3-{[5-(dimethylcarbamoyl)pyrrolidin-3-yl]sulfanyl}-6-(1-hydroxyethyl)-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid

AlkaPlorer ID: AK000935

Synonym: None

IUPAC Name: (4R,5S,6S)-3-[(3S,5S)-5-(dimethylcarbamoyl)pyrrolidin-3-yl]sulfanyl-6-[(1R)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid

Structure

SMILES: C[C@@H](O)[C@H]1C(=O)N2C(C(=O)O)=C(S[C@@H]3CN[C@H](C(=O)N(C)C)C3)[C@H](C)[C@H]12

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InChI: InChI=1S/C17H25N3O5S/c1-7-12-11(8(2)21)16(23)20(12)13(17(24)25)14(7)26-9-5-10(18-6-9)15(22)19(3)4/h7-12,18,21H,5-6H2,1-4H3,(H,24,25)/t7-,8-,9+,10+,11-,12-/m1/s1

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InChIKey: DMJNNHOOLUXYBV-PQTSNVLCSA-N

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Reference

PubChem CID: 40466974

CAS: 119478-56-7

NPASS: NPC478435

Source

Species Genus Family Order Class Phylum Kingdom Domain

Properties Information

Molecule Weight: 383.4700000000002

TPSA: 110.18

MolLogP: -0.3079999999999994

Number of H-Donors: 3

Number of H-Acceptors: 6

RingCount: 3

Activities Information

Organism Target Name Standard Type Standard Value Standard Units doi
Acinetobacter Acinetobacter Activity 0.0 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter Activity 0.4 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter Activity 1.4 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter Activity 1.7 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter Activity 18.0 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter Activity 80.6 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter Activity 97.9 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter Activity 100.0 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter MIC 0.015 ug.mL-1 10.1128/aac.00381-08
Acinetobacter Acinetobacter MIC 16.0 ug.mL-1 10.1128/aac.00381-08
Acinetobacter Acinetobacter MIC 64.0 ug.mL-1 10.1016/j.bmc.2021.116142
Acinetobacter Acinetobacter MIC 128.0 ug.mL-1 10.1016/j.bmc.2021.116142
Acinetobacter Acinetobacter MIC50 1.0 ug.mL-1 10.1128/aac.00381-08
Acinetobacter Acinetobacter MIC50 32.0 ug.mL-1 10.1128/aac.00381-08
Acinetobacter Acinetobacter MIC90 4.0 ug.mL-1 10.1128/aac.00381-08
Acinetobacter Acinetobacter MIC90 32.0 ug.mL-1 10.1128/aac.00381-08
Acinetobacter baumannii Acinetobacter baumannii Activity 0.0 % 10.1128/aac.00400-09
Acinetobacter baumannii Acinetobacter baumannii Activity 4.0 % 10.1128/aac.01099-06
Acinetobacter baumannii Acinetobacter baumannii Activity 8.0 % 10.1128/aac.00400-09
Acinetobacter baumannii Acinetobacter baumannii Activity 12.0 % 10.1128/aac.01533-08
Acinetobacter baumannii Acinetobacter baumannii Activity 22.4 % 10.1128/aac.00570-08
Acinetobacter baumannii Acinetobacter baumannii Activity 22.9 % 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii Activity 77.1 % 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii Activity 92.0 % 10.1128/aac.00400-09
Acinetobacter baumannii Acinetobacter baumannii Activity nan None 10.1128/aac.00748-09
Acinetobacter baumannii Acinetobacter baumannii Activity nan None 10.1128/aac.00764-10
Acinetobacter baumannii Acinetobacter baumannii Activity nan None 10.1128/aac.00963-09
Acinetobacter baumannii Acinetobacter baumannii Activity nan None 10.1128/aac.01525-09
Acinetobacter baumannii Acinetobacter baumannii Activity nan None 10.1128/aac.01533-08
Acinetobacter baumannii Acinetobacter baumannii ED90 25.0 mg kg-1 10.1021/acs.jmedchem.8b00091
Acinetobacter baumannii Acinetobacter baumannii ED90 50.0 mg kg-1 10.1021/acs.jmedchem.8b00091
Acinetobacter baumannii Acinetobacter baumannii FC 0.1 None 10.1021/jm501050e
Acinetobacter baumannii Acinetobacter baumannii FC 2.0 None 10.1128/aac.01512-06
Acinetobacter baumannii Acinetobacter baumannii FICI 0.281 None 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii FICI 0.5 None 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii Inhibition 10.36 % 10.6019/CHEMBL4513141
Acinetobacter baumannii Acinetobacter baumannii Inhibition 100.0 % 10.1021/acs.jmedchem.2c01905
Acinetobacter baumannii Acinetobacter baumannii MIC 0.06 ug.mL-1 10.1128/aac.00400-09
Acinetobacter baumannii Acinetobacter baumannii MIC 0.064 ug.mL-1 10.1128/aac.00072-09
Acinetobacter baumannii Acinetobacter baumannii MIC 0.094 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 0.12 ug.mL-1 10.1128/aac.00336-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.12 ug.mL-1 10.1128/aac.00689-07
Acinetobacter baumannii Acinetobacter baumannii MIC 0.125 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.125 ug.mL-1 10.1128/aac.00570-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.125 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 0.19 ug.mL-1 10.1128/aac.00598-10
Acinetobacter baumannii Acinetobacter baumannii MIC 0.19 ug.mL-1 10.1128/aac.00856-09
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1016/j.ejmech.2018.08.025
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1021/acs.jmedchem.8b00091
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1021/jm400560z
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1021/ml200012f
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1039/C5MD00377F
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1128/aac.00050-10
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1128/aac.00393-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1128/aac.00491-10
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1128/aac.00598-10
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1128/aac.00689-07
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1128/aac.00978-07
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1128/aac.01004-09
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1128/aac.01398-09
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1128/aac.01684-07
Acinetobacter baumannii Acinetobacter baumannii MIC 0.38 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.38 ug.mL-1 10.1128/aac.01512-06
Acinetobacter baumannii Acinetobacter baumannii MIC 0.38 ug.mL-1 10.1128/aac.01684-07
Acinetobacter baumannii Acinetobacter baumannii MIC 0.5 ug.mL-1 10.1021/acs.jmedchem.6b00746
Acinetobacter baumannii Acinetobacter baumannii MIC 0.5 ug.mL-1 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii MIC 0.5 ug.mL-1 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii MIC 0.5 ug.mL-1 10.1128/aac.00393-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.5 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.5 ug.mL-1 10.1128/aac.00491-10
Acinetobacter baumannii Acinetobacter baumannii MIC 0.5 ug.mL-1 10.1128/aac.00689-07
Acinetobacter baumannii Acinetobacter baumannii MIC 0.5 ug.mL-1 10.1128/aac.01407-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.5 ug.mL-1 10.1128/aac.01512-06
Acinetobacter baumannii Acinetobacter baumannii MIC 0.5 ug.mL-1 10.1128/aac.01663-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.75 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 0.75 ug.mL-1 10.1128/aac.01512-06
Acinetobacter baumannii Acinetobacter baumannii MIC 0.75 ug.mL-1 10.1128/aac.01684-07
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1016/j.ejmech.2018.08.025
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1039/C5MD00377F
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1128/aac.00050-10
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1128/aac.00178-09
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1128/aac.00689-07
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1128/aac.01433-06
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1128/aac.01525-09
Acinetobacter baumannii Acinetobacter baumannii MIC 1.5 ug.mL-1 10.1128/aac.00072-09
Acinetobacter baumannii Acinetobacter baumannii MIC 1.5 ug.mL-1 10.1128/aac.01512-06
Acinetobacter baumannii Acinetobacter baumannii MIC 1.5 ug.mL-1 10.1128/aac.01684-07
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1039/C5MD00377F
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.00050-10
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.00267-07
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.00689-07
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.00978-07
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.01139-06
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.01684-07
Acinetobacter baumannii Acinetobacter baumannii MIC 3.0 ug.mL-1 10.1128/aac.01512-06
Acinetobacter baumannii Acinetobacter baumannii MIC 3.0 ug.mL-1 10.1128/aac.01663-08
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1016/j.ejmech.2018.08.025
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.00267-07
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.00292-09
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.00366-08
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.00689-07
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.01512-06
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.01684-07
Acinetobacter baumannii Acinetobacter baumannii MIC 6.0 ug.mL-1 10.1128/aac.00072-09
Acinetobacter baumannii Acinetobacter baumannii MIC 6.0 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 6.0 ug.mL-1 10.1128/aac.00570-08
Acinetobacter baumannii Acinetobacter baumannii MIC 6.0 ug.mL-1 10.1128/aac.01512-06
Acinetobacter baumannii Acinetobacter baumannii MIC 6.0 ug.mL-1 10.1128/aac.01663-08
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1039/C5MD00377F
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.00072-08
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.00292-09
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.00491-10
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.00689-07
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.00838-06
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.01512-06
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.01799-09
Acinetobacter baumannii Acinetobacter baumannii MIC 12.0 ug.mL-1 10.1128/aac.00292-09
Acinetobacter baumannii Acinetobacter baumannii MIC 12.0 ug.mL-1 10.1128/aac.01684-07
Acinetobacter baumannii Acinetobacter baumannii MIC 12.5 ug.mL-1 10.1016/j.ejmech.2007.02.001
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1016/j.bmc.2013.09.041
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1016/j.bmcl.2021.127928
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1016/j.ejmech.2018.06.014
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1016/j.ejmech.2018.08.025
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.2c01905
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.8b00091
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.00292-09
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.00393-08
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.00491-10
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.00689-07
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.00978-07
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.01259-06
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.01398-09
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.01414-07
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.01512-06
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.01684-07
Acinetobacter baumannii Acinetobacter baumannii MIC 24.0 ug.mL-1 10.1128/aac.00292-09
Acinetobacter baumannii Acinetobacter baumannii MIC 24.0 ug.mL-1 10.1128/aac.00861-09
Acinetobacter baumannii Acinetobacter baumannii MIC 24.0 ug.mL-1 10.1128/aac.01684-07
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1016/j.bmcl.2021.127928
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.08.025
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1021/acs.jmedchem.9b00720
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1021/jm501050e
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.00267-07
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.00292-09
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.00393-08
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.00598-10
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.00689-07
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.00856-09
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.01121-08
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.01259-06
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.01464-06
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.01512-06
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.01525-09
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.01684-07
Acinetobacter baumannii Acinetobacter baumannii MIC 64.0 ug.mL-1 10.1016/j.bmcl.2021.127928
Acinetobacter baumannii Acinetobacter baumannii MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.08.025
Acinetobacter baumannii Acinetobacter baumannii MIC 64.0 ug.mL-1 10.1021/acs.jmedchem.6b01261
Acinetobacter baumannii Acinetobacter baumannii MIC 64.0 ug.mL-1 10.1021/acs.jmedchem.8b00091
Acinetobacter baumannii Acinetobacter baumannii MIC 64.0 ug.mL-1 10.1128/aac.00292-09
Acinetobacter baumannii Acinetobacter baumannii MIC 64.0 ug.mL-1 10.1128/aac.00978-07
Acinetobacter baumannii Acinetobacter baumannii MIC 64.0 ug.mL-1 10.1128/aac.01004-09
Acinetobacter baumannii Acinetobacter baumannii MIC 64.0 ug.mL-1 10.1128/aac.01259-06
Acinetobacter baumannii Acinetobacter baumannii MIC 128.0 ug.mL-1 10.1128/aac.00178-09
Acinetobacter baumannii Acinetobacter baumannii MIC 128.0 ug.mL-1 10.1128/aac.01259-06
Acinetobacter baumannii Acinetobacter baumannii MIC 128.0 ug.mL-1 10.1128/aac.01525-09
Acinetobacter baumannii Acinetobacter baumannii MIC 256.0 ug.mL-1 10.1128/aac.00178-09
Acinetobacter baumannii Acinetobacter baumannii MIC 256.0 ug.mL-1 10.1128/aac.00689-07
Acinetobacter baumannii Acinetobacter baumannii MIC 500.0 ug.mL-1 10.1128/aac.01502-06
Acinetobacter baumannii Acinetobacter baumannii MIC 1000.0 nM 10.1021/acs.jmedchem.1c00614
Acinetobacter baumannii Acinetobacter baumannii MIC 3000.0 ug.mL-1 10.1128/aac.01502-06
Acinetobacter baumannii Acinetobacter baumannii MIC 4000.0 ug.mL-1 10.1128/aac.01502-06
Acinetobacter baumannii Acinetobacter baumannii MIC 8000.0 ug.mL-1 10.1128/aac.01502-06
Acinetobacter baumannii Acinetobacter baumannii MIC 12000.0 ug.mL-1 10.1128/aac.01502-06
Acinetobacter baumannii Acinetobacter baumannii MIC 32000.0 nM 10.1021/acs.jmedchem.1c00621
Acinetobacter baumannii Acinetobacter baumannii MIC50 0.5 ug.mL-1 10.1128/aac.00400-09
Acinetobacter baumannii Acinetobacter baumannii MIC50 2.0 ug.mL-1 10.1128/aac.00336-08
Acinetobacter baumannii Acinetobacter baumannii MIC50 8.0 ug.mL-1 10.1016/j.ejmech.2021.113436
Acinetobacter baumannii Acinetobacter baumannii MIC50 8.0 ug.mL-1 10.1128/aac.00366-08
Acinetobacter baumannii Acinetobacter baumannii MIC50 16.0 ug.mL-1 10.1128/aac.01099-06
Acinetobacter baumannii Acinetobacter baumannii MIC50 32.0 ug.mL-1 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii MIC50 64.0 ug.mL-1 10.1016/j.ejmech.2021.113436
Acinetobacter baumannii Acinetobacter baumannii MIC90 1.0 ug.mL-1 10.1016/j.bmcl.2016.06.019
Acinetobacter baumannii Acinetobacter baumannii MIC90 4.0 ug.mL-1 10.1128/aac.00400-09
Acinetobacter baumannii Acinetobacter baumannii MIC90 8.0 ug.mL-1 10.1128/aac.00366-08
Acinetobacter baumannii Acinetobacter baumannii MIC90 32.0 ug.mL-1 10.1128/aac.00336-08
Acinetobacter baumannii Acinetobacter baumannii MIC90 64.0 ug.mL-1 10.1016/j.bmcl.2012.07.005
Acinetobacter baumannii Acinetobacter baumannii MIC90 64.0 ug.mL-1 10.1016/j.bmcl.2016.06.019
Acinetobacter baumannii Acinetobacter baumannii MIC90 64.0 ug.mL-1 10.1016/j.ejmech.2021.113436
Acinetobacter baumannii Acinetobacter baumannii MIC90 64.0 ug.mL-1 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii MIC90 128.0 ug.mL-1 10.1128/aac.01099-06
Acinetobacter baumannii Acinetobacter baumannii MPC 1.0 ug ml-1 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii MPC 2.0 ug ml-1 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii MPC 4.0 ug ml-1 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii MPC 8.0 ug ml-1 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii MPC 16.0 ug ml-1 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii MPC 32.0 ug ml-1 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii MPC 128.0 ug ml-1 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii PD50 25.0 mg kg-1 10.1021/acs.jmedchem.8b00091
Acinetobacter baumannii Acinetobacter baumannii PD50 50.0 mg kg-1 10.1021/acs.jmedchem.8b00091
Acinetobacter baumannii Acinetobacter baumannii Ratio 2.0 None 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii Ratio 4.0 None 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii Ratio 8.0 None 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii Ratio 16.0 None 10.1128/aac.00033-10
Acinetobacter baumannii Acinetobacter baumannii Ratio 64.0 None 10.1128/aac.00491-10
Acinetobacter baumannii Beta-lactamase OXA-23 Activity 0.029 % 10.1128/aac.01004-09
Acinetobacter baumannii Beta-lactamase OXA-23 Activity 10.0 % 10.1128/aac.01004-09
Acinetobacter baumannii Beta-lactamase OXA-23 Activity 14.9 % 10.1128/aac.01004-09
Acinetobacter baumannii Beta-lactamase OXA-23 Activity 140.0 % 10.1128/aac.01004-09
Acinetobacter baumannii Beta-lactamase OXA-23 Kcat 0.13 nmol/min 10.1128/aac.01004-09
Acinetobacter baumannii Beta-lactamase OXA-23 Kcat 170.0 /s 10.1128/aac.01004-09
Acinetobacter baumannii Beta-lactamase OXA-23 Kcat/Km 0.052 /s/microM 10.1128/aac.01004-09
Acinetobacter baumannii Beta-lactamase OXA-23 Kcat/Km 1.3 /s/microM 10.1128/aac.01004-09
Acinetobacter baumannii Beta-lactamase OXA-23 Km 2500.0 nM 10.1128/aac.01004-09
Acinetobacter baumannii Beta-lactamase OXA-23 Km 130000.0 nM 10.1128/aac.01004-09
Acinetobacter baylyi Acinetobacter baylyi MIC 0.25 ug.mL-1 10.1128/aac.01674-09
Acinetobacter baylyi Acinetobacter baylyi MIC 32.0 ug.mL-1 10.1128/aac.01674-09
Acinetobacter calcoaceticus Acinetobacter calcoaceticus MIC 0.5 ug.mL-1 10.1016/S0960-894X(97)00282-5
Acinetobacter calcoaceticus Acinetobacter calcoaceticus MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.03.031
Acinetobacter calcoaceticus Acinetobacter calcoaceticus MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.03.031
Acinetobacter haemolyticus Acinetobacter haemolyticus MIC 32.0 ug.mL-1 10.1128/aac.00267-07
Acinetobacter lwoffii Acinetobacter lwoffii MIC 2.0 ug.mL-1 10.1128/aac.00598-10
Acinetobacter lwoffii Acinetobacter lwoffii MIC 4.0 ug.mL-1 10.1128/aac.00598-10
Acinetobacter lwoffii Acinetobacter lwoffii MIC 8.0 ug.mL-1 10.1128/aac.00598-10
Acinetobacter lwoffii Acinetobacter lwoffii MIC 16.0 ug.mL-1 10.1128/aac.00598-10
Acinetobacter lwoffii Acinetobacter lwoffii MIC 32.0 ug.mL-1 10.1128/aac.00598-10
Acinetobacter lwoffii Acinetobacter lwoffii MIC 64.0 ug.mL-1 10.1128/aac.00598-10
Acinetobacter pittii Acinetobacter pittii Activity 57.9 % 10.1128/aac.01624-09
Acinetobacter pittii Acinetobacter pittii MIC 0.094 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 0.125 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 0.19 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 0.25 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 0.38 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 0.47 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 0.5 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 0.5 ug.mL-1 10.1128/aac.01624-09
Acinetobacter pittii Acinetobacter pittii MIC 0.64 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 0.75 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 1.0 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 1.5 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 3.0 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 4.0 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 6.0 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 8.0 ug.mL-1 10.1128/aac.00072-08
Acinetobacter pittii Acinetobacter pittii MIC 16.0 ug.mL-1 10.1128/aac.01624-09
Acinetobacter pittii Acinetobacter pittii MIC 32.0 ug.mL-1 10.1128/aac.01624-09
Acinetobacter pittii Acinetobacter pittii MIC 64.0 ug.mL-1 10.1128/aac.01624-09
Acinetobacter pittii Acinetobacter pittii MIC50 16.0 ug.mL-1 10.1128/aac.01624-09
Acinetobacter pittii Acinetobacter pittii MIC90 32.0 ug.mL-1 10.1128/aac.01624-09
Acinetobacter pittii Acinetobacter pittii Ratio 3.0 None 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii Ratio 4.0 None 10.1128/aac.00485-08
Acinetobacter radioresistens Acinetobacter radioresistens GI nan None 10.1128/aac.01304-07
Acinetobacter radioresistens Acinetobacter radioresistens MIC 0.25 ug.mL-1 10.1128/aac.00999-08
Acinetobacter radioresistens Acinetobacter radioresistens MIC 1.0 ug.mL-1 10.1128/aac.00999-08
Acinetobacter sp. Acinetobacter sp. MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Acinetobacter sp. Acinetobacter sp. MIC 8.0 ug.mL-1 10.1128/aac.00838-06
Acinetobacter sp. Acinetobacter sp. MIC50 1.0 ug.mL-1 10.1021/jm400560z
Acinetobacter sp. Acinetobacter sp. MIC50 1.0 ug.mL-1 10.1021/ml200012f
Acinetobacter sp. Acinetobacter sp. MIC50 1.0 ug.mL-1 10.1128/aac.01525-09
Acinetobacter sp. Acinetobacter sp. MIC90 32.0 ug.mL-1 10.1021/jm400560z
Acinetobacter sp. Acinetobacter sp. MIC90 32.0 ug.mL-1 10.1021/ml200012f
Acinetobacter sp. Acinetobacter sp. MIC90 32.0 ug.mL-1 10.1128/aac.01525-09
Actinomyces israelii Actinomyces israelii Activity 8.0 % 10.1128/aac.00481-10
Actinomyces israelii Actinomyces israelii Activity 92.0 % 10.1128/aac.00481-10
Actinomyces israelii Actinomyces israelii MIC 0.008 ug.mL-1 10.1128/aac.00481-10
Actinomyces israelii Actinomyces israelii MIC50 0.125 ug.mL-1 10.1128/aac.00481-10
Actinomyces israelii Actinomyces israelii MIC90 2.0 ug.mL-1 10.1128/aac.00481-10
Actinomyces naeslundii Actinomyces naeslundii Activity 8.0 % 10.1128/aac.00481-10
Actinomyces naeslundii Actinomyces naeslundii Activity 92.0 % 10.1128/aac.00481-10
Actinomyces naeslundii Actinomyces naeslundii MIC 0.008 ug.mL-1 10.1128/aac.00481-10
Actinomyces naeslundii Actinomyces naeslundii MIC50 0.125 ug.mL-1 10.1128/aac.00481-10
Actinomyces naeslundii Actinomyces naeslundii MIC90 2.0 ug.mL-1 10.1128/aac.00481-10
Aeromonas allosaccharophila Extended-spectrum beta-lactamase PER-6 Kcat 0.004 /s 10.1128/aac.01585-09
Aeromonas allosaccharophila Extended-spectrum beta-lactamase PER-6 Kcat/Km 0.4 /uM/s 10.1128/aac.01585-09
Aeromonas allosaccharophila Extended-spectrum beta-lactamase PER-6 Km 10000.0 nM 10.1128/aac.01585-09
Aeromonas caviae Aeromonas caviae MIC 0.125 ug.mL-1 10.1016/j.bmc.2013.09.041
Aeromonas caviae Aeromonas caviae MIC 1.0 ug.mL-1 10.1016/j.bmc.2013.09.041
Aeromonas caviae Aeromonas caviae MIC 1024.0 ug.mL-1 10.1128/aac.01462-06
Aeromonas caviae IMP-19 Kcat 1.0 /s 10.1128/aac.01462-06
Aeromonas caviae IMP-19 Kcat/Km 0.14 None 10.1128/aac.01462-06
Aeromonas caviae IMP-19 Km 7000.0 nM 10.1128/aac.01462-06
Aeromonas hydrophila Aeromonas hydrophila MIC 0.06 ug.mL-1 10.1016/j.bmc.2013.09.041
Anaerococcus prevotii Anaerococcus prevotii Activity 0.0 % 10.1128/aac.00481-10
Anaerococcus prevotii Anaerococcus prevotii Activity 0.0 % 10.1128/aac.00696-08
Anaerococcus prevotii Anaerococcus prevotii Activity 0.0 % 10.1128/aac.01128-07
Anaerococcus prevotii Anaerococcus prevotii Activity 100.0 % 10.1128/aac.00481-10
Anaerococcus prevotii Anaerococcus prevotii MIC 0.008 ug.mL-1 10.1128/aac.00481-10
Anaerococcus prevotii Anaerococcus prevotii MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Anaerococcus prevotii Anaerococcus prevotii MIC 0.06 ug.mL-1 10.1128/aac.00696-08
Anaerococcus prevotii Anaerococcus prevotii MIC 0.25 ug.mL-1 10.1128/aac.00595-08
Anaerococcus prevotii Anaerococcus prevotii MIC50 0.03 ug.mL-1 10.1128/aac.01128-07
Anaerococcus prevotii Anaerococcus prevotii MIC50 0.06 ug.mL-1 10.1128/aac.00481-10
Anaerococcus prevotii Anaerococcus prevotii MIC50 0.125 ug.mL-1 10.1128/aac.00696-08
Anaerococcus prevotii Anaerococcus prevotii MIC90 0.125 ug.mL-1 10.1128/aac.00481-10
Anaerococcus prevotii Anaerococcus prevotii MIC90 0.125 ug.mL-1 10.1128/aac.01128-07
Anaerococcus prevotii Anaerococcus prevotii MIC90 0.5 ug.mL-1 10.1128/aac.00696-08
Anaerococcus tetradius Anaerococcus tetradius Activity 0.0 % 10.1128/aac.01128-07
Anaerococcus tetradius Anaerococcus tetradius MIC 0.03 ug.mL-1 10.1128/aac.00910-07
Anaerococcus tetradius Anaerococcus tetradius MIC50 0.03 ug.mL-1 10.1128/aac.00910-07
Anaerococcus tetradius Anaerococcus tetradius MIC50 0.03 ug.mL-1 10.1128/aac.01128-07
Anaerococcus tetradius Anaerococcus tetradius MIC90 0.125 ug.mL-1 10.1128/aac.01128-07
Anaerococcus vaginalis Anaerococcus vaginalis Activity 0.0 % 10.1128/aac.01128-07
Anaerococcus vaginalis Anaerococcus vaginalis MIC50 0.03 ug.mL-1 10.1128/aac.01128-07
Anaerococcus vaginalis Anaerococcus vaginalis MIC90 0.125 ug.mL-1 10.1128/aac.01128-07
Anaerocolumna aminovalerica Anaerocolumna aminovalerica Activity 0.0 % 10.1128/aac.01128-07
Anaerocolumna aminovalerica Anaerocolumna aminovalerica MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Anaerocolumna aminovalerica Anaerocolumna aminovalerica MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
Aspergillus fumigatus Aspergillus fumigatus IC50 300.0 nM 10.1021/acs.jnatprod.9b00187
Bacillus anthracis Bacillus anthracis MIC 0.06 ug.mL-1 10.1128/aac.00737-08
Bacillus anthracis Bacillus anthracis MIC 0.12 ug.mL-1 10.1128/aac.00737-08
Bacillus anthracis Bacillus anthracis MIC 0.25 ug.mL-1 10.1128/aac.00737-08
Bacillus anthracis Bacillus anthracis MIC 0.5 ug.mL-1 10.1128/aac.00737-08
Bacillus anthracis Bacillus anthracis MIC 4.0 ug.mL-1 10.1128/aac.00737-08
Bacillus anthracis Bacillus anthracis MIC 8.0 ug.mL-1 10.1128/aac.00737-08
Bacillus anthracis Bacillus anthracis MIC 32.0 ug.mL-1 10.1128/aac.00737-08
Bacillus subtilis Bacillus subtilis MIC 0.05 ug.mL-1 10.1016/j.ejmech.2006.10.006
Bacillus subtilis Bacillus subtilis MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
Bacillus subtilis Bacillus subtilis MIC 3.125 ug.mL-1 10.1016/j.bmc.2016.02.013
Bacillus subtilis Bacillus subtilis MIC 1000.0 nM 10.1021/acs.jmedchem.1c00614
Bacillus subtilis Bacillus subtilis MIC 1000.0 nM 10.1021/acs.jmedchem.1c02140
Bacteria Cell membrane Activity 12.2 % 10.1016/j.ejmech.2022.114278
Bacteria Cell membrane Activity 14.7 % 10.1016/j.ejmech.2022.114278
Bacteria Cell membrane Activity 17.2 % 10.1016/j.ejmech.2022.114278
Bacteria Cell membrane Activity 22.1 % 10.1016/j.ejmech.2022.114278
Bacteria Cell membrane Activity nan None 10.1016/j.ejmech.2018.06.054
Bacteroides caccae Bacteroides caccae Activity 0.0 % 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae Activity 0.0 % 10.1128/aac.00696-08
Bacteroides caccae Bacteroides caccae Activity 0.0 % 10.1128/aac.01128-07
Bacteroides caccae Bacteroides caccae Activity 0.5 % 10.1128/aac.01435-06
Bacteroides caccae Bacteroides caccae Activity 4.0 % 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae Activity 96.0 % 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae Activity 98.0 % 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae MIC 0.12 ug.mL-1 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae MIC 0.125 ug.mL-1 10.1128/aac.00696-08
Bacteroides caccae Bacteroides caccae MIC 0.13 ug.mL-1 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae MIC 0.4 ug.mL-1 10.1128/aac.01435-06
Bacteroides caccae Bacteroides caccae MIC50 0.25 ug.mL-1 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae MIC50 0.25 ug.mL-1 10.1128/aac.00595-08
Bacteroides caccae Bacteroides caccae MIC50 0.25 ug.mL-1 10.1128/aac.00696-08
Bacteroides caccae Bacteroides caccae MIC50 0.25 ug.mL-1 10.1128/aac.01128-07
Bacteroides caccae Bacteroides caccae MIC50 0.5 ug.mL-1 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
Bacteroides caccae Bacteroides caccae MIC90 1.0 ug.mL-1 10.1128/aac.01435-06
Bacteroides caccae Bacteroides caccae MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae MIC90 2.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae MIC90 2.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides caccae Bacteroides caccae MIC90 4.0 ug.mL-1 10.1128/aac.00595-08
Bacteroides fragilis Bacteroides fragilis Activity 0.0 % 10.1128/aac.01128-07
Bacteroides fragilis Bacteroides fragilis Activity 1.0 % 10.1128/aac.01435-06
Bacteroides fragilis Bacteroides fragilis Activity 1.5 % 10.1128/aac.00696-08
Bacteroides fragilis Bacteroides fragilis Activity 3.0 % 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis Activity 5.0 % 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis Activity 88.0 % 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis Activity 90.0 % 10.1128/aac.00910-07
Bacteroides fragilis Bacteroides fragilis Activity 92.0 % 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis Activity 99.0 % 10.1128/aac.00910-07
Bacteroides fragilis Bacteroides fragilis MIC 0.05 ug.mL-1 10.1128/aac.00595-08
Bacteroides fragilis Bacteroides fragilis MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis MIC 0.06 ug.mL-1 10.1128/aac.00910-07
Bacteroides fragilis Bacteroides fragilis MIC 0.12 ug.mL-1 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis MIC 0.125 ug.mL-1 10.1128/aac.00595-08
Bacteroides fragilis Bacteroides fragilis MIC 0.125 ug.mL-1 10.1128/aac.00696-08
Bacteroides fragilis Bacteroides fragilis MIC 0.125 ug.mL-1 10.1128/aac.00910-07
Bacteroides fragilis Bacteroides fragilis MIC 0.25 ug.mL-1 10.1128/aac.00595-08
Bacteroides fragilis Bacteroides fragilis MIC 0.38 ug.mL-1 10.1128/aac.01435-06
Bacteroides fragilis Bacteroides fragilis MIC 2.0 ug.mL-1 10.1128/aac.00595-08
Bacteroides fragilis Bacteroides fragilis MIC 128.0 ug.mL-1 10.1128/aac.00595-08
Bacteroides fragilis Bacteroides fragilis MIC50 0.125 ug.mL-1 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis MIC50 0.125 ug.mL-1 10.1128/aac.00910-07
Bacteroides fragilis Bacteroides fragilis MIC50 0.125 ug.mL-1 10.1128/aac.01128-07
Bacteroides fragilis Bacteroides fragilis MIC50 0.25 ug.mL-1 10.1128/aac.00595-08
Bacteroides fragilis Bacteroides fragilis MIC50 0.25 ug.mL-1 10.1128/aac.00696-08
Bacteroides fragilis Bacteroides fragilis MIC50 0.28 ug.mL-1 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis MIC90 0.25 ug.mL-1 10.1128/aac.01128-07
Bacteroides fragilis Bacteroides fragilis MIC90 0.5 ug.mL-1 10.1128/aac.00595-08
Bacteroides fragilis Bacteroides fragilis MIC90 1.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides fragilis Bacteroides fragilis MIC90 1.0 ug.mL-1 10.1128/aac.00910-07
Bacteroides fragilis Bacteroides fragilis MIC90 1.0 ug.mL-1 10.1128/aac.01435-06
Bacteroides fragilis Bacteroides fragilis MIC90 4.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis MIC90 8.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides ovatus Bacteroides ovatus Activity 0.0 % 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus Activity 0.0 % 10.1128/aac.00696-08
Bacteroides ovatus Bacteroides ovatus Activity 0.0 % 10.1128/aac.01128-07
Bacteroides ovatus Bacteroides ovatus Activity 98.0 % 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus MIC 0.125 ug.mL-1 10.1128/aac.00696-08
Bacteroides ovatus Bacteroides ovatus MIC 0.13 ug.mL-1 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus MIC 0.25 ug.mL-1 10.1128/aac.00595-08
Bacteroides ovatus Bacteroides ovatus MIC 0.25 ug.mL-1 10.1128/aac.00910-07
Bacteroides ovatus Bacteroides ovatus MIC50 0.25 ug.mL-1 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus MIC50 0.25 ug.mL-1 10.1128/aac.00910-07
Bacteroides ovatus Bacteroides ovatus MIC50 0.25 ug.mL-1 10.1128/aac.01128-07
Bacteroides ovatus Bacteroides ovatus MIC50 0.5 ug.mL-1 10.1128/aac.00696-08
Bacteroides ovatus Bacteroides ovatus MIC90 0.5 ug.mL-1 10.1128/aac.00910-07
Bacteroides ovatus Bacteroides ovatus MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
Bacteroides ovatus Bacteroides ovatus MIC90 2.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus MIC90 2.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides stercoris Bacteroides stercoris Activity 0.0 % 10.1128/aac.01128-07
Bacteroides stercoris Bacteroides stercoris Activity 0.5 % 10.1128/aac.01435-06
Bacteroides stercoris Bacteroides stercoris MIC 0.4 ug.mL-1 10.1128/aac.01435-06
Bacteroides stercoris Bacteroides stercoris MIC50 0.25 ug.mL-1 10.1128/aac.00595-08
Bacteroides stercoris Bacteroides stercoris MIC50 0.25 ug.mL-1 10.1128/aac.01128-07
Bacteroides stercoris Bacteroides stercoris MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
Bacteroides stercoris Bacteroides stercoris MIC90 1.0 ug.mL-1 10.1128/aac.01435-06
Bacteroides stercoris Bacteroides stercoris MIC90 4.0 ug.mL-1 10.1128/aac.00595-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 0.0 % 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 0.0 % 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 0.0 % 10.1128/aac.00696-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 0.0 % 10.1128/aac.01128-07
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 0.1 % 10.1128/aac.01435-06
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 90.0 % 10.1128/aac.00910-07
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 97.0 % 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 98.0 % 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 99.0 % 10.1128/aac.00910-07
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 0.12 ug.mL-1 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 0.125 ug.mL-1 10.1128/aac.00696-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 0.125 ug.mL-1 10.1128/aac.00910-07
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 0.13 ug.mL-1 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 0.25 ug.mL-1 10.1128/aac.00595-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 0.25 ug.mL-1 10.1128/aac.00910-07
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 0.47 ug.mL-1 10.1128/aac.01435-06
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 0.25 ug.mL-1 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 0.25 ug.mL-1 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 0.25 ug.mL-1 10.1128/aac.00910-07
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 0.25 ug.mL-1 10.1128/aac.01128-07
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 0.5 ug.mL-1 10.1128/aac.00595-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 0.5 ug.mL-1 10.1128/aac.00696-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 0.5 ug.mL-1 10.1128/aac.00910-07
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 1.0 ug.mL-1 10.1128/aac.01435-06
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 2.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 2.0 ug.mL-1 10.1128/aac.00595-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 2.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides uniformis Bacteroides uniformis Activity 0.0 % 10.1128/aac.00696-08
Bacteroides uniformis Bacteroides uniformis Activity 0.0 % 10.1128/aac.01128-07
Bacteroides uniformis Bacteroides uniformis Activity 0.5 % 10.1128/aac.01435-06
Bacteroides uniformis Bacteroides uniformis Activity 4.0 % 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis Activity 96.0 % 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis MIC 0.12 ug.mL-1 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis MIC 0.125 ug.mL-1 10.1128/aac.00595-08
Bacteroides uniformis Bacteroides uniformis MIC 0.125 ug.mL-1 10.1128/aac.00696-08
Bacteroides uniformis Bacteroides uniformis MIC 0.41 ug.mL-1 10.1128/aac.01435-06
Bacteroides uniformis Bacteroides uniformis MIC50 0.25 ug.mL-1 10.1128/aac.00595-08
Bacteroides uniformis Bacteroides uniformis MIC50 0.25 ug.mL-1 10.1128/aac.00696-08
Bacteroides uniformis Bacteroides uniformis MIC50 0.25 ug.mL-1 10.1128/aac.01128-07
Bacteroides uniformis Bacteroides uniformis MIC50 0.5 ug.mL-1 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis MIC90 0.5 ug.mL-1 10.1128/aac.00696-08
Bacteroides uniformis Bacteroides uniformis MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
Bacteroides uniformis Bacteroides uniformis MIC90 1.0 ug.mL-1 10.1128/aac.01435-06
Bacteroides uniformis Bacteroides uniformis MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis MIC90 4.0 ug.mL-1 10.1128/aac.00595-08
Bifidobacterium bifidum Bifidobacterium bifidum MIC 0.06 ug.mL-1 10.1128/aac.00595-08
Bifidobacterium breve Bifidobacterium breve MIC 1.0 ug.mL-1 10.1128/aac.00595-08
Bos taurus Progesterone receptor IC50 nan None None
Bos taurus Progesterone receptor Ki nan None None
Burkholderia cenocepacia PenB class A beta-lactamase Kcat 1.0 /s 10.1128/aac.00946-08
Burkholderia cenocepacia PenB class A beta-lactamase Kcat/Km 0.5 /uM/s 10.1128/aac.00946-08
Burkholderia cenocepacia PenB class A beta-lactamase Km 2500000.0 nM 10.1128/aac.00946-08
Burkholderia cepacia Burkholderia cepacia Activity 26.0 % 10.1128/aac.00954-06
Burkholderia cepacia Burkholderia cepacia Activity 48.0 % 10.1128/aac.00954-06
Burkholderia cepacia Burkholderia cepacia MIC 0.4 ug.mL-1 10.1016/j.ejmech.2006.10.006
Burkholderia cepacia Burkholderia cepacia MIC 0.4 ug.mL-1 10.1016/j.ejmech.2007.02.001
Burkholderia cepacia Burkholderia cepacia MIC50 8.0 ug.mL-1 10.1128/aac.00954-06
Burkholderia cepacia Burkholderia cepacia MIC90 32.0 ug.mL-1 10.1128/aac.00954-06
