| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00072-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00861-09 |
| Acinetobacter baumannii |
ADC-11 |
Kcat |
550.0 |
/s |
10.1128/aac.00050-10 |
| Acinetobacter baumannii |
ADC-11 |
Kcat/Km |
2.5 |
/uM/s |
10.1128/aac.00050-10 |
| Acinetobacter baumannii |
ADC-11 |
Km |
210000.0 |
nM |
10.1128/aac.00050-10 |
| Acinetobacter baumannii |
Beta-lactamase ADC-33 |
Kcat |
140.0 |
/s |
10.1128/aac.00050-10 |
| Acinetobacter baumannii |
Beta-lactamase ADC-33 |
Kcat/Km |
1.0 |
/uM/s |
10.1128/aac.00050-10 |
| Acinetobacter baumannii |
Beta-lactamase ADC-33 |
Km |
120000.0 |
nM |
10.1128/aac.00050-10 |
| Acinetobacter genomosp. 3 |
ADC-14 protein |
Kcat |
56.52 |
/s |
10.1128/aac.00485-08 |
| Acinetobacter genomosp. 3 |
ADC-14 protein |
Kcat/Km |
8398.16 |
/mM/s |
10.1128/aac.00485-08 |
| Acinetobacter genomosp. 3 |
ADC-14 protein |
Km |
6730.0 |
nM |
10.1128/aac.00485-08 |
| Acinetobacter genomosp. 3 |
ADC-16 protein |
Kcat |
1380.8 |
/s |
10.1128/aac.00485-08 |
| Acinetobacter genomosp. 3 |
ADC-16 protein |
Kcat/Km |
9916.65 |
/mM/s |
10.1128/aac.00485-08 |
| Acinetobacter genomosp. 3 |
ADC-16 protein |
Km |
139240.0 |
nM |
10.1128/aac.00485-08 |
| Acinetobacter genomosp. 3 |
ADC-18 protein |
Kcat |
1418.36 |
/s |
10.1128/aac.00485-08 |
| Acinetobacter genomosp. 3 |
ADC-18 protein |
Kcat/Km |
9566.33 |
/mM/s |
10.1128/aac.00485-08 |
| Acinetobacter genomosp. 3 |
ADC-18 protein |
Km |
148270.0 |
nM |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
24.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
28.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
48.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
96.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
192.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00072-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Aeromonas allosaccharophila |
Extended-spectrum beta-lactamase PER-6 |
Kcat |
8.0 |
/s |
10.1128/aac.01585-09 |
| Aeromonas allosaccharophila |
Extended-spectrum beta-lactamase PER-6 |
Kcat/Km |
145.0 |
/uM/s |
10.1128/aac.01585-09 |
| Aeromonas allosaccharophila |
Extended-spectrum beta-lactamase PER-6 |
Km |
55000.0 |
nM |
10.1128/aac.01585-09 |
| Aeromonas caviae |
IMP-19 |
Kcat |
11.0 |
/s |
10.1128/aac.01462-06 |
| Aeromonas caviae |
IMP-19 |
Kcat/Km |
0.14 |
None |
10.1128/aac.01462-06 |
| Aeromonas caviae |
IMP-19 |
Km |
76000.0 |
nM |
10.1128/aac.01462-06 |
| Aeromonas sp. |
Aeromonas sp. |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00770-08 |
| Aspergillus fumigatus |
Aspergillus fumigatus |
IZ |
nan |
None |
10.1016/j.ejmech.2010.05.018 |
| Aspergillus fumigatus |
Aspergillus fumigatus |
MIC |
nan |
None |
10.1016/j.ejmech.2010.05.018 |
| Aspergillus niger |
Aspergillus niger |
DIZ |
nan |
None |
10.1007/s00044-012-9978-0 |
| Aspergillus niger |
Aspergillus niger |
MIC |
nan |
None |
10.1007/s00044-012-9978-0 |
| Bacillus clausii |
Beta-lactamase |
Activity |
18.0 |
None |
10.1128/aac.00537-07 |
| Bacillus clausii |
Beta-lactamase |
Activity |
35.0 |
U |
10.1128/aac.00537-07 |
| Bacillus clausii |
Beta-lactamase |
Kcat |
22.0 |
/s |
10.1128/aac.00537-07 |
| Bacillus clausii |
Beta-lactamase |
Kcat/Km |
1.5 |
/uM/s |
10.1128/aac.00537-07 |
| Bacillus clausii |
Beta-lactamase |
Km |
15000.0 |
nM |
10.1128/aac.00537-07 |
| Bacillus subtilis |
4'-phosphopantetheinyl transferase ffp |
Potency |
56234.1 |
nM |
None |
| Bacillus subtilis |
Bacillus subtilis |
IZ |
36.0 |
mm |
10.1016/j.ejmech.2011.03.045 |
| Bacillus subtilis |
Bacillus subtilis |
IZ |
36.0 |
mm |
10.1016/j.ejmech.2012.11.017 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2011.03.045 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2012.11.017 |
| Bacillus thuringiensis |
Bacillus thuringiensis |
IZ |
37.0 |
mm |
10.1016/j.ejmech.2011.03.045 |
| Bacillus thuringiensis |
Bacillus thuringiensis |
IZ |
37.0 |
mm |
10.1016/j.ejmech.2012.11.017 |
| Bacillus thuringiensis |
Bacillus thuringiensis |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2011.03.045 |
| Bacillus thuringiensis |
Bacillus thuringiensis |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2012.11.017 |
| Botrytis fabae |
Botrytis fabae |
DIZ |
nan |
None |
10.1016/j.ejmech.2012.11.017 |
| Botrytis fabae |
Botrytis fabae |
IZ |
nan |
None |
10.1016/j.ejmech.2011.03.045 |
| Botrytis fabae |
Botrytis fabae |
MIC |
nan |
None |
10.1016/j.ejmech.2011.03.045 |
| Botrytis fabae |
Botrytis fabae |
MIC |
nan |
None |
10.1016/j.ejmech.2012.11.017 |
| Brachyspira pilosicoli |
Class D beta-lactamase |
Kcat |
nan |
None |
10.1128/aac.00684-07 |
| Burkholderia cenocepacia |
PenB class A beta-lactamase |
Kcat |
300.0 |
/s |
10.1128/aac.00946-08 |
| Burkholderia cenocepacia |
PenB class A beta-lactamase |
Kcat/Km |
3000.0 |
/uM/s |
10.1128/aac.00946-08 |
| Burkholderia cenocepacia |
PenB class A beta-lactamase |
Km |
100000.0 |
nM |
10.1128/aac.00946-08 |
| Campylobacter coli |
Campylobacter coli |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter coli |
Campylobacter coli |
MIC50 |
256.0 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter coli |
Campylobacter coli |
MIC90 |
256.0 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC50 |
256.0 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC90 |
256.0 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Caulobacter vibrioides |
Metallo-beta-lactamase |
Kcat/Km |
4.3 |
10'5/M/s |
10.1128/aac.01062-07 |
| Chryseobacterium indologenes |
Chryseobacterium indologenes |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01607-08 |
| Chryseobacterium indologenes |
Metallo-beta-lactamase IND-2 |
Kcat/Km |
1.2 |
10'6/M/s |
10.1128/aac.01607-08 |
| Chryseobacterium indologenes |
Metallo-beta-lactamase IND-6 |
Kcat |
415.0 |
/s |
10.1128/aac.01607-08 |
| Chryseobacterium indologenes |
Metallo-beta-lactamase IND-6 |
Kcat/Km |
6.9 |
10'6/M/s |
10.1128/aac.01607-08 |
| Chryseobacterium indologenes |
Metallo-beta-lactamase IND-6 |
Km |
60000.0 |
nM |
10.1128/aac.01607-08 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01395-06 |
| Citrobacter freundii |
PER-2 beta-lactamase |
Activity |
100.0 |
% |
10.1128/aac.01395-06 |
| Citrobacter freundii |
PER-2 beta-lactamase |
Kcat |
6.0 |
/s |
10.1128/aac.01395-06 |
| Citrobacter freundii |
PER-2 beta-lactamase |
Kcat/Km |
0.67 |
/uM/s |
10.1128/aac.01395-06 |
| Citrobacter freundii |
PER-2 beta-lactamase |
Km |
9000.0 |
nM |
10.1128/aac.01395-06 |
| Citrobacter gillenii |
Gil1 |
Kcat |
37.0 |
/s |
10.1128/aac.01152-06 |
| Citrobacter gillenii |
Gil1 |
Kcat/Km |
598.0 |
/mM/s |
10.1128/aac.01152-06 |
| Citrobacter gillenii |
Gil1 |
Km |
62000.0 |
nM |
10.1128/aac.01152-06 |
| Citrobacter gillenii |
Gil1 |
Ratio |
11.0 |
None |
10.1128/aac.01152-06 |
| Dialister invisus |
Dialister invisus |
Activity |
8.0 |
ug ml-1 |
10.1128/aac.00538-07 |
| Dialister invisus |
Dialister invisus |
Activity |
nan |
None |
10.1128/aac.00538-07 |
| Dialister invisus |
Dialister invisus |
MIC |
nan |
None |
10.1128/aac.00538-07 |
| Dialister micraerophilus |
Dialister micraerophilus |
Activity |
8.0 |
ug ml-1 |
10.1128/aac.00538-07 |
| Dialister micraerophilus |
Dialister micraerophilus |
Activity |
nan |
None |
10.1128/aac.00538-07 |
| Dialister micraerophilus |
Dialister micraerophilus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Dialister pneumosintes |
Dialister pneumosintes |
Activity |
8.0 |
ug ml-1 |
10.1128/aac.00538-07 |
| Dialister pneumosintes |
Dialister pneumosintes |
Activity |
nan |
None |
10.1128/aac.00538-07 |
| Dialister pneumosintes |
Dialister pneumosintes |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Dialister pneumosintes |
Dialister pneumosintes |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Dialister pneumosintes |
Dialister pneumosintes |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Dialister propionicifaciens |
Dialister propionicifaciens |
Activity |
8.0 |
ug ml-1 |
10.1128/aac.00538-07 |
| Dialister propionicifaciens |
Dialister propionicifaciens |
Activity |
nan |
None |
10.1128/aac.00538-07 |
| Dialister propionicifaciens |
Dialister propionicifaciens |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Elizabethkingia meningoseptica |
GOB-1 metallo-beta-lactamase |
Kcat/Km |
6.7 |
10'5/M/s |
10.1128/aac.01062-07 |
| Enterobacter |
Enterobacter |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01614-06 |
| Enterobacter cloacae |
Beta-lactamase |
K cat |
200.0 |
s-1 |
10.1016/j.bmcl.2004.07.067 |
| Enterobacter cloacae |
Beta-lactamase |
Km |
9000.0 |
nM |
10.1016/j.bmcl.2004.07.067 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00178a011 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00193a001 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00207a022 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
125.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
125.0 |
ug.mL-1 |
10.1021/jm00375a026 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
128.0 |
ug.mL-1 |
10.1021/jm00346a024 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01082-06 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Enterobacter cloacae |
IMI-1 |
Kcat |
120.0 |
/s |
10.1128/aac.00491-07 |
| Enterobacter cloacae |
IMI-1 |
Kcat/Km |
920.0 |
/mM/s |
10.1128/aac.00491-07 |
| Enterobacter cloacae |
IMI-1 |
Km |
130000.0 |
nM |
10.1128/aac.00491-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm00346a024 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
13.0 |
ug.mL-1 |
10.1021/jm00211a006 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm00375a026 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00178a011 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00207a022 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
14000.0 |
nM |
10.1021/jm00203a001 |
| Escherichia coli |
Beta-lactamase ACC-4 |
Kcat |
96.0 |
/s |
10.1128/aac.00389-07 |
| Escherichia coli |
Beta-lactamase ACC-4 |
Kcat/Km |
3.2 |
/s/microM |
10.1128/aac.00389-07 |
| Escherichia coli |
Beta-lactamase ACC-4 |
Km |
30000.0 |
nM |
10.1128/aac.00389-07 |
| Escherichia coli |
Beta-lactamase OXA-1 |
K cat |
1.2 |
s-1 |
10.1016/j.bmcl.2004.07.067 |
| Escherichia coli |
Beta-lactamase OXA-1 |
Km |
10000.0 |
nM |
10.1016/j.bmcl.2004.07.067 |
| Escherichia coli |
Beta-lactamase SCO-1 |
Activity |
3.0 |
None |
10.1128/aac.01439-06 |
| Escherichia coli |
Beta-lactamase SHV-1 |
Kcat |
128.0 |
/s |
10.1128/aac.01442-09 |
| Escherichia coli |
Beta-lactamase SHV-1 |
Kcat/Km |
3.2 |
/uM/s |
10.1128/aac.01442-09 |
| Escherichia coli |
Beta-lactamase SHV-1 |
Km |
40000.0 |
nM |
10.1128/aac.01442-09 |
| Escherichia coli |
Beta-lactamase SHV-11 |
Kcat |
0.5 |
/s |
10.1128/aac.00387-08 |
| Escherichia coli |
Beta-lactamase SHV-11 |
Kcat/Km |
10.0 |
/uM/s |
10.1128/aac.00387-08 |
| Escherichia coli |
Beta-lactamase SHV-11 |
Km |
50000.0 |
nM |
10.1128/aac.00387-08 |
| Escherichia coli |
Beta-lactamase TEM |
Activity |
27.0 |
None |
10.1128/aac.01439-06 |
| Escherichia coli |
Beta-lactamase TEM |
K cat |
115.0 |
1/S |
10.1021/jm0493663 |
| Escherichia coli |
Beta-lactamase TEM |
K cat |
120.0 |
s-1 |
10.1016/j.bmcl.2004.07.067 |
| Escherichia coli |
Beta-lactamase TEM |
Kcat |
165.0 |
/s |
10.1128/aac.00614-07 |
| Escherichia coli |
Beta-lactamase TEM |
Kcat/Km |
0.7 |
None |
10.1128/aac.00614-07 |
| Escherichia coli |
Beta-lactamase TEM |
Km |
242.0 |
/s/microM |
10.1128/aac.00614-07 |
| Escherichia coli |
Beta-lactamase TEM |
Km |
200000.0 |
nM |
10.1016/j.bmcl.2004.07.067 |
| Escherichia coli |
Beta-lactamase TEM |
Km |
347000.0 |
nM |
10.1021/jm0493663 |
| Escherichia coli |
Beta-lactamase TEM |
Ratio |
7.7 |
10'5/M/s |
10.1128/aac.00011-07 |
| Escherichia coli |
Beta-lactamase Toho-1 |
Kcat |
790.0 |
/s |
10.1128/aac.00098-10 |
| Escherichia coli |
Beta-lactamase Toho-1 |
Kcat/Km |
4.3 |
10'6/s/M |
10.1128/aac.00098-10 |
| Escherichia coli |
Beta-lactamase Toho-1 |
Km |
190000.0 |
nM |
10.1128/aac.00098-10 |
| Escherichia coli |
BlaVIM-1 |
Kcat |
281.0 |
/s |
10.1128/aac.00017-09 |
| Escherichia coli |
BlaVIM-1 |
Kcat/Km |
5.3 |
/s/microM |
10.1128/aac.00017-09 |
| Escherichia coli |
CMT-type beta lactamase |
Kcat |
0.26 |
/s |
10.1128/aac.00614-07 |
| Escherichia coli |
CMT-type beta lactamase |
Kcat/Km |
0.0015 |
None |
10.1128/aac.00614-07 |
| Escherichia coli |
CMT-type beta lactamase |
Km |
170.4 |
/s/microM |
10.1128/aac.00614-07 |
| Escherichia coli |
Escherichia coli |
Activity |
100.0 |
% |
10.1128/aac.01412-06 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1128/aac.00614-07 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1128/aac.01195-06 |
| Escherichia coli |
Escherichia coli |
Antibiotic resistance |
nan |
None |
10.1016/s0960-894x(98)00536-8 |
| Escherichia coli |
Escherichia coli |
IZ |
11.0 |
mm |
10.1016/j.bmcl.2016.05.053 |
| Escherichia coli |
Escherichia coli |
IZ |
38.0 |
mm |
10.1016/j.ejmech.2011.03.045 |
| Escherichia coli |
Escherichia coli |
IZ |
38.0 |
mm |
10.1016/j.ejmech.2012.11.017 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01395-06 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00787-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01180-07 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01442-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.2 |
ug.mL-1 |
10.1128/aac.00787-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.3 |
ug.mL-1 |
10.1128/aac.00787-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.03.008 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm301490d |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00098-10 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00219-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00389-07 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00608-08 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00642-08 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00787-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00859-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00961-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01152-06 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01439-06 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01463-07 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01585-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01600-06 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01615-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2.3 |
