| Acinetobacter |
Acinetobacter |
Activity |
0.0 |
% |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
Activity |
0.4 |
% |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
Activity |
1.4 |
% |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
Activity |
1.7 |
% |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
Activity |
18.0 |
% |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
Activity |
80.6 |
% |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
Activity |
97.9 |
% |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
Activity |
100.0 |
% |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116142 |
| Acinetobacter |
Acinetobacter |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116142 |
| Acinetobacter |
Acinetobacter |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
MIC50 |
32.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Acinetobacter |
Acinetobacter |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
0.0 |
% |
10.1128/aac.00400-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
4.0 |
% |
10.1128/aac.01099-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
8.0 |
% |
10.1128/aac.00400-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
12.0 |
% |
10.1128/aac.01533-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
22.4 |
% |
10.1128/aac.00570-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
22.9 |
% |
10.1128/aac.00264-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
77.1 |
% |
10.1128/aac.00264-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
92.0 |
% |
10.1128/aac.00400-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
nan |
None |
10.1128/aac.00748-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
nan |
None |
10.1128/aac.00764-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
nan |
None |
10.1128/aac.00963-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
nan |
None |
10.1128/aac.01525-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
nan |
None |
10.1128/aac.01533-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
ED90 |
25.0 |
mg kg-1 |
10.1021/acs.jmedchem.8b00091 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
ED90 |
50.0 |
mg kg-1 |
10.1021/acs.jmedchem.8b00091 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
FC |
0.1 |
None |
10.1021/jm501050e |
| Acinetobacter baumannii |
Acinetobacter baumannii |
FC |
2.0 |
None |
10.1128/aac.01512-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
FICI |
0.281 |
None |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
FICI |
0.5 |
None |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Inhibition |
10.36 |
% |
10.6019/CHEMBL4513141 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Inhibition |
100.0 |
% |
10.1021/acs.jmedchem.2c01905 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.00072-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.094 |
ug.mL-1 |
10.1128/aac.01198-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00570-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01198-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.00598-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.00856-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.8b00091 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm400560z |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1021/ml200012f |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1039/C5MD00377F |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00050-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00393-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00491-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00598-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00978-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01198-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01398-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01684-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.01512-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.01684-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00746 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00264-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00393-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00491-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01407-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01512-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01663-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.01198-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.01512-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.01684-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.0 |
ug.mL-1 |
10.1039/C5MD00377F |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00050-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00178-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01198-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01433-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.00072-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.01512-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.01684-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1039/C5MD00377F |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00050-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00267-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00978-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01139-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01198-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01684-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.01512-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.01663-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00267-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00292-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00366-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01198-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01512-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01684-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.00072-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.00570-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.01512-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.01663-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1039/C5MD00377F |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00072-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00292-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00491-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00838-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01512-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01799-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.00292-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.01684-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmc.2013.09.041 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.014 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01905 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b00091 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00292-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00393-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00491-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00978-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01259-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01398-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01414-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01512-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01684-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
24.0 |
ug.mL-1 |
10.1128/aac.00292-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
24.0 |
ug.mL-1 |
10.1128/aac.00861-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
24.0 |
ug.mL-1 |
10.1128/aac.01684-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm501050e |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00267-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00292-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00393-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00598-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00856-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01121-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01259-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01464-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01512-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01684-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01261 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b00091 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00292-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00978-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01259-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00178-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01259-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00178-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
500.0 |
ug.mL-1 |
10.1128/aac.01502-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
3000.0 |
ug.mL-1 |
10.1128/aac.01502-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4000.0 |
ug.mL-1 |
10.1128/aac.01502-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8000.0 |
ug.mL-1 |
10.1128/aac.01502-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
12000.0 |
ug.mL-1 |
10.1128/aac.01502-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32000.0 |
nM |
10.1021/acs.jmedchem.1c00621 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC50 |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113436 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00366-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.01099-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC50 |
32.0 |
ug.mL-1 |
10.1128/aac.00264-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC50 |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113436 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00366-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.07.005 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113436 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00264-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
128.0 |
ug.mL-1 |
10.1128/aac.01099-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MPC |
1.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MPC |
2.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MPC |
4.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MPC |
8.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MPC |
16.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MPC |
32.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MPC |
128.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
PD50 |
25.0 |
mg kg-1 |
10.1021/acs.jmedchem.8b00091 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
PD50 |
50.0 |
mg kg-1 |
10.1021/acs.jmedchem.8b00091 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Ratio |
2.0 |
None |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Ratio |
4.0 |
None |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Ratio |
8.0 |
None |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Ratio |
16.0 |
None |
10.1128/aac.00033-10 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Ratio |
64.0 |
None |
10.1128/aac.00491-10 |
| Acinetobacter baumannii |
Beta-lactamase OXA-23 |
Activity |
0.029 |
% |
10.1128/aac.01004-09 |
| Acinetobacter baumannii |
Beta-lactamase OXA-23 |
Activity |
10.0 |
% |
10.1128/aac.01004-09 |
| Acinetobacter baumannii |
Beta-lactamase OXA-23 |
Activity |
14.9 |
% |
10.1128/aac.01004-09 |
| Acinetobacter baumannii |
Beta-lactamase OXA-23 |
Activity |
140.0 |
% |
10.1128/aac.01004-09 |
| Acinetobacter baumannii |
Beta-lactamase OXA-23 |
Kcat |
0.13 |
nmol/min |
10.1128/aac.01004-09 |
| Acinetobacter baumannii |
Beta-lactamase OXA-23 |
Kcat |
170.0 |
/s |
10.1128/aac.01004-09 |
| Acinetobacter baumannii |
Beta-lactamase OXA-23 |
Kcat/Km |
0.052 |
/s/microM |
10.1128/aac.01004-09 |
| Acinetobacter baumannii |
Beta-lactamase OXA-23 |
Kcat/Km |
1.3 |
/s/microM |
10.1128/aac.01004-09 |
| Acinetobacter baumannii |
Beta-lactamase OXA-23 |
Km |
2500.0 |
nM |
10.1128/aac.01004-09 |
| Acinetobacter baumannii |
Beta-lactamase OXA-23 |
Km |
130000.0 |
nM |
10.1128/aac.01004-09 |
| Acinetobacter baylyi |
Acinetobacter baylyi |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01674-09 |
| Acinetobacter baylyi |
Acinetobacter baylyi |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01674-09 |
| Acinetobacter calcoaceticus |
Acinetobacter calcoaceticus |
MIC |
0.5 |
ug.mL-1 |
10.1016/S0960-894X(97)00282-5 |
| Acinetobacter calcoaceticus |
Acinetobacter calcoaceticus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.031 |
| Acinetobacter calcoaceticus |
Acinetobacter calcoaceticus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.031 |
| Acinetobacter haemolyticus |
Acinetobacter haemolyticus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00267-07 |
| Acinetobacter lwoffii |
Acinetobacter lwoffii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00598-10 |
| Acinetobacter lwoffii |
Acinetobacter lwoffii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00598-10 |
| Acinetobacter lwoffii |
Acinetobacter lwoffii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00598-10 |
| Acinetobacter lwoffii |
Acinetobacter lwoffii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00598-10 |
| Acinetobacter lwoffii |
Acinetobacter lwoffii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00598-10 |
| Acinetobacter lwoffii |
Acinetobacter lwoffii |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00598-10 |
| Acinetobacter pittii |
Acinetobacter pittii |
Activity |
57.9 |
% |
10.1128/aac.01624-09 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
0.094 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
0.47 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01624-09 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
0.64 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00072-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01624-09 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01624-09 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01624-09 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.01624-09 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.01624-09 |
| Acinetobacter pittii |
Acinetobacter pittii |
Ratio |
3.0 |
None |
10.1128/aac.00485-08 |
| Acinetobacter pittii |
Acinetobacter pittii |
Ratio |
4.0 |
None |
10.1128/aac.00485-08 |
| Acinetobacter radioresistens |
Acinetobacter radioresistens |
GI |
nan |
None |
10.1128/aac.01304-07 |
| Acinetobacter radioresistens |
Acinetobacter radioresistens |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00999-08 |
| Acinetobacter radioresistens |
Acinetobacter radioresistens |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00999-08 |
| Acinetobacter sp. |
Acinetobacter sp. |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Acinetobacter sp. |
Acinetobacter sp. |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00838-06 |
| Acinetobacter sp. |
Acinetobacter sp. |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm400560z |
| Acinetobacter sp. |
Acinetobacter sp. |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/ml200012f |
| Acinetobacter sp. |
Acinetobacter sp. |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Acinetobacter sp. |
Acinetobacter sp. |
MIC90 |
32.0 |
ug.mL-1 |
10.1021/jm400560z |
| Acinetobacter sp. |
Acinetobacter sp. |
MIC90 |
32.0 |
ug.mL-1 |
10.1021/ml200012f |
| Acinetobacter sp. |
Acinetobacter sp. |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Actinomyces israelii |
Actinomyces israelii |
Activity |
8.0 |
% |
10.1128/aac.00481-10 |
| Actinomyces israelii |
Actinomyces israelii |
Activity |
92.0 |
% |
10.1128/aac.00481-10 |
| Actinomyces israelii |
Actinomyces israelii |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Actinomyces israelii |
Actinomyces israelii |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Actinomyces israelii |
Actinomyces israelii |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Actinomyces naeslundii |
Actinomyces naeslundii |
Activity |
8.0 |
% |
10.1128/aac.00481-10 |
| Actinomyces naeslundii |
Actinomyces naeslundii |
Activity |
92.0 |
% |
10.1128/aac.00481-10 |
| Actinomyces naeslundii |
Actinomyces naeslundii |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Actinomyces naeslundii |
Actinomyces naeslundii |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Actinomyces naeslundii |
Actinomyces naeslundii |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Aeromonas allosaccharophila |
Extended-spectrum beta-lactamase PER-6 |
Kcat |
0.004 |
/s |
10.1128/aac.01585-09 |
| Aeromonas allosaccharophila |
Extended-spectrum beta-lactamase PER-6 |
Kcat/Km |
0.4 |
/uM/s |
10.1128/aac.01585-09 |
| Aeromonas allosaccharophila |
Extended-spectrum beta-lactamase PER-6 |
Km |
10000.0 |
nM |
10.1128/aac.01585-09 |
| Aeromonas caviae |
Aeromonas caviae |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmc.2013.09.041 |
| Aeromonas caviae |
Aeromonas caviae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2013.09.041 |
| Aeromonas caviae |
Aeromonas caviae |
MIC |
1024.0 |
ug.mL-1 |
10.1128/aac.01462-06 |
| Aeromonas caviae |
IMP-19 |
Kcat |
1.0 |
/s |
10.1128/aac.01462-06 |
| Aeromonas caviae |
IMP-19 |
Kcat/Km |
0.14 |
None |
10.1128/aac.01462-06 |
| Aeromonas caviae |
IMP-19 |
Km |
7000.0 |
nM |
10.1128/aac.01462-06 |
| Aeromonas hydrophila |
Aeromonas hydrophila |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmc.2013.09.041 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
Activity |
100.0 |
% |
10.1128/aac.00481-10 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Anaerococcus tetradius |
Anaerococcus tetradius |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Anaerococcus tetradius |
Anaerococcus tetradius |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Anaerococcus tetradius |
Anaerococcus tetradius |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Anaerococcus tetradius |
Anaerococcus tetradius |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Anaerococcus tetradius |
Anaerococcus tetradius |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Anaerococcus vaginalis |
Anaerococcus vaginalis |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Anaerococcus vaginalis |
Anaerococcus vaginalis |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Anaerococcus vaginalis |
Anaerococcus vaginalis |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Anaerocolumna aminovalerica |
Anaerocolumna aminovalerica |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Anaerocolumna aminovalerica |
Anaerocolumna aminovalerica |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Anaerocolumna aminovalerica |
Anaerocolumna aminovalerica |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Aspergillus fumigatus |
Aspergillus fumigatus |
IC50 |
300.0 |
nM |
10.1021/acs.jnatprod.9b00187 |
| Bacillus anthracis |
Bacillus anthracis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00737-08 |
| Bacillus anthracis |
Bacillus anthracis |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00737-08 |
| Bacillus anthracis |
Bacillus anthracis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00737-08 |
| Bacillus anthracis |
Bacillus anthracis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00737-08 |
| Bacillus anthracis |
Bacillus anthracis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00737-08 |
| Bacillus anthracis |
Bacillus anthracis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00737-08 |
| Bacillus anthracis |
Bacillus anthracis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00737-08 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
3.125 |
ug.mL-1 |
10.1016/j.bmc.2016.02.013 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Bacteria |
Cell membrane |
Activity |
12.2 |
% |
10.1016/j.ejmech.2022.114278 |
| Bacteria |
Cell membrane |
Activity |
14.7 |
% |
10.1016/j.ejmech.2022.114278 |
| Bacteria |
Cell membrane |
Activity |
17.2 |
% |
10.1016/j.ejmech.2022.114278 |
| Bacteria |
Cell membrane |
Activity |
22.1 |
% |
10.1016/j.ejmech.2022.114278 |
| Bacteria |
Cell membrane |
Activity |
nan |
None |
10.1016/j.ejmech.2018.06.054 |
| Bacteroides caccae |
Bacteroides caccae |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Bacteroides caccae |
Bacteroides caccae |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Bacteroides caccae |
Bacteroides caccae |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Bacteroides caccae |
Bacteroides caccae |
Activity |
0.5 |
% |
10.1128/aac.01435-06 |
| Bacteroides caccae |
Bacteroides caccae |
Activity |
4.0 |
% |
10.1128/aac.00355-08 |
| Bacteroides caccae |
Bacteroides caccae |
Activity |
96.0 |
% |
10.1128/aac.00355-08 |
| Bacteroides caccae |
Bacteroides caccae |
Activity |
98.0 |
% |
10.1128/aac.00481-10 |
| Bacteroides caccae |
Bacteroides caccae |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Bacteroides caccae |
Bacteroides caccae |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides caccae |
Bacteroides caccae |
MIC |
0.13 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Bacteroides caccae |
Bacteroides caccae |
MIC |
0.4 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Bacteroides caccae |
Bacteroides caccae |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Bacteroides caccae |
Bacteroides caccae |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides caccae |
Bacteroides caccae |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides caccae |
Bacteroides caccae |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Bacteroides caccae |
Bacteroides caccae |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Bacteroides caccae |
Bacteroides caccae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Bacteroides caccae |
Bacteroides caccae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Bacteroides caccae |
Bacteroides caccae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Bacteroides caccae |
Bacteroides caccae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Bacteroides caccae |
Bacteroides caccae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides caccae |
Bacteroides caccae |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Bacteroides fragilis |
Bacteroides fragilis |
Activity |
1.0 |
% |
10.1128/aac.01435-06 |
| Bacteroides fragilis |
Bacteroides fragilis |
Activity |
1.5 |
% |
10.1128/aac.00696-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
Activity |
3.0 |
% |
10.1128/aac.00481-10 |
| Bacteroides fragilis |
Bacteroides fragilis |
Activity |
5.0 |
% |
10.1128/aac.00355-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
Activity |
88.0 |
% |
10.1128/aac.00355-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
Activity |
90.0 |
% |
10.1128/aac.00910-07 |
| Bacteroides fragilis |
Bacteroides fragilis |
Activity |
92.0 |
% |
10.1128/aac.00481-10 |
| Bacteroides fragilis |
Bacteroides fragilis |
Activity |
99.0 |
% |
10.1128/aac.00910-07 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
0.05 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC50 |
0.28 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Bacteroides ovatus |
Bacteroides ovatus |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Bacteroides ovatus |
Bacteroides ovatus |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Bacteroides ovatus |
Bacteroides ovatus |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Bacteroides ovatus |
Bacteroides ovatus |
Activity |
98.0 |
% |
10.1128/aac.00481-10 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC |
0.13 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides stercoris |
Bacteroides stercoris |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Bacteroides stercoris |
Bacteroides stercoris |
Activity |
0.5 |
% |
10.1128/aac.01435-06 |
| Bacteroides stercoris |
Bacteroides stercoris |
MIC |
0.4 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Bacteroides stercoris |
Bacteroides stercoris |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides stercoris |
Bacteroides stercoris |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Bacteroides stercoris |
Bacteroides stercoris |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Bacteroides stercoris |
Bacteroides stercoris |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Bacteroides stercoris |
Bacteroides stercoris |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
Activity |
0.1 |
% |
10.1128/aac.01435-06 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
Activity |
90.0 |
% |
10.1128/aac.00910-07 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
Activity |
97.0 |
% |
10.1128/aac.00355-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
Activity |
98.0 |
% |
10.1128/aac.00481-10 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
Activity |
99.0 |
% |
10.1128/aac.00910-07 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC |
0.13 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC |
0.47 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides uniformis |
Bacteroides uniformis |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Bacteroides uniformis |
Bacteroides uniformis |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Bacteroides uniformis |
Bacteroides uniformis |
Activity |
0.5 |
% |
10.1128/aac.01435-06 |
| Bacteroides uniformis |
Bacteroides uniformis |
Activity |
4.0 |
% |
10.1128/aac.00355-08 |
| Bacteroides uniformis |
Bacteroides uniformis |
Activity |
96.0 |
% |
10.1128/aac.00355-08 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC |
0.41 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bifidobacterium bifidum |
Bifidobacterium bifidum |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bifidobacterium breve |
Bifidobacterium breve |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Bos taurus |
Progesterone receptor |
IC50 |
nan |
None |
None |
| Bos taurus |
Progesterone receptor |
Ki |
nan |
None |
None |
| Burkholderia cenocepacia |
PenB class A beta-lactamase |
Kcat |
1.0 |
/s |
10.1128/aac.00946-08 |
| Burkholderia cenocepacia |
PenB class A beta-lactamase |
Kcat/Km |
0.5 |
/uM/s |
10.1128/aac.00946-08 |
| Burkholderia cenocepacia |
PenB class A beta-lactamase |
Km |
2500000.0 |
nM |
10.1128/aac.00946-08 |
| Burkholderia cepacia |
Burkholderia cepacia |
Activity |
26.0 |
% |
10.1128/aac.00954-06 |
| Burkholderia cepacia |
Burkholderia cepacia |
Activity |
48.0 |
% |
10.1128/aac.00954-06 |
| Burkholderia cepacia |
Burkholderia cepacia |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Burkholderia cepacia |
Burkholderia cepacia |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Burkholderia cepacia |
Burkholderia cepacia |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00954-06 |
| Burkholderia cepacia |
Burkholderia cepacia |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00954-06 |
| Burkholderia pseudomallei |
Burkholderia pseudomallei |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00893-08 |
| Burkholderia pseudomallei |
Burkholderia pseudomallei |
MIC50 |
3.0 |
ug.mL-1 |
10.1128/aac.00893-08 |
| Burkholderia pseudomallei |
Burkholderia pseudomallei |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00893-08 |
| Burkholderia pseudomallei |
Burkholderia pseudomallei |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00893-08 |
| Burkholderia pseudomallei |
Burkholderia pseudomallei |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01582-09 |
| Campylobacter coli |
Campylobacter coli |
Activity |
0.0 |
% |
10.1128/aac.00898-09 |
| Campylobacter coli |
Campylobacter coli |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter coli |
Campylobacter coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter coli |
Campylobacter coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter coli |
Campylobacter coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter coli |
Campylobacter coli |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter coli |
Campylobacter coli |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
Activity |
0.0 |
% |
10.1128/aac.00898-09 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC |
0.08 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Campylobacter jejuni |
Campylobacter jejuni |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.01655-08 |
| Candida albicans |
Candida albicans |
IC50 |
300.0 |
nM |
10.1021/acs.jnatprod.9b00187 |
| Candida albicans |
Candida albicans |
Inhibition |
3.42 |
% |
10.6019/CHEMBL4513141 |
| Capnocytophaga ochracea |
Capnocytophaga ochracea |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Caulobacter vibrioides |
Metallo-beta-lactamase |
Kcat/Km |
2.6 |
10'5/M/s |
10.1128/aac.01062-07 |
| Cavia porcellus |
Leukotriene C4 synthase |
IC50 |
nan |
None |
None |
| Cavia porcellus |
Leukotriene C4 synthase |
Ki |
nan |
None |
None |
| Cavia porcellus |
Serotonin 4 (5-HT4) receptor |
IC50 |
nan |
None |
None |
| Cavia porcellus |
Serotonin 4 (5-HT4) receptor |
Ki |
nan |
None |
None |
| Chryseobacterium indologenes |
Chryseobacterium indologenes |
Activity |
16.0 |
ug ml-1 |
10.1128/aac.00083-07 |
| Chryseobacterium indologenes |
Chryseobacterium indologenes |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01607-08 |
| Chryseobacterium indologenes |
IND-like metallo-beta-lactamase |
Kcat/Km |
1.5 |
10'4/M/s |
10.1128/aac.01607-08 |
| Chryseobacterium indologenes |
Metallo-beta-lactamase IND-2 |
Kcat/Km |
1.8 |
10'5/M/s |
10.1128/aac.01607-08 |
| Chryseobacterium indologenes |
Metallo-beta-lactamase IND-6 |
Kcat |
25.0 |
/s |
10.1128/aac.01607-08 |
| Chryseobacterium indologenes |
Metallo-beta-lactamase IND-6 |
Kcat/Km |
1.7 |
10'5/M/s |
10.1128/aac.01607-08 |
| Chryseobacterium indologenes |
Metallo-beta-lactamase IND-6 |
Km |
145000.0 |
nM |
10.1128/aac.01607-08 |
| Citrobacter |
Citrobacter |
Activity |
0.0 |
% |
10.1128/aac.00381-08 |
| Citrobacter |
Citrobacter |
Activity |
100.0 |
% |
10.1128/aac.00381-08 |
| Citrobacter |
Citrobacter |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Citrobacter |
Citrobacter |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Citrobacter |