Burkholderia pseudomallei Burkholderia pseudomallei MIC50 1.0 ug.mL-1 10.1128/aac.00893-08
Burkholderia pseudomallei Burkholderia pseudomallei MIC50 3.0 ug.mL-1 10.1128/aac.00893-08
Burkholderia pseudomallei Burkholderia pseudomallei MIC90 2.0 ug.mL-1 10.1128/aac.00893-08
Burkholderia pseudomallei Burkholderia pseudomallei MIC90 4.0 ug.mL-1 10.1128/aac.00893-08
Burkholderia pseudomallei Burkholderia pseudomallei MIC90 4.0 ug.mL-1 10.1128/aac.01582-09
Campylobacter coli Campylobacter coli Activity 0.0 % 10.1128/aac.00898-09
Campylobacter coli Campylobacter coli MIC 0.015 ug.mL-1 10.1128/aac.01655-08
Campylobacter coli Campylobacter coli MIC 0.03 ug.mL-1 10.1128/aac.01655-08
Campylobacter coli Campylobacter coli MIC 0.06 ug.mL-1 10.1128/aac.01655-08
Campylobacter coli Campylobacter coli MIC 0.12 ug.mL-1 10.1128/aac.01655-08
Campylobacter coli Campylobacter coli MIC50 0.12 ug.mL-1 10.1128/aac.01655-08
Campylobacter coli Campylobacter coli MIC90 0.12 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni Activity 0.0 % 10.1128/aac.00898-09
Campylobacter jejuni Campylobacter jejuni MIC 0.008 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC 0.015 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC 0.03 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC 0.06 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC 0.08 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC 0.12 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC 0.25 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC 0.5 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC50 0.015 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC90 0.12 ug.mL-1 10.1128/aac.01655-08
Candida albicans Candida albicans IC50 300.0 nM 10.1021/acs.jnatprod.9b00187
Candida albicans Candida albicans Inhibition 3.42 % 10.6019/CHEMBL4513141
Capnocytophaga ochracea Capnocytophaga ochracea MIC 0.03 ug.mL-1 10.1128/aac.00595-08
Caulobacter vibrioides Metallo-beta-lactamase Kcat/Km 2.6 10'5/M/s 10.1128/aac.01062-07
Cavia porcellus Leukotriene C4 synthase IC50 nan None None
Cavia porcellus Leukotriene C4 synthase Ki nan None None
Cavia porcellus Serotonin 4 (5-HT4) receptor IC50 nan None None
Cavia porcellus Serotonin 4 (5-HT4) receptor Ki nan None None
Chryseobacterium indologenes Chryseobacterium indologenes Activity 16.0 ug ml-1 10.1128/aac.00083-07
Chryseobacterium indologenes Chryseobacterium indologenes MIC 8.0 ug.mL-1 10.1128/aac.01607-08
Chryseobacterium indologenes IND-like metallo-beta-lactamase Kcat/Km 1.5 10'4/M/s 10.1128/aac.01607-08
Chryseobacterium indologenes Metallo-beta-lactamase IND-2 Kcat/Km 1.8 10'5/M/s 10.1128/aac.01607-08
Chryseobacterium indologenes Metallo-beta-lactamase IND-6 Kcat 25.0 /s 10.1128/aac.01607-08
Chryseobacterium indologenes Metallo-beta-lactamase IND-6 Kcat/Km 1.7 10'5/M/s 10.1128/aac.01607-08
Chryseobacterium indologenes Metallo-beta-lactamase IND-6 Km 145000.0 nM 10.1128/aac.01607-08
Citrobacter Citrobacter Activity 0.0 % 10.1128/aac.00381-08
Citrobacter Citrobacter Activity 100.0 % 10.1128/aac.00381-08
Citrobacter Citrobacter MIC 0.015 ug.mL-1 10.1128/aac.00381-08
Citrobacter Citrobacter MIC 0.03 ug.mL-1 10.1128/aac.00381-08
Citrobacter Citrobacter MIC50 0.06 ug.mL-1 10.1128/aac.00381-08
Citrobacter Citrobacter MIC50 0.12 ug.mL-1 10.1128/aac.00381-08
Citrobacter Citrobacter MIC90 0.06 ug.mL-1 10.1128/aac.00381-08
Citrobacter Citrobacter MIC90 0.12 ug.mL-1 10.1128/aac.00381-08
Citrobacter Citrobacter MIC90 0.25 ug.mL-1 10.1128/aac.00381-08
Citrobacter freundii Citrobacter freundii MIC 0.015 ug.mL-1 10.1128/aac.00336-08
Citrobacter freundii Citrobacter freundii MIC 0.016 ug.mL-1 10.1128/aac.00830-08
Citrobacter freundii Citrobacter freundii MIC 0.025 ug.mL-1 10.1016/j.ejmech.2007.02.001
Citrobacter freundii Citrobacter freundii MIC 0.032 ug.mL-1 10.1128/aac.00830-08
Citrobacter freundii Citrobacter freundii MIC 0.06 ug.mL-1 10.1016/S0960-894X(97)00282-5
Citrobacter freundii Citrobacter freundii MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Citrobacter freundii Citrobacter freundii MIC 0.125 ug.mL-1 10.1128/aac.00830-08
Citrobacter freundii Citrobacter freundii MIC 0.25 ug.mL-1 10.1128/aac.00830-08
Citrobacter freundii Citrobacter freundii MIC 2.0 ug.mL-1 10.1128/aac.01099-09
Citrobacter freundii Citrobacter freundii MIC 4.0 ug.mL-1 10.1128/aac.01099-09
Citrobacter freundii Citrobacter freundii MIC 4.0 ug.mL-1 10.1128/aac.01337-07
Citrobacter freundii Citrobacter freundii MIC 8.0 ug.mL-1 10.1128/aac.01405-06
Citrobacter freundii Citrobacter freundii MIC 32.0 ug.mL-1 10.1128/aac.01305-10
Citrobacter freundii Citrobacter freundii MIC 32.0 ug.mL-1 10.1128/aac.01312-09
Citrobacter freundii Citrobacter freundii MIC50 0.03 ug.mL-1 10.1128/aac.00336-08
Citrobacter freundii Citrobacter freundii MIC50 0.06 ug.mL-1 10.1021/ml200012f
Citrobacter freundii Citrobacter freundii MIC50 0.06 ug.mL-1 10.1128/aac.01525-09
Citrobacter freundii Citrobacter freundii MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
Citrobacter freundii Citrobacter freundii MIC90 0.25 ug.mL-1 10.1021/ml200012f
Citrobacter freundii Citrobacter freundii MIC90 0.25 ug.mL-1 10.1128/aac.01525-09
Clostridioides difficile Clostridioides difficile Activity 0.0 % 10.1128/aac.00481-10
Clostridioides difficile Clostridioides difficile Activity 90.0 % 10.1128/aac.00910-07
Clostridioides difficile Clostridioides difficile Activity 99.0 % 10.1128/aac.00910-07
Clostridioides difficile Clostridioides difficile Activity 100.0 % 10.1128/aac.00481-10
Clostridioides difficile Clostridioides difficile Activity nan None 10.1128/aac.00696-08
Clostridioides difficile Clostridioides difficile Activity nan None 10.1128/aac.00910-07
Clostridioides difficile Clostridioides difficile MIC 0.25 ug.mL-1 10.1128/aac.00481-10
Clostridioides difficile Clostridioides difficile MIC 1.0 ug.mL-1 10.1128/aac.00476-08
Clostridioides difficile Clostridioides difficile MIC 1.0 ug.mL-1 10.1128/aac.00595-08
Clostridioides difficile Clostridioides difficile MIC 1.0 ug.mL-1 10.1128/aac.00696-08
Clostridioides difficile Clostridioides difficile MIC 1.0 ug.mL-1 10.1128/aac.00910-07
Clostridioides difficile Clostridioides difficile MIC 4.0 ug.mL-1 10.1128/aac.00595-08
Clostridioides difficile Clostridioides difficile MIC50 2.0 ug.mL-1 10.1128/aac.00476-08
Clostridioides difficile Clostridioides difficile MIC50 2.0 ug.mL-1 10.1128/aac.00481-10
Clostridioides difficile Clostridioides difficile MIC50 2.0 ug.mL-1 10.1128/aac.00595-08
Clostridioides difficile Clostridioides difficile MIC50 2.0 ug.mL-1 10.1128/aac.00910-07
Clostridioides difficile Clostridioides difficile MIC50 2.0 ug.mL-1 10.1128/aac.01623-06
Clostridioides difficile Clostridioides difficile MIC90 2.0 ug.mL-1 10.1128/aac.00476-08
Clostridioides difficile Clostridioides difficile MIC90 2.0 ug.mL-1 10.1128/aac.00481-10
Clostridioides difficile Clostridioides difficile MIC90 2.0 ug.mL-1 10.1128/aac.01623-06
Clostridioides difficile Clostridioides difficile MIC90 4.0 ug.mL-1 10.1128/aac.00595-08
Clostridioides difficile Clostridioides difficile MIC90 4.0 ug.mL-1 10.1128/aac.00910-07
Clostridium cadaveris Clostridium cadaveris Activity 0.0 % 10.1128/aac.01128-07
Clostridium cadaveris Clostridium cadaveris MIC 0.03 ug.mL-1 10.1128/aac.00910-07
Clostridium cadaveris Clostridium cadaveris MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Clostridium cadaveris Clostridium cadaveris MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
[Clostridium] innocuum [Clostridium] innocuum Activity 0.0 % 10.1128/aac.00696-08
[Clostridium] innocuum [Clostridium] innocuum Activity 0.0 % 10.1128/aac.01128-07
[Clostridium] innocuum [Clostridium] innocuum MIC 0.06 ug.mL-1 10.1128/aac.00696-08
[Clostridium] innocuum [Clostridium] innocuum MIC 1.0 ug.mL-1 10.1128/aac.00910-07
[Clostridium] innocuum [Clostridium] innocuum MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
[Clostridium] innocuum [Clostridium] innocuum MIC50 2.0 ug.mL-1 10.1128/aac.00696-08
[Clostridium] innocuum [Clostridium] innocuum MIC50 2.0 ug.mL-1 10.1128/aac.00910-07
[Clostridium] innocuum [Clostridium] innocuum MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
[Clostridium] innocuum [Clostridium] innocuum MIC90 2.0 ug.mL-1 10.1128/aac.00696-08
Clostridium malenominatum Clostridium malenominatum Activity 0.0 % 10.1128/aac.01128-07
Clostridium malenominatum Clostridium malenominatum MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Clostridium malenominatum Clostridium malenominatum MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
Clostridium paraputrificum Clostridium paraputrificum Activity 0.0 % 10.1128/aac.00355-08
Clostridium paraputrificum Clostridium paraputrificum Activity 0.0 % 10.1128/aac.00696-08
Clostridium paraputrificum Clostridium paraputrificum Activity 100.0 % 10.1128/aac.00355-08
Clostridium paraputrificum Clostridium paraputrificum MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Clostridium paraputrificum Clostridium paraputrificum MIC 0.06 ug.mL-1 10.1128/aac.00696-08
Clostridium paraputrificum Clostridium paraputrificum MIC 0.25 ug.mL-1 10.1128/aac.00910-07
Clostridium paraputrificum Clostridium paraputrificum MIC50 0.03 ug.mL-1 10.1128/aac.00355-08
Clostridium paraputrificum Clostridium paraputrificum MIC50 2.0 ug.mL-1 10.1128/aac.00696-08
Clostridium paraputrificum Clostridium paraputrificum MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Clostridium paraputrificum Clostridium paraputrificum MIC90 2.0 ug.mL-1 10.1128/aac.00696-08
Clostridium perfringens Clostridium perfringens Activity 0.0 % 10.1128/aac.00355-08
Clostridium perfringens Clostridium perfringens Activity 0.0 % 10.1128/aac.00481-10
Clostridium perfringens Clostridium perfringens Activity 0.0 % 10.1128/aac.00696-08
Clostridium perfringens Clostridium perfringens Activity 0.0 % 10.1128/aac.01128-07
Clostridium perfringens Clostridium perfringens Activity 90.0 % 10.1128/aac.00910-07
Clostridium perfringens Clostridium perfringens Activity 99.0 % 10.1128/aac.00910-07
Clostridium perfringens Clostridium perfringens Activity 100.0 % 10.1128/aac.00355-08
Clostridium perfringens Clostridium perfringens Activity 100.0 % 10.1128/aac.00481-10
Clostridium perfringens Clostridium perfringens MIC 0.008 ug.mL-1 10.1128/aac.00481-10
Clostridium perfringens Clostridium perfringens MIC 0.015 ug.mL-1 10.1128/aac.00595-08
Clostridium perfringens Clostridium perfringens MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Clostridium perfringens Clostridium perfringens MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Clostridium perfringens Clostridium perfringens MIC 0.03 ug.mL-1 10.1128/aac.00910-07
Clostridium perfringens Clostridium perfringens MIC 0.06 ug.mL-1 10.1128/aac.00696-08
Clostridium perfringens Clostridium perfringens MIC50 0.015 ug.mL-1 10.1128/aac.00481-10
Clostridium perfringens Clostridium perfringens MIC50 0.015 ug.mL-1 10.1128/aac.00595-08
Clostridium perfringens Clostridium perfringens MIC50 0.015 ug.mL-1 10.1128/aac.01128-07
Clostridium perfringens Clostridium perfringens MIC50 0.016 ug.mL-1 10.1128/aac.00910-07
Clostridium perfringens Clostridium perfringens MIC50 0.03 ug.mL-1 10.1128/aac.00355-08
Clostridium perfringens Clostridium perfringens MIC50 0.06 ug.mL-1 10.1128/aac.00696-08
Clostridium perfringens Clostridium perfringens MIC90 0.015 ug.mL-1 10.1128/aac.00481-10
Clostridium perfringens Clostridium perfringens MIC90 0.015 ug.mL-1 10.1128/aac.01128-07
Clostridium perfringens Clostridium perfringens MIC90 0.016 ug.mL-1 10.1128/aac.00910-07
Clostridium perfringens Clostridium perfringens MIC90 0.03 ug.mL-1 10.1128/aac.00595-08
Clostridium perfringens Clostridium perfringens MIC90 0.125 ug.mL-1 10.1128/aac.00696-08
Clostridium perfringens Clostridium perfringens MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Clostridium septicum Clostridium septicum Activity 0.0 % 10.1128/aac.00355-08
Clostridium septicum Clostridium septicum Activity 100.0 % 10.1128/aac.00355-08
Clostridium septicum Clostridium septicum MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Clostridium septicum Clostridium septicum MIC 0.06 ug.mL-1 10.1128/aac.00595-08
Clostridium septicum Clostridium septicum MIC50 0.03 ug.mL-1 10.1128/aac.00355-08
Clostridium septicum Clostridium septicum MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Clostridium tertium Clostridium tertium Activity 0.0 % 10.1128/aac.00355-08
Clostridium tertium Clostridium tertium Activity 0.0 % 10.1128/aac.00696-08
Clostridium tertium Clostridium tertium Activity 100.0 % 10.1128/aac.00355-08
Clostridium tertium Clostridium tertium MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Clostridium tertium Clostridium tertium MIC 0.06 ug.mL-1 10.1128/aac.00696-08
Clostridium tertium Clostridium tertium MIC50 0.03 ug.mL-1 10.1128/aac.00355-08
Clostridium tertium Clostridium tertium MIC50 2.0 ug.mL-1 10.1128/aac.00696-08
Clostridium tertium Clostridium tertium MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Clostridium tertium Clostridium tertium MIC90 2.0 ug.mL-1 10.1128/aac.00696-08
Corynebacterium accolens Corynebacterium accolens Activity 0.0 % 10.1128/aac.01128-07
Corynebacterium accolens Corynebacterium accolens MIC50 0.125 ug.mL-1 10.1128/aac.01128-07
Corynebacterium accolens Corynebacterium accolens MIC90 0.25 ug.mL-1 10.1128/aac.01128-07
Corynebacterium amycolatum Corynebacterium amycolatum Activity 7.0 % 10.1128/aac.01128-07
Corynebacterium amycolatum Corynebacterium amycolatum MIC50 1.0 ug.mL-1 10.1128/aac.01128-07
Corynebacterium amycolatum Corynebacterium amycolatum MIC50 16.0 ug.mL-1 10.1128/aac.01128-07
Corynebacterium aurimucosum Corynebacterium aurimucosum Activity 20.0 % 10.1128/aac.01128-07
Corynebacterium aurimucosum Corynebacterium aurimucosum MIC50 1.0 ug.mL-1 10.1128/aac.01128-07
Corynebacterium aurimucosum Corynebacterium aurimucosum MIC90 16.0 ug.mL-1 10.1128/aac.01128-07
Corynebacterium diphtheriae Corynebacterium diphtheriae MIC 0.02 ug.mL-1 10.1016/j.ejmech.2007.02.001
Corynebacterium diphtheriae Corynebacterium diphtheriae MIC 0.05 ug.mL-1 10.1016/j.ejmech.2006.10.006
Corynebacterium jeikeium Corynebacterium jeikeium Activity 20.0 % 10.1128/aac.01128-07
Corynebacterium jeikeium Corynebacterium jeikeium MIC50 1.0 ug.mL-1 10.1128/aac.01128-07
Corynebacterium jeikeium Corynebacterium jeikeium MIC90 16.0 ug.mL-1 10.1128/aac.01128-07
Corynebacterium minutissimum Corynebacterium minutissimum Activity 20.0 % 10.1128/aac.01128-07
Corynebacterium minutissimum Corynebacterium minutissimum MIC50 1.0 ug.mL-1 10.1128/aac.01128-07
Corynebacterium minutissimum Corynebacterium minutissimum MIC90 16.0 ug.mL-1 10.1128/aac.01128-07
Corynebacterium simulans Corynebacterium simulans Activity 0.0 % 10.1128/aac.01128-07
Corynebacterium simulans Corynebacterium simulans MIC50 0.125 ug.mL-1 10.1128/aac.01128-07
Corynebacterium simulans Corynebacterium simulans MIC90 0.25 ug.mL-1 10.1128/aac.01128-07
Corynebacterium striatum Corynebacterium striatum Activity 0.0 % 10.1128/aac.01128-07
Corynebacterium striatum Corynebacterium striatum MIC50 0.125 ug.mL-1 10.1128/aac.01128-07
Corynebacterium striatum Corynebacterium striatum MIC90 0.25 ug.mL-1 10.1128/aac.01128-07
Corynebacterium urealyticum Corynebacterium urealyticum Activity 20.0 % 10.1128/aac.01128-07
Corynebacterium urealyticum Corynebacterium urealyticum MIC50 1.0 ug.mL-1 10.1128/aac.01128-07
Corynebacterium urealyticum Corynebacterium urealyticum MIC90 16.0 ug.mL-1 10.1128/aac.01128-07
Corynebacterium xerosis Corynebacterium xerosis Activity 0.0 % 10.1128/aac.01128-07
Corynebacterium xerosis Corynebacterium xerosis MIC50 0.125 ug.mL-1 10.1128/aac.01128-07
Corynebacterium xerosis Corynebacterium xerosis MIC90 0.25 ug.mL-1 10.1128/aac.01128-07
Cronobacter sakazakii Cronobacter sakazakii MIC 0.0625 ug.mL-1 10.1016/j.ejmech.2022.114495
Cryptococcus neoformans Cryptococcus neoformans IC50 300.0 nM 10.1021/acs.jnatprod.9b00187
Cryptococcus neoformans Cryptococcus neoformans Inhibition 2.76 % 10.6019/CHEMBL4513141
Cutibacterium acnes Cutibacterium acnes Activity 0.0 % 10.1128/aac.00696-08
Cutibacterium acnes Cutibacterium acnes Activity 0.0 % 10.1128/aac.01128-07
Cutibacterium acnes Cutibacterium acnes MIC 0.06 ug.mL-1 10.1128/aac.00696-08
Cutibacterium acnes Cutibacterium acnes MIC 2.0 ug.mL-1 10.1128/aac.00595-08
Cutibacterium acnes Cutibacterium acnes MIC50 0.06 ug.mL-1 10.1128/aac.00696-08
Cutibacterium acnes Cutibacterium acnes MIC50 0.125 ug.mL-1 10.1128/aac.01128-07
Cutibacterium acnes Cutibacterium acnes MIC90 0.06 ug.mL-1 10.1128/aac.00696-08
Cutibacterium acnes Cutibacterium acnes MIC90 0.25 ug.mL-1 10.1128/aac.01128-07
Eggerthella lenta Eggerthella lenta Activity 8.0 % 10.1128/aac.00481-10
Eggerthella lenta Eggerthella lenta Activity 92.0 % 10.1128/aac.00481-10
Eggerthella lenta Eggerthella lenta MIC 0.008 ug.mL-1 10.1128/aac.00481-10
Eggerthella lenta Eggerthella lenta MIC 0.03 ug.mL-1 10.1128/aac.00595-08
Eggerthella lenta Eggerthella lenta MIC 1.0 ug.mL-1 10.1128/aac.00595-08
Eggerthella lenta Eggerthella lenta MIC50 0.125 ug.mL-1 10.1128/aac.00481-10
Eggerthella lenta Eggerthella lenta MIC50 0.5 ug.mL-1 10.1128/aac.00595-08
Eggerthella lenta Eggerthella lenta MIC90 1.0 ug.mL-1 10.1128/aac.00595-08
Eggerthella lenta Eggerthella lenta MIC90 2.0 ug.mL-1 10.1128/aac.00481-10
Elizabethkingia meningoseptica GOB-1 metallo-beta-lactamase Kcat/Km 5.3 10'6/M/s 10.1128/aac.01062-07
Enterobacter cloacae Beta-lactamase Activity 1.2e-05 % 10.1128/aac.01004-09
Enterobacter cloacae Beta-lactamase Activity 0.00042 % 10.1128/aac.01004-09
Enterobacter cloacae Beta-lactamase Kcat 0.00031 /s 10.1128/aac.01004-09
Enterobacter cloacae Beta-lactamase Kcat/Km 3.2e-05 /s/microM 10.1128/aac.01004-09
Enterobacter cloacae Beta-lactamase Km 9800.0 nM 10.1128/aac.01004-09
Enterobacter cloacae Enterobacter cloacae Activity 0.0 % 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae Activity 0.0 % 10.1128/aac.00400-09
Enterobacter cloacae Enterobacter cloacae Activity 0.0 % 10.1128/aac.01128-07
Enterobacter cloacae Enterobacter cloacae Activity 0.0 % 10.1128/aac.01538-07
Enterobacter cloacae Enterobacter cloacae Activity 0.4 % 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae Activity 0.5 % 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae Activity 7.0 ug ml-1 10.1128/aac.01525-09
Enterobacter cloacae Enterobacter cloacae Activity 9.0 ug ml-1 10.1128/aac.01525-09
Enterobacter cloacae Enterobacter cloacae Activity 99.5 % 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae Activity 99.6 % 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae Activity 100.0 % 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae Activity 100.0 % 10.1128/aac.00400-09
Enterobacter cloacae Enterobacter cloacae Activity nan None 10.1128/aac.01525-09
Enterobacter cloacae Enterobacter cloacae Inhibition nan % 10.1128/aac.01452-08
Enterobacter cloacae Enterobacter cloacae MBC 0.03 ug ml-1 10.1128/aac.01452-08
Enterobacter cloacae Enterobacter cloacae MBC 0.125 ug ml-1 10.1128/aac.01452-08
Enterobacter cloacae Enterobacter cloacae MBC 0.25 ug ml-1 10.1128/aac.01525-09
Enterobacter cloacae Enterobacter cloacae MBC 0.5 ug ml-1 10.1128/aac.01452-08
Enterobacter cloacae Enterobacter cloacae MBC 2.0 ug ml-1 10.1128/aac.01525-09
Enterobacter cloacae Enterobacter cloacae MIC 0.01 ug.mL-1 10.1016/j.ejmech.2006.10.006
Enterobacter cloacae Enterobacter cloacae MIC 0.01 ug.mL-1 10.1016/j.ejmech.2007.02.001
Enterobacter cloacae Enterobacter cloacae MIC 0.015 ug.mL-1 10.1128/aac.00336-08
Enterobacter cloacae Enterobacter cloacae MIC 0.015 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC 0.016 ug.mL-1 10.1128/aac.00830-08
Enterobacter cloacae Enterobacter cloacae MIC 0.025 ug.mL-1 10.1016/j.bmcl.2003.09.039
Enterobacter cloacae Enterobacter cloacae MIC 0.025 ug.mL-1 10.1016/j.bmcl.2004.09.092
Enterobacter cloacae Enterobacter cloacae MIC 0.025 ug.mL-1 10.1016/j.ejmech.2006.10.006
Enterobacter cloacae Enterobacter cloacae MIC 0.025 ug.mL-1 10.1016/j.ejmech.2007.02.001
Enterobacter cloacae Enterobacter cloacae MIC 0.025 ug.mL-1 10.1016/s0960-894x(00)00253-5
Enterobacter cloacae Enterobacter cloacae MIC 0.025 ug.mL-1 10.1016/s0960-894x(00)00575-8
Enterobacter cloacae Enterobacter cloacae MIC 0.025 ug.mL-1 10.1016/s0960-894x(01)00451-6
Enterobacter cloacae Enterobacter cloacae MIC 0.025 ug.mL-1 10.1016/s0960-894x(02)00948-4
Enterobacter cloacae Enterobacter cloacae MIC 0.025 ug.mL-1 10.1016/s0960-894x(99)00407-2
Enterobacter cloacae Enterobacter cloacae MIC 0.025 ug.mL-1 10.1016/s0960-894x(99)00646-0
Enterobacter cloacae Enterobacter cloacae MIC 0.025 ug.mL-1 10.1016/s0960-894x(99)00692-7
Enterobacter cloacae Enterobacter cloacae MIC 0.03 ug.mL-1 10.1016/j.bmcl.2003.09.039
Enterobacter cloacae Enterobacter cloacae MIC 0.03 ug.mL-1 10.1016/j.bmcl.2021.127928
Enterobacter cloacae Enterobacter cloacae MIC 0.03 ug.mL-1 10.1016/j.ejmech.2006.10.006
Enterobacter cloacae Enterobacter cloacae MIC 0.03 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC 0.03 ug.mL-1 10.1128/aac.01452-08
Enterobacter cloacae Enterobacter cloacae MIC 0.031 ug.mL-1 10.1016/j.bmc.2021.116343
Enterobacter cloacae Enterobacter cloacae MIC 0.032 ug.mL-1 10.1128/aac.00830-08
Enterobacter cloacae Enterobacter cloacae MIC 0.06 ug.mL-1 10.1016/j.bmcl.2021.127928
Enterobacter cloacae Enterobacter cloacae MIC 0.06 ug.mL-1 10.1016/S0960-894X(97)00282-5
Enterobacter cloacae Enterobacter cloacae MIC 0.06 ug.mL-1 10.1128/aac.00400-09
Enterobacter cloacae Enterobacter cloacae MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Enterobacter cloacae Enterobacter cloacae MIC 0.064 ug.mL-1 10.1128/aac.00830-08
Enterobacter cloacae Enterobacter cloacae MIC 0.125 ug.mL-1 10.1016/j.bmcl.2021.127928
Enterobacter cloacae Enterobacter cloacae MIC 0.125 ug.mL-1 10.1128/aac.00830-08
Enterobacter cloacae Enterobacter cloacae MIC 0.125 ug.mL-1 10.1128/aac.01099-09
Enterobacter cloacae Enterobacter cloacae MIC 0.125 ug.mL-1 10.1128/aac.01452-08
Enterobacter cloacae Enterobacter cloacae MIC 0.125 ug.mL-1 10.1128/aac.01525-09
Enterobacter cloacae Enterobacter cloacae MIC 0.25 ug.mL-1 10.1016/j.bmc.2013.09.041
Enterobacter cloacae Enterobacter cloacae MIC 0.25 ug.mL-1 10.1016/j.bmcl.2021.127928
Enterobacter cloacae Enterobacter cloacae MIC 0.25 ug.mL-1 10.1021/acs.jmedchem.9b01518
Enterobacter cloacae Enterobacter cloacae MIC 0.25 ug.mL-1 10.1128/aac.00830-08
Enterobacter cloacae Enterobacter cloacae MIC 0.25 ug.mL-1 10.1128/aac.01004-09
Enterobacter cloacae Enterobacter cloacae MIC 0.25 ug.mL-1 10.1128/aac.01452-08
Enterobacter cloacae Enterobacter cloacae MIC 0.5 ug.mL-1 10.1016/j.bmc.2013.09.041
Enterobacter cloacae Enterobacter cloacae MIC 0.5 ug.mL-1 10.1128/aac.01312-09
Enterobacter cloacae Enterobacter cloacae MIC 0.75 ug.mL-1 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae MIC 0.75 ug.mL-1 10.1128/aac.01312-09
Enterobacter cloacae Enterobacter cloacae MIC 1.0 ug.mL-1 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae MIC 1.0 ug.mL-1 10.1128/aac.00830-08
Enterobacter cloacae Enterobacter cloacae MIC 1.0 ug.mL-1 10.1128/aac.01525-09
Enterobacter cloacae Enterobacter cloacae MIC 2.0 ug.mL-1 10.1016/j.ejmech.2018.03.031
Enterobacter cloacae Enterobacter cloacae MIC 2.0 ug.mL-1 10.1128/aac.00707-08
Enterobacter cloacae Enterobacter cloacae MIC 2.0 ug.mL-1 10.1128/aac.01099-09
Enterobacter cloacae Enterobacter cloacae MIC 2.0 ug.mL-1 10.1128/aac.01341-07
Enterobacter cloacae Enterobacter cloacae MIC 4.0 ug.mL-1 10.1128/aac.00931-08
Enterobacter cloacae Enterobacter cloacae MIC 4.0 ug.mL-1 10.1128/aac.01099-09
Enterobacter cloacae Enterobacter cloacae MIC 4.0 ug.mL-1 10.1128/aac.01341-07
Enterobacter cloacae Enterobacter cloacae MIC 4.0 ug.mL-1 10.1128/aac.01525-09
Enterobacter cloacae Enterobacter cloacae MIC 6.0 ug.mL-1 10.1128/aac.01341-07
Enterobacter cloacae Enterobacter cloacae MIC 8.0 ug.mL-1 10.1021/acs.jmedchem.5b00127
Enterobacter cloacae Enterobacter cloacae MIC 8.0 ug.mL-1 10.1128/aac.01099-09
Enterobacter cloacae Enterobacter cloacae MIC 8.0 ug.mL-1 10.1128/aac.01341-07
Enterobacter cloacae Enterobacter cloacae MIC 16.0 ug.mL-1 10.1016/j.bmc.2021.116343
Enterobacter cloacae Enterobacter cloacae MIC 16.0 ug.mL-1 10.1128/aac.01099-09
Enterobacter cloacae Enterobacter cloacae MIC 24.0 ug.mL-1 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae MIC 24.0 ug.mL-1 10.1128/aac.01341-07
Enterobacter cloacae Enterobacter cloacae MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.03.031
Enterobacter cloacae Enterobacter cloacae MIC 32.0 ug.mL-1 10.1039/C5MD00380F
Enterobacter cloacae Enterobacter cloacae MIC 32.0 ug.mL-1 10.1128/aac.00033-09
Enterobacter cloacae Enterobacter cloacae MIC 32.0 ug.mL-1 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae MIC 32.0 ug.mL-1 10.1128/aac.00260-09
Enterobacter cloacae Enterobacter cloacae MIC 32.0 ug.mL-1 10.1128/aac.01341-07
Enterobacter cloacae Enterobacter cloacae MIC50 0.03 ug.mL-1 10.1128/aac.00336-08
Enterobacter cloacae Enterobacter cloacae MIC50 0.06 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC50 0.06 ug.mL-1 10.1128/aac.00400-09
Enterobacter cloacae Enterobacter cloacae MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Enterobacter cloacae Enterobacter cloacae MIC50 0.06 ug.mL-1 10.1128/aac.01525-09
Enterobacter cloacae Enterobacter cloacae MIC50 0.25 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC90 0.06 ug.mL-1 10.1128/aac.00400-09
Enterobacter cloacae Enterobacter cloacae MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
Enterobacter cloacae Enterobacter cloacae MIC90 0.12 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC90 0.13 ug.mL-1 10.1016/j.bmcl.2016.06.019
Enterobacter cloacae Enterobacter cloacae MIC90 0.25 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC90 0.25 ug.mL-1 10.1128/aac.01525-09
Enterobacter cloacae Enterobacter cloacae MIC90 0.5 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC90 0.5 ug.mL-1 10.1128/aac.01128-07
Enterobacter cloacae IMI-1 Kcat 10.0 /s 10.1128/aac.00491-07
Enterobacter cloacae IMI-1 Kcat/Km 380.0 /mM/s 10.1128/aac.00491-07
Enterobacter cloacae IMI-1 Km 26000.0 nM 10.1128/aac.00491-07
Enterobacteriaceae Enterobacteriaceae Activity 0.0 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 0.1 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 0.7 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 1.3 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 2.0 % 10.1128/aac.00044-07
Enterobacteriaceae Enterobacteriaceae Activity 6.0 % 10.1128/aac.00044-07
Enterobacteriaceae Enterobacteriaceae Activity 32.7 % 10.1128/aac.01114-07
Enterobacteriaceae Enterobacteriaceae Activity 50.0 % 10.1128/aac.01114-07
Enterobacteriaceae Enterobacteriaceae Activity 62.5 % 10.1128/aac.01450-09
Enterobacteriaceae Enterobacteriaceae Activity 77.9 % 10.1128/aac.01450-09
Enterobacteriaceae Enterobacteriaceae Activity 81.3 % 10.1128/aac.01450-09
Enterobacteriaceae Enterobacteriaceae Activity 85.0 % 10.1128/aac.01450-09
Enterobacteriaceae Enterobacteriaceae Activity 91.7 % 10.1128/aac.01450-09
Enterobacteriaceae Enterobacteriaceae Activity 98.0 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 99.6 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 99.8 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 100.0 % 10.1128/aac.01450-09
Enterobacteriaceae Enterobacteriaceae MIC 0.015 ug.mL-1 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae MIC 2.0 ug.mL-1 10.1016/j.ejmech.2018.06.054
Enterobacteriaceae Enterobacteriaceae MIC 2.0 ug.mL-1 10.1128/aac.01114-07
Enterobacteriaceae Enterobacteriaceae MIC 8.0 ug.mL-1 10.1016/j.ejmech.2018.06.054
Enterobacteriaceae Enterobacteriaceae MIC 16.0 ug.mL-1 10.1016/j.ejmech.2018.06.054
Enterobacteriaceae Enterobacteriaceae MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.06.054
Enterobacteriaceae Enterobacteriaceae MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.06.054
Enterobacteriaceae Enterobacteriaceae MIC nan None 10.1016/j.ejmech.2017.10.044
Enterobacteriaceae Enterobacteriaceae MIC50 0.03 ug.mL-1 10.1128/aac.01450-09
Enterobacteriaceae Enterobacteriaceae MIC50 0.06 ug.mL-1 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae MIC50 0.12 ug.mL-1 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae MIC50 8.0 ug.mL-1 10.1128/aac.01114-07
Enterobacteriaceae Enterobacteriaceae MIC90 0.12 ug.mL-1 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae MIC90 0.12 ug.mL-1 10.1128/aac.01450-09
Enterobacteriaceae Enterobacteriaceae MIC90 0.25 ug.mL-1 10.1128/aac.01450-09
Enterobacteriaceae Enterobacteriaceae MIC90 0.5 ug.mL-1 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae MIC90 8.0 ug.mL-1 10.1128/aac.01114-07
Enterobacteriaceae Enterobacteriaceae MIC90 32.0 ug.mL-1 10.1016/j.bmcl.2018.01.006
Enterobacter sp. Enterobacter sp. Activity 33.3 % 10.1128/aac.01114-07
Enterobacter sp. Enterobacter sp. Activity 41.7 % 10.1128/aac.01114-07
Enterobacter sp. Enterobacter sp. MIC50 8.0 ug.mL-1 10.1128/aac.01114-07
Enterobacter sp. Enterobacter sp. MIC90 8.0 ug.mL-1 10.1128/aac.01114-07
Enterocloster clostridioformis Enterocloster clostridioformis Activity 0.0 % 10.1128/aac.01128-07
Enterocloster clostridioformis Enterocloster clostridioformis MIC 0.25 ug.mL-1 10.1128/aac.00595-08
Enterocloster clostridioformis Enterocloster clostridioformis MIC 1.0 ug.mL-1 10.1128/aac.00910-07
Enterocloster clostridioformis Enterocloster clostridioformis MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Enterocloster clostridioformis Enterocloster clostridioformis MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
Enterococcus durans Enterococcus durans MIC 0.8 ug.mL-1 10.1016/j.ejmech.2006.10.006
Enterococcus durans Enterococcus durans MIC 0.8 ug.mL-1 10.1016/j.ejmech.2007.02.001
Enterococcus faecalis Enterococcus faecalis MIC 2.0 ug.mL-1 10.1016/S0960-894X(97)00282-5
Enterococcus faecalis Enterococcus faecalis MIC 2.0 ug.mL-1 10.1039/D1MD00230A
Enterococcus faecalis Enterococcus faecalis MIC 4.0 ug.mL-1 10.1016/j.ejmech.2018.06.054
Enterococcus faecalis Enterococcus faecalis MIC 4.0 ug.mL-1 10.1039/D1MD00230A
Enterococcus faecalis Enterococcus faecalis MIC 8.0 ug.mL-1 10.1039/D1MD00230A
Enterococcus faecalis Enterococcus faecalis MIC 12.5 ug.mL-1 10.1016/j.ejmech.2007.02.001
Enterococcus faecalis Enterococcus faecalis MIC 4000.0 nM 10.1021/acs.jmedchem.1c00614
Enterococcus faecalis Enterococcus faecalis MIC 16000.0 nM 10.1021/acs.jmedchem.1c02140
Enterococcus faecalis Enterococcus faecalis MIC nan None 10.1016/j.ejmech.2017.10.044
Enterococcus faecalis Enterococcus faecalis MIC nan None 10.1016/j.ejmech.2017.12.009
Enterococcus faecalis Enterococcus faecalis MIC nan None 10.1021/acs.jmedchem.2c01674
Enterococcus faecalis Enterococcus faecalis MIC90 4.0 ug.mL-1 10.1016/j.bmcl.2016.06.019
Enterococcus faecium Enterococcus faecium MIC 0.01 ug.mL-1 10.1016/j.ejmech.2006.10.006
Enterococcus faecium Enterococcus faecium MIC 0.01 ug.mL-1 10.1016/j.ejmech.2007.02.001
Enterococcus faecium Enterococcus faecium MIC 1.0 ug.mL-1 10.1074/jbc.m704286200
Enterococcus faecium Enterococcus faecium MIC 2.0 ug.mL-1 10.1016/j.ejmech.2021.113402
Enterococcus faecium Enterococcus faecium MIC 4.0 ug.mL-1 10.1016/j.ejmech.2021.113402
Enterococcus faecium Enterococcus faecium MIC 6.25 ug.mL-1 10.1016/s0960-894x(99)00692-7
Enterococcus faecium Enterococcus faecium MIC 6.25 ug.mL-1 10.1021/np049577a
Enterococcus faecium Enterococcus faecium MIC 8.0 ug.mL-1 10.1016/j.ejmech.2021.113402
Enterococcus faecium Enterococcus faecium MIC 8.0 ug.mL-1 10.1016/j.ejmech.2022.114495
Enterococcus faecium Enterococcus faecium MIC 8.0 ug.mL-1 10.1074/jbc.m704286200
Enterococcus faecium Enterococcus faecium MIC 12.5 ug.mL-1 10.1016/s0960-894x(98)00270-4
Enterococcus faecium Enterococcus faecium MIC 12.5 ug.mL-1 10.1016/s0960-894x(99)00407-2
Enterococcus faecium Enterococcus faecium MIC 128.0 ug.mL-1 10.1016/j.ejmech.2021.113402
Enterococcus faecium Enterococcus faecium MIC 128.0 ug.mL-1 10.1016/S0960-894X(97)00282-5
Enterococcus faecium Enterococcus faecium MIC 128.0 ug.mL-1 10.1039/D1MD00230A
Enterococcus faecium Enterococcus faecium MIC 256.0 ug.mL-1 10.1016/j.bmc.2021.116128
Enterococcus faecium Enterococcus faecium MIC nan None 10.1021/np800503z
Enterococcus sp. Enterococcus sp. Activity nan None 10.1128/aac.01538-07
Escherichia coli Beta-lactamase Activity 1.1e-05 % 10.1128/aac.01004-09
Escherichia coli Beta-lactamase Activity 0.058 % 10.1128/aac.01004-09
Escherichia coli Beta-lactamase Kcat 8.1e-05 /s 10.1128/aac.01004-09
Escherichia coli Beta-lactamase Kcat/Km 0.0014 /s/microM 10.1128/aac.01004-09
Escherichia coli Beta-lactamase Km 60.0 nM 10.1128/aac.01004-09
Escherichia coli Beta-lactamase CTX-M Activity 0.0022 % 10.1128/aac.01004-09
Escherichia coli Beta-lactamase CTX-M Activity 0.0078 % 10.1128/aac.01004-09
Escherichia coli Beta-lactamase CTX-M Kcat 0.0042 /s 10.1128/aac.01004-09
Escherichia coli Beta-lactamase CTX-M Kcat/Km 0.00038 /s/microM 10.1128/aac.01004-09
Escherichia coli Beta-lactamase CTX-M Km 11000.0 nM 10.1128/aac.01004-09
Escherichia coli Beta-lactamase TEM Activity 2.3e-05 % 10.1128/aac.01004-09
Escherichia coli Beta-lactamase TEM Activity 0.00083 % 10.1128/aac.01004-09
Escherichia coli Beta-lactamase TEM Kcat 0.00023 /s 10.1128/aac.01004-09
Escherichia coli Beta-lactamase TEM Kcat/Km 1.5e-05 /s/microM 10.1128/aac.01004-09
Escherichia coli Beta-lactamase TEM Km 15000.0 nM 10.1128/aac.01004-09
Escherichia coli BlaVIM-1 Kcat 13.0 /s 10.1128/aac.00017-09
Escherichia coli BlaVIM-1 Kcat 15.0 /s 10.1128/aac.00458-09
Escherichia coli BlaVIM-1 Kcat/Km 0.27 /s/microM 10.1128/aac.00017-09
Escherichia coli BlaVIM-1 Kcat/Km 0.3 /uM/s 10.1128/aac.00458-09
Escherichia coli BlaVIM-1 Km 50000.0 nM 10.1128/aac.00458-09
Escherichia coli Escherichia coli Activity -1.46 log10CFU/g 10.1021/acs.jmedchem.0c00579
Escherichia coli Escherichia coli Activity 0.0 % 10.1128/aac.00063-08
Escherichia coli Escherichia coli Activity 0.0 % 10.1128/aac.00381-08
Escherichia coli Escherichia coli Activity 0.0 % 10.1128/aac.00400-09
Escherichia coli Escherichia coli Activity 0.0 % 10.1128/aac.00551-10
Escherichia coli Escherichia coli Activity 0.0 % 10.1128/aac.01128-07
Escherichia coli Escherichia coli Activity 0.0 % 10.1128/aac.01412-06
Escherichia coli Escherichia coli Activity 0.0 % 10.1128/aac.01538-07
Escherichia coli Escherichia coli Activity 0.125 ug ml-1 10.1128/aac.00083-07
Escherichia coli Escherichia coli Activity 1.0 CFU/ml 10.1016/j.ejmech.2022.114495
Escherichia coli Escherichia coli Activity 1.0 ug ml-1 10.1128/aac.00083-07
Escherichia coli Escherichia coli Activity 95.0 % 10.1016/j.ejmech.2019.01.083
Escherichia coli Escherichia coli Activity 100.0 % 10.1128/aac.00381-08
Escherichia coli Escherichia coli Activity 100.0 % 10.1128/aac.00400-09
Escherichia coli Escherichia coli Activity 100.0 % 10.1128/aac.01176-07
Escherichia coli Escherichia coli Activity 100.0 % 10.1128/aac.01509-06
Escherichia coli Escherichia coli Activity nan None 10.1016/j.bmcl.2016.10.004
Escherichia coli Escherichia coli Activity nan None 10.1016/j.ejmech.2022.114278
Escherichia coli Escherichia coli Activity nan None 10.1016/j.ejmech.2022.114571
Escherichia coli Escherichia coli Activity nan None 10.1128/aac.00220-10
Escherichia coli Escherichia coli Activity nan None 10.1128/aac.01525-09
Escherichia coli Escherichia coli Activity nan None 10.1128/aac.01529-07
Escherichia coli Escherichia coli ED50 2.04 mg.kg-1 10.1021/acs.jmedchem.6b01261
Escherichia coli Escherichia coli ED50 nan mg.kg-1 10.1016/S0960-894X(97)00282-5
Escherichia coli Escherichia coli fT>MIC 70.0 % 10.1128/aac.00752-06
Escherichia coli Escherichia coli fT>MIC 85.0 % 10.1128/aac.00752-06
Escherichia coli Escherichia coli fT>MIC 90.0 % 10.1128/aac.00752-06
Escherichia coli Escherichia coli fT>MIC 93.0 % 10.1128/aac.00752-06
Escherichia coli Escherichia coli IC50 0.03 ug.mL-1 10.1128/aac.01433-08
Escherichia coli Escherichia coli IC50 10.0 nM 10.1021/acs.jnatprod.9b00187
Escherichia coli Escherichia coli Inhibition 7.87 % 10.6019/CHEMBL4513141
Escherichia coli Escherichia coli Inhibition nan % 10.1128/aac.01452-08
Escherichia coli Escherichia coli MBC 0.03 ug ml-1 10.1128/aac.01433-08
Escherichia coli Escherichia coli MBC 0.06 ug ml-1 10.1128/aac.01452-08
Escherichia coli Escherichia coli MBC 2.0 ug ml-1 10.1021/acs.jmedchem.2c01469
Escherichia coli Escherichia coli MIC 0.0 ug.mL-1 10.1128/aac.01585-09
Escherichia coli Escherichia coli MIC 1e-05 ug.mL-1 10.1016/j.ejmech.2022.114108
Escherichia coli Escherichia coli MIC 6e-05 ug.mL-1 10.1128/aac.00294-06
Escherichia coli Escherichia coli MIC 0.002 ug.mL-1 10.1128/aac.01451-07
Escherichia coli Escherichia coli MIC 0.004 ug.mL-1 10.1128/aac.01337-07
Escherichia coli Escherichia coli MIC 0.008 ug.mL-1 10.1016/j.bmc.2021.116142
Escherichia coli Escherichia coli MIC 0.008 ug.mL-1 10.1016/j.ejmech.2021.113975
Escherichia coli Escherichia coli MIC 0.008 ug.mL-1 10.1128/aac.00485-08