ug.mL-1 |
10.1128/aac.00787-09 |
| Escherichia coli |
Escherichia coli |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Escherichia coli |
Escherichia coli |
MIC |
3.1 |
ug.mL-1 |
10.1021/jm00211a006 |
| Escherichia coli |
Escherichia coli |
MIC |
3.1 |
ug.mL-1 |
10.1021/jm00219a010 |
| Escherichia coli |
Escherichia coli |
MIC |
3.1 |
ug.mL-1 |
10.1021/jm00228a003 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00011-07 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00387-08 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00427-09 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00543-08 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00614-07 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00638-08 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00642-08 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00774-09 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00791-09 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00858-10 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01025-07 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01058-06 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01082-06 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01164-08 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01252-09 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01381-07 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01607-08 |
| Escherichia coli |
Escherichia coli |
MIC |
4.7 |
ug.mL-1 |
10.1128/aac.00787-09 |
| Escherichia coli |
Escherichia coli |
MIC |
5.0 |
ug.mL-1 |
10.1021/jm00218a018 |
| Escherichia coli |
Escherichia coli |
MIC |
5.3 |
ug.mL-1 |
10.1128/aac.00787-09 |
| Escherichia coli |
Escherichia coli |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.00787-09 |
| Escherichia coli |
Escherichia coli |
MIC |
6.2 |
ug.mL-1 |
10.1021/jm00207a022 |
| Escherichia coli |
Escherichia coli |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2011.03.045 |
| Escherichia coli |
Escherichia coli |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2012.11.017 |
| Escherichia coli |
Escherichia coli |
MIC |
6.3 |
ug.mL-1 |
10.1021/jm00193a001 |
| Escherichia coli |
Escherichia coli |
MIC |
6.7 |
ug.mL-1 |
10.1128/aac.00787-09 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.05.110 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm301490d |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00387-08 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00543-08 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00614-07 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00638-08 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00642-08 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00770-08 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00774-09 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01058-06 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01152-06 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01164-08 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01381-07 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01412-06 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01439-06 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01442-09 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01463-07 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01600-06 |
| Escherichia coli |
Escherichia coli |
MIC |
9.3 |
ug.mL-1 |
10.1128/aac.00787-09 |
| Escherichia coli |
Escherichia coli |
MIC |
10.7 |
ug.mL-1 |
10.1128/aac.00787-09 |
| Escherichia coli |
Escherichia coli |
MIC |
12.5 |
ug.mL-1 |
10.1021/jm00178a011 |
| Escherichia coli |
Escherichia coli |
MIC |
15.0 |
ug.mL-1 |
10.1021/jm00217a021 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm00375a026 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm301490d |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00614-07 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00642-08 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01058-06 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01062-07 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01082-06 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01336-09 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01381-07 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01442-09 |
| Escherichia coli |
Escherichia coli |
MIC |
30.0 |
ug.mL-1 |
10.1021/jm00211a041 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm00375a026 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00427-09 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00614-07 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00642-08 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00858-10 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01058-06 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00011-07 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00642-08 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00770-08 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01025-07 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01058-06 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01062-07 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01164-08 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01607-08 |
| Escherichia coli |
Escherichia coli |
MIC |
106.0 |
ug.mL-1 |
10.1128/aac.01336-09 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1021/jm00346a024 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00098-10 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00642-08 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00961-09 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01058-06 |
| Escherichia coli |
Escherichia coli |
MIC |
192.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1021/jm301490d |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00638-08 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00642-08 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00774-09 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00858-10 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00859-09 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01180-07 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01252-09 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01336-09 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01439-06 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01585-09 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01615-09 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00098-10 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00219-09 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00389-07 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00608-08 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00642-08 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00791-09 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01395-06 |
| Escherichia coli |
Escherichia coli |
MIC |
1000.0 |
ug.mL-1 |
10.1128/aac.00537-07 |
| Escherichia coli |
Escherichia coli |
MIC |
1024.0 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1024.0 |
ug.mL-1 |
10.1128/aac.00642-08 |
| Escherichia coli |
Escherichia coli |
MIC |
1024.0 |
ug.mL-1 |
10.1128/aac.01412-06 |
| Escherichia coli |
Escherichia coli |
MIC |
2048.0 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2048.0 |
ug.mL-1 |
10.1128/aac.00098-10 |
| Escherichia coli |
Escherichia coli |
MIC |
4000.0 |
ug.mL-1 |
10.1128/aac.00537-07 |
| Escherichia coli |
Escherichia coli |
MIC |
7000.0 |
nM |
10.1021/jm00203a001 |
| Escherichia coli |
Escherichia coli |
MIC |
12500.0 |
nM |
10.1021/acs.jmedchem.8b01923 |
| Escherichia coli |
Escherichia coli |
MIC |
16000.0 |
ug.mL-1 |
10.1128/aac.00537-07 |
| Escherichia coli |
Escherichia coli |
MIC |
25000.0 |
nM |
10.1021/acs.jmedchem.8b01923 |
| Escherichia coli |
Escherichia coli |
MIC |
64000.0 |
ug.mL-1 |
10.1128/aac.00537-07 |
| Escherichia coli |
Escherichia coli |
MIC |
100000.0 |
nM |
10.1021/acs.jmedchem.8b01923 |
| Escherichia coli |
Escherichia coli |
MIC |
400000.0 |
nM |
10.1021/acs.jmedchem.8b01923 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1128/aac.00787-09 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1128/aac.01472-06 |
| Escherichia coli |
Escherichia coli |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.01412-06 |
| Escherichia coli |
Escherichia coli |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.01412-06 |
| Escherichia coli |
Escherichia coli |
PD50 |
50.0 |
mg kg-1 |
10.1021/jm00211a006 |
| Escherichia coli |
Escherichia coli |
PD50 |
50.0 |
mg kg-1 |
10.1021/jm00219a010 |
| Escherichia coli |
Escherichia coli |
PD50 |
50.0 |
mg kg-1 |
10.1021/jm00228a003 |
| Escherichia coli |
Escherichia coli |
Ratio |
1.0 |
None |
10.1016/j.ejmech.2012.03.008 |
| Escherichia coli |
Escherichia coli |
Ratio |
16.0 |
None |
10.1128/aac.00734-08 |
| Escherichia coli |
Escherichia coli |
Stability |
6.0 |
nmol/min |
10.1128/aac.00734-08 |
| Escherichia coli |
Escherichia coli |
Stability |
7.0 |
nmol/min |
10.1128/aac.00734-08 |
| Escherichia coli |
Escherichia coli |
Stability |
25.0 |
nmol/min |
10.1128/aac.00734-08 |
| Escherichia coli |
Escherichia coli |
Stability |
50.0 |
nmol/min |
10.1128/aac.00734-08 |
| Escherichia coli |
Escherichia coli |
Stability |
53.0 |
nmol/min |
10.1128/aac.00734-08 |
| Escherichia coli |
Escherichia coli |
Stability |
65.0 |
nmol/min |
10.1128/aac.00734-08 |
| Escherichia coli |
Metallo-beta-lactamase |
Activity |
141.0 |
umol |
10.1128/aac.01025-07 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat |
56.2 |
/s |
10.1128/aac.00017-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat |
130.0 |
/s |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat |
320.0 |
/s |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat/Km |
1.28 |
/s/microM |
10.1128/aac.00017-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat/Km |
11.0 |
/uM/s |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat/Km |
12.0 |
uM/hr |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat/Km |
12.0 |
/uM/s |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat/Km |
13.0 |
/uM/s |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Km |
10000.0 |
nM |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Km |
11000.0 |
nM |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Km |
28000.0 |
nM |
10.1128/aac.01336-09 |
| Escherichia coli K-12 |
Beta-lactamase AmpC |
Kcat/Km |
2.86 |
microM/s |
10.1021/acs.jmedchem.8b01923 |
| Flavobacterium meningosepticum |
Carbapenem-hydrolyzing beta-lactamase BlaB-1 |
Kcat/Km |
1.6 |
10'6/M/s |
10.1128/aac.01607-08 |
| Fluoribacter gormanii |
FEZ-1 protein |
Kcat/Km |
2.5 |
10'6/M/s |
10.1128/aac.01062-07 |
| Fusarium oxysporum |
Fusarium oxysporum |
DIZ |
nan |
None |
10.1007/s00044-012-9978-0 |
| Fusarium oxysporum |
Fusarium oxysporum |
DIZ |
nan |
None |
10.1016/j.ejmech.2012.11.017 |
| Fusarium oxysporum |
Fusarium oxysporum |
IZ |
nan |
None |
10.1016/j.ejmech.2010.05.018 |
| Fusarium oxysporum |
Fusarium oxysporum |
IZ |
nan |
None |
10.1016/j.ejmech.2011.03.045 |
| Fusarium oxysporum |
Fusarium oxysporum |
MIC |
nan |
None |
10.1007/s00044-012-9978-0 |
| Fusarium oxysporum |
Fusarium oxysporum |
MIC |
nan |
None |
10.1016/j.ejmech.2010.05.018 |
| Fusarium oxysporum |
Fusarium oxysporum |
MIC |
nan |
None |
10.1016/j.ejmech.2011.03.045 |
| Fusarium oxysporum |
Fusarium oxysporum |
MIC |
nan |
None |
10.1016/j.ejmech.2012.11.017 |
| Giardia intestinalis |
Putative fructose-1,6-bisphosphate aldolase |
Potency |
28117.1 |
nM |
None |
| Homo sapiens |
15-hydroxyprostaglandin dehydrogenase [NAD+] |
Potency |
19952.6 |
nM |
None |
| Homo sapiens |
Adenosine A1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A2a receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2b adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2c adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-1 adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-2 adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bradykinin B2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cannabinoid CB1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 |
IC50 |
2786.0 |
nM |
None |
| Homo sapiens |
Cerebroside-sulfatase |
Potency |
37933.0 |
nM |
None |
| Homo sapiens |
Cholecystokinin A receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cholecystokinin B receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Delta opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
DNA (cytosine-5)-methyltransferase 1 |
IC50 |
7280.0 |
nM |
None |
| Homo sapiens |
DNA polymerase eta |
Potency |
5358.2 |
nM |
None |
| Homo sapiens |
DNA polymerase eta |
Potency |
7079.5 |
nM |
None |
| Homo sapiens |
DNA polymerase iota |
Potency |
15003.0 |
nM |
None |
| Homo sapiens |
DNA polymerase iota |
Potency |
31622.8 |
nM |
None |
| Homo sapiens |
DNA polymerase kappa |
Potency |
39810.7 |
nM |
None |
| Homo sapiens |
DNA polymerase kappa |
Potency |
50118.7 |
nM |
None |
| Homo sapiens |
Dopamine D1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Endothelin receptor ET-A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Equilibrative nucleoside transporter 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Flap endonuclease 1 |
Potency |
70794.6 |
nM |
None |
| Homo sapiens |
Gamma-aminobutyric acid receptor subunit alpha-1/alpha-2/beta-2/gamma-2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Ghrelin receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glutaminase kidney isoform, mitochondrial |
Potency |
19952.6 |
nM |
None |
| Homo sapiens |
Glutaminase kidney isoform, mitochondrial |
Potency |
35481.3 |
nM |
None |
| Homo sapiens |
HepG2 |
LD50 |
100.0 |
ug ml-1 |
10.1021/acs.jmedchem.5b01833 |
| Homo sapiens |
HERG |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histone deacetylase 6 |
Inhibition |
-26.47 |
% |
10.6019/CHEMBL4808148 |
| Homo sapiens |
Histone deacetylase 6 |
Inhibition |
-1.53 |
% |
10.6019/CHEMBL4808148 |
| Homo sapiens |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Potency |
