| Acinetobacter baumannii |
Acinetobacter baumannii |
Inhibition |
2.64 |
% |
10.6019/CHEMBL4513141 |
| Bacillus subtilis |
4'-phosphopantetheinyl transferase ffp |
Potency |
70794.6 |
nM |
None |
| Bos taurus |
Progesterone receptor |
IC50 |
nan |
None |
None |
| Bos taurus |
Progesterone receptor |
Ki |
nan |
None |
None |
| Candida albicans |
Candida albicans |
Inhibition |
3.01 |
% |
10.6019/CHEMBL4513141 |
| Canis lupus familiaris |
Canis familiaris |
ED50 |
0.0087 |
mg.kg-1 |
10.1021/jm00393a018 |
| Canis lupus familiaris |
Canis familiaris |
ED50 |
0.042 |
mg.kg-1 |
10.1021/jm00027a007 |
| Canis lupus familiaris |
Canis familiaris |
Inhibition |
96.0 |
% |
10.1021/jm00027a007 |
| Canis lupus familiaris |
MDCK |
logPapp |
-7.36 |
None |
10.1021/jm901846t |
| Cavia porcellus |
Histamine H2 receptor |
ED50 |
2.7e-06 |
M |
10.1021/jm00393a018 |
| Cavia porcellus |
Histamine H2 receptor |
IC50 |
300.0 |
nM |
10.1021/jm00027a007 |
| Cavia porcellus |
Histamine H2 receptor |
Inhibition |
87.0 |
% |
10.1021/jm00027a007 |
| Cavia porcellus |
Histamine H2 receptor |
Kd |
18.2 |
nM |
10.1016/s0960-894x(03)00235-x |
| Cavia porcellus |
Histamine H2 receptor |
Kd |
100.0 |
nM |
10.1021/jm00091a012 |
| Cavia porcellus |
Leukotriene C4 synthase |
IC50 |
nan |
None |
None |
| Cavia porcellus |
Leukotriene C4 synthase |
Ki |
nan |
None |
None |
| Cavia porcellus |
Serotonin 4 (5-HT4) receptor |
IC50 |
nan |
None |
None |
| Cavia porcellus |
Serotonin 4 (5-HT4) receptor |
Ki |
nan |
None |
None |
| Cryptococcus neoformans |
Cryptococcus neoformans |
Inhibition |
-2.8 |
% |
10.6019/CHEMBL4513141 |
| Escherichia coli |
Escherichia coli |
Inhibition |
3.55 |
% |
10.6019/CHEMBL4513141 |
| Homo sapiens |
Acetylcholinesterase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Acetylcholinesterase |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A2a receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A2a receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A2a receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A3 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A3 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adhesion G-protein coupled receptor F1 |
%Inhib (Mean) |
-53.73 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Adhesion G-protein coupled receptor F1 |
%Inhib (Mean) |
-48.78 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Adhesion G-protein coupled receptor F1 |
%Inhib (Mean) |
-37.63 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Adhesion G-protein coupled receptor F1 |
%Inhib (Mean) |
-35.84 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Adhesion G-protein coupled receptor F1 |
%Max (Mean) |
-0.02135 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1d adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-1d adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
%Inhib (Mean) |
-31.78 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
%Inhib (Mean) |
-14.76 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
%Inhib (Mean) |
-10.3 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
%Inhib (Mean) |
-7.95 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
%Max (Mean) |
4.6 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Alpha-2b adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2b adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2b adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2c adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2c adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2c adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Angiotensin II type 2 (AT-2) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Angiotensin II type 2 (AT-2) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Apelin receptor |
%Inhib (Mean) |
-23.19 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Apelin receptor |
%Inhib (Mean) |
-21.8 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Apelin receptor |
%Inhib (Mean) |
-15.29 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Apelin receptor |
%Inhib (Mean) |
6.27 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Apelin receptor |
%Max (Mean) |
-0.162 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Beta-1 adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-1 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-1 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-2 adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-2 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
%Inhib (Mean) |
-71.34 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Beta-2 adrenergic receptor |
%Inhib (Mean) |
-18.53 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Beta-2 adrenergic receptor |
%Inhib (Mean) |
-6.38 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Beta-2 adrenergic receptor |
%Inhib (Mean) |
14.64 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Beta-2 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
%Max (Mean) |
-2.02 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Beta-3 adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-3 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-3 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Bile salt export pump |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bile salt export pump |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Bile salt export pump |
IC50 |
135000.0 |
nM |
10.1093/toxsci/kfq269 |
| Homo sapiens |
Bile salt export pump |
IC50 |
1000000.0 |
nM |
10.1124/dmd.111.040758 |
| Homo sapiens |
Bloom syndrome protein |
Potency |
1.6 |
nM |
None |
| Homo sapiens |
Bradykinin B1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bradykinin B2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bradykinin B2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Bradykinin B2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Bromodomain-containing protein 4 |
Delta TM |
-1.43 |
C |
None |
| Homo sapiens |
C5a anaphylatoxin chemotactic receptor |
%Inhib (Mean) |
-27.84 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
C5a anaphylatoxin chemotactic receptor |
%Inhib (Mean) |
-25.37 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
C5a anaphylatoxin chemotactic receptor |
%Inhib (Mean) |
-23.39 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
C5a anaphylatoxin chemotactic receptor |
%Inhib (Mean) |
-3.981 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
C5a anaphylatoxin chemotactic receptor |
%Max (Mean) |
-3.059 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Calcitonin receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Calcitonin receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Canalicular multispecific organic anion transporter 1 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 2 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Cannabinoid CB1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cannabinoid CB1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cannabinoid CB1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cannabinoid CB1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase I |
Ki |
922.4 |
nM |
10.1021/acsmedchemlett.8b00334 |
| Homo sapiens |
Carbonic anhydrase II |
IC50 |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase II |
Ki |
57.9 |
nM |
10.1021/acsmedchemlett.8b00334 |
| Homo sapiens |
Carbonic anhydrase II |
Ki |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase III |
Ki |
10000.0 |
nM |
10.1021/acsmedchemlett.8b00334 |
| Homo sapiens |
Carbonic anhydrase IV |
Ki |
938.8 |
nM |
10.1021/acsmedchemlett.8b00334 |
| Homo sapiens |
Carbonic anhydrase IX |
Ki |
126.3 |
nM |
10.1021/acsmedchemlett.8b00334 |
| Homo sapiens |
Carbonic anhydrase VA |
Ki |
1429.5 |
nM |
10.1021/acsmedchemlett.8b00334 |
| Homo sapiens |
Carbonic anhydrase VB |
Ki |
5328.2 |
nM |
10.1021/acsmedchemlett.8b00334 |
| Homo sapiens |
Carbonic anhydrase VI |
Ki |
98.2 |
nM |
10.1021/acsmedchemlett.8b00334 |
| Homo sapiens |
Carbonic anhydrase VII |
Ki |
3.0 |
nM |
10.1021/acsmedchemlett.8b00334 |
| Homo sapiens |
Carbonic anhydrase XII |
Ki |
45.3 |
nM |
10.1021/acsmedchemlett.8b00334 |
| Homo sapiens |
Carbonic anhydrase XIII |
Ki |
171.5 |
nM |
10.1021/acsmedchemlett.8b00334 |
| Homo sapiens |
Carbonic anhydrase XIV |
Ki |
677.2 |
nM |
10.1021/acsmedchemlett.8b00334 |
| Homo sapiens |
Casein kinase I delta |
Delta TM |
0.05 |
C |
None |
| Homo sapiens |
Caspase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Caspase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cathepsin G |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cathepsin G |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 2 |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 4 |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin A receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cholecystokinin A receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin A receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin B receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cholesterol 24-hydroxylase |
Activity |
60.0 |
% |
None |
| Homo sapiens |
Corticotropin releasing factor receptor 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Corticotropin releasing factor receptor 2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
C-X3-C chemokine receptor 1 |
%Inhib (Mean) |
-36.18 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
C-X3-C chemokine receptor 1 |
%Inhib (Mean) |
-22.14 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
C-X3-C chemokine receptor 1 |
%Inhib (Mean) |
-5.56 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
C-X3-C chemokine receptor 1 |
%Inhib (Mean) |
3.168 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
C-X3-C chemokine receptor 1 |
%Max (Mean) |
-1.787 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Cyclin-dependent kinase 2 |
Delta TM |
1.16 |
C |
None |
| Homo sapiens |
Cyclooxygenase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cysteinyl leukotriene receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cysteinyl leukotriene receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