Escherichia coli Escherichia coli MIC 0.008 ug.mL-1 10.1128/aac.00771-10
Escherichia coli Escherichia coli MIC 0.01 ug.mL-1 10.1016/j.ejmech.2006.10.006
Escherichia coli Escherichia coli MIC 0.01 ug.mL-1 10.1016/j.ejmech.2007.02.001
Escherichia coli Escherichia coli MIC 0.01 ug.mL-1 10.1016/j.ejmech.2022.114108
Escherichia coli Escherichia coli MIC 0.01 ug.mL-1 10.1128/aac.01451-07
Escherichia coli Escherichia coli MIC 0.012 ug.mL-1 10.1128/aac.00598-10
Escherichia coli Escherichia coli MIC 0.012 ug.mL-1 10.1128/aac.01818-09
Escherichia coli Escherichia coli MIC 0.013 ug.mL-1 10.1016/s0960-894x(99)00407-2
Escherichia coli Escherichia coli MIC 0.013 ug.mL-1 10.1016/s0960-894x(99)00692-7
Escherichia coli Escherichia coli MIC 0.013 ug.mL-1 10.1021/np060206z
Escherichia coli Escherichia coli MIC 0.015 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 0.015 ug.mL-1 10.1128/aac.00336-08
Escherichia coli Escherichia coli MIC 0.015 ug.mL-1 10.1128/aac.00381-08
Escherichia coli Escherichia coli MIC 0.015 ug.mL-1 10.1128/aac.00768-10
Escherichia coli Escherichia coli MIC 0.015 ug.mL-1 10.1128/aac.00858-10
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1016/j.bmcl.2003.09.039
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1016/j.ejmech.2022.114108
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1128/aac.00033-10
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1128/aac.00072-09
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1128/aac.00175-08
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1128/aac.00458-09
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1128/aac.00461-09
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1128/aac.00684-07
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1128/aac.00771-10
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1128/aac.00830-08
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1128/aac.01341-07
Escherichia coli Escherichia coli MIC 0.02 ug.mL-1 10.1016/j.ejmech.2007.02.001
Escherichia coli Escherichia coli MIC 0.02133 ug.mL-1 10.1016/j.ejmech.2022.114108
Escherichia coli Escherichia coli MIC 0.023 ug.mL-1 10.1128/aac.00050-10
Escherichia coli Escherichia coli MIC 0.023 ug.mL-1 10.1128/aac.00374-07
Escherichia coli Escherichia coli MIC 0.023 ug.mL-1 10.1128/aac.00485-08
Escherichia coli Escherichia coli MIC 0.023 ug.mL-1 10.1128/aac.00771-10
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/0960-894X(95)00380-C
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/j.bmcl.2003.09.039
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/j.bmcl.2004.09.092
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/j.ejmech.2006.10.006
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/s0960-894x(00)00253-5
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/s0960-894x(00)00575-8
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/s0960-894x(01)00451-6
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/s0960-894x(02)00948-4
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/S0960-894X(97)00230-8
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/s0960-894x(98)00270-4
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/s0960-894x(99)00407-2
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/s0960-894x(99)00646-0
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1016/s0960-894x(99)00692-7
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1021/np049577a
Escherichia coli Escherichia coli MIC 0.025 ug.mL-1 10.1128/aac.00780-06
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1016/j.bmcl.2003.09.039
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1016/j.bmcl.2021.127928
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1016/j.ejmech.2006.10.006
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1021/acs.jmedchem.6b00746
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1021/acs.jmedchem.9b01518
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1021/np800503z
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.00033-09
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.00033-10
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.00175-08
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.00461-09
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.00543-08
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.00752-06
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.00768-10
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.01004-09
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.01025-07
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.01062-07
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.01099-09
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.01180-07
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.01336-09
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.01433-08
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.01452-08
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.01529-07
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.01585-09
Escherichia coli Escherichia coli MIC 0.03 ug.mL-1 10.1128/aac.01607-08
Escherichia coli Escherichia coli MIC 0.031 ug.mL-1 10.1016/j.bmc.2021.116343
Escherichia coli Escherichia coli MIC 0.031 ug.mL-1 10.1016/j.ejmech.2022.114174
Escherichia coli Escherichia coli MIC 0.032 ug.mL-1 10.1128/aac.00050-10
Escherichia coli Escherichia coli MIC 0.032 ug.mL-1 10.1128/aac.00374-07
Escherichia coli Escherichia coli MIC 0.032 ug.mL-1 10.1128/aac.00436-09
Escherichia coli Escherichia coli MIC 0.032 ug.mL-1 10.1128/aac.00485-08
Escherichia coli Escherichia coli MIC 0.032 ug.mL-1 10.1128/aac.00598-10
Escherichia coli Escherichia coli MIC 0.032 ug.mL-1 10.1128/aac.00684-07
Escherichia coli Escherichia coli MIC 0.032 ug.mL-1 10.1128/aac.00752-06
Escherichia coli Escherichia coli MIC 0.032 ug.mL-1 10.1128/aac.00771-10
Escherichia coli Escherichia coli MIC 0.032 ug.mL-1 10.1128/aac.00830-08
Escherichia coli Escherichia coli MIC 0.032 ug.mL-1 10.1128/aac.01011-08
Escherichia coli Escherichia coli MIC 0.032 ug.mL-1 10.1128/aac.01099-09
Escherichia coli Escherichia coli MIC 0.032 ug.mL-1 10.1128/aac.01762-09
Escherichia coli Escherichia coli MIC 0.03733 ug.mL-1 10.1016/j.ejmech.2022.114108
Escherichia coli Escherichia coli MIC 0.0375 ug.mL-1 10.1039/c9md00455f
Escherichia coli Escherichia coli MIC 0.04 ug.mL-1 10.1021/jm010546b
Escherichia coli Escherichia coli MIC 0.047 ug.mL-1 10.1128/aac.00072-09
Escherichia coli Escherichia coli MIC 0.047 ug.mL-1 10.1128/aac.00158-08
Escherichia coli Escherichia coli MIC 0.047 ug.mL-1 10.1128/aac.00436-09
Escherichia coli Escherichia coli MIC 0.047 ug.mL-1 10.1128/aac.00752-06
Escherichia coli Escherichia coli MIC 0.047 ug.mL-1 10.1128/aac.00771-10
Escherichia coli Escherichia coli MIC 0.047 ug.mL-1 10.1128/aac.01304-07
Escherichia coli Escherichia coli MIC 0.049 ug.mL-1 10.1016/j.ejmech.2007.02.001
Escherichia coli Escherichia coli MIC 0.05 ug.mL-1 10.1016/j.bmc.2016.02.013
Escherichia coli Escherichia coli MIC 0.05 ug.mL-1 10.1016/j.ejmech.2006.10.006
Escherichia coli Escherichia coli MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1016/j.bmcl.2021.127928
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1016/j.bmcl.2021.127956
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1016/S0960-894X(97)00282-5
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1021/acs.jmedchem.9b01518
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.00033-09
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.00033-10
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.00400-09
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.00688-09
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.00734-08
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.00858-10
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.00878-10
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.01004-09
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.01025-07
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.01053-06
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.01062-07
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.01433-08
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.01452-08
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.01561-09
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1128/aac.01585-09
Escherichia coli Escherichia coli MIC 0.0625 ug.mL-1 10.1016/j.ejmech.2022.114495
Escherichia coli Escherichia coli MIC 0.063 ug.mL-1 10.1016/j.ejmech.2018.06.014
Escherichia coli Escherichia coli MIC 0.064 ug.mL-1 10.1128/aac.00465-08
Escherichia coli Escherichia coli MIC 0.064 ug.mL-1 10.1128/aac.00774-09
Escherichia coli Escherichia coli MIC 0.064 ug.mL-1 10.1128/aac.01011-08
Escherichia coli Escherichia coli MIC 0.064 ug.mL-1 10.1128/aac.01099-09
Escherichia coli Escherichia coli MIC 0.064 ug.mL-1 10.1128/aac.01762-09
Escherichia coli Escherichia coli MIC 0.094 ug.mL-1 10.1128/aac.00137-10
Escherichia coli Escherichia coli MIC 0.094 ug.mL-1 10.1128/aac.00752-06
Escherichia coli Escherichia coli MIC 0.094 ug.mL-1 10.1128/aac.00771-10
Escherichia coli Escherichia coli MIC 0.094 ug.mL-1 10.1128/aac.01304-07
Escherichia coli Escherichia coli MIC 0.094 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 0.1 ug.mL-1 10.1128/aac.01451-07
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1016/j.bmc.2013.09.041
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1128/aac.00017-09
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1128/aac.00856-09
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1128/aac.00961-09
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1128/aac.00978-07
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1128/aac.01176-07
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1128/aac.01247-10
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1128/aac.01433-08
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1128/aac.01451-07
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1128/aac.01586-08
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1128/aac.01607-08
Escherichia coli Escherichia coli MIC 0.12 ug.mL-1 10.1128/aac.01672-07
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1016/j.ejmech.2007.03.023
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1016/j.ejmech.2017.10.044
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1016/j.ejmech.2017.12.009
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1016/j.ejmech.2018.03.058
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1016/j.ejmech.2018.06.054
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1016/j.ejmech.2019.02.024
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1016/j.ejmech.2022.114495
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1021/acs.jmedchem.2c01674
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1021/acs.jmedchem.6b01261
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1128/aac.00752-06
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1128/aac.01011-08
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1128/aac.01025-07
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1128/aac.01525-09
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1128/aac.01539-07
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1128/aac.01762-09
Escherichia coli Escherichia coli MIC 0.19 ug.mL-1 10.1128/aac.00465-08
Escherichia coli Escherichia coli MIC 0.19 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00033-09
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00072-09
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00158-08
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00299-07
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00374-07
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00393-08
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00458-09
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00465-08
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00736-08
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00961-09
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.01359-09
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.01451-07
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.01525-09
Escherichia coli Escherichia coli MIC 0.38 ug.mL-1 10.1128/aac.00158-08
Escherichia coli Escherichia coli MIC 0.38 ug.mL-1 10.1128/aac.01180-07
Escherichia coli Escherichia coli MIC 0.38 ug.mL-1 10.1128/aac.01451-07
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1016/j.ejmech.2019.02.024
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00033-10
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00227-08
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00458-09
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00543-08
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00736-08
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.01336-09
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.01359-09
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.01762-09
Escherichia coli Escherichia coli MIC 0.625 ug.mL-1 10.1016/j.bmcl.2021.128192
Escherichia coli Escherichia coli MIC 0.75 ug.mL-1 10.1128/aac.00436-09
Escherichia coli Escherichia coli MIC 0.75 ug.mL-1 10.1128/aac.00752-06
Escherichia coli Escherichia coli MIC 0.75 ug.mL-1 10.1128/aac.01762-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1016/j.bmc.2013.09.041
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1016/j.ejmech.2018.03.058
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1016/j.ejmech.2022.114278
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1021/acs.jmedchem.2c01469
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1021/acsmedchemlett.7b00428
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00017-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00033-10
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00158-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00458-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00734-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00899-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01359-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01433-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01462-06
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01672-07
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01762-09
Escherichia coli Escherichia coli MIC 1.5 ug.mL-1 10.1128/aac.01247-10
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1016/j.ejmech.2018.03.031
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00137-10
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00734-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00856-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00858-10
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00896-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01341-07
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01359-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01433-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01451-07
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01539-07
Escherichia coli Escherichia coli MIC 3.0 ug.mL-1 10.1128/aac.00878-10
Escherichia coli Escherichia coli MIC 3.0 ug.mL-1 10.1128/aac.01341-07
Escherichia coli Escherichia coli MIC 3.0 ug.mL-1 10.1128/aac.01451-07
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1016/j.ejmech.2018.03.031
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1021/acs.jmedchem.5b00127
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00072-09
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00158-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00458-09
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01053-06
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01337-07
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01359-09
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01433-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01762-09
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1016/j.ejmech.2018.03.058
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1021/acs.jmedchem.8b00091
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00017-09
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00734-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.01099-09
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.01359-09
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.01762-09
Escherichia coli Escherichia coli MIC 12.0 ug.mL-1 10.1128/aac.00774-09
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1016/j.bmcl.2021.127956
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1016/j.ejmech.2022.114278
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.8b00091
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1039/C5MD00380F
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00017-09
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00878-10
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.01099-09
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.01359-09
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.01525-09
Escherichia coli Escherichia coli MIC 24.0 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1021/acs.jmedchem.9b00720
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.00774-09
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.01525-09
Escherichia coli Escherichia coli MIC 60.0 nM 10.1021/acs.jmedchem.1c00621
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/j.bmc.2021.116128
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/j.bmcl.2021.127956
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/j.ejmech.2022.114599
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1021/acs.jmedchem.2c01257
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1016/j.bmc.2021.116128
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1021/acs.jmedchem.2c01469
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1021/acs.jmedchem.9b00338
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1021/acsmedchemlett.7b00428
Escherichia coli Escherichia coli MIC 250.0 nM 10.1021/acs.jmedchem.1c00621
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01462-06
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.01462-06
Escherichia coli Escherichia coli MIC 1000.0 nM 10.1021/acs.jmedchem.1c00614
Escherichia coli Escherichia coli MIC 1000.0 nM 10.1021/acs.jmedchem.1c02140
Escherichia coli Escherichia coli MIC 4000.0 nM 10.1021/acs.jmedchem.1c00621
Escherichia coli Escherichia coli MIC nan None 10.1021/np800503z
Escherichia coli Escherichia coli MIC nan None 10.1128/aac.01512-06
Escherichia coli Escherichia coli MIC50 0.015 ug.mL-1 10.1128/aac.00336-08
Escherichia coli Escherichia coli MIC50 0.03 ug.mL-1 10.1021/jm400560z
Escherichia coli Escherichia coli MIC50 0.03 ug.mL-1 10.1128/aac.00381-08
Escherichia coli Escherichia coli MIC50 0.03 ug.mL-1 10.1128/aac.01128-07
Escherichia coli Escherichia coli MIC50 0.03 ug.mL-1 10.1128/aac.01509-06
Escherichia coli Escherichia coli MIC50 0.047 ug.mL-1 10.1128/aac.00171-08
Escherichia coli Escherichia coli MIC50 0.06 ug.mL-1 10.1021/ml200012f
Escherichia coli Escherichia coli MIC50 0.06 ug.mL-1 10.1128/aac.00381-08
Escherichia coli Escherichia coli MIC50 0.06 ug.mL-1 10.1128/aac.00400-09
Escherichia coli Escherichia coli MIC50 0.06 ug.mL-1 10.1128/aac.01525-09
Escherichia coli Escherichia coli MIC50 0.12 ug.mL-1 10.1128/aac.01176-07
Escherichia coli Escherichia coli MIC50 0.5 ug.mL-1 10.1021/acs.jmedchem.9b00338
Escherichia coli Escherichia coli MIC50 1.0 ug.mL-1 10.1021/acs.jmedchem.0c00255
Escherichia coli Escherichia coli MIC50 1.0 ug.mL-1 10.1128/aac.01412-06
Escherichia coli Escherichia coli MIC90 0.03 ug.mL-1 10.1128/aac.01128-07
Escherichia coli Escherichia coli MIC90 0.06 ug.mL-1 10.1016/j.bmcl.2012.07.005
Escherichia coli Escherichia coli MIC90 0.06 ug.mL-1 10.1021/jm400560z
Escherichia coli Escherichia coli MIC90 0.06 ug.mL-1 10.1021/ml200012f
Escherichia coli Escherichia coli MIC90 0.06 ug.mL-1 10.1128/aac.00381-08
Escherichia coli Escherichia coli MIC90 0.06 ug.mL-1 10.1128/aac.00400-09
Escherichia coli Escherichia coli MIC90 0.064 ug.mL-1 10.1128/aac.00171-08
Escherichia coli Escherichia coli MIC90 0.094 ug.mL-1 10.1128/aac.00171-08
Escherichia coli Escherichia coli MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
Escherichia coli Escherichia coli MIC90 0.12 ug.mL-1 10.1128/aac.01176-07
Escherichia coli Escherichia coli MIC90 0.125 ug.mL-1 10.1128/aac.00171-08
Escherichia coli Escherichia coli MIC90 0.19 ug.mL-1 10.1128/aac.00171-08
Escherichia coli Escherichia coli MIC90 0.25 ug.mL-1 10.1128/aac.01509-06
Escherichia coli Escherichia coli MIC90 0.5 ug.mL-1 10.1128/aac.01525-09
Escherichia coli Escherichia coli MIC90 1.0 ug.mL-1 10.1128/aac.01412-06
Escherichia coli Escherichia coli MIC90 8.0 ug.mL-1 10.1021/acs.jmedchem.0c00255
Escherichia coli Escherichia coli MIC90 32.0 ug.mL-1 10.1021/acs.jmedchem.9b00338
Escherichia coli Escherichia coli MPC 0.03 ug ml-1 10.1128/aac.00033-10
Escherichia coli Escherichia coli MPC 0.06 ug ml-1 10.1128/aac.00033-10
Escherichia coli Escherichia coli MPC 0.125 ug ml-1 10.1128/aac.00033-10
Escherichia coli Escherichia coli MPC 0.25 ug ml-1 10.1128/aac.00033-10
Escherichia coli Escherichia coli MPC 1.0 ug ml-1 10.1128/aac.00033-10
Escherichia coli Escherichia coli MPC 4.0 ug ml-1 10.1128/aac.00033-10
Escherichia coli Escherichia coli MPC 16.0 ug ml-1 10.1128/aac.00033-10
Escherichia coli Escherichia coli PD50 1.24 mg kg-1 10.1016/s0960-894x(98)00270-4
Escherichia coli Escherichia coli Ratio 2.0 None 10.1128/aac.00033-10
Escherichia coli Escherichia coli Ratio 4.0 None 10.1128/aac.00033-10
Escherichia coli Escherichia coli Ratio 8.0 None 10.1128/aac.00033-10
Escherichia coli Escherichia coli Ratio 16.0 None 10.1128/aac.00033-10
Escherichia coli Escherichia coli Ratio 16.0 None 10.1128/aac.00734-08
Escherichia coli Escherichia coli Survival 44.0 % 10.1039/C5MD00380F
Escherichia coli Metallo-beta-lactamase Kcat 1.4 /s 10.1128/aac.00017-09
Escherichia coli Metallo-beta-lactamase Kcat 5.0 /s 10.1128/aac.01336-09
Escherichia coli Metallo-beta-lactamase Kcat 35.0 /s 10.1128/aac.01336-09
Escherichia coli Metallo-beta-lactamase Kcat 45.0 /s 10.1128/aac.01336-09
Escherichia coli Metallo-beta-lactamase Kcat/Km 0.28 /s/microM 10.1128/aac.00017-09
Escherichia coli Metallo-beta-lactamase Kcat/Km 1.9 /uM/s 10.1128/aac.01336-09
Escherichia coli Metallo-beta-lactamase Kcat/Km 2.5 uM/hr 10.1128/aac.01336-09
Escherichia coli Metallo-beta-lactamase Kcat/Km 2.5 /uM/s 10.1128/aac.01336-09
Escherichia coli Metallo-beta-lactamase Kcat/Km 4.5 /uM/s 10.1128/aac.01336-09
Escherichia coli Metallo-beta-lactamase Km 2000.0 nM 10.1128/aac.01336-09
Escherichia coli Metallo-beta-lactamase Km 10000.0 nM 10.1128/aac.01336-09
Escherichia coli Metallo-beta-lactamase Km 18000.0 nM 10.1128/aac.01336-09
Escherichia coli Metallo-beta-lactamase MIC 64.0 ug.mL-1 10.1016/j.bmc.2021.116128
Escherichia coli Metallo-beta-lactamase VIM-19 Kcat 25.0 /s 10.1128/aac.00458-09
Escherichia coli Metallo-beta-lactamase VIM-19 Kcat/Km 2.0 /uM/s 10.1128/aac.00458-09
Escherichia coli Metallo-beta-lactamase VIM-19 Km 15000.0 nM 10.1128/aac.00458-09
Eubacterium limosum Eubacterium limosum MIC 0.03 ug.mL-1 10.1128/aac.00595-08
Eubacterium limosum Eubacterium limosum MIC50 0.5 ug.mL-1 10.1128/aac.00595-08
Eubacterium limosum Eubacterium limosum MIC90 1.0 ug.mL-1 10.1128/aac.00595-08
Eubacterium sp. Eubacterium sp. Activity 8.0 % 10.1128/aac.00481-10
Eubacterium sp. Eubacterium sp. Activity 92.0 % 10.1128/aac.00481-10
Eubacterium sp. Eubacterium sp. MIC 0.008 ug.mL-1 10.1128/aac.00481-10
Eubacterium sp. Eubacterium sp. MIC50 0.125 ug.mL-1 10.1128/aac.00481-10
Eubacterium sp. Eubacterium sp. MIC90 2.0 ug.mL-1 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna Activity 0.0 % 10.1128/aac.00355-08
Finegoldia magna Finegoldia magna Activity 0.0 % 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna Activity 0.0 % 10.1128/aac.00696-08
Finegoldia magna Finegoldia magna Activity 0.0 % 10.1128/aac.01128-07
Finegoldia magna Finegoldia magna Activity 90.0 % 10.1128/aac.00910-07
Finegoldia magna Finegoldia magna Activity 99.0 % 10.1128/aac.00910-07
Finegoldia magna Finegoldia magna Activity 100.0 % 10.1128/aac.00355-08
Finegoldia magna Finegoldia magna Activity 100.0 % 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna Activity nan None 10.1128/aac.00910-07
Finegoldia magna Finegoldia magna MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Finegoldia magna Finegoldia magna MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna MIC 0.06 ug.mL-1 10.1128/aac.00696-08
Finegoldia magna Finegoldia magna MIC 0.06 ug.mL-1 10.1128/aac.00910-07
Finegoldia magna Finegoldia magna MIC50 0.06 ug.mL-1 10.1128/aac.00355-08
Finegoldia magna Finegoldia magna MIC50 0.06 ug.mL-1 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna MIC50 0.06 ug.mL-1 10.1128/aac.00910-07
Finegoldia magna Finegoldia magna MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Finegoldia magna Finegoldia magna MIC50 0.125 ug.mL-1 10.1128/aac.00595-08
Finegoldia magna Finegoldia magna MIC50 0.125 ug.mL-1 10.1128/aac.00696-08
Finegoldia magna Finegoldia magna MIC90 0.125 ug.mL-1 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna MIC90 0.125 ug.mL-1 10.1128/aac.00595-08
Finegoldia magna Finegoldia magna MIC90 0.125 ug.mL-1 10.1128/aac.00696-08
Finegoldia magna Finegoldia magna MIC90 0.125 ug.mL-1 10.1128/aac.00910-07
Finegoldia magna Finegoldia magna MIC90 0.125 ug.mL-1 10.1128/aac.01128-07
Finegoldia magna Finegoldia magna MIC90 0.5 ug.mL-1 10.1128/aac.00355-08
Flavobacterium meningosepticum Carbapenem-hydrolyzing beta-lactamase BlaB-1 Kcat/Km 7.6 10'5/M/s 10.1128/aac.01607-08
Fluoribacter gormanii FEZ-1 protein Kcat/Km 5.0 10'5/M/s 10.1128/aac.01062-07
Fusobacterium mortiferum Fusobacterium mortiferum Activity 8.0 % 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum Activity 92.0 % 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC 0.008 ug.mL-1 10.1128/aac.00481-10
Fusobacterium mortiferum Fusobacterium mortiferum MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC 0.06 ug.mL-1 10.1128/aac.00910-07
Fusobacterium mortiferum Fusobacterium mortiferum MIC50 0.03 ug.mL-1 10.1128/aac.00595-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC50 0.06 ug.mL-1 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC50 0.125 ug.mL-1 10.1128/aac.00910-07
Fusobacterium mortiferum Fusobacterium mortiferum MIC90 0.12 ug.mL-1 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC90 0.125 ug.mL-1 10.1128/aac.00595-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC90 0.5 ug.mL-1 10.1128/aac.00910-07
Fusobacterium necrophorum Fusobacterium necrophorum Activity 8.0 % 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum Activity 92.0 % 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC 0.015 ug.mL-1 10.1128/aac.00595-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Fusobacterium necrophorum Fusobacterium necrophorum MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC50 0.016 ug.mL-1 10.1128/aac.00910-07
Fusobacterium necrophorum Fusobacterium necrophorum MIC50 0.03 ug.mL-1 10.1128/aac.00595-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC50 0.06 ug.mL-1 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC90 0.12 ug.mL-1 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC90 0.125 ug.mL-1 10.1128/aac.00595-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC90 0.125 ug.mL-1 10.1128/aac.00910-07
Fusobacterium nucleatum Fusobacterium nucleatum Activity 8.0 % 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum Activity 90.0 % 10.1128/aac.00910-07
Fusobacterium nucleatum Fusobacterium nucleatum Activity 92.0 % 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum Activity 99.0 % 10.1128/aac.00910-07
Fusobacterium nucleatum Fusobacterium nucleatum MIC 0.008 ug.mL-1 10.1128/aac.00481-10
Fusobacterium nucleatum Fusobacterium nucleatum MIC 0.008 ug.mL-1 10.1128/aac.00910-07
Fusobacterium nucleatum Fusobacterium nucleatum MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Fusobacterium nucleatum Fusobacterium nucleatum MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC 8.0 ug.mL-1 10.1128/aac.00595-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC50 0.016 ug.mL-1 10.1128/aac.00910-07
Fusobacterium nucleatum Fusobacterium nucleatum MIC50 0.03 ug.mL-1 10.1128/aac.00595-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC50 0.06 ug.mL-1 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC90 0.03 ug.mL-1 10.1128/aac.00910-07
Fusobacterium nucleatum Fusobacterium nucleatum MIC90 0.12 ug.mL-1 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC90 0.125 ug.mL-1 10.1128/aac.00595-08
Fusobacterium sp. Fusobacterium sp. MIC50 0.03 ug.mL-1 10.1128/aac.00595-08
Fusobacterium sp. Fusobacterium sp. MIC90 0.125 ug.mL-1 10.1128/aac.00595-08
Fusobacterium varium Fusobacterium varium Activity 8.0 % 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium Activity 92.0 % 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium MIC 0.008 ug.mL-1 10.1128/aac.00481-10
Fusobacterium varium Fusobacterium varium MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium MIC 0.06 ug.mL-1 10.1128/aac.00910-07
Fusobacterium varium Fusobacterium varium MIC 0.25 ug.mL-1 10.1128/aac.00595-08
Fusobacterium varium Fusobacterium varium MIC50 0.03 ug.mL-1 10.1128/aac.00595-08
Fusobacterium varium Fusobacterium varium MIC50 0.06 ug.mL-1 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium MIC50 0.125 ug.mL-1 10.1128/aac.00910-07
Fusobacterium varium Fusobacterium varium MIC90 0.12 ug.mL-1 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium MIC90 0.125 ug.mL-1 10.1128/aac.00595-08
Fusobacterium varium Fusobacterium varium MIC90 0.25 ug.mL-1 10.1128/aac.00910-07
Haemophilus influenzae Haemophilus influenzae Activity 0.0 % 10.1128/aac.00422-07
Haemophilus influenzae Haemophilus influenzae Activity 0.0 % 10.1128/aac.01538-07
Haemophilus influenzae Haemophilus influenzae Activity 9.5 % 10.1128/aac.00422-07
Haemophilus influenzae Haemophilus influenzae Activity 90.5 % 10.1128/aac.00422-07
Haemophilus influenzae Haemophilus influenzae Activity 99.0 % 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae Activity 99.6 % 10.1128/aac.00971-07
Haemophilus influenzae Haemophilus influenzae Activity 99.7 % 10.1128/aac.00971-07
Haemophilus influenzae Haemophilus influenzae Activity 100.0 % 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae Activity 100.0 % 10.1128/aac.00422-07
Haemophilus influenzae Haemophilus influenzae Activity 100.0 % 10.1128/aac.00971-07
Haemophilus influenzae Haemophilus influenzae MIC 6e-05 ug.mL-1 10.1128/aac.00294-06
Haemophilus influenzae Haemophilus influenzae MIC 0.016 ug.mL-1 10.1128/aac.00054-10
Haemophilus influenzae Haemophilus influenzae MIC 0.031 ug.mL-1 10.1128/aac.00054-10
Haemophilus influenzae Haemophilus influenzae MIC 0.06 ug.mL-1 10.1021/np800503z
Haemophilus influenzae Haemophilus influenzae MIC 0.06 ug.mL-1 10.1128/aac.00190-07
Haemophilus influenzae Haemophilus influenzae MIC 0.063 ug.mL-1 10.1128/aac.00054-10
Haemophilus influenzae Haemophilus influenzae MIC 0.064 ug.mL-1 10.1128/aac.00190-07
Haemophilus influenzae Haemophilus influenzae MIC 0.12 ug.mL-1 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC 0.125 ug.mL-1 10.1021/acs.jmedchem.6b00746
Haemophilus influenzae Haemophilus influenzae MIC 0.125 ug.mL-1 10.1128/aac.00190-07
Haemophilus influenzae Haemophilus influenzae MIC 3.125 ug.mL-1 10.1016/j.ejmech.2007.02.001
Haemophilus influenzae Haemophilus influenzae MIC50 0.03 ug.mL-1 10.1128/aac.00971-07
Haemophilus influenzae Haemophilus influenzae MIC50 0.06 ug.mL-1 10.1128/aac.00422-07
Haemophilus influenzae Haemophilus influenzae MIC50 0.06 ug.mL-1 10.1128/aac.00971-07
Haemophilus influenzae Haemophilus influenzae MIC50 0.063 ug.mL-1 10.1128/aac.00054-10
Haemophilus influenzae Haemophilus influenzae MIC50 0.064 ug.mL-1 10.1128/aac.00960-06
Haemophilus influenzae Haemophilus influenzae MIC50 0.094 ug.mL-1 10.1128/aac.00960-06
Haemophilus influenzae Haemophilus influenzae MIC50 0.12 ug.mL-1 10.1128/aac.00054-10
Haemophilus influenzae Haemophilus influenzae MIC50 0.12 ug.mL-1 10.1128/aac.00422-07
Haemophilus influenzae Haemophilus influenzae MIC50 0.125 ug.mL-1 10.1128/aac.00960-06
Haemophilus influenzae Haemophilus influenzae MIC50 0.19 ug.mL-1 10.1128/aac.00960-06
Haemophilus influenzae Haemophilus influenzae MIC50 0.25 ug.mL-1 10.1128/aac.00054-10
Haemophilus influenzae Haemophilus influenzae MIC50 0.25 ug.mL-1 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC50 0.25 ug.mL-1 10.1128/aac.00422-07
Haemophilus influenzae Haemophilus influenzae MIC90 0.06 ug.mL-1 10.1128/aac.00422-07
Haemophilus influenzae Haemophilus influenzae MIC90 0.06 ug.mL-1 10.1128/aac.00971-07
Haemophilus influenzae Haemophilus influenzae MIC90 0.12 ug.mL-1 10.1128/aac.00054-10
Haemophilus influenzae Haemophilus influenzae MIC90 0.12 ug.mL-1 10.1128/aac.00971-07
Haemophilus influenzae Haemophilus influenzae MIC90 0.125 ug.mL-1 10.1128/aac.00960-06
Haemophilus influenzae Haemophilus influenzae MIC90 0.25 ug.mL-1 10.1128/aac.00054-10
Haemophilus influenzae Haemophilus influenzae MIC90 0.25 ug.mL-1 10.1128/aac.00422-07
Haemophilus influenzae Haemophilus influenzae MIC90 0.38 ug.mL-1 10.1128/aac.00960-06
Haemophilus influenzae Haemophilus influenzae MIC90 0.5 ug.mL-1 10.1128/aac.00054-10
Haemophilus influenzae Haemophilus influenzae MIC90 0.5 ug.mL-1 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC90 0.5 ug.mL-1 10.1128/aac.00422-07
Haemophilus influenzae Haemophilus influenzae MIC90 32.0 ug.mL-1 10.1128/aac.00960-06
Haemophilus parainfluenzae Haemophilus parainfluenzae MIC 0.03 ug.mL-1 10.1021/np800503z
Homo sapiens Acetylcholinesterase AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Acetylcholinesterase IC50 nan None None
Homo sapiens Acetylcholinesterase Ki nan None None
Homo sapiens Adenosine A1 receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Adenosine A1 receptor IC50 nan None None
Homo sapiens Adenosine A1 receptor Ki nan None None
Homo sapiens Adenosine A2a receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Adenosine A2a receptor IC50 nan None None
Homo sapiens Adenosine A2a receptor Ki nan None None
Homo sapiens Adenosine A3 receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Adenosine A3 receptor IC50 nan None None
Homo sapiens Adenosine A3 receptor Ki nan None None
Homo sapiens Alpha-1a adrenergic receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-1a adrenergic receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-1d adrenergic receptor IC50 nan None None
Homo sapiens Alpha-1d adrenergic receptor Ki nan None None
Homo sapiens Alpha-2a adrenergic receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-2a adrenergic receptor IC50 nan None None
Homo sapiens Alpha-2a adrenergic receptor Ki nan None None
Homo sapiens Alpha-2b adrenergic receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-2b adrenergic receptor IC50 nan None None
Homo sapiens Alpha-2b adrenergic receptor Ki nan None None
Homo sapiens Alpha-2c adrenergic receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-2c adrenergic receptor IC50 nan None None
Homo sapiens Alpha-2c adrenergic receptor Ki nan None None
Homo sapiens Angiotensin II type 2 (AT-2) receptor IC50 nan None None
Homo sapiens Angiotensin II type 2 (AT-2) receptor Ki nan None None
Homo sapiens Beta-1 adrenergic receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Beta-1 adrenergic receptor IC50 nan None None
Homo sapiens Beta-1 adrenergic receptor Ki nan None None
Homo sapiens Beta-2 adrenergic receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Beta-2 adrenergic receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Beta-2 adrenergic receptor IC50 nan None None
Homo sapiens Beta-2 adrenergic receptor Ki nan None None
Homo sapiens Beta-3 adrenergic receptor IC50 nan None None
Homo sapiens Beta-3 adrenergic receptor Ki nan None None
Homo sapiens Bile salt export pump AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Bile salt export pump IC50 133000.0 nM 10.1093/toxsci/kft176
Homo sapiens Bradykinin B2 receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Bradykinin B2 receptor IC50 nan None None
Homo sapiens Bradykinin B2 receptor Ki nan None None
Homo sapiens Calcitonin receptor IC50 nan None None
Homo sapiens Calcitonin receptor Ki nan None None
Homo sapiens Canalicular multispecific organic anion transporter 1 IC50 133000.0 nM 10.1093/toxsci/kft176
Homo sapiens Canalicular multispecific organic anion transporter 2 IC50 133000.0 nM 10.1093/toxsci/kft176
Homo sapiens Cannabinoid CB1 receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Cannabinoid CB1 receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Cannabinoid CB1 receptor IC50 nan None None
Homo sapiens Cannabinoid CB1 receptor Ki nan None None
Homo sapiens Carbonic anhydrase II IC50 nan None None