7519.3 |
nM |
None |
| Homo sapiens |
Homo sapiens |
AUC |
9890.0 |
ng.hr.mL-1 |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
AUC |
12050.0 |
ng.hr.mL-1 |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
CL_renal |
98.0 |
ml/min |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
CL_renal |
148.0 |
ml/min |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
Cmax |
53726.83 |
nM |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
Cmax |
97616.35 |
nM |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
MRT |
0.38 |
hr |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
MRT |
0.59 |
hr |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
T1/2 |
0.26 |
hr |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
T1/2 |
0.41 |
hr |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
T1/2 |
0.74 |
hr |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
T1/2 |
0.91 |
hr |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
Vdss |
0.6 |
L.kg-1 |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
Vdss |
0.63 |
L.kg-1 |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
Vz |
1.19 |
L/hr/kg |
10.1128/aac.01600-08 |
| Homo sapiens |
Homo sapiens |
Vz |
1.58 |
L/hr/kg |
10.1128/aac.01600-08 |
| Homo sapiens |
Importin subunit beta-1/Snurportin-1 |
Potency |
112201.8 |
nM |
None |
| Homo sapiens |
Kappa opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Lysine-specific demethylase 4A |
Potency |
79432.8 |
nM |
None |
| Homo sapiens |
Melanocortin receptor 3 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Microtubule-associated protein tau |
Potency |
22387.2 |
nM |
None |
| Homo sapiens |
Microtubule-associated protein tau |
Potency |
28183.8 |
nM |
None |
| Homo sapiens |
Monoamine oxidase A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Motilin receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Mu opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuronal acetylcholine receptor protein alpha-4 subunit |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Norepinephrine transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Oligopeptide transporter small intestine isoform |
Ki |
10000000.0 |
nM |
10.1016/j.ejpb.2004.07.008 |
| Homo sapiens |
Oligopeptide transporter small intestine isoform |
Ki |
10000000.0 |
nM |
10.1021/jm048982w |
| Homo sapiens |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
Potency |
21331.3 |
nM |
None |
| Homo sapiens |
Peroxisome proliferator-activated receptor gamma |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 3A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 4D |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Plasma |
Cp |
17.6 |
mg/L |
10.1128/aac.00718-08 |
| Homo sapiens |
Plasma |
Cp |
38.7 |
mg/L |
10.1128/aac.00718-08 |
| Homo sapiens |
Plasma |
PPB |
58.0 |
% |
10.1128/aac.00718-08 |
| Homo sapiens |
Plasma |
PPB |
59.0 |
% |
10.1128/aac.01600-08 |
| Homo sapiens |
Plasma |
PPB |
70.8 |
% |
10.1128/aac.00718-08 |
| Homo sapiens |
Plasma |
PPB |
71.0 |
% |
10.1128/aac.01600-08 |
| Homo sapiens |
Pregnane X receptor |
AC50 |
21999.9 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Pregnane X receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Progesterone receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Regulator of G-protein signaling 4 |
Potency |
18887.6 |
nM |
None |
| Homo sapiens |
Serine/threonine-protein kinase PLK1 |
Potency |
23778.1 |
nM |
None |
| Homo sapiens |
Serotonin 1a (5-HT1a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 3a (5-HT3a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Solute carrier family 15 member 2 |
Ki |
8300000.0 |
nM |
10.1016/j.bmc.2011.06.027 |
| Homo sapiens |
Solute carrier family 15 member 2 |
Ki |
8317637.71 |
nM |
10.1016/j.bmc.2011.06.027 |
| Homo sapiens |
Solute carrier family 22 member 11 |
Ki |
200.0 |
nM |
10.1016/s0014-2999(02)01306-7 |
| Homo sapiens |
Solute carrier family 22 member 5 |
Activity |
nan |
None |
None |
| Homo sapiens |
Solute carrier family 22 member 6 |
Ki |
220.0 |
nM |
10.1016/s0014-2999(02)01306-7 |
| Homo sapiens |
Solute carrier family 22 member 7 |
IC50 |
1410000.0 |
nM |
10.1016/s0014-2999(03)01381-5 |
| Homo sapiens |
Solute carrier family 22 member 8 |
Inhibition |
nan |
% |
10.1124/dmd.112.049569 |
| Homo sapiens |
Solute carrier family 22 member 8 |
Ki |
40.0 |
nM |
10.1016/s0014-2999(02)01306-7 |
| Homo sapiens |
Type-1 angiotensin II receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Tyrosyl-DNA phosphodiesterase 1 |
Potency |
25118.9 |
nM |
None |
| Homo sapiens |
Vasopressin V1a receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vasopressin V2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vitamin D receptor |
Potency |
56234.1 |
nM |
None |
| Homo sapiens |
Vitamin D receptor |
Potency |
63095.7 |
nM |
None |
| Homo sapiens |
Werner syndrome ATP-dependent helicase |
Potency |
50118.7 |
nM |
None |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
3.0 |
ug.mL-1 |
10.1021/jm00217a021 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
5.0 |
ug.mL-1 |
10.1021/jm00218a018 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
12.5 |
ug.mL-1 |
10.1021/jm00219a010 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm00346a024 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
50.0 |
ug.mL-1 |
10.1021/jm00207a022 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
50.0 |
ug.mL-1 |
10.1021/jm00211a006 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
50.0 |
ug.mL-1 |
10.1021/jm00228a003 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00178a011 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
14000.0 |
nM |
10.1021/jm00203a001 |
| Klebsiella pneumoniae |
Beta-lactamase NDM-1 |
Kcat |
4.0 |
/s |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
Beta-lactamase NDM-1 |
Kcat/Km |
0.4 |
/s/microM |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
Beta-lactamase NDM-1 |
Km |
10000.0 |
nM |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-1 |
Kcat |
128.0 |
/s |
10.1128/aac.01381-07 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-1 |
Kcat |
128.0 |
/s |
10.1128/aac.01525-07 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-1 |
Kcat/Km |
3.2 |
/uM/s |
10.1128/aac.01381-07 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-1 |
Kcat/Km |
3.2 |
/uM/s |
10.1128/aac.01525-07 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-1 |
Km |
40000.0 |
nM |
10.1128/aac.01381-07 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-1 |
Km |
40000.0 |
nM |
10.1128/aac.01525-07 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-55 |
Kcat |
38.0 |
/s |
10.1128/aac.01525-07 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-55 |
Kcat/Km |
4.4 |
/uM/s |
10.1128/aac.01525-07 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-55 |
Km |
9000.0 |
nM |
10.1128/aac.01525-07 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-72 |
Kcat |
38.0 |
/s |
10.1128/aac.01381-07 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-72 |
Kcat/Km |
0.3 |
/uM/s |
10.1128/aac.01381-07 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-72 |
Km |
141000.0 |
nM |
10.1128/aac.01381-07 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Kcat |
44.0 |
/s |
10.1128/aac.00197-10 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Kcat |
75.0 |
/s |
10.1128/aac.00491-07 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Kcat/Km |
3.1 |
/uM/s |
10.1128/aac.00197-10 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Kcat/Km |
1400.0 |
/mM/s |
10.1128/aac.00491-07 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Km |
14000.0 |
nM |
10.1128/aac.00197-10 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Km |
53000.0 |
nM |
10.1128/aac.00491-07 |
| Klebsiella pneumoniae |
Class C beta-lactamase CMY-36 |
Kcat |
140.0 |
/s |
10.1128/aac.01284-08 |
| Klebsiella pneumoniae |
Class C beta-lactamase CMY-36 |
Kcat/Km |
31.8 |
/uM/s |
10.1128/aac.01284-08 |
| Klebsiella pneumoniae |
Class C beta-lactamase CMY-36 |
Km |
4400.0 |
nM |
10.1128/aac.01284-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm00346a024 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.8 |
ug.mL-1 |
10.1021/jm00193a001 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm00211a041 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm00217a021 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.6 |
ug.mL-1 |
10.1021/jm00219a010 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
3.1 |
ug.mL-1 |
10.1021/jm00178a011 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
3.1 |
ug.mL-1 |
10.1021/jm00207a022 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
3.1 |
ug.mL-1 |
10.1021/jm00211a006 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
3.1 |
ug.mL-1 |
10.1021/jm00228a003 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00387-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01381-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm00375a026 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00543-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00193a001 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
125.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
125.0 |
ug.mL-1 |
10.1021/jm00375a026 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00543-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01180-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1024.0 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2048.0 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
3600.0 |
nM |
10.1021/jm00203a001 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase VIM-2 |
Kcat |
57.0 |
/s |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase VIM-2 |
Kcat/Km |
1.28 |
/s/microM |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase VIM-2 |
Km |
44000.0 |
nM |
10.1128/aac.00774-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
IZ |
30.3 |
mm |
10.1128/aac.00503-10 |
| Listeria monocytogenes |
Listeria monocytogenes |
IZ |
33.6 |
mm |
10.1128/aac.00503-10 |
| Morganella morganii |
Morganella morganii |
MIC |
63.0 |
ug.mL-1 |
10.1021/jm00375a026 |
| Morganella morganii |
Morganella morganii |
MIC |
125.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Morganella morganii |
Morganella morganii |
MIC |
125.0 |
ug.mL-1 |
10.1021/jm00375a026 |
| Morganella morganii |
Morganella morganii |
MIC |
128.0 |
ug.mL-1 |
10.1021/jm00346a024 |
| Morganella morganii |
Morganella morganii |
MIC |
200.0 |
ug.mL-1 |
10.1021/jm00219a010 |
| Morganella morganii |
Morganella morganii |
MIC |
453000.0 |
nM |
10.1021/jm00203a001 |
| Mus musculus |
Monoamine oxidase A |
Activity |
nan |
None |
10.1021/jm800656v |
| Mus musculus |
Solute carrier family 22 member 6 |
Inhibition |
nan |
% |
10.1124/dmd.112.049569 |
| Mus musculus |
Solute carrier family 22 member 8 |
Drug uptake |
nan |
None |
10.1124/dmd.112.049569 |
| Mus musculus |
Solute carrier family 22 member 8 |
IC50 |
33300.0 |
nM |
10.1124/dmd.112.049569 |
| Mus musculus |
Solute carrier family 22 member 8 |
Inhibition |
nan |
% |
10.1124/dmd.112.049569 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
95.53 |
ug.mL-1 |
10.1021/acs.jmedchem.5b01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
100.0 |
ug.mL-1 |
10.1021/acs.jmedchem.5b01833 |
| Pectobacterium atrosepticum |
Pectobacterium atrosepticum |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01062-07 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm00375a026 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
3.1 |
ug.mL-1 |
10.1021/jm00193a001 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
5.0 |
ug.mL-1 |
10.1021/jm00218a018 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
6.2 |
ug.mL-1 |
10.1021/jm00207a022 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm00375a026 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
12.5 |
ug.mL-1 |
10.1021/jm00178a011 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01399-07 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm00346a024 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
50.0 |
ug.mL-1 |
10.1021/jm00193a001 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00207a022 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00211a041 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
128.0 |
ug.mL-1 |
10.1021/jm00346a024 |
| Providencia rettgeri |
Providencia rettgeri |
MIC |
63.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Providencia rettgeri |
Providencia rettgeri |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Providencia stuartii |
Providencia stuartii |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00207a022 |
| Providencia stuartii |
Providencia stuartii |
MIC |
2048.0 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Pseudomonas |
Pseudomonas |
IZ |
38.0 |
mm |
10.1007/s00044-012-9978-0 |
| Pseudomonas |
Pseudomonas |
IZ |
38.0 |
mm |
10.1016/j.ejmech.2010.05.018 |
| Pseudomonas |
Pseudomonas |
MIC |
6.25 |
ug.mL-1 |
10.1007/s00044-012-9978-0 |
| Pseudomonas |
Pseudomonas |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2010.05.018 |
| Pseudomonas aeruginosa |
Beta-lactamase |
Kcat |
4.3 |
/s |
10.1128/aac.00859-09 |
| Pseudomonas aeruginosa |
Beta-lactamase |
Kcat |
115.0 |
/s |
10.1128/aac.01410-08 |
| Pseudomonas aeruginosa |
Beta-lactamase |
Kcat/Km |
2200.0 |
/mM/s |
10.1128/aac.00859-09 |
| Pseudomonas aeruginosa |
Beta-lactamase |
Kcat/Km |
2300.0 |
/uM/s |
10.1128/aac.01410-08 |
| Pseudomonas aeruginosa |
Beta-lactamase |
Km |
2000.0 |
nM |
10.1128/aac.00859-09 |
| Pseudomonas aeruginosa |
Beta-lactamase |
Km |
50000.0 |
nM |
10.1128/aac.01410-08 |
| Pseudomonas aeruginosa |
Beta-lactamase bla(BEL1) |
Kcat |
150.0 |
/s |
10.1128/aac.00859-09 |
| Pseudomonas aeruginosa |
Beta-lactamase bla(BEL1) |
Kcat/Km |
540.0 |
/mM/s |
10.1128/aac.00859-09 |
| Pseudomonas aeruginosa |
Beta-lactamase bla(BEL1) |
Km |
280000.0 |
nM |
10.1128/aac.00859-09 |
| Pseudomonas aeruginosa |
Beta-lactamase GES-13 |
Kcat |
10.1 |
/s |
10.1128/aac.01561-09 |
| Pseudomonas aeruginosa |
Beta-lactamase GES-13 |
Kcat/Km |
0.1 |
/uM/s |
10.1128/aac.01561-09 |
| Pseudomonas aeruginosa |
Beta-lactamase GES-13 |
Km |
106000.0 |
nM |
10.1128/aac.01561-09 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-1 |