Citrobacter |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Citrobacter |
Citrobacter |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Citrobacter |
Citrobacter |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Citrobacter |
Citrobacter |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Citrobacter |
Citrobacter |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
0.06 |
ug.mL-1 |
10.1016/S0960-894X(97)00282-5 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01337-07 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01405-06 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01305-10 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Citrobacter freundii |
Citrobacter freundii |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Citrobacter freundii |
Citrobacter freundii |
MIC50 |
0.06 |
ug.mL-1 |
10.1021/ml200012f |
| Citrobacter freundii |
Citrobacter freundii |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Citrobacter freundii |
Citrobacter freundii |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Citrobacter freundii |
Citrobacter freundii |
MIC90 |
0.25 |
ug.mL-1 |
10.1021/ml200012f |
| Citrobacter freundii |
Citrobacter freundii |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Clostridioides difficile |
Clostridioides difficile |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Clostridioides difficile |
Clostridioides difficile |
Activity |
90.0 |
% |
10.1128/aac.00910-07 |
| Clostridioides difficile |
Clostridioides difficile |
Activity |
99.0 |
% |
10.1128/aac.00910-07 |
| Clostridioides difficile |
Clostridioides difficile |
Activity |
100.0 |
% |
10.1128/aac.00481-10 |
| Clostridioides difficile |
Clostridioides difficile |
Activity |
nan |
None |
10.1128/aac.00696-08 |
| Clostridioides difficile |
Clostridioides difficile |
Activity |
nan |
None |
10.1128/aac.00910-07 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00476-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00476-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Clostridioides difficile |
Clostridioides difficile |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Clostridioides difficile |
Clostridioides difficile |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01623-06 |
| Clostridioides difficile |
Clostridioides difficile |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00476-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Clostridioides difficile |
Clostridioides difficile |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01623-06 |
| Clostridioides difficile |
Clostridioides difficile |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Clostridium cadaveris |
Clostridium cadaveris |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Clostridium cadaveris |
Clostridium cadaveris |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Clostridium cadaveris |
Clostridium cadaveris |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Clostridium cadaveris |
Clostridium cadaveris |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00910-07 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00910-07 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium malenominatum |
Clostridium malenominatum |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Clostridium malenominatum |
Clostridium malenominatum |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Clostridium malenominatum |
Clostridium malenominatum |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
Activity |
100.0 |
% |
10.1128/aac.00355-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium perfringens |
Clostridium perfringens |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Clostridium perfringens |
Clostridium perfringens |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Clostridium perfringens |
Clostridium perfringens |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Clostridium perfringens |
Clostridium perfringens |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Clostridium perfringens |
Clostridium perfringens |
Activity |
90.0 |
% |
10.1128/aac.00910-07 |
| Clostridium perfringens |
Clostridium perfringens |
Activity |
99.0 |
% |
10.1128/aac.00910-07 |
| Clostridium perfringens |
Clostridium perfringens |
Activity |
100.0 |
% |
10.1128/aac.00355-08 |
| Clostridium perfringens |
Clostridium perfringens |
Activity |
100.0 |
% |
10.1128/aac.00481-10 |
| Clostridium perfringens |
Clostridium perfringens |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Clostridium perfringens |
Clostridium perfringens |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Clostridium perfringens |
Clostridium perfringens |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Clostridium perfringens |
Clostridium perfringens |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Clostridium perfringens |
Clostridium perfringens |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Clostridium perfringens |
Clostridium perfringens |
MIC50 |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Clostridium perfringens |
Clostridium perfringens |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC90 |
0.015 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Clostridium perfringens |
Clostridium perfringens |
MIC90 |
0.015 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Clostridium perfringens |
Clostridium perfringens |
MIC90 |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Clostridium perfringens |
Clostridium perfringens |
MIC90 |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Clostridium septicum |
Clostridium septicum |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Clostridium septicum |
Clostridium septicum |
Activity |
100.0 |
% |
10.1128/aac.00355-08 |
| Clostridium septicum |
Clostridium septicum |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Clostridium septicum |
Clostridium septicum |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Clostridium septicum |
Clostridium septicum |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Clostridium septicum |
Clostridium septicum |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Clostridium tertium |
Clostridium tertium |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Clostridium tertium |
Clostridium tertium |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Clostridium tertium |
Clostridium tertium |
Activity |
100.0 |
% |
10.1128/aac.00355-08 |
| Clostridium tertium |
Clostridium tertium |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Clostridium tertium |
Clostridium tertium |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium tertium |
Clostridium tertium |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Clostridium tertium |
Clostridium tertium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium tertium |
Clostridium tertium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Clostridium tertium |
Clostridium tertium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Corynebacterium accolens |
Corynebacterium accolens |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Corynebacterium accolens |
Corynebacterium accolens |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium accolens |
Corynebacterium accolens |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium amycolatum |
Corynebacterium amycolatum |
Activity |
7.0 |
% |
10.1128/aac.01128-07 |
| Corynebacterium amycolatum |
Corynebacterium amycolatum |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium amycolatum |
Corynebacterium amycolatum |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium aurimucosum |
Corynebacterium aurimucosum |
Activity |
20.0 |
% |
10.1128/aac.01128-07 |
| Corynebacterium aurimucosum |
Corynebacterium aurimucosum |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium aurimucosum |
Corynebacterium aurimucosum |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium diphtheriae |
Corynebacterium diphtheriae |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Corynebacterium diphtheriae |
Corynebacterium diphtheriae |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
Activity |
20.0 |
% |
10.1128/aac.01128-07 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium minutissimum |
Corynebacterium minutissimum |
Activity |
20.0 |
% |
10.1128/aac.01128-07 |
| Corynebacterium minutissimum |
Corynebacterium minutissimum |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium minutissimum |
Corynebacterium minutissimum |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium simulans |
Corynebacterium simulans |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Corynebacterium simulans |
Corynebacterium simulans |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium simulans |
Corynebacterium simulans |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium striatum |
Corynebacterium striatum |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Corynebacterium striatum |
Corynebacterium striatum |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium striatum |
Corynebacterium striatum |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium urealyticum |
Corynebacterium urealyticum |
Activity |
20.0 |
% |
10.1128/aac.01128-07 |
| Corynebacterium urealyticum |
Corynebacterium urealyticum |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium urealyticum |
Corynebacterium urealyticum |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium xerosis |
Corynebacterium xerosis |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Corynebacterium xerosis |
Corynebacterium xerosis |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Corynebacterium xerosis |
Corynebacterium xerosis |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Cronobacter sakazakii |
Cronobacter sakazakii |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Cryptococcus neoformans |
Cryptococcus neoformans |
IC50 |
300.0 |
nM |
10.1021/acs.jnatprod.9b00187 |
| Cryptococcus neoformans |
Cryptococcus neoformans |
Inhibition |
2.76 |
% |
10.6019/CHEMBL4513141 |
| Cutibacterium acnes |
Cutibacterium acnes |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Cutibacterium acnes |
Cutibacterium acnes |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Cutibacterium acnes |
Cutibacterium acnes |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Cutibacterium acnes |
Cutibacterium acnes |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Cutibacterium acnes |
Cutibacterium acnes |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Cutibacterium acnes |
Cutibacterium acnes |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Cutibacterium acnes |
Cutibacterium acnes |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Cutibacterium acnes |
Cutibacterium acnes |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Eggerthella lenta |
Eggerthella lenta |
Activity |
8.0 |
% |
10.1128/aac.00481-10 |
| Eggerthella lenta |
Eggerthella lenta |
Activity |
92.0 |
% |
10.1128/aac.00481-10 |
| Eggerthella lenta |
Eggerthella lenta |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Eggerthella lenta |
Eggerthella lenta |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Eggerthella lenta |
Eggerthella lenta |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Eggerthella lenta |
Eggerthella lenta |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Eggerthella lenta |
Eggerthella lenta |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Eggerthella lenta |
Eggerthella lenta |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Eggerthella lenta |
Eggerthella lenta |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Elizabethkingia meningoseptica |
GOB-1 metallo-beta-lactamase |
Kcat/Km |
5.3 |
10'6/M/s |
10.1128/aac.01062-07 |
| Enterobacter cloacae |
Beta-lactamase |
Activity |
1.2e-05 |
% |
10.1128/aac.01004-09 |
| Enterobacter cloacae |
Beta-lactamase |
Activity |
0.00042 |
% |
10.1128/aac.01004-09 |
| Enterobacter cloacae |
Beta-lactamase |
Kcat |
0.00031 |
/s |
10.1128/aac.01004-09 |
| Enterobacter cloacae |
Beta-lactamase |
Kcat/Km |
3.2e-05 |
/s/microM |
10.1128/aac.01004-09 |
| Enterobacter cloacae |
Beta-lactamase |
Km |
9800.0 |
nM |
10.1128/aac.01004-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
0.0 |
% |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
0.0 |
% |
10.1128/aac.00400-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
0.0 |
% |
10.1128/aac.01538-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
0.4 |
% |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
0.5 |
% |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
7.0 |
ug ml-1 |
10.1128/aac.01525-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
9.0 |
ug ml-1 |
10.1128/aac.01525-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
99.5 |
% |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
99.6 |
% |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
100.0 |
% |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
100.0 |
% |
10.1128/aac.00400-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
Activity |
nan |
None |
10.1128/aac.01525-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
Inhibition |
nan |
% |
10.1128/aac.01452-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MBC |
0.03 |
ug ml-1 |
10.1128/aac.01452-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MBC |
0.125 |
ug ml-1 |
10.1128/aac.01452-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.01525-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MBC |
0.5 |
ug ml-1 |
10.1128/aac.01452-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MBC |
2.0 |
ug ml-1 |
10.1128/aac.01525-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(00)00253-5 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(00)00575-8 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(01)00451-6 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(02)00948-4 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(99)00407-2 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(99)00646-0 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(99)00692-7 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01452-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.031 |
ug.mL-1 |
10.1016/j.bmc.2021.116343 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.06 |
ug.mL-1 |
10.1016/S0960-894X(97)00282-5 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01452-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2013.09.041 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01452-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2013.09.041 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.031 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00707-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01341-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00931-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01341-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.01341-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.5b00127 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01341-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116343 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
24.0 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
24.0 |
ug.mL-1 |
10.1128/aac.01341-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.031 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
32.0 |
ug.mL-1 |
10.1039/C5MD00380F |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00033-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00260-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01341-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC90 |
0.13 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Enterobacter cloacae |
IMI-1 |
Kcat |
10.0 |
/s |
10.1128/aac.00491-07 |
| Enterobacter cloacae |
IMI-1 |
Kcat/Km |
380.0 |
/mM/s |
10.1128/aac.00491-07 |
| Enterobacter cloacae |
IMI-1 |
Km |
26000.0 |
nM |
10.1128/aac.00491-07 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
0.0 |
% |
10.1128/aac.00381-08 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
0.1 |
% |
10.1128/aac.00381-08 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
0.7 |
% |
10.1128/aac.00381-08 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
1.3 |
% |
10.1128/aac.00381-08 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
2.0 |
% |
10.1128/aac.00044-07 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
6.0 |
% |
10.1128/aac.00044-07 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
32.7 |
% |
10.1128/aac.01114-07 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
50.0 |
% |
10.1128/aac.01114-07 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
62.5 |
% |
10.1128/aac.01450-09 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
77.9 |
% |
10.1128/aac.01450-09 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
81.3 |
% |
10.1128/aac.01450-09 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
85.0 |
% |
10.1128/aac.01450-09 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
91.7 |
% |
10.1128/aac.01450-09 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
98.0 |
% |
10.1128/aac.00381-08 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
99.6 |
% |
10.1128/aac.00381-08 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
99.8 |
% |
10.1128/aac.00381-08 |
| Enterobacteriaceae |
Enterobacteriaceae |
Activity |
100.0 |
% |
10.1128/aac.01450-09 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01114-07 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC |
nan |
None |
10.1016/j.ejmech.2017.10.044 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01450-09 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.01114-07 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.01450-09 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01450-09 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01114-07 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC90 |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.006 |
| Enterobacter sp. |
Enterobacter sp. |
Activity |
33.3 |
% |
10.1128/aac.01114-07 |
| Enterobacter sp. |
Enterobacter sp. |
Activity |
41.7 |
% |
10.1128/aac.01114-07 |
| Enterobacter sp. |
Enterobacter sp. |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.01114-07 |
| Enterobacter sp. |
Enterobacter sp. |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01114-07 |
| Enterocloster clostridioformis |
Enterocloster clostridioformis |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Enterocloster clostridioformis |
Enterocloster clostridioformis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Enterocloster clostridioformis |
Enterocloster clostridioformis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Enterocloster clostridioformis |
Enterocloster clostridioformis |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Enterocloster clostridioformis |
Enterocloster clostridioformis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Enterococcus durans |
Enterococcus durans |
MIC |
0.8 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Enterococcus durans |
Enterococcus durans |
MIC |
0.8 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/S0960-894X(97)00282-5 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1039/D1MD00230A |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1039/D1MD00230A |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1039/D1MD00230A |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1016/j.ejmech.2017.10.044 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1016/j.ejmech.2017.12.009 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1021/acs.jmedchem.2c01674 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1074/jbc.m704286200 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113402 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113402 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
6.25 |
ug.mL-1 |
10.1016/s0960-894x(99)00692-7 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
6.25 |
ug.mL-1 |
10.1021/np049577a |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113402 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
8.0 |
ug.mL-1 |
10.1074/jbc.m704286200 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
12.5 |
ug.mL-1 |
10.1016/s0960-894x(98)00270-4 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
12.5 |
ug.mL-1 |
10.1016/s0960-894x(99)00407-2 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113402 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
128.0 |
ug.mL-1 |
10.1016/S0960-894X(97)00282-5 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
128.0 |
ug.mL-1 |
10.1039/D1MD00230A |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116128 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
nan |
None |
10.1021/np800503z |
| Enterococcus sp. |
Enterococcus sp. |
Activity |
nan |
None |
10.1128/aac.01538-07 |
| Escherichia coli |
Beta-lactamase |
Activity |
1.1e-05 |
% |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase |
Activity |
0.058 |
% |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase |
Kcat |
8.1e-05 |
/s |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase |
Kcat/Km |
0.0014 |
/s/microM |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase |
Km |
60.0 |
nM |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase CTX-M |
Activity |
0.0022 |
% |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase CTX-M |
Activity |
0.0078 |
% |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase CTX-M |
Kcat |
0.0042 |
/s |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase CTX-M |
Kcat/Km |
0.00038 |
/s/microM |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase CTX-M |
Km |
11000.0 |
nM |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase TEM |
Activity |
2.3e-05 |
% |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase TEM |
Activity |
0.00083 |
% |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase TEM |
Kcat |
0.00023 |
/s |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase TEM |
Kcat/Km |
1.5e-05 |
/s/microM |
10.1128/aac.01004-09 |
| Escherichia coli |
Beta-lactamase TEM |
Km |
15000.0 |
nM |
10.1128/aac.01004-09 |
| Escherichia coli |
BlaVIM-1 |
Kcat |
13.0 |
/s |
10.1128/aac.00017-09 |
| Escherichia coli |
BlaVIM-1 |
Kcat |
15.0 |
/s |
10.1128/aac.00458-09 |
| Escherichia coli |
BlaVIM-1 |
Kcat/Km |
0.27 |
/s/microM |
10.1128/aac.00017-09 |
| Escherichia coli |
BlaVIM-1 |
Kcat/Km |
0.3 |
/uM/s |
10.1128/aac.00458-09 |
| Escherichia coli |
BlaVIM-1 |
Km |
50000.0 |
nM |
10.1128/aac.00458-09 |
| Escherichia coli |
Escherichia coli |
Activity |
-1.46 |
log10CFU/g |
10.1021/acs.jmedchem.0c00579 |
| Escherichia coli |
Escherichia coli |
Activity |
0.0 |
% |
10.1128/aac.00063-08 |
| Escherichia coli |
Escherichia coli |
Activity |
0.0 |
% |
10.1128/aac.00381-08 |
| Escherichia coli |
Escherichia coli |
Activity |
0.0 |
% |
10.1128/aac.00400-09 |
| Escherichia coli |
Escherichia coli |
Activity |
0.0 |
% |
10.1128/aac.00551-10 |
| Escherichia coli |
Escherichia coli |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Escherichia coli |
Escherichia coli |
Activity |
0.0 |
% |
10.1128/aac.01412-06 |
| Escherichia coli |
Escherichia coli |
Activity |
0.0 |
% |
10.1128/aac.01538-07 |
| Escherichia coli |
Escherichia coli |
Activity |
0.125 |
ug ml-1 |
10.1128/aac.00083-07 |
| Escherichia coli |
Escherichia coli |
Activity |
1.0 |
CFU/ml |
10.1016/j.ejmech.2022.114495 |
| Escherichia coli |
Escherichia coli |
Activity |
1.0 |
ug ml-1 |
10.1128/aac.00083-07 |
| Escherichia coli |
Escherichia coli |
Activity |
95.0 |
% |
10.1016/j.ejmech.2019.01.083 |
| Escherichia coli |
Escherichia coli |
Activity |
100.0 |
% |
10.1128/aac.00381-08 |
| Escherichia coli |
Escherichia coli |
Activity |
100.0 |
% |
10.1128/aac.00400-09 |
| Escherichia coli |
Escherichia coli |
Activity |
100.0 |
% |
10.1128/aac.01176-07 |
| Escherichia coli |
Escherichia coli |
Activity |
100.0 |
% |
10.1128/aac.01509-06 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1016/j.bmcl.2016.10.004 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1016/j.ejmech.2022.114278 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1016/j.ejmech.2022.114571 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1128/aac.00220-10 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1128/aac.01525-09 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1128/aac.01529-07 |
| Escherichia coli |
Escherichia coli |
ED50 |
2.04 |
mg.kg-1 |
10.1021/acs.jmedchem.6b01261 |
| Escherichia coli |
Escherichia coli |
ED50 |
nan |
mg.kg-1 |
10.1016/S0960-894X(97)00282-5 |
| Escherichia coli |
Escherichia coli |
fT>MIC |
70.0 |
% |
10.1128/aac.00752-06 |
| Escherichia coli |
Escherichia coli |
fT>MIC |
85.0 |
% |
10.1128/aac.00752-06 |
| Escherichia coli |
Escherichia coli |
fT>MIC |
90.0 |
% |
10.1128/aac.00752-06 |
| Escherichia coli |
Escherichia coli |
fT>MIC |
93.0 |
% |
10.1128/aac.00752-06 |
| Escherichia coli |
Escherichia coli |
IC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Escherichia coli |
Escherichia coli |
IC50 |
10.0 |
nM |
10.1021/acs.jnatprod.9b00187 |
| Escherichia coli |
Escherichia coli |
Inhibition |
7.87 |
% |
10.6019/CHEMBL4513141 |
| Escherichia coli |
Escherichia coli |
Inhibition |
nan |
% |
10.1128/aac.01452-08 |
| Escherichia coli |
Escherichia coli |
MBC |
0.03 |
ug ml-1 |
10.1128/aac.01433-08 |
| Escherichia coli |
Escherichia coli |
MBC |
0.06 |
ug ml-1 |
10.1128/aac.01452-08 |
| Escherichia coli |
Escherichia coli |
MBC |
2.0 |
ug ml-1 |
10.1021/acs.jmedchem.2c01469 |
| Escherichia coli |
Escherichia coli |
MIC |
0.0 |
ug.mL-1 |
10.1128/aac.01585-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1e-05 |
ug.mL-1 |
10.1016/j.ejmech.2022.114108 |
| Escherichia coli |
Escherichia coli |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.00294-06 |
| Escherichia coli |
Escherichia coli |
MIC |
0.002 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.004 |
ug.mL-1 |
10.1128/aac.01337-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.008 |
ug.mL-1 |
10.1016/j.bmc.2021.116142 |
| Escherichia coli |
Escherichia coli |
MIC |
0.008 |
ug.mL-1 |
10.1016/j.ejmech.2021.113975 |
| Escherichia coli |
Escherichia coli |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00771-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Escherichia coli |
Escherichia coli |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Escherichia coli |
Escherichia coli |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2022.114108 |
| Escherichia coli |
Escherichia coli |
MIC |
0.01 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.012 |
ug.mL-1 |
10.1128/aac.00598-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.012 |
ug.mL-1 |
10.1128/aac.01818-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.013 |
ug.mL-1 |
10.1016/s0960-894x(99)00407-2 |
| Escherichia coli |
Escherichia coli |
MIC |
0.013 |
ug.mL-1 |
10.1016/s0960-894x(99)00692-7 |
| Escherichia coli |
Escherichia coli |
MIC |
0.013 |
ug.mL-1 |
10.1021/np060206z |
| Escherichia coli |
Escherichia coli |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.006 |
| Escherichia coli |
Escherichia coli |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00768-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00858-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1016/j.ejmech.2022.114108 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00072-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00175-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00458-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00461-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00684-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00771-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.01341-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Escherichia coli |
Escherichia coli |
MIC |
0.02133 |
ug.mL-1 |
10.1016/j.ejmech.2022.114108 |
| Escherichia coli |
Escherichia coli |
MIC |
0.023 |
ug.mL-1 |
10.1128/aac.00050-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.023 |
ug.mL-1 |
10.1128/aac.00374-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.023 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.023 |
ug.mL-1 |
10.1128/aac.00771-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/0960-894X(95)00380-C |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(00)00253-5 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(00)00575-8 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(01)00451-6 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(02)00948-4 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/S0960-894X(97)00230-8 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(98)00270-4 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(99)00407-2 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(99)00646-0 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(99)00692-7 |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1021/np049577a |
| Escherichia coli |
Escherichia coli |
MIC |
0.025 |
ug.mL-1 |
10.1128/aac.00780-06 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00746 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1021/np800503z |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00033-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00175-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00461-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00543-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00768-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01025-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01062-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01180-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01336-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01431-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01452-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01529-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01585-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01607-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.031 |
ug.mL-1 |
10.1016/j.bmc.2021.116343 |
| Escherichia coli |
Escherichia coli |
MIC |
0.031 |
ug.mL-1 |
10.1016/j.ejmech.2022.114174 |
| Escherichia coli |