Activity |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2A6 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2A6 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2E1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2E1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Delta opioid receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Delta opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Delta opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
DNA-(apurinic or apyrimidinic site) lyase |
Potency |
2511.9 |
nM |
None |
| Homo sapiens |
DNA polymerase iota |
Potency |
10000.0 |
nM |
None |
| Homo sapiens |
Dopamine D1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D2 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D3 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D3 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D3 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D4 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D4 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D4 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D5 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine transporter |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Endothelin receptor ET-A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-A |
Ki |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-B |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Equilibrative nucleoside transporter 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor beta |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor beta |
IC50 |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor beta |
Ki |
nan |
None |
None |
| Homo sapiens |
Fibroblast |
Growth Rate |
0.17 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
Fibroblast |
Growth Rate |
0.22 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
Fibroblast |
Growth Rate |
0.4 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
Fibroblast |
Growth Rate |
0.41 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
Fibroblast |
Growth Rate |
0.42 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
Fibroblast |
Growth Rate |
0.55 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
Fibroblast |
Growth Rate |
0.89 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
Fibroblast growth factor receptor 3 |
Delta TM |
0.15 |
C |
None |
| Homo sapiens |
Gastric inhibitory polypeptide receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Geminin |
Potency |
580.5 |
nM |
None |
| Homo sapiens |
Ghrelin receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucagon-like peptide 1 receptor |
%Inhib (Mean) |
-27.9 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Glucagon-like peptide 1 receptor |
%Inhib (Mean) |
-27.63 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Glucagon-like peptide 1 receptor |
%Inhib (Mean) |
-11.95 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Glucagon-like peptide 1 receptor |
%Inhib (Mean) |
-7.46 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Glucagon-like peptide 1 receptor |
%Max (Mean) |
-0.48 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Glucagon receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Glucocorticoid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Glucose-dependent insulinotropic receptor |
%Inhib (Mean) |
-19.12 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Glucose-dependent insulinotropic receptor |
%Inhib (Mean) |
-3.01 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Glucose-dependent insulinotropic receptor |
%Inhib (Mean) |
-2.015 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Glucose-dependent insulinotropic receptor |
%Inhib (Mean) |
1.61 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Glucose-dependent insulinotropic receptor |
%Max (Mean) |
0.5819 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Glycogen synthase kinase-3 beta |
Delta TM |
0.06 |
C |
None |
| Homo sapiens |
G-protein coupled receptor 120 |
%Inhib (Mean) |
-39.4 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
G-protein coupled receptor 120 |
%Inhib (Mean) |
-25.96 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
G-protein coupled receptor 120 |
%Inhib (Mean) |
-22.73 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
G-protein coupled receptor 120 |
%Inhib (Mean) |
-12.11 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
G-protein coupled receptor 120 |
%Max (Mean) |
0.1 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
G-protein coupled receptor 35 |
%Inhib (Mean) |
-26.08 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
G-protein coupled receptor 35 |
%Max (Mean) |
19.14 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
HEK293 |
Drug uptake |
nan |
None |
10.1021/acs.jmedchem.2c01075 |
| Homo sapiens |
HEK-293T |
Growth Rate |
0.45 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
HEK-293T |
Growth Rate |
0.65 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
HEK-293T |
Growth Rate |
0.72 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
HEK-293T |
Growth Rate |
0.89 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
HEK-293T |
Growth Rate |
0.96 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
HERG |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
HERG |
IC50 |
nan |
None |
None |
| Homo sapiens |
HERG |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Histamine H1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H2 receptor |
AC50 |
6.3 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H2 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H2 receptor |
IC50 |
42.0 |
nM |
None |
| Homo sapiens |
Histamine H2 receptor |
Ki |
41.0 |
nM |
None |
| Homo sapiens |
Histamine H3 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histone deacetylase 6 |
Inhibition |
-45.31 |
% |
10.6019/CHEMBL4808148 |
| Homo sapiens |
Histone deacetylase 6 |
Inhibition |
-4.29 |
% |
10.6019/CHEMBL4808148 |
| Homo sapiens |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Potency |
25.1 |
nM |
None |
| Homo sapiens |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Potency |
843.7 |
nM |
None |
| Homo sapiens |
HMG-CoA reductase |
IC50 |
nan |
None |
None |
| Homo sapiens |
HMG-CoA reductase |
Ki |
nan |
None |
None |
| Homo sapiens |
Homo sapiens |
% absorbed |
45.0 |
% |
10.1021/jm001020e |
| Homo sapiens |
Homo sapiens |
Activity |
0.28 |
% |
10.1016/j.ejmech.2009.11.034 |
| Homo sapiens |
Homo sapiens |
CL |
6.6 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
CL_renal |
4.42 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
DILI_Concern |
nan |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
DILI_severity_class |
3.0 |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
F |
42.0 |
% |
10.1021/jm901421c |
| Homo sapiens |
Homo sapiens |
F |
42.0 |
% |
10.1021/jm901846t |
| Homo sapiens |
Homo sapiens |
LBF |
16.0 |
% |
10.1021/jm901421c |
| Homo sapiens |
Homo sapiens |
Vdss |
1.2 |
L.kg-1 |
10.1016/j.ejmech.2009.06.004 |
| Homo sapiens |
Interleukin-8 receptor A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor A |
Ki |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor B |
IC50 |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor B |
Ki |
nan |
None |
None |
| Homo sapiens |
Kappa opioid receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Kappa opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Kappa opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Leukocyte common antigen |
IC50 |
nan |
None |
None |
| Homo sapiens |
Leukocyte common antigen |
Ki |
nan |
None |
None |
| Homo sapiens |
Leukocyte elastase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Leukocyte elastase |
Ki |
nan |
None |
None |
| Homo sapiens |
Lipoxin A4 receptor |
%Inhib (Mean) |
-25.64 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Lipoxin A4 receptor |
%Inhib (Mean) |
-22.56 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Lipoxin A4 receptor |
%Inhib (Mean) |
-17.16 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Lipoxin A4 receptor |
%Inhib (Mean) |
-14.22 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Lipoxin A4 receptor |
%Max (Mean) |
-3.41 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Lysine-specific demethylase 4A |
Potency |
22387.2 |
nM |
None |
| Homo sapiens |
MAP kinase ERK1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK1 |
Ki |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK2 |
Delta TM |
0.11 |
C |
None |
| Homo sapiens |
MAP kinase ERK2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK2 |
Ki |
nan |
None |
None |
| Homo sapiens |
MAP kinase p38 alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase p38 alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase 9 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase 9 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 3 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Melanocortin receptor 3 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 3 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 4 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Melanocortin receptor 4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Monoamine oxidase A |
AC50 |
8100.1 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Monoamine oxidase A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Monoamine oxidase A |
Ki |
nan |
None |
None |
| Homo sapiens |
Motilin receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Multidrug and toxin extrusion protein 1 |
IC50 |
760.0 |
nM |
10.1021/jm301302s |
| Homo sapiens |
Multidrug and toxin extrusion protein 2 |
IC50 |
36200.0 |
nM |
10.1021/jm301302s |
| Homo sapiens |