Kcat |
449.0 |
/s |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-1 |
Kcat/Km |
3.3 |
/M/s |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-1 |
Km |
135000.0 |
nM |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Kcat |
130.0 |
/s |
10.1128/aac.00166-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Kcat/Km |
12.0 |
/uM/s |
10.1128/aac.00166-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Km |
11000.0 |
nM |
10.1128/aac.00166-08 |
| Pseudomonas aeruginosa |
Class B carbapenemase VIM-13 |
Kcat |
656.0 |
/s |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Class B carbapenemase VIM-13 |
Kcat/Km |
8.6 |
/M/s |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Class B carbapenemase VIM-13 |
Km |
76000.0 |
nM |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Metallo-beta-lactamase VIM-11 |
Kcat |
81.0 |
/s |
10.1128/aac.01025-07 |
| Pseudomonas aeruginosa |
Metallo-beta-lactamase VIM-11 |
Kcat/Km |
1.8 |
10'6/M/s |
10.1128/aac.01025-07 |
| Pseudomonas aeruginosa |
Metallo-beta-lactamase VIM-11 |
Km |
4500.0 |
nM |
10.1128/aac.01025-07 |
| Pseudomonas aeruginosa |
Metallo-beta-lactamase VIM-2 |
Kcat |
96.4 |
/s |
10.1128/aac.01025-07 |
| Pseudomonas aeruginosa |
Metallo-beta-lactamase VIM-2 |
Kcat/Km |
1.6 |
10'6/M/s |
10.1128/aac.01025-07 |
| Pseudomonas aeruginosa |
Metallo-beta-lactamase VIM-2 |
Km |
6200.0 |
nM |
10.1128/aac.01025-07 |
| Pseudomonas aeruginosa |
Metallo-b-lactamase |
Kcat |
180.0 |
/s |
10.1128/aac.00166-08 |
| Pseudomonas aeruginosa |
Metallo-b-lactamase |
Kcat/Km |
4.0 |
/uM/s |
10.1128/aac.00166-08 |
| Pseudomonas aeruginosa |
Metallo-b-lactamase |
Km |
45000.0 |
nM |
10.1128/aac.00166-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
nan |
None |
10.1021/jm00211a006 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
37.0 |
mm |
10.1016/j.ejmech.2011.03.045 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
37.0 |
mm |
10.1016/j.ejmech.2012.11.017 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2011.03.045 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2012.11.017 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00193a001 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00207a022 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
125.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
128.0 |
ug.mL-1 |
10.1021/jm00346a024 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
200.0 |
ug.mL-1 |
10.1021/jm00219a010 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00859-09 |
| Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) |
Beta-lactamase |
Kcat |
44.0 |
/s |
10.1128/aac.01410-08 |
| Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) |
Beta-lactamase |
Kcat/Km |
510.0 |
/uM/s |
10.1128/aac.01410-08 |
| Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) |
Beta-lactamase |
Km |
85000.0 |
nM |
10.1128/aac.01410-08 |
| Pseudomonas fluorescens |
Beta-lactamase |
Kcat/Km |
500.0 |
/mM/s |
10.1128/aac.00961-09 |
| Pseudomonas fluorescens |
Pseudomonas fluorescens |
IZ |
37.0 |
mm |
10.1007/s00044-012-0079-x |
| Pseudomonas fluorescens |
Pseudomonas fluorescens |
IZ |
37.0 |
mm |
10.1007/s00044-012-9978-0 |
| Pseudomonas fluorescens |
Pseudomonas fluorescens |
IZ |
37.0 |
mm |
10.1016/j.ejmech.2010.05.018 |
| Pseudomonas fluorescens |
Pseudomonas fluorescens |
MIC |
6.25 |
ug.mL-1 |
10.1007/s00044-012-9978-0 |
| Pseudomonas fluorescens |
Pseudomonas fluorescens |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2010.05.018 |
| Pseudomonas fluorescens |
Pseudomonas fluorescens |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00961-09 |
| Pseudomonas fluorescens |
Pseudomonas fluorescens |
MIC |
6250.0 |
ug.mL-1 |
10.1007/s00044-012-0079-x |
| Pseudomonas luteola |
Beta-lactamase |
Kcat |
543.0 |
/s |
10.1128/aac.00427-09 |
| Pseudomonas luteola |
Beta-lactamase |
Kcat/Km |
25.86 |
/s/microM |
10.1128/aac.00427-09 |
| Pseudomonas luteola |
Beta-lactamase |
Km |
21000.0 |
nM |
10.1128/aac.00427-09 |
| Pseudomonas savastanoi pv. phaseolicola |
Pseudomonas savastanoi pv. phaseolicola |
IZ |
38.0 |
mm |
10.1007/s00044-012-0079-x |
| Pseudomonas savastanoi pv. phaseolicola |
Pseudomonas savastanoi pv. phaseolicola |
MIC |
6250.0 |
ug.mL-1 |
10.1007/s00044-012-0079-x |
| Pseudomonas stutzeri |
Metallo-beta-lactamase |
Kcat |
30.0 |
/s |
10.1128/aac.01456-09 |
| Pseudomonas stutzeri |
Metallo-beta-lactamase |
Km |
6000.0 |
nM |
10.1128/aac.01456-09 |
| Pseudomonas stutzeri |
Metallo-beta-lactamase |
Ratio |
5000.0 |
None |
10.1128/aac.01456-09 |
| Rattus norvegicus |
Androgen Receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Cyclooxygenase-1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
GABA receptor alpha-1 subunit |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Glutamate (NMDA) receptor subunit zeta 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Oligopeptide transporter, kidney isoform |
Ki |
8300000.0 |
nM |
10.1016/j.ejpb.2004.07.008 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
28000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
29000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
30000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
31000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
32000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.1 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.2 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.3 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
899.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
967.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1007.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1075.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1157.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1210.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1218.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1231.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1283.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1293.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1313.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1320.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1321.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1347.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1371.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1381.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1382.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1398.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1407.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1413.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1425.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1462.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1472.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1511.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1513.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1549.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1558.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1568.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1573.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1605.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1638.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1655.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
29.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
30.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
33.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
36.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
37.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
37.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
38.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
38.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
39.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
39.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
40.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
41.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
42.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
42.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
43.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
44.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
44.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
44.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
46.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
48.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
49.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
52.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
53.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
21.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
21.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
21.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
21.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
21.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
21.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
22.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
22.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
22.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
22.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
22.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
22.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
22.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
22.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
23.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
23.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
23.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
23.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
23.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
24.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
24.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
24.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
24.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
24.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
25.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
26.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
57.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
58.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
62.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
63.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
64.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
64.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
66.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
68.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
69.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
69.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
71.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
72.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
72.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
75.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
76.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
76.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
77.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
78.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
78.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
80.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
81.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
85.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
87.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
90.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
91.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
94.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
95.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
101.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.02 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.04 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.02 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.04 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.06 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.08 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.1 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.12 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.16 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.18 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.2 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.22 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.28 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.3 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
0.34 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
92.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
96.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
100.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
104.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
110.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
120.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
122.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
124.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
126.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
128.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
156.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
158.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
160.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
162.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
166.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
168.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
170.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
172.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
176.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
178.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
180.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
182.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
186.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
196.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
102.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
103.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
104.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
105.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
106.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