Escherichia coli |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00050-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00374-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00436-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00485-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00598-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00684-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Escherichia coli |
Escherichia coli |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00771-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.01011-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.01762-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.03733 |
ug.mL-1 |
10.1016/j.ejmech.2022.114108 |
| Escherichia coli |
Escherichia coli |
MIC |
0.0375 |
ug.mL-1 |
10.1039/c9md00455f |
| Escherichia coli |
Escherichia coli |
MIC |
0.04 |
ug.mL-1 |
10.1021/jm010546b |
| Escherichia coli |
Escherichia coli |
MIC |
0.047 |
ug.mL-1 |
10.1128/aac.00072-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.047 |
ug.mL-1 |
10.1128/aac.00158-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.047 |
ug.mL-1 |
10.1128/aac.00436-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.047 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Escherichia coli |
Escherichia coli |
MIC |
0.047 |
ug.mL-1 |
10.1128/aac.00771-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.047 |
ug.mL-1 |
10.1128/aac.01304-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Escherichia coli |
Escherichia coli |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmc.2016.02.013 |
| Escherichia coli |
Escherichia coli |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Escherichia coli |
Escherichia coli |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.006 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2021.127956 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1016/S0960-894X(97)00282-5 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00033-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00688-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00734-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00858-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00878-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01025-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01053-06 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01062-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01431-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01452-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01561-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01585-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Escherichia coli |
Escherichia coli |
MIC |
0.063 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.014 |
| Escherichia coli |
Escherichia coli |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.00465-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.00774-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.01011-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.01762-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.094 |
ug.mL-1 |
10.1128/aac.00137-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.094 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Escherichia coli |
Escherichia coli |
MIC |
0.094 |
ug.mL-1 |
10.1128/aac.00771-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.094 |
ug.mL-1 |
10.1128/aac.01304-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.094 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.1 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.bmc.2013.09.041 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00856-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00961-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00978-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01176-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01247-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01586-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01607-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01672-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.006 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2007.03.023 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2017.10.044 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2017.12.009 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.058 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2019.02.024 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01674 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01261 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01011-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01025-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01431-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01539-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01762-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.00465-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.006 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00033-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00072-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00158-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00299-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00374-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00393-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00458-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00465-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00736-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00961-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01359-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01431-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00158-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.01180-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.006 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.02.024 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00227-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00458-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00543-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00736-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01336-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01359-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01762-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.625 |
ug.mL-1 |
10.1016/j.bmcl.2021.128192 |
| Escherichia coli |
Escherichia coli |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.00436-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Escherichia coli |
Escherichia coli |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.01762-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2013.09.041 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.006 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.058 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114278 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01469 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1021/acsmedchemlett.7b00428 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00158-08 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00458-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00734-08 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00899-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01359-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01462-06 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01672-07 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01762-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.01247-10 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.006 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.031 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00137-10 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00734-08 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00856-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00858-10 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00896-08 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01341-07 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01359-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01539-07 |
| Escherichia coli |
Escherichia coli |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.00878-10 |
| Escherichia coli |
Escherichia coli |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.01341-07 |
| Escherichia coli |
Escherichia coli |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.006 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.031 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.5b00127 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00072-09 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00158-08 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00458-09 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01053-06 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01337-07 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01359-09 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01762-09 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.006 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.058 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b00091 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00734-08 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01359-09 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01762-09 |
| Escherichia coli |
Escherichia coli |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.00774-09 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.006 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127956 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114278 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b00091 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1039/C5MD00380F |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00878-10 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01359-09 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Escherichia coli |
Escherichia coli |
MIC |
24.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00774-09 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Escherichia coli |
Escherichia coli |
MIC |
60.0 |
nM |
10.1021/acs.jmedchem.1c00621 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116128 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.006 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127956 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114599 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01257 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116128 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01469 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00338 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1021/acsmedchemlett.7b00428 |
| Escherichia coli |
Escherichia coli |
MIC |
250.0 |
nM |
10.1021/acs.jmedchem.1c00621 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01462-06 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01462-06 |
| Escherichia coli |
Escherichia coli |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Escherichia coli |
Escherichia coli |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Escherichia coli |
Escherichia coli |
MIC |
4000.0 |
nM |
10.1021/acs.jmedchem.1c00621 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1021/np800503z |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1128/aac.01512-06 |
| Escherichia coli |
Escherichia coli |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Escherichia coli |
Escherichia coli |
MIC50 |
0.03 |
ug.mL-1 |
10.1021/jm400560z |
| Escherichia coli |
Escherichia coli |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Escherichia coli |
Escherichia coli |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Escherichia coli |
Escherichia coli |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01509-06 |
| Escherichia coli |
Escherichia coli |
MIC50 |
0.047 |
ug.mL-1 |
10.1128/aac.00171-08 |
| Escherichia coli |
Escherichia coli |
MIC50 |
0.06 |
ug.mL-1 |
10.1021/ml200012f |
| Escherichia coli |
Escherichia coli |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Escherichia coli |
Escherichia coli |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Escherichia coli |
Escherichia coli |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Escherichia coli |
Escherichia coli |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.01176-07 |
| Escherichia coli |
Escherichia coli |
MIC50 |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00338 |
| Escherichia coli |
Escherichia coli |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00255 |
| Escherichia coli |
Escherichia coli |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01412-06 |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.03 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2012.07.005 |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.06 |
ug.mL-1 |
10.1021/jm400560z |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.06 |
ug.mL-1 |
10.1021/ml200012f |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.064 |
ug.mL-1 |
10.1128/aac.00171-08 |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.094 |
ug.mL-1 |
10.1128/aac.00171-08 |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.01176-07 |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00171-08 |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.19 |
ug.mL-1 |
10.1128/aac.00171-08 |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01509-06 |
| Escherichia coli |
Escherichia coli |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Escherichia coli |
Escherichia coli |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01412-06 |
| Escherichia coli |
Escherichia coli |
MIC90 |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00255 |
| Escherichia coli |
Escherichia coli |
MIC90 |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00338 |
| Escherichia coli |
Escherichia coli |
MPC |
0.03 |
ug ml-1 |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
MPC |
0.06 |
ug ml-1 |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
MPC |
0.125 |
ug ml-1 |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
MPC |
0.25 |
ug ml-1 |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
MPC |
1.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
MPC |
4.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
MPC |
16.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
PD50 |
1.24 |
mg kg-1 |
10.1016/s0960-894x(98)00270-4 |
| Escherichia coli |
Escherichia coli |
Ratio |
2.0 |
None |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
Ratio |
4.0 |
None |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
Ratio |
8.0 |
None |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
Ratio |
16.0 |
None |
10.1128/aac.00033-10 |
| Escherichia coli |
Escherichia coli |
Ratio |
16.0 |
None |
10.1128/aac.00734-08 |
| Escherichia coli |
Escherichia coli |
Survival |
44.0 |
% |
10.1039/C5MD00380F |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat |
1.4 |
/s |
10.1128/aac.00017-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat |
5.0 |
/s |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat |
35.0 |
/s |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat |
45.0 |
/s |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat/Km |
0.28 |
/s/microM |
10.1128/aac.00017-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat/Km |
1.9 |
/uM/s |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat/Km |
2.5 |
uM/hr |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat/Km |
2.5 |
/uM/s |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Kcat/Km |
4.5 |
/uM/s |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Km |
2000.0 |
nM |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Km |
10000.0 |
nM |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
Km |
18000.0 |
nM |
10.1128/aac.01336-09 |
| Escherichia coli |
Metallo-beta-lactamase |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116128 |
| Escherichia coli |
Metallo-beta-lactamase VIM-19 |
Kcat |
25.0 |
/s |
10.1128/aac.00458-09 |
| Escherichia coli |
Metallo-beta-lactamase VIM-19 |
Kcat/Km |
2.0 |
/uM/s |
10.1128/aac.00458-09 |
| Escherichia coli |
Metallo-beta-lactamase VIM-19 |
Km |
15000.0 |
nM |
10.1128/aac.00458-09 |
| Eubacterium limosum |
Eubacterium limosum |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Eubacterium limosum |
Eubacterium limosum |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Eubacterium limosum |
Eubacterium limosum |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Eubacterium sp. |
Eubacterium sp. |
Activity |
8.0 |
% |
10.1128/aac.00481-10 |
| Eubacterium sp. |
Eubacterium sp. |
Activity |
92.0 |
% |
10.1128/aac.00481-10 |
| Eubacterium sp. |
Eubacterium sp. |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Eubacterium sp. |
Eubacterium sp. |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Eubacterium sp. |
Eubacterium sp. |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Finegoldia magna |
Finegoldia magna |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Finegoldia magna |
Finegoldia magna |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Finegoldia magna |
Finegoldia magna |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Finegoldia magna |
Finegoldia magna |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Finegoldia magna |
Finegoldia magna |
Activity |
90.0 |
% |
10.1128/aac.00910-07 |
| Finegoldia magna |
Finegoldia magna |
Activity |
99.0 |
% |
10.1128/aac.00910-07 |
| Finegoldia magna |
Finegoldia magna |
Activity |
100.0 |
% |
10.1128/aac.00355-08 |
| Finegoldia magna |
Finegoldia magna |
Activity |
100.0 |
% |
10.1128/aac.00481-10 |
| Finegoldia magna |
Finegoldia magna |
Activity |
nan |
None |
10.1128/aac.00910-07 |
| Finegoldia magna |
Finegoldia magna |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Finegoldia magna |
Finegoldia magna |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Finegoldia magna |
Finegoldia magna |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Finegoldia magna |
Finegoldia magna |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Finegoldia magna |
Finegoldia magna |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Finegoldia magna |
Finegoldia magna |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Finegoldia magna |
Finegoldia magna |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Finegoldia magna |
Finegoldia magna |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Finegoldia magna |
Finegoldia magna |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Finegoldia magna |
Finegoldia magna |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Finegoldia magna |
Finegoldia magna |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Finegoldia magna |
Finegoldia magna |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Finegoldia magna |
Finegoldia magna |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Finegoldia magna |
Finegoldia magna |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Finegoldia magna |
Finegoldia magna |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Finegoldia magna |
Finegoldia magna |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Flavobacterium meningosepticum |
Carbapenem-hydrolyzing beta-lactamase BlaB-1 |
Kcat/Km |
7.6 |
10'5/M/s |
10.1128/aac.01607-08 |
| Fluoribacter gormanii |
FEZ-1 protein |
Kcat/Km |
5.0 |
10'5/M/s |
10.1128/aac.01062-07 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
Activity |
8.0 |
% |
10.1128/aac.00355-08 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
Activity |
92.0 |
% |
10.1128/aac.00355-08 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Fusobacterium necrophorum |
Fusobacterium necrophorum |
Activity |
8.0 |
% |
10.1128/aac.00355-08 |
| Fusobacterium necrophorum |
Fusobacterium necrophorum |
Activity |
92.0 |
% |
10.1128/aac.00355-08 |
| Fusobacterium necrophorum |
Fusobacterium necrophorum |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium necrophorum |
Fusobacterium necrophorum |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Fusobacterium necrophorum |
Fusobacterium necrophorum |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Fusobacterium necrophorum |
Fusobacterium necrophorum |
MIC50 |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Fusobacterium necrophorum |
Fusobacterium necrophorum |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium necrophorum |
Fusobacterium necrophorum |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Fusobacterium necrophorum |
Fusobacterium necrophorum |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Fusobacterium necrophorum |
Fusobacterium necrophorum |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium necrophorum |
Fusobacterium necrophorum |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
Activity |
8.0 |
% |
10.1128/aac.00355-08 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
Activity |
90.0 |
% |
10.1128/aac.00910-07 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
Activity |
92.0 |
% |
10.1128/aac.00355-08 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
Activity |
99.0 |
% |
10.1128/aac.00910-07 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC50 |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC90 |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium sp. |
Fusobacterium sp. |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium sp. |
Fusobacterium sp. |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium varium |
Fusobacterium varium |
Activity |
8.0 |
% |
10.1128/aac.00355-08 |
| Fusobacterium varium |
Fusobacterium varium |
Activity |
92.0 |
% |
10.1128/aac.00355-08 |
| Fusobacterium varium |
Fusobacterium varium |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Fusobacterium varium |
Fusobacterium varium |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Fusobacterium varium |
Fusobacterium varium |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Fusobacterium varium |
Fusobacterium varium |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium varium |
Fusobacterium varium |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium varium |
Fusobacterium varium |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Fusobacterium varium |
Fusobacterium varium |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Fusobacterium varium |
Fusobacterium varium |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Fusobacterium varium |
Fusobacterium varium |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Fusobacterium varium |
Fusobacterium varium |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
Activity |
0.0 |
% |
10.1128/aac.00422-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
Activity |
0.0 |
% |
10.1128/aac.01538-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
Activity |
9.5 |
% |
10.1128/aac.00422-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
Activity |
90.5 |
% |
10.1128/aac.00422-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
Activity |
99.0 |
% |
10.1128/aac.00192-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
Activity |
99.6 |
% |
10.1128/aac.00971-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
Activity |
99.7 |
% |
10.1128/aac.00971-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
Activity |
100.0 |
% |
10.1128/aac.00192-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
Activity |
100.0 |
% |
10.1128/aac.00422-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
Activity |
100.0 |
% |
10.1128/aac.00971-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.00294-06 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00054-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.031 |
ug.mL-1 |
10.1128/aac.00054-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.06 |
ug.mL-1 |
10.1021/np800503z |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00190-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.063 |
ug.mL-1 |
10.1128/aac.00054-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.00190-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00192-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.125 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00746 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00190-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
3.125 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00422-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.063 |
ug.mL-1 |
10.1128/aac.00054-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.064 |
ug.mL-1 |
10.1128/aac.00960-06 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.094 |
ug.mL-1 |
10.1128/aac.00960-06 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00054-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00422-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00960-06 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.19 |
ug.mL-1 |
10.1128/aac.00960-06 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00054-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00192-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00422-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00422-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00054-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00960-06 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00054-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00422-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.38 |
ug.mL-1 |
10.1128/aac.00960-06 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00054-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00192-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00422-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00960-06 |
| Haemophilus parainfluenzae |
Haemophilus parainfluenzae |
MIC |
0.03 |
ug.mL-1 |
10.1021/np800503z |
| Homo sapiens |
Acetylcholinesterase |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Acetylcholinesterase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Acetylcholinesterase |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A1 receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A2a receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A2a receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A2a receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A3 receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A3 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A3 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1d adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-1d adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2b adrenergic receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2b adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2b adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2c adrenergic receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2c adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2c adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Angiotensin II type 2 (AT-2) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Angiotensin II type 2 (AT-2) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-1 adrenergic receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-1 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-1 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-2 adrenergic receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-2 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-3 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-3 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Bile salt export pump |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bile salt export pump |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Bradykinin B2 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bradykinin B2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Bradykinin B2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Calcitonin receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Calcitonin receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Canalicular multispecific organic anion transporter 1 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 2 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Cannabinoid CB1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cannabinoid CB1 receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cannabinoid CB1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cannabinoid CB1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase II |
IC50 |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase II |
Ki |
nan |
None |
None |
| Homo sapiens |
Caspase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Caspase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cathepsin G |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cathepsin G |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 2 |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 4 |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin A receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cholecystokinin A receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin A receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-2 |
AC50 |
109999.3 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cysteinyl leukotriene receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cysteinyl leukotriene receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 1A2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2A6 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2A6 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2C19 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2C9 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2D6 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2E1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2E1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 3A4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Delta opioid receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Delta opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Delta opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dihydropyrimidine dehydrogenase |
Activity |
1.0 |
None |
10.1016/s0960-894x(00)00575-8 |
| Homo sapiens |