Homo sapiens Carbonic anhydrase II Ki nan None None
Homo sapiens Caspase-1 IC50 nan None None
Homo sapiens Caspase-1 Ki nan None None
Homo sapiens Cathepsin G IC50 nan None None
Homo sapiens Cathepsin G Ki nan None None
Homo sapiens C-C chemokine receptor type 2 IC50 nan None None
Homo sapiens C-C chemokine receptor type 2 Ki nan None None
Homo sapiens C-C chemokine receptor type 4 IC50 nan None None
Homo sapiens C-C chemokine receptor type 4 Ki nan None None
Homo sapiens C-C chemokine receptor type 5 IC50 nan None None
Homo sapiens C-C chemokine receptor type 5 Ki nan None None
Homo sapiens Cholecystokinin A receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Cholecystokinin A receptor IC50 nan None None
Homo sapiens Cholecystokinin A receptor Ki nan None None
Homo sapiens Cyclooxygenase-1 IC50 nan None None
Homo sapiens Cyclooxygenase-1 Ki nan None None
Homo sapiens Cyclooxygenase-2 AC50 109999.3 nM 10.1038/s41467-023-40064-9
Homo sapiens Cyclooxygenase-2 IC50 nan None None
Homo sapiens Cyclooxygenase-2 Ki nan None None
Homo sapiens Cysteinyl leukotriene receptor 1 IC50 nan None None
Homo sapiens Cysteinyl leukotriene receptor 1 Ki nan None None
Homo sapiens Cytochrome P450 1A2 IC50 nan None None
Homo sapiens Cytochrome P450 1A2 Inhibition nan % 10.1021/tx300075j
Homo sapiens Cytochrome P450 1A2 Ki nan None None
Homo sapiens Cytochrome P450 2A6 IC50 nan None None
Homo sapiens Cytochrome P450 2A6 Ki nan None None
Homo sapiens Cytochrome P450 2C19 IC50 nan None None
Homo sapiens Cytochrome P450 2C19 Inhibition nan % 10.1021/tx300075j
Homo sapiens Cytochrome P450 2C19 Ki nan None None
Homo sapiens Cytochrome P450 2C9 IC50 nan None None
Homo sapiens Cytochrome P450 2C9 Inhibition nan % 10.1021/tx300075j
Homo sapiens Cytochrome P450 2C9 Ki nan None None
Homo sapiens Cytochrome P450 2D6 IC50 nan None None
Homo sapiens Cytochrome P450 2D6 Inhibition nan % 10.1021/tx300075j
Homo sapiens Cytochrome P450 2D6 Ki nan None None
Homo sapiens Cytochrome P450 2E1 IC50 nan None None
Homo sapiens Cytochrome P450 2E1 Ki nan None None
Homo sapiens Cytochrome P450 3A4 IC50 nan None None
Homo sapiens Cytochrome P450 3A4 Inhibition nan % 10.1021/tx300075j
Homo sapiens Cytochrome P450 3A4 Ki nan None None
Homo sapiens Delta opioid receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Delta opioid receptor IC50 nan None None
Homo sapiens Delta opioid receptor Ki nan None None
Homo sapiens Dihydropyrimidine dehydrogenase Activity 1.0 None 10.1016/s0960-894x(00)00575-8
Homo sapiens Dopamine D1 receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine D1 receptor IC50 nan None None
Homo sapiens Dopamine D1 receptor Ki nan None None
Homo sapiens Dopamine D2 receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine D2 receptor IC50 nan None None
Homo sapiens Dopamine D2 receptor Ki nan None None
Homo sapiens Dopamine D3 receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine D3 receptor IC50 nan None None
Homo sapiens Dopamine D3 receptor Ki nan None None
Homo sapiens Dopamine D4 receptor IC50 nan None None
Homo sapiens Dopamine D4 receptor Ki nan None None
Homo sapiens Dopamine transporter AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine transporter IC50 nan None None
Homo sapiens Dopamine transporter Ki nan None None
Homo sapiens Endothelin receptor ET-A AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Endothelin receptor ET-A IC50 nan None None
Homo sapiens Endothelin receptor ET-A Ki nan None None
Homo sapiens Epidermal growth factor receptor erbB1 AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Epidermal growth factor receptor erbB1 IC50 nan None None
Homo sapiens Epidermal growth factor receptor erbB1 Ki nan None None
Homo sapiens Equilibrative nucleoside transporter 1 AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Estrogen receptor alpha AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Estrogen receptor alpha AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Estrogen receptor alpha IC50 nan None None
Homo sapiens Estrogen receptor alpha Ki nan None None
Homo sapiens Estrogen receptor beta IC50 nan None None
Homo sapiens Estrogen receptor beta Ki nan None None
Homo sapiens Gamma-aminobutyric acid receptor subunit alpha-1/alpha-2/beta-2/gamma-2 AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Ghrelin receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Glucocorticoid receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Glucocorticoid receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Glucocorticoid receptor IC50 nan None None
Homo sapiens Glucocorticoid receptor Ki nan None None
Homo sapiens HEK293 Activity nan None 10.1016/j.ejmech.2022.114278
Homo sapiens HepaRG Activity nan None 10.1016/j.ejmech.2022.114278
Homo sapiens HERG AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens HERG IC50 nan None None
Homo sapiens HERG Ki nan None None
Homo sapiens Histamine H1 receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Histamine H1 receptor IC50 nan None None
Homo sapiens Histamine H1 receptor Ki nan None None
Homo sapiens Histamine H2 receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Histamine H2 receptor IC50 nan None None
Homo sapiens Histamine H2 receptor Ki nan None None
Homo sapiens Histamine H3 receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens HMG-CoA reductase IC50 nan None None
Homo sapiens HMG-CoA reductase Ki nan None None
Homo sapiens Homo sapiens Activity 2.0 % 10.1128/aac.01582-09
Homo sapiens Homo sapiens Activity 4.4 L/hr 10.1128/aac.01582-09
Homo sapiens Homo sapiens AUC 129500.0 ng.hr.mL-1 10.1128/aac.01582-09
Homo sapiens Homo sapiens AUC 166500.0 ng.hr.mL-1 10.1128/aac.01582-09
Homo sapiens Homo sapiens AUMC 26709.7 mg.hr/L 10.1128/aac.01582-09
Homo sapiens Homo sapiens AUMC 31378.3 mg.hr/L 10.1128/aac.01582-09
Homo sapiens Homo sapiens CL 2.4 L/hr 10.1128/aac.01582-09
Homo sapiens Homo sapiens CL 3.5 L/hr 10.1128/aac.01582-09
Homo sapiens Homo sapiens CL 3.9 mL.min-1.kg-1 10.1021/jm900403j
Homo sapiens Homo sapiens CL 6.0 L/hr 10.1128/aac.01582-09
Homo sapiens Homo sapiens CL_renal 0.005 L/hr 10.1128/aac.01582-09
Homo sapiens Homo sapiens CL_renal 2.73 mL.min-1.kg-1 10.1021/jm900403j
Homo sapiens Homo sapiens Cmax 147599.55 nM 10.1128/aac.01582-09
Homo sapiens Homo sapiens Cmin 7.6 mg/L 10.1128/aac.01582-09
Homo sapiens Homo sapiens DILI_Concern nan None 10.1016/j.drudis.2016.02.015
Homo sapiens Homo sapiens DILI_severity_class 3.0 None 10.1016/j.drudis.2016.02.015
Homo sapiens Homo sapiens fAUC 157430.0 ng.hr.mL-1 10.1128/aac.00294-06
Homo sapiens Homo sapiens fCmax 32.27 ug ml-1 10.1128/aac.00294-06
Homo sapiens Homo sapiens fCmin 0.91 ug ml-1 10.1128/aac.00294-06
Homo sapiens Homo sapiens fT>MIC 91.0 % 10.1128/aac.00294-06
Homo sapiens Homo sapiens Kel 0.16 /hr 10.1128/aac.01582-09
Homo sapiens Homo sapiens MRT 163.3 hr 10.1128/aac.01582-09
Homo sapiens Homo sapiens MRT 174.3 hr 10.1128/aac.01582-09
Homo sapiens Homo sapiens Ratio 0.74 None 10.1128/aac.01582-09
Homo sapiens Homo sapiens T1/2 4.32 hr 10.1128/aac.01582-09
Homo sapiens Homo sapiens Vd 0.37 L.kg-1 10.1128/aac.01582-09
Homo sapiens Interleukin-8 receptor A IC50 nan None None
Homo sapiens Interleukin-8 receptor A Ki nan None None
Homo sapiens Interleukin-8 receptor B IC50 nan None None
Homo sapiens Interleukin-8 receptor B Ki nan None None
Homo sapiens Kappa opioid receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Kappa opioid receptor IC50 nan None None
Homo sapiens Kappa opioid receptor Ki nan None None
Homo sapiens Leukocyte common antigen IC50 nan None None
Homo sapiens Leukocyte common antigen Ki nan None None
Homo sapiens Leukocyte elastase IC50 nan None None
Homo sapiens Leukocyte elastase Ki nan None None
Homo sapiens Liver microsomes Activity nan None 10.1021/tx300075j
Homo sapiens Liver microsomes Stability nan % 10.1021/tx300075j
Homo sapiens MAP kinase ERK1 IC50 nan None None
Homo sapiens MAP kinase ERK1 Ki nan None None
Homo sapiens MAP kinase ERK2 IC50 nan None None
Homo sapiens MAP kinase ERK2 Ki nan None None
Homo sapiens MAP kinase p38 alpha IC50 nan None None
Homo sapiens MAP kinase p38 alpha Ki nan None None
Homo sapiens Matrix metalloproteinase-1 IC50 nan None None
Homo sapiens Matrix metalloproteinase-1 Ki nan None None
Homo sapiens Matrix metalloproteinase 9 IC50 nan None None
Homo sapiens Matrix metalloproteinase 9 Ki nan None None
Homo sapiens Melanocortin receptor 3 AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Melanocortin receptor 3 IC50 nan None None
Homo sapiens Melanocortin receptor 3 Ki nan None None
Homo sapiens Melanocortin receptor 4 AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Melanocortin receptor 4 IC50 nan None None
Homo sapiens Melanocortin receptor 4 Ki nan None None
Homo sapiens Melanocortin receptor 5 IC50 nan None None
Homo sapiens Melanocortin receptor 5 Ki nan None None
Homo sapiens Monoamine oxidase A AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Monoamine oxidase A IC50 nan None None
Homo sapiens Monoamine oxidase A Ki nan None None
Homo sapiens Motilin receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Multidrug resistance-associated protein 4 IC50 133000.0 nM 10.1093/toxsci/kft176
Homo sapiens Mu opioid receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Mu opioid receptor IC50 nan None None
Homo sapiens Mu opioid receptor Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M1 AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Muscarinic acetylcholine receptor M1 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M1 Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M2 AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Muscarinic acetylcholine receptor M2 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M2 Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M3 AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Muscarinic acetylcholine receptor M3 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M3 Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M4 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M4 Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M5 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M5 Ki nan None None
Homo sapiens Neurokinin 1 receptor IC50 nan None None
Homo sapiens Neurokinin 1 receptor Ki nan None None
Homo sapiens Neurokinin 2 receptor IC50 nan None None
Homo sapiens Neurokinin 2 receptor Ki nan None None
Homo sapiens Neuronal acetylcholine receptor protein alpha-4 subunit AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Neuropeptide Y receptor type 1 AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Neuropeptide Y receptor type 1 IC50 nan None None
Homo sapiens Neuropeptide Y receptor type 1 Ki nan None None
Homo sapiens Neuropeptide Y receptor type 2 IC50 nan None None
Homo sapiens Neuropeptide Y receptor type 2 Ki nan None None
Homo sapiens Norepinephrine transporter AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Norepinephrine transporter IC50 nan None None
Homo sapiens Norepinephrine transporter Ki nan None None
Homo sapiens Peroxisome proliferator-activated receptor gamma AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Phosphodiesterase 3A AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Phosphodiesterase 4D AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Phosphodiesterase 5A IC50 nan None None
Homo sapiens Phosphodiesterase 5A Ki nan None None
Homo sapiens Plasma Fu nan None 10.1021/acsmedchemlett.5b00026
Homo sapiens Platelet activating factor receptor IC50 nan None None
Homo sapiens Platelet activating factor receptor Ki nan None None
Homo sapiens Pregnane X receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Pregnane X receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Progesterone receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Protein kinase C alpha IC50 nan None None
Homo sapiens Protein kinase C alpha Ki nan None None
Homo sapiens Receptor protein-tyrosine kinase erbB-2 AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Receptor protein-tyrosine kinase erbB-2 IC50 nan None None
Homo sapiens Receptor protein-tyrosine kinase erbB-2 Ki nan None None
Homo sapiens Renal dipeptidase Stability 100.0 % 10.1016/0960-894X(95)00380-C
Homo sapiens Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform IC50 nan None None
Homo sapiens Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform Ki nan None None
Homo sapiens Serotonin 1a (5-HT1a) receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2a (5-HT2a) receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2a (5-HT2a) receptor IC50 nan None None
Homo sapiens Serotonin 2a (5-HT2a) receptor Ki nan None None
Homo sapiens Serotonin 2b (5-HT2b) receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2b (5-HT2b) receptor IC50 nan None None
Homo sapiens Serotonin 2b (5-HT2b) receptor Ki nan None None
Homo sapiens Serotonin 2c (5-HT2c) receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2c (5-HT2c) receptor IC50 nan None None
Homo sapiens Serotonin 2c (5-HT2c) receptor Ki nan None None
Homo sapiens Serotonin 3a (5-HT3a) receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 6 (5-HT6) receptor IC50 nan None None
Homo sapiens Serotonin 6 (5-HT6) receptor Ki nan None None
Homo sapiens Serotonin transporter AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin transporter IC50 nan None None
Homo sapiens Serotonin transporter Ki nan None None
Homo sapiens Sigma opioid receptor IC50 nan None None
Homo sapiens Sigma opioid receptor Ki nan None None
Homo sapiens THP-1 Ratio 0.2 None 10.1128/aac.00123-08
Homo sapiens Thromboxane A2 receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Thromboxane A2 receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Thromboxane-A synthase IC50 nan None None
Homo sapiens Thromboxane-A synthase Ki nan None None
Homo sapiens Type-1 angiotensin II receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Tyrosine-protein kinase FYN IC50 nan None None
Homo sapiens Tyrosine-protein kinase FYN Ki nan None None
Homo sapiens Tyrosine-protein kinase LCK IC50 nan None None
Homo sapiens Tyrosine-protein kinase LCK Ki nan None None
Homo sapiens Vascular endothelial growth factor receptor 1 IC50 nan None None
Homo sapiens Vascular endothelial growth factor receptor 1 Ki nan None None
Homo sapiens Vascular endothelial growth factor receptor 2 AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Vasoactive intestinal polypeptide receptor 1 IC50 nan None None
Homo sapiens Vasoactive intestinal polypeptide receptor 1 Ki nan None None
Homo sapiens Vasopressin V1a receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Vasopressin V1a receptor IC50 nan None None
Homo sapiens Vasopressin V1a receptor Ki nan None None
Homo sapiens Vasopressin V2 receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Hoylesella oralis Hoylesella oralis Activity 0.0 % 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis Activity 100.0 % 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis MIC 0.03 ug.mL-1 10.1128/aac.00595-08
Hoylesella oralis Hoylesella oralis MIC50 0.125 ug.mL-1 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis MIC90 0.5 ug.mL-1 10.1128/aac.00481-10
Janthinobacterium lividum THIN-B proetin Kcat/Km 5.0 10'6/M/s 10.1128/aac.01062-07
Klebsiella aerogenes Klebsiella aerogenes Activity 0.0 % 10.1128/aac.01128-07
Klebsiella aerogenes Klebsiella aerogenes MIC 0.015 ug.mL-1 10.1128/aac.00336-08
Klebsiella aerogenes Klebsiella aerogenes MIC 0.03 ug.mL-1 10.1016/j.bmcl.2021.127928
Klebsiella aerogenes Klebsiella aerogenes MIC 0.032 ug.mL-1 10.1128/aac.01099-09
Klebsiella aerogenes Klebsiella aerogenes MIC 0.049 ug.mL-1 10.1016/j.bmcl.2003.09.039
Klebsiella aerogenes Klebsiella aerogenes MIC 0.049 ug.mL-1 10.1016/j.bmcl.2004.09.092
Klebsiella aerogenes Klebsiella aerogenes MIC 0.049 ug.mL-1 10.1016/j.ejmech.2006.10.006
Klebsiella aerogenes Klebsiella aerogenes MIC 0.049 ug.mL-1 10.1016/s0960-894x(00)00253-5
Klebsiella aerogenes Klebsiella aerogenes MIC 0.049 ug.mL-1 10.1016/s0960-894x(00)00575-8
Klebsiella aerogenes Klebsiella aerogenes MIC 0.049 ug.mL-1 10.1016/s0960-894x(01)00451-6
Klebsiella aerogenes Klebsiella aerogenes MIC 0.049 ug.mL-1 10.1016/s0960-894x(02)00948-4
Klebsiella aerogenes Klebsiella aerogenes MIC 0.049 ug.mL-1 10.1016/s0960-894x(98)00270-4
Klebsiella aerogenes Klebsiella aerogenes MIC 0.049 ug.mL-1 10.1016/s0960-894x(99)00407-2
Klebsiella aerogenes Klebsiella aerogenes MIC 0.049 ug.mL-1 10.1016/s0960-894x(99)00646-0
Klebsiella aerogenes Klebsiella aerogenes MIC 0.049 ug.mL-1 10.1016/s0960-894x(99)00692-7
Klebsiella aerogenes Klebsiella aerogenes MIC 0.06 ug.mL-1 10.1016/j.bmcl.2021.127928
Klebsiella aerogenes Klebsiella aerogenes MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Klebsiella aerogenes Klebsiella aerogenes MIC 0.125 ug.mL-1 10.1016/j.bmcl.2021.127928
Klebsiella aerogenes Klebsiella aerogenes MIC 2.0 ug.mL-1 10.1021/acs.jmedchem.9b01518
Klebsiella aerogenes Klebsiella aerogenes MIC 4.0 ug.mL-1 10.1016/j.bmcl.2021.127928
Klebsiella aerogenes Klebsiella aerogenes MIC 8.0 ug.mL-1 10.1128/aac.01099-09
Klebsiella aerogenes Klebsiella aerogenes MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.03.031
Klebsiella aerogenes Klebsiella aerogenes MIC50 0.03 ug.mL-1 10.1128/aac.00336-08
Klebsiella aerogenes Klebsiella aerogenes MIC50 0.06 ug.mL-1 10.1021/ml200012f
Klebsiella aerogenes Klebsiella aerogenes MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Klebsiella aerogenes Klebsiella aerogenes MIC50 0.25 ug.mL-1 10.1128/aac.01525-09
Klebsiella aerogenes Klebsiella aerogenes MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
Klebsiella aerogenes Klebsiella aerogenes MIC90 0.25 ug.mL-1 10.1021/ml200012f
Klebsiella aerogenes Klebsiella aerogenes MIC90 0.5 ug.mL-1 10.1128/aac.01128-07
Klebsiella aerogenes Klebsiella aerogenes MIC90 4.0 ug.mL-1 10.1128/aac.01525-09
Klebsiella oxytoca Klebsiella oxytoca Activity 0.0 % 10.1128/aac.00400-09
Klebsiella oxytoca Klebsiella oxytoca Activity 0.0 % 10.1128/aac.01128-07
Klebsiella oxytoca Klebsiella oxytoca Activity 100.0 % 10.1128/aac.00400-09
Klebsiella oxytoca Klebsiella oxytoca MIC 0.015 ug.mL-1 10.1128/aac.00336-08
Klebsiella oxytoca Klebsiella oxytoca MIC 0.049 ug.mL-1 10.1016/s0960-894x(99)00692-7
Klebsiella oxytoca Klebsiella oxytoca MIC 0.049 ug.mL-1 10.1021/np049577a
Klebsiella oxytoca Klebsiella oxytoca MIC 0.049 ug.mL-1 10.1021/np060206z
Klebsiella oxytoca Klebsiella oxytoca MIC 0.06 ug.mL-1 10.1016/j.bmcl.2003.09.039
Klebsiella oxytoca Klebsiella oxytoca MIC 0.06 ug.mL-1 10.1128/aac.00400-09
Klebsiella oxytoca Klebsiella oxytoca MIC 0.06 ug.mL-1 10.1128/aac.01004-09
Klebsiella oxytoca Klebsiella oxytoca MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Klebsiella oxytoca Klebsiella oxytoca MIC 0.125 ug.mL-1 10.1128/aac.01525-09
Klebsiella oxytoca Klebsiella oxytoca MIC 4.0 ug.mL-1 10.1021/acs.jmedchem.5b00127
Klebsiella oxytoca Klebsiella oxytoca MIC 32.0 ug.mL-1 10.1039/C5MD00380F
Klebsiella oxytoca Klebsiella oxytoca MIC 32.0 ug.mL-1 10.1128/aac.00260-09
Klebsiella oxytoca Klebsiella oxytoca MIC 32.0 ug.mL-1 10.1128/aac.01355-08
Klebsiella oxytoca Klebsiella oxytoca MIC50 0.03 ug.mL-1 10.1128/aac.00336-08
Klebsiella oxytoca Klebsiella oxytoca MIC50 0.03 ug.mL-1 10.1128/aac.01128-07
Klebsiella oxytoca Klebsiella oxytoca MIC50 0.06 ug.mL-1 10.1128/aac.00400-09
Klebsiella oxytoca Klebsiella oxytoca MIC50 0.06 ug.mL-1 10.1128/aac.01525-09
Klebsiella oxytoca Klebsiella oxytoca MIC90 0.06 ug.mL-1 10.1128/aac.00400-09
Klebsiella oxytoca Klebsiella oxytoca MIC90 0.06 ug.mL-1 10.1128/aac.01128-07
Klebsiella oxytoca Klebsiella oxytoca MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
Klebsiella oxytoca Klebsiella oxytoca MIC90 1.0 ug.mL-1 10.1128/aac.01525-09
Klebsiella pneumoniae Beta-lactamase AH27 CTX-M-15 Kcat 0.004 /s 10.1128/aac.00461-09
Klebsiella pneumoniae Beta-lactamase AH27 CTX-M-15 Km nan None 10.1128/aac.00461-09
Klebsiella pneumoniae Beta-lactamase AH27 CTX-M-15 Ratio nan None 10.1128/aac.00461-09
Klebsiella pneumoniae Beta-lactamase NDM-1 Kcat 12.0 /s 10.1128/aac.00774-09
Klebsiella pneumoniae Beta-lactamase NDM-1 Kcat/Km 0.25 /s/microM 10.1128/aac.00774-09
Klebsiella pneumoniae Beta-lactamase NDM-1 Kd 11000.0 nM 10.1016/j.bmcl.2016.03.004
Klebsiella pneumoniae Beta-lactamase NDM-1 Km 49000.0 nM 10.1128/aac.00774-09
Klebsiella pneumoniae Beta-lactamase NDM-1 MIC 32.0 ug.mL-1 10.1016/j.bmc.2020.115598
Klebsiella pneumoniae Beta-lactamase NDM-1 MIC 64.0 ug.mL-1 10.1016/j.bmc.2020.115598
Klebsiella pneumoniae Beta-lactamase SHV-1 Activity 0.00041 % 10.1128/aac.01004-09
Klebsiella pneumoniae Beta-lactamase SHV-1 Activity 0.015 % 10.1128/aac.01004-09
Klebsiella pneumoniae Beta-lactamase SHV-1 Kcat 0.0017 /s 10.1128/aac.01004-09
Klebsiella pneumoniae Beta-lactamase SHV-1 Kcat/Km 0.0004 /s/microM 10.1128/aac.01004-09
Klebsiella pneumoniae Beta-lactamase SHV-1 Km 4200.0 nM 10.1128/aac.01004-09
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Activity 0.92 % 10.1128/aac.01004-09
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Activity 2.0 % 10.1128/aac.00690-09
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Activity 31.0 U 10.1128/aac.00690-09
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Activity 37.0 % 10.1128/aac.01004-09
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Activity 55.0 U 10.1128/aac.00690-09
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Activity 57.0 % 10.1128/aac.00690-09
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Activity 64.0 % 10.1128/aac.00690-09
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Activity 76.0 U 10.1128/aac.00690-09
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Kcat 3.0 /s 10.1128/aac.00491-07
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Kcat 3.6 /s 10.1128/aac.01004-09
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Kcat/Km 0.28 /s/microM 10.1128/aac.01004-09
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Kcat/Km 250.0 /mM/s 10.1128/aac.00491-07
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Km 12000.0 nM 10.1128/aac.00491-07
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Km 13000.0 nM 10.1128/aac.01004-09
Klebsiella pneumoniae Class A carbapenemase Activity 0.06 umol 10.1128/aac.01180-07
Klebsiella pneumoniae Extended spectrum beta-lactamase CTX-M-71 Kcat 0.07 /s 10.1128/aac.00461-09
Klebsiella pneumoniae Extended spectrum beta-lactamase CTX-M-71 Km nan None 10.1128/aac.00461-09
Klebsiella pneumoniae Extended spectrum beta-lactamase CTX-M-71 Ratio nan None 10.1128/aac.00461-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 0.0 % 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 0.0 % 10.1128/aac.00400-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 0.0 % 10.1128/aac.01128-07
Klebsiella pneumoniae Klebsiella pneumoniae Activity 0.2 % 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 0.3 % 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 4.5 % 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 9.1 % 10.1128/aac.01538-07
Klebsiella pneumoniae Klebsiella pneumoniae Activity 12.5 % 10.1128/aac.01538-07
Klebsiella pneumoniae Klebsiella pneumoniae Activity 13.6 % 10.1128/aac.01538-07
Klebsiella pneumoniae Klebsiella pneumoniae Activity 17.8 % 10.1128/aac.01538-07
Klebsiella pneumoniae Klebsiella pneumoniae Activity 18.9 % 10.1128/aac.01538-07
Klebsiella pneumoniae Klebsiella pneumoniae Activity 95.5 % 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 99.7 % 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 99.8 % 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 100.0 % 10.1128/aac.00400-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 100.0 % 10.1128/aac.01509-06
Klebsiella pneumoniae Klebsiella pneumoniae Activity nan None 10.1016/j.ejmech.2022.114571
Klebsiella pneumoniae Klebsiella pneumoniae Activity nan None 10.1128/aac.01525-09
Klebsiella pneumoniae Klebsiella pneumoniae deltalog10CFU 1.41 None 10.1021/acs.jmedchem.5b00127
Klebsiella pneumoniae Klebsiella pneumoniae ED50 100.0 mg.kg-1 10.1021/acs.jmedchem.6b01261
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 0.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 3.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 5.0 % 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 12.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 16.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 18.0 % 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 30.0 % 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 38.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 45.0 % 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 47.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 50.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 56.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 58.0 % 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 59.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 62.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 65.0 % 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 68.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 69.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 72.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 75.0 % 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 78.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 80.0 % 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 85.0 % 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 88.0 % 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 90.0 % 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae fT>MIC 100.0 % 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae Inhibition 0.03 % 10.6019/CHEMBL4513141
Klebsiella pneumoniae Klebsiella pneumoniae Inhibition nan % 10.1016/j.bmc.2021.116128
Klebsiella pneumoniae Klebsiella pneumoniae Inhibition nan % 10.1128/aac.01452-08
Klebsiella pneumoniae Klebsiella pneumoniae IZ 13.0 mm 10.1128/aac.01325-08
Klebsiella pneumoniae Klebsiella pneumoniae IZ 14.0 mm 10.1128/aac.01325-08
Klebsiella pneumoniae Klebsiella pneumoniae IZ 23.0 mm 10.1128/aac.00543-08
Klebsiella pneumoniae Klebsiella pneumoniae IZ 27.0 mm 10.1128/aac.01325-08
Klebsiella pneumoniae Klebsiella pneumoniae log10cfu 3.0 None 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae MBC 0.06 ug ml-1 10.1128/aac.01452-08
Klebsiella pneumoniae Klebsiella pneumoniae MBC 16.0 ug ml-1 10.1128/aac.01452-08
Klebsiella pneumoniae Klebsiella pneumoniae MBC 64.0 ug ml-1 10.1021/acs.jmedchem.2c01469
Klebsiella pneumoniae Klebsiella pneumoniae MIC 6e-05 ug.mL-1 10.1128/aac.00294-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.015 ug.mL-1 10.1128/aac.00083-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.015 ug.mL-1 10.1128/aac.00336-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.015 ug.mL-1 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.016 ug.mL-1 10.1016/j.bmcl.2003.09.039
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.016 ug.mL-1 10.1128/aac.00830-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.016 ug.mL-1 10.1128/aac.01099-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.025 ug.mL-1 10.1016/j.ejmech.2007.02.001
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.03 ug.mL-1 10.1016/j.bmcl.2003.09.039
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.03 ug.mL-1 10.1016/j.bmcl.2021.127928
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.03 ug.mL-1 10.1021/acs.jmedchem.6b00746
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.03 ug.mL-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.03 ug.mL-1 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.03 ug.mL-1 10.1128/aac.00715-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.03 ug.mL-1 10.1128/aac.01004-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.03 ug.mL-1 10.1128/aac.01452-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.031 ug.mL-1 10.1016/j.bmc.2021.116343
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.032 ug.mL-1 10.1128/aac.00830-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.032 ug.mL-1 10.1128/aac.01099-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.032 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.04 ug.mL-1 10.1021/jm010546b
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.047 ug.mL-1 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.047 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.05 ug.mL-1 10.1016/j.ejmech.2006.10.006
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.06 ug.mL-1 10.1016/j.bmcl.2003.09.039
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.06 ug.mL-1 10.1016/j.bmcl.2021.127928
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.06 ug.mL-1 10.1021/acs.jmedchem.9b01518
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.06 ug.mL-1 10.1021/np800503z
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.06 ug.mL-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.06 ug.mL-1 10.1128/aac.00083-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.06 ug.mL-1 10.1128/aac.00400-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.06 ug.mL-1 10.1128/aac.01004-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.06 ug.mL-1 10.1128/aac.01452-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.0625 ug.mL-1 10.1016/j.ejmech.2022.114495
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.064 ug.mL-1 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.064 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.094 ug.mL-1 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.094 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.12 ug.mL-1 10.1016/j.bmc.2013.09.041
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.12 ug.mL-1 10.1128/aac.00017-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.125 ug.mL-1 10.1016/j.bmcl.2021.127928
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.125 ug.mL-1 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.125 ug.mL-1 10.1128/aac.00830-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.128 ug.mL-1 10.1016/j.ejmech.2021.113975
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.25 ug.mL-1 10.1021/jm400560z
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.25 ug.mL-1 10.1128/aac.00008-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.25 ug.mL-1 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.25 ug.mL-1 10.1128/aac.01325-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.5 ug.mL-1 10.1016/j.ejmech.2022.114571
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.5 ug.mL-1 10.1128/aac.00461-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.5 ug.mL-1 10.1128/aac.00543-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.5 ug.mL-1 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.5 ug.mL-1 10.1128/aac.01312-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.75 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1016/j.bmc.2021.116343
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1016/j.bmcl.2021.127928
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1016/j.ejmech.2019.02.024
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1016/j.ejmech.2022.114278
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1021/acs.jmedchem.8b00091
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1021/ml200012f
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1039/C5MD00380F
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.00008-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.00158-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.01099-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.01451-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.5 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1016/j.ejmech.2018.06.054
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1021/acs.jmedchem.8b00091
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.00008-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.00026-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.00158-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.00260-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.00299-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.00690-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.01099-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.01312-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.01451-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.01818-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 3.0 ug.mL-1 10.1128/aac.00436-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 3.0 ug.mL-1 10.1128/aac.01451-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1021/acs.jmedchem.5b00127
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1039/C5MD00380F
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00008-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00017-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00158-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00197-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00299-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00458-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00461-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00736-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.01099-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.01325-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.01451-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.01452-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.01525-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.01539-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.01818-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 6.0 ug.mL-1 10.1128/aac.01180-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 6.0 ug.mL-1 10.1128/aac.01451-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 6.0 ug.mL-1 10.1128/aac.01672-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1016/j.bmc.2021.116142
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1016/j.ejmech.2018.03.031
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1021/acs.jmedchem.5b00127
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.00008-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.00158-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.00299-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.00690-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.01099-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.01325-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.01818-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 12.0 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1016/j.ejmech.2018.03.031
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1016/j.ejmech.2018.06.014
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1016/j.ejmech.2022.114278
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.2c01257
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.2c01469
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.5b00127
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.8b00091
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.9b01518
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1039/C5MD00380F
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.00008-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.00011-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.00260-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.00690-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.01004-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.01099-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.01312-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.01355-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.01672-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1016/j.bmcl.2021.127928
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.03.031
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.06.054
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1016/j.ejmech.2019.02.024
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1021/acs.jmedchem.6b01261
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1021/acs.jmedchem.9b00720
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1039/C5MD00380F
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.00008-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.00017-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.00137-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.00260-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.00299-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.00736-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.00752-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01053-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01247-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01312-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01355-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01451-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01525-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01672-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01818-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1016/j.bmcl.2021.127928