Multidrug resistance-associated protein 4 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Mu opioid receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Mu opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Mu opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurokinin 1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neurokinin 1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neurokinin 1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurokinin 2 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neurokinin 2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neurokinin 2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurotensin receptor 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Norepinephrine transporter |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Norepinephrine transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Norepinephrine transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Peregrin |
Delta TM |
-1.92 |
C |
None |
| Homo sapiens |
Peripheral myelin protein 22 |
Potency |
95283.4 |
nM |
None |
| Homo sapiens |
Peroxisome proliferator-activated receptor gamma/Nuclear receptor coactivator 1 |
EC50 |
79370.0 |
nM |
None |
| Homo sapiens |
Peroxisome proliferator-activated receptor gamma/Nuclear receptor coactivator 2 |
EC50 |
79370.0 |
nM |
None |
| Homo sapiens |
Peroxisome proliferator-activated receptor gamma/Nuclear receptor coactivator 3 |
EC50 |
79370.0 |
nM |
None |
| Homo sapiens |
Phosphodiesterase 3A |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 4D |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 5A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Phosphodiesterase 5A |
Ki |
nan |
None |
None |
| Homo sapiens |
Phosphodiesterase 6A |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Plasma |
fCmax |
0.492 |
uM |
10.1124/dmd.111.040758 |
| Homo sapiens |
Platelet activating factor receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Platelet activating factor receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
POU domain, class 2, transcription factor 1 |
Activity |
nan |
None |
10.1021/acs.jmedchem.2c01075 |
| Homo sapiens |
POU domain, class 2, transcription factor 1 |
CL |
87.4 |
mL.min-1.g-1 |
10.1021/acs.jmedchem.0c02047 |
| Homo sapiens |
POU domain, class 2, transcription factor 1 |
Km |
35700.0 |
nM |
10.1021/acs.jmedchem.0c02047 |
| Homo sapiens |
POU domain, class 2, transcription factor 1 |
Vmax |
3121.0 |
pmol/mg/min |
10.1021/acs.jmedchem.0c02047 |
| Homo sapiens |
POU domain, class 2, transcription factor 2 |
Activity |
nan |
None |
10.1021/acs.jmedchem.2c01075 |
| Homo sapiens |
Prelamin-A/C |
Potency |
28.2 |
nM |
None |
| Homo sapiens |
Prelamin-A/C |
Potency |
281.8 |
nM |
None |
| Homo sapiens |
Prelamin-A/C |
Potency |
5623.4 |
nM |
None |
| Homo sapiens |
Progesterone receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Protein kinase C alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
Protein kinase C alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Runt-related transcription factor 1/Core-binding factor subunit beta |
Potency |
44668.4 |
nM |
None |
| Homo sapiens |
Serine/threonine-protein kinase Aurora-A |
Delta TM |
-0.15 |
C |
None |
| Homo sapiens |
Serine/threonine-protein kinase PLK1 |
Potency |
23778.1 |
nM |
None |
| Homo sapiens |
Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 1a (5-HT1a) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 3a (5-HT3a) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 5a (5-HT5a) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 7 (5-HT7) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Serum albumin |
pKa |
0.02 |
None |
10.1021/acs.jmedchem.0c00046 |
| Homo sapiens |
Serum albumin |
PPB |
4.4 |
% |
10.1021/acs.jmedchem.0c00046 |
| Homo sapiens |
Serum albumin |
PPB |
25.1 |
% |
10.1021/acs.jmedchem.0c00046 |
| Homo sapiens |
Sigma opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Sigma opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Solute carrier family 22 member 1 |
IC50 |
300000.0 |
nM |
10.1021/jm301302s |
| Homo sapiens |
Solute carrier family 22 member 1 |
Inhibition |
13.9 |
% |
10.1021/jm8003152 |
| Homo sapiens |
Solute carrier family 22 member 2 |
IC50 |
36100.0 |
nM |
10.1021/jm301302s |
| Homo sapiens |
Solute carrier family 22 member 2 |
Ki |
1800000.0 |
nM |
10.1016/j.ejphar.2004.09.032 |
| Homo sapiens |
Solute carrier family 22 member 3 |
Activity |
nan |
None |
10.1021/acs.jmedchem.2c01075 |
| Homo sapiens |
Solute carrier family 22 member 3 |
Drug uptake |
nan |
None |
10.1021/acs.jmedchem.2c01075 |
| Homo sapiens |
Solute carrier family 22 member 3 |
IC50 |
10700.0 |
nM |
10.1021/jm301302s |
| Homo sapiens |
Solute carrier family 22 member 3 |
Inhibition |
6.0 |
% |
10.1021/acs.jmedchem.2c01075 |
| Homo sapiens |
Solute carrier family 22 member 3 |
Inhibition |
29.0 |
% |
10.1021/acs.jmedchem.2c01075 |
| Homo sapiens |
Solute carrier family 22 member 3 |
Inhibition |
55.0 |
% |
10.1021/acs.jmedchem.2c01075 |
| Homo sapiens |
Solute carrier family 22 member 3 |
Inhibition |
56.0 |
% |
10.1021/acs.jmedchem.2c01075 |
| Homo sapiens |
Solute carrier family 22 member 8 |
Activity |
nan |
None |
10.1016/j.ejphar.2004.09.032 |
| Homo sapiens |
Solute carrier family 22 member 8 |
Ki |
300000.0 |
nM |
10.1016/j.ejphar.2004.09.032 |
| Homo sapiens |
Solute carrier family 22 member 8 |
Km |
124000.0 |
nM |
10.1124/jpet.105.094052 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Inhibition |
97.53 |
% |
10.1124/mol.112.084152 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
Inhibition |
86.68 |
% |
10.1124/mol.112.084152 |
| Homo sapiens |
Sphingosine 1-phosphate receptor Edg-1 |
%Inhib (Mean) |
-31.41 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Sphingosine 1-phosphate receptor Edg-1 |
%Inhib (Mean) |
-29.61 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Sphingosine 1-phosphate receptor Edg-1 |
%Inhib (Mean) |
-23.13 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Sphingosine 1-phosphate receptor Edg-1 |
%Inhib (Mean) |
-16.6 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Sphingosine 1-phosphate receptor Edg-1 |
%Max (Mean) |
1.384 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Thromboxane A2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Thromboxane-A synthase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Thromboxane-A synthase |
Ki |
nan |
None |
None |
| Homo sapiens |
Thyroid stimulating hormone receptor |
Potency |
31622.8 |
nM |
None |
| Homo sapiens |
Transcription intermediary factor 1-alpha |
Delta TM |
0.08 |
C |
None |
| Homo sapiens |
Type-1 angiotensin II receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Type-1 angiotensin II receptor |
%Inhib (Mean) |
-11.32 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Type-1 angiotensin II receptor |
%Inhib (Mean) |
-4.185 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Type-1 angiotensin II receptor |
%Inhib (Mean) |
1.37 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Type-1 angiotensin II receptor |
%Inhib (Mean) |
5.92 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Type-1 angiotensin II receptor |
%Max (Mean) |
-7.139 |
% |
10.6019/CHEMBL5209801 |
| Homo sapiens |
Tyrosine-protein kinase ABL |
Delta TM |
-0.04 |
C |
None |
| Homo sapiens |
Tyrosine-protein kinase FYN |
IC50 |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase FYN |
Ki |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase LCK |
IC50 |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase LCK |
Ki |
nan |
None |
None |
| Homo sapiens |
Tyrosyl-DNA phosphodiesterase 1 |
Potency |
33498.3 |
nM |
None |
| Homo sapiens |
U2OS |
Growth Rate |
-1.0 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
U2OS |
Growth Rate |
0.18 |
None |
10.6019/CHEMBL5058564 |
| Homo sapiens |
Vascular endothelial growth factor receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vascular endothelial growth factor receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasoactive intestinal polypeptide receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vasoactive intestinal polypeptide receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasopressin V1a receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vasopressin V1a receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vasopressin V1a receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasopressin V2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vitamin D receptor |
Potency |
22387.2 |
nM |
None |
| Human immunodeficiency virus 1 |
Human immunodeficiency virus type 1 integrase |
Inhibition |
50.0 |
% |
10.1021/jm990322h |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Inhibition |
2.4 |
% |
10.6019/CHEMBL4513141 |
| Mus musculus |
Nitric oxide synthase, inducible |
IC50 |
nan |
None |
None |
| Mus musculus |
Nitric oxide synthase, inducible |
Ki |
nan |
None |
None |
| Mus musculus |
Solute carrier family 22 member 8 |
Activity |
75.0 |
% |
10.1124/dmd.32.5.479 |
| Oryctolagus cuniculus |
Angiotensin-converting enzyme |
IC50 |
nan |
None |
None |
| Oryctolagus cuniculus |
Angiotensin-converting enzyme |
Ki |
nan |
None |
None |
| Oryctolagus cuniculus |
Arachidonate 15-lipoxygenase |
IC50 |
nan |
None |
None |
| Oryctolagus cuniculus |
Arachidonate 15-lipoxygenase |
Ki |
nan |
None |
None |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
22750.0 |
nM |
10.1128/aac.00431-10 |
| Plasmodium falciparum |
Plasmodium falciparum |
Potency |
4256.2 |
nM |
None |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Inhibition |
4.47 |
% |
10.6019/CHEMBL4513141 |
| Rattus norvegicus |
Aldose reductase |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Aldose reductase |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1a adrenergic receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1a adrenergic receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1b adrenergic receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1b adrenergic receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Androgen Receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Androgen Receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Androgen Receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Bile salt export pump |
IC50 |