Dopamine D1 receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D2 receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D3 receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D3 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D3 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D4 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D4 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine transporter |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-A |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Endothelin receptor ET-A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-A |
Ki |
nan |
None |
None |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Equilibrative nucleoside transporter 1 |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor beta |
IC50 |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor beta |
Ki |
nan |
None |
None |
| Homo sapiens |
Gamma-aminobutyric acid receptor subunit alpha-1/alpha-2/beta-2/gamma-2 |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Ghrelin receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Glucocorticoid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
HEK293 |
Activity |
nan |
None |
10.1016/j.ejmech.2022.114278 |
| Homo sapiens |
HepaRG |
Activity |
nan |
None |
10.1016/j.ejmech.2022.114278 |
| Homo sapiens |
HERG |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
HERG |
IC50 |
nan |
None |
None |
| Homo sapiens |
HERG |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H1 receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Histamine H1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H2 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Histamine H2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H3 receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
HMG-CoA reductase |
IC50 |
nan |
None |
None |
| Homo sapiens |
HMG-CoA reductase |
Ki |
nan |
None |
None |
| Homo sapiens |
Homo sapiens |
Activity |
2.0 |
% |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
Activity |
4.4 |
L/hr |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
AUC |
129500.0 |
ng.hr.mL-1 |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
AUC |
166500.0 |
ng.hr.mL-1 |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
AUMC |
26709.7 |
mg.hr/L |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
AUMC |
31378.3 |
mg.hr/L |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
CL |
2.4 |
L/hr |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
CL |
3.5 |
L/hr |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
CL |
3.9 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
CL |
6.0 |
L/hr |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
CL_renal |
0.005 |
L/hr |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
CL_renal |
2.73 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
Cmax |
147599.55 |
nM |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
Cmin |
7.6 |
mg/L |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
DILI_Concern |
nan |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
DILI_severity_class |
3.0 |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
fAUC |
157430.0 |
ng.hr.mL-1 |
10.1128/aac.00294-06 |
| Homo sapiens |
Homo sapiens |
fCmax |
32.27 |
ug ml-1 |
10.1128/aac.00294-06 |
| Homo sapiens |
Homo sapiens |
fCmin |
0.91 |
ug ml-1 |
10.1128/aac.00294-06 |
| Homo sapiens |
Homo sapiens |
fT>MIC |
91.0 |
% |
10.1128/aac.00294-06 |
| Homo sapiens |
Homo sapiens |
Kel |
0.16 |
/hr |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
MRT |
163.3 |
hr |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
MRT |
174.3 |
hr |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
Ratio |
0.74 |
None |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
T1/2 |
4.32 |
hr |
10.1128/aac.01582-09 |
| Homo sapiens |
Homo sapiens |
Vd |
0.37 |
L.kg-1 |
10.1128/aac.01582-09 |
| Homo sapiens |
Interleukin-8 receptor A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor A |
Ki |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor B |
IC50 |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor B |
Ki |
nan |
None |
None |
| Homo sapiens |
Kappa opioid receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Kappa opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Kappa opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Leukocyte common antigen |
IC50 |
nan |
None |
None |
| Homo sapiens |
Leukocyte common antigen |
Ki |
nan |
None |
None |
| Homo sapiens |
Leukocyte elastase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Leukocyte elastase |
Ki |
nan |
None |
None |
| Homo sapiens |
Liver microsomes |
Activity |
nan |
None |
10.1021/tx300075j |
| Homo sapiens |
Liver microsomes |
Stability |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
MAP kinase ERK1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK1 |
Ki |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK2 |
Ki |
nan |
None |
None |
| Homo sapiens |
MAP kinase p38 alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase p38 alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase 9 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase 9 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 3 |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Melanocortin receptor 3 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 3 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 4 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Melanocortin receptor 4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Monoamine oxidase A |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Monoamine oxidase A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Monoamine oxidase A |
Ki |
nan |
None |
None |
| Homo sapiens |
Motilin receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Multidrug resistance-associated protein 4 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Mu opioid receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Mu opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Mu opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurokinin 1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neurokinin 1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurokinin 2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neurokinin 2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Neuronal acetylcholine receptor protein alpha-4 subunit |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Norepinephrine transporter |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Norepinephrine transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Norepinephrine transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Peroxisome proliferator-activated receptor gamma |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 3A |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 4D |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 5A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Phosphodiesterase 5A |
Ki |
nan |
None |
None |
| Homo sapiens |
Plasma |
Fu |
nan |
None |
10.1021/acsmedchemlett.5b00026 |
| Homo sapiens |
Platelet activating factor receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Platelet activating factor receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Pregnane X receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Pregnane X receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Progesterone receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Protein kinase C alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
Protein kinase C alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Renal dipeptidase |
Stability |
100.0 |
% |
10.1016/0960-894X(95)00380-C |
| Homo sapiens |
Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 1a (5-HT1a) receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 3a (5-HT3a) receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin transporter |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Sigma opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Sigma opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
THP-1 |
Ratio |
0.2 |
None |
10.1128/aac.00123-08 |
| Homo sapiens |
Thromboxane A2 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Thromboxane A2 receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Thromboxane-A synthase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Thromboxane-A synthase |
Ki |
nan |
None |
None |
| Homo sapiens |
Type-1 angiotensin II receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Tyrosine-protein kinase FYN |
IC50 |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase FYN |
Ki |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase LCK |
IC50 |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase LCK |
Ki |
nan |
None |
None |
| Homo sapiens |
Vascular endothelial growth factor receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vascular endothelial growth factor receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Vascular endothelial growth factor receptor 2 |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vasoactive intestinal polypeptide receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vasoactive intestinal polypeptide receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasopressin V1a receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vasopressin V1a receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vasopressin V1a receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasopressin V2 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Hoylesella oralis |
Hoylesella oralis |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Hoylesella oralis |
Hoylesella oralis |
Activity |
100.0 |
% |
10.1128/aac.00481-10 |
| Hoylesella oralis |
Hoylesella oralis |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Hoylesella oralis |
Hoylesella oralis |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Hoylesella oralis |
Hoylesella oralis |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Hoylesella oralis |
Hoylesella oralis |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Janthinobacterium lividum |
THIN-B proetin |
Kcat/Km |
5.0 |
10'6/M/s |
10.1128/aac.01062-07 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(00)00253-5 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(00)00575-8 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(01)00451-6 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(02)00948-4 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(98)00270-4 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(99)00407-2 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(99)00646-0 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(99)00692-7 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.031 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC50 |
0.06 |
ug.mL-1 |
10.1021/ml200012f |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC90 |
0.25 |
ug.mL-1 |
10.1021/ml200012f |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
Activity |
0.0 |
% |
10.1128/aac.00400-09 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
Activity |
100.0 |
% |
10.1128/aac.00400-09 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(99)00692-7 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
0.049 |
ug.mL-1 |
10.1021/np049577a |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
0.049 |
ug.mL-1 |
10.1021/np060206z |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.5b00127 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
32.0 |
ug.mL-1 |
10.1039/C5MD00380F |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00260-09 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01355-08 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Klebsiella pneumoniae |
Beta-lactamase AH27 CTX-M-15 |
Kcat |
0.004 |
/s |
10.1128/aac.00461-09 |
| Klebsiella pneumoniae |
Beta-lactamase AH27 CTX-M-15 |
Km |
nan |
None |
10.1128/aac.00461-09 |
| Klebsiella pneumoniae |
Beta-lactamase AH27 CTX-M-15 |
Ratio |
nan |
None |
10.1128/aac.00461-09 |
| Klebsiella pneumoniae |
Beta-lactamase NDM-1 |
Kcat |
12.0 |
/s |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
Beta-lactamase NDM-1 |
Kcat/Km |
0.25 |
/s/microM |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
Beta-lactamase NDM-1 |
Kd |
11000.0 |
nM |
10.1016/j.bmcl.2016.03.004 |
| Klebsiella pneumoniae |
Beta-lactamase NDM-1 |
Km |
49000.0 |
nM |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
Beta-lactamase NDM-1 |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115598 |
| Klebsiella pneumoniae |
Beta-lactamase NDM-1 |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115598 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-1 |
Activity |
0.00041 |
% |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-1 |
Activity |
0.015 |
% |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-1 |
Kcat |
0.0017 |
/s |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-1 |
Kcat/Km |
0.0004 |
/s/microM |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Beta-lactamase SHV-1 |
Km |
4200.0 |
nM |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Activity |
0.92 |
% |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Activity |
2.0 |
% |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Activity |
31.0 |
U |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Activity |
37.0 |
% |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Activity |
55.0 |
U |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Activity |
57.0 |
% |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Activity |
64.0 |
% |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Activity |
76.0 |
U |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Kcat |
3.0 |
/s |
10.1128/aac.00491-07 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Kcat |
3.6 |
/s |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Kcat/Km |
0.28 |
/s/microM |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Kcat/Km |
250.0 |
/mM/s |
10.1128/aac.00491-07 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Km |
12000.0 |
nM |
10.1128/aac.00491-07 |
| Klebsiella pneumoniae |
Carbepenem-hydrolyzing beta-lactamase KPC |
Km |
13000.0 |
nM |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Class A carbapenemase |
Activity |
0.06 |
umol |
10.1128/aac.01180-07 |
| Klebsiella pneumoniae |
Extended spectrum beta-lactamase CTX-M-71 |
Kcat |
0.07 |
/s |
10.1128/aac.00461-09 |
| Klebsiella pneumoniae |
Extended spectrum beta-lactamase CTX-M-71 |
Km |
nan |
None |
10.1128/aac.00461-09 |
| Klebsiella pneumoniae |
Extended spectrum beta-lactamase CTX-M-71 |
Ratio |
nan |
None |
10.1128/aac.00461-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
0.0 |
% |
10.1128/aac.00381-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
0.0 |
% |
10.1128/aac.00400-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
0.2 |
% |
10.1128/aac.00381-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
0.3 |
% |
10.1128/aac.00381-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
4.5 |
% |
10.1128/aac.00381-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
9.1 |
% |
10.1128/aac.01538-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
12.5 |
% |
10.1128/aac.01538-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
13.6 |
% |
10.1128/aac.01538-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
17.8 |
% |
10.1128/aac.01538-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
18.9 |
% |
10.1128/aac.01538-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
95.5 |
% |
10.1128/aac.00381-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
99.7 |
% |
10.1128/aac.00381-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
99.8 |
% |
10.1128/aac.00381-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
100.0 |
% |
10.1128/aac.00400-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
100.0 |
% |
10.1128/aac.01509-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
nan |
None |
10.1016/j.ejmech.2022.114571 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
nan |
None |
10.1128/aac.01525-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
deltalog10CFU |
1.41 |
None |
10.1021/acs.jmedchem.5b00127 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
ED50 |
100.0 |
mg.kg-1 |
10.1021/acs.jmedchem.6b01261 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
0.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
3.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
5.0 |
% |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
12.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
16.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
18.0 |
% |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
30.0 |
% |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
38.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
45.0 |
% |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
47.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
50.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
56.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
58.0 |
% |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
59.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
62.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
65.0 |
% |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
68.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
69.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
72.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
75.0 |
% |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
78.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
80.0 |
% |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
85.0 |
% |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
88.0 |
% |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
90.0 |
% |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
fT>MIC |
100.0 |
% |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Inhibition |
0.03 |
% |
10.6019/CHEMBL4513141 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Inhibition |
nan |
% |
10.1016/j.bmc.2021.116128 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Inhibition |
nan |
% |
10.1128/aac.01452-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
IZ |
13.0 |
mm |
10.1128/aac.01325-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
IZ |
14.0 |
mm |
10.1128/aac.01325-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
IZ |
23.0 |
mm |
10.1128/aac.00543-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
IZ |
27.0 |
mm |
10.1128/aac.01325-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
log10cfu |
3.0 |
None |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MBC |
0.06 |
ug ml-1 |
10.1128/aac.01452-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MBC |
16.0 |
ug ml-1 |
10.1128/aac.01452-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MBC |
64.0 |
ug ml-1 |
10.1021/acs.jmedchem.2c01469 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.00294-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00083-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.016 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00746 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00715-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01452-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.031 |
ug.mL-1 |
10.1016/j.bmc.2021.116343 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.01301-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.04 |
ug.mL-1 |
10.1021/jm010546b |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.047 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.047 |
ug.mL-1 |
10.1128/aac.01301-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1021/np800503z |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00083-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01452-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.01301-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.094 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.094 |
ug.mL-1 |
10.1128/aac.01301-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.bmc.2013.09.041 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00830-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.128 |
ug.mL-1 |
10.1016/j.ejmech.2021.113975 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm400560z |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00008-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01325-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2022.114571 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00461-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00543-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.01301-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116343 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.02.024 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114278 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b00091 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/ml200012f |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1039/C5MD00380F |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00008-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00158-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01301-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.01301-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b00091 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00008-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00026-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00158-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00260-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00299-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01198-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01301-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01818-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.00436-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.5b00127 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1039/C5MD00380F |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00008-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00158-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00197-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00299-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00458-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00461-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00736-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01198-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01301-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01325-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01452-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01539-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01818-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.01180-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.01672-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116142 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.031 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.5b00127 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00008-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00158-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00299-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01325-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01818-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.01301-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.031 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.014 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114278 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01257 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01469 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.5b00127 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b00091 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1039/C5MD00380F |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00008-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00011-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00260-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01355-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01672-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.031 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.02.024 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01261 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1039/C5MD00380F |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00008-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00137-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00260-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00299-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00736-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00752-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01053-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01247-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01355-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01672-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01818-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.031 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.058 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114599 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jmedchem.5b00127 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01261 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm400560z |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1021/np800503z |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00008-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00543-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01190-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01355-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01818-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127956 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
128.0 |
ug.mL-1 |
10.1021/np4000944 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
128.0 |
ug.mL-1 |
10.1039/C5MD00380F |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00008-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01198-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01818-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116128 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01469 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00008-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01099-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01198-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01539-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00008-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16000.0 |
nM |
10.1021/acs.jmedchem.1c00621 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64000.0 |
nM |
10.1021/acs.jmedchem.1c00621 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
nan |
None |
10.1016/j.ejmech.2017.10.044 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.03 |
ug.mL-1 |
10.1021/jm400560z |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00083-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01450-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01509-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.047 |
ug.mL-1 |
10.1128/aac.00171-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.06 |
ug.mL-1 |
10.1021/ml200012f |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00083-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00255 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC50 |
32.0 |
ug.mL-1 |
10.1021/jm400560z |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00083-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.01450-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.064 |
ug.mL-1 |
10.1128/aac.00171-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.094 |
ug.mL-1 |
10.1128/aac.00171-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00171-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.19 |
ug.mL-1 |
10.1128/aac.00171-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.25 |
ug.mL-1 |
10.1021/jm400560z |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01509-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00083-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.07.005 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
32.0 |
ug.mL-1 |
10.1021/ml200012f |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
64.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00255 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
64.0 |
ug.mL-1 |
10.1021/jm400560z |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MPC |
0.06 |
ug ml-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MPC |
0.125 |
ug ml-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MPC |
0.5 |
ug ml-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MPC |
8.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MPC |
16.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MPC |
32.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MPC |
64.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Ratio |
1.0 |
None |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Ratio |
2.0 |
None |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Ratio |
4.0 |
None |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Ratio |
8.0 |
None |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Ratio |
16.0 |
None |
10.1128/aac.00033-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Survival |
0.0 |
% |
10.1021/acs.jmedchem.6b01261 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Survival |
69.0 |
% |
10.1039/C5MD00380F |
| Klebsiella pneumoniae |
Metallo-beta-lactamase |
Activity |
42.0 |
U |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase |
Activity |
55.0 |
U |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase |
Activity |
57.0 |
% |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase |
Activity |
64.0 |
% |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase |
Activity |
76.0 |
U |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase |
Activity |
80.0 |
% |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase |
Activity |
80.0 |
U |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase |
Activity |
100.0 |
% |
10.1128/aac.00690-09 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase VIM-2 |