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.03.031
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.03.058
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.06.054
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1016/j.ejmech.2022.114599
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1021/acs.jmedchem.5b00127
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1021/acs.jmedchem.6b01261
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1021/acs.jmedchem.9b00720
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1021/acs.jmedchem.9b01518
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1021/jm400560z
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1021/np800503z
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1128/aac.00008-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1128/aac.00543-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1128/aac.00690-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1128/aac.01190-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1128/aac.01312-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1128/aac.01355-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1128/aac.01818-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1016/j.bmcl.2021.127956
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1021/acs.jmedchem.9b01518
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1021/np4000944
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1039/C5MD00380F
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1128/aac.00008-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1128/aac.01818-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1016/j.bmc.2021.116128
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1021/acs.jmedchem.2c01469
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.00008-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.00774-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.01099-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.01539-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 512.0 ug.mL-1 10.1128/aac.00008-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1000.0 nM 10.1021/acs.jmedchem.1c00614
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1000.0 nM 10.1021/acs.jmedchem.1c02140
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16000.0 nM 10.1021/acs.jmedchem.1c00621
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64000.0 nM 10.1021/acs.jmedchem.1c00621
Klebsiella pneumoniae Klebsiella pneumoniae MIC nan None 10.1016/j.ejmech.2017.10.044
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.03 ug.mL-1 10.1016/j.bmcl.2004.09.092
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.03 ug.mL-1 10.1021/jm400560z
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.03 ug.mL-1 10.1128/aac.00083-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.03 ug.mL-1 10.1128/aac.00336-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.03 ug.mL-1 10.1128/aac.01128-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.03 ug.mL-1 10.1128/aac.01450-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.03 ug.mL-1 10.1128/aac.01509-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.047 ug.mL-1 10.1128/aac.00171-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.06 ug.mL-1 10.1021/ml200012f
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.06 ug.mL-1 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.06 ug.mL-1 10.1128/aac.00400-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.06 ug.mL-1 10.1128/aac.01525-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 0.12 ug.mL-1 10.1128/aac.00083-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 16.0 ug.mL-1 10.1021/acs.jmedchem.0c00255
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 32.0 ug.mL-1 10.1021/jm400560z
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.06 ug.mL-1 10.1016/j.bmcl.2004.09.092
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.06 ug.mL-1 10.1016/j.bmcl.2016.06.019
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.06 ug.mL-1 10.1128/aac.00083-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.06 ug.mL-1 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.06 ug.mL-1 10.1128/aac.00400-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.06 ug.mL-1 10.1128/aac.01128-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.06 ug.mL-1 10.1128/aac.01450-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.064 ug.mL-1 10.1128/aac.00171-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.094 ug.mL-1 10.1128/aac.00171-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.125 ug.mL-1 10.1128/aac.00171-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.19 ug.mL-1 10.1128/aac.00171-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.25 ug.mL-1 10.1021/jm400560z
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.25 ug.mL-1 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.25 ug.mL-1 10.1128/aac.01509-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 0.5 ug.mL-1 10.1128/aac.00083-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 16.0 ug.mL-1 10.1128/aac.01525-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 32.0 ug.mL-1 10.1016/j.bmcl.2012.07.005
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 32.0 ug.mL-1 10.1021/ml200012f
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 64.0 ug.mL-1 10.1021/acs.jmedchem.0c00255
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 64.0 ug.mL-1 10.1021/jm400560z
Klebsiella pneumoniae Klebsiella pneumoniae MPC 0.06 ug ml-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MPC 0.125 ug ml-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MPC 0.5 ug ml-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MPC 8.0 ug ml-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MPC 16.0 ug ml-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MPC 32.0 ug ml-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae MPC 64.0 ug ml-1 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae Ratio 1.0 None 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae Ratio 2.0 None 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae Ratio 4.0 None 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae Ratio 8.0 None 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae Ratio 16.0 None 10.1128/aac.00033-10
Klebsiella pneumoniae Klebsiella pneumoniae Survival 0.0 % 10.1021/acs.jmedchem.6b01261
Klebsiella pneumoniae Klebsiella pneumoniae Survival 69.0 % 10.1039/C5MD00380F
Klebsiella pneumoniae Metallo-beta-lactamase Activity 42.0 U 10.1128/aac.00690-09
Klebsiella pneumoniae Metallo-beta-lactamase Activity 55.0 U 10.1128/aac.00690-09
Klebsiella pneumoniae Metallo-beta-lactamase Activity 57.0 % 10.1128/aac.00690-09
Klebsiella pneumoniae Metallo-beta-lactamase Activity 64.0 % 10.1128/aac.00690-09
Klebsiella pneumoniae Metallo-beta-lactamase Activity 76.0 U 10.1128/aac.00690-09
Klebsiella pneumoniae Metallo-beta-lactamase Activity 80.0 % 10.1128/aac.00690-09
Klebsiella pneumoniae Metallo-beta-lactamase Activity 80.0 U 10.1128/aac.00690-09
Klebsiella pneumoniae Metallo-beta-lactamase Activity 100.0 % 10.1128/aac.00690-09
Klebsiella pneumoniae Metallo-beta-lactamase VIM-2 Kcat 1.0 /s 10.1128/aac.00774-09
Klebsiella pneumoniae Metallo-beta-lactamase VIM-2 Kcat/Km 0.28 /s/microM 10.1128/aac.00774-09
Klebsiella pneumoniae Metallo-beta-lactamase VIM-2 Km 5000.0 nM 10.1128/aac.00774-09
Klebsiella pneumoniae OXA-48 Activity 0.05 umol/min/mg 10.1128/aac.00543-08
Klebsiella pneumoniae OXA-48 Ka 4.0 10'4/M/s 10.1021/acs.jmedchem.6b00660
Klebsiella pneumoniae OXA-48 Kcat 0.098 /s 10.1021/acs.jmedchem.6b00660
Klebsiella pneumoniae OXA-48 Kcat/Km 9.8 10'4/M/s 10.1021/acs.jmedchem.6b00660
Klebsiella pneumoniae OXA-48 Kd 0.3463 /s 10.1021/acs.jmedchem.6b00660
Klebsiella pneumoniae OXA-48 Kd 850.0 nM 10.1021/acs.jmedchem.6b00660
Klebsiella pneumoniae OXA-48 Km 1000.0 nM 10.1021/acs.jmedchem.6b00660
Klebsiella sp. Klebsiella sp. Activity 20.0 % 10.1128/aac.01114-07
Klebsiella sp. Klebsiella sp. Activity 61.7 % 10.1128/aac.01114-07
Klebsiella sp. Klebsiella sp. MIC50 8.0 ug.mL-1 10.1128/aac.01114-07
Klebsiella sp. Klebsiella sp. MIC90 8.0 ug.mL-1 10.1128/aac.01114-07
Lacrimispora sphenoides Lacrimispora sphenoides Activity 0.0 % 10.1128/aac.01128-07
Lacrimispora sphenoides Lacrimispora sphenoides MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Lacrimispora sphenoides Lacrimispora sphenoides MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
Lacticaseibacillus casei Lacticaseibacillus casei MIC 2.0 ug.mL-1 10.1128/aac.00595-08
Lactiplantibacillus plantarum Lactiplantibacillus plantarum MIC 0.25 ug.mL-1 10.1128/aac.00595-08
Lactobacillus acidophilus Lactobacillus acidophilus MIC 0.25 ug.mL-1 10.1128/aac.00595-08
Limosilactobacillus fermentum Limosilactobacillus fermentum MIC 0.25 ug.mL-1 10.1128/aac.00595-08
Limosilactobacillus reuteri Limosilactobacillus reuteri MIC 0.5 ug.mL-1 10.1128/aac.00595-08
Micrococcus luteus Micrococcus luteus MIC 0.05 ug.mL-1 10.1016/j.ejmech.2006.10.006
Micrococcus luteus Micrococcus luteus MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
Micrococcus luteus Micrococcus luteus MIC nan None 10.1021/acs.jmedchem.2c01674
Moraxella catarrhalis Moraxella catarrhalis MIC 0.004 ug.mL-1 10.1021/np800503z
Moraxella catarrhalis Moraxella catarrhalis MIC 0.008 ug.mL-1 10.1021/acs.jmedchem.6b00746
Moraxella catarrhalis Moraxella catarrhalis MIC 0.06 ug.mL-1 10.1128/aac.00400-09
Moraxella catarrhalis Moraxella catarrhalis MIC50 0.004 ug.mL-1 10.1128/aac.00971-07
Moraxella catarrhalis Moraxella catarrhalis MIC50 0.008 ug.mL-1 10.1016/j.bmcl.2004.09.092
Moraxella catarrhalis Moraxella catarrhalis MIC50 0.06 ug.mL-1 10.1128/aac.00400-09
Moraxella catarrhalis Moraxella catarrhalis MIC90 0.008 ug.mL-1 10.1016/j.bmcl.2004.09.092
Moraxella catarrhalis Moraxella catarrhalis MIC90 0.008 ug.mL-1 10.1128/aac.00971-07
Moraxella catarrhalis Moraxella catarrhalis MIC90 0.06 ug.mL-1 10.1128/aac.00400-09
Morganella morganii Morganella morganii MIC 0.06 ug.mL-1 10.1016/S0960-894X(97)00282-5
Morganella morganii Morganella morganii MIC 0.06 ug.mL-1 10.1128/aac.00336-08
Morganella morganii Morganella morganii MIC50 0.12 ug.mL-1 10.1128/aac.00336-08
Morganella morganii Morganella morganii MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
Mus musculus Mus musculus AUC 0.0 hr 10.1016/s0960-894x(99)00407-2
Mus musculus Mus musculus AUC 3.29 ug ml-1 10.1016/s0960-894x(99)00692-7
Mus musculus Mus musculus AUC 6860.0 ng.hr.mL-1 10.1016/s0960-894x(99)00407-2
Mus musculus Mus musculus Cmax 19819.02 nM 10.1016/s0960-894x(99)00692-7
Mus musculus Mus musculus Cmax 40602.92 nM 10.1016/s0960-894x(99)00407-2
Mus musculus Mus musculus ED50 7.88 mg.kg-1 10.1016/S0960-894X(97)00230-8
Mus musculus Mus musculus PD50 0.65 mg kg-1 10.1016/s0960-894x(99)00407-2
Mus musculus Mus musculus PD50 1.11 mg kg-1 10.1016/s0960-894x(02)00948-4
Mus musculus Mus musculus PD50 1.24 mg kg-1 10.1016/s0960-894x(99)00692-7
Mus musculus Mus musculus PD50 4.26 mg kg-1 10.1016/s0960-894x(99)00407-2
Mus musculus Mus musculus PD50 4.49 mg kg-1 10.1016/s0960-894x(02)00948-4
Mus musculus Mus musculus PD50 4.55 mg kg-1 10.1016/s0960-894x(99)00407-2
Mus musculus Mus musculus PD50 4.6 mg kg-1 10.1016/s0960-894x(99)00692-7
Mus musculus Mus musculus PD50 4.72 mg kg-1 10.1016/s0960-894x(02)00948-4
Mus musculus Mus musculus PD50 5.43 mg kg-1 10.1016/s0960-894x(02)00948-4
Mus musculus Mus musculus PD50 11.1 mg kg-1 10.1016/s0960-894x(99)00407-2
Mus musculus Mus musculus PD50 nan None 10.1016/s0960-894x(99)00692-7
Mus musculus Mus musculus Recovery 25.0 % 10.1016/0960-894X(95)00380-C
Mus musculus Mus musculus T1/2 0.24 hr 10.1016/s0960-894x(99)00692-7
Mus musculus Mus musculus T1/2 0.27 hr 10.1016/s0960-894x(99)00407-2
Mus musculus Mus musculus Tmax 0.17 hr 10.1016/s0960-894x(99)00407-2
Mus musculus Mus musculus Tmax 0.21 hr 10.1016/s0960-894x(99)00692-7
Mus musculus Nitric oxide synthase, inducible IC50 nan None None
Mus musculus Nitric oxide synthase, inducible Ki nan None None
Mus musculus Plasma fAUC 4466.67 ng.hr.mL-1 10.1128/aac.00642-09
Mus musculus Plasma fAUC 30616.67 ng.hr.mL-1 10.1128/aac.00642-09
Mus musculus Plasma fCmax 11.0 ug ml-1 10.1128/aac.00642-09
Mus musculus Plasma fCmax 72.0 ug ml-1 10.1128/aac.00642-09
Mus musculus Plasma T1/2 0.1433 hr 10.1128/aac.00642-09
Mus musculus Plasma T1/2 0.2267 hr 10.1128/aac.00642-09
Mus musculus Plasma Tmax 0.125 hr 10.1128/aac.00642-09
Mycobacterium avium Mycobacterium avium MIC90 64.0 ug.mL-1 10.1016/j.bmcl.2016.06.019
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 1.7 log10CFU 10.1021/acs.jmedchem.2c00227
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 2.0 log10CFU 10.1021/acs.jmedchem.2c00227
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1016/j.bmc.2013.05.024
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.ejmech.2017.06.005
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 4.0 ug.mL-1 10.1016/j.bmcl.2016.06.019
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 8.0 ug.mL-1 10.1016/j.bmcl.2016.06.019
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 10000.0 nM 10.1021/acs.jmedchem.2c00227
Mycobacteroides abscessus Mycobacteroides abscessus MIC90 64.0 ug.mL-1 10.1016/j.bmcl.2016.06.019
Neisseria meningitidis Neisseria meningitidis MIC50 0.008 ug.mL-1 10.1128/aac.01315-06
Neisseria meningitidis Neisseria meningitidis MIC90 0.015 ug.mL-1 10.1128/aac.01315-06
Nocardia brasiliensis Nocardia brasiliensis MIC 0.001 ug.mL-1 10.1128/aac.01102-06
Nocardia brasiliensis Nocardia brasiliensis MIC50 2.0 ug.mL-1 10.1128/aac.01520-09
Nocardia brasiliensis Nocardia brasiliensis MIC90 8.0 ug.mL-1 10.1128/aac.01520-09
Nocardia carnea Nocardia carnea MIC 0.001 ug.mL-1 10.1128/aac.01102-06
Nocardia cyriacigeorgica Nocardia cyriacigeorgica MIC 6e-05 ug.mL-1 10.1128/aac.01102-06
Nocardia farcinica Nocardia farcinica MIC 0.002 ug.mL-1 10.1128/aac.01102-06
Nocardia nova Nocardia nova MIC 0.0005 ug.mL-1 10.1128/aac.01102-06
Nocardia otitidiscaviarum Nocardia otitidiscaviarum MIC 0.001 ug.mL-1 10.1128/aac.01102-06
Nocardia sp. Nocardia sp. MIC 6e-05 ug.mL-1 10.1128/aac.01102-06
Nocardia transvalensis Nocardia transvalensis MIC 0.064 ug.mL-1 10.1128/aac.01102-06
Oryctolagus cuniculus Angiotensin-converting enzyme IC50 nan None None
Oryctolagus cuniculus Angiotensin-converting enzyme Ki nan None None
Oryctolagus cuniculus Arachidonate 15-lipoxygenase IC50 nan None None
Oryctolagus cuniculus Arachidonate 15-lipoxygenase Ki nan None None
Paeniclostridium sordellii Paeniclostridium sordellii MIC 0.03 ug.mL-1 10.1128/aac.00595-08
Paeniclostridium sordellii Paeniclostridium sordellii MIC 0.06 ug.mL-1 10.1128/aac.00910-07
Parabacteroides distasonis Parabacteroides distasonis Activity 0.0 % 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis Activity 0.0 % 10.1128/aac.00696-08
Parabacteroides distasonis Parabacteroides distasonis Activity 0.0 % 10.1128/aac.01128-07
Parabacteroides distasonis Parabacteroides distasonis Activity 1.1 % 10.1128/aac.01435-06
Parabacteroides distasonis Parabacteroides distasonis Activity 98.0 % 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis MIC 0.125 ug.mL-1 10.1128/aac.00910-07
Parabacteroides distasonis Parabacteroides distasonis MIC 0.13 ug.mL-1 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis MIC 0.25 ug.mL-1 10.1128/aac.00696-08
Parabacteroides distasonis Parabacteroides distasonis MIC50 0.125 ug.mL-1 10.1128/aac.00910-07
Parabacteroides distasonis Parabacteroides distasonis MIC50 0.25 ug.mL-1 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis MIC50 0.25 ug.mL-1 10.1128/aac.00595-08
Parabacteroides distasonis Parabacteroides distasonis MIC50 0.25 ug.mL-1 10.1128/aac.01128-07
Parabacteroides distasonis Parabacteroides distasonis MIC50 1.0 ug.mL-1 10.1128/aac.00696-08
Parabacteroides distasonis Parabacteroides distasonis MIC90 0.5 ug.mL-1 10.1128/aac.00910-07
Parabacteroides distasonis Parabacteroides distasonis MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
Parabacteroides distasonis Parabacteroides distasonis MIC90 2.0 ug.mL-1 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis MIC90 2.0 ug.mL-1 10.1128/aac.00696-08
Parabacteroides distasonis Parabacteroides distasonis MIC90 2.0 ug.mL-1 10.1128/aac.01435-06
Parabacteroides distasonis Parabacteroides distasonis MIC90 4.0 ug.mL-1 10.1128/aac.00595-08
Parabacteroides merdae Parabacteroides merdae Activity 0.0 % 10.1128/aac.00696-08
Parabacteroides merdae Parabacteroides merdae Activity 0.0 % 10.1128/aac.01128-07
Parabacteroides merdae Parabacteroides merdae Activity 0.5 % 10.1128/aac.01435-06
Parabacteroides merdae Parabacteroides merdae MIC 0.125 ug.mL-1 10.1128/aac.00696-08
Parabacteroides merdae Parabacteroides merdae MIC 0.4 ug.mL-1 10.1128/aac.01435-06
Parabacteroides merdae Parabacteroides merdae MIC50 0.25 ug.mL-1 10.1128/aac.00696-08
Parabacteroides merdae Parabacteroides merdae MIC50 0.25 ug.mL-1 10.1128/aac.01128-07
Parabacteroides merdae Parabacteroides merdae MIC90 1.0 ug.mL-1 10.1128/aac.00696-08
Parabacteroides merdae Parabacteroides merdae MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
Parabacteroides merdae Parabacteroides merdae MIC90 1.0 ug.mL-1 10.1128/aac.01435-06
Paraclostridium bifermentans Paraclostridium bifermentans MIC 0.125 ug.mL-1 10.1128/aac.00910-07
Parvimonas micra Parvimonas micra Activity 0.0 % 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra Activity 0.0 % 10.1128/aac.00481-10
Parvimonas micra Parvimonas micra Activity 0.0 % 10.1128/aac.00696-08
Parvimonas micra Parvimonas micra Activity 0.0 % 10.1128/aac.01128-07
Parvimonas micra Parvimonas micra Activity 100.0 % 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra MIC 0.01 ug.mL-1 10.1128/aac.00481-10
Parvimonas micra Parvimonas micra MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra MIC 0.03 ug.mL-1 10.1128/aac.00910-07
Parvimonas micra Parvimonas micra MIC 0.06 ug.mL-1 10.1128/aac.00696-08
Parvimonas micra Parvimonas micra MIC 0.125 ug.mL-1 10.1128/aac.00595-08
Parvimonas micra Parvimonas micra MIC50 0.03 ug.mL-1 10.1128/aac.00910-07
Parvimonas micra Parvimonas micra MIC50 0.06 ug.mL-1 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra MIC50 0.06 ug.mL-1 10.1128/aac.00595-08
Parvimonas micra Parvimonas micra MIC50 0.125 ug.mL-1 10.1128/aac.00696-08
Parvimonas micra Parvimonas micra MIC50 0.125 ug.mL-1 10.1128/aac.01128-07
Parvimonas micra Parvimonas micra MIC50 0.25 ug.mL-1 10.1128/aac.00481-10
Parvimonas micra Parvimonas micra MIC90 0.125 ug.mL-1 10.1128/aac.00595-08
Parvimonas micra Parvimonas micra MIC90 0.25 ug.mL-1 10.1128/aac.00910-07
Parvimonas micra Parvimonas micra MIC90 0.25 ug.mL-1 10.1128/aac.01128-07
Parvimonas micra Parvimonas micra MIC90 0.5 ug.mL-1 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra MIC90 0.5 ug.mL-1 10.1128/aac.00696-08
Parvimonas micra Parvimonas micra MIC90 4.0 ug.mL-1 10.1128/aac.00481-10
Pasteurella multocida Pasteurella multocida MIC 0.05 ug.mL-1 10.1016/j.ejmech.2006.10.006
Pasteurella multocida Pasteurella multocida MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
Pectobacterium atrosepticum Pectobacterium atrosepticum MIC 0.25 ug.mL-1 10.1128/aac.01062-07
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus Activity 0.0 % 10.1128/aac.00355-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus Activity 0.0 % 10.1128/aac.00481-10
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus Activity 0.0 % 10.1128/aac.00696-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus Activity 0.0 % 10.1128/aac.01128-07
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus Activity 100.0 % 10.1128/aac.00355-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus Activity 100.0 % 10.1128/aac.00481-10
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC 0.008 ug.mL-1 10.1128/aac.00481-10
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC 0.015 ug.mL-1 10.1128/aac.00595-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC 0.06 ug.mL-1 10.1128/aac.00696-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC50 0.008 ug.mL-1 10.1128/aac.00481-10
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC50 0.015 ug.mL-1 10.1128/aac.00595-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC50 0.015 ug.mL-1 10.1128/aac.01128-07
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC50 0.016 ug.mL-1 10.1128/aac.00910-07
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC50 0.06 ug.mL-1 10.1128/aac.00355-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC50 0.125 ug.mL-1 10.1128/aac.00696-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC90 0.03 ug.mL-1 10.1128/aac.00481-10
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC90 0.03 ug.mL-1 10.1128/aac.00910-07
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC90 0.125 ug.mL-1 10.1128/aac.00595-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC90 0.125 ug.mL-1 10.1128/aac.01128-07
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC90 0.5 ug.mL-1 10.1128/aac.00355-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC90 0.5 ug.mL-1 10.1128/aac.00696-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius Activity 0.0 % 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius Activity 0.0 % 10.1128/aac.01128-07
Peptostreptococcus anaerobius Peptostreptococcus anaerobius Activity 100.0 % 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius Activity 100.0 % 10.1128/aac.00481-10
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC 0.01 ug.mL-1 10.1128/aac.00481-10
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC 0.25 ug.mL-1 10.1128/aac.00910-07
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC 0.5 ug.mL-1 10.1128/aac.00595-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC50 0.06 ug.mL-1 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC50 0.125 ug.mL-1 10.1128/aac.01128-07
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC50 0.25 ug.mL-1 10.1128/aac.00481-10
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC50 0.25 ug.mL-1 10.1128/aac.00595-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC50 0.25 ug.mL-1 10.1128/aac.00910-07
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC90 0.25 ug.mL-1 10.1128/aac.01128-07
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC90 0.5 ug.mL-1 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC90 2.0 ug.mL-1 10.1128/aac.00595-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC90 2.0 ug.mL-1 10.1128/aac.00910-07
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC90 4.0 ug.mL-1 10.1128/aac.00481-10
Peptostreptococcus sp. Peptostreptococcus sp. Activity 0.0 % 10.1128/aac.00696-08
Peptostreptococcus sp. Peptostreptococcus sp. MIC 0.06 ug.mL-1 10.1128/aac.00696-08
Peptostreptococcus sp. Peptostreptococcus sp. MIC50 0.125 ug.mL-1 10.1128/aac.00696-08
Peptostreptococcus sp. Peptostreptococcus sp. MIC90 0.5 ug.mL-1 10.1128/aac.00696-08
Phocaeicola vulgatus Phocaeicola vulgatus Activity 0.0 % 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus Activity 0.0 % 10.1128/aac.00696-08
Phocaeicola vulgatus Phocaeicola vulgatus Activity 0.0 % 10.1128/aac.01128-07
Phocaeicola vulgatus Phocaeicola vulgatus Activity 0.0 % 10.1128/aac.01435-06
Phocaeicola vulgatus Phocaeicola vulgatus Activity 4.0 % 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus Activity 96.0 % 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus Activity 98.0 % 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus MIC 0.12 ug.mL-1 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC 0.125 ug.mL-1 10.1128/aac.00595-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC 0.125 ug.mL-1 10.1128/aac.00910-07
Phocaeicola vulgatus Phocaeicola vulgatus MIC 0.13 ug.mL-1 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus MIC 0.25 ug.mL-1 10.1128/aac.00696-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC 0.47 ug.mL-1 10.1128/aac.01435-06
Phocaeicola vulgatus Phocaeicola vulgatus MIC50 0.25 ug.mL-1 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus MIC50 0.25 ug.mL-1 10.1128/aac.00595-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC50 0.25 ug.mL-1 10.1128/aac.00910-07
Phocaeicola vulgatus Phocaeicola vulgatus MIC50 0.25 ug.mL-1 10.1128/aac.01128-07
Phocaeicola vulgatus Phocaeicola vulgatus MIC50 0.5 ug.mL-1 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC50 0.5 ug.mL-1 10.1128/aac.00696-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 1.0 ug.mL-1 10.1128/aac.00910-07
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 1.0 ug.mL-1 10.1128/aac.01128-07
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 1.0 ug.mL-1 10.1128/aac.01435-06
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 2.0 ug.mL-1 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 2.0 ug.mL-1 10.1128/aac.00696-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 4.0 ug.mL-1 10.1128/aac.00595-08
Porphyromonas asaccharolytica Porphyromonas asaccharolytica Activity 0.0 % 10.1128/aac.01128-07
Porphyromonas asaccharolytica Porphyromonas asaccharolytica MIC 0.008 ug.mL-1 10.1128/aac.00481-10
Porphyromonas asaccharolytica Porphyromonas asaccharolytica MIC 0.015 ug.mL-1 10.1128/aac.00595-08
Porphyromonas asaccharolytica Porphyromonas asaccharolytica MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Porphyromonas asaccharolytica Porphyromonas asaccharolytica MIC50 0.015 ug.mL-1 10.1128/aac.00595-08
Porphyromonas asaccharolytica Porphyromonas asaccharolytica MIC50 0.015 ug.mL-1 10.1128/aac.01128-07
Porphyromonas asaccharolytica Porphyromonas asaccharolytica MIC90 0.015 ug.mL-1 10.1128/aac.01128-07
Porphyromonas asaccharolytica Porphyromonas asaccharolytica MIC90 0.03 ug.mL-1 10.1128/aac.00595-08
Porphyromonas gingivalis Porphyromonas gingivalis MIC 0.015 ug.mL-1 10.1128/aac.00595-08
Porphyromonas gingivalis Porphyromonas gingivalis MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Porphyromonas gingivalis Porphyromonas gingivalis MIC50 0.015 ug.mL-1 10.1128/aac.00595-08
Porphyromonas gingivalis Porphyromonas gingivalis MIC90 0.03 ug.mL-1 10.1128/aac.00595-08
Porphyromonas levii Porphyromonas levii MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Porphyromonas somerae Porphyromonas somerae Activity 0.0 % 10.1128/aac.01128-07
Porphyromonas somerae Porphyromonas somerae MIC50 0.015 ug.mL-1 10.1128/aac.01128-07
Porphyromonas somerae Porphyromonas somerae MIC90 0.015 ug.mL-1 10.1128/aac.01128-07
Prevotella bivia Prevotella bivia Activity 0.0 % 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia Activity 0.0 % 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia Activity 0.0 % 10.1128/aac.01128-07
Prevotella bivia Prevotella bivia Activity 100.0 % 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia Activity 100.0 % 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia MIC 0.03 ug.mL-1 10.1128/aac.00910-07
Prevotella bivia Prevotella bivia MIC 0.06 ug.mL-1 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia MIC 0.25 ug.mL-1 10.1128/aac.00595-08
Prevotella bivia Prevotella bivia MIC50 0.06 ug.mL-1 10.1128/aac.00910-07
Prevotella bivia Prevotella bivia MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Prevotella bivia Prevotella bivia MIC50 0.12 ug.mL-1 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia MIC50 0.125 ug.mL-1 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia MIC90 0.125 ug.mL-1 10.1128/aac.00910-07
Prevotella bivia Prevotella bivia MIC90 0.125 ug.mL-1 10.1128/aac.01128-07
Prevotella bivia Prevotella bivia MIC90 0.25 ug.mL-1 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia MIC90 0.5 ug.mL-1 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae Activity 0.0 % 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae Activity 0.0 % 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae Activity 100.0 % 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae Activity 100.0 % 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae MIC 0.06 ug.mL-1 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae MIC 0.06 ug.mL-1 10.1128/aac.00910-07
Prevotella buccae Prevotella buccae MIC 0.25 ug.mL-1 10.1128/aac.00595-08
Prevotella buccae Prevotella buccae MIC50 0.06 ug.mL-1 10.1128/aac.00910-07
Prevotella buccae Prevotella buccae MIC50 0.12 ug.mL-1 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae MIC50 0.125 ug.mL-1 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae MIC90 0.06 ug.mL-1 10.1128/aac.00910-07
Prevotella buccae Prevotella buccae MIC90 0.25 ug.mL-1 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae MIC90 0.5 ug.mL-1 10.1128/aac.00481-10
Prevotella corporis Prevotella corporis MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Prevotella corporis Prevotella corporis MIC 0.03 ug.mL-1 10.1128/aac.00595-08
Prevotella corporis Prevotella corporis MIC50 0.03 ug.mL-1 10.1128/aac.00910-07
Prevotella corporis Prevotella corporis MIC90 0.06 ug.mL-1 10.1128/aac.00910-07
Prevotella denticola Prevotella denticola MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Prevotella denticola Prevotella denticola MIC 0.06 ug.mL-1 10.1128/aac.00595-08
Prevotella denticola Prevotella denticola MIC50 0.06 ug.mL-1 10.1128/aac.00910-07
Prevotella denticola Prevotella denticola MIC90 0.25 ug.mL-1 10.1128/aac.00910-07
Prevotella disiens Prevotella disiens MIC 0.03 ug.mL-1 10.1128/aac.00910-07
Prevotella disiens Prevotella disiens MIC50 0.03 ug.mL-1 10.1128/aac.00910-07
Prevotella disiens Prevotella disiens MIC90 0.125 ug.mL-1 10.1128/aac.00910-07
Prevotella intermedia Prevotella intermedia Activity 0.0 % 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia Activity 0.0 % 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia Activity 90.0 % 10.1128/aac.00910-07
Prevotella intermedia Prevotella intermedia Activity 99.0 % 10.1128/aac.00910-07
Prevotella intermedia Prevotella intermedia Activity 100.0 % 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia Activity 100.0 % 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Prevotella intermedia Prevotella intermedia MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia MIC 0.03 ug.mL-1 10.1128/aac.00910-07
Prevotella intermedia Prevotella intermedia MIC 0.06 ug.mL-1 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia MIC 0.06 ug.mL-1 10.1128/aac.00595-08
Prevotella intermedia Prevotella intermedia MIC50 0.03 ug.mL-1 10.1128/aac.00910-07
Prevotella intermedia Prevotella intermedia MIC50 0.06 ug.mL-1 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia MIC50 0.06 ug.mL-1 10.1128/aac.00595-08
Prevotella intermedia Prevotella intermedia MIC50 0.12 ug.mL-1 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia MIC90 0.06 ug.mL-1 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia MIC90 0.125 ug.mL-1 10.1128/aac.00595-08
Prevotella intermedia Prevotella intermedia MIC90 0.125 ug.mL-1 10.1128/aac.00910-07
Prevotella intermedia Prevotella intermedia MIC90 0.25 ug.mL-1 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica Activity 0.0 % 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica Activity 100.0 % 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Prevotella melaninogenica Prevotella melaninogenica MIC 0.06 ug.mL-1 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica MIC 0.125 ug.mL-1 10.1128/aac.00595-08
Prevotella melaninogenica Prevotella melaninogenica MIC50 0.06 ug.mL-1 10.1128/aac.00910-07
Prevotella melaninogenica Prevotella melaninogenica MIC50 0.12 ug.mL-1 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica MIC50 0.125 ug.mL-1 10.1128/aac.00595-08
Prevotella melaninogenica Prevotella melaninogenica MIC90 0.06 ug.mL-1 10.1128/aac.00910-07
Prevotella melaninogenica Prevotella melaninogenica MIC90 0.25 ug.mL-1 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica MIC90 0.25 ug.mL-1 10.1128/aac.00595-08
Prevotella nigrescens Prevotella nigrescens MIC 0.016 ug.mL-1 10.1128/aac.00910-07
Prevotella nigrescens Prevotella nigrescens MIC50 0.03 ug.mL-1 10.1128/aac.00910-07
Prevotella nigrescens Prevotella nigrescens MIC90 0.06 ug.mL-1 10.1128/aac.00910-07
Priestia megaterium Priestia megaterium MIC 0.05 ug.mL-1 10.1016/j.ejmech.2006.10.006
Priestia megaterium Priestia megaterium MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
Propionibacterium Propionibacterium Activity 0.0 % 10.1128/aac.00696-08
Propionibacterium Propionibacterium MIC 0.06 ug.mL-1 10.1128/aac.00696-08
Propionibacterium Propionibacterium MIC50 0.06 ug.mL-1 10.1128/aac.00696-08
Propionibacterium Propionibacterium MIC90 0.25 ug.mL-1 10.1128/aac.00696-08
Proteus mirabilis Proteus mirabilis Activity 0.0 % 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis Activity 0.0 % 10.1128/aac.00400-09
Proteus mirabilis Proteus mirabilis Activity 0.0 % 10.1128/aac.01128-07
Proteus mirabilis Proteus mirabilis Activity 100.0 % 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis Activity 100.0 % 10.1128/aac.00400-09
Proteus mirabilis Proteus mirabilis Activity 100.0 % 10.1128/aac.01509-06
Proteus mirabilis Proteus mirabilis MIC 0.015 ug.mL-1 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis MIC 0.03 ug.mL-1 10.1128/aac.00336-08
Proteus mirabilis Proteus mirabilis MIC 0.06 ug.mL-1 10.1128/aac.00400-09
Proteus mirabilis Proteus mirabilis MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Proteus mirabilis Proteus mirabilis MIC 0.1 ug.mL-1 10.1016/j.ejmech.2006.10.006
Proteus mirabilis Proteus mirabilis MIC 0.1 ug.mL-1 10.1016/j.ejmech.2007.02.001
Proteus mirabilis Proteus mirabilis MIC 0.12 ug.mL-1 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis MIC 0.25 ug.mL-1 10.1016/j.ejmech.2022.114571
Proteus mirabilis Proteus mirabilis MIC 16.0 ug.mL-1 10.1128/aac.01114-07
Proteus mirabilis Proteus mirabilis MIC50 0.03 ug.mL-1 10.1128/aac.01509-06
Proteus mirabilis Proteus mirabilis MIC50 0.06 ug.mL-1 10.1128/aac.00336-08
Proteus mirabilis Proteus mirabilis MIC50 0.06 ug.mL-1 10.1128/aac.00400-09
Proteus mirabilis Proteus mirabilis MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Proteus mirabilis Proteus mirabilis MIC50 0.12 ug.mL-1 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis MIC50 0.125 ug.mL-1 10.1128/aac.01525-09
Proteus mirabilis Proteus mirabilis MIC90 0.06 ug.mL-1 10.1128/aac.00400-09
Proteus mirabilis Proteus mirabilis MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
Proteus mirabilis Proteus mirabilis MIC90 0.125 ug.mL-1 10.1128/aac.01128-07
Proteus mirabilis Proteus mirabilis MIC90 0.25 ug.mL-1 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis MIC90 0.25 ug.mL-1 10.1128/aac.01509-06
Proteus mirabilis Proteus mirabilis MIC90 0.5 ug.mL-1 10.1128/aac.01525-09
Proteus vulgaris Proteus vulgaris Activity 0.0 % 10.1128/aac.01128-07
Proteus vulgaris Proteus vulgaris MIC 0.015 ug.mL-1 10.1128/aac.00336-08
Proteus vulgaris Proteus vulgaris MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Proteus vulgaris Proteus vulgaris MIC 0.1 ug.mL-1 10.1016/0960-894X(95)00380-C
Proteus vulgaris Proteus vulgaris MIC 0.1 ug.mL-1 10.1016/j.ejmech.2006.10.006
Proteus vulgaris Proteus vulgaris MIC 0.1 ug.mL-1 10.1016/j.ejmech.2007.02.001
Proteus vulgaris Proteus vulgaris MIC 0.1 ug.mL-1 10.1016/S0960-894X(97)00230-8
Proteus vulgaris Proteus vulgaris MIC50 0.03 ug.mL-1 10.1128/aac.00336-08
Proteus vulgaris Proteus vulgaris MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Proteus vulgaris Proteus vulgaris MIC50 0.125 ug.mL-1 10.1128/aac.01525-09
Proteus vulgaris Proteus vulgaris MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
Proteus vulgaris Proteus vulgaris MIC90 0.125 ug.mL-1 10.1128/aac.01128-07
Proteus vulgaris Proteus vulgaris MIC90 0.5 ug.mL-1 10.1128/aac.01525-09
Providencia rettgeri Providencia rettgeri Activity 0.0 % 10.1128/aac.01128-07
Providencia rettgeri Providencia rettgeri MIC 0.05 ug.mL-1 10.1016/j.ejmech.2006.10.006
Providencia rettgeri Providencia rettgeri MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
Providencia rettgeri Providencia rettgeri MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Providencia rettgeri Providencia rettgeri MIC 0.1 ug.mL-1 10.1016/j.ejmech.2006.10.006
Providencia rettgeri Providencia rettgeri MIC 0.1 ug.mL-1 10.1016/j.ejmech.2007.02.001
Providencia rettgeri Providencia rettgeri MIC 32.0 ug.mL-1 10.1128/aac.01312-09
Providencia rettgeri Providencia rettgeri MIC 32.0 ug.mL-1 10.1128/aac.01525-09
Providencia rettgeri Providencia rettgeri MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Providencia rettgeri Providencia rettgeri MIC50 0.25 ug.mL-1 10.1128/aac.01525-09
Providencia rettgeri Providencia rettgeri MIC90 0.125 ug.mL-1 10.1128/aac.01128-07
Providencia rettgeri Providencia rettgeri MIC90 32.0 ug.mL-1 10.1128/aac.01525-09
Providencia stuartii Providencia stuartii MIC 0.015 ug.mL-1 10.1128/aac.00336-08