107.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
108.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
109.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
110.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
606.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
608.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
616.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
624.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
640.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
648.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
656.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
664.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
674.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
676.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
678.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
682.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
688.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
692.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
698.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
704.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
706.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
712.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
720.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
736.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
744.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
746.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
750.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
758.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
792.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
806.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
852.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
106.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
106.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
106.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
106.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
107.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
107.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
107.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
107.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
1.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2576.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2608.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2666.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2682.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2692.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2746.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2776.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2786.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2792.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2794.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2816.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2838.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2840.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2908.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2912.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2914.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2924.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2932.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2938.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2944.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2946.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
3024.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
3030.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
3038.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
3054.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
3084.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
3098.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
3100.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
3114.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
3230.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
3392.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
3472.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
2.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
2.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
3.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1600.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1668.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1684.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1692.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1702.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1716.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1718.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1730.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1732.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1736.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1744.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1754.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1760.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1762.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1766.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1768.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1790.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1794.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1808.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1820.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1830.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1844.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1848.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1858.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1866.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1886.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1894.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1908.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
42.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
42.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
42.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
129000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
130000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
131000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
132000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
134000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
135000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
136000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
137000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
139000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
142000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
144000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
149000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
154000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
156000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
96.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
105.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
109.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
119.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
128.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
142.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
146.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
147.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
148.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
148.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
150.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
152.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
152.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
153.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
157.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
158.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
162.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
162.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
162.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
166.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
171.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
176.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
176.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
177.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
178.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
181.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
182.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
204.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
207.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
214.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
221.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
66.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
67.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
70.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
72.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
73.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
74.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
75.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
76.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
79.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
80.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
82.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
83.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
83.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
84.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
84.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
84.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
87.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
87.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
88.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
88.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
89.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
89.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
19.1 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
19.6 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
19.8 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.2 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.3 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.4 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.5 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.6 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.7 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.8 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.1 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.2 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.3 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
37.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
52.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
52.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
53.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
53.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
56.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
56.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
57.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
58.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
58.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
59.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
59.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
59.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.8 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
1.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
1.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
6.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
7.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
7.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
8.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
9.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
10.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
10.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
12.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
12.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
12.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
13.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
17.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
18.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
18.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
19.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
20.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
22.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
22.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
23.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
25.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
28.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
56.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
59.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
61.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
63.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
67.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
69.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
70.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
71.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
72.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
73.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
75.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
76.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
78.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
85.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
89.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
90.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
91.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
93.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
94.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