Kcat |
1.0 |
/s |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase VIM-2 |
Kcat/Km |
0.28 |
/s/microM |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
Metallo-beta-lactamase VIM-2 |
Km |
5000.0 |
nM |
10.1128/aac.00774-09 |
| Klebsiella pneumoniae |
OXA-48 |
Activity |
0.05 |
umol/min/mg |
10.1128/aac.00543-08 |
| Klebsiella pneumoniae |
OXA-48 |
Ka |
4.0 |
10'4/M/s |
10.1021/acs.jmedchem.6b00660 |
| Klebsiella pneumoniae |
OXA-48 |
Kcat |
0.098 |
/s |
10.1021/acs.jmedchem.6b00660 |
| Klebsiella pneumoniae |
OXA-48 |
Kcat/Km |
9.8 |
10'4/M/s |
10.1021/acs.jmedchem.6b00660 |
| Klebsiella pneumoniae |
OXA-48 |
Kd |
0.3463 |
/s |
10.1021/acs.jmedchem.6b00660 |
| Klebsiella pneumoniae |
OXA-48 |
Kd |
850.0 |
nM |
10.1021/acs.jmedchem.6b00660 |
| Klebsiella pneumoniae |
OXA-48 |
Km |
1000.0 |
nM |
10.1021/acs.jmedchem.6b00660 |
| Klebsiella sp. |
Klebsiella sp. |
Activity |
20.0 |
% |
10.1128/aac.01114-07 |
| Klebsiella sp. |
Klebsiella sp. |
Activity |
61.7 |
% |
10.1128/aac.01114-07 |
| Klebsiella sp. |
Klebsiella sp. |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.01114-07 |
| Klebsiella sp. |
Klebsiella sp. |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01114-07 |
| Lacrimispora sphenoides |
Lacrimispora sphenoides |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Lacrimispora sphenoides |
Lacrimispora sphenoides |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Lacrimispora sphenoides |
Lacrimispora sphenoides |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Lacticaseibacillus casei |
Lacticaseibacillus casei |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Lactiplantibacillus plantarum |
Lactiplantibacillus plantarum |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Lactobacillus acidophilus |
Lactobacillus acidophilus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Limosilactobacillus fermentum |
Limosilactobacillus fermentum |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Limosilactobacillus reuteri |
Limosilactobacillus reuteri |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Micrococcus luteus |
Micrococcus luteus |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Micrococcus luteus |
Micrococcus luteus |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Micrococcus luteus |
Micrococcus luteus |
MIC |
nan |
None |
10.1021/acs.jmedchem.2c01674 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
0.004 |
ug.mL-1 |
10.1021/np800503z |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
0.008 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00746 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
0.004 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
0.008 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
0.008 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
0.008 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Morganella morganii |
Morganella morganii |
MIC |
0.06 |
ug.mL-1 |
10.1016/S0960-894X(97)00282-5 |
| Morganella morganii |
Morganella morganii |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Morganella morganii |
Morganella morganii |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Morganella morganii |
Morganella morganii |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Mus musculus |
Mus musculus |
AUC |
0.0 |
hr |
10.1016/s0960-894x(99)00407-2 |
| Mus musculus |
Mus musculus |
AUC |
3.29 |
ug ml-1 |
10.1016/s0960-894x(99)00692-7 |
| Mus musculus |
Mus musculus |
AUC |
6860.0 |
ng.hr.mL-1 |
10.1016/s0960-894x(99)00407-2 |
| Mus musculus |
Mus musculus |
Cmax |
19819.02 |
nM |
10.1016/s0960-894x(99)00692-7 |
| Mus musculus |
Mus musculus |
Cmax |
40602.92 |
nM |
10.1016/s0960-894x(99)00407-2 |
| Mus musculus |
Mus musculus |
ED50 |
7.88 |
mg.kg-1 |
10.1016/S0960-894X(97)00230-8 |
| Mus musculus |
Mus musculus |
PD50 |
0.65 |
mg kg-1 |
10.1016/s0960-894x(99)00407-2 |
| Mus musculus |
Mus musculus |
PD50 |
1.11 |
mg kg-1 |
10.1016/s0960-894x(02)00948-4 |
| Mus musculus |
Mus musculus |
PD50 |
1.24 |
mg kg-1 |
10.1016/s0960-894x(99)00692-7 |
| Mus musculus |
Mus musculus |
PD50 |
4.26 |
mg kg-1 |
10.1016/s0960-894x(99)00407-2 |
| Mus musculus |
Mus musculus |
PD50 |
4.49 |
mg kg-1 |
10.1016/s0960-894x(02)00948-4 |
| Mus musculus |
Mus musculus |
PD50 |
4.55 |
mg kg-1 |
10.1016/s0960-894x(99)00407-2 |
| Mus musculus |
Mus musculus |
PD50 |
4.6 |
mg kg-1 |
10.1016/s0960-894x(99)00692-7 |
| Mus musculus |
Mus musculus |
PD50 |
4.72 |
mg kg-1 |
10.1016/s0960-894x(02)00948-4 |
| Mus musculus |
Mus musculus |
PD50 |
5.43 |
mg kg-1 |
10.1016/s0960-894x(02)00948-4 |
| Mus musculus |
Mus musculus |
PD50 |
11.1 |
mg kg-1 |
10.1016/s0960-894x(99)00407-2 |
| Mus musculus |
Mus musculus |
PD50 |
nan |
None |
10.1016/s0960-894x(99)00692-7 |
| Mus musculus |
Mus musculus |
Recovery |
25.0 |
% |
10.1016/0960-894X(95)00380-C |
| Mus musculus |
Mus musculus |
T1/2 |
0.24 |
hr |
10.1016/s0960-894x(99)00692-7 |
| Mus musculus |
Mus musculus |
T1/2 |
0.27 |
hr |
10.1016/s0960-894x(99)00407-2 |
| Mus musculus |
Mus musculus |
Tmax |
0.17 |
hr |
10.1016/s0960-894x(99)00407-2 |
| Mus musculus |
Mus musculus |
Tmax |
0.21 |
hr |
10.1016/s0960-894x(99)00692-7 |
| Mus musculus |
Nitric oxide synthase, inducible |
IC50 |
nan |
None |
None |
| Mus musculus |
Nitric oxide synthase, inducible |
Ki |
nan |
None |
None |
| Mus musculus |
Plasma |
fAUC |
4466.67 |
ng.hr.mL-1 |
10.1128/aac.00642-09 |
| Mus musculus |
Plasma |
fAUC |
30616.67 |
ng.hr.mL-1 |
10.1128/aac.00642-09 |
| Mus musculus |
Plasma |
fCmax |
11.0 |
ug ml-1 |
10.1128/aac.00642-09 |
| Mus musculus |
Plasma |
fCmax |
72.0 |
ug ml-1 |
10.1128/aac.00642-09 |
| Mus musculus |
Plasma |
T1/2 |
0.1433 |
hr |
10.1128/aac.00642-09 |
| Mus musculus |
Plasma |
T1/2 |
0.2267 |
hr |
10.1128/aac.00642-09 |
| Mus musculus |
Plasma |
Tmax |
0.125 |
hr |
10.1128/aac.00642-09 |
| Mycobacterium avium |
Mycobacterium avium |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.7 |
log10CFU |
10.1021/acs.jmedchem.2c00227 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.0 |
log10CFU |
10.1021/acs.jmedchem.2c00227 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmc.2013.05.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2017.06.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
10000.0 |
nM |
10.1021/acs.jmedchem.2c00227 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC50 |
0.008 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC90 |
0.015 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Nocardia brasiliensis |
Nocardia brasiliensis |
MIC |
0.001 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia brasiliensis |
Nocardia brasiliensis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01520-09 |
| Nocardia brasiliensis |
Nocardia brasiliensis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01520-09 |
| Nocardia carnea |
Nocardia carnea |
MIC |
0.001 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia cyriacigeorgica |
Nocardia cyriacigeorgica |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia farcinica |
Nocardia farcinica |
MIC |
0.002 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia nova |
Nocardia nova |
MIC |
0.0005 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia otitidiscaviarum |
Nocardia otitidiscaviarum |
MIC |
0.001 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia sp. |
Nocardia sp. |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia transvalensis |
Nocardia transvalensis |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Oryctolagus cuniculus |
Angiotensin-converting enzyme |
IC50 |
nan |
None |
None |
| Oryctolagus cuniculus |
Angiotensin-converting enzyme |
Ki |
nan |
None |
None |
| Oryctolagus cuniculus |
Arachidonate 15-lipoxygenase |
IC50 |
nan |
None |
None |
| Oryctolagus cuniculus |
Arachidonate 15-lipoxygenase |
Ki |
nan |
None |
None |
| Paeniclostridium sordellii |
Paeniclostridium sordellii |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Paeniclostridium sordellii |
Paeniclostridium sordellii |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
Activity |
1.1 |
% |
10.1128/aac.01435-06 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
Activity |
98.0 |
% |
10.1128/aac.00481-10 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC |
0.13 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Parabacteroides merdae |
Parabacteroides merdae |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Parabacteroides merdae |
Parabacteroides merdae |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Parabacteroides merdae |
Parabacteroides merdae |
Activity |
0.5 |
% |
10.1128/aac.01435-06 |
| Parabacteroides merdae |
Parabacteroides merdae |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Parabacteroides merdae |
Parabacteroides merdae |
MIC |
0.4 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Parabacteroides merdae |
Parabacteroides merdae |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Parabacteroides merdae |
Parabacteroides merdae |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Parabacteroides merdae |
Parabacteroides merdae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Parabacteroides merdae |
Parabacteroides merdae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Parabacteroides merdae |
Parabacteroides merdae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Paraclostridium bifermentans |
Paraclostridium bifermentans |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Parvimonas micra |
Parvimonas micra |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Parvimonas micra |
Parvimonas micra |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Parvimonas micra |
Parvimonas micra |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Parvimonas micra |
Parvimonas micra |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Parvimonas micra |
Parvimonas micra |
Activity |
100.0 |
% |
10.1128/aac.00355-08 |
| Parvimonas micra |
Parvimonas micra |
MIC |
0.01 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Parvimonas micra |
Parvimonas micra |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Parvimonas micra |
Parvimonas micra |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Parvimonas micra |
Parvimonas micra |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Parvimonas micra |
Parvimonas micra |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Parvimonas micra |
Parvimonas micra |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Parvimonas micra |
Parvimonas micra |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Parvimonas micra |
Parvimonas micra |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Parvimonas micra |
Parvimonas micra |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Parvimonas micra |
Parvimonas micra |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Parvimonas micra |
Parvimonas micra |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Parvimonas micra |
Parvimonas micra |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Parvimonas micra |
Parvimonas micra |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Parvimonas micra |
Parvimonas micra |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Parvimonas micra |
Parvimonas micra |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Parvimonas micra |
Parvimonas micra |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Parvimonas micra |
Parvimonas micra |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Pasteurella multocida |
Pasteurella multocida |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Pasteurella multocida |
Pasteurella multocida |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Pectobacterium atrosepticum |
Pectobacterium atrosepticum |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01062-07 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
Activity |
100.0 |
% |
10.1128/aac.00355-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
Activity |
100.0 |
% |
10.1128/aac.00481-10 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC50 |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC50 |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC90 |
0.03 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC90 |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
Activity |
100.0 |
% |
10.1128/aac.00355-08 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
Activity |
100.0 |
% |
10.1128/aac.00481-10 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC |
0.01 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Peptostreptococcus sp. |
Peptostreptococcus sp. |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Peptostreptococcus sp. |
Peptostreptococcus sp. |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Peptostreptococcus sp. |
Peptostreptococcus sp. |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Peptostreptococcus sp. |
Peptostreptococcus sp. |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
Activity |
0.0 |
% |
10.1128/aac.01435-06 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
Activity |
4.0 |
% |
10.1128/aac.00355-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
Activity |
96.0 |
% |
10.1128/aac.00355-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
Activity |
98.0 |
% |
10.1128/aac.00481-10 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC |
0.13 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC |
0.47 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01435-06 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Porphyromonas asaccharolytica |
Porphyromonas asaccharolytica |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Porphyromonas asaccharolytica |
Porphyromonas asaccharolytica |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Porphyromonas asaccharolytica |
Porphyromonas asaccharolytica |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Porphyromonas asaccharolytica |
Porphyromonas asaccharolytica |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Porphyromonas asaccharolytica |
Porphyromonas asaccharolytica |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Porphyromonas asaccharolytica |
Porphyromonas asaccharolytica |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Porphyromonas asaccharolytica |
Porphyromonas asaccharolytica |
MIC90 |
0.015 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Porphyromonas asaccharolytica |
Porphyromonas asaccharolytica |
MIC90 |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Porphyromonas gingivalis |
Porphyromonas gingivalis |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Porphyromonas gingivalis |
Porphyromonas gingivalis |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Porphyromonas gingivalis |
Porphyromonas gingivalis |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Porphyromonas gingivalis |
Porphyromonas gingivalis |
MIC90 |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Porphyromonas levii |
Porphyromonas levii |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Porphyromonas somerae |
Porphyromonas somerae |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Porphyromonas somerae |
Porphyromonas somerae |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Porphyromonas somerae |
Porphyromonas somerae |
MIC90 |
0.015 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Prevotella bivia |
Prevotella bivia |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Prevotella bivia |
Prevotella bivia |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Prevotella bivia |
Prevotella bivia |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Prevotella bivia |
Prevotella bivia |
Activity |
100.0 |
% |
10.1128/aac.00355-08 |
| Prevotella bivia |
Prevotella bivia |
Activity |
100.0 |
% |
10.1128/aac.00481-10 |
| Prevotella bivia |
Prevotella bivia |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Prevotella bivia |
Prevotella bivia |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella bivia |
Prevotella bivia |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Prevotella bivia |
Prevotella bivia |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Prevotella bivia |
Prevotella bivia |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella bivia |
Prevotella bivia |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Prevotella bivia |
Prevotella bivia |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Prevotella bivia |
Prevotella bivia |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Prevotella bivia |
Prevotella bivia |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella bivia |
Prevotella bivia |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Prevotella bivia |
Prevotella bivia |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Prevotella bivia |
Prevotella bivia |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Prevotella buccae |
Prevotella buccae |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Prevotella buccae |
Prevotella buccae |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Prevotella buccae |
Prevotella buccae |
Activity |
100.0 |
% |
10.1128/aac.00355-08 |
| Prevotella buccae |
Prevotella buccae |
Activity |
100.0 |
% |
10.1128/aac.00481-10 |
| Prevotella buccae |
Prevotella buccae |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Prevotella buccae |
Prevotella buccae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Prevotella buccae |
Prevotella buccae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella buccae |
Prevotella buccae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Prevotella buccae |
Prevotella buccae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella buccae |
Prevotella buccae |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Prevotella buccae |
Prevotella buccae |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Prevotella buccae |
Prevotella buccae |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella buccae |
Prevotella buccae |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Prevotella buccae |
Prevotella buccae |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Prevotella corporis |
Prevotella corporis |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella corporis |
Prevotella corporis |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Prevotella corporis |
Prevotella corporis |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella corporis |
Prevotella corporis |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella denticola |
Prevotella denticola |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella denticola |
Prevotella denticola |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Prevotella denticola |
Prevotella denticola |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella denticola |
Prevotella denticola |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella disiens |
Prevotella disiens |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella disiens |
Prevotella disiens |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella disiens |
Prevotella disiens |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella intermedia |
Prevotella intermedia |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Prevotella intermedia |
Prevotella intermedia |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| Prevotella intermedia |
Prevotella intermedia |
Activity |
90.0 |
% |
10.1128/aac.00910-07 |
| Prevotella intermedia |
Prevotella intermedia |
Activity |
99.0 |
% |
10.1128/aac.00910-07 |
| Prevotella intermedia |
Prevotella intermedia |
Activity |
100.0 |
% |
10.1128/aac.00355-08 |
| Prevotella intermedia |
Prevotella intermedia |
Activity |
100.0 |
% |
10.1128/aac.00481-10 |
| Prevotella intermedia |
Prevotella intermedia |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella intermedia |
Prevotella intermedia |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Prevotella intermedia |
Prevotella intermedia |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella intermedia |
Prevotella intermedia |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Prevotella intermedia |
Prevotella intermedia |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Prevotella intermedia |
Prevotella intermedia |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella intermedia |
Prevotella intermedia |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Prevotella intermedia |
Prevotella intermedia |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Prevotella intermedia |
Prevotella intermedia |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Prevotella intermedia |
Prevotella intermedia |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Prevotella intermedia |
Prevotella intermedia |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Prevotella intermedia |
Prevotella intermedia |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella intermedia |
Prevotella intermedia |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
Activity |
0.0 |
% |
10.1128/aac.00355-08 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
Activity |
100.0 |
% |
10.1128/aac.00355-08 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00355-08 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Prevotella nigrescens |
Prevotella nigrescens |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella nigrescens |
Prevotella nigrescens |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Prevotella nigrescens |
Prevotella nigrescens |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Priestia megaterium |
Priestia megaterium |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Priestia megaterium |
Priestia megaterium |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Propionibacterium |
Propionibacterium |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Propionibacterium |
Propionibacterium |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Propionibacterium |
Propionibacterium |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Propionibacterium |
Propionibacterium |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Proteus mirabilis |
Proteus mirabilis |
Activity |
0.0 |
% |
10.1128/aac.00381-08 |
| Proteus mirabilis |
Proteus mirabilis |
Activity |
0.0 |
% |
10.1128/aac.00400-09 |
| Proteus mirabilis |
Proteus mirabilis |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Proteus mirabilis |
Proteus mirabilis |
Activity |
100.0 |
% |
10.1128/aac.00381-08 |
| Proteus mirabilis |
Proteus mirabilis |
Activity |
100.0 |
% |
10.1128/aac.00400-09 |
| Proteus mirabilis |
Proteus mirabilis |
Activity |
100.0 |
% |
10.1128/aac.01509-06 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2022.114571 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01114-07 |
| Proteus mirabilis |
Proteus mirabilis |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01509-06 |
| Proteus mirabilis |
Proteus mirabilis |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Proteus mirabilis |
Proteus mirabilis |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Proteus mirabilis |
Proteus mirabilis |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Proteus mirabilis |
Proteus mirabilis |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Proteus mirabilis |
Proteus mirabilis |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Proteus mirabilis |
Proteus mirabilis |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Proteus mirabilis |
Proteus mirabilis |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Proteus mirabilis |
Proteus mirabilis |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Proteus mirabilis |
Proteus mirabilis |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Proteus mirabilis |
Proteus mirabilis |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01509-06 |
| Proteus mirabilis |
Proteus mirabilis |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Proteus vulgaris |
Proteus vulgaris |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
0.1 |
ug.mL-1 |
10.1016/0960-894X(95)00380-C |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
0.1 |
ug.mL-1 |
10.1016/S0960-894X(97)00230-8 |
| Proteus vulgaris |
Proteus vulgaris |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Proteus vulgaris |
Proteus vulgaris |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Proteus vulgaris |
Proteus vulgaris |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Proteus vulgaris |
Proteus vulgaris |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Proteus vulgaris |
Proteus vulgaris |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Proteus vulgaris |
Proteus vulgaris |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Providencia rettgeri |
Providencia rettgeri |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Providencia rettgeri |
Providencia rettgeri |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Providencia rettgeri |
Providencia rettgeri |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Providencia rettgeri |
Providencia rettgeri |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Providencia rettgeri |
Providencia rettgeri |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Providencia rettgeri |
Providencia rettgeri |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Providencia rettgeri |
Providencia rettgeri |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01312-09 |
| Providencia rettgeri |
Providencia rettgeri |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Providencia rettgeri |
Providencia rettgeri |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Providencia rettgeri |
Providencia rettgeri |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Providencia rettgeri |
Providencia rettgeri |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Providencia rettgeri |
Providencia rettgeri |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Providencia stuartii |
Providencia stuartii |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Providencia stuartii |
Providencia stuartii |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Providencia stuartii |
Providencia stuartii |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Providencia stuartii |
Providencia stuartii |
MIC |
8.0 |
ug.mL-1 |
10.1039/C5MD00380F |
| Providencia stuartii |
Providencia stuartii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00017-09 |
| Providencia stuartii |
Providencia stuartii |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Providencia stuartii |
Providencia stuartii |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Providencia stuartii |
Providencia stuartii |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Providencia stuartii |
Providencia stuartii |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Beta-lactamase |
Kcat |
nan |
None |
10.1128/aac.01397-09 |
| Pseudomonas aeruginosa |
Beta-lactamase |
Kcat/Km |
0.2 |
/uM/s |
10.1128/aac.01397-09 |
| Pseudomonas aeruginosa |
Beta-lactamase |
Km |
nan |
None |
10.1128/aac.01397-09 |
| Pseudomonas aeruginosa |
Beta-lactamase IMP-1 |
Activity |
9.6 |
% |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase IMP-1 |
Activity |
31.0 |
% |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase IMP-1 |
Kcat |
26.0 |
/s |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase IMP-1 |
Kcat/Km |
4.0 |
/s/microM |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase IMP-1 |
Km |
6500.0 |
nM |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase OXA-10 |
Activity |
0.031 |
% |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase OXA-10 |
Activity |
nan |
None |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase OXA-10 |
Kcat |
0.005 |
/s |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase OXA-10 |
Kcat/Km |
nan |
None |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase OXA-10 |
Km |
nan |
None |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-1 |
Kcat |
20.0 |
/s |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-1 |
Kcat/Km |
2.8 |
/M/s |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-1 |
Km |
72000.0 |
nM |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Activity |
1.8 |
% |
10.1128/aac.00175-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Activity |
1.8 |
% |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Activity |
62.0 |
% |
10.1128/aac.00175-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Activity |
62.0 |
% |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Kcat |
2.1 |
/s |
10.1128/aac.00175-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Kcat |
2.1 |
/s |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Kcat |
5.0 |
/s |
10.1128/aac.00166-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Kcat |
8.5 |
/s |
10.1128/aac.01397-09 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Kcat/Km |
0.053 |
/s/microM |
10.1128/aac.00175-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Kcat/Km |
0.053 |
/s/microM |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Kcat/Km |
0.9 |
/uM/s |
10.1128/aac.01397-09 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Kcat/Km |
2.5 |
/uM/s |
10.1128/aac.00166-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Kd |
12000.0 |
nM |
10.1021/acs.jmedchem.5b01289 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Km |
2000.0 |
nM |
10.1021/acs.jmedchem.5b01289 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Km |
2000.0 |
nM |
10.1128/aac.00166-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Km |
9400.0 |
nM |
10.1128/aac.01397-09 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Km |
40000.0 |
nM |
10.1128/aac.00175-08 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
Km |
40000.0 |
nM |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115598 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115598 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115598 |
| Pseudomonas aeruginosa |
Beta-lactamase VIM-2 |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115598 |
| Pseudomonas aeruginosa |
Class B carbapenemase VIM-13 |
Kcat |
9.0 |
/s |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Class B carbapenemase VIM-13 |
Kcat/Km |
5.92 |
/M/s |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Class B carbapenemase VIM-13 |
Km |
15500.0 |
nM |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Metallo-beta-lactamase VIM-11 |
Kcat |
3.2 |
/s |
10.1128/aac.01025-07 |
| Pseudomonas aeruginosa |