Providencia stuartii Providencia stuartii MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Providencia stuartii Providencia stuartii MIC 0.12 ug.mL-1 10.1128/aac.00017-09
Providencia stuartii Providencia stuartii MIC 8.0 ug.mL-1 10.1039/C5MD00380F
Providencia stuartii Providencia stuartii MIC 8.0 ug.mL-1 10.1128/aac.00017-09
Providencia stuartii Providencia stuartii MIC50 0.03 ug.mL-1 10.1128/aac.00336-08
Providencia stuartii Providencia stuartii MIC50 0.25 ug.mL-1 10.1128/aac.01525-09
Providencia stuartii Providencia stuartii MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
Providencia stuartii Providencia stuartii MIC90 32.0 ug.mL-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Beta-lactamase Kcat nan None 10.1128/aac.01397-09
Pseudomonas aeruginosa Beta-lactamase Kcat/Km 0.2 /uM/s 10.1128/aac.01397-09
Pseudomonas aeruginosa Beta-lactamase Km nan None 10.1128/aac.01397-09
Pseudomonas aeruginosa Beta-lactamase IMP-1 Activity 9.6 % 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase IMP-1 Activity 31.0 % 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase IMP-1 Kcat 26.0 /s 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase IMP-1 Kcat/Km 4.0 /s/microM 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase IMP-1 Km 6500.0 nM 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase OXA-10 Activity 0.031 % 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase OXA-10 Activity nan None 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase OXA-10 Kcat 0.005 /s 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase OXA-10 Kcat/Km nan None 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase OXA-10 Km nan None 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase VIM-1 Kcat 20.0 /s 10.1128/aac.00465-08
Pseudomonas aeruginosa Beta-lactamase VIM-1 Kcat/Km 2.8 /M/s 10.1128/aac.00465-08
Pseudomonas aeruginosa Beta-lactamase VIM-1 Km 72000.0 nM 10.1128/aac.00465-08
Pseudomonas aeruginosa Beta-lactamase VIM-2 Activity 1.8 % 10.1128/aac.00175-08
Pseudomonas aeruginosa Beta-lactamase VIM-2 Activity 1.8 % 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase VIM-2 Activity 62.0 % 10.1128/aac.00175-08
Pseudomonas aeruginosa Beta-lactamase VIM-2 Activity 62.0 % 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase VIM-2 Kcat 2.1 /s 10.1128/aac.00175-08
Pseudomonas aeruginosa Beta-lactamase VIM-2 Kcat 2.1 /s 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase VIM-2 Kcat 5.0 /s 10.1128/aac.00166-08
Pseudomonas aeruginosa Beta-lactamase VIM-2 Kcat 8.5 /s 10.1128/aac.01397-09
Pseudomonas aeruginosa Beta-lactamase VIM-2 Kcat/Km 0.053 /s/microM 10.1128/aac.00175-08
Pseudomonas aeruginosa Beta-lactamase VIM-2 Kcat/Km 0.053 /s/microM 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase VIM-2 Kcat/Km 0.9 /uM/s 10.1128/aac.01397-09
Pseudomonas aeruginosa Beta-lactamase VIM-2 Kcat/Km 2.5 /uM/s 10.1128/aac.00166-08
Pseudomonas aeruginosa Beta-lactamase VIM-2 Kd 12000.0 nM 10.1021/acs.jmedchem.5b01289
Pseudomonas aeruginosa Beta-lactamase VIM-2 Km 2000.0 nM 10.1021/acs.jmedchem.5b01289
Pseudomonas aeruginosa Beta-lactamase VIM-2 Km 2000.0 nM 10.1128/aac.00166-08
Pseudomonas aeruginosa Beta-lactamase VIM-2 Km 9400.0 nM 10.1128/aac.01397-09
Pseudomonas aeruginosa Beta-lactamase VIM-2 Km 40000.0 nM 10.1128/aac.00175-08
Pseudomonas aeruginosa Beta-lactamase VIM-2 Km 40000.0 nM 10.1128/aac.01004-09
Pseudomonas aeruginosa Beta-lactamase VIM-2 MIC 1.0 ug.mL-1 10.1016/j.bmc.2020.115598
Pseudomonas aeruginosa Beta-lactamase VIM-2 MIC 8.0 ug.mL-1 10.1016/j.bmc.2020.115598
Pseudomonas aeruginosa Beta-lactamase VIM-2 MIC 16.0 ug.mL-1 10.1016/j.bmc.2020.115598
Pseudomonas aeruginosa Beta-lactamase VIM-2 MIC 64.0 ug.mL-1 10.1016/j.bmc.2020.115598
Pseudomonas aeruginosa Class B carbapenemase VIM-13 Kcat 9.0 /s 10.1128/aac.00465-08
Pseudomonas aeruginosa Class B carbapenemase VIM-13 Kcat/Km 5.92 /M/s 10.1128/aac.00465-08
Pseudomonas aeruginosa Class B carbapenemase VIM-13 Km 15500.0 nM 10.1128/aac.00465-08
Pseudomonas aeruginosa Metallo-beta-lactamase VIM-11 Kcat 3.2 /s 10.1128/aac.01025-07
Pseudomonas aeruginosa Metallo-beta-lactamase VIM-11 Kcat/Km 1.4 10'6/M/s 10.1128/aac.01025-07
Pseudomonas aeruginosa Metallo-beta-lactamase VIM-11 Km 22700.0 nM 10.1128/aac.01025-07
Pseudomonas aeruginosa Metallo-beta-lactamase VIM-2 Kcat 3.5 /s 10.1128/aac.01025-07
Pseudomonas aeruginosa Metallo-beta-lactamase VIM-2 Kcat/Km 1.4 10'6/M/s 10.1128/aac.01025-07
Pseudomonas aeruginosa Metallo-beta-lactamase VIM-2 Km 24500.0 nM 10.1128/aac.01025-07
Pseudomonas aeruginosa Metallo-b-lactamase Kcat 42.0 /s 10.1128/aac.00166-08
Pseudomonas aeruginosa Metallo-b-lactamase Kcat/Km 1.1 /uM/s 10.1128/aac.00166-08
Pseudomonas aeruginosa Metallo-b-lactamase Km 38000.0 nM 10.1128/aac.00166-08
Pseudomonas aeruginosa Pseudomonas aeruginosa AAC -22.46 deltalog10CFU/ml.hr 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa AAC -19.58 deltalog10CFU/ml.hr 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa AAC 5.3 deltalog10CFU/ml.hr 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 0.0 % 10.1128/aac.01538-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 0.7 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 1.0 10'-5 ug/ml 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 1.0 10'-7 ug/ml 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 2.0 ug ml-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 2.9 deltalog10CFU 10.1021/acs.jmedchem.6b01903
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 3.0 ug ml-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 3.6 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 3.7 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 4.1 % 10.1128/aac.00400-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 4.2 deltalog10CFU 10.1021/acs.jmedchem.6b01903
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 4.6 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 4.7 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 4.9 deltalog10CFU 10.1021/acs.jmedchem.6b01903
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 6.5 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 7.0 % 10.1128/aac.01128-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 7.9 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 8.1 % 10.1128/aac.00400-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 10.2 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 12.4 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 13.33 % 10.1016/j.ejmech.2020.112252
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 15.67 % 10.1016/j.ejmech.2020.112252
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 16.9 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 17.2 % 10.1128/aac.00851-06
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 18.0 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 32.0 ug ml-1 10.1128/aac.01043-06
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 35.5 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 40.6 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 42.5 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 52.0 % 10.1128/aac.01104-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 52.1 % 10.1128/aac.00834-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 56.1 % 10.1128/aac.00851-06
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 59.5 % 10.1128/aac.01483-06
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 60.9 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 68.0 % 10.1128/aac.00810-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 74.1 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 76.9 % 10.1128/aac.00851-06
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 83.9 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 85.3 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 87.0 % 10.1128/aac.00679-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 87.8 % 10.1128/aac.00400-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 88.8 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 95.0 % 10.1128/aac.00453-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 98.5 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 602.0 mm3 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 810.0 mm3 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 862.0 mm3 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 926.0 mm3 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 992.0 mm3 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 1030.0 mm3 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 1190.0 mm3 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 1316.0 mm3 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity nan None 10.1016/0960-894X(95)00202-5
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity nan None 10.1016/j.ejmech.2020.112252
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity nan None 10.1016/j.ejmech.2022.114278
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity nan None 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity nan None 10.1128/aac.01278-06
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity nan None 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity nan None 10.1128/aac.01529-07
Pseudomonas aeruginosa Pseudomonas aeruginosa deltalog10CFU -1.23 /ml 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa deltalog10CFU -1.1 None 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa deltalog10CFU -1.09 /ml 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa deltalog10CFU -1.0 None 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa deltalog10CFU -0.9 None 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa deltalog10CFU -0.83 /ml 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa deltalog10CFU 0.2 None 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa deltalog10CFU 0.5 None 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa deltalog10CFU 0.7 None 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa FC 0.2 None 10.1021/jm501050e
Pseudomonas aeruginosa Pseudomonas aeruginosa FC 1.0 None 10.1021/acs.jmedchem.1c00888
Pseudomonas aeruginosa Pseudomonas aeruginosa fT>MIC 38.0 % 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa fT>MIC 47.0 % 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa fT>MIC 50.0 % 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa fT>MIC 56.0 % 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa fT>MIC 63.0 % 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa fT>MIC 69.0 % 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa fT>MIC 75.0 % 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa fT>MIC 78.0 % 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa fT>MIC 82.0 % 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa fT>MIC 94.0 % 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa fT>MIC 100.0 % 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa IC50 1.0 ug.mL-1 10.1128/aac.01433-08
Pseudomonas aeruginosa Pseudomonas aeruginosa IC50 20.0 nM 10.1021/acs.jnatprod.9b00187
Pseudomonas aeruginosa Pseudomonas aeruginosa Inhibition 8.16 % 10.6019/CHEMBL4513141
Pseudomonas aeruginosa Pseudomonas aeruginosa Inhibition nan % 10.1128/aac.01452-08
Pseudomonas aeruginosa Pseudomonas aeruginosa IZ 6.0 mm 10.1128/aac.00399-09
Pseudomonas aeruginosa Pseudomonas aeruginosa IZ 16.0 mm 10.1128/aac.00399-09
Pseudomonas aeruginosa Pseudomonas aeruginosa IZ 16.0 mm 10.1128/aac.00893-08
Pseudomonas aeruginosa Pseudomonas aeruginosa IZ 17.0 mm 10.1128/aac.00399-09
Pseudomonas aeruginosa Pseudomonas aeruginosa IZ 18.0 mm 10.1128/aac.00399-09
Pseudomonas aeruginosa Pseudomonas aeruginosa IZ 19.0 mm 10.1128/aac.00399-09
Pseudomonas aeruginosa Pseudomonas aeruginosa IZ 20.0 mm 10.1128/aac.00399-09
Pseudomonas aeruginosa Pseudomonas aeruginosa IZ 21.0 mm 10.1128/aac.00399-09
Pseudomonas aeruginosa Pseudomonas aeruginosa log10cfu 3.0 None 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa log10CFU/g 2.0 None 10.1021/acs.jmedchem.5b00262
Pseudomonas aeruginosa Pseudomonas aeruginosa MBC 0.125 ug ml-1 10.1128/aac.01452-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MBC 1.0 ug ml-1 10.1128/aac.01433-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MBC 1.0 ug ml-1 10.1128/aac.01452-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MBC 2.0 ug ml-1 10.1128/aac.01452-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MBC 2.0 ug ml-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MBC 4.0 ug ml-1 10.1021/acs.jmedchem.2c01469
Pseudomonas aeruginosa Pseudomonas aeruginosa MBC 32.0 ug ml-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 6e-05 ug.mL-1 10.1128/aac.00294-06
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.01 ug.mL-1 10.1128/aac.01451-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.023 ug.mL-1 10.1128/aac.00257-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.03 ug.mL-1 10.1128/aac.00336-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.03 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.03 ug.mL-1 10.1128/aac.00413-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.047 ug.mL-1 10.1128/aac.00257-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.049 ug.mL-1 10.1016/j.bmcl.2003.09.039
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.049 ug.mL-1 10.1016/j.bmcl.2004.09.092
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.049 ug.mL-1 10.1016/s0960-894x(00)00253-5
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.049 ug.mL-1 10.1016/s0960-894x(00)00575-8
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.049 ug.mL-1 10.1016/s0960-894x(01)00451-6
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.049 ug.mL-1 10.1016/s0960-894x(02)00948-4
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.049 ug.mL-1 10.1016/s0960-894x(98)00270-4
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.049 ug.mL-1 10.1016/s0960-894x(99)00407-2
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.049 ug.mL-1 10.1016/s0960-894x(99)00646-0
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.049 ug.mL-1 10.1016/s0960-894x(99)00692-7
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.049 ug.mL-1 10.1021/np060206z
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.05 ug.mL-1 10.1128/aac.01451-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.06 ug.mL-1 10.1016/j.bmcl.2021.127928
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.06 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.06 ug.mL-1 10.1128/aac.00400-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.06 ug.mL-1 10.1128/aac.00816-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.0625 ug.mL-1 10.1016/j.ejmech.2022.114495
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.063 ug.mL-1 10.1016/j.ejmech.2018.06.014
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.064 ug.mL-1 10.1128/aac.00257-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.064 ug.mL-1 10.1128/aac.00912-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.094 ug.mL-1 10.1128/aac.00257-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.098 ug.mL-1 10.1021/np049577a
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.098 ug.mL-1 10.1021/np060206z
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.1 ug.mL-1 10.1021/np020507i
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.12 ug.mL-1 10.1016/j.bmc.2021.116142
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.12 ug.mL-1 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.12 ug.mL-1 10.1128/aac.00689-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.12 ug.mL-1 10.1128/aac.00816-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.12 ug.mL-1 10.1128/aac.01410-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.125 ug.mL-1 10.1016/j.ejmech.2018.06.014
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.125 ug.mL-1 10.1021/acs.jmedchem.6b01903
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.125 ug.mL-1 10.1128/aac.00257-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.125 ug.mL-1 10.1128/aac.00912-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.125 ug.mL-1 10.1128/aac.01452-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.125 ug.mL-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.19 ug.mL-1 10.1128/aac.00257-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.19 ug.mL-1 10.1128/aac.00419-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.195 ug.mL-1 10.1016/j.bmcl.2003.09.039
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.195 ug.mL-1 10.1016/j.bmcl.2004.09.092
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.195 ug.mL-1 10.1016/j.ejmech.2006.10.006
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.195 ug.mL-1 10.1016/s0960-894x(00)00253-5
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.195 ug.mL-1 10.1016/s0960-894x(00)00575-8
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.195 ug.mL-1 10.1016/s0960-894x(01)00451-6
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.195 ug.mL-1 10.1016/s0960-894x(02)00948-4
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.195 ug.mL-1 10.1016/s0960-894x(98)00270-4
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.195 ug.mL-1 10.1016/s0960-894x(99)00407-2
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.195 ug.mL-1 10.1016/s0960-894x(99)00646-0
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.2 ug.mL-1 10.1016/0960-894X(95)00380-C
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.2 ug.mL-1 10.1016/j.ejmech.2006.10.006
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.2 ug.mL-1 10.1016/j.ejmech.2007.02.001
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.2 ug.mL-1 10.1016/S0960-894X(97)00230-8
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.2 ug.mL-1 10.1021/jm010546b
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.2 ug.mL-1 10.1021/np020507i
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.2 ug.mL-1 10.1128/aac.00464-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1016/j.bmcl.2021.127928
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1016/j.ejmech.2018.08.025
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1016/j.ejmech.2020.112252
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1016/S0960-894X(97)00282-5
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1039/C5MD00373C
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00257-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00405-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00415-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00419-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00689-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00816-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00834-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00900-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00912-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.01410-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.01452-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.01529-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.361 ug.mL-1 10.1016/s0960-894x(99)00692-7
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.38 ug.mL-1 10.1128/aac.00257-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.38 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.38 ug.mL-1 10.1128/aac.00419-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.38 ug.mL-1 10.1128/aac.00465-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.38 ug.mL-1 10.1128/aac.00810-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.38 ug.mL-1 10.1128/aac.00822-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.39 ug.mL-1 10.1021/np020507i
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.391 ug.mL-1 10.1021/np060206z
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.4 ug.mL-1 10.1016/j.ejmech.2006.10.006
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.4 ug.mL-1 10.1016/j.ejmech.2007.02.001
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.4 ug.mL-1 10.1021/jm010546b
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1016/j.bmcl.2003.09.039
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1021/acs.jmedchem.6b00746
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1021/acs.jmedchem.6b01742
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1021/ml200012f
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1039/C5MD00373C
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00033-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00174-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00257-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00413-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00419-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00642-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00689-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00816-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00822-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00834-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00912-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.01004-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.01104-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.01172-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.01452-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.01529-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.75 ug.mL-1 10.1128/aac.00174-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.75 ug.mL-1 10.1128/aac.00822-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.8 ug.mL-1 10.1016/j.ejmech.2006.10.006
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.8 ug.mL-1 10.1016/j.ejmech.2007.02.001
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1016/j.bmcl.2003.09.039
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1016/j.bmcl.2021.127928
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1016/j.ejmech.2022.114278
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1021/acs.jmedchem.2c01469
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1021/acs.jmedchem.6b00867
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1021/acs.jmedchem.8b01093
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1021/acs.jmedchem.9b01518
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1021/acsmedchemlett.5b00026
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1039/C5MD00373C
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.00257-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.00413-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.00574-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.00689-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.00816-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.00899-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.00912-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.01104-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.01360-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.01410-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.01433-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.01452-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.5 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.56 ug.mL-1 10.1016/S0960-894X(97)00230-8
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.563 ug.mL-1 10.1016/j.ejmech.2007.02.001
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.6 ug.mL-1 10.1128/aac.00464-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1016/j.bmcl.2021.127928
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1016/j.ejmech.2018.08.025
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1021/acs.jmedchem.1c00888
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1021/jm400560z
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1039/C5MD00373C
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00399-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00413-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00574-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00689-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00816-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00837-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.01004-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.01104-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.01410-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.01433-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 3.0 ug.mL-1 10.1128/aac.00837-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 3.0 ug.mL-1 10.1128/aac.01451-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 3.1 ug.mL-1 10.1128/aac.00464-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1016/j.ejmech.2018.08.025
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1016/S0960-894X(97)00282-5
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1021/acs.jmedchem.5b00262
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1021/acs.jmedchem.6b00867
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1021/np800503z
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1039/C5MD00373C
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00080-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00399-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00413-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00574-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00689-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00816-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00834-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.01104-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.01433-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 6.0 ug.mL-1 10.1128/aac.00822-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 6.0 ug.mL-1 10.1128/aac.00837-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 6.3 ug.mL-1 10.1128/aac.00464-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1016/j.bmc.2013.09.041
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1016/j.bmc.2021.116128
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1016/j.bmcl.2003.09.039
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1016/j.ejmech.2018.08.025
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1016/j.ejmech.2020.112252
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1016/j.ejmech.2022.114278
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1021/acs.jmedchem.6b00867
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1039/C5MD00373C
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.00080-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.00299-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.00399-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.00574-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.00707-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.00810-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.00816-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.00822-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.01011-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.01104-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.01172-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.01433-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.01483-06
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 12.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 12.0 ug.mL-1 10.1128/aac.00465-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 12.5 ug.mL-1 10.1128/aac.00464-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1016/j.bmcl.2021.127928
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1016/j.ejmech.2018.06.014
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1016/j.ejmech.2018.08.025
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.6b00867
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.8b00091
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.9b00720
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1039/C5MD00373C
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00080-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00413-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00574-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00689-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00810-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00816-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00834-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.01172-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.01190-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.01360-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.01433-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 24.0 ug.mL-1 10.1128/aac.01573-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1016/j.bmcl.2021.127928
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.03.058
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.08.025
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1021/acs.jmedchem.2c01469
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1021/acs.jmedchem.6b00867
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1021/acs.jmedchem.6b01261
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1039/C5MD00373C
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1039/C5MD00380F
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00033-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00299-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00465-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00574-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00707-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00816-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00834-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00837-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00900-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01004-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01172-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01230-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01267-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01345-06
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01451-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01561-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01573-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 61.0 ug.mL-1 10.1016/j.ejmech.2018.03.058
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.03.058
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.06.014
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.08.025
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1021/acs.jmedchem.9b00338
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1021/acs.jmedchem.9b01518
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1021/jm400560z
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1039/C5MD00373C
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1039/C5MD00380F
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.00574-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.00734-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.00834-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.01172-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1021/acs.jmedchem.2c01257
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1039/C5MD00380F
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.00175-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.00399-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.00679-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.00689-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.01004-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.01405-06
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 512.0 ug.mL-1 10.1128/aac.01360-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1000.0 nM 10.1021/acs.jmedchem.1c00614
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1000.0 nM 10.1021/acs.jmedchem.1c00621
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2000.0 nM 10.1021/acs.jmedchem.1c02140
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8000.0 nM 10.1021/acs.jmedchem.1c00621
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC nan None 10.1021/acs.jmedchem.6b00867
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 0.5 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 0.5 ug.mL-1 10.1128/aac.00400-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 0.5 ug.mL-1 10.1128/aac.01128-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 1.0 ug.mL-1 10.1021/jm400560z
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 1.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 1.0 ug.mL-1 10.1128/aac.00413-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 2.0 ug.mL-1 10.1016/j.bmcl.2004.09.092
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 2.0 ug.mL-1 10.1021/acs.jmedchem.0c00255
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 2.0 ug.mL-1 10.1021/acs.jmedchem.7b00377
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 2.0 ug.mL-1 10.1128/aac.00912-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 4.0 ug.mL-1 10.1128/aac.00336-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 4.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 4.0 ug.mL-1 10.1128/aac.00912-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 4.0 ug.mL-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 8.0 ug.mL-1 10.1021/acs.jmedchem.9b00338
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 8.0 ug.mL-1 10.1021/ml200012f
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 8.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 8.0 ug.mL-1 10.1128/aac.00912-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 16.0 ug.mL-1 10.1128/aac.00912-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 64.0 ug.mL-1 10.1021/jm400560z
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 0.06 ug.mL-1 10.1039/C1MD00095K
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 0.125 ug.mL-1 10.1039/C1MD00095K
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 0.25 ug.mL-1 10.1016/j.bmcl.2016.06.019
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 0.25 ug.mL-1 10.1039/C1MD00095K
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 0.5 ug.mL-1 10.1016/j.bmcl.2012.07.005
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 0.5 ug.mL-1 10.1039/C1MD00095K
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 1.0 ug.mL-1 10.1039/C1MD00095K
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 2.0 ug.mL-1 10.1039/C1MD00095K
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 2.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 4.0 ug.mL-1 10.1039/C1MD00095K
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 4.0 ug.mL-1 10.1128/aac.01128-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 8.0 ug.mL-1 10.1021/acs.jmedchem.0c00255
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 8.0 ug.mL-1 10.1039/C1MD00095K
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 8.0 ug.mL-1 10.1128/aac.00336-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 8.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 8.0 ug.mL-1 10.1128/aac.00400-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 16.0 ug.mL-1 10.1016/j.bmcl.2004.09.092
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 16.0 ug.mL-1 10.1021/jm400560z
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 16.0 ug.mL-1 10.1039/C1MD00095K
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 16.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 16.0 ug.mL-1 10.1128/aac.00413-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 32.0 ug.mL-1 10.1021/acs.jmedchem.7b00377
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 32.0 ug.mL-1 10.1021/acs.jmedchem.9b00338
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 32.0 ug.mL-1 10.1039/C1MD00095K
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 32.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 32.0 ug.mL-1 10.1128/aac.00912-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 32.0 ug.mL-1 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 64.0 ug.mL-1 10.1016/j.bmcl.2012.07.005
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 64.0 ug.mL-1 10.1021/jm400560z
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 64.0 ug.mL-1 10.1021/ml200012f
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 64.0 ug.mL-1 10.1039/C1MD00095K
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 128.0 ug.mL-1 10.1128/aac.00912-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 nan None 10.1016/j.bmcl.2012.07.005
Pseudomonas aeruginosa Pseudomonas aeruginosa MPC 4.0 ug ml-1 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MPC 8.0 ug ml-1 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MPC 16.0 ug ml-1 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MPC 32.0 ug ml-1 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MPC 64.0 ug ml-1 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa PD50 1.04 mg kg-1 10.1021/ml200012f