96.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1158.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1172.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1218.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1220.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1254.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1278.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1298.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1328.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1342.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1344.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1346.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1348.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1352.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1354.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1356.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1360.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1380.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1386.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1388.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1400.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1412.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1416.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1424.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1426.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1430.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1438.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1446.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1450.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1458.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1472.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1488.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1005000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1071000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1080000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1138000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1165000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1173000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1179000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1183000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1200000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1202000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1203000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1211000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1213000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1221000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1239000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1243000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1261000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1281000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1283000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1287000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1288000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1291000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1315000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1317000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1325000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1326000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1350000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1357000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1359000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1399000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.1 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.3 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.5 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
51000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
52000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
53000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
54000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
55000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
56000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
57000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
58000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
59000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
61000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
15.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
16.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
16.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
16.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
16.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
16.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
16.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
16.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
16.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
17.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6072000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6116000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6188000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6196000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6204000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6220000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6272000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6296000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6302000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6330000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6368000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6388000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6398000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6406000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6416000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6420000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6426000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6428000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6440000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6452000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6470000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6518000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6614000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6898000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6940000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6952000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6986000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7628000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7892000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7978000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
8054000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
3.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
143.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
143.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
208.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
210.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
211.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
212.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
213.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
214.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
214.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
214.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
214.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
215.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
217.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
218.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
219.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
223.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
225.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
226.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
226.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
230.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
233.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
236.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
255.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
260.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
261.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
261.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
294.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
302.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
304.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
318.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
341.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
376.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
376.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
378.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Tissue Severity Score |
nan |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
404.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
410.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
600.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
658.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
692.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
712.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
746.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
752.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
760.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
794.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
798.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
876.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
900.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
902.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
920.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
938.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
946.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
968.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1012.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1032.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1034.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1064.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1084.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1098.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1102.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1152.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1164.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1310.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1328.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1366.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1412.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1468.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
6320.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
6950.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7150.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7350.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7460.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7580.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7630.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7730.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7770.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7870.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8010.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8120.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8170.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8480.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8920.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8960.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9060.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9100.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9230.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9310.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9680.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9800.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9830.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10040.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10320.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10370.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10390.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10770.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10840.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10960.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11040.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11820.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
0.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
13.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Solute carrier family 22 member 6 |
Ki |
290000.0 |
nM |
None |
| Rattus norvegicus |
Solute carrier family 22 member 6 |
Ki |
530000.0 |
nM |
10.1016/s0024-3205(02)01500-x |
| Rattus norvegicus |
Solute carrier family 22 member 7 |
IC50 |
1500000.0 |
nM |
10.1016/s0014-2999(03)01381-5 |
| Rattus norvegicus |
Solute carrier family 22 member 8 |
Ki |
48000.0 |
nM |
10.1016/s0024-3205(02)01500-x |
| Rattus norvegicus |
Thioredoxin reductase 1, cytoplasmic |
Potency |
16833.6 |
nM |
None |
| Rattus norvegicus |
Thioredoxin reductase 1, cytoplasmic |
Potency |
44668.4 |
nM |
None |
| Salmonella |
Salmonella |
MIC |
0.8 |
ug.mL-1 |
10.1021/jm00207a022 |
| Salmonella |
Salmonella |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm00346a024 |
| Salmonella |
Salmonella |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00207a022 |
| Salmonella enterica subsp. enterica serovar Paratyphi A |
Salmonella paratyphi |
MIC |
0.8 |
ug.mL-1 |
10.1021/jm00219a010 |
| Salmonella enterica subsp. enterica serovar Paratyphi A |
Salmonella paratyphi |
MIC |
1.6 |
ug.mL-1 |
10.1021/jm00211a006 |
| Salmonella enterica subsp. enterica serovar Paratyphi A |
Salmonella paratyphi |
MIC |
1.6 |
ug.mL-1 |
10.1021/jm00228a003 |
| Salmonella enterica subsp. enterica serovar Typhi |
Salmonella typhi |
MIC |
12.5 |
ug.mL-1 |
10.1021/jm00218a018 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00600-06 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.00205-08 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00079-09 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00600-06 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00600-06 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00600-06 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00600-06 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00079-09 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00079-09 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