Metallo-beta-lactamase VIM-11 |
Kcat/Km |
1.4 |
10'6/M/s |
10.1128/aac.01025-07 |
| Pseudomonas aeruginosa |
Metallo-beta-lactamase VIM-11 |
Km |
22700.0 |
nM |
10.1128/aac.01025-07 |
| Pseudomonas aeruginosa |
Metallo-beta-lactamase VIM-2 |
Kcat |
3.5 |
/s |
10.1128/aac.01025-07 |
| Pseudomonas aeruginosa |
Metallo-beta-lactamase VIM-2 |
Kcat/Km |
1.4 |
10'6/M/s |
10.1128/aac.01025-07 |
| Pseudomonas aeruginosa |
Metallo-beta-lactamase VIM-2 |
Km |
24500.0 |
nM |
10.1128/aac.01025-07 |
| Pseudomonas aeruginosa |
Metallo-b-lactamase |
Kcat |
42.0 |
/s |
10.1128/aac.00166-08 |
| Pseudomonas aeruginosa |
Metallo-b-lactamase |
Kcat/Km |
1.1 |
/uM/s |
10.1128/aac.00166-08 |
| Pseudomonas aeruginosa |
Metallo-b-lactamase |
Km |
38000.0 |
nM |
10.1128/aac.00166-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
AAC |
-22.46 |
deltalog10CFU/ml.hr |
10.1128/aac.00160-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
AAC |
-19.58 |
deltalog10CFU/ml.hr |
10.1128/aac.00160-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
AAC |
5.3 |
deltalog10CFU/ml.hr |
10.1128/aac.00160-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
0.0 |
% |
10.1128/aac.01538-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
0.7 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
1.0 |
10'-5 ug/ml |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
1.0 |
10'-7 ug/ml |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
2.0 |
ug ml-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
2.9 |
deltalog10CFU |
10.1021/acs.jmedchem.6b01903 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
3.0 |
ug ml-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
3.6 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
3.7 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
4.1 |
% |
10.1128/aac.00400-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
4.2 |
deltalog10CFU |
10.1021/acs.jmedchem.6b01903 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
4.6 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
4.7 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
4.9 |
deltalog10CFU |
10.1021/acs.jmedchem.6b01903 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
6.5 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
7.0 |
% |
10.1128/aac.01128-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
7.9 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
8.1 |
% |
10.1128/aac.00400-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
10.2 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
12.4 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
13.33 |
% |
10.1016/j.ejmech.2020.112252 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
15.67 |
% |
10.1016/j.ejmech.2020.112252 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
16.9 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
17.2 |
% |
10.1128/aac.00851-06 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
18.0 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
32.0 |
ug ml-1 |
10.1128/aac.01043-06 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
35.5 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
40.6 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
42.5 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
52.0 |
% |
10.1128/aac.01104-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
52.1 |
% |
10.1128/aac.00834-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
56.1 |
% |
10.1128/aac.00851-06 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
59.5 |
% |
10.1128/aac.01483-06 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
60.9 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
68.0 |
% |
10.1128/aac.00810-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
74.1 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
76.9 |
% |
10.1128/aac.00851-06 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
83.9 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
85.3 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
87.0 |
% |
10.1128/aac.00679-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
87.8 |
% |
10.1128/aac.00400-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
88.8 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
95.0 |
% |
10.1128/aac.00453-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
98.5 |
% |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
602.0 |
mm3 |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
810.0 |
mm3 |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
862.0 |
mm3 |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
926.0 |
mm3 |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
992.0 |
mm3 |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
1030.0 |
mm3 |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
1190.0 |
mm3 |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
1316.0 |
mm3 |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
nan |
None |
10.1016/0960-894X(95)00202-5 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
nan |
None |
10.1016/j.ejmech.2020.112252 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
nan |
None |
10.1016/j.ejmech.2022.114278 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
nan |
None |
10.1128/aac.00160-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
nan |
None |
10.1128/aac.01278-06 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
nan |
None |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
nan |
None |
10.1128/aac.01529-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
deltalog10CFU |
-1.23 |
/ml |
10.1128/aac.00160-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
deltalog10CFU |
-1.1 |
None |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
deltalog10CFU |
-1.09 |
/ml |
10.1128/aac.00160-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
deltalog10CFU |
-1.0 |
None |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
deltalog10CFU |
-0.9 |
None |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
deltalog10CFU |
-0.83 |
/ml |
10.1128/aac.00160-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
deltalog10CFU |
0.2 |
None |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
deltalog10CFU |
0.5 |
None |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
deltalog10CFU |
0.7 |
None |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
FC |
0.2 |
None |
10.1021/jm501050e |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
FC |
1.0 |
None |
10.1021/acs.jmedchem.1c00888 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
fT>MIC |
38.0 |
% |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
fT>MIC |
47.0 |
% |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
fT>MIC |
50.0 |
% |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
fT>MIC |
56.0 |
% |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
fT>MIC |
63.0 |
% |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
fT>MIC |
69.0 |
% |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
fT>MIC |
75.0 |
% |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
fT>MIC |
78.0 |
% |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
fT>MIC |
82.0 |
% |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
fT>MIC |
94.0 |
% |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
fT>MIC |
100.0 |
% |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IC50 |
20.0 |
nM |
10.1021/acs.jnatprod.9b00187 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Inhibition |
8.16 |
% |
10.6019/CHEMBL4513141 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Inhibition |
nan |
% |
10.1128/aac.01452-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
6.0 |
mm |
10.1128/aac.00399-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
16.0 |
mm |
10.1128/aac.00399-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
16.0 |
mm |
10.1128/aac.00893-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
17.0 |
mm |
10.1128/aac.00399-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
18.0 |
mm |
10.1128/aac.00399-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
19.0 |
mm |
10.1128/aac.00399-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
20.0 |
mm |
10.1128/aac.00399-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
21.0 |
mm |
10.1128/aac.00399-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
log10cfu |
3.0 |
None |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
log10CFU/g |
2.0 |
None |
10.1021/acs.jmedchem.5b00262 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MBC |
0.125 |
ug ml-1 |
10.1128/aac.01452-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MBC |
1.0 |
ug ml-1 |
10.1128/aac.01433-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MBC |
1.0 |
ug ml-1 |
10.1128/aac.01452-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MBC |
2.0 |
ug ml-1 |
10.1128/aac.01452-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MBC |
2.0 |
ug ml-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MBC |
4.0 |
ug ml-1 |
10.1021/acs.jmedchem.2c01469 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MBC |
32.0 |
ug ml-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.00294-06 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.01 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.023 |
ug.mL-1 |
10.1128/aac.00257-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.047 |
ug.mL-1 |
10.1128/aac.00257-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(00)00253-5 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(00)00575-8 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(01)00451-6 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(02)00948-4 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(98)00270-4 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(99)00407-2 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(99)00646-0 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(99)00692-7 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.049 |
ug.mL-1 |
10.1021/np060206z |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.05 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00816-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.063 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.014 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.00257-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.00912-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.094 |
ug.mL-1 |
10.1128/aac.00257-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.098 |
ug.mL-1 |
10.1021/np049577a |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.098 |
ug.mL-1 |
10.1021/np060206z |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.1 |
ug.mL-1 |
10.1021/np020507i |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.bmc.2021.116142 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00816-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01410-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.014 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.125 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01903 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00257-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00912-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01452-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.00257-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.00419-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.195 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.195 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.195 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(00)00253-5 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(00)00575-8 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(01)00451-6 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(02)00948-4 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(98)00270-4 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(99)00407-2 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(99)00646-0 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.2 |
ug.mL-1 |
10.1016/0960-894X(95)00380-C |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.2 |
ug.mL-1 |
10.1016/S0960-894X(97)00230-8 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.2 |
ug.mL-1 |
10.1021/jm010546b |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.2 |
ug.mL-1 |
10.1021/np020507i |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.2 |
ug.mL-1 |
10.1128/aac.00464-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2020.112252 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1016/S0960-894X(97)00282-5 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1039/C5MD00373C |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00257-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00385-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00415-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00419-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00816-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00834-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00900-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00912-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01410-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01452-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01529-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.361 |
ug.mL-1 |
10.1016/s0960-894x(99)00692-7 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00257-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00385-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00419-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00810-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00822-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.39 |
ug.mL-1 |
10.1021/np020507i |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.391 |
ug.mL-1 |
10.1021/np060206z |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.4 |
ug.mL-1 |
10.1021/jm010546b |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00746 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01742 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1021/ml200012f |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1039/C5MD00373C |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00033-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00160-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00174-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00257-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00385-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00419-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00816-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00822-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00834-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00912-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01104-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01172-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01452-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01529-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.00174-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.00822-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.8 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.8 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114278 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01469 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00867 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b01093 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00026 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1039/C5MD00373C |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00257-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00385-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00574-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00816-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00899-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00912-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01104-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01360-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01410-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01452-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.00385-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.56 |
ug.mL-1 |
10.1016/S0960-894X(97)00230-8 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.563 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.6 |
ug.mL-1 |
10.1128/aac.00464-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c00888 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm400560z |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1039/C5MD00373C |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00160-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00399-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00574-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00816-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00837-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01104-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01410-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.00837-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
3.1 |
ug.mL-1 |
10.1128/aac.00464-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1016/S0960-894X(97)00282-5 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.5b00262 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00867 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1021/np800503z |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1039/C5MD00373C |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00080-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00160-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00282-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00399-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00574-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00816-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00834-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01104-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.00822-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.00837-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
6.3 |
ug.mL-1 |
10.1128/aac.00464-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmc.2013.09.041 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116128 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112252 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114278 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00867 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1039/C5MD00373C |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00080-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00299-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00399-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00574-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00707-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00810-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00816-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00822-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01011-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01104-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01172-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01483-06 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.00282-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
12.5 |
ug.mL-1 |
10.1128/aac.00464-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.014 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00867 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b00091 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1039/C5MD00373C |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00080-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00160-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00282-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00574-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00810-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00816-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00834-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01172-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01190-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01360-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
24.0 |
ug.mL-1 |
10.1128/aac.01573-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127928 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.058 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01469 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00867 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01261 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1039/C5MD00373C |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1039/C5MD00380F |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00033-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00282-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00299-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00465-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00574-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00707-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00816-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00834-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00837-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00900-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01172-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01230-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01267-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01345-06 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01451-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01561-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01573-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
61.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.058 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.058 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.014 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00338 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm400560z |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1039/C5MD00373C |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1039/C5MD00380F |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00574-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00734-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00834-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01172-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01257 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
128.0 |
ug.mL-1 |
10.1039/C5MD00380F |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00175-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00399-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00679-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00689-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01405-06 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01360-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00621 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8000.0 |
nM |
10.1021/acs.jmedchem.1c00621 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1021/acs.jmedchem.6b00867 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm400560z |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00255 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.7b00377 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00912-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00912-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00338 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
8.0 |
ug.mL-1 |
10.1021/ml200012f |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00912-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.00912-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC50 |
64.0 |
ug.mL-1 |
10.1021/jm400560z |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
0.06 |
ug.mL-1 |
10.1039/C1MD00095K |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
0.125 |
ug.mL-1 |
10.1039/C1MD00095K |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
0.25 |
ug.mL-1 |
10.1039/C1MD00095K |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2012.07.005 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
0.5 |
ug.mL-1 |
10.1039/C1MD00095K |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
1.0 |
ug.mL-1 |
10.1039/C1MD00095K |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
2.0 |
ug.mL-1 |
10.1039/C1MD00095K |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
4.0 |
ug.mL-1 |
10.1039/C1MD00095K |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00255 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
8.0 |
ug.mL-1 |
10.1039/C1MD00095K |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
16.0 |
ug.mL-1 |
10.1021/jm400560z |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
16.0 |
ug.mL-1 |
10.1039/C1MD00095K |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.7b00377 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00338 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
32.0 |
ug.mL-1 |
10.1039/C1MD00095K |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00912-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.07.005 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
64.0 |
ug.mL-1 |
10.1021/jm400560z |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
64.0 |
ug.mL-1 |
10.1021/ml200012f |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
64.0 |
ug.mL-1 |
10.1039/C1MD00095K |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
128.0 |
ug.mL-1 |
10.1128/aac.00912-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
nan |
None |
10.1016/j.bmcl.2012.07.005 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MPC |
4.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MPC |
8.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MPC |
16.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MPC |
32.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MPC |
64.0 |
ug ml-1 |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
PD50 |
1.04 |
mg kg-1 |
10.1021/ml200012f |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
PD50 |
1.3 |
mg kg-1 |
10.1021/ml200012f |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
PD50 |
1.76 |
mg kg-1 |
10.1016/s0960-894x(98)00270-4 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Ratio |
4.0 |
None |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Ratio |
8.0 |
None |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Ratio |
16.0 |
None |
10.1128/aac.00033-10 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Ratio |
32.0 |
None |
10.1016/j.ejmech.2020.112252 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Survival |
23.0 |
% |
10.1039/C5MD00380F |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Survival |
25.0 |
% |
10.1016/j.ejmech.2019.111814 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
TIME |
1.5 |
hr |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
TIME |
3.8 |
hr |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
TIME |
4.1 |
hr |
10.1128/aac.01525-09 |
| Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) |
Beta-lactamase |
Activity |
0.0063 |
% |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) |
Beta-lactamase |
Activity |
1.6 |
% |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) |
Beta-lactamase |
Kcat |
0.006 |
/s |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) |
Beta-lactamase |
Kcat/Km |
0.0043 |
/s/microM |
10.1128/aac.01004-09 |
| Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) |
Beta-lactamase |
Km |
1400.0 |
nM |
10.1128/aac.01004-09 |
| Pseudomonas fluorescens |
Beta-lactamase |
Kcat/Km |
80.0 |
/mM/s |
10.1128/aac.00961-09 |
| Pseudomonas fluorescens |
Pseudomonas fluorescens |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Pseudomonas fluorescens |
Pseudomonas fluorescens |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00961-09 |
| Pseudomonas fluorescens |
Pseudomonas fluorescens |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Pseudomonas fluorescens |
Pseudomonas fluorescens |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Pseudomonas putida |
Pseudomonas putida |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00931-08 |
| Pseudomonas putida |
Pseudomonas putida |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00838-06 |
| Pseudomonas putida |
Pseudomonas putida |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00707-08 |
| Pseudomonas stutzeri |
Metallo-beta-lactamase |
Kcat |
4.0 |
/s |
10.1128/aac.01456-09 |
| Pseudomonas stutzeri |
Metallo-beta-lactamase |
Km |
20000.0 |
nM |
10.1128/aac.01456-09 |
| Pseudomonas stutzeri |
Metallo-beta-lactamase |
Ratio |
200.0 |
None |
10.1128/aac.01456-09 |
| Rattus norvegicus |
Aldose reductase |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Aldose reductase |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1a adrenergic receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1a adrenergic receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1b adrenergic receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1b adrenergic receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Androgen Receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Androgen Receptor |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Androgen Receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Androgen Receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Cyclooxygenase-1 |
AC50 |
33424.5 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
GABA receptor alpha-1 subunit |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Glutamate (NMDA) receptor subunit zeta 1 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Glycine receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Glycine receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Insulin receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Insulin receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Nitric-oxide synthase, brain |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Nitric-oxide synthase, brain |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