Pseudomonas aeruginosa Pseudomonas aeruginosa PD50 1.3 mg kg-1 10.1021/ml200012f
Pseudomonas aeruginosa Pseudomonas aeruginosa PD50 1.76 mg kg-1 10.1016/s0960-894x(98)00270-4
Pseudomonas aeruginosa Pseudomonas aeruginosa Ratio 4.0 None 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa Ratio 8.0 None 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa Ratio 16.0 None 10.1128/aac.00033-10
Pseudomonas aeruginosa Pseudomonas aeruginosa Ratio 32.0 None 10.1016/j.ejmech.2020.112252
Pseudomonas aeruginosa Pseudomonas aeruginosa Survival 23.0 % 10.1039/C5MD00380F
Pseudomonas aeruginosa Pseudomonas aeruginosa Survival 25.0 % 10.1016/j.ejmech.2019.111814
Pseudomonas aeruginosa Pseudomonas aeruginosa TIME 1.5 hr 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa TIME 3.8 hr 10.1128/aac.01525-09
Pseudomonas aeruginosa Pseudomonas aeruginosa TIME 4.1 hr 10.1128/aac.01525-09
Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) Beta-lactamase Activity 0.0063 % 10.1128/aac.01004-09
Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) Beta-lactamase Activity 1.6 % 10.1128/aac.01004-09
Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) Beta-lactamase Kcat 0.006 /s 10.1128/aac.01004-09
Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) Beta-lactamase Kcat/Km 0.0043 /s/microM 10.1128/aac.01004-09
Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) Beta-lactamase Km 1400.0 nM 10.1128/aac.01004-09
Pseudomonas fluorescens Beta-lactamase Kcat/Km 80.0 /mM/s 10.1128/aac.00961-09
Pseudomonas fluorescens Pseudomonas fluorescens MIC 0.12 ug.mL-1 10.1128/aac.00336-08
Pseudomonas fluorescens Pseudomonas fluorescens MIC 16.0 ug.mL-1 10.1128/aac.00961-09
Pseudomonas fluorescens Pseudomonas fluorescens MIC50 2.0 ug.mL-1 10.1128/aac.00336-08
Pseudomonas fluorescens Pseudomonas fluorescens MIC90 32.0 ug.mL-1 10.1128/aac.00336-08
Pseudomonas putida Pseudomonas putida MIC 4.0 ug.mL-1 10.1128/aac.00931-08
Pseudomonas putida Pseudomonas putida MIC 8.0 ug.mL-1 10.1128/aac.00838-06
Pseudomonas putida Pseudomonas putida MIC 32.0 ug.mL-1 10.1128/aac.00707-08
Pseudomonas stutzeri Metallo-beta-lactamase Kcat 4.0 /s 10.1128/aac.01456-09
Pseudomonas stutzeri Metallo-beta-lactamase Km 20000.0 nM 10.1128/aac.01456-09
Pseudomonas stutzeri Metallo-beta-lactamase Ratio 200.0 None 10.1128/aac.01456-09
Rattus norvegicus Aldose reductase IC50 nan None None
Rattus norvegicus Aldose reductase Ki nan None None
Rattus norvegicus Alpha-1a adrenergic receptor IC50 nan None None
Rattus norvegicus Alpha-1a adrenergic receptor Ki nan None None
Rattus norvegicus Alpha-1b adrenergic receptor IC50 nan None None
Rattus norvegicus Alpha-1b adrenergic receptor Ki nan None None
Rattus norvegicus Androgen Receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Androgen Receptor AC50 300000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Androgen Receptor IC50 nan None None
Rattus norvegicus Androgen Receptor Ki nan None None
Rattus norvegicus Cyclooxygenase-1 AC50 33424.5 nM 10.1038/s41467-023-40064-9
Rattus norvegicus GABA receptor alpha-1 subunit AC50 10000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Glutamate (NMDA) receptor subunit zeta 1 AC50 10000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Glycine receptor IC50 nan None None
Rattus norvegicus Glycine receptor Ki nan None None
Rattus norvegicus Insulin receptor IC50 nan None None
Rattus norvegicus Insulin receptor Ki nan None None
Rattus norvegicus Nitric-oxide synthase, brain IC50 nan None None
Rattus norvegicus Nitric-oxide synthase, brain Ki nan None None
Rattus norvegicus Rattus norvegicus ALB 41300.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALB 42700.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALB 43300.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALB 43800.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALB 44700.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALP 317.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALP 336.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALP 367.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALP 370.33 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALP 398.83 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALP 443.33 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALT 43.83 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALT 46.5 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALT 52.33 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALT 52.67 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALT 61.33 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus AST 75.67 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus AST 76.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus AST 76.5 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus AST 81.17 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus AST 85.67 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus AST 86.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus AUC 6383.33 ng.hr.mL-1 10.1016/s0960-894x(00)00253-5
Rattus norvegicus Rattus norvegicus AUC 6383.33 ng.hr.mL-1 10.1016/s0960-894x(01)00451-6
Rattus norvegicus Rattus norvegicus AUC 6383.33 ng.hr.mL-1 10.1016/s0960-894x(02)00948-4
Rattus norvegicus Rattus norvegicus BASO 0.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BASOLE 0.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BILI 1.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BILI 1.5 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BILI 1.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BILI 2.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BUN 133.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BUN 163.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BUN 166.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BUN 176.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BUN 190.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BUN 200.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHLORIDE 99.17 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHLORIDE 99.67 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHLORIDE 101.0 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHLORIDE 101.33 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHLORIDE 101.67 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHOL 606.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHOL 700.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHOL 713.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHOL 740.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHOL 783.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHOL 853.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CK 176.67 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CK 199.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CK 231.83 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CK 254.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CK 300.67 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CK 331.5 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CL 54.16 mL.min-1.kg-1 10.1016/s0960-894x(00)00253-5
Rattus norvegicus Rattus norvegicus CL 54.16 mL.min-1.kg-1 10.1016/s0960-894x(01)00451-6
Rattus norvegicus Rattus norvegicus CL 54.2 mL.min-1.kg-1 10.1016/s0960-894x(02)00948-4
Rattus norvegicus Rattus norvegicus CO2 25330000.0 nM 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CO2 27000000.0 nM 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CO2 27500000.0 nM 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CO2 28330000.0 nM 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CO2 29330000.0 nM 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CREAT 1.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CREAT 2.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CREAT 2.2 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CREAT 2.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CREAT 3.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOS 148.67 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOS 214.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOS 222.83 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOS 276.67 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOS 351.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOS 455.67 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOSLE 1.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOSLE 1.33 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOSLE 2.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOSLE 2.33 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOSLE 2.67 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus GLUC 1543.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus GLUC 1550.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus GLUC 1606.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus GLUC 1610.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus GLUC 1688.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus GLUC 1713.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HCT 34.4 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HCT 35.5 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HCT 35.53 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HCT 35.77 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HCT 36.37 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HCT 36.52 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HGB 131000.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HGB 132700.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HGB 134000.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HGB 134500.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HGB 135300.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HGB 136700.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LDH 71.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LDH 127.33 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LDH 174.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LDH 187.67 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LDH 241.67 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LDH 406.33 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LIPASE 8.67 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LIPASE 9.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LIPASE 9.5 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYM 12444.67 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYM 12982.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYM 13228.33 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYM 14286.67 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYM 14453.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYM 16020.5 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYMLE 85.67 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYMLE 88.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYMLE 89.33 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYMLE 90.5 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYMLE 92.33 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCH 23.22 pg 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCH 23.37 pg 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCH 23.8 pg 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCH 24.03 pg 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCH 24.07 pg 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCHC 368500.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCHC 373700.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCHC 374700.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCHC 376000.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCHC 381000.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCHC 382000.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCV 61.33 fL 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCV 61.92 fL 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCV 62.23 fL 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCV 63.47 fL 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCV 63.97 fL 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCV 64.3 fL 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MONO 0.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MONO 29.17 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MONO 45.33 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MONOLE 0.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MONOLE 0.17 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MONOLE 0.33 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTLE 6.33 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTLE 8.33 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTLE 9.33 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTLE 9.67 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTLE 10.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTLE 11.33 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTSG 841.33 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTSG 1468.33 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTSG 1474.67 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTSG 1490.83 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTSG 1520.67 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTSG 1912.33 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PHOS 114.8 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PHOS 118.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PHOS 119.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PHOS 122.5 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PHOS 122.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PHOS 123.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PLAT 1149330.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PLAT 1178000.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PLAT 1189000.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PLAT 1239500.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PLAT 1255500.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PLAT 1310330.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus POTASSIUM 6.26 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus POTASSIUM 6.33 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus POTASSIUM 6.59 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus POTASSIUM 6.82 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus POTASSIUM 6.87 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PROT 59000.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PROT 59300.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PROT 59800.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PROT 60300.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PROT 63000.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus RBC 5530000.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus RBC 5620000.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus RBC 5690000.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus RBC 5720000.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus RBC 5760000.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus RBC 5780000.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus RBCNUC 0.0 /100WBC 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus RBCNUC 0.17 /100WBC 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus SODIUM 141.28 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus SODIUM 142.3 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus SODIUM 143.0 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus SODIUM 143.8 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus SODIUM 144.6 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus SODIUM 147.07 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus T1/2 0.0665 hr 10.1016/s0960-894x(00)00253-5
Rattus norvegicus Rattus norvegicus T1/2 0.0665 hr 10.1016/s0960-894x(01)00451-6
Rattus norvegicus Rattus norvegicus T1/2 0.0665 hr 10.1016/s0960-894x(02)00948-4
Rattus norvegicus Rattus norvegicus URATE 16.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus URATE 16.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus URATE 18.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus URATE 19.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus URATE 20.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus WBC 13500.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus WBC 14730.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus WBC 15100.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus WBC 16170.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus WBC 16700.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus WBC 17670.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Serotonin 1a (5-HT1a) receptor IC50 nan None None
Rattus norvegicus Serotonin 1a (5-HT1a) receptor Ki nan None None
Rattus norvegicus Serotonin 1b (5-HT1b) receptor IC50 nan None None
Rattus norvegicus Serotonin 1b (5-HT1b) receptor Ki nan None None
Rattus norvegicus Voltage-gated L-type calcium channel alpha-1C subunit AC50 10000.0 nM 10.1038/s41467-023-40064-9
Salmonella Salmonella MIC 0.015 ug.mL-1 10.1128/aac.00336-08
Salmonella Salmonella MIC 0.1 ug.mL-1 10.1016/j.ejmech.2006.10.006
Salmonella Salmonella MIC 0.1 ug.mL-1 10.1016/j.ejmech.2007.02.001
Salmonella Salmonella MIC50 0.03 ug.mL-1 10.1128/aac.00336-08
Salmonella Salmonella MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
Salmonella enterica Salmonella enterica MIC 0.125 ug.mL-1 10.1016/j.ejmech.2018.06.054
Salmonella enterica Salmonella enterica MIC 0.125 ug.mL-1 10.1021/acs.jmedchem.2c01674
Salmonella enterica Salmonella enterica MIC nan None 10.1016/j.ejmech.2017.10.044
Salmonella enterica Salmonella enterica MIC nan None 10.1016/j.ejmech.2017.12.009
Salmonella enterica subsp. enterica serovar Enteritidis Salmonella enteritidis MIC 0.016 ug.mL-1 10.1016/j.bmcl.2003.09.039
Salmonella enterica subsp. enterica serovar Enteritidis Salmonella enteritidis MIC 0.03 ug.mL-1 10.1016/j.bmcl.2003.09.039
Salmonella enterica subsp. enterica serovar Paratyphi A Salmonella paratyphi MIC 0.02 ug.mL-1 10.1016/j.ejmech.2007.02.001
Salmonella enterica subsp. enterica serovar Paratyphi A Salmonella paratyphi MIC 0.03 ug.mL-1 10.1016/j.ejmech.2006.10.006
Salmonella enterica subsp. enterica serovar Typhi Salmonella typhi MIC 0.01 ug.mL-1 10.1016/j.ejmech.2006.10.006
Salmonella enterica subsp. enterica serovar Typhi Salmonella typhi MIC 0.01 ug.mL-1 10.1016/j.ejmech.2007.02.001
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.016 ug.mL-1 10.1016/j.bmcl.2003.09.039
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.025 ug.mL-1 10.1016/j.ejmech.2006.10.006
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.025 ug.mL-1 10.1016/s0960-894x(98)00270-4
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.025 ug.mL-1 10.1016/s0960-894x(99)00407-2
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.03 ug.mL-1 10.1016/j.bmcl.2003.09.039
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.049 ug.mL-1 10.1016/j.bmcl.2003.09.039
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.049 ug.mL-1 10.1016/j.bmcl.2004.09.092
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.049 ug.mL-1 10.1016/s0960-894x(00)00253-5
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.049 ug.mL-1 10.1016/s0960-894x(00)00575-8
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.049 ug.mL-1 10.1016/s0960-894x(01)00451-6
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.049 ug.mL-1 10.1016/s0960-894x(02)00948-4
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.049 ug.mL-1 10.1016/s0960-894x(99)00646-0
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.049 ug.mL-1 10.1016/s0960-894x(99)00692-7
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
Schaalia meyeri Schaalia meyeri Activity 8.0 % 10.1128/aac.00481-10
Schaalia meyeri Schaalia meyeri Activity 92.0 % 10.1128/aac.00481-10
Schaalia meyeri Schaalia meyeri MIC 0.008 ug.mL-1 10.1128/aac.00481-10
Schaalia meyeri Schaalia meyeri MIC50 0.125 ug.mL-1 10.1128/aac.00481-10
Schaalia meyeri Schaalia meyeri MIC90 2.0 ug.mL-1 10.1128/aac.00481-10
Serratia fonticola Carbapenem-hydrolizing beta-lactamase SFC-1 Kcat 6.5 /s 10.1128/aac.00491-07
Serratia fonticola Carbapenem-hydrolizing beta-lactamase SFC-1 Kcat/Km 250.0 /mM/s 10.1128/aac.00491-07
Serratia fonticola Carbapenem-hydrolizing beta-lactamase SFC-1 Km 26000.0 nM 10.1128/aac.00491-07
Serratia marcescens Carbapenem-hydrolyzing beta-lactamase SME-3 Activity 0.27 % 10.1128/aac.01004-09
Serratia marcescens Carbapenem-hydrolyzing beta-lactamase SME-3 Activity 18.0 % 10.1128/aac.01004-09
Serratia marcescens Carbapenem-hydrolyzing beta-lactamase SME-3 Kcat 3.2 /s 10.1128/aac.01004-09
Serratia marcescens Carbapenem-hydrolyzing beta-lactamase SME-3 Kcat/Km 0.55 /s/microM 10.1128/aac.01004-09
Serratia marcescens Carbapenem-hydrolyzing beta-lactamase SME-3 Km 5800.0 nM 10.1128/aac.01004-09
Serratia marcescens Serratia marcescens Activity 0.0 % 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens Activity 0.0 % 10.1128/aac.00400-09
Serratia marcescens Serratia marcescens Activity 0.8 % 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens Activity 99.2 % 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens Activity 100.0 % 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens Activity 100.0 % 10.1128/aac.00400-09
Serratia marcescens Serratia marcescens MIC 0.008 ug.mL-1 10.1128/aac.00768-10
Serratia marcescens Serratia marcescens MIC 0.015 ug.mL-1 10.1128/aac.00336-08
Serratia marcescens Serratia marcescens MIC 0.015 ug.mL-1 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens MIC 0.015 ug.mL-1 10.1128/aac.00768-10
Serratia marcescens Serratia marcescens MIC 0.03 ug.mL-1 10.1128/aac.01004-09
Serratia marcescens Serratia marcescens MIC 0.049 ug.mL-1 10.1016/j.ejmech.2007.02.001
Serratia marcescens Serratia marcescens MIC 0.05 ug.mL-1 10.1016/j.ejmech.2006.10.006
Serratia marcescens Serratia marcescens MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
Serratia marcescens Serratia marcescens MIC 0.06 ug.mL-1 10.1021/jm010546b
Serratia marcescens Serratia marcescens MIC 0.06 ug.mL-1 10.1021/np800503z
Serratia marcescens Serratia marcescens MIC 0.06 ug.mL-1 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens MIC 0.06 ug.mL-1 10.1128/aac.00400-09
Serratia marcescens Serratia marcescens MIC 0.06 ug.mL-1 10.1128/aac.01525-09
Serratia marcescens Serratia marcescens MIC 0.125 ug.mL-1 10.1128/aac.01525-09
Serratia marcescens Serratia marcescens MIC 0.2 ug.mL-1 10.1016/j.ejmech.2006.10.006
Serratia marcescens Serratia marcescens MIC 0.2 ug.mL-1 10.1016/j.ejmech.2007.02.001
Serratia marcescens Serratia marcescens MIC 0.25 ug.mL-1 10.1128/aac.00768-10
Serratia marcescens Serratia marcescens MIC 1.0 ug.mL-1 10.1128/aac.00768-10
Serratia marcescens Serratia marcescens MIC 2.0 ug.mL-1 10.1128/aac.01539-07
Serratia marcescens Serratia marcescens MIC 8.0 ug.mL-1 10.1128/aac.00309-07
Serratia marcescens Serratia marcescens MIC 8.0 ug.mL-1 10.1128/aac.00768-10
Serratia marcescens Serratia marcescens MIC 16.0 ug.mL-1 10.1128/aac.00768-10
Serratia marcescens Serratia marcescens MIC 32.0 ug.mL-1 10.1128/aac.00768-10
Serratia marcescens Serratia marcescens MIC 32.0 ug.mL-1 10.1128/aac.01525-09
Serratia marcescens Serratia marcescens MIC 128.0 ug.mL-1 10.1128/aac.01004-09
Serratia marcescens Serratia marcescens MIC50 0.03 ug.mL-1 10.1128/aac.00336-08
Serratia marcescens Serratia marcescens MIC50 0.06 ug.mL-1 10.1021/ml200012f
Serratia marcescens Serratia marcescens MIC50 0.06 ug.mL-1 10.1128/aac.00400-09
Serratia marcescens Serratia marcescens MIC50 0.12 ug.mL-1 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens MIC50 0.125 ug.mL-1 10.1128/aac.01525-09
Serratia marcescens Serratia marcescens MIC50 0.25 ug.mL-1 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens MIC90 0.06 ug.mL-1 10.1128/aac.00400-09
Serratia marcescens Serratia marcescens MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
Serratia marcescens Serratia marcescens MIC90 0.25 ug.mL-1 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens MIC90 4.0 ug.mL-1 10.1128/aac.01525-09
Serratia marcescens Serratia marcescens MIC90 64.0 ug.mL-1 10.1021/ml200012f
Severe acute respiratory syndrome coronavirus 2 Replicase polyprotein 1ab Inhibition -4.064 % 10.6019/CHEMBL4495564
Severe acute respiratory syndrome coronavirus 2 Replicase polyprotein 1ab Inhibition 10.85 % 10.6019/CHEMBL4495564
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 IC50 19952.62 nM 10.6019/CHEMBL4651402
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 IC50 20000.0 nM 10.6019/CHEMBL4651402
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Inhibition -0.09 % 10.6019/CHEMBL4495565
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Inhibition 0.12 % 10.6019/CHEMBL4495565
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Inhibition 10.13 % 10.21203/rs.3.rs-23951/v1
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Inhibition index 0.4369 None 10.1101/2020.04.03.023846
Shigella flexneri Shigella flexneri MIC 0.03 ug.mL-1 10.1016/j.bmcl.2003.09.039
Shigella sonnei Shigella sonnei MIC 0.03 ug.mL-1 10.1016/j.bmcl.2003.09.039
Shigella sonnei Shigella sonnei MIC 0.5 ug.mL-1 10.1128/aac.00227-08
Staphylococcus Staphylococcus Activity 99.4 % 10.1128/aac.00381-08
Staphylococcus Staphylococcus MIC 0.098 ug.mL-1 10.1016/j.ejmech.2007.02.001
Staphylococcus Staphylococcus MIC50 0.06 ug.mL-1 10.1128/aac.00381-08
Staphylococcus Staphylococcus MIC50 0.12 ug.mL-1 10.1128/aac.00381-08
Staphylococcus Staphylococcus MIC50 2.0 ug.mL-1 10.1128/aac.00381-08
Staphylococcus Staphylococcus MIC50 16.0 ug.mL-1 10.1128/aac.00381-08
Staphylococcus aureus MecA IC50 53.0 ug.mL-1 10.1128/aac.00413-08
Staphylococcus aureus MecA IC50 130.0 ug.mL-1 10.1128/aac.00413-08
Staphylococcus aureus Staphylococcus aureus Activity 0.0 % 10.1128/aac.01128-07
Staphylococcus aureus Staphylococcus aureus Activity 0.0 % 10.1128/aac.01351-07
Staphylococcus aureus Staphylococcus aureus Activity 0.0 % 10.1128/aac.01538-07
Staphylococcus aureus Staphylococcus aureus Activity 98.0 % 10.1128/aac.01351-07
Staphylococcus aureus Staphylococcus aureus Activity 100.0 % 10.1128/aac.00381-08
Staphylococcus aureus Staphylococcus aureus Activity 100.0 % 10.1128/aac.01128-07
Staphylococcus aureus Staphylococcus aureus Activity 100.0 % 10.1128/aac.01538-07
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1016/j.ejmech.2022.114278
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1021/acsmedchemlett.1c00648
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.01192-06
Staphylococcus aureus Staphylococcus aureus EC50 0.14 ug.mL-1 10.1128/aac.01192-06
Staphylococcus aureus Staphylococcus aureus EC50 0.16 ug.mL-1 10.1128/aac.01192-06
Staphylococcus aureus Staphylococcus aureus EC50 0.2 ug.mL-1 10.1128/aac.01192-06
Staphylococcus aureus Staphylococcus aureus EC50 0.29 ug.mL-1 10.1128/aac.01192-06
Staphylococcus aureus Staphylococcus aureus EC50 0.33 ug.mL-1 10.1128/aac.01192-06
Staphylococcus aureus Staphylococcus aureus EC50 nan None 10.1128/aac.01192-06
Staphylococcus aureus Staphylococcus aureus FIC 2.0 None 10.1021/acs.jnatprod.2c00621
Staphylococcus aureus Staphylococcus aureus IC50 0.06 ug.mL-1 10.1128/aac.01433-08
Staphylococcus aureus Staphylococcus aureus IC50 10.0 nM 10.1021/acs.jnatprod.9b00187
Staphylococcus aureus Staphylococcus aureus Inhibition -14.17 % 10.6019/CHEMBL4513141
Staphylococcus aureus Staphylococcus aureus MBC 0.12 ug ml-1 10.1128/aac.01433-08
Staphylococcus aureus Staphylococcus aureus MBC 8.0 ug ml-1 10.1021/acs.jmedchem.2c01469
Staphylococcus aureus Staphylococcus aureus MIC 6e-05 ug.mL-1 10.1128/aac.00294-06
Staphylococcus aureus Staphylococcus aureus MIC 0.013 ug.mL-1 10.1016/s0960-894x(99)00692-7
Staphylococcus aureus Staphylococcus aureus MIC 0.049 ug.mL-1 10.1021/np049577a
Staphylococcus aureus Staphylococcus aureus MIC 0.049 ug.mL-1 10.1021/np060206z
Staphylococcus aureus Staphylococcus aureus MIC 0.05 ug.mL-1 10.1016/j.ejmech.2006.10.006
Staphylococcus aureus Staphylococcus aureus MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
Staphylococcus aureus Staphylococcus aureus MIC 0.06 ug.mL-1 10.1016/j.ejmech.2021.113402
Staphylococcus aureus Staphylococcus aureus MIC 0.06 ug.mL-1 10.1016/S0960-894X(97)00282-5
Staphylococcus aureus Staphylococcus aureus MIC 0.06 ug.mL-1 10.1021/acs.jmedchem.9b01518
Staphylococcus aureus Staphylococcus aureus MIC 0.06 ug.mL-1 10.1039/D1MD00230A
Staphylococcus aureus Staphylococcus aureus MIC 0.06 ug.mL-1 10.1128/aac.01433-08
Staphylococcus aureus Staphylococcus aureus MIC 0.0625 ug.mL-1 10.1016/j.ejmech.2020.112996
Staphylococcus aureus Staphylococcus aureus MIC 0.0625 ug.mL-1 10.1016/j.ejmech.2022.114495
Staphylococcus aureus Staphylococcus aureus MIC 0.098 ug.mL-1 10.1016/j.bmcl.2003.09.039
Staphylococcus aureus Staphylococcus aureus MIC 0.098 ug.mL-1 10.1016/j.ejmech.2006.10.006
Staphylococcus aureus Staphylococcus aureus MIC 0.098 ug.mL-1 10.1016/s0960-894x(00)00253-5
Staphylococcus aureus Staphylococcus aureus MIC 0.098 ug.mL-1 10.1016/s0960-894x(00)00575-8
Staphylococcus aureus Staphylococcus aureus MIC 0.098 ug.mL-1 10.1016/s0960-894x(01)00451-6
Staphylococcus aureus Staphylococcus aureus MIC 0.098 ug.mL-1 10.1016/s0960-894x(02)00948-4
Staphylococcus aureus Staphylococcus aureus MIC 0.098 ug.mL-1 10.1016/s0960-894x(98)00270-4
Staphylococcus aureus Staphylococcus aureus MIC 0.098 ug.mL-1 10.1016/s0960-894x(99)00407-2
Staphylococcus aureus Staphylococcus aureus MIC 0.098 ug.mL-1 10.1016/s0960-894x(99)00646-0
Staphylococcus aureus Staphylococcus aureus MIC 0.098 ug.mL-1 10.1021/np049577a
Staphylococcus aureus Staphylococcus aureus MIC 0.098 ug.mL-1 10.1021/np060206z
Staphylococcus aureus Staphylococcus aureus MIC 0.1 ug.mL-1 10.1016/0960-894X(95)00380-C
Staphylococcus aureus Staphylococcus aureus MIC 0.1 ug.mL-1 10.1016/j.ejmech.2006.10.006
Staphylococcus aureus Staphylococcus aureus MIC 0.1 ug.mL-1 10.1016/j.ejmech.2007.02.001
Staphylococcus aureus Staphylococcus aureus MIC 0.1 ug.mL-1 10.1016/S0960-894X(97)00230-8
Staphylococcus aureus Staphylococcus aureus MIC 0.1 ug.mL-1 10.1021/jm010546b
Staphylococcus aureus Staphylococcus aureus MIC 0.12 ug.mL-1 10.1016/j.ejmech.2021.113402
Staphylococcus aureus Staphylococcus aureus MIC 0.12 ug.mL-1 10.1039/D1MD00230A
Staphylococcus aureus Staphylococcus aureus MIC 0.12 ug.mL-1 10.1128/aac.01433-08
Staphylococcus aureus Staphylococcus aureus MIC 0.125 ug.mL-1 10.1016/j.ejmech.2018.06.054
Staphylococcus aureus Staphylococcus aureus MIC 0.125 ug.mL-1 10.1021/acs.jmedchem.6b00746
Staphylococcus aureus Staphylococcus aureus MIC 0.13 ug.mL-1 10.1016/j.ejmech.2018.11.052
Staphylococcus aureus Staphylococcus aureus MIC 0.19 ug.mL-1 10.1016/S0960-894X(01)80919-7
Staphylococcus aureus Staphylococcus aureus MIC 0.195 ug.mL-1 10.1016/j.bmcl.2003.09.039
Staphylococcus aureus Staphylococcus aureus MIC 0.195 ug.mL-1 10.1016/j.bmcl.2004.09.092
Staphylococcus aureus Staphylococcus aureus MIC 0.195 ug.mL-1 10.1016/s0960-894x(00)00253-5
Staphylococcus aureus Staphylococcus aureus MIC 0.195 ug.mL-1 10.1016/s0960-894x(00)00575-8
Staphylococcus aureus Staphylococcus aureus MIC 0.195 ug.mL-1 10.1016/s0960-894x(01)00451-6
Staphylococcus aureus Staphylococcus aureus MIC 0.195 ug.mL-1 10.1016/s0960-894x(02)00948-4
Staphylococcus aureus Staphylococcus aureus MIC 0.195 ug.mL-1 10.1016/s0960-894x(99)00646-0
Staphylococcus aureus Staphylococcus aureus MIC 0.195 ug.mL-1 10.1016/s0960-894x(99)00692-7
Staphylococcus aureus Staphylococcus aureus MIC 0.195 ug.mL-1 10.1021/np049577a
Staphylococcus aureus Staphylococcus aureus MIC 0.25 ug.mL-1 10.1016/j.ejmech.2019.04.067
Staphylococcus aureus Staphylococcus aureus MIC 0.25 ug.mL-1 10.1021/np800503z
Staphylococcus aureus Staphylococcus aureus MIC 0.25 ug.mL-1 10.1128/aac.01433-08
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1016/j.bmcl.2015.04.046
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1016/j.ejmech.2018.11.052
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1016/j.ejmech.2019.04.067
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1128/aac.01351-07
Staphylococcus aureus Staphylococcus aureus MIC 0.78 ug.mL-1 10.1016/j.bmc.2016.02.013
Staphylococcus aureus Staphylococcus aureus MIC 1.0 ug.mL-1 10.1016/j.bmcl.2015.04.046
Staphylococcus aureus Staphylococcus aureus MIC 1.0 ug.mL-1 10.1016/j.ejmech.2007.03.023
Staphylococcus aureus Staphylococcus aureus MIC 1.0 ug.mL-1 10.1016/j.ejmech.2018.11.052
Staphylococcus aureus Staphylococcus aureus MIC 1.0 ug.mL-1 10.1016/j.ejmech.2020.112996
Staphylococcus aureus Staphylococcus aureus MIC 1.0 ug.mL-1 10.1021/acs.jnatprod.1c00578
Staphylococcus aureus Staphylococcus aureus MIC 1.0 ug.mL-1 10.1021/acs.jnatprod.2c00621
Staphylococcus aureus Staphylococcus aureus MIC 1.56 ug.mL-1 10.1016/S0960-894X(01)80919-7
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1016/j.ejmech.2018.11.052
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1016/j.ejmech.2021.113402
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1016/j.ejmech.2022.114278
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1021/acs.jmedchem.2c01469
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1021/acs.jmedchem.6b00746
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1021/acs.jnatprod.2c00621
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1039/D1MD00230A
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1128/aac.00413-08
Staphylococcus aureus Staphylococcus aureus MIC 3.1 ug.mL-1 10.1021/np030162j
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1016/j.bmcl.2015.04.046
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1016/j.ejmech.2018.08.070
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1016/j.ejmech.2018.11.052
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1016/j.ejmech.2019.04.067
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1016/j.ejmech.2020.112996
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1016/j.ejmech.2021.113402
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1021/np800503z
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1039/D1MD00230A
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1128/aac.01433-08
Staphylococcus aureus Staphylococcus aureus MIC 6.25 ug.mL-1 10.1016/j.ejmech.2007.02.001
Staphylococcus aureus Staphylococcus aureus MIC 8.0 ug.mL-1 10.1016/j.ejmech.2018.11.052
Staphylococcus aureus Staphylococcus aureus MIC 8.0 ug.mL-1 10.1016/j.ejmech.2020.112996
Staphylococcus aureus Staphylococcus aureus MIC 8.0 ug.mL-1 10.1016/j.ejmech.2021.113402
Staphylococcus aureus Staphylococcus aureus MIC 8.0 ug.mL-1 10.1016/S0960-894X(97)00282-5
Staphylococcus aureus Staphylococcus aureus MIC 8.0 ug.mL-1 10.1039/D1MD00230A
Staphylococcus aureus Staphylococcus aureus MIC 8.0 ug.mL-1 10.1128/aac.01433-08
Staphylococcus aureus Staphylococcus aureus MIC 16.0 ug.mL-1 10.1016/j.bmcl.2015.04.046
Staphylococcus aureus Staphylococcus aureus MIC 16.0 ug.mL-1 10.1016/j.ejmech.2018.08.070
Staphylococcus aureus Staphylococcus aureus MIC 16.0 ug.mL-1 10.1016/j.ejmech.2018.11.052
Staphylococcus aureus Staphylococcus aureus MIC 16.0 ug.mL-1 10.1016/j.ejmech.2019.04.067
Staphylococcus aureus Staphylococcus aureus MIC 16.0 ug.mL-1 10.1016/j.ejmech.2020.112996
Staphylococcus aureus Staphylococcus aureus MIC 16.0 ug.mL-1 10.1128/aac.00413-08
Staphylococcus aureus Staphylococcus aureus MIC 25.0 ug.mL-1 10.1016/0960-894X(95)00380-C
Staphylococcus aureus Staphylococcus aureus MIC 25.0 ug.mL-1 10.1016/S0960-894X(01)80919-7
Staphylococcus aureus Staphylococcus aureus MIC 25.0 ug.mL-1 10.1016/S0960-894X(97)00230-8
Staphylococcus aureus Staphylococcus aureus MIC 25.0 ug.mL-1 10.1021/np030162j
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1016/j.bmcl.2015.04.046
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.06.054
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.11.052
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1016/j.ejmech.2019.04.067
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1016/j.ejmech.2020.112996
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1021/acs.jmedchem.2c01469
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1021/acs.jmedchem.9b01518
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1128/aac.00413-08
Staphylococcus aureus Staphylococcus aureus MIC 50.0 ug.mL-1 10.1021/np030162j
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1016/j.bmc.2021.116128
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.06.054
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.08.070
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.11.052
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1016/j.ejmech.2019.04.067
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1016/j.ejmech.2020.112996
Staphylococcus aureus Staphylococcus aureus MIC 100.0 ug.mL-1 10.1016/S0960-894X(01)80919-7
