| Bos mutus |
Dipeptidyl peptidase 3 |
IC50 |
300000.0 |
nM |
10.1007/s00044-010-9454-7 |
| Bos mutus |
Dipeptidyl peptidase 3 |
Inhibition |
96.0 |
% |
10.1007/s00044-010-9454-7 |
| Bos mutus |
Dipeptidyl peptidase 3 |
Ki |
245000.0 |
nM |
10.1007/s00044-010-9454-7 |
| Bos taurus |
Progesterone receptor |
IC50 |
nan |
None |
None |
| Bos taurus |
Progesterone receptor |
Ki |
nan |
None |
None |
| Canis lupus familiaris |
MDCK |
logPapp |
-4.04 |
None |
10.1021/jm901846t |
| Cavia porcellus |
Leukotriene C4 synthase |
IC50 |
nan |
None |
None |
| Cavia porcellus |
Leukotriene C4 synthase |
Ki |
nan |
None |
None |
| Cavia porcellus |
Serotonin 4 (5-HT4) receptor |
IC50 |
nan |
None |
None |
| Cavia porcellus |
Serotonin 4 (5-HT4) receptor |
Ki |
nan |
None |
None |
| Cryptosporidium parvum |
Cryptosporidium parvum |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Danio rerio |
Danio rerio |
Activity |
nan |
None |
10.1016/j.bmcl.2014.07.050 |
| Entamoeba histolytica |
Entamoeba histolytica |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Gallus gallus |
Chorioallantoic membrane |
ID50 |
396.9 |
fmol |
10.1016/j.bmcl.2014.05.005 |
| Gallus gallus |
Chorioallantoic membrane |
Inhibition |
77.9 |
% |
10.1016/j.bmcl.2014.05.005 |
| Homo sapiens |
5-lipoxygenase activating protein |
IC50 |
44000.0 |
nM |
10.1021/jm800197b |
| Homo sapiens |
Acetylcholinesterase |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Acetylcholinesterase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Acetylcholinesterase |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A2a receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A2a receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A2a receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A3 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A3 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Aldehyde dehydrogenase 1A1 |
Potency |
28183.8 |
nM |
None |
| Homo sapiens |
Aldo-keto-reductase family 1 member C3 |
Inhibition |
8.0 |
% |
10.1016/j.bmcl.2005.08.063 |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1d adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-1d adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2b adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2b adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2b adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2c adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2c adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2c adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Androgen Receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Angiotensin II type 2 (AT-2) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Angiotensin II type 2 (AT-2) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
ATPase family AAA domain-containing protein 5 |
Potency |
20587.8 |
nM |
None |
| Homo sapiens |
ATPase family AAA domain-containing protein 5 |
Potency |
23099.9 |
nM |
None |
| Homo sapiens |
Beta-1 adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-1 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-1 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-2 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-3 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-3 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Bile acid receptor FXR |
AC50 |
26999.8 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bile acid receptor FXR |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bile salt export pump |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bile salt export pump |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Bile salt export pump |
IC50 |
135000.0 |
nM |
10.1093/toxsci/kfq269 |
| Homo sapiens |
Bile salt export pump |
IC50 |
1000000.0 |
nM |
10.1124/dmd.111.040758 |
| Homo sapiens |
Bile salt export pump |
IC50 |
1000000.0 |
nM |
10.1124/dmd.112.047068 |
| Homo sapiens |
Blood |
IC50 |
44000.0 |
nM |
10.1021/jm800197b |
| Homo sapiens |
Blood |
IC50 |
94000.0 |
nM |
10.1021/jm800197b |
| Homo sapiens |
Bradykinin B2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Bradykinin B2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Bromodomain-containing protein 2 |
Activity |
11.0 |
% |
10.1021/jm201320w |
| Homo sapiens |
Bromodomain-containing protein 2 |
Activity |
nan |
None |
10.1021/jm201320w |
| Homo sapiens |
Bromodomain-containing protein 2 |
Inhibition |
6.0 |
% |
10.1021/jm201320w |
| Homo sapiens |
Bromodomain-containing protein 3 |
Activity |
7.0 |
% |
10.1021/jm201320w |
| Homo sapiens |
Bromodomain-containing protein 3 |
Inhibition |
19.0 |
% |
10.1021/jm201320w |
| Homo sapiens |
Bromodomain-containing protein 4 |
Activity |
5.0 |
% |
10.1021/jm201320w |
| Homo sapiens |
Bromodomain-containing protein 4 |
Inhibition |
12.0 |
% |
10.1021/jm201320w |
| Homo sapiens |
Bromodomain-containing protein 4 |
Kd |
250000.0 |
nM |
10.1039/C5MD00209E |
| Homo sapiens |
Caco-2 |
logPapp |
-4.0 |
None |
10.1016/j.bmc.2011.03.011 |
| Homo sapiens |
Calcitonin receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Calcitonin receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Canalicular multispecific organic anion transporter 1 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 2 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Cannabinoid CB1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cannabinoid CB1 receptor |
Activity |
13.0 |
% |
10.1021/jm800807k |
| Homo sapiens |
Cannabinoid CB1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cannabinoid CB1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Cannabinoid CB2 receptor |
Activity |
15.0 |
% |
10.1021/jm800807k |
| Homo sapiens |
Carbonic anhydrase I |
Ki |
10000.0 |
nM |
10.1016/j.bmc.2008.06.013 |
| Homo sapiens |
Carbonic anhydrase I |
Ki |
10000.0 |
nM |
10.1016/j.bmcl.2008.04.077 |
| Homo sapiens |
Carbonic anhydrase I |
Ki |
10000.0 |
nM |
10.1016/j.bmcl.2015.10.021 |
| Homo sapiens |
Carbonic anhydrase II |
IC50 |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase II |
Ki |
6200.0 |
nM |
10.1016/j.bmc.2008.06.013 |
| Homo sapiens |
Carbonic anhydrase II |
Ki |
6200.0 |
nM |
10.1016/j.bmcl.2008.04.077 |
| Homo sapiens |
Carbonic anhydrase II |
Ki |
6200.0 |
nM |
10.1016/j.bmcl.2015.10.021 |
| Homo sapiens |
Carbonic anhydrase II |
Ki |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase III |
Ki |
7100.0 |
nM |
10.1016/j.bmc.2008.06.013 |
| Homo sapiens |
Carbonic anhydrase IV |
Ki |
11400.0 |
nM |
10.1016/j.bmc.2008.06.013 |
| Homo sapiens |
Carbonic anhydrase IX |
Ki |
70700.0 |
nM |
10.1016/j.bmc.2008.06.013 |
| Homo sapiens |
Carbonic anhydrase IX |
Ki |
70700.0 |
nM |
10.1016/j.bmcl.2015.10.021 |
| Homo sapiens |
Carbonic anhydrase VA |
Ki |
802000.0 |
nM |
10.1016/j.bmc.2008.06.013 |
| Homo sapiens |
Carbonic anhydrase VB |
Ki |
296000.0 |
nM |
10.1016/j.bmc.2008.06.013 |
| Homo sapiens |
Carbonic anhydrase VI |
Ki |
658000.0 |
nM |
10.1016/j.bmc.2008.06.013 |
| Homo sapiens |
Carbonic anhydrase VII |
Ki |
9100.0 |
nM |
10.1016/j.bmc.2008.06.013 |
| Homo sapiens |
Carbonic anhydrase XII |
Ki |
4100.0 |
nM |
10.1016/j.bmc.2008.06.013 |
| Homo sapiens |
Carbonic anhydrase XIV |
Ki |
10600.0 |
nM |
10.1016/j.bmc.2008.06.013 |
| Homo sapiens |
Caspase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Caspase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cathepsin G |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cathepsin G |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 2 |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 4 |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin A receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cholecystokinin A receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin A receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Cholesterol 24-hydroxylase |
Activity |
132.0 |
% |
None |
| Homo sapiens |
Chromobox protein homolog 1 |
Potency |
39810.7 |
nM |
None |
| Homo sapiens |
Cyclooxygenase |
Control |
67.0 |
% |
10.1021/jm00385a031 |
| Homo sapiens |
Cyclooxygenase-1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-1 |
Activity |
nan |
None |
10.1021/jm800807k |
| Homo sapiens |
Cyclooxygenase-1 |
IC50 |
200000.0 |
nM |
10.1021/acs.jmedchem.6b00078 |
| Homo sapiens |
Cyclooxygenase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-2 |
IC50 |
141000.0 |
nM |
10.1021/jm800807k |
| Homo sapiens |
Cyclooxygenase-2 |
IC50 |
141253.75 |
nM |
10.1021/jm800807k |
| Homo sapiens |
Cyclooxygenase-2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-2 |
INH |
26.0 |
uM |
10.1021/jm201320w |
| Homo sapiens |
Cyclooxygenase-2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cysteinyl leukotriene receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cysteinyl leukotriene receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A1 |
Kcat |
0.84 |
/min |
10.1124/dmd.112.047308 |
| Homo sapiens |
Cytochrome P450 1A1 |
Kcat/Km |
0.001 |
None |
10.1124/dmd.112.047308 |
| Homo sapiens |
Cytochrome P450 1A1 |
Kd |
19100.0 |
nM |
10.1016/j.ejmech.2010.07.055 |
| Homo sapiens |
Cytochrome P450 1A1 |
Km |
803000.0 |
nM |
10.1124/dmd.112.047308 |
| Homo sapiens |
Cytochrome P450 1A2 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
IC50 |
25000.0 |
nM |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
Inhibition |
10.0 |
% |
10.1124/dmd.111.039180 |
| Homo sapiens |
Cytochrome P450 1A2 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 1A2 |
Kcat |
2.2 |
/min |
10.1124/dmd.112.047308 |
| Homo sapiens |
Cytochrome P450 1A2 |
Kcat/Km |
0.018 |
None |
10.1124/dmd.112.047308 |
| Homo sapiens |
Cytochrome P450 1A2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
Km |
120000.0 |
nM |
10.1124/dmd.112.047308 |
| Homo sapiens |
Cytochrome P450 2A6 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2A6 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2B6 |
Inhibition |
10.0 |
% |
10.1124/dmd.111.039180 |
| Homo sapiens |
Cytochrome P450 2C19 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
Inhibition |
10.0 |
% |
10.1124/dmd.111.039180 |
| Homo sapiens |
Cytochrome P450 2C19 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2C19 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C8 |
Inhibition |
10.0 |
% |
10.1124/dmd.111.039180 |
| Homo sapiens |
Cytochrome P450 2C9 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
Inhibition |
10.0 |
% |
10.1124/dmd.111.039180 |
| Homo sapiens |
Cytochrome P450 2C9 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2C9 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
IC50 |
10000.0 |
nM |
10.1016/j.ejmech.2020.112600 |
| Homo sapiens |
Cytochrome P450 2D6 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
Inhibition |
10.0 |
% |
10.1124/dmd.111.039180 |
| Homo sapiens |
Cytochrome P450 2D6 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2D6 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2E1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2E1 |
Inhibition |
50.0 |
% |
10.1016/j.ejmech.2020.112600 |
| Homo sapiens |
Cytochrome P450 2E1 |
Inhibition |
nan |
% |
10.1016/j.bmcl.2018.09.020 |
| Homo sapiens |
Cytochrome P450 2E1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2J2 |
IC50 |
50000.0 |
nM |
10.1124/dmd.112.048264 |
| Homo sapiens |
Cytochrome P450 3A4 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
IC50 |
10000.0 |
nM |
10.1016/j.ejmech.2020.112600 |
| Homo sapiens |
Cytochrome P450 3A4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
Inhibition |
10.0 |
% |
10.1124/dmd.111.039180 |
| Homo sapiens |
Cytochrome P450 3A4 |
Inhibition |
50.0 |
% |
10.1016/j.ejmech.2020.112600 |
| Homo sapiens |
Cytochrome P450 3A4 |
Inhibition |
nan |
% |
10.1016/j.bmcl.2018.09.020 |
| Homo sapiens |
Cytochrome P450 3A4 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 3A4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
Potency |
15848.9 |
nM |
None |
| Homo sapiens |
Delta opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Delta opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Delta opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D3 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D3 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D4 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D4 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Endothelin receptor ET-A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-A |
Ki |
nan |
None |
None |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Equilibrative nucleoside transporter 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor alpha |
Potency |
31622.8 |
nM |
None |
| Homo sapiens |
Estrogen receptor beta |
IC50 |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor beta |
Ki |
nan |
None |
None |
| Homo sapiens |