41300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
42700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
43300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
43800.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
44700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
317.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
336.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
367.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
370.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
398.83 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
443.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
43.83 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
46.5 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
52.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
52.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
61.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
75.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
76.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
76.5 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
81.17 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
85.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
86.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AUC |
6383.33 |
ng.hr.mL-1 |
10.1016/s0960-894x(00)00253-5 |
| Rattus norvegicus |
Rattus norvegicus |
AUC |
6383.33 |
ng.hr.mL-1 |
10.1016/s0960-894x(01)00451-6 |
| Rattus norvegicus |
Rattus norvegicus |
AUC |
6383.33 |
ng.hr.mL-1 |
10.1016/s0960-894x(02)00948-4 |
| Rattus norvegicus |
Rattus norvegicus |
BASO |
0.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
1.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
1.5 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
1.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
133.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
163.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
166.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
176.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
190.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
200.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
99.17 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
99.67 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
101.0 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
101.33 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
101.67 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
606.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
713.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
740.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
783.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
853.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
176.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
199.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
231.83 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
254.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
300.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
331.5 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CL |
54.16 |
mL.min-1.kg-1 |
10.1016/s0960-894x(00)00253-5 |
| Rattus norvegicus |
Rattus norvegicus |
CL |
54.16 |
mL.min-1.kg-1 |
10.1016/s0960-894x(01)00451-6 |
| Rattus norvegicus |
Rattus norvegicus |
CL |
54.2 |
mL.min-1.kg-1 |
10.1016/s0960-894x(02)00948-4 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
25330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
27000000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
27500000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
28330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
29330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
1.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.2 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
3.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
148.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
214.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
222.83 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
276.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
351.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
455.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
2.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
2.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
2.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1543.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1550.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1606.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1610.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1688.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1713.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
34.4 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
35.5 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
35.53 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
35.77 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.37 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.52 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
131000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
132700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
134000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
134500.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
135300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
136700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
71.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
127.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
174.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
187.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
241.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
406.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
8.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
9.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
9.5 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
12444.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
12982.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
13228.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
14286.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
14453.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
16020.5 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
85.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
88.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
89.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
90.5 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
92.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
23.22 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
23.37 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
23.8 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.03 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.07 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
368500.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
373700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
374700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
376000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
381000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
382000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.33 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.92 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.23 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.47 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.97 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.3 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
0.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
29.17 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
45.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
0.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
0.17 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
0.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
6.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
8.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
9.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
9.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
10.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
11.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
841.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1468.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1474.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1490.83 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1520.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1912.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
114.8 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
118.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
119.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
122.5 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
122.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
123.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1149330.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1178000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1189000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1239500.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1255500.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1310330.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.26 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.33 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.59 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.82 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.87 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
59000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
59300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
59800.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
60300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
63000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5530000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5620000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5690000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5720000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5760000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5780000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
0.0 |
/100WBC |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
0.17 |
/100WBC |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.28 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.3 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
143.0 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
143.8 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
144.6 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
147.07 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
0.0665 |
hr |
10.1016/s0960-894x(00)00253-5 |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
0.0665 |
hr |
10.1016/s0960-894x(01)00451-6 |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
0.0665 |
hr |
10.1016/s0960-894x(02)00948-4 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
16.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
16.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
18.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
19.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
20.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
13500.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
14730.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
15100.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
16170.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
16700.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
17670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Serotonin 1a (5-HT1a) receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1a (5-HT1a) receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1b (5-HT1b) receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1b (5-HT1b) receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Voltage-gated L-type calcium channel alpha-1C subunit |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Salmonella |
Salmonella |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Salmonella |
Salmonella |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Salmonella |
Salmonella |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Salmonella |
Salmonella |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Salmonella |
Salmonella |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Salmonella enterica |
Salmonella enterica |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Salmonella enterica |
Salmonella enterica |
MIC |
0.125 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01674 |
| Salmonella enterica |
Salmonella enterica |
MIC |
nan |
None |
10.1016/j.ejmech.2017.10.044 |
| Salmonella enterica |
Salmonella enterica |
MIC |
nan |
None |
10.1016/j.ejmech.2017.12.009 |
| Salmonella enterica subsp. enterica serovar Enteritidis |
Salmonella enteritidis |
MIC |
0.016 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Salmonella enterica subsp. enterica serovar Enteritidis |
Salmonella enteritidis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Salmonella enterica subsp. enterica serovar Paratyphi A |
Salmonella paratyphi |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Salmonella enterica subsp. enterica serovar Paratyphi A |
Salmonella paratyphi |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Salmonella enterica subsp. enterica serovar Typhi |
Salmonella typhi |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Salmonella enterica subsp. enterica serovar Typhi |
Salmonella typhi |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.016 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(98)00270-4 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(99)00407-2 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(00)00253-5 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(00)00575-8 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(01)00451-6 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(02)00948-4 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(99)00646-0 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.049 |
ug.mL-1 |
10.1016/s0960-894x(99)00692-7 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Schaalia meyeri |
Schaalia meyeri |
Activity |
8.0 |
% |
10.1128/aac.00481-10 |
| Schaalia meyeri |
Schaalia meyeri |
Activity |
92.0 |
% |
10.1128/aac.00481-10 |
| Schaalia meyeri |
Schaalia meyeri |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Schaalia meyeri |
Schaalia meyeri |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Schaalia meyeri |
Schaalia meyeri |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| Serratia fonticola |
Carbapenem-hydrolizing beta-lactamase SFC-1 |
Kcat |
6.5 |
/s |
10.1128/aac.00491-07 |
| Serratia fonticola |
Carbapenem-hydrolizing beta-lactamase SFC-1 |
Kcat/Km |
250.0 |
/mM/s |
10.1128/aac.00491-07 |
| Serratia fonticola |
Carbapenem-hydrolizing beta-lactamase SFC-1 |
Km |
26000.0 |
nM |
10.1128/aac.00491-07 |
| Serratia marcescens |
Carbapenem-hydrolyzing beta-lactamase SME-3 |
Activity |
0.27 |
% |
10.1128/aac.01004-09 |
| Serratia marcescens |
Carbapenem-hydrolyzing beta-lactamase SME-3 |
Activity |
18.0 |
% |
10.1128/aac.01004-09 |
| Serratia marcescens |
Carbapenem-hydrolyzing beta-lactamase SME-3 |
Kcat |
3.2 |
/s |
10.1128/aac.01004-09 |
| Serratia marcescens |
Carbapenem-hydrolyzing beta-lactamase SME-3 |
Kcat/Km |
0.55 |
/s/microM |
10.1128/aac.01004-09 |
| Serratia marcescens |
Carbapenem-hydrolyzing beta-lactamase SME-3 |
Km |
5800.0 |
nM |
10.1128/aac.01004-09 |
| Serratia marcescens |
Serratia marcescens |
Activity |
0.0 |
% |
10.1128/aac.00381-08 |
| Serratia marcescens |
Serratia marcescens |
Activity |
0.0 |
% |
10.1128/aac.00400-09 |
| Serratia marcescens |
Serratia marcescens |
Activity |
0.8 |
% |
10.1128/aac.00381-08 |
| Serratia marcescens |
Serratia marcescens |
Activity |
99.2 |
% |
10.1128/aac.00381-08 |
| Serratia marcescens |
Serratia marcescens |
Activity |
100.0 |
% |
10.1128/aac.00381-08 |
| Serratia marcescens |
Serratia marcescens |
Activity |
100.0 |
% |
10.1128/aac.00400-09 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00768-10 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00768-10 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.06 |
ug.mL-1 |
10.1021/jm010546b |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.06 |
ug.mL-1 |
10.1021/np800503z |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Serratia marcescens |
Serratia marcescens |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00768-10 |
| Serratia marcescens |
Serratia marcescens |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00768-10 |
| Serratia marcescens |
Serratia marcescens |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01539-07 |
| Serratia marcescens |
Serratia marcescens |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00309-07 |
| Serratia marcescens |
Serratia marcescens |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00768-10 |
| Serratia marcescens |
Serratia marcescens |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00768-10 |
| Serratia marcescens |
Serratia marcescens |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00768-10 |
| Serratia marcescens |
Serratia marcescens |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Serratia marcescens |
Serratia marcescens |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01004-09 |
| Serratia marcescens |
Serratia marcescens |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Serratia marcescens |
Serratia marcescens |
MIC50 |
0.06 |
ug.mL-1 |
10.1021/ml200012f |
| Serratia marcescens |
Serratia marcescens |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Serratia marcescens |
Serratia marcescens |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Serratia marcescens |
Serratia marcescens |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Serratia marcescens |
Serratia marcescens |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Serratia marcescens |
Serratia marcescens |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Serratia marcescens |
Serratia marcescens |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Serratia marcescens |
Serratia marcescens |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Serratia marcescens |
Serratia marcescens |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Serratia marcescens |
Serratia marcescens |
MIC90 |
64.0 |
ug.mL-1 |
10.1021/ml200012f |
| Severe acute respiratory syndrome coronavirus 2 |
Replicase polyprotein 1ab |
Inhibition |
-4.064 |
% |
10.6019/CHEMBL4495564 |
| Severe acute respiratory syndrome coronavirus 2 |
Replicase polyprotein 1ab |
Inhibition |
10.85 |
% |
10.6019/CHEMBL4495564 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
19952.62 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
20000.0 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
-0.09 |
% |
10.6019/CHEMBL4495565 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
0.12 |
% |
10.6019/CHEMBL4495565 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
10.13 |
% |
10.21203/rs.3.rs-23951/v1 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition index |
0.4369 |
None |
10.1101/2020.04.03.023846 |
| Shigella flexneri |
Shigella flexneri |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Shigella sonnei |
Shigella sonnei |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Shigella sonnei |
Shigella sonnei |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00227-08 |
| Staphylococcus |
Staphylococcus |
Activity |
99.4 |
% |
10.1128/aac.00381-08 |
| Staphylococcus |
Staphylococcus |
MIC |
0.098 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Staphylococcus |
Staphylococcus |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Staphylococcus |
Staphylococcus |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Staphylococcus |
Staphylococcus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Staphylococcus |
Staphylococcus |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Staphylococcus aureus |
MecA |
IC50 |
53.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Staphylococcus aureus |
MecA |
IC50 |
130.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.01351-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.01538-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
98.0 |
% |
10.1128/aac.01351-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00381-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.01128-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.01538-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.ejmech.2022.114278 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/acsmedchemlett.1c00648 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01192-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.14 |
ug.mL-1 |
10.1128/aac.01192-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.16 |
ug.mL-1 |
10.1128/aac.01192-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.2 |
ug.mL-1 |
10.1128/aac.01192-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.29 |
ug.mL-1 |
10.1128/aac.01192-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.33 |
ug.mL-1 |
10.1128/aac.01192-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
nan |
None |
10.1128/aac.01192-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
FIC |
2.0 |
None |
10.1021/acs.jnatprod.2c00621 |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
10.0 |
nM |
10.1021/acs.jnatprod.9b00187 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
-14.17 |
% |
10.6019/CHEMBL4513141 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.12 |
ug ml-1 |
10.1128/aac.01433-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
8.0 |
ug ml-1 |
10.1021/acs.jmedchem.2c01469 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.00294-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.013 |
ug.mL-1 |
10.1016/s0960-894x(99)00692-7 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.049 |
ug.mL-1 |
10.1021/np049577a |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.049 |
ug.mL-1 |
10.1021/np060206z |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2021.113402 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1016/S0960-894X(97)00282-5 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1039/D1MD00230A |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.ejmech.2020.112996 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.098 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.098 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.098 |
ug.mL-1 |
10.1016/s0960-894x(00)00253-5 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.098 |
ug.mL-1 |
10.1016/s0960-894x(00)00575-8 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.098 |
ug.mL-1 |
10.1016/s0960-894x(01)00451-6 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.098 |
ug.mL-1 |
10.1016/s0960-894x(02)00948-4 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.098 |
ug.mL-1 |
10.1016/s0960-894x(98)00270-4 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.098 |
ug.mL-1 |
10.1016/s0960-894x(99)00407-2 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.098 |
ug.mL-1 |
10.1016/s0960-894x(99)00646-0 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.098 |
ug.mL-1 |
10.1021/np049577a |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.098 |
ug.mL-1 |
10.1021/np060206z |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.1 |
ug.mL-1 |
10.1016/0960-894X(95)00380-C |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.1 |
ug.mL-1 |
10.1016/S0960-894X(97)00230-8 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm010546b |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.ejmech.2021.113402 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1039/D1MD00230A |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00746 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.13 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.052 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.19 |
ug.mL-1 |
10.1016/S0960-894X(01)80919-7 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.195 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.195 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(00)00253-5 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(00)00575-8 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(01)00451-6 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(02)00948-4 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(99)00646-0 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.195 |
ug.mL-1 |
10.1016/s0960-894x(99)00692-7 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.195 |
ug.mL-1 |
10.1021/np049577a |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1021/np800503z |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2015.04.046 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.052 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01351-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.bmc.2016.02.013 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.04.046 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.03.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.052 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112996 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jnatprod.1c00578 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00621 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.56 |
ug.mL-1 |
10.1016/S0960-894X(01)80919-7 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.052 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113402 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114278 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01469 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00746 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00621 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1039/D1MD00230A |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.1 |
ug.mL-1 |
10.1021/np030162j |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.04.046 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.070 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.052 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112996 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113402 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/np800503z |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1039/D1MD00230A |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.052 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112996 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113402 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1016/S0960-894X(97)00282-5 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1039/D1MD00230A |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.04.046 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.070 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.052 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112996 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
25.0 |
ug.mL-1 |
10.1016/0960-894X(95)00380-C |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
25.0 |
ug.mL-1 |
10.1016/S0960-894X(01)80919-7 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
25.0 |
ug.mL-1 |
10.1016/S0960-894X(97)00230-8 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
25.0 |
ug.mL-1 |
10.1021/np030162j |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.04.046 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.052 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112996 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01469 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
50.0 |
ug.mL-1 |
10.1021/np030162j |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116128 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.070 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.052 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112996 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
100.0 |
ug.mL-1 |
10.1016/S0960-894X(01)80919-7 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.ejmech.2017.10.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.ejmech.2017.12.009 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1021/acs.jmedchem.2c01674 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1021/np800503z |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01351-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01351-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00413-08 |
| Staphylococcus chromogenes |
Staphylococcus chromogenes |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
0.0 |
% |
10.1128/aac.01538-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
1.8 |
% |
10.1128/aac.01538-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
9.3 |
% |
10.1128/aac.01538-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
29.2 |
% |
10.1128/aac.01538-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
67.0 |
% |
10.1128/aac.01128-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
100.0 |
% |
10.1128/aac.01538-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.8 |
ug.mL-1 |
10.1021/np030162j |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.6 |
ug.mL-1 |
10.1021/np030162j |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
73.0 |
% |
10.1128/aac.01128-07 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Stenotrophomonas maltophilia |
Beta-lactamase L1 |
Kcat/Km |
4.5 |
10'6/M/s |
10.1128/aac.01062-07 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
Activity |
nan |
None |
10.1128/aac.01525-09 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MBC |
16.0 |
ug ml-1 |
10.1128/aac.01525-09 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.01283-09 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00682-07 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01283-09 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.01283-09 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01485-07 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00682-07 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01283-09 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01513-08 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.014 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01485-07 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm010546b |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.bmc.2013.09.041 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