1000000.0 |
nM |
10.1124/dmd.111.040758 |
| Rattus norvegicus |
Cyclooxygenase-1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
GABA receptor alpha-1 subunit |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Glutamate (NMDA) receptor subunit zeta 1 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Glycine receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Glycine receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Inositol monophosphatase 1 |
Potency |
5011.9 |
nM |
None |
| Rattus norvegicus |
Insulin receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Insulin receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Nitric-oxide synthase, brain |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Nitric-oxide synthase, brain |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Peripheral myelin protein 22 |
Potency |
12579.7 |
nM |
None |
| Rattus norvegicus |
Plasma |
logFu |
0.83 |
None |
10.1016/j.ejmech.2009.06.004 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
32000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
33000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
34000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
35000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
36000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
41700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
43300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
44000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
44300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.3 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.4 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.5 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.6 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.7 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
326.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
343.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
383.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
396.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
577.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
609.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
664.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
722.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
794.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
808.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
809.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
814.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
838.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
851.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
861.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
873.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
883.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
885.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
896.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
898.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
907.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
917.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
918.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
921.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
928.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
940.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
987.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
990.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
998.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
999.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1002.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1057.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1062.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1109.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1126.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1146.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
26.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
28.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
28.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
30.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
30.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
32.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
32.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
32.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
33.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
33.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
33.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
36.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
36.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
38.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
39.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
39.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
40.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
40.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
55.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
56.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
57.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
59.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
18.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
18.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
18.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
18.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
21.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
21.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
21.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
22.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
22.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
23.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
56.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
59.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
59.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
59.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
60.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
61.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
62.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
62.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
62.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
63.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
64.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
64.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
64.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
64.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
65.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
65.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
65.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
65.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
66.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
66.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
66.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
66.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
67.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
68.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
68.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
69.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
71.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
71.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
85.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
87.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
89.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
90.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BASO |
0.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.52 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.56 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.64 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.68 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.7 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.72 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.74 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.76 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.78 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.82 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.86 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.88 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.92 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.94 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.96 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.98 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
1.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
1.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
1.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
84.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
86.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
88.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
92.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
94.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
96.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
98.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
100.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
102.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
108.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
132.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
134.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
138.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
142.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
144.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
146.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
152.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
154.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
156.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
158.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
160.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
163.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
164.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