nan |
None |
10.1128/aac.01472-06 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
Ratio |
4.0 |
None |
10.1016/j.ejmech.2012.03.008 |
| Salmonella enterica subsp. enterica serovar Westhampton |
Extended-spectrum beta-lactamase CTX-M-53 |
Kcat |
2000.0 |
/s |
10.1128/aac.01581-08 |
| Salmonella enterica subsp. enterica serovar Westhampton |
Extended-spectrum beta-lactamase CTX-M-53 |
Kcat/Km |
16.4 |
/s/microM |
10.1128/aac.01581-08 |
| Salmonella enterica subsp. enterica serovar Westhampton |
Extended-spectrum beta-lactamase CTX-M-53 |
Km |
122000.0 |
nM |
10.1128/aac.01581-08 |
| Salmonella newport |
Efflux transporter |
Kcat |
150.0 |
/s |
10.1128/aac.01284-08 |
| Salmonella newport |
Efflux transporter |
Kcat/Km |
29.4 |
/uM/s |
10.1128/aac.01284-08 |
| Salmonella newport |
Efflux transporter |
Km |
5100.0 |
nM |
10.1128/aac.01284-08 |
| Serratia fonticola |
Carbapenem-hydrolizing beta-lactamase SFC-1 |
Kcat |
280.0 |
/s |
10.1128/aac.00491-07 |
| Serratia fonticola |
Carbapenem-hydrolizing beta-lactamase SFC-1 |
Kcat/Km |
2171.0 |
/mM/s |
10.1128/aac.00491-07 |
| Serratia fonticola |
Carbapenem-hydrolizing beta-lactamase SFC-1 |
Km |
129000.0 |
nM |
10.1128/aac.00491-07 |
| Serratia marcescens |
Serratia marcescens |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00193a001 |
| Serratia marcescens |
Serratia marcescens |
MIC |
125.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Serratia marcescens |
Serratia marcescens |
MIC |
125.0 |
ug.mL-1 |
10.1021/jm00375a026 |
| Serratia marcescens |
Serratia marcescens |
MIC |
453000.0 |
nM |
10.1021/jm00203a001 |
| Severe acute respiratory syndrome coronavirus 2 |
Replicase polyprotein 1ab |
Inhibition |
-8.837 |
% |
10.6019/CHEMBL4495564 |
| Severe acute respiratory syndrome coronavirus 2 |
Replicase polyprotein 1ab |
Inhibition |
-5.45 |
% |
10.6019/CHEMBL4495564 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Hit score |
0.1524 |
None |
10.1101/2020.04.21.054387 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
-3.82 |
% |
10.21203/rs.3.rs-23951/v1 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
0.04 |
% |
10.6019/CHEMBL4495565 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
0.06 |
% |
10.6019/CHEMBL4495565 |
| Shigella flexneri |
Shigella flexneri |
MIC |
6.2 |
ug.mL-1 |
10.1021/jm00228a003 |
| Shigella flexneri |
Shigella flexneri |
MIC |
6.3 |
ug.mL-1 |
10.1021/jm00211a006 |
| Shigella sonnei |
Shigella sonnei |
MIC |
5.0 |
ug.mL-1 |
10.1021/jm00218a018 |
| Shigella sp. |
Shigella sp. |
MIC |
14.0 |
ug.mL-1 |
10.1021/jm00217a021 |
| Shouchella clausii |
Shouchella clausii |
MIC |
8000.0 |
ug.mL-1 |
10.1128/aac.00537-07 |
| Staphylococcus aureus |
Beta-lactamase |
K cat |
0.001 |
s-1 |
10.1016/j.bmcl.2004.07.067 |
| Staphylococcus aureus |
Beta-lactamase |
Km |
1000.0 |
nM |
10.1016/j.bmcl.2004.07.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/jm00228a003 |
| Staphylococcus aureus |
Staphylococcus aureus |
Antibiotic resistance |
nan |
None |
10.1016/s0960-894x(98)00536-8 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
31.0 |
mm |
10.1016/j.bmcl.2016.05.053 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
36.0 |
mm |
10.1007/s00044-012-0079-x |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
36.0 |
mm |
10.1007/s00044-012-9978-0 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
36.0 |
mm |
10.1016/j.ejmech.2010.05.018 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.00025 |
ug.mL-1 |
10.1128/aac.01173-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.00038 |
ug.mL-1 |
10.1128/aac.01173-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.015 |
ug.mL-1 |
10.1021/jm00346a024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.05 |
ug.mL-1 |
10.1021/jm00193a001 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1021/jm00346a024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1021/jm00375a026 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm00207a022 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1021/jm00218a018 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.128 |
ug.mL-1 |
10.1128/aac.01173-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.13 |
ug.mL-1 |
10.1021/jm00192a025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.2 |
ug.mL-1 |
10.1021/jm00178a011 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.2 |
ug.mL-1 |
10.1021/jm00193a001 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.2 |
ug.mL-1 |
10.1021/jm00211a006 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.2 |
ug.mL-1 |
10.1021/jm00219a010 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.2 |
ug.mL-1 |
10.1021/jm00228a003 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.2 |
ug.mL-1 |
10.1128/aac.00718-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2010.05.110 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.256 |
ug.mL-1 |
10.1128/aac.01173-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.3 |
ug.mL-1 |
10.1021/jm00211a041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.3 |
ug.mL-1 |
10.1128/aac.01325-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.4 |
ug.mL-1 |
10.1021/jm00207a022 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.4 |
ug.mL-1 |
10.1128/aac.01325-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2010.05.110 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm00192a025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm00218a018 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm00375a026 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01325-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01472-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.6 |
ug.mL-1 |
10.1128/aac.01325-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.8 |
ug.mL-1 |
10.1021/jm00178a011 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01472-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.3 |
ug.mL-1 |
10.1128/aac.01325-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.9 |
ug.mL-1 |
10.1128/aac.01325-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm00375a026 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01325-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.01325-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6.25 |
ug.mL-1 |
10.1007/s00044-012-9978-0 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2010.05.018 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.05.110 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm00192a025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01472-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
200.0 |
nM |
10.1021/jm00203a001 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6250.0 |
ug.mL-1 |
10.1007/s00044-012-0079-x |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01325-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01325-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01325-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01325-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.4 |
ug.mL-1 |
10.1021/jm00207a022 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.03 |
ug.mL-1 |
10.1021/jm00375a026 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1021/jm00192a025 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm00178a011 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm00193a001 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm00207a022 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2010.05.110 |
| Streptococcus pneumoniae R6 |
Penicillin-binding protein 2X |
Activity |
nan |
None |
10.1021/jm900625q |
| Streptococcus pneumoniae serotype 4 (strain ATCC BAA-334 / TIGR4) |
Penicillin-binding protein 2x |
Activity |
nan |
None |
10.1021/jm900625q |
| Streptococcus pyogenes |
Streptococcus pyogenes |
IZ |
37.0 |
mm |
10.1007/s00044-012-0079-x |
| Streptococcus pyogenes |
Streptococcus pyogenes |
IZ |
37.0 |
mm |
10.1007/s00044-012-9978-0 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
IZ |
37.0 |
mm |
10.1016/j.ejmech.2010.05.018 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.06 |
ug.mL-1 |
10.1021/jm00375a026 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm00178a011 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm00207a022 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm00211a041 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.13 |
ug.mL-1 |
10.1021/jm00192a025 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
6.25 |
ug.mL-1 |
10.1007/s00044-012-9978-0 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2010.05.018 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
6250.0 |
ug.mL-1 |
10.1007/s00044-012-0079-x |
| Trypanosoma brucei |
6-phospho-1-fructokinase |
Potency |
8492.1 |
nM |
None |
| Trypanosoma brucei brucei |
Phosphoglycerate kinase, glycosomal |
Potency |
35481.3 |
nM |
None |
| None |
ADMET |
CL |
1.8 |
mL.min-1.kg-1 |
10.1124/dmd.108.020479 |
| None |
ADMET |
Cp |
8.6 |
mg/L |
10.1128/aac.00718-08 |
| None |
ADMET |
Cp |
8.9 |
mg/L |
10.1128/aac.00718-08 |
| None |
ADMET |
Cp |
14.5 |
mg/L |
10.1128/aac.00718-08 |
| None |
ADMET |
Drug metabolism |
0.0 |
% |
10.1021/acs.jmedchem.8b01923 |
| None |
ADMET |
Drug uptake |
0.54 |
mg/L |
10.1128/aac.00718-08 |
| None |
ADMET |
Drug uptake |
2.84 |
mg/L |
10.1128/aac.00718-08 |
| None |
ADMET |
Drug uptake |
3.06 |
mg/L |
10.1128/aac.00718-08 |
| None |
ADMET |
k |
0.317 |
hr-1 |
10.1021/jm00401a026 |
| None |
ADMET |
k cat |
0.001 |
s-1 |
10.1016/s0960-894x(98)00739-2 |
| None |
ADMET |
k cat |
120.0 |
s-1 |
10.1016/s0960-894x(98)00739-2 |
| None |
ADMET |
k cat |
200.0 |
s-1 |
10.1016/s0960-894x(98)00739-2 |
| None |
ADMET |
Km |
1000.0 |
nM |
10.1016/s0960-894x(98)00739-2 |
| None |
ADMET |
Km |
9000.0 |
nM |
10.1016/s0960-894x(98)00739-2 |
| None |
ADMET |
Km |
200000.0 |
nM |
10.1016/s0960-894x(98)00739-2 |
| None |
ADMET |
MRT |
0.65 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
Ratio |
1000.0 |
M-1 s-1 |
10.1016/s0960-894x(98)00739-2 |
| None |
ADMET |
Ratio |
600000.0 |
M-1 s-1 |
10.1016/s0960-894x(98)00739-2 |
| None |
ADMET |
Ratio |
22000000.0 |
M-1 s-1 |
10.1016/s0960-894x(98)00739-2 |
| None |
ADMET |
T1/2 |
0.95 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
T1/2 |
1.1 |
hr |
10.1021/jm00400a015 |
| None |
ADMET |
T1/2 |
29.0 |
hr |
10.1021/jm00400a015 |
| None |
ADMET |
Vdss |
0.07 |
L.kg-1 |
10.1124/dmd.108.020479 |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1021/tx900326k |
| None |
NON-PROTEIN TARGET |
Fu |
0.22 |
None |
10.1124/dmd.108.020479 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (acute) |
0.0 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (animal toxicity known) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (benign tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (granulomatous hepatitis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (mechanism) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
1.5 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
4.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (time to onset) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00791-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00791-09 |
| None |
NON-PROTEIN TARGET |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm00217a021 |
| None |
NON-PROTEIN TARGET |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01152-06 |
| None |
NON-PROTEIN TARGET |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
MIC |
3.1 |
ug.mL-1 |
10.1021/jm00178a011 |
| None |
NON-PROTEIN TARGET |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01615-09 |
| None |
NON-PROTEIN TARGET |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01585-09 |
| None |
NON-PROTEIN TARGET |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01463-07 |
| None |
NON-PROTEIN TARGET |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00427-09 |
| None |
NON-PROTEIN TARGET |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00791-09 |
| None |
NON-PROTEIN TARGET |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01463-07 |
| None |
NON-PROTEIN TARGET |
MIC |
96.0 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00427-09 |
| None |
NON-PROTEIN TARGET |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01252-09 |
| None |
NON-PROTEIN TARGET |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01600-06 |
| None |
NON-PROTEIN TARGET |
MIC50 |
256.0 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
MIC90 |
256.0 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
T>MIC |
160.0 |
min |
10.1128/aac.00718-08 |
| None |
NON-PROTEIN TARGET |
T>MIC |
285.0 |
min |
10.1128/aac.00718-08 |
| None |
NON-PROTEIN TARGET |
T>MIC |
336.0 |
min |
10.1128/aac.00718-08 |
| None |
No relevant target |
K |
9.7 |
10'5/s |
10.1021/jm00217a021 |
| None |
No relevant target |
Solubility |
457.0 |
ug.mL-1 |
10.1016/j.bmc.2010.08.003 |
| None |
Unchecked |
Ac50 |
5.012 |
uM |
None |
| None |
Unchecked |
Ac50 |
15.85 |
uM |
None |
| None |
Unchecked |
AC50 |
5011.9 |
nM |
None |
| None |
Unchecked |
AC50 |
15848.9 |
nM |
None |
| None |
Unchecked |
Activity |
0.04 |
% |
10.1128/aac.01164-08 |
| None |
Unchecked |
Activity |
0.1 |
% |
10.1128/aac.00684-07 |
| None |
Unchecked |
Activity |
1.6 |
% |
10.1128/aac.01164-08 |
| None |
Unchecked |
Activity |
5.4 |
umol |
10.1128/aac.01025-07 |
| None |
Unchecked |
Activity |
6.0 |
None |
10.1128/aac.01439-06 |
| None |
Unchecked |
Activity |
10.0 |
mU |
10.1128/aac.00978-07 |
| None |
Unchecked |
Activity |
15.0 |
mU |
10.1128/aac.00978-07 |
| None |
Unchecked |
Activity |
20.0 |
mU |
10.1128/aac.00978-07 |
| None |
Unchecked |
Activity |
nan |
None |
10.1128/aac.00978-07 |
| None |
Unchecked |
Drug metabolism |
61.0 |
% |
10.1021/acs.jmedchem.8b01923 |
| None |
Unchecked |
Drug metabolism |
68.0 |
% |
10.1021/acs.jmedchem.8b01923 |
| None |
Unchecked |
Drug metabolism |
100.0 |
% |
10.1021/acs.jmedchem.8b01923 |
| None |
Unchecked |
FC |
2.7 |
None |
10.1128/aac.00197-10 |
| None |
Unchecked |
FC |
100.0 |
None |
10.1128/aac.00537-07 |
| None |
Unchecked |
Hepatotoxicity (acute) |