128.0 |
ug.mL-1 |
10.1016/S0960-894X(97)00282-5 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC50 |
64.0 |
ug.mL-1 |
10.1021/ml200012f |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC90 |
64.0 |
ug.mL-1 |
10.1021/ml200012f |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Streptococcus |
Streptococcus |
EC50 |
1154.0 |
nM |
None |
| Streptococcus agalactiae |
Streptococcus agalactiae |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00185-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.031 |
ug.mL-1 |
10.1128/aac.01716-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00185-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00185-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00185-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
0.063 |
ug.mL-1 |
10.1128/aac.01716-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
0.063 |
ug.mL-1 |
10.1128/aac.01716-08 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC |
0.05 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Streptococcus dysgalactiae |
Streptococcus dysgalactiae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Streptococcus dysgalactiae subsp. equisimilis |
Streptococcus dysgalactiae subsp. equisimilis |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Streptococcus dysgalactiae subsp. equisimilis |
Streptococcus dysgalactiae subsp. equisimilis |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Streptococcus dysgalactiae subsp. equisimilis |
Streptococcus dysgalactiae subsp. equisimilis |
MIC90 |
0.015 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Streptococcus intermedius |
Streptococcus intermedius |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
0.0 |
% |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
0.0 |
% |
10.1128/aac.01538-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
0.4 |
% |
10.1128/aac.01384-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
0.4 |
% |
10.1128/aac.01538-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
0.5 |
% |
10.1128/aac.01538-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
2.3 |
% |
10.1128/aac.00381-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
4.5 |
% |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
9.5 |
% |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
33.3 |
% |
10.1128/aac.01268-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
34.3 |
% |
10.1128/aac.01268-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
59.5 |
% |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
75.9 |
% |
10.1128/aac.01387-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
83.2 |
% |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
83.9 |
% |
10.1128/aac.00381-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
86.8 |
% |
10.1128/aac.01384-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
93.2 |
% |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
100.0 |
% |
10.1128/aac.00381-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
100.0 |
% |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.00294-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.015 |
ug.mL-1 |
10.1021/np800503z |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.016 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00746 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01387-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00185-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01082-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01082-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01324-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2020.115776 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01082-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01268-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01082-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/np800503z |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.01384-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.016 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2020.115776 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01268-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01387-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00381-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01324-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
0.015 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
0.016 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01384-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115776 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00971-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01268-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01387-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01531-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01324-08 |
| Streptococcus pneumoniae R6 |
Penicillin-binding protein 2X |
Activity |
nan |
None |
10.1021/jm900625q |
| Streptococcus pneumoniae serotype 4 (strain ATCC BAA-334 / TIGR4) |
Penicillin-binding protein 2x |
Activity |
nan |
None |
10.1021/jm900625q |
| Streptococcus pyogenes |
Streptococcus pyogenes |
Activity |
0.0 |
% |
10.1128/aac.01128-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.002 |
ug.mL-1 |
10.1016/s0960-894x(98)00270-4 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.002 |
ug.mL-1 |
10.1016/s0960-894x(99)00407-2 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.004 |
ug.mL-1 |
10.1021/np020507i |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.004 |
ug.mL-1 |
10.1021/np060206z |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.007 |
ug.mL-1 |
10.1021/np049577a |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.008 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00746 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.01 |
ug.mL-1 |
10.1021/np020507i |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.013 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.013 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.013 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.013 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.013 |
ug.mL-1 |
10.1016/s0960-894x(00)00253-5 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.013 |
ug.mL-1 |
10.1016/s0960-894x(00)00575-8 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.013 |
ug.mL-1 |
10.1016/s0960-894x(01)00451-6 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.013 |
ug.mL-1 |
10.1016/s0960-894x(02)00948-4 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.013 |
ug.mL-1 |
10.1016/s0960-894x(99)00646-0 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.013 |
ug.mL-1 |
10.1016/s0960-894x(99)00692-7 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
0.015 |
ug.mL-1 |
10.1128/aac.01128-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
PD50 |
7.16 |
mg kg-1 |
10.1016/s0960-894x(98)00270-4 |
| Streptococcus pyogenes serotype M1 |
Streptokinase A |
EC50 |
127.0 |
nM |
None |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
EC50 |
153.0 |
nM |
None |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00596-08 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00596-08 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00596-08 |
| Sus scrofa |
Renal dipeptidase |
Activity |
32.0 |
None |
10.1016/s0960-894x(99)00692-7 |
| Sus scrofa |
Renal dipeptidase |
DHP-I stability |
1.0 |
None |
10.1016/S0960-894X(97)00230-8 |
| Sus scrofa |
Renal dipeptidase |
Relative t1/2 |
1.0 |
None |
10.1016/s0960-894x(99)00646-0 |
| Sus scrofa |
Renal dipeptidase |
Stability |
100.0 |
% |
10.1016/s0960-894x(99)00407-2 |
| Sus scrofa |
Renal dipeptidase |
Stability |
3200.0 |
% |
10.1016/s0960-894x(98)00270-4 |
| Thomasclavelia ramosa |
Thomasclavelia ramosa |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Thomasclavelia ramosa |
Thomasclavelia ramosa |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Thomasclavelia ramosa |
Thomasclavelia ramosa |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00910-07 |
| Trueperella pyogenes |
Trueperella pyogenes |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| Trueperella pyogenes |
Trueperella pyogenes |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| Veillonella parvula |
Veillonella parvula |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| Veillonella parvula |
Veillonella parvula |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00355-08 |
| None |
ADMET |
AUC |
2.0 |
hr |
10.1016/s0960-894x(98)00270-4 |
| None |
ADMET |
AUC |
3.29 |
ug ml-1 |
10.1016/s0960-894x(98)00270-4 |
| None |
ADMET |
AUC |
6383.33 |
ng.hr.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| None |
ADMET |
AUC |
6383.33 |
ng.hr.mL-1 |
10.1016/j.ejmech.2019.111744 |
| None |
ADMET |
AUC |
11583.33 |
ng.hr.mL-1 |
10.1016/j.bmcl.2004.09.092 |
| None |
ADMET |
CL |
3.9 |
mL.min-1.kg-1 |
10.1124/dmd.108.020479 |
| None |
ADMET |
CL |
4.0 |
mL.min-1.kg-1 |
10.1002/jps.20373 |
| None |
ADMET |
CL |
7.0 |
mL.min-1.kg-1 |
10.1002/jps.20373 |
| None |
ADMET |
CL |
7.0 |
mL.min-1.kg-1 |
10.1016/j.bmcl.2004.09.092 |
| None |
ADMET |
CL |
47.0 |
mL.min-1.kg-1 |
10.1002/jps.20373 |
| None |
ADMET |
CL |
51.16 |
mL.min-1.kg-1 |
10.1016/j.ejmech.2019.111744 |
| None |
ADMET |
CL |
52.0 |
mL.min-1.kg-1 |
10.1016/j.bmcl.2004.09.092 |
| None |
ADMET |
Cmax |
19819.02 |
nM |
10.1016/s0960-894x(98)00270-4 |
| None |
ADMET |
Cmax |
146295.67 |
nM |
10.1128/aac.00160-07 |
| None |
ADMET |
log10(%HIA +10) |
1.0 |
None |
10.1016/j.ejmech.2010.11.005 |
| None |
ADMET |
mortality |
100.0 |
% |
10.1016/j.ejmech.2019.04.034 |
| None |
ADMET |
MRT |
1.3 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
Ratio |
34.24 |
None |
10.1128/aac.00294-06 |
| None |
ADMET |
Ratio |
1427.66 |
None |
10.1128/aac.00294-06 |
| None |
ADMET |
Ratio |
6683.38 |
None |
10.1128/aac.00294-06 |
| None |
ADMET |
Relative t1/2 |
1.0 |
None |
10.1016/s0960-894x(02)00948-4 |
| None |
ADMET |
T1/2 |
0.01667 |
hr |
10.1016/j.bmcl.2004.09.092 |
| None |
ADMET |
T1/2 |
0.06667 |
hr |
10.1016/j.bmcl.2004.09.092 |
| None |
ADMET |
T1/2 |
0.24 |
hr |
10.1016/s0960-894x(98)00270-4 |
| None |
ADMET |
T1/2 |
0.45 |
hr |
10.1128/aac.00160-07 |
| None |
ADMET |
T1/2 |
0.46 |
hr |
10.1021/acs.jmedchem.2c00227 |
| None |
ADMET |
T1/2 |
0.55 |
hr |
10.1016/j.bmcl.2004.09.092 |
| None |
ADMET |
T1/2 |
1.0 |
hr |
10.1016/j.ejmech.2020.112829 |
| None |
ADMET |
T1/2 |
1.0 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
T1/2 |
3.99 |
hr |
10.1016/j.ejmech.2019.111744 |
| None |
ADMET |
Tmax |
0.21 |
hr |
10.1016/s0960-894x(98)00270-4 |
| None |
ADMET |
Vdss |
0.25 |
L.kg-1 |
10.1002/jps.20373 |
| None |
ADMET |
Vdss |
0.3 |
L.kg-1 |
10.1002/jps.20373 |
| None |
ADMET |
Vdss |
0.3 |
L.kg-1 |
10.1124/dmd.108.020479 |
| None |
ADMET |
Vdss |
0.3 |
mL/min/kg |
10.1002/jps.20373 |
| None |
Erythrocyte |
HC50 |
500.0 |
ug ml-1 |
10.1016/j.ejmech.2022.114278 |
| None |
Erythrocyte |
HC50 |
nan |
None |
10.1016/j.ejmech.2017.10.044 |
| None |
Erythrocyte |
HC50 |
nan |
None |
10.1016/j.ejmech.2017.12.009 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Index Value |
0.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Active |
2.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Marginal |
1.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Index Value |
0.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1021/tx900326k |
| None |
Hepatotoxicity |
HepSE_bilirubinemia |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholecystitis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholelithiasis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cirrhosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_Combined Scores |
3.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_elevated liver function tests |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic failure |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic necrosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatitis |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatomegaly |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_jaundice |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver disease |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver fatty |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver function tests abnormal |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
LDH Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LDH Increase - Index Value |
33.8 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LDH Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Index Value |
50.8 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Index Value |
50.8 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
NON-PROTEIN TARGET |
Activity |
0.0 |
% |
10.1128/aac.00481-10 |
| None |
NON-PROTEIN TARGET |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| None |
NON-PROTEIN TARGET |
Activity |
0.0 |
% |
10.1128/aac.00898-09 |
| None |
NON-PROTEIN TARGET |
Activity |
0.5 |
% |
10.1128/aac.01435-06 |
| None |
NON-PROTEIN TARGET |
Activity |
8.0 |
% |
10.1128/aac.00481-10 |
| None |
NON-PROTEIN TARGET |
Activity |
9.0 |
ug ml-1 |
10.1128/aac.01525-09 |
| None |
NON-PROTEIN TARGET |
Activity |
16.0 |
ug ml-1 |
10.1128/aac.00898-09 |
| None |
NON-PROTEIN TARGET |
Activity |
53.7 |
% |
10.1128/aac.01173-09 |
| None |
NON-PROTEIN TARGET |
Activity |
92.0 |
% |
10.1128/aac.00481-10 |
| None |
NON-PROTEIN TARGET |
Activity |
nan |
None |
10.1128/aac.00128-10 |
| None |
NON-PROTEIN TARGET |
Activity |
nan |
None |
10.1128/aac.01525-09 |
| None |
NON-PROTEIN TARGET |
FICI |
0.5 |
None |
10.1128/aac.01173-09 |
| None |
NON-PROTEIN TARGET |
fT>MIC |
1.9 |
hr |
10.1128/aac.00642-09 |
| None |
NON-PROTEIN TARGET |
fT>MIC |
2.0 |
hr |
10.1128/aac.00642-09 |
| None |
NON-PROTEIN TARGET |
fT>MIC |
8.0 |
% |
10.1128/aac.00642-09 |
| None |
NON-PROTEIN TARGET |
fT>MIC |
8.5 |
% |
10.1128/aac.00642-09 |
| None |
NON-PROTEIN TARGET |
fT>MIC |
40.0 |
% |
10.1128/aac.01582-09 |
| None |
NON-PROTEIN TARGET |
Fu |
0.87 |
None |
10.1124/dmd.108.020479 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (acute) |
5.3 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (animal toxicity known) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (benign tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (granulomatous hepatitis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (mechanism) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
48.1 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
92.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (time to onset) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
MIC |
0.00012 |
ug.mL-1 |
10.1128/aac.01102-06 |
| None |
NON-PROTEIN TARGET |
MIC |
0.00025 |
ug.mL-1 |
10.1128/aac.01102-06 |
| None |
NON-PROTEIN TARGET |
MIC |
0.002 |
ug.mL-1 |
10.1128/aac.01102-06 |
| None |
NON-PROTEIN TARGET |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00481-10 |
| None |
NON-PROTEIN TARGET |
MIC |
0.0094 |
ug.mL-1 |
10.1128/aac.00570-10 |
| None |
NON-PROTEIN TARGET |
MIC |
0.013 |
ug.mL-1 |
10.1016/s0960-894x(98)00270-4 |
| None |
NON-PROTEIN TARGET |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| None |
NON-PROTEIN TARGET |
MIC |
0.023 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(98)00270-4 |
| None |
NON-PROTEIN TARGET |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| None |
NON-PROTEIN TARGET |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00570-10 |
| None |
NON-PROTEIN TARGET |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00684-07 |
| None |
NON-PROTEIN TARGET |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.006 |
| None |
NON-PROTEIN TARGET |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2007.02.001 |
| None |
NON-PROTEIN TARGET |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00696-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00978-07 |
| None |
NON-PROTEIN TARGET |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01525-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01585-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.bmc.2013.09.041 |
| None |
NON-PROTEIN TARGET |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00570-10 |
| None |
NON-PROTEIN TARGET |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00696-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00570-10 |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01525-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00570-10 |
| None |
NON-PROTEIN TARGET |
MIC |
0.4 |
ug.mL-1 |
10.1128/aac.01435-06 |
| None |
NON-PROTEIN TARGET |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00128-10 |
| None |
NON-PROTEIN TARGET |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00978-07 |
| None |
NON-PROTEIN TARGET |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00570-10 |
| None |
NON-PROTEIN TARGET |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00899-09 |
| None |
NON-PROTEIN TARGET |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00570-10 |
| None |
NON-PROTEIN TARGET |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00899-09 |
| None |
NON-PROTEIN TARGET |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00128-10 |
| None |
NON-PROTEIN TARGET |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00899-09 |
| None |
NON-PROTEIN TARGET |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00128-10 |
| None |
NON-PROTEIN TARGET |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00734-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00336-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00898-09 |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00481-10 |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.01525-09 |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.19 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00696-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| None |
NON-PROTEIN TARGET |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00898-09 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.03 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00898-09 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01525-09 |
| None |
NON-PROTEIN TARGET |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01435-06 |
| None |
NON-PROTEIN TARGET |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00481-10 |
| None |
NON-PROTEIN TARGET |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00595-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00630-09 |
| None |
NON-PROTEIN TARGET |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01525-09 |
| None |
NON-PROTEIN TARGET |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00898-09 |
| None |
NON-PROTEIN TARGET |
T>MIC |
41.67 |
% |
10.1128/aac.00160-07 |
| None |
NON-PROTEIN TARGET |
T>MIC |
66.67 |
% |
10.1128/aac.00160-07 |
| None |
No relevant target |
Activity |
40.3 |
% |
10.1128/aac.00123-08 |
| None |
No relevant target |
Activity |
49.3 |
% |
10.1128/aac.00123-08 |
| None |
No relevant target |
Drug degradation |
30.0 |
% |
10.1021/acs.jmedchem.0c00255 |
| None |
No relevant target |
Drug degradation |
50.0 |
% |
10.1021/ml200012f |
| None |
No relevant target |
Drug degradation |
60.0 |
% |
10.1016/j.ejmech.2020.112829 |
| None |
No relevant target |
Drug degradation |
80.0 |
% |
10.1016/j.bmc.2013.05.024 |
| None |
No relevant target |
LogD |
2.5 |
None |
10.1016/j.bmc.2013.05.024 |
| None |
No relevant target |
Stability |
5.0 |
% |
10.1016/j.bmc.2013.05.024 |
| None |
No relevant target |
T1/2 |
78.0 |
hr |
10.1016/j.bmcl.2018.01.006 |
| None |
No relevant target |
T1/2 |
95.0 |
hr |
10.1021/acsmedchemlett.5b00026 |
| None |
Unchecked |
Ac50 |
0.3162 |
uM |
None |
| None |
Unchecked |
Ac50 |
0.7079 |
uM |
None |
| None |
Unchecked |
Ac50 |
0.8913 |
uM |
None |
| None |
Unchecked |
AC50 |
316.2 |
nM |
None |
| None |
Unchecked |
AC50 |
320.0 |
nM |
None |
| None |
Unchecked |
AC50 |
707.9 |
nM |
None |
| None |
Unchecked |
AC50 |
891.3 |
nM |
None |
| None |
Unchecked |
Activity |
0.0011 |
% |
10.1128/aac.01004-09 |
| None |
Unchecked |
Activity |
0.002 |
% |
10.1128/aac.01004-09 |
| None |
Unchecked |
Activity |
0.0024 |
% |
10.1128/aac.01004-09 |
| None |
Unchecked |
Activity |
0.0079 |
% |
10.1128/aac.01004-09 |
| None |
Unchecked |
Activity |
1.0 |
mU |
10.1128/aac.00978-07 |
| None |
Unchecked |
Activity |
1.5 |
mU |
10.1128/aac.00978-07 |
| None |
Unchecked |
Activity |
1.7 |
mU |
10.1128/aac.00978-07 |
| None |
Unchecked |
Activity |
1.8 |
% |
10.1128/aac.00083-07 |
| None |
Unchecked |
Activity |
3.4 |
% |
10.1128/aac.00175-08 |
| None |
Unchecked |
Activity |
9.4 |
% |
10.1128/aac.00175-08 |
| None |
Unchecked |
Activity |
83.0 |
% |
10.1128/aac.00175-08 |
| None |
Unchecked |
Activity |
110.0 |
% |
10.1128/aac.00175-08 |
| None |
Unchecked |
Activity |
nan |
None |
10.1021/acs.jmedchem.1c02140 |
| None |
Unchecked |
Activity |
nan |
None |
10.1128/aac.00978-07 |
| None |
Unchecked |
HC50 |
nan |
None |
10.1021/acs.jmedchem.2c01469 |
| None |
Unchecked |
HC50 |
nan |
None |
10.1021/acs.jmedchem.2c01674 |
| None |
Unchecked |
Hepatotoxicity (acute) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (association with vascular disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (choleostasis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (chronic liver disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cirrhosis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (comment) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cytolytic) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (malignant tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (severe hepatitis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (steatosis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (successful reintroduction) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
IC50 |
0.0033 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
0.008 |
ug.mL-1 |
10.1128/aac.01529-07 |
| None |
Unchecked |
IC50 |
0.013 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
0.016 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
0.018 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
0.02 |
ug.mL-1 |
10.1128/aac.01529-07 |
| None |
Unchecked |
IC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01529-07 |
| None |
Unchecked |
IC50 |
0.044 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
0.047 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
0.05 |
ug.mL-1 |
10.1128/aac.01529-07 |
| None |
Unchecked |
IC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01529-07 |
| None |
Unchecked |
IC50 |
0.071 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
0.08 |
ug.mL-1 |
10.1128/aac.01529-07 |
| None |
Unchecked |
IC50 |
0.11 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
0.12 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
0.26 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
0.39 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01529-07 |
| None |
Unchecked |
IC50 |
0.6 |
ug.mL-1 |
10.1128/aac.01529-07 |
| None |
Unchecked |
IC50 |
0.77 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
0.82 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
1.2 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
1.3 |
ug.mL-1 |
10.1128/aac.01529-07 |
| None |
Unchecked |
IC50 |
1.7 |
ug.mL-1 |
10.1128/aac.01529-07 |
| None |
Unchecked |
IC50 |
4.0 |
ug.mL-1 |
10.1128/aac.01529-07 |
| None |
Unchecked |
IC50 |
4.5 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
15.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
16.0 |
ug.mL-1 |
10.1128/aac.01529-07 |
| None |
Unchecked |
IC50 |
130.0 |
ug.mL-1 |
10.1128/aac.01433-08 |
| None |
Unchecked |
IC50 |
nan |
None |
None |
| None |
Unchecked |
Inhibition |
90.0 |
% |
10.1016/j.bmc.2021.116128 |
| None |
Unchecked |
K |
1.1 |
10'3/uM/s |
10.1021/acs.jmedchem.6b00096 |
| None |
Unchecked |
K |
4.9 |
10'4/M/s |
10.1021/acsmedchemlett.5b00026 |
| None |
Unchecked |
K |
60.0 |
10'3/s |
10.1021/acs.jmedchem.6b00096 |
| None |
Unchecked |
Kcat |
0.00039 |
/s |
10.1128/aac.01004-09 |
| None |
Unchecked |
Kcat |
0.0096 |
/s |
10.1128/aac.01004-09 |
| None |
Unchecked |
Kcat |
0.01 |
/s |
10.1128/aac.01600-06 |
| None |
Unchecked |
Kcat |
0.05 |
/s |
10.1128/aac.00858-10 |
| None |
Unchecked |
Kcat |
0.3 |
/s |
10.1128/aac.00856-09 |
| None |
Unchecked |
Kcat |
0.4 |
/s |
10.1128/aac.01337-07 |
| None |
Unchecked |
Kcat |
0.92 |
10'3/s |
10.1021/acs.jmedchem.6b00096 |
| None |
Unchecked |
Kcat |
1.0 |
/s |
10.1128/aac.00961-09 |
| None |
Unchecked |
Kcat |
1.0 |
/s |
10.1128/aac.01009-09 |
| None |
Unchecked |
Kcat |
1.0 |
/s |
10.1128/aac.01062-07 |
| None |
Unchecked |
Kcat |
1.0 |
/s |
10.1128/aac.01462-06 |
| None |
Unchecked |
Kcat |
1.3 |
/s |
10.1128/aac.00017-09 |
| None |
Unchecked |
Kcat |
4.13 |
/s |
10.1128/aac.00083-07 |
| None |
Unchecked |
Kcat |
5.0 |
/s |
10.1128/aac.00858-10 |
| None |
Unchecked |
Kcat |
5.0 |
/s |
10.1128/aac.01336-09 |
| None |
Unchecked |
Kcat |
6.0 |
/s |
10.1128/aac.01336-09 |
| None |
Unchecked |
Kcat |
6.5 |
/s |
10.1128/aac.00175-08 |
| None |
Unchecked |
Kcat |
8.4 |
/s |
10.1128/aac.00175-08 |
| None |
Unchecked |
Kcat |
13.0 |
/s |
10.1128/aac.00166-08 |
| None |
Unchecked |
Kcat |
50.0 |
/s |
10.1128/aac.00774-09 |
| None |
Unchecked |
Kcat/Km |
4.4e-05 |
/s/microM |
10.1128/aac.01004-09 |
| None |
Unchecked |
Kcat/Km |
0.00011 |
/s/microM |
10.1128/aac.01004-09 |
| None |
Unchecked |
Kcat/Km |
0.003 |
/s/microM |
10.1128/aac.00856-09 |
| None |
Unchecked |
Kcat/Km |
0.015 |
/uM/s |
10.1128/aac.00083-07 |
| None |
Unchecked |
Kcat/Km |
0.07 |
/s/microM |
10.1128/aac.00175-08 |
| None |
Unchecked |
Kcat/Km |
0.12 |
/s/microM |
10.1128/aac.00774-09 |
| None |
Unchecked |
Kcat/Km |
0.14 |
/s/microM |
10.1128/aac.00017-09 |
| None |
Unchecked |
Kcat/Km |
0.26 |
/uM/s |
10.1128/aac.00166-08 |
| None |
Unchecked |
Kcat/Km |
0.5 |
uM/hr |
10.1128/aac.01336-09 |
| None |
Unchecked |
Kcat/Km |
1.0 |
/s/M |
10.1128/aac.01025-07 |
| None |
Unchecked |
Kcat/Km |
1.9 |
/s/microM |
10.1128/aac.00175-08 |
| None |
Unchecked |
Kcat/Km |
3.0 |
uM/hr |
10.1128/aac.01336-09 |
| None |
Unchecked |
Kcat/Km |
3.3 |
10'4/M/s |
10.1128/aac.01337-07 |
| None |
Unchecked |
Kcat/Km |
3.3 |
None |
10.1128/aac.01462-06 |
| None |
Unchecked |
Kcat/Km |
4.5 |
10'6/M/s |
10.1128/aac.00409-10 |
| None |
Unchecked |
Kcat/Km |
5.0 |
10'5/M/s |
10.1128/aac.00409-10 |
| None |
Unchecked |
Kcat/Km |
5.0 |
10'5/M/s |
10.1128/aac.00858-10 |
| None |
Unchecked |
Kcat/Km |
5.3 |
10'6/M/s |
10.1128/aac.00409-10 |
| None |
Unchecked |
Kcat/Km |
6.0 |
10'3/M/s |
10.1128/aac.00858-10 |
| None |
Unchecked |
Kcat/Km |
8.3 |
10'5/M/s |
10.1128/aac.00409-10 |
| None |
Unchecked |
Kcat/Km |
8.3 |
10'5/M/s |
10.1128/aac.01062-07 |
| None |
Unchecked |
Kcat/Km |
9.6 |
10'2/M/s |
10.1128/aac.01062-07 |
| None |
Unchecked |
Kcat/Km |
1000.0 |
/M/s |
10.1021/acs.jmedchem.6b00096 |
| None |
Unchecked |
Kd |
75000.0 |
nM |
10.1016/j.bmc.2020.115437 |
| None |
Unchecked |
Ki |
nan |
None |
None |
| None |
Unchecked |
Km |
300.0 |
nM |
10.1128/aac.01462-06 |
| None |
Unchecked |
Km |
920.0 |
nM |
10.1021/acs.jmedchem.6b00096 |
| None |
Unchecked |
Km |
2000.0 |
nM |
10.1128/aac.01336-09 |
| None |
Unchecked |
Km |
3400.0 |
nM |
10.1128/aac.00175-08 |
| None |
Unchecked |
Km |
5000.0 |
nM |
10.1128/aac.00409-10 |
| None |
Unchecked |
Km |
8400.0 |
nM |
10.1128/aac.00858-10 |
| None |
Unchecked |
Km |
8800.0 |
nM |
10.1128/aac.01004-09 |
| None |
Unchecked |
Km |
10000.0 |
nM |
10.1128/aac.00409-10 |
| None |
Unchecked |
Km |
10000.0 |
nM |
10.1128/aac.00774-09 |
| None |
Unchecked |
Km |
10000.0 |
nM |
10.1128/aac.00858-10 |
| None |
Unchecked |
Km |
10000.0 |
nM |
10.1128/aac.01336-09 |
| None |
Unchecked |
Km |
12000.0 |
nM |
10.1128/aac.00961-09 |
| None |
Unchecked |
Km |
12000.0 |
nM |
10.1128/aac.01337-07 |
| None |
Unchecked |
Km |
50000.0 |
nM |
10.1128/aac.00166-08 |
| None |
Unchecked |
Km |
85000.0 |
nM |
10.1128/aac.00409-10 |
| None |
Unchecked |
Km |
90000.0 |
nM |
10.1128/aac.01004-09 |
| None |
Unchecked |
Km |
100000.0 |
nM |
10.1128/aac.00856-09 |
| None |
Unchecked |
Km |
120000.0 |
nM |
10.1128/aac.00175-08 |
| None |
Unchecked |
Km |
190000.0 |
nM |
10.1128/aac.00409-10 |
| None |
Unchecked |
Km |
280000.0 |
nM |
10.1128/aac.00083-07 |
| None |
Unchecked |
Km |
990000.0 |
nM |
10.1128/aac.01062-07 |
| None |
Unchecked |
Km |
nan |
None |
10.1128/aac.01600-06 |
| None |
Unchecked |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115598 |
| None |
Unchecked |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.09.039 |
| None |
Unchecked |
MIC |
1.0 |
ug.mL-1 |
10.1016/s0960-894x(00)00253-5 |
| None |
Unchecked |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115598 |
| None |
Unchecked |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116128 |
| None |
Unchecked |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116128 |
| None |
Unchecked |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.007 |
| None |
Unchecked |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116128 |
| None |
Unchecked |
MIC |
nan |
None |
10.1016/j.bmc.2020.115598 |
| None |
Unchecked |
Ratio |
1.0 |
None |
10.1128/aac.00413-08 |
| None |
Unchecked |
Ratio |
2.0 |
None |
10.1128/aac.00413-08 |
| None |
Unchecked |
Ratio |
4.0 |
None |
10.1128/aac.00413-08 |
| None |
Unchecked |
Ratio |
8.0 |
None |
10.1128/aac.00413-08 |
| None |
Unchecked |
Ratio |
28.05 |
None |
10.1128/aac.00160-07 |
| None |
Unchecked |
Ratio |
32.0 |
None |
10.1128/aac.00413-08 |
| None |
Unchecked |
Ratio |
112.2 |
None |
10.1128/aac.00160-07 |
| None |
Unchecked |
Ratio |
1300.0 |
/M/s |
10.1021/acs.jmedchem.6b00096 |
| None |
Unchecked |
Ratio |
nan |
None |
10.1021/acs.jmedchem.2c01674 |
| None |
Unchecked |
Relative hydrolysis |
28.0 |
None |
10.1016/S0960-894X(97)00282-5 |
| None |
Unchecked |
Stability |
100.0 |
% |
10.1016/s0960-894x(01)00451-6 |