166.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
170.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
174.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
180.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
186.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
99.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
102.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
103.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
104.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
105.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
106.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
107.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
108.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
109.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
103.67 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
106.33 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
106.67 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
578.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
593.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
624.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
626.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
670.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
678.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
686.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
706.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
724.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
730.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
732.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
738.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
742.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
746.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
746.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
750.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
760.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
762.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
766.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
772.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
774.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
776.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
780.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
786.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
790.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
806.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
812.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
818.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
820.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
828.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
838.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
852.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
853.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
213.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
218.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
259.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
662.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
102.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
102.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
24330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
25670000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
26330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
27330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
1.9 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
3.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
4.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
5.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
6.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ED50 |
3.5 |
mg.kg-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
ED50 |
100.0 |
mg.kg-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
121.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
169.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
179.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
254.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2046.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2098.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2132.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2174.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2176.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2178.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2184.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2186.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2194.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2206.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2214.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2220.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2222.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2234.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2240.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2250.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2252.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2254.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2258.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2262.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2280.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2282.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2294.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2296.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2300.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2322.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2324.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2336.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Flow rate |
43.4 |
ml min-1 100g-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Flow rate |
46.9 |
ml min-1 100g-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Flow rate |
50.5 |
ml min-1 100g-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Flow rate |
58.4 |
ml min-1 100g-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Flow rate |
60.5 |
ml min-1 100g-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Flow rate |
62.5 |
ml min-1 100g-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Flow rate |
68.6 |
ml min-1 100g-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Flow rate |
73.0 |
ml min-1 100g-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
0.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
0.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
2.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
2.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1523.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1620.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1794.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1820.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1826.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1828.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1836.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1862.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1864.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1894.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1904.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1906.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1924.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1928.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1938.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1942.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1944.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1950.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1952.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1962.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1966.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1972.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1978.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1994.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1996.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2006.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2008.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2052.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2056.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2080.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2082.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2174.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2178.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2200.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2418.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
32.47 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
34.6 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
34.9 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.73 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
42.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
43.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
43.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
43.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
44.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
121000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
129000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
131000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
131700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
132000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
133000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
134000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
134300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
135000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
136000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
137000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
139000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
139700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