Gamma-aminobutyric acid receptor subunit alpha-1/alpha-2/beta-2/gamma-2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Ghrelin receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Glucocorticoid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Glutaminase kidney isoform, mitochondrial |
Potency |
17782.8 |
nM |
None |
| Homo sapiens |
Glutaminase kidney isoform, mitochondrial |
Potency |
28183.8 |
nM |
None |
| Homo sapiens |
HepaRG |
Activity |
nan |
None |
10.1016/j.bmcl.2018.09.020 |
| Homo sapiens |
HepaRG |
Activity |
nan |
None |
10.1016/j.ejmech.2020.112600 |
| Homo sapiens |
Hepatocyte |
Activity |
nan |
None |
10.1016/j.bmc.2006.07.054 |
| Homo sapiens |
Hepatocyte |
Activity |
nan |
None |
10.1016/j.ejmech.2020.112600 |
| Homo sapiens |
Hepatocyte |
CL |
4.0 |
mL.min-1.kg-1 |
10.1016/j.ejmech.2008.07.027 |
| Homo sapiens |
Hepatocyte |
logCL |
0.6021 |
None |
10.1016/j.ejmech.2008.07.027 |
| Homo sapiens |
HepG2 |
Activity |
nan |
None |
10.1016/j.bmc.2006.07.054 |
| Homo sapiens |
HepG2 |
EC50 |
594000.0 |
nM |
10.1021/ml4000904 |
| Homo sapiens |
HERG |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
HERG |
IC50 |
nan |
None |
None |
| Homo sapiens |
HERG |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Histamine H1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Histamine H2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histone deacetylase 6 |
Inhibition |
-27.16 |
% |
10.6019/CHEMBL4808148 |
| Homo sapiens |
Histone deacetylase 6 |
Inhibition |
-2.28 |
% |
10.6019/CHEMBL4808148 |
| Homo sapiens |
HMG-CoA reductase |
IC50 |
nan |
None |
None |
| Homo sapiens |
HMG-CoA reductase |
Ki |
nan |
None |
None |
| Homo sapiens |
Homo sapiens |
Activity |
0.8 |
% |
10.1016/j.ejmech.2009.11.034 |
| Homo sapiens |
Homo sapiens |
Activity |
1.3 |
None |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
Activity |
nan |
None |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
AUC |
3700.0 |
ng.hr.mL-1 |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
AUC |
21000.0 |
ng.hr.mL-1 |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
AUC |
28000.0 |
ng.hr.mL-1 |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
AUC |
36700.0 |
ng.hr.mL-1 |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
AUC |
66000.0 |
ng.hr.mL-1 |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
AUC |
77800.0 |
ng.hr.mL-1 |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
CL |
4.9 |
mL.min-1.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
CL |
5.0 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
CL |
5.0 |
mL.min-1.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
CL |
5.45 |
mL.min-1.kg-1 |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
CL |
13.0 |
ml/min |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
CL |
380.0 |
ml/min |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
CL/F |
13.2 |
L/hr |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
CL/F |
18.7 |
L/hr |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
CL/F |
365.0 |
mL/min |
None |
| Homo sapiens |
Homo sapiens |
CL_renal |
0.15 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
CL_renal |
0.2 |
mL.min-1.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Cmax |
27785.13 |
nM |
None |
| Homo sapiens |
Homo sapiens |
Cmax |
117094.47 |
nM |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
DILI_Concern |
nan |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
DILI_severity_class |
5.0 |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
Drug metabolism |
0.2 |
ug ml-1 |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
Drug recovery |
5.0 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
6.4 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
6.9 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
8.0 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
8.1 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
8.2 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
8.6 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
8.7 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
9.1 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
9.3 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
9.4 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
9.7 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
10.1 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
10.3 |
g |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
10.6 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
11.2 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
11.8 |
g |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
11.9 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
13.0 |
g |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
13.3 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
13.4 |
g |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
13.7 |
g |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
13.8 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
14.5 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
14.5 |
g |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
15.2 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
16.5 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
32.3 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
54.7 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
60.9 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
63.6 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
66.5 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
68.9 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
72.4 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
73.9 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
75.3 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug recovery |
93.0 |
%ID |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Drug uptake |
6.7 |
ug ml-1 |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
Drug uptake |
120.0 |
ug ml-1 |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
EC50 |
2.0 |
ug.mL-1 |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
Emax |
4.6 |
None |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
F |
75.0 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
F |
76.0 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
F |
85.0 |
% |
10.1021/jm901846t |
| Homo sapiens |
Homo sapiens |
F |
88.0 |
% |
10.1016/j.bmc.2007.08.060 |
| Homo sapiens |
Homo sapiens |
Fa |
1.0 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
F_fraction |
0.82 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Fg |
1.04 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Fh |
0.79 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
ka |
2.4 |
L/hr |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
Kel |
1.3 |
L/hr |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
T1/2 |
0.13 |
hr |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
T1/2 |
0.53 |
hr |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
T1/2 |
0.88 |
hr |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.3 |
hr |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.97 |
hr |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.98 |
hr |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.0 |
hr |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.17 |
hr |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.5 |
hr |
None |
| Homo sapiens |
Homo sapiens |
Tmax |
0.25 |
hr |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Tmax |
0.5 |
hr |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
Tmax |
0.9 |
hr |
None |
| Homo sapiens |
Homo sapiens |
Vd |
0.509 |
L.kg-1 |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Vd |
0.9 |
L.kg-1 |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Vd |
65.0 |
l |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Vd/F |
30.9 |
l |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
Vd/F |
69.7 |
l |
10.1248/bpb.30.157 |
| Homo sapiens |
Homo sapiens |
Vdss |
0.897 |
L.kg-1 |
10.1111/j.1365-2125.1980.tb01812.x |
| Homo sapiens |
Homo sapiens |
Vdss |
0.95 |
L.kg-1 |
10.1016/j.ejmech.2009.06.004 |
| Homo sapiens |
Homo sapiens |
Vdss |
1.0 |
L.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
HUVEC |
Activity |
25.93 |
% |
10.1016/j.bmcl.2017.07.036 |
| Homo sapiens |
HUVEC |
Activity |
nan |
None |
10.1016/j.bmcl.2017.07.036 |
| Homo sapiens |
HUVEC |
Inhibition |
10.47 |
% |
10.1016/j.bmcl.2017.07.036 |
| Homo sapiens |
Interleukin-8 receptor A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor A |
Ki |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor B |
IC50 |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor B |
Ki |
nan |
None |
None |
| Homo sapiens |
Kappa opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Kappa opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
KB |
TD50 |
nan |
None |
10.1021/jm7009292 |
| Homo sapiens |
L02 |
Activity |
nan |
None |
10.1021/acs.jnatprod.0c01117 |
| Homo sapiens |
Leukocyte common antigen |
IC50 |
nan |
None |
None |
| Homo sapiens |
Leukocyte common antigen |
Ki |
nan |
None |
None |
| Homo sapiens |
Leukocyte elastase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Leukocyte elastase |
Ki |
nan |
None |
None |
| Homo sapiens |
Liver |
Stability |
74.5 |
% |
10.1039/c5md00349k |
| Homo sapiens |
Liver |
T1/2 |
4.4 |
hr |
10.1039/c5md00349k |
| Homo sapiens |
Liver microsome |
CL |
0.000198 |
mL.min-1.g-1 |
10.1124/dmd.111.039180 |
| Homo sapiens |
Liver microsome |
Drug metabolism |
19.8 |
pmol/min |
10.1124/dmd.111.039180 |
| Homo sapiens |
Liver microsome |
PB |
71.3 |
pmol |
10.1124/dmd.111.039180 |
| Homo sapiens |
Liver microsome |
Retention_time |
3.3 |
min |
10.1124/dmd.111.044057 |
| Homo sapiens |
Liver microsomes |
Activity |
113.0 |
pmol |
10.1021/tx300075j |
| Homo sapiens |
Liver microsomes |
Stability |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
LXR-alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
LXR-beta |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
MAP kinase ERK1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK1 |
Ki |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK2 |
Ki |
nan |
None |
None |
| Homo sapiens |
MAP kinase p38 alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase p38 alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase 9 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase 9 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 3 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Melanocortin receptor 3 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 3 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Menin/Histone-lysine N-methyltransferase MLL |
Potency |
39810.7 |
nM |
None |
| Homo sapiens |
Microtubule-associated protein tau |
Potency |
44668.4 |
nM |
None |
| Homo sapiens |
Monoamine oxidase A |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Monoamine oxidase A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Monoamine oxidase A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Monoamine oxidase A |
Ki |
nan |
None |
None |
| Homo sapiens |
Monoglyceride lipase |
Inhibition |
20.0 |
% |
10.1021/jm901891p |
| Homo sapiens |
Monoglyceride lipase |
Inhibition |
34.0 |
% |
10.1021/jm901891p |
| Homo sapiens |
Mothers against decapentaplegic homolog 3 |
Potency |
3548.1 |
nM |
None |
| Homo sapiens |
Motilin receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Multidrug resistance-associated protein 4 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Mu opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Mu opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Mu opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Myoglobin |
IC50 |
2300.0 |
nM |
10.1021/ml4000904 |
| Homo sapiens |
Neurokinin 1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neurokinin 1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurokinin 2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neurokinin 2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Neuronal acetylcholine receptor protein alpha-4 subunit |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Norepinephrine transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Norepinephrine transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Norepinephrine transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Nuclear receptor ROR-gamma |
Potency |
21131.7 |
nM |
None |
| Homo sapiens |
Nuclear receptor subfamily 1 group I member 3 |
AC50 |
15000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Peroxisome proliferator-activated receptor alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Peroxisome proliferator-activated receptor gamma |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
nan |
None |
10.1016/s0378-5173(03)00372-7 |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
nan |
None |
10.1021/tx010125x |
| Homo sapiens |
Phosphodiesterase 3A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 4A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 4D |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 5A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Phosphodiesterase 5A |