4.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (association with vascular disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (choleostasis) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (chronic liver disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cirrhosis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (comment) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cytolytic) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (malignant tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (severe hepatitis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (steatosis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (successful reintroduction) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
IC50 |
99000.0 |
nM |
None |
| None |
Unchecked |
Inhibition |
nan |
% |
10.1016/j.ejmech.2022.114174 |
| None |
Unchecked |
Kcat |
0.1 |
/s |
10.1128/aac.00387-08 |
| None |
Unchecked |
Kcat |
0.1 |
/s |
10.1128/aac.01145-07 |
| None |
Unchecked |
Kcat |
0.1 |
/s |
10.1128/aac.01600-06 |
| None |
Unchecked |
Kcat |
0.2 |
/s |
10.1128/aac.00856-09 |
| None |
Unchecked |
Kcat |
0.3 |
/s |
10.1128/aac.01164-08 |
| None |
Unchecked |
Kcat |
0.4 |
/s |
10.1128/aac.00858-10 |
| None |
Unchecked |
Kcat |
0.5 |
/s |
10.1128/aac.01463-07 |
| None |
Unchecked |
Kcat |
2.94 |
/s |
10.1128/aac.00771-10 |
| None |
Unchecked |
Kcat |
4.0 |
/s |
10.1128/aac.01058-06 |
| None |
Unchecked |
Kcat |
4.0 |
/s |
10.1128/aac.01442-09 |
| None |
Unchecked |
Kcat |
4.1 |
/s |
10.1128/aac.00684-07 |
| None |
Unchecked |
Kcat |
4.6 |
/s |
10.1021/jm301490d |
| None |
Unchecked |
Kcat |
10.0 |
/s |
10.1128/aac.00608-08 |
| None |
Unchecked |
Kcat |
10.1 |
/s |
10.1128/aac.00771-10 |
| None |
Unchecked |
Kcat |
15.0 |
/s |
10.1128/aac.01058-06 |
| None |
Unchecked |
Kcat |
18.4 |
/s |
10.1128/aac.01058-06 |
| None |
Unchecked |
Kcat |
21.2 |
/s |
10.1128/aac.00017-09 |
| None |
Unchecked |
Kcat |
26.0 |
/s |
10.1128/aac.00197-10 |
| None |
Unchecked |
Kcat |
32.0 |
/s |
10.1128/aac.01336-09 |
| None |
Unchecked |
Kcat |
42.6 |
/s |
10.1021/jm301490d |
| None |
Unchecked |
Kcat |
46.0 |
/s |
10.1128/aac.00614-07 |
| None |
Unchecked |
Kcat |
48.0 |
/s |
10.1128/aac.00774-09 |
| None |
Unchecked |
Kcat |
52.0 |
/s |
10.1128/aac.00614-07 |
| None |
Unchecked |
Kcat |
65.0 |
/s |
10.1128/aac.00197-10 |
| None |
Unchecked |
Kcat |
65.0 |
/s |
10.1128/aac.00608-08 |
| None |
Unchecked |
Kcat |
106.0 |
/s |
10.1128/aac.00163-08 |
| None |
Unchecked |
Kcat |
110.0 |
/s |
10.1128/aac.01410-08 |
| None |
Unchecked |
Kcat |
120.0 |
/s |
10.1128/aac.01410-08 |
| None |
Unchecked |
Kcat |
126.0 |
/s |
10.1128/aac.01058-06 |
| None |
Unchecked |
Kcat |
135.0 |
/s |
10.1128/aac.01336-09 |
| None |
Unchecked |
Kcat |
160.0 |
/s |
10.1128/aac.01284-08 |
| None |
Unchecked |
Kcat |
165.0 |
/s |
10.1128/aac.01058-06 |
| None |
Unchecked |
Kcat |
167.0 |
/s |
10.1128/aac.00771-10 |
| None |
Unchecked |
Kcat |
180.0 |
/s |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat |
185.0 |
/s |
10.1128/aac.00227-08 |
| None |
Unchecked |
Kcat |
194.0 |
/s |
10.1128/aac.01058-06 |
| None |
Unchecked |
Kcat |
200.0 |
/s |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat |
218.0 |
/s |
10.1128/aac.00771-10 |
| None |
Unchecked |
Kcat |
240.0 |
/s |
10.1128/aac.01062-07 |
| None |
Unchecked |
Kcat |
250.0 |
/s |
10.1128/aac.00961-09 |
| None |
Unchecked |
Kcat |
250.0 |
/s |
10.1128/aac.01336-09 |
| None |
Unchecked |
Kcat |
256.0 |
/s |
10.1128/aac.00219-09 |
| None |
Unchecked |
Kcat |
260.0 |
/s |
10.1128/aac.00771-10 |
| None |
Unchecked |
Kcat |
267.0 |
/s |
10.1128/aac.00219-09 |
| None |
Unchecked |
Kcat |
280.0 |
/s |
10.1128/aac.00166-08 |
| None |
Unchecked |
Kcat |
300.0 |
/s |
10.1128/aac.01252-09 |
| None |
Unchecked |
Kcat |
313.0 |
/s |
10.1128/aac.00771-10 |
| None |
Unchecked |
Kcat |
320.0 |
/s |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat |
370.0 |
/s |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat |
410.0 |
/s |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat |
470.0 |
/s |
10.1128/aac.01252-09 |
| None |
Unchecked |
Kcat |
500.0 |
/s |
10.1128/aac.00608-08 |
| None |
Unchecked |
Kcat |
540.0 |
/s |
10.1128/aac.00608-08 |
| None |
Unchecked |
Kcat |
540.0 |
/s |
10.1128/aac.01252-09 |
| None |
Unchecked |
Kcat |
620.0 |
/s |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat |
690.0 |
/s |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat |
780.0 |
/s |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat/Km |
0.001 |
/s/microM |
10.1128/aac.00856-09 |
| None |
Unchecked |
Kcat/Km |
0.006 |
/uM/s |
10.1128/aac.01164-08 |
| None |
Unchecked |
Kcat/Km |
0.02 |
/uM/s |
10.1128/aac.01058-06 |
| None |
Unchecked |
Kcat/Km |
0.02 |
/uM/s |
10.1128/aac.01442-09 |
| None |
Unchecked |
Kcat/Km |
0.02 |
None |
10.1128/aac.00614-07 |
| None |
Unchecked |
Kcat/Km |
0.04 |
/uM/s |
10.1128/aac.01058-06 |
| None |
Unchecked |
Kcat/Km |
0.04 |
None |
10.1128/aac.00614-07 |
| None |
Unchecked |
Kcat/Km |
0.05 |
/uM/s |
10.1128/aac.00771-10 |
| None |
Unchecked |
Kcat/Km |
0.05 |
/uM/s |
10.1128/aac.01058-06 |
| None |
Unchecked |
Kcat/Km |
0.06 |
None |
10.1128/aac.01145-07 |
| None |
Unchecked |
Kcat/Km |
0.1 |
/uM/s |
10.1128/aac.00771-10 |
| None |
Unchecked |
Kcat/Km |
0.16 |
/uM/s |
10.1021/jm301490d |
| None |
Unchecked |
Kcat/Km |
0.2 |
/mM/s |
10.1128/aac.00608-08 |
| None |
Unchecked |
Kcat/Km |
0.31 |
uM/hr |
10.1128/aac.01336-09 |
| None |
Unchecked |
Kcat/Km |
0.5 |
/uM/s |
10.1128/aac.00050-10 |
| None |
Unchecked |
Kcat/Km |
0.61 |
/uM/s |
10.1128/aac.01058-06 |
| None |
Unchecked |
Kcat/Km |
0.67 |
/uM/s |
10.1128/aac.01058-06 |
| None |
Unchecked |
Kcat/Km |
0.7 |
/uM/s |
10.1128/aac.01058-06 |
| None |
Unchecked |
Kcat/Km |
0.87 |
/uM/s |
10.1021/jm301490d |
| None |
Unchecked |
Kcat/Km |
0.9 |
/uM/s |
10.1128/aac.00197-10 |
| None |
Unchecked |
Kcat/Km |
1.0 |
10'7/M/s |
10.1128/aac.01252-09 |
| None |
Unchecked |
Kcat/Km |
1.1 |
10'6/M/s |
10.1128/aac.01252-09 |
| None |
Unchecked |
Kcat/Km |
1.12 |
/s/M |
10.1128/aac.01025-07 |
| None |
Unchecked |
Kcat/Km |
1.2 |
10'6/M/s |
10.1128/aac.01062-07 |
| None |
Unchecked |
Kcat/Km |
1.2 |
10'6/s/M |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat/Km |
1.4 |
/s/microM |
10.1128/aac.00017-09 |
| None |
Unchecked |
Kcat/Km |
2.4 |
10'6/M/s |
10.1128/aac.00858-10 |
| None |
Unchecked |
Kcat/Km |
2.4 |
/s/microM |
10.1128/aac.00774-09 |
| None |
Unchecked |
Kcat/Km |
2.48 |
/uM/s |
10.1128/aac.00771-10 |
| None |
Unchecked |
Kcat/Km |
2.5 |
10'6/M/s |
10.1128/aac.00409-10 |
| None |
Unchecked |
Kcat/Km |
2.73 |
/uM/s |
10.1128/aac.00771-10 |
| None |
Unchecked |
Kcat/Km |
2.8 |
10'6/s/M |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat/Km |
3.3 |
10'6/s/M |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat/Km |
3.6 |
/uM/s |
10.1128/aac.00197-10 |
| None |
Unchecked |
Kcat/Km |
4.0 |
10'6/M/s |
10.1128/aac.00858-10 |
| None |
Unchecked |
Kcat/Km |
4.0 |
10'6/s/M |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat/Km |
4.0 |
/mM/s |
10.1128/aac.01145-07 |
| None |
Unchecked |
Kcat/Km |
4.1 |
10'6/s/M |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat/Km |
4.8 |
10'6/s/M |
10.1128/aac.00098-10 |
| None |
Unchecked |
Kcat/Km |
4.81 |
/uM/s |
10.1128/aac.00771-10 |
| None |
Unchecked |
Kcat/Km |
4.9 |
10'6/M/s |
10.1128/aac.00227-08 |
| None |
Unchecked |
Kcat/Km |
5.0 |
/uM/s |
10.1128/aac.00387-08 |
| None |
Unchecked |
Kcat/Km |
5.1 |
/uM/s |
10.1128/aac.00166-08 |
| None |
Unchecked |
Kcat/Km |
5.8 |
10'5/M/s |
10.1128/aac.00409-10 |
| None |
Unchecked |
Kcat/Km |
5.8 |
10'5/M/s |
10.1128/aac.01062-07 |
| None |
Unchecked |
Kcat/Km |
6.0 |
/mM/s |
10.1128/aac.00608-08 |
| None |
Unchecked |
Kcat/Km |
6.4 |
uM/hr |
10.1128/aac.01336-09 |
| None |
Unchecked |
Kcat/Km |
6.7 |
10'5/M/s |
10.1128/aac.00409-10 |
| None |
Unchecked |
Kcat/Km |
7.0 |
10'6/M/s |
10.1128/aac.01252-09 |
| None |
Unchecked |
Kcat/Km |
8.7 |
10'5/M/s |
10.1128/aac.00684-07 |
| None |
Unchecked |
Kcat/Km |
9.2 |
10'6/M/s |
10.1128/aac.00409-10 |
| None |
Unchecked |
Kcat/Km |
10.0 |
/uM/s |
10.1128/aac.00219-09 |
| None |
Unchecked |
Kcat/Km |
12.0 |
/mM/s |
10.1128/aac.00608-08 |
| None |
Unchecked |
Kcat/Km |
13.2 |
/uM/s |
10.1128/aac.00771-10 |
| None |
Unchecked |
Kcat/Km |
16.0 |
/mM/s |
10.1128/aac.00608-08 |
| None |
Unchecked |
Kcat/Km |
16.0 |
/uM/s |
10.1128/aac.00219-09 |
| None |
Unchecked |
Kcat/Km |
22.0 |
uM/hr |
10.1128/aac.01336-09 |
| None |
Unchecked |
Kcat/Km |
32.0 |
/uM/s |
10.1128/aac.01284-08 |
| None |
Unchecked |
Kcat/Km |
90.0 |
/mM/s |
10.1128/aac.01082-06 |
| None |
Unchecked |
Kcat/Km |
670.0 |
/uM/s |
10.1128/aac.01585-09 |
| None |
Unchecked |
Kcat/Km |
750.0 |
/mM/s |
10.1128/aac.00961-09 |
| None |
Unchecked |
Kcat/Km |
750.0 |
/uM/s |
10.1128/aac.00163-08 |
| None |
Unchecked |
Kcat/Km |
2200.0 |
/uM/s |
10.1128/aac.01410-08 |
| None |
Unchecked |
Kcat/Km |
2750.0 |
/uM/s |
10.1128/aac.01410-08 |
| None |
Unchecked |
Ki |
0.5 |
/M/s |
10.1021/ml400408c |
| None |
Unchecked |
Ki |
320.0 |
nM |
10.1016/j.bmc.2007.10.075 |
| None |
Unchecked |
Ki |
320.0 |
nM |
10.1039/C0MD00119H |
| None |
Unchecked |
Km |
100.0 |
nM |
10.1128/aac.00858-10 |
| None |
Unchecked |
Km |
327.0 |
/s/microM |
10.1128/aac.00614-07 |
| None |
Unchecked |
Km |
1200.0 |
/s/microM |
10.1128/aac.00614-07 |
| None |
Unchecked |
Km |
5000.0 |
nM |
10.1128/aac.01284-08 |
| None |
Unchecked |
Km |
5000.0 |
nM |
10.1128/aac.01336-09 |
| None |
Unchecked |
Km |
6000.0 |
nM |
10.1128/aac.01336-09 |
| None |
Unchecked |
Km |
8900.0 |
nM |
10.1128/aac.00409-10 |
| None |
Unchecked |
Km |
15000.0 |
nM |
10.1128/aac.01463-07 |
| None |
Unchecked |
Km |
17000.0 |
nM |
10.1128/aac.00219-09 |
| None |
Unchecked |
Km |
18000.0 |
nM |
10.1128/aac.00197-10 |
| None |
Unchecked |
Km |
20000.0 |
nM |
10.1128/aac.00387-08 |
| None |
Unchecked |
Km |
21000.0 |
nM |
10.1128/aac.00774-09 |
| None |
Unchecked |
Km |
21000.0 |
nM |
10.1128/aac.00858-10 |
| None |
Unchecked |
Km |
23700.0 |
nM |
10.1128/aac.00771-10 |
| None |
Unchecked |
Km |
24000.0 |
nM |
10.1128/aac.00409-10 |
| None |
Unchecked |
Km |
24000.0 |
nM |
10.1128/aac.01145-07 |
| None |
Unchecked |
Km |
26000.0 |
nM |
10.1128/aac.00219-09 |
| None |
Unchecked |
Km |
29000.0 |
nM |
10.1021/jm301490d |
| None |
Unchecked |
Km |
30000.0 |
nM |
10.1128/aac.00197-10 |
| None |
Unchecked |
Km |
37900.0 |
nM |
10.1128/aac.00227-08 |
| None |
Unchecked |
Km |
42000.0 |
nM |
10.1128/aac.01252-09 |
| None |
Unchecked |
Km |
45000.0 |
nM |
10.1128/aac.01252-09 |
| None |
Unchecked |
Km |
45000.0 |
nM |
10.1128/aac.01410-08 |
| None |
Unchecked |
Km |
47000.0 |
nM |
10.1128/aac.00684-07 |
| None |
Unchecked |
Km |
48900.0 |
nM |
10.1021/jm301490d |
| None |
Unchecked |
Km |
50000.0 |
nM |
10.1128/aac.01164-08 |
| None |
Unchecked |
Km |
50000.0 |
nM |
10.1128/aac.01410-08 |
| None |
Unchecked |
Km |
53900.0 |
nM |
10.1128/aac.00771-10 |
| None |
Unchecked |
Km |
54000.0 |
nM |
10.1128/aac.00771-10 |
| None |
Unchecked |
Km |
55000.0 |
nM |
10.1128/aac.00166-08 |
| None |
Unchecked |
Km |
61100.0 |
nM |
10.1128/aac.00771-10 |
| None |
Unchecked |
Km |
70000.0 |
nM |
10.1128/aac.00098-10 |
| None |
Unchecked |
Km |
77000.0 |
nM |
10.1128/aac.00098-10 |
| None |
Unchecked |
Km |
87800.0 |
nM |
10.1128/aac.00771-10 |
| None |
Unchecked |
Km |
98000.0 |
nM |
10.1128/aac.00098-10 |
| None |
Unchecked |
Km |
106000.0 |
nM |
10.1128/aac.00771-10 |
| None |
Unchecked |
Km |
120000.0 |
nM |
10.1128/aac.00098-10 |
| None |
Unchecked |
Km |
120000.0 |
nM |
10.1128/aac.00409-10 |
| None |
Unchecked |
Km |
120000.0 |
nM |
10.1128/aac.01600-06 |
| None |
Unchecked |
Km |
140000.0 |
nM |
10.1128/aac.00098-10 |
| None |
Unchecked |
Km |
141000.0 |
nM |
10.1128/aac.00163-08 |
| None |
Unchecked |
Km |
150000.0 |
nM |
10.1128/aac.00098-10 |
| None |
Unchecked |
Km |
169000.0 |
nM |
10.1128/aac.01442-09 |
| None |
Unchecked |
Km |
170000.0 |
nM |
10.1128/aac.00098-10 |
| None |
Unchecked |
Km |
200000.0 |
nM |
10.1128/aac.00098-10 |
| None |
Unchecked |
Km |
200000.0 |
nM |
10.1128/aac.01062-07 |
| None |
Unchecked |
Km |
205000.0 |
nM |
10.1128/aac.01058-06 |
| None |
Unchecked |
Km |
220000.0 |
nM |
10.1128/aac.00856-09 |
| None |
Unchecked |
Km |
230000.0 |
nM |
10.1128/aac.00409-10 |
| None |
Unchecked |
Km |
242000.0 |
nM |
10.1128/aac.01058-06 |
| None |
Unchecked |
Km |
260000.0 |
nM |
10.1128/aac.01058-06 |
| None |
Unchecked |
Km |
288000.0 |
nM |
10.1128/aac.01058-06 |
| None |
Unchecked |
Km |
330000.0 |
nM |
10.1128/aac.01058-06 |
| None |
Unchecked |
Km |
335000.0 |
nM |
10.1128/aac.01058-06 |
| None |
Unchecked |
Km |
400000.0 |
nM |
10.1128/aac.01082-06 |
| None |
Unchecked |
Km |
500000.0 |
nM |
10.1128/aac.01252-09 |
| None |
Unchecked |
Km |
500000.0 |
nM |
10.1128/aac.01336-09 |
| None |
Unchecked |
Km |
550000.0 |
nM |
10.1128/aac.00961-09 |
| None |
Unchecked |
Km |
5500000.0 |
nM |
10.1128/aac.00608-08 |
| None |
Unchecked |
Km |
30000000.0 |
nM |
10.1128/aac.00608-08 |
| None |
Unchecked |
Km |
45000000.0 |
nM |
10.1128/aac.00608-08 |
| None |
Unchecked |
Km |
85000000.0 |
nM |
10.1128/aac.00608-08 |
| None |
Unchecked |
Km |
nan |
None |
10.1128/aac.00389-07 |
| None |
Unchecked |
Potency |
562.3 |
nM |
None |
| None |
Unchecked |
Ratio |
1.0 |
/mM/s |
10.1128/aac.01600-06 |
| None |
Unchecked |
Ratio |
4.0 |
None |
10.1128/aac.00614-07 |
| None |
Unchecked |
Ratio |
30.0 |
None |
10.1128/aac.01463-07 |
| None |
Unchecked |
Ratio |
176.0 |
None |
10.1128/aac.00614-07 |
| None |
Unchecked |
Ratio |
1000.0 |
1/sM |
10.1016/j.bmcl.2004.07.067 |
| None |
Unchecked |
Ratio |
86000.0 |
1/sM |
10.1016/j.bmcl.2004.07.067 |
| None |
Unchecked |
Ratio |
600000.0 |
1/sM |
10.1016/j.bmcl.2004.07.067 |
| None |
Unchecked |
Ratio |
22000000.0 |
1/sM |
10.1016/j.bmcl.2004.07.067 |
| None |
Unchecked |
Selectivity ratio |
2.0 |
None |
10.1021/acs.jmedchem.8b01923 |
| None |
Unchecked |
T |
96.0 |
min |
10.1128/aac.00718-08 |
| None |
Unchecked |
T |
191.0 |
min |
10.1128/aac.00718-08 |
| None |
Unchecked |
T |
219.0 |
min |
10.1128/aac.00718-08 |
| None |
Unchecked |
Vmax |
nan |
None |
10.1128/aac.00389-07 |
| None |
Unchecked |
Vmax/Km |
nan |
None |
10.1128/aac.00389-07 |