143000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
144000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
154000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
155000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
157000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
7.9 |
% |
10.1021/jm00091a012 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
22.0 |
% |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
59.0 |
% |
10.1016/j.bmcl.2008.10.007 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
90.7 |
% |
10.1021/jm00091a012 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
96.0 |
% |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
62.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
123.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
125.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
132.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
132.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
135.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
137.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
138.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
150.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
151.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
153.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
160.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
162.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
165.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
176.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
176.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
177.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
181.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
183.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
184.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
185.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
186.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
188.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
190.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
190.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
193.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
194.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
194.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
196.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
198.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
202.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
203.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
204.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
205.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
230.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
250.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
8.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
8.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
9.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
9906.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
12766.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
13320.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
15699.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
64.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
65.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
71.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
71.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
73.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
74.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
74.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
75.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
76.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
76.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
77.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
77.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
79.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
79.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
79.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
80.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
80.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
82.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
82.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
84.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
85.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
90.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
92.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
19.4 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
19.7 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.8 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.2 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.5 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.7 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.8 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.1 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.2 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.3 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.4 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.5 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.6 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
23.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
23.73 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.43 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.87 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
372700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
380300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
385000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
54.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
55.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
56.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
56.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
59.8 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.8 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.5 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.57 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.2 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.63 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
48.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
74.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
113.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
233.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
0.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
0.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
1.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
1.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
1.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
5.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
8.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
11.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
12.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
13.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
13.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
17.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
17.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
17.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
18.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
18.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
19.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
19.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
20.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
22.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
24.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
26.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
29.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
713.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1366.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1405.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
2530.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
67.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
70.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
71.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
72.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
73.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
74.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
75.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
76.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
77.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
78.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
80.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
82.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
88.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
89.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
90.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
91.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
92.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
94.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
137.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
140.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
145.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
146.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1212.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1300.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1312.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1330.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1338.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1348.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1368.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1376.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1378.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1390.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1396.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1404.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1408.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1412.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1414.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1418.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1428.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1446.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1458.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1460.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1466.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1472.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1476.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1494.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1510.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1514.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1530.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1566.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1610.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