Ki |
nan |
None |
None |
| Homo sapiens |
Plasma |
fCmax |
165.39 |
uM |
10.1124/dmd.111.040758 |
| Homo sapiens |
Platelet activating factor receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Platelet activating factor receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Pregnane X receptor |
AC50 |
23999.9 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Pregnane X receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Progesterone receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Protein kinase C alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
Protein kinase C alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Retinoic acid receptor alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Retinoic acid receptor beta |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Retinoic acid receptor gamma |
AC50 |
25999.8 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Retinoic acid receptor gamma |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 1a (5-HT1a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 3a (5-HT3a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Serum albumin |
Log K' |
0.81 |
None |
10.1021/jm010960b |
| Homo sapiens |
Sigma opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Sigma opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Skin |
log Kp |
-7.22 |
None |
10.1016/j.bmc.2007.07.050 |
| Homo sapiens |
Solute carrier family 22 member 1 |
Inhibition |
-9.2 |
% |
10.1021/jm8003152 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Inhibition |
99.98 |
% |
10.1124/mol.112.084152 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
Inhibition |
96.68 |
% |
10.1124/mol.112.084152 |
| Homo sapiens |
Sulfotransferase 1A1 |
Activity |
nan |
None |
None |
| Homo sapiens |
Thrombin |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Thromboxane A2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Thromboxane-A synthase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Thromboxane-A synthase |
Ki |
nan |
None |
None |
| Homo sapiens |
Thyroid stimulating hormone receptor |
Potency |
158.5 |
nM |
None |
| Homo sapiens |
Type-1 angiotensin II receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Tyrosine-protein kinase FYN |
IC50 |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase FYN |
Ki |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase LCK |
IC50 |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase LCK |
Ki |
nan |
None |
None |
| Homo sapiens |
UDP-glucuronosyltransferase 1-1 |
Activity |
0.0 |
pm/min/mg |
10.1146/annurev.pharmtox.40.1.581 |
| Homo sapiens |
UDP-glucuronosyltransferase 1-1 |
Activity |
nan |
None |
None |
| Homo sapiens |
UDP-glucuronosyltransferase 1-1 |
Km |
9400000.0 |
nM |
10.1016/j.pharmthera.2004.10.013 |
| Homo sapiens |
UDP-glucuronosyltransferase 1-1 |
Vmax |
1300.0 |
pmol/min/mg protein |
10.1016/j.pharmthera.2004.10.013 |
| Homo sapiens |
UDP-glucuronosyltransferase 1-10 |
Activity |
0.0 |
pm/min/mg |
10.1146/annurev.pharmtox.40.1.581 |
| Homo sapiens |
UDP-glucuronosyltransferase 1-6 |
Activity |
nan |
None |
None |
| Homo sapiens |
UDP-glucuronosyltransferase 1-6 |
Km |
2200000.0 |
nM |
10.1016/j.pharmthera.2004.10.013 |
| Homo sapiens |
UDP-glucuronosyltransferase 1-6 |
Vmax |
100.0 |
pmol/min/mg protein |
10.1016/j.pharmthera.2004.10.013 |
| Homo sapiens |
UDP-glucuronosyltransferase 1-7 |
Activity |
0.0 |
pm/min/mg |
10.1146/annurev.pharmtox.40.1.581 |
| Homo sapiens |
UDP-glucuronosyltransferase 1-8 |
Activity |
0.0 |
pm/min/mg |
10.1146/annurev.pharmtox.40.1.581 |
| Homo sapiens |
UDP-glucuronosyltransferase 1-9 |
Activity |
nan |
None |
None |
| Homo sapiens |
UDP-glucuronosyltransferase 1-9 |
Km |
20900000.0 |
nM |
10.1016/j.pharmthera.2004.10.013 |
| Homo sapiens |
UDP-glucuronosyltransferase 1-9 |
Vmax |
6300.0 |
pmol/min/mg protein |
10.1016/j.pharmthera.2004.10.013 |
| Homo sapiens |
UDP-glucuronosyltransferase 1A4 |
Activity |
0.0 |
pm/min/mg |
10.1146/annurev.pharmtox.40.1.581 |
| Homo sapiens |
UDP-glucuronosyltransferase 2B10 |
Activity |
0.0 |
pm/min/mg |
10.1146/annurev.pharmtox.40.1.581 |
| Homo sapiens |
UDP-glucuronosyltransferase 2B15 |
Activity |
0.0 |
pm/min/mg |
10.1146/annurev.pharmtox.40.1.581 |
| Homo sapiens |
UDP-glucuronosyltransferase 2B4 |
Activity |
0.0 |
pm/min/mg |
10.1146/annurev.pharmtox.40.1.581 |
| Homo sapiens |
UDP-glucuronosyltransferase 2B7 |
Activity |
0.0 |
pm/min/mg |
10.1146/annurev.pharmtox.40.1.581 |
| Homo sapiens |
Vascular endothelial growth factor receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vascular endothelial growth factor receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Vascular endothelial growth factor receptor 2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vasoactive intestinal polypeptide receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vasoactive intestinal polypeptide receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasopressin V1a receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vasopressin V1a receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vasopressin V1a receptor |
Ki |
nan |
None |
None |
| Leishmania amazonensis |
Leishmania amazonensis |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Leishmania donovani |
Leishmania donovani |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Leishmania infantum |
Leishmania infantum |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Leishmania major |
Leishmania major |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Leishmania mexicana |
Leishmania mexicana |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Mus musculus |
Carbonic anhydrase 15 |
Ki |
9230.0 |
nM |
10.1016/j.bmcl.2008.04.077 |
| Mus musculus |
Carbonic anhydrase XIII |
Ki |
30300.0 |
nM |
10.1016/j.bmc.2008.06.013 |
| Mus musculus |
L1210 |
Activity |
15.0 |
% |
10.1021/jm050567w |
| Mus musculus |
L1210 |
log(1/ID50) |
3.73 |
None |
10.1021/jm050567w |
| Mus musculus |
Liver |
Stability |
97.7 |
% |
10.1021/acs.jmedchem.6b00015 |
| Mus musculus |
Monoamine oxidase A |
Activity |
nan |
None |
10.1021/jm800656v |
| Mus musculus |
Monoamine oxidase B |
Activity |
nan |
None |
10.1021/jm800656v |
| Mus musculus |
Mus musculus |
Activity |
-1.1 |
degrees C |
10.1016/j.ejmech.2009.02.026 |
| Mus musculus |
Mus musculus |
Activity |
13.0 |
% |
10.1016/j.bmcl.2007.07.058 |
| Mus musculus |
Mus musculus |
Activity |
13.0 |
% |
10.1016/j.ejmech.2020.113042 |
| Mus musculus |
Mus musculus |
Activity |
17.0 |
% |
10.1016/j.ejmech.2020.113042 |
| Mus musculus |
Mus musculus |
Activity |
18.0 |
% |
10.1016/j.ejmech.2020.113042 |
| Mus musculus |
Mus musculus |
Activity |
34.0 |
% |
10.1016/j.ejmech.2009.02.026 |
| Mus musculus |
Mus musculus |
Activity |
36.0 |
% |
10.1016/j.ejmech.2020.113042 |
| Mus musculus |
Mus musculus |
Activity |
40.0 |
% |
10.1016/j.bmc.2006.07.054 |
| Mus musculus |
Mus musculus |
Activity |
47.0 |
% |
10.1021/jm800807k |
| Mus musculus |
Mus musculus |
Activity |
47.76 |
% |
10.1016/j.ejmech.2008.03.043 |
| Mus musculus |
Mus musculus |
Activity |
51.61 |
% |
10.1007/s00044-010-9300-y |
| Mus musculus |
Mus musculus |
Activity |
51.8 |
% |
10.1016/j.ejmech.2009.02.026 |
| Mus musculus |
Mus musculus |
Activity |
54.6 |
% |
10.1016/j.ejmech.2009.02.026 |
| Mus musculus |
Mus musculus |
Activity |
60.6 |
% |
10.1016/j.ejmech.2009.02.026 |
| Mus musculus |
Mus musculus |
Activity |
61.32 |
% |
10.1016/j.bmc.2006.07.054 |
| Mus musculus |
Mus musculus |
Activity |
100.0 |
% |
10.1021/jm800807k |
| Mus musculus |
Mus musculus |
Activity |
299.01 |
U/ml |
10.1016/j.bmc.2006.07.054 |
| Mus musculus |
Mus musculus |
Activity |
nan |
None |
10.1007/s00044-010-9300-y |
| Mus musculus |
Mus musculus |
Activity |
nan |
None |
10.1016/j.bmc.2006.07.054 |
| Mus musculus |
Mus musculus |
Activity |
nan |
None |
10.1016/j.bmc.2008.08.019 |
| Mus musculus |
Mus musculus |
Activity |
nan |
None |
10.1016/j.bmcl.2018.09.020 |
| Mus musculus |
Mus musculus |
Activity |
nan |
None |
10.1016/j.ejmech.2009.02.026 |
| Mus musculus |
Mus musculus |
Activity |
nan |
None |
10.1016/j.ejmech.2020.112600 |
| Mus musculus |
Mus musculus |
Activity |
nan |
None |
10.1016/j.ejmech.2020.113042 |
| Mus musculus |
Mus musculus |
Activity |
nan |
None |
10.1021/np9804177 |
| Mus musculus |
Mus musculus |
Administered dose |
0.4 |
% |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Administered dose |
1.1 |
% |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Administered dose |
2.0 |
% |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Administered dose |
2.3 |
% |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Administered dose |
18.5 |
% |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Administered dose |
68.8 |
% |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
BBR |
0.68 |
None |
10.1016/j.bmcl.2006.01.033 |
| Mus musculus |
Mus musculus |
Deaths |
11.0 |
None |
10.1021/jm00347a001 |
| Mus musculus |
Mus musculus |
Dose |
59.8 |
% |
10.1021/jm00140a014 |
| Mus musculus |
Mus musculus |
Drug uptake |
43.0 |
uM |
10.1016/j.bmcl.2006.01.033 |
| Mus musculus |
Mus musculus |
Drug uptake |
64.0 |
uM |
10.1016/j.bmcl.2006.01.033 |
| Mus musculus |
Mus musculus |
ED50 |
68.6 |
umol.kg-1 |
10.1016/j.ejmech.2020.112600 |
| Mus musculus |
Mus musculus |
ED50 |
84.3 |
mg.kg-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
ED50 |
1290.0 |
umol.kg-1 |
10.1016/j.bmc.2006.07.054 |
| Mus musculus |
Mus musculus |
ED50 |
1903.0 |
umol.kg-1 |
10.1016/j.bmc.2006.07.054 |
| Mus musculus |
Mus musculus |
Hepatic necrosis in survivors |
1.13 |
None |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Hepatic necrosis in survivors |
3.25 |
None |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
ID50 |
120.0 |
umol.kg-1 |
10.1016/j.ejmech.2009.06.029 |
| Mus musculus |
Mus musculus |
ID50 |
120.0 |
umol.kg-1 |
10.1021/np9804177 |
| Mus musculus |
Mus musculus |
ID50 |
125.0 |
umol.kg-1 |
10.1016/j.bmc.2008.08.019 |
| Mus musculus |
Mus musculus |
ID50 |
125.0 |
umol.kg-1 |
10.1021/np9804177 |
| Mus musculus |
Mus musculus |
ID50 |
133.0 |
umol.kg-1 |
10.1016/j.ejmech.2009.06.029 |
| Mus musculus |
Mus musculus |
ID50 |
1145.0 |
umol.kg-1 |
10.1016/j.bmc.2008.08.019 |
| Mus musculus |
Mus musculus |
ID50 |
1145.0 |
umol.kg-1 |
10.1016/j.ejmech.2009.06.029 |
| Mus musculus |
Mus musculus |
Inhibition |
29.38 |
% |
10.1007/s00044-010-9300-y |
| Mus musculus |
Mus musculus |
Inhibition |
36.0 |
% |
10.1016/j.bmcl.2009.07.075 |
| Mus musculus |
Mus musculus |
Inhibition |
38.0 |
% |
10.1016/j.bmc.2008.08.019 |
| Mus musculus |
Mus musculus |
Inhibition |
38.0 |
% |
10.1016/j.ejmech.2009.06.029 |
| Mus musculus |
Mus musculus |
Inhibition |
85.0 |
% |
10.1021/np9804177 |
| Mus musculus |
Mus musculus |
Inhibition |
88.0 |
% |
10.1021/np9804177 |
| Mus musculus |
Mus musculus |
LD50 |
3700.0 |
umol.kg-1 |
10.1016/j.bmc.2006.07.054 |
| Mus musculus |
Mus musculus |
MPE |
32.02 |
% |
10.1007/s00044-010-9300-y |
| Mus musculus |
Mus musculus |
No. of animals |
0.0 |
None |
10.1021/jm00393a034 |
| Mus musculus |
Mus musculus |
No. of animals |
1.0 |
None |
10.1021/jm00393a034 |
| Mus musculus |
Mus musculus |
No. of animals |
11.0 |
None |
10.1021/jm00393a034 |
| Mus musculus |
Mus musculus |
No. of animals with liver necrosis |
1.0 |
None |
10.1021/jm00347a001 |
| Mus musculus |
Mus musculus |
No. of animals with liver necrosis |
7.0 |
None |
10.1021/jm00347a001 |
| Mus musculus |
Mus musculus |
No. of animals with liver necrosis |
8.0 |
None |
10.1021/jm00347a001 |
| Mus musculus |
Mus musculus |
No. of survivors |
2.0 |
None |
10.1021/jm00393a034 |
| Mus musculus |
Mus musculus |
permeability |
0.51 |
umol cm2/hr |
10.1016/j.bmcl.2006.03.061 |
| Mus musculus |
Mus musculus |
Plasma ALT at 24 h |
1552.0 |
mU ml-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Plasma ALT at 24 h |
4030.0 |
mU ml-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.04 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.05 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.09 |
nM equiv mg-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.11 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.15 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.2 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.21 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.24 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.29 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.58 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.71 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.73 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
0.92 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
1.08 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
1.13 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