Staphylococcus aureus Staphylococcus aureus MIC 1000.0 nM 10.1021/acs.jmedchem.1c00614
Staphylococcus aureus Staphylococcus aureus MIC 1000.0 nM 10.1021/acs.jmedchem.1c02140
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1016/j.ejmech.2017.10.044
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1016/j.ejmech.2017.12.009
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1021/acs.jmedchem.2c01674
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1021/np800503z
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1128/aac.00642-09
Staphylococcus aureus Staphylococcus aureus MIC50 0.06 ug.mL-1 10.1128/aac.00381-08
Staphylococcus aureus Staphylococcus aureus MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Staphylococcus aureus Staphylococcus aureus MIC50 0.12 ug.mL-1 10.1128/aac.00381-08
Staphylococcus aureus Staphylococcus aureus MIC50 1.0 ug.mL-1 10.1128/aac.00381-08
Staphylococcus aureus Staphylococcus aureus MIC50 2.0 ug.mL-1 10.1128/aac.01128-07
Staphylococcus aureus Staphylococcus aureus MIC50 2.0 ug.mL-1 10.1128/aac.01351-07
Staphylococcus aureus Staphylococcus aureus MIC50 8.0 ug.mL-1 10.1128/aac.00381-08
Staphylococcus aureus Staphylococcus aureus MIC50 8.0 ug.mL-1 10.1128/aac.00413-08
Staphylococcus aureus Staphylococcus aureus MIC90 0.06 ug.mL-1 10.1016/j.bmcl.2016.06.019
Staphylococcus aureus Staphylococcus aureus MIC90 0.125 ug.mL-1 10.1128/aac.01128-07
Staphylococcus aureus Staphylococcus aureus MIC90 2.0 ug.mL-1 10.1128/aac.01351-07
Staphylococcus aureus Staphylococcus aureus MIC90 16.0 ug.mL-1 10.1128/aac.01128-07
Staphylococcus aureus Staphylococcus aureus MIC90 32.0 ug.mL-1 10.1128/aac.00413-08
Staphylococcus chromogenes Staphylococcus chromogenes MIC 0.0625 ug.mL-1 10.1016/j.ejmech.2022.114495
Staphylococcus epidermidis Staphylococcus epidermidis Activity 0.0 % 10.1128/aac.01538-07
Staphylococcus epidermidis Staphylococcus epidermidis Activity 1.8 % 10.1128/aac.01538-07
Staphylococcus epidermidis Staphylococcus epidermidis Activity 9.3 % 10.1128/aac.01538-07
Staphylococcus epidermidis Staphylococcus epidermidis Activity 29.2 % 10.1128/aac.01538-07
Staphylococcus epidermidis Staphylococcus epidermidis Activity 67.0 % 10.1128/aac.01128-07
Staphylococcus epidermidis Staphylococcus epidermidis Activity 100.0 % 10.1128/aac.01538-07
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.8 ug.mL-1 10.1021/np030162j
Staphylococcus epidermidis Staphylococcus epidermidis MIC 1.6 ug.mL-1 10.1021/np030162j
Staphylococcus epidermidis Staphylococcus epidermidis MIC 1000.0 nM 10.1021/acs.jmedchem.1c00614
Staphylococcus epidermidis Staphylococcus epidermidis MIC 1000.0 nM 10.1021/acs.jmedchem.1c02140
Staphylococcus epidermidis Staphylococcus epidermidis MIC50 1.0 ug.mL-1 10.1128/aac.01128-07
Staphylococcus epidermidis Staphylococcus epidermidis MIC90 4.0 ug.mL-1 10.1128/aac.01128-07
Staphylococcus haemolyticus Staphylococcus haemolyticus Activity 73.0 % 10.1128/aac.01128-07
Staphylococcus haemolyticus Staphylococcus haemolyticus MIC50 1.0 ug.mL-1 10.1128/aac.01128-07
Staphylococcus haemolyticus Staphylococcus haemolyticus MIC90 32.0 ug.mL-1 10.1128/aac.01128-07
Staphylococcus lugdunensis Staphylococcus lugdunensis Activity 0.0 % 10.1128/aac.01128-07
Staphylococcus lugdunensis Staphylococcus lugdunensis MIC50 0.25 ug.mL-1 10.1128/aac.01128-07
Staphylococcus lugdunensis Staphylococcus lugdunensis MIC90 0.5 ug.mL-1 10.1128/aac.01128-07
Stenotrophomonas maltophilia Beta-lactamase L1 Kcat/Km 4.5 10'6/M/s 10.1128/aac.01062-07
Stenotrophomonas maltophilia Stenotrophomonas maltophilia Activity nan None 10.1128/aac.01525-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MBC 16.0 ug ml-1 10.1128/aac.01525-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 0.06 ug.mL-1 10.1128/aac.00400-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 0.12 ug.mL-1 10.1128/aac.00336-08
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 0.25 ug.mL-1 10.1128/aac.01525-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 0.38 ug.mL-1 10.1128/aac.01283-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 0.5 ug.mL-1 10.1128/aac.00682-07
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 0.5 ug.mL-1 10.1128/aac.01283-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 0.75 ug.mL-1 10.1128/aac.01283-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 4.0 ug.mL-1 10.1128/aac.01485-07
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 32.0 ug.mL-1 10.1128/aac.00682-07
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 32.0 ug.mL-1 10.1128/aac.01283-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 32.0 ug.mL-1 10.1128/aac.01513-08
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 32.0 ug.mL-1 10.1128/aac.01525-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.06.014
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 64.0 ug.mL-1 10.1128/aac.01485-07
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 100.0 ug.mL-1 10.1021/jm010546b
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 128.0 ug.mL-1 10.1016/j.bmc.2013.09.041
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 128.0 ug.mL-1 10.1016/S0960-894X(97)00282-5
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC50 2.0 ug.mL-1 10.1128/aac.00336-08
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC50 8.0 ug.mL-1 10.1128/aac.01525-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC50 64.0 ug.mL-1 10.1021/ml200012f
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC50 64.0 ug.mL-1 10.1128/aac.00400-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC90 32.0 ug.mL-1 10.1128/aac.00336-08
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC90 32.0 ug.mL-1 10.1128/aac.01525-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC90 64.0 ug.mL-1 10.1021/ml200012f
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC90 64.0 ug.mL-1 10.1128/aac.00400-09
Streptococcus Streptococcus EC50 1154.0 nM None
Streptococcus agalactiae Streptococcus agalactiae Activity 0.0 % 10.1128/aac.01128-07
Streptococcus agalactiae Streptococcus agalactiae MIC 0.03 ug.mL-1 10.1128/aac.00185-08
Streptococcus agalactiae Streptococcus agalactiae MIC 0.031 ug.mL-1 10.1128/aac.01716-08
Streptococcus agalactiae Streptococcus agalactiae MIC 0.049 ug.mL-1 10.1016/j.ejmech.2007.02.001
Streptococcus agalactiae Streptococcus agalactiae MIC 0.05 ug.mL-1 10.1016/j.ejmech.2006.10.006
Streptococcus agalactiae Streptococcus agalactiae MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
Streptococcus agalactiae Streptococcus agalactiae MIC 0.06 ug.mL-1 10.1128/aac.00185-08
Streptococcus agalactiae Streptococcus agalactiae MIC 0.12 ug.mL-1 10.1128/aac.00185-08
Streptococcus agalactiae Streptococcus agalactiae MIC 0.25 ug.mL-1 10.1128/aac.00185-08
Streptococcus agalactiae Streptococcus agalactiae MIC50 0.06 ug.mL-1 10.1128/aac.01128-07
Streptococcus agalactiae Streptococcus agalactiae MIC50 0.063 ug.mL-1 10.1128/aac.01716-08
Streptococcus agalactiae Streptococcus agalactiae MIC90 0.06 ug.mL-1 10.1128/aac.01128-07
Streptococcus agalactiae Streptococcus agalactiae MIC90 0.063 ug.mL-1 10.1128/aac.01716-08
Streptococcus constellatus Streptococcus constellatus MIC 0.05 ug.mL-1 10.1128/aac.00595-08
Streptococcus dysgalactiae Streptococcus dysgalactiae MIC 8.0 ug.mL-1 10.1016/j.ejmech.2022.114495
Streptococcus dysgalactiae subsp. equisimilis Streptococcus dysgalactiae subsp. equisimilis Activity 0.0 % 10.1128/aac.01128-07
Streptococcus dysgalactiae subsp. equisimilis Streptococcus dysgalactiae subsp. equisimilis MIC50 0.015 ug.mL-1 10.1128/aac.01128-07
Streptococcus dysgalactiae subsp. equisimilis Streptococcus dysgalactiae subsp. equisimilis MIC90 0.015 ug.mL-1 10.1128/aac.01128-07
Streptococcus intermedius Streptococcus intermedius MIC 0.25 ug.mL-1 10.1128/aac.00595-08
Streptococcus pneumoniae Streptococcus pneumoniae Activity 0.0 % 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae Activity 0.0 % 10.1128/aac.01538-07
Streptococcus pneumoniae Streptococcus pneumoniae Activity 0.4 % 10.1128/aac.01384-06
Streptococcus pneumoniae Streptococcus pneumoniae Activity 0.4 % 10.1128/aac.01538-07
Streptococcus pneumoniae Streptococcus pneumoniae Activity 0.5 % 10.1128/aac.01538-07
Streptococcus pneumoniae Streptococcus pneumoniae Activity 2.3 % 10.1128/aac.00381-08
Streptococcus pneumoniae Streptococcus pneumoniae Activity 4.5 % 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae Activity 9.5 % 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae Activity 33.3 % 10.1128/aac.01268-09
Streptococcus pneumoniae Streptococcus pneumoniae Activity 34.3 % 10.1128/aac.01268-09
Streptococcus pneumoniae Streptococcus pneumoniae Activity 59.5 % 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae Activity 75.9 % 10.1128/aac.01387-07
Streptococcus pneumoniae Streptococcus pneumoniae Activity 83.2 % 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae Activity 83.9 % 10.1128/aac.00381-08
Streptococcus pneumoniae Streptococcus pneumoniae Activity 86.8 % 10.1128/aac.01384-06
Streptococcus pneumoniae Streptococcus pneumoniae Activity 93.2 % 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae Activity 100.0 % 10.1128/aac.00381-08
Streptococcus pneumoniae Streptococcus pneumoniae Activity 100.0 % 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC 6e-05 ug.mL-1 10.1128/aac.00294-06
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.008 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.01 ug.mL-1 10.1016/j.ejmech.2007.02.001
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.015 ug.mL-1 10.1021/np800503z
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.016 ug.mL-1 10.1021/acs.jmedchem.6b00746
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.016 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.03 ug.mL-1 10.1128/aac.01387-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.06 ug.mL-1 10.1128/aac.00185-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.06 ug.mL-1 10.1128/aac.01082-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.06 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.12 ug.mL-1 10.1128/aac.01082-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.12 ug.mL-1 10.1128/aac.01324-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.12 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.125 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.25 ug.mL-1 10.1016/j.bmc.2020.115776
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.25 ug.mL-1 10.1128/aac.01082-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.25 ug.mL-1 10.1128/aac.01268-09
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.25 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.5 ug.mL-1 10.1128/aac.01082-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.5 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 1.0 ug.mL-1 10.1021/np800503z
Streptococcus pneumoniae Streptococcus pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.015 ug.mL-1 10.1128/aac.00381-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.015 ug.mL-1 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.015 ug.mL-1 10.1128/aac.01384-06
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.016 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.06 ug.mL-1 10.1128/aac.00381-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.06 ug.mL-1 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.06 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.5 ug.mL-1 10.1016/j.bmc.2020.115776
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.5 ug.mL-1 10.1016/j.bmcl.2004.09.092
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.5 ug.mL-1 10.1128/aac.00381-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.5 ug.mL-1 10.1128/aac.01268-09
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.5 ug.mL-1 10.1128/aac.01387-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.5 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 1.0 ug.mL-1 10.1128/aac.00381-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 1.0 ug.mL-1 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 1.0 ug.mL-1 10.1128/aac.01324-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 1.0 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.015 ug.mL-1 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.016 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.25 ug.mL-1 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.25 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.5 ug.mL-1 10.1016/j.bmcl.2004.09.092
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.5 ug.mL-1 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.5 ug.mL-1 10.1128/aac.01384-06
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.5 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 1.0 ug.mL-1 10.1016/j.bmc.2020.115776
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 1.0 ug.mL-1 10.1128/aac.00971-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 1.0 ug.mL-1 10.1128/aac.01268-09
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 1.0 ug.mL-1 10.1128/aac.01387-07
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 1.0 ug.mL-1 10.1128/aac.01531-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 2.0 ug.mL-1 10.1128/aac.01324-08
Streptococcus pneumoniae R6 Penicillin-binding protein 2X Activity nan None 10.1021/jm900625q
Streptococcus pneumoniae serotype 4 (strain ATCC BAA-334 / TIGR4) Penicillin-binding protein 2x Activity nan None 10.1021/jm900625q
Streptococcus pyogenes Streptococcus pyogenes Activity 0.0 % 10.1128/aac.01128-07
Streptococcus pyogenes Streptococcus pyogenes MIC 0.002 ug.mL-1 10.1016/s0960-894x(98)00270-4
Streptococcus pyogenes Streptococcus pyogenes MIC 0.002 ug.mL-1 10.1016/s0960-894x(99)00407-2
Streptococcus pyogenes Streptococcus pyogenes MIC 0.004 ug.mL-1 10.1021/np020507i
Streptococcus pyogenes Streptococcus pyogenes MIC 0.004 ug.mL-1 10.1021/np060206z
Streptococcus pyogenes Streptococcus pyogenes MIC 0.007 ug.mL-1 10.1021/np049577a
Streptococcus pyogenes Streptococcus pyogenes MIC 0.008 ug.mL-1 10.1021/acs.jmedchem.6b00746
Streptococcus pyogenes Streptococcus pyogenes MIC 0.01 ug.mL-1 10.1016/j.ejmech.2006.10.006
Streptococcus pyogenes Streptococcus pyogenes MIC 0.01 ug.mL-1 10.1021/np020507i
Streptococcus pyogenes Streptococcus pyogenes MIC 0.013 ug.mL-1 10.1016/j.bmcl.2003.09.039
Streptococcus pyogenes Streptococcus pyogenes MIC 0.013 ug.mL-1 10.1016/j.bmcl.2004.09.092
Streptococcus pyogenes Streptococcus pyogenes MIC 0.013 ug.mL-1 10.1016/j.ejmech.2006.10.006
Streptococcus pyogenes Streptococcus pyogenes MIC 0.013 ug.mL-1 10.1016/j.ejmech.2007.02.001
Streptococcus pyogenes Streptococcus pyogenes MIC 0.013 ug.mL-1 10.1016/s0960-894x(00)00253-5
Streptococcus pyogenes Streptococcus pyogenes MIC 0.013 ug.mL-1 10.1016/s0960-894x(00)00575-8
Streptococcus pyogenes Streptococcus pyogenes MIC 0.013 ug.mL-1 10.1016/s0960-894x(01)00451-6
Streptococcus pyogenes Streptococcus pyogenes MIC 0.013 ug.mL-1 10.1016/s0960-894x(02)00948-4
Streptococcus pyogenes Streptococcus pyogenes MIC 0.013 ug.mL-1 10.1016/s0960-894x(99)00646-0
Streptococcus pyogenes Streptococcus pyogenes MIC 0.013 ug.mL-1 10.1016/s0960-894x(99)00692-7
Streptococcus pyogenes Streptococcus pyogenes MIC50 0.015 ug.mL-1 10.1128/aac.01128-07
Streptococcus pyogenes Streptococcus pyogenes MIC90 0.015 ug.mL-1 10.1128/aac.01128-07
Streptococcus pyogenes Streptococcus pyogenes PD50 7.16 mg kg-1 10.1016/s0960-894x(98)00270-4
Streptococcus pyogenes serotype M1 Streptokinase A EC50 127.0 nM None
Streptococcus sp. 'group A' Streptococcus sp. 'group A' EC50 153.0 nM None
Streptococcus sp. 'group B' Streptococcus sp. 'group B' MIC 0.12 ug.mL-1 10.1128/aac.00596-08
Streptococcus sp. 'group B' Streptococcus sp. 'group B' MIC 0.25 ug.mL-1 10.1128/aac.00596-08
Streptococcus sp. 'group B' Streptococcus sp. 'group B' MIC 0.5 ug.mL-1 10.1128/aac.00596-08
Sus scrofa Renal dipeptidase Activity 32.0 None 10.1016/s0960-894x(99)00692-7
Sus scrofa Renal dipeptidase DHP-I stability 1.0 None 10.1016/S0960-894X(97)00230-8
Sus scrofa Renal dipeptidase Relative t1/2 1.0 None 10.1016/s0960-894x(99)00646-0
Sus scrofa Renal dipeptidase Stability 100.0 % 10.1016/s0960-894x(99)00407-2
Sus scrofa Renal dipeptidase Stability 3200.0 % 10.1016/s0960-894x(98)00270-4
Thomasclavelia ramosa Thomasclavelia ramosa MIC 0.5 ug.mL-1 10.1128/aac.00910-07
Thomasclavelia ramosa Thomasclavelia ramosa MIC 1.0 ug.mL-1 10.1128/aac.00595-08
Thomasclavelia ramosa Thomasclavelia ramosa MIC50 1.0 ug.mL-1 10.1128/aac.00910-07
Trueperella pyogenes Trueperella pyogenes MIC 0.03 ug.mL-1 10.1016/j.ejmech.2006.10.006
Trueperella pyogenes Trueperella pyogenes MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
Veillonella parvula Veillonella parvula MIC 0.03 ug.mL-1 10.1128/aac.00595-08
Veillonella parvula Veillonella parvula MIC 0.06 ug.mL-1 10.1128/aac.00355-08
None ADMET AUC 2.0 hr 10.1016/s0960-894x(98)00270-4
None ADMET AUC 3.29 ug ml-1 10.1016/s0960-894x(98)00270-4
None ADMET AUC 6383.33 ng.hr.mL-1 10.1016/j.bmcl.2004.09.092
None ADMET AUC 6383.33 ng.hr.mL-1 10.1016/j.ejmech.2019.111744
None ADMET AUC 11583.33 ng.hr.mL-1 10.1016/j.bmcl.2004.09.092
None ADMET CL 3.9 mL.min-1.kg-1 10.1124/dmd.108.020479
None ADMET CL 4.0 mL.min-1.kg-1 10.1002/jps.20373
None ADMET CL 7.0 mL.min-1.kg-1 10.1002/jps.20373
None ADMET CL 7.0 mL.min-1.kg-1 10.1016/j.bmcl.2004.09.092
None ADMET CL 47.0 mL.min-1.kg-1 10.1002/jps.20373
None ADMET CL 51.16 mL.min-1.kg-1 10.1016/j.ejmech.2019.111744
None ADMET CL 52.0 mL.min-1.kg-1 10.1016/j.bmcl.2004.09.092
None ADMET Cmax 19819.02 nM 10.1016/s0960-894x(98)00270-4
None ADMET Cmax 146295.67 nM 10.1128/aac.00160-07
None ADMET log10(%HIA +10) 1.0 None 10.1016/j.ejmech.2010.11.005
None ADMET mortality 100.0 % 10.1016/j.ejmech.2019.04.034
None ADMET MRT 1.3 hr 10.1124/dmd.108.020479
None ADMET Ratio 34.24 None 10.1128/aac.00294-06
None ADMET Ratio 1427.66 None 10.1128/aac.00294-06
None ADMET Ratio 6683.38 None 10.1128/aac.00294-06
None ADMET Relative t1/2 1.0 None 10.1016/s0960-894x(02)00948-4
None ADMET T1/2 0.01667 hr 10.1016/j.bmcl.2004.09.092
None ADMET T1/2 0.06667 hr 10.1016/j.bmcl.2004.09.092
None ADMET T1/2 0.24 hr 10.1016/s0960-894x(98)00270-4
None ADMET T1/2 0.45 hr 10.1128/aac.00160-07
None ADMET T1/2 0.46 hr 10.1021/acs.jmedchem.2c00227
None ADMET T1/2 0.55 hr 10.1016/j.bmcl.2004.09.092
None ADMET T1/2 1.0 hr 10.1016/j.ejmech.2020.112829
None ADMET T1/2 1.0 hr 10.1124/dmd.108.020479
None ADMET T1/2 3.99 hr 10.1016/j.ejmech.2019.111744
None ADMET Tmax 0.21 hr 10.1016/s0960-894x(98)00270-4
None ADMET Vdss 0.25 L.kg-1 10.1002/jps.20373
None ADMET Vdss 0.3 L.kg-1 10.1002/jps.20373
None ADMET Vdss 0.3 L.kg-1 10.1124/dmd.108.020479
None ADMET Vdss 0.3 mL/min/kg 10.1002/jps.20373
None Erythrocyte HC50 500.0 ug ml-1 10.1016/j.ejmech.2022.114278
None Erythrocyte HC50 nan None 10.1016/j.ejmech.2017.10.044
None Erythrocyte HC50 nan None 10.1016/j.ejmech.2017.12.009
None Hepatotoxicity Alkaline Phosphatase Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity Alkaline Phosphatase Increase - Index Value 0.0 None 10.2174/1570163043334794
None Hepatotoxicity Alkaline Phosphatase Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None Hepatotoxicity Composite Activity - Active 2.0 None 10.2174/1570163043334794
None Hepatotoxicity Composite Activity - Marginal 1.0 None 10.2174/1570163043334794
None Hepatotoxicity Composite Activity - Score nan None 10.2174/1570163043334794
None Hepatotoxicity GGT Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity GGT Increase - Index Value 0.0 None 10.2174/1570163043334794
None Hepatotoxicity GGT Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None Hepatotoxicity Hepatotoxicity nan None 10.1021/tx900326k
None Hepatotoxicity HepSE_bilirubinemia 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_cholecystitis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_cholelithiasis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_cirrhosis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_Combined Scores 3.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_elevated liver function tests 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatic failure 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatic necrosis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatitis 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatomegaly 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_jaundice 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_liver disease 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_liver fatty 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_liver function tests abnormal 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity LDH Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity LDH Increase - Index Value 33.8 None 10.2174/1570163043334794
None Hepatotoxicity LDH Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None Hepatotoxicity SGOT Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity SGOT Increase - Index Value 50.8 None 10.2174/1570163043334794
None Hepatotoxicity SGOT Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None Hepatotoxicity SGPT Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity SGPT Increase - Index Value 50.8 None 10.2174/1570163043334794
None Hepatotoxicity SGPT Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None NON-PROTEIN TARGET Activity 0.0 % 10.1128/aac.00481-10
None NON-PROTEIN TARGET Activity 0.0 % 10.1128/aac.00696-08
None NON-PROTEIN TARGET Activity 0.0 % 10.1128/aac.00898-09
None NON-PROTEIN TARGET Activity 0.5 % 10.1128/aac.01435-06
None NON-PROTEIN TARGET Activity 8.0 % 10.1128/aac.00481-10
None NON-PROTEIN TARGET Activity 9.0 ug ml-1 10.1128/aac.01525-09
None NON-PROTEIN TARGET Activity 16.0 ug ml-1 10.1128/aac.00898-09
None NON-PROTEIN TARGET Activity 53.7 % 10.1128/aac.01173-09
None NON-PROTEIN TARGET Activity 92.0 % 10.1128/aac.00481-10
None NON-PROTEIN TARGET Activity nan None 10.1128/aac.00128-10
None NON-PROTEIN TARGET Activity nan None 10.1128/aac.01525-09
None NON-PROTEIN TARGET FICI 0.5 None 10.1128/aac.01173-09
None NON-PROTEIN TARGET fT>MIC 1.9 hr 10.1128/aac.00642-09
None NON-PROTEIN TARGET fT>MIC 2.0 hr 10.1128/aac.00642-09
None NON-PROTEIN TARGET fT>MIC 8.0 % 10.1128/aac.00642-09
None NON-PROTEIN TARGET fT>MIC 8.5 % 10.1128/aac.00642-09
None NON-PROTEIN TARGET fT>MIC 40.0 % 10.1128/aac.01582-09
None NON-PROTEIN TARGET Fu 0.87 None 10.1124/dmd.108.020479
None NON-PROTEIN TARGET Hepatotoxicity (acute) 5.3 % 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (animal toxicity known) nan None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (benign tumour) 0.0 None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (granulomatous hepatitis) 0.0 None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (mechanism) nan None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (moderate) 48.1 % 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (moderate) 92.0 None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (time to onset) nan None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET MIC 0.00012 ug.mL-1 10.1128/aac.01102-06
None NON-PROTEIN TARGET MIC 0.00025 ug.mL-1 10.1128/aac.01102-06
None NON-PROTEIN TARGET MIC 0.002 ug.mL-1 10.1128/aac.01102-06
None NON-PROTEIN TARGET MIC 0.008 ug.mL-1 10.1128/aac.00481-10
None NON-PROTEIN TARGET MIC 0.0094 ug.mL-1 10.1128/aac.00570-10
None NON-PROTEIN TARGET MIC 0.013 ug.mL-1 10.1016/s0960-894x(98)00270-4
None NON-PROTEIN TARGET MIC 0.015 ug.mL-1 10.1128/aac.00336-08
None NON-PROTEIN TARGET MIC 0.015 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC 0.02 ug.mL-1 10.1016/j.ejmech.2007.02.001
None NON-PROTEIN TARGET MIC 0.023 ug.mL-1 10.1128/aac.00630-09
None NON-PROTEIN TARGET MIC 0.025 ug.mL-1 10.1016/s0960-894x(98)00270-4
None NON-PROTEIN TARGET MIC 0.03 ug.mL-1 10.1016/j.ejmech.2006.10.006
None NON-PROTEIN TARGET MIC 0.03 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC 0.032 ug.mL-1 10.1128/aac.00570-10
None NON-PROTEIN TARGET MIC 0.032 ug.mL-1 10.1128/aac.00630-09
None NON-PROTEIN TARGET MIC 0.032 ug.mL-1 10.1128/aac.00684-07
None NON-PROTEIN TARGET MIC 0.05 ug.mL-1 10.1016/j.ejmech.2006.10.006
None NON-PROTEIN TARGET MIC 0.05 ug.mL-1 10.1016/j.ejmech.2007.02.001
None NON-PROTEIN TARGET MIC 0.06 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC 0.06 ug.mL-1 10.1128/aac.00696-08
None NON-PROTEIN TARGET MIC 0.06 ug.mL-1 10.1128/aac.00978-07
None NON-PROTEIN TARGET MIC 0.06 ug.mL-1 10.1128/aac.01525-09
None NON-PROTEIN TARGET MIC 0.06 ug.mL-1 10.1128/aac.01585-09
None NON-PROTEIN TARGET MIC 0.064 ug.mL-1 10.1128/aac.00630-09
None NON-PROTEIN TARGET MIC 0.12 ug.mL-1 10.1016/j.bmc.2013.09.041
None NON-PROTEIN TARGET MIC 0.125 ug.mL-1 10.1128/aac.00570-10
None NON-PROTEIN TARGET MIC 0.125 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC 0.125 ug.mL-1 10.1128/aac.00696-08
None NON-PROTEIN TARGET MIC 0.25 ug.mL-1 10.1128/aac.00570-10
None NON-PROTEIN TARGET MIC 0.25 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC 0.25 ug.mL-1 10.1128/aac.01525-09
None NON-PROTEIN TARGET MIC 0.38 ug.mL-1 10.1128/aac.00570-10
None NON-PROTEIN TARGET MIC 0.4 ug.mL-1 10.1128/aac.01435-06
None NON-PROTEIN TARGET MIC 0.5 ug.mL-1 10.1128/aac.00128-10
None NON-PROTEIN TARGET MIC 0.5 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC 0.5 ug.mL-1 10.1128/aac.00978-07
None NON-PROTEIN TARGET MIC 1.0 ug.mL-1 10.1128/aac.00570-10
None NON-PROTEIN TARGET MIC 1.0 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC 1.0 ug.mL-1 10.1128/aac.00899-09
None NON-PROTEIN TARGET MIC 2.0 ug.mL-1 10.1128/aac.00630-09
None NON-PROTEIN TARGET MIC 4.0 ug.mL-1 10.1128/aac.00570-10
None NON-PROTEIN TARGET MIC 4.0 ug.mL-1 10.1128/aac.00899-09
None NON-PROTEIN TARGET MIC 8.0 ug.mL-1 10.1128/aac.00128-10
None NON-PROTEIN TARGET MIC 8.0 ug.mL-1 10.1128/aac.00899-09
None NON-PROTEIN TARGET MIC 16.0 ug.mL-1 10.1128/aac.00128-10
None NON-PROTEIN TARGET MIC 32.0 ug.mL-1 10.1128/aac.00734-08
None NON-PROTEIN TARGET MIC50 0.015 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC50 0.03 ug.mL-1 10.1128/aac.00336-08
None NON-PROTEIN TARGET MIC50 0.03 ug.mL-1 10.1128/aac.00898-09
None NON-PROTEIN TARGET MIC50 0.06 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC50 0.125 ug.mL-1 10.1128/aac.00481-10
None NON-PROTEIN TARGET MIC50 0.125 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC50 0.125 ug.mL-1 10.1128/aac.01525-09
None NON-PROTEIN TARGET MIC50 0.19 ug.mL-1 10.1128/aac.00630-09
None NON-PROTEIN TARGET MIC50 0.25 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC50 0.25 ug.mL-1 10.1128/aac.00696-08
None NON-PROTEIN TARGET MIC50 2.0 ug.mL-1 10.1128/aac.00696-08
None NON-PROTEIN TARGET MIC50 2.0 ug.mL-1 10.1128/aac.01525-09
None NON-PROTEIN TARGET MIC50 4.0 ug.mL-1 10.1128/aac.00898-09
None NON-PROTEIN TARGET MIC90 0.03 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC90 0.12 ug.mL-1 10.1128/aac.00336-08
None NON-PROTEIN TARGET MIC90 0.125 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC90 0.25 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC90 0.25 ug.mL-1 10.1128/aac.00898-09
None NON-PROTEIN TARGET MIC90 0.5 ug.mL-1 10.1128/aac.01525-09
None NON-PROTEIN TARGET MIC90 1.0 ug.mL-1 10.1128/aac.00696-08
None NON-PROTEIN TARGET MIC90 1.0 ug.mL-1 10.1128/aac.01435-06
None NON-PROTEIN TARGET MIC90 2.0 ug.mL-1 10.1128/aac.00481-10
None NON-PROTEIN TARGET MIC90 2.0 ug.mL-1 10.1128/aac.00696-08
None NON-PROTEIN TARGET MIC90 4.0 ug.mL-1 10.1128/aac.00595-08
None NON-PROTEIN TARGET MIC90 4.0 ug.mL-1 10.1128/aac.00630-09
None NON-PROTEIN TARGET MIC90 4.0 ug.mL-1 10.1128/aac.01525-09
None NON-PROTEIN TARGET MIC90 64.0 ug.mL-1 10.1128/aac.00898-09
None NON-PROTEIN TARGET T>MIC 41.67 % 10.1128/aac.00160-07
None NON-PROTEIN TARGET T>MIC 66.67 % 10.1128/aac.00160-07
None No relevant target Activity 40.3 % 10.1128/aac.00123-08
None No relevant target Activity 49.3 % 10.1128/aac.00123-08
None No relevant target Drug degradation 30.0 % 10.1021/acs.jmedchem.0c00255
None No relevant target Drug degradation 50.0 % 10.1021/ml200012f
None No relevant target Drug degradation 60.0 % 10.1016/j.ejmech.2020.112829
None No relevant target Drug degradation 80.0 % 10.1016/j.bmc.2013.05.024
None No relevant target LogD 2.5 None 10.1016/j.bmc.2013.05.024
None No relevant target Stability 5.0 % 10.1016/j.bmc.2013.05.024
None No relevant target T1/2 78.0 hr 10.1016/j.bmcl.2018.01.006
None No relevant target T1/2 95.0 hr 10.1021/acsmedchemlett.5b00026
None Unchecked Ac50 0.3162 uM None
None Unchecked Ac50 0.7079 uM None
None Unchecked Ac50 0.8913 uM None
None Unchecked AC50 316.2 nM None
None Unchecked AC50 320.0 nM None
None Unchecked AC50 707.9 nM None
None Unchecked AC50 891.3 nM None
None Unchecked Activity 0.0011 % 10.1128/aac.01004-09
None Unchecked Activity 0.002 % 10.1128/aac.01004-09
None Unchecked Activity 0.0024 % 10.1128/aac.01004-09
None Unchecked Activity 0.0079 % 10.1128/aac.01004-09
None Unchecked Activity 1.0 mU 10.1128/aac.00978-07
None Unchecked Activity 1.5 mU 10.1128/aac.00978-07
None Unchecked Activity 1.7 mU 10.1128/aac.00978-07
None Unchecked Activity 1.8 % 10.1128/aac.00083-07
None Unchecked Activity 3.4 % 10.1128/aac.00175-08
None Unchecked Activity 9.4 % 10.1128/aac.00175-08
None Unchecked Activity 83.0 % 10.1128/aac.00175-08
None Unchecked Activity 110.0 % 10.1128/aac.00175-08
None Unchecked Activity nan None 10.1021/acs.jmedchem.1c02140
None Unchecked Activity nan None 10.1128/aac.00978-07
None Unchecked HC50 nan None 10.1021/acs.jmedchem.2c01469
None Unchecked HC50 nan None 10.1021/acs.jmedchem.2c01674
None Unchecked Hepatotoxicity (acute) 1.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (association with vascular disease) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (choleostasis) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (chronic liver disease) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (cirrhosis) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (comment) nan None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (cytolytic) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (malignant tumour) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (severe hepatitis) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (steatosis) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (successful reintroduction) nan None 10.1016/s0399-8320(04)95062-2
None Unchecked IC50 0.0033 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 0.008 ug.mL-1 10.1128/aac.01529-07
None Unchecked IC50 0.013 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 0.016 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 0.018 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 0.02 ug.mL-1 10.1128/aac.01529-07
None Unchecked IC50 0.03 ug.mL-1 10.1128/aac.01529-07
None Unchecked IC50 0.044 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 0.047 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 0.05 ug.mL-1 10.1128/aac.01529-07
None Unchecked IC50 0.06 ug.mL-1 10.1128/aac.01529-07
None Unchecked IC50 0.071 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 0.08 ug.mL-1 10.1128/aac.01529-07
None Unchecked IC50 0.11 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 0.12 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 0.26 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 0.39 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 0.5 ug.mL-1 10.1128/aac.01529-07
None Unchecked IC50 0.6 ug.mL-1 10.1128/aac.01529-07
None Unchecked IC50 0.77 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 0.82 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 1.2 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 1.3 ug.mL-1 10.1128/aac.01529-07
None Unchecked IC50 1.7 ug.mL-1 10.1128/aac.01529-07
None Unchecked IC50 4.0 ug.mL-1 10.1128/aac.01529-07
None Unchecked IC50 4.5 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 15.0 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 16.0 ug.mL-1 10.1128/aac.01529-07
None Unchecked IC50 130.0 ug.mL-1 10.1128/aac.01433-08
None Unchecked IC50 nan None None
None Unchecked Inhibition 90.0 % 10.1016/j.bmc.2021.116128
None Unchecked K 1.1 10'3/uM/s 10.1021/acs.jmedchem.6b00096
None Unchecked K 4.9 10'4/M/s 10.1021/acsmedchemlett.5b00026
None Unchecked K 60.0 10'3/s 10.1021/acs.jmedchem.6b00096
None Unchecked Kcat 0.00039 /s 10.1128/aac.01004-09
None Unchecked Kcat 0.0096 /s 10.1128/aac.01004-09
None Unchecked Kcat 0.01 /s 10.1128/aac.01600-06
None Unchecked Kcat 0.05 /s 10.1128/aac.00858-10
None Unchecked Kcat 0.3 /s 10.1128/aac.00856-09
None Unchecked Kcat 0.4 /s 10.1128/aac.01337-07
None Unchecked Kcat 0.92 10'3/s 10.1021/acs.jmedchem.6b00096
None Unchecked Kcat 1.0 /s 10.1128/aac.00961-09
None Unchecked Kcat 1.0 /s 10.1128/aac.01009-09
None Unchecked Kcat 1.0 /s 10.1128/aac.01062-07
None Unchecked Kcat 1.0 /s 10.1128/aac.01462-06
None Unchecked Kcat 1.3 /s 10.1128/aac.00017-09
None Unchecked Kcat 4.13 /s 10.1128/aac.00083-07
None Unchecked Kcat 5.0 /s 10.1128/aac.00858-10
None Unchecked Kcat 5.0 /s 10.1128/aac.01336-09
None Unchecked Kcat 6.0 /s 10.1128/aac.01336-09
None Unchecked Kcat 6.5 /s 10.1128/aac.00175-08
None Unchecked Kcat 8.4 /s 10.1128/aac.00175-08
None Unchecked Kcat 13.0 /s 10.1128/aac.00166-08
None Unchecked Kcat 50.0 /s 10.1128/aac.00774-09
None Unchecked Kcat/Km 4.4e-05 /s/microM 10.1128/aac.01004-09
None Unchecked Kcat/Km 0.00011 /s/microM 10.1128/aac.01004-09
None Unchecked Kcat/Km 0.003 /s/microM 10.1128/aac.00856-09
None Unchecked Kcat/Km 0.015 /uM/s 10.1128/aac.00083-07
None Unchecked Kcat/Km 0.07 /s/microM 10.1128/aac.00175-08
None Unchecked Kcat/Km 0.12 /s/microM 10.1128/aac.00774-09
None Unchecked Kcat/Km 0.14 /s/microM 10.1128/aac.00017-09
None Unchecked Kcat/Km 0.26 /uM/s 10.1128/aac.00166-08
None Unchecked Kcat/Km 0.5 uM/hr 10.1128/aac.01336-09
None Unchecked Kcat/Km 1.0 /s/M 10.1128/aac.01025-07
None Unchecked Kcat/Km 1.9 /s/microM 10.1128/aac.00175-08
None Unchecked Kcat/Km 3.0 uM/hr 10.1128/aac.01336-09
None Unchecked Kcat/Km 3.3 10'4/M/s 10.1128/aac.01337-07
None Unchecked Kcat/Km 3.3 None 10.1128/aac.01462-06
None Unchecked Kcat/Km 4.5 10'6/M/s 10.1128/aac.00409-10
None Unchecked Kcat/Km 5.0 10'5/M/s 10.1128/aac.00409-10
None Unchecked Kcat/Km 5.0 10'5/M/s 10.1128/aac.00858-10
None Unchecked Kcat/Km 5.3 10'6/M/s 10.1128/aac.00409-10
None Unchecked Kcat/Km 6.0 10'3/M/s 10.1128/aac.00858-10
None Unchecked Kcat/Km 8.3 10'5/M/s 10.1128/aac.00409-10
None Unchecked Kcat/Km 8.3 10'5/M/s 10.1128/aac.01062-07
None Unchecked Kcat/Km 9.6 10'2/M/s 10.1128/aac.01062-07
None Unchecked Kcat/Km 1000.0 /M/s 10.1021/acs.jmedchem.6b00096
None Unchecked Kd 75000.0 nM 10.1016/j.bmc.2020.115437
None Unchecked Ki nan None None
None Unchecked Km 300.0 nM 10.1128/aac.01462-06
None Unchecked Km 920.0 nM 10.1021/acs.jmedchem.6b00096
None Unchecked Km 2000.0 nM 10.1128/aac.01336-09
None Unchecked Km 3400.0 nM 10.1128/aac.00175-08
None Unchecked Km 5000.0 nM 10.1128/aac.00409-10
None Unchecked Km 8400.0 nM 10.1128/aac.00858-10
None Unchecked Km 8800.0 nM 10.1128/aac.01004-09
None Unchecked Km 10000.0 nM 10.1128/aac.00409-10
None Unchecked Km 10000.0 nM 10.1128/aac.00774-09
None Unchecked Km 10000.0 nM 10.1128/aac.00858-10
None Unchecked Km 10000.0 nM 10.1128/aac.01336-09
None Unchecked Km 12000.0 nM 10.1128/aac.00961-09
None Unchecked Km 12000.0 nM 10.1128/aac.01337-07
None Unchecked Km 50000.0 nM 10.1128/aac.00166-08
None Unchecked Km 85000.0 nM 10.1128/aac.00409-10
None Unchecked Km 90000.0 nM 10.1128/aac.01004-09
None Unchecked Km 100000.0 nM 10.1128/aac.00856-09
None Unchecked Km 120000.0 nM 10.1128/aac.00175-08
None Unchecked Km 190000.0 nM 10.1128/aac.00409-10
None Unchecked Km 280000.0 nM 10.1128/aac.00083-07
None Unchecked Km 990000.0 nM 10.1128/aac.01062-07
None Unchecked Km nan None 10.1128/aac.01600-06
None Unchecked MIC 1.0 ug.mL-1 10.1016/j.bmc.2020.115598
None Unchecked MIC 1.0 ug.mL-1 10.1016/j.bmcl.2003.09.039
None Unchecked MIC 1.0 ug.mL-1 10.1016/s0960-894x(00)00253-5
None Unchecked MIC 16.0 ug.mL-1 10.1016/j.bmc.2020.115598
None Unchecked MIC 32.0 ug.mL-1 10.1016/j.bmc.2021.116128
None Unchecked MIC 64.0 ug.mL-1 10.1016/j.bmc.2021.116128
None Unchecked MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.06.007
None Unchecked MIC 128.0 ug.mL-1 10.1016/j.bmc.2021.116128
None Unchecked MIC nan None 10.1016/j.bmc.2020.115598
None Unchecked Ratio 1.0 None 10.1128/aac.00413-08
None Unchecked Ratio 2.0 None 10.1128/aac.00413-08
None Unchecked Ratio 4.0 None 10.1128/aac.00413-08
None Unchecked Ratio 8.0 None 10.1128/aac.00413-08
None Unchecked Ratio 28.05 None 10.1128/aac.00160-07
None Unchecked Ratio 32.0 None 10.1128/aac.00413-08
None Unchecked Ratio 112.2 None 10.1128/aac.00160-07
None Unchecked Ratio 1300.0 /M/s 10.1021/acs.jmedchem.6b00096
None Unchecked Ratio nan None 10.1021/acs.jmedchem.2c01674
None Unchecked Relative hydrolysis 28.0 None 10.1016/S0960-894X(97)00282-5
None Unchecked Stability 100.0 % 10.1016/s0960-894x(01)00451-6

Metabolism Information