966000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
984000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1002000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1003000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1096000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1105000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1110000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1116000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1121000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1124000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1126000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1142000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1146000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1159670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1162000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1167000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1176000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1177000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1182000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1184000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1196000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1205000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1207000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1218000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1226000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1241000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1242000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1251000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1262000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1267000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1269000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1277000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1294000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1325670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1387000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
3.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
3.7 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
3.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
3.9 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.1 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.93 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.01 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.03 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
7.04 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
52000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
53000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
54000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
55000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
56000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
57000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
58700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
59000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
60000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
60700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
61000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
63000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
64000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5110000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5400000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5420000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5808000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5880000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5898000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5900000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5936000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5942000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5962000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5980000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5994000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6006000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6016000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6026000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6044000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6046000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6066000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6070000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6102000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6120000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6122000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6170000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6182000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6202000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6296000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6344000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6562000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6890000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6894000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6918000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7682000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7690000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7960000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7966000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
0.0 |
/100WBC |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
1.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
145.8 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
146.63 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
148.03 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
209.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
209.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
209.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
211.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
211.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
212.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
212.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
212.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
213.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
215.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
216.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
217.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
223.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
224.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
225.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
225.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
226.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
226.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
227.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
257.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
259.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
261.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
262.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
310.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
314.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
316.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
322.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
376.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
376.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
389.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
394.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Tissue Severity Score |
nan |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Tissue Severity Score |
nan |
None |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
272.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
462.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
466.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
476.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
508.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
518.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
558.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
566.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
600.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
624.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
632.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
668.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
674.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
694.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
722.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
776.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
784.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
796.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
826.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
828.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
856.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
862.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
868.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
910.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
964.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