1.19 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
1.22 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
1.52 |
nM equiv mg-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
1.55 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
2.19 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
2.45 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
2.89 |
nM equiv (mg of tissue)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
12.4 |
nM equiv (ml of urine)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
15.3 |
nM equiv mg-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
19.2 |
nM equiv (ml of blood)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
544.0 |
nM equiv (ml of blood)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
1605.0 |
nM equiv (ml of blood)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
3880.0 |
nM equiv (ml of urine)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Radioactivity |
6005.0 |
nM equiv (ml of urine)-1 |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Survival |
17.0 |
% |
10.1021/jm00393a034 |
| Mus musculus |
Mus musculus |
Survivors at 24 h |
4.0 |
None |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Survivors at 24 h |
8.0 |
None |
10.1021/jm00159a029 |
| Mus musculus |
Mus musculus |
Toxicity |
0.0 |
None |
10.1021/jm00140a014 |
| Mus musculus |
Mus musculus |
Toxicity |
2.0 |
None |
10.1021/jm00140a014 |
| Mus musculus |
Mus musculus |
Toxicity |
3.0 |
None |
10.1021/jm00140a014 |
| Mus musculus |
Mus musculus |
Toxicity |
nan |
None |
10.1021/jm00185a001 |
| Mus musculus |
Nitric oxide synthase, inducible |
IC50 |
nan |
None |
None |
| Mus musculus |
Nitric oxide synthase, inducible |
Ki |
nan |
None |
None |
| Mus musculus |
RAW264.7 |
GI50 |
1002000.0 |
nM |
10.1039/C3MD00251A |
| Mus musculus |
Skin |
permeability |
0.51 |
umol/cm2/hr |
10.1016/j.bmcl.2011.04.118 |
| Mus musculus |
Skin |
permeability |
0.74 |
umol/cm2/hr |
10.1016/j.bmcl.2011.04.118 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
661000.0 |
nM |
10.1039/C3MD00251A |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
661000.0 |
nM |
10.1039/C3MD00251A |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
600000.0 |
nM |
10.1039/C3MD00251A |
| Oryctolagus cuniculus |
Angiotensin-converting enzyme |
IC50 |
nan |
None |
None |
| Oryctolagus cuniculus |
Angiotensin-converting enzyme |
Ki |
nan |
None |
None |
| Oryctolagus cuniculus |
Arachidonate 15-lipoxygenase |
IC50 |
28380.0 |
nM |
None |
| Oryctolagus cuniculus |
Arachidonate 15-lipoxygenase |
Ki |
nan |
None |
None |
| Ovis aries |
Cyclooxygenase-1 |
IC50 |
372000.0 |
nM |
10.1021/ml4000904 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
86700.0 |
nM |
10.1021/jm7009292 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
198400.0 |
nM |
10.1021/jm7009292 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Plasmodium falciparum |
Plasmodium falciparum |
Potency |
10417.9 |
nM |
None |
| Plasmodium falciparum |
Plasmodium falciparum |
Potency |
11689.1 |
nM |
None |
| Plasmodium falciparum |
Plasmodium falciparum |
Ratio IC50 |
0.4 |
None |
10.1021/jm7009292 |
| Pneumocystis carinii |
Pneumocystis carinii |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Rattus norvegicus |
Aldose reductase |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Aldose reductase |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1a adrenergic receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1a adrenergic receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1b adrenergic receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1b adrenergic receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Anandamide amidohydrolase |
IC50 |
300000.0 |
nM |
10.1021/jm901891p |
| Rattus norvegicus |
Anandamide amidohydrolase |
Inhibition |
4.0 |
% |
10.1021/jm901891p |
| Rattus norvegicus |
Anandamide amidohydrolase |
Inhibition |
22.0 |
% |
10.1021/jm800807k |
| Rattus norvegicus |
Androgen Receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Androgen Receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Androgen Receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Aryl sulfotransferase |
Km |
92000.0 |
nM |
10.1021/jm010481c |
| Rattus norvegicus |
Aryl sulfotransferase |
Ratio |
66.7 |
None |
10.1021/jm010481c |
| Rattus norvegicus |
Aryl sulfotransferase |
Vmax |
181.0 |
nM min-1 |
10.1021/jm010481c |
| Rattus norvegicus |
Bile salt export pump |
IC50 |
1000000.0 |
nM |
10.1124/dmd.111.040758 |
| Rattus norvegicus |
Cyclooxygenase-1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Cytochrome P450 1A1 |
Ks |
0.87 |
mM |
10.1021/jm00032a021 |
| Rattus norvegicus |
Cytochrome P450 2B1 |
Ks |
0.8 |
mM |
10.1021/jm00032a021 |
| Rattus norvegicus |
GABA receptor alpha-1 subunit |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Glycine receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Glycine receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
H9c2 |
Activity |
nan |
None |
10.1039/C8MD00611C |
| Rattus norvegicus |
Insulin receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Insulin receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Liver |
Stability |
43.0 |
% |
10.1039/c5md00349k |
| Rattus norvegicus |
Liver |
T1/2 |
1.48 |
hr |
10.1039/c5md00349k |
| Rattus norvegicus |
Liver microsomes |
Stability |
65.0 |
% |
10.1021/ml4000904 |
| Rattus norvegicus |
Nitric-oxide synthase, brain |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Nitric-oxide synthase, brain |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Peripheral myelin protein 22 |
Potency |
12.8 |
nM |
None |
| Rattus norvegicus |
Plasma |
Fu |
0.52 |
None |
10.1021/jm901371v |
| Rattus norvegicus |
Plasma |
logFu |
1.0 |
None |
10.1016/j.ejmech.2009.06.004 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
-6.7 |
degrees C |
10.1016/j.ejmech.2008.09.020 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
4.18 |
% |
10.1007/s00044-004-0123-6 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
5.14 |
% |
10.1007/s00044-004-0123-6 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
5.47 |
% |
10.1007/s00044-004-0123-6 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
6.06 |
% |
10.1007/s00044-004-0123-6 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
37.0 |
degrees C |
10.1016/j.ejmech.2008.09.020 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
37.16 |
degrees C |
10.1016/j.bmc.2009.05.073 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
37.2 |
degrees C |
10.1016/j.bmc.2009.05.073 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
37.27 |
degrees C |
10.1016/j.bmc.2009.05.073 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
37.3 |
degrees C |
10.1016/j.ejmech.2008.09.020 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
37.38 |
degrees C |
10.1016/j.bmc.2009.05.073 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
37.6 |
degrees C |
10.1016/j.ejmech.2008.09.020 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
38.0 |
degrees C |
10.1016/j.ejmech.2008.09.020 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
38.4 |
degrees C |
10.1016/j.ejmech.2008.09.020 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
66.0 |
% |
10.1021/acs.jmedchem.9b00017 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
34000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
35000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
36000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
37000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
38000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
39300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
40000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
41000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
41000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
41500.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
43000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
44000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
44600.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.3 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.4 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.5 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.6 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.7 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.8 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.9 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
2.3 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
2.4 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
2.5 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
326.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
340.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
341.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
356.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
359.83 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
430.5 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
485.6 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
536.6 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
576.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
592.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
594.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
638.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
702.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
758.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
798.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
800.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
800.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
810.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
813.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
821.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
832.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
835.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
842.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
888.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
900.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
902.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
908.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
910.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
923.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
940.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
945.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
983.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
985.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
990.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
994.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
997.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1005.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1050.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1110.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1272.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
25.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
28.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
28.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
28.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
28.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
29.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
29.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
29.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
30.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
30.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
30.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
30.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
32.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
33.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
36.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
37.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
38.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
39.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
39.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
42.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
45.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
51.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
54.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
58.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
61.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
62.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
69.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
72.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
85.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
100.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
14.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
14.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
14.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
17.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
17.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
17.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
18.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
51.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
53.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
54.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
55.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
55.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
56.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
56.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
57.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
57.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
57.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
58.5 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
58.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
59.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
60.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
60.5 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
61.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
61.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
61.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
61.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
62.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
63.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
63.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
66.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
73.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
74.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
76.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
77.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
83.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
84.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
90.83 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
92.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
93.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
108.4 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
123.8 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BASO |
0.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
1.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.14 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.18 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.2 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.24 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.26 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.28 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.3 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.34 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.36 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.38 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.4 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.44 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.46 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.48 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.54 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.56 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.575 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.62 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.64 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.68 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.9 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
1.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
1.4 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.2 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
3.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
108.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
110.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
114.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
120.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
122.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
124.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
128.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
130.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
132.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
133.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
134.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
135.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
136.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
140.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
142.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
142.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
150.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
153.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
160.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
164.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
168.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
170.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
174.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
178.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
180.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
182.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
184.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
186.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
194.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
200.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
210.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
218.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
101.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
103.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
104.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
105.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
106.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
107.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
108.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
109.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
110.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
97.67 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
98.33 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
98.5 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
98.67 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
99.0 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
99.17 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
99.67 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
104.0 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
610.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
664.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
668.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
705.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
716.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
728.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
748.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
752.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
753.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
762.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
770.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
776.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
782.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
790.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
800.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
804.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
810.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
813.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
816.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
818.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
822.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
824.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
830.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
848.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
850.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
854.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
858.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
872.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
874.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
876.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
886.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
894.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
904.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
914.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
918.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
968.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
974.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
1040.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
201.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
222.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
248.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
253.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
256.17 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
273.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
298.8 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
328.8 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
102.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
102.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.7 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.5 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
106.9 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
27170000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
27330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
28330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
29000000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
31200000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
33000000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
33330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
33670000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
1.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
1.5 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
1.6 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
1.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
1.8 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
1.9 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
3.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
4.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
5.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Dose |
58.8 |
% |
10.1021/jm00140a014 |
| Rattus norvegicus |
Rattus norvegicus |
ED50 |
245.1 |
umol.kg-1 |
10.1016/j.ejmech.2020.112600 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
0.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
17.8 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
47.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
65.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.2 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
2.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
2.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
2.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
3.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
4.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
5.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
5.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
5.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
5.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
6.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
6.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
8.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
9.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
10.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
11.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
1808.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
1888.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
1916.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
1954.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
1962.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
1970.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
1982.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2005.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2064.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2072.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2076.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2078.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2118.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2122.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2198.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2206.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2212.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2250.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2310.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2314.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2336.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2362.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2370.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2392.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2400.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2406.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2412.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2422.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2460.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2484.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2496.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
0.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.5 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
2.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
2.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1540.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1560.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1571.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1573.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1586.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1610.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1650.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1713.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1824.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1868.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1878.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1888.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1906.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1912.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1922.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1928.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1930.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1940.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1946.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1948.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1950.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1952.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1966.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1970.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1974.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1982.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1984.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1990.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1992.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1996.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2010.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2014.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2022.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2028.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2035.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2044.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2045.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2050.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2054.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2056.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
31.17 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
32.6 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
32.78 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
34.53 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
34.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
34.87 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
34.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
35.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
35.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
35.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.4 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.4 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
42.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
43.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
43.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
118000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
119000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
120000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
121000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
123000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
124000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
125000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
125700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
126000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
128000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
129000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
129000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
129800.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
130000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
132700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
134000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
135000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
135000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
135700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
136200.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
137000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
138000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
140000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
142000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
144000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
145000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
147000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
148600.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
59.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
66.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
72.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
79.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
80.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
81.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
82.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
84.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
84.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
85.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
86.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
86.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
88.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
91.5 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
96.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
100.5 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
102.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
103.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
104.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
105.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
105.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
106.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
107.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
107.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
109.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
110.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
111.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
111.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
114.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
119.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
124.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
126.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
128.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
132.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
134.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
138.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
142.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
161.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
199.2 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
9.8 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
10.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
10.5 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
10.8 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
13.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
6275.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
7022.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
8402.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
8609.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
8879.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
10212.2 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
10431.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
12444.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
56.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
59.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
60.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
62.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
62.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
63.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
63.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
63.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
65.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
65.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
65.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
66.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
68.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
68.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
69.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
70.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
71.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
72.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
73.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
73.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
74.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
76.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
77.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
80.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
82.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
82.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
85.2 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
85.6 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
88.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
89.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
90.17 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
92.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
93.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
19.5 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.4 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.5 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.3 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.4 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.5 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.6 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.7 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.8 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.1 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.2 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.3 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.4 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.46 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.5 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.6 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.9 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.27 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.43 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.5 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.97 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
25.13 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
26.13 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
368200.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
374400.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
384300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
389000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
389500.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
395700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
396200.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
403300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
57.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.0 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.28 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.8 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.87 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.03 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.13 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.53 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.8 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.87 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.8 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
66.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
66.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
66.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
66.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
67.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
67.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
67.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
40.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
40.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
68.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
90.5 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
128.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
135.4 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
158.2 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
162.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
0.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
0.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
1.2 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
4.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
4.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
4.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
5.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
5.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
5.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
6.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
7.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
7.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
7.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
7.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
8.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
8.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
9.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
10.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
10.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
11.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
11.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
12.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
12.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
13.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
15.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
16.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
17.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
22.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
5.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
6.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
7.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
9.17 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
9.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
9.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
11.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
11.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
12.4 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
13.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
13.4 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
13.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
17.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
17.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
17.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
18.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
18.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
18.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
19.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
20.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
20.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
20.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
21.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
21.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
23.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
24.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
25.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
28.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
548.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
633.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
649.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
715.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1094.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1111.83 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1212.8 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1674.6 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
79.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
83.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
87.2 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
88.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
89.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
90.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
91.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
91.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
92.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
93.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
95.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
96.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
97.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
99.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
101.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
102.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
105.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
108.2 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
110.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
110.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
114.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
116.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
117.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
118.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
119.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
120.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
132.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
135.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1366.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1435.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1444.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1446.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1452.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1492.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1494.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1562.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1564.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1570.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1582.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1592.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1614.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1630.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1632.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1650.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1666.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1680.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1736.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1742.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1750.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1756.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1770.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1790.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1828.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1852.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
2002.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
2088.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
2110.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
989330.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1006400.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1052670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1081000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1082000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1082830.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1084000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1085000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1109000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1118000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1129000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1141000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1148000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1156000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1160000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1163000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1171000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1182000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1183000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1188000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1190000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1191670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1198000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1199000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1203000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1208000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1217000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1230000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1237330.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1244000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1257000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1267000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1269000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1275000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1289000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1297000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1312000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1437600.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.5 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.9 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.1 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.3 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.34 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.5 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.63 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.65 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.7 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.71 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.75 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.78 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.81 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.3 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.73 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
54000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
55000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
56000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
57000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
57000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
58000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
58000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
59000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
59000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
60000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
60400.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
60500.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
61000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
62700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
63000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
64000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
64200.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
66000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
68000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
4800000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5130000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5192000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5200000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5368000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5375000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5406000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5422000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5470000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5510000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5520000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5538000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5554000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5560000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5594000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5656000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5666000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5688000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5720000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5742000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5890000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5906000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5916000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5930000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5940000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5944000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6018000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6020000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6126000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6218000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6402000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6406000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6438000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6552000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6630000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6650000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6680000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7080000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7202000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7438000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
0.0 |
/100WBC |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
3.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
3.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
9.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
9.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
9.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.5 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.9 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.53 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.7 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
143.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
143.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
143.6 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
143.87 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
144.12 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
144.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
144.74 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
145.03 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
145.13 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
T |
6.7 |
degrees C |
10.1016/j.bmc.2014.03.043 |
| Rattus norvegicus |
Rattus norvegicus |
T |
36.4 |
degrees C |
10.1007/s00044-013-0468-9 |
| Rattus norvegicus |
Rattus norvegicus |
T |
36.8 |
degrees C |
10.1007/s00044-013-0468-9 |
| Rattus norvegicus |
Rattus norvegicus |
T |
37.0 |
degrees C |
10.1007/s00044-013-0468-9 |
| Rattus norvegicus |
Rattus norvegicus |
T |
37.0 |
degrees C |
10.1016/j.bmc.2014.03.043 |
| Rattus norvegicus |
Rattus norvegicus |
T |
37.1 |
degrees C |
10.1016/j.ejmech.2014.05.080 |
| Rattus norvegicus |
Rattus norvegicus |
T |
37.14 |
degrees C |
10.1016/j.ejmech.2014.05.080 |
| Rattus norvegicus |
Rattus norvegicus |
T |
37.3 |
degrees C |
10.1016/j.bmc.2014.03.043 |
| Rattus norvegicus |
Rattus norvegicus |
T |
37.6 |
degrees C |
10.1016/j.bmc.2014.03.043 |
| Rattus norvegicus |
Rattus norvegicus |
T |
37.7 |
degrees C |
10.1007/s00044-012-0449-4 |
| Rattus norvegicus |
Rattus norvegicus |
T |
37.88 |
degrees C |
10.1016/j.ejmech.2014.05.080 |
| Rattus norvegicus |
Rattus norvegicus |
T |
37.9 |
degrees C |
10.1007/s00044-012-0449-4 |
| Rattus norvegicus |
Rattus norvegicus |
T |
38.0 |
degrees C |
10.1007/s00044-012-0449-4 |
| Rattus norvegicus |
Rattus norvegicus |
T |
38.0 |
degrees C |
10.1016/j.bmc.2014.03.043 |
| Rattus norvegicus |
Rattus norvegicus |
T |
38.4 |
degrees C |
10.1016/j.bmc.2014.03.043 |
| Rattus norvegicus |
Rattus norvegicus |
T |
39.6 |
degrees C |
10.1007/s00044-012-0449-4 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
195.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
197.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
198.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
198.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
199.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
199.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
200.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
200.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
200.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
201.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
202.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
204.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
205.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
205.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
208.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
215.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
216.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
219.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
228.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
229.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
237.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
245.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
266.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
267.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
286.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
297.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
313.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
314.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
349.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
371.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
373.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
399.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Tissue Severity Score |
nan |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Tissue Severity Score |
nan |
None |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
Toxicity |
nan |
None |
10.1021/jm00185a001 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
324.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
338.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
362.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
392.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
418.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
428.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
434.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
466.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
470.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
548.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
620.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
966.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1036.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1050.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1128.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1136.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1222.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1254.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1264.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1266.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1402.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1418.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1452.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1556.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1600.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1686.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1828.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1836.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
2096.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
2348.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
2756.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
3.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
5.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
6.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
6.8 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
7.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
7.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
8.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
33.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
1740.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
2010.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
2110.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
2260.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
2280.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
2340.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
2430.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
2510.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
2540.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
2830.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
2840.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
2860.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
3020.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
3050.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
3100.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
3220.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
3740.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
3830.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
3890.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
3980.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
4010.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
4240.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
4510.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
4690.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
4890.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
5080.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
6210.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
6660.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
6950.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7110.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7900.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9170.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9530.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9980.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11160.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11630.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
12040.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
13670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
0.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
0.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
7.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
13.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
13.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
15.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
16.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
16.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
17.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Serotonin 1a (5-HT1a) receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1a (5-HT1a) receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1b (5-HT1b) receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1b (5-HT1b) receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Solute carrier family 22 member 6 |
Ki |
2099000.0 |
nM |
None |
| Severe acute respiratory syndrome coronavirus 2 |
Replicase polyprotein 1ab |
Inhibition |
16.03 |
% |
10.6019/CHEMBL4495564 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Hit score |
0.1305 |
None |
10.1101/2020.04.21.054387 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
19952.62 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
20000.0 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
-1.06 |
% |
10.21203/rs.3.rs-23951/v1 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
-0.3 |
% |
10.6019/CHEMBL4495565 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition index |
0.1595 |
None |
10.1101/2020.04.03.023846 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
13.2 |
% |
10.1128/aac.01293-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
44.2 |
% |
10.1128/aac.01293-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
10.8 |
% |
10.1128/aac.01293-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
56.3 |
% |
10.1128/aac.01293-08 |
| Toxoplasma gondii |
Toxoplasma gondii |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Trichomonas vaginalis |
Trichomonas vaginalis |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Trichomonas vaginalis |