974.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
982.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1018.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1114.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
11.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
16.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
21.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
23.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
6850.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7380.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7510.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7730.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7760.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7830.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8120.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8200.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8220.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8410.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8440.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8480.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8590.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8680.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8730.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8750.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9020.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9080.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9420.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9450.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9510.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9790.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9860.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10630.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10640.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10750.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11170.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11230.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11410.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11500.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11640.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11700.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
13830.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
16130.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
17430.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
0.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
13.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
15.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
15.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Serotonin 1a (5-HT1a) receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1a (5-HT1a) receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1b (5-HT1b) receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1b (5-HT1b) receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Voltage-gated L-type calcium channel alpha-1C subunit |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Voltage-gated N-type calcium channel alpha-1B subunit |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Severe acute respiratory syndrome coronavirus 2 |
Replicase polyprotein 1ab |
Inhibition |
11.54 |
% |
10.6019/CHEMBL4495564 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Hit score |
0.1617 |
None |
10.1101/2020.04.21.054387 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
19952.62 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
20000.0 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
-0.04 |
% |
10.6019/CHEMBL4495565 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
12.2 |
% |
10.21203/rs.3.rs-23951/v1 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition index |
0.07228 |
None |
10.1101/2020.04.03.023846 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
6.96 |
% |
10.6019/CHEMBL4513141 |
| Trypanosoma brucei |
6-phospho-1-fructokinase |
Potency |
37933.0 |
nM |
None |
| Trypanosoma cruzi |
Cruzipain |
Potency |
10000.0 |
nM |
None |
| Trypanosoma cruzi |
Cruzipain |
Potency |
12589.3 |
nM |
None |
| Trypanosoma cruzi |
Cruzipain |
Potency |
15848.9 |
nM |
None |
| Trypanosoma cruzi |
Cruzipain |
Potency |
25118.9 |
nM |
None |
| None |
ADMET |
CL |
6.6 |
mL.min-1.kg-1 |
10.1124/dmd.108.020479 |
| None |
ADMET |
delta logD |
-0.52 |
None |
10.1021/jm0000564 |
| None |
ADMET |
F |
49.0 |
% |
10.1021/jm0000564 |
| None |
ADMET |
log10(%HIA +10) |
1.681 |
None |
10.1016/j.ejmech.2010.11.005 |
| None |
ADMET |
Log Pe |
-4.6 |
cm s-1 |
10.1021/jm001020e |
| None |
ADMET |
Log Pe |
-4.3 |
cm s-1 |
10.1021/jm001020e |
| None |
ADMET |
MRT |
3.0 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
permeability |
0.6 |
10'-6 cm/s |
10.1021/jm901421c |
| None |
ADMET |
PPB |
20.0 |
% |
10.1021/acs.jmedchem.0c00046 |
| None |
ADMET |
T1/2 |
2.8 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
Vdss |
1.2 |
L.kg-1 |
10.1124/dmd.108.020479 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Index Value |
0.8 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Active |
0.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Marginal |
0.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Index Value |
0.4 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1021/tx1000865 |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1021/tx900326k |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1124/dmd.110.035113 |
| None |
Hepatotoxicity |
HepSE_bilirubinemia |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholecystitis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholelithiasis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cirrhosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_Combined Scores |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_elevated liver function tests |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic failure |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic necrosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatitis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatomegaly |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_jaundice |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver disease |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver fatty |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver function tests abnormal |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
LDH Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LDH Increase - Index Value |
0.4 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LDH Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LTKB_BD DILI severity score |
3.0 |
None |
10.1016/j.drudis.2011.05.007 |
| None |
Hepatotoxicity |
SGOT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Index Value |
0.8 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Index Value |
0.7 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
NON-PROTEIN TARGET |
Fu |
0.84 |
None |
10.1124/dmd.108.020479 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (acute) |
0.0 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (animal toxicity known) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (benign tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (granulomatous hepatitis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (mechanism) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
2.8 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
12.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (time to onset) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Potency |
0.7 |
nM |
None |
| None |
NON-PROTEIN TARGET |
Potency |
6.0 |
nM |
None |
| None |
NON-PROTEIN TARGET |
Potency |
10583.9 |
nM |
None |
| None |
No relevant target |
LogD |
-1.27 |
None |
10.1021/jm0000564 |
| None |
No relevant target |
LogD |
-0.8 |
None |
10.1021/jm001020e |
| None |
No relevant target |
LogD7.4 |
-0.6 |
None |
10.6019/CHEMBL3301361 |
| None |
No relevant target |
pKa |
7.1 |
None |
10.1016/j.ejmech.2009.06.004 |
| None |
No relevant target |
pKa |
7.1 |
None |
10.1021/jm0000564 |
| None |
No relevant target |
Solubility |
760.0 |
ug.mL-1 |
10.1016/j.bmc.2010.08.003 |
| None |
Phospholipidosis |
Phospholipidosis |
nan |
None |
10.1021/ci6004542 |
| None |
Phospholipidosis |
Phospholipidosis |
nan |
None |
10.1021/mp100103e |
| None |
Unchecked |
Ac50 |
0.7943 |
uM |
None |
| None |
Unchecked |
Ac50 |
1.778 |
uM |
None |
| None |
Unchecked |
Ac50 |
25.12 |
uM |
None |
| None |
Unchecked |
AC50 |
794.3 |
nM |
None |
| None |
Unchecked |
AC50 |
1780.0 |
nM |
None |
| None |
Unchecked |
AC50 |
25118.9 |
nM |
None |
| None |
Unchecked |
Hepatotoxicity (acute) |
5.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (association with vascular disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (choleostasis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (chronic liver disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cirrhosis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (comment) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cytolytic) |
4.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (malignant tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (severe hepatitis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (steatosis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (successful reintroduction) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
IC50 |
nan |
None |
None |
| None |
Unchecked |
Inhibition |
nan |
% |
10.1038/nchembio873 |
| None |
Unchecked |
Ki |
20.7 |
nM |
10.1021/acsmedchemlett.8b00334 |
| None |
Unchecked |
Ki |
49.8 |
nM |
10.1021/acsmedchemlett.8b00334 |
| None |
Unchecked |
Ki |
nan |
None |
None |
| None |
Unchecked |
Potency |
2511.9 |
nM |
None |
| None |
Unchecked |
Potency |
15848.9 |
nM |
None |
| None |
Unchecked |
Ratio |
34.2 |
None |
10.1021/acs.jmedchem.0c02047 |
| None |
Unchecked |
Ratio IC50 |
5.0 |
None |
10.1021/jm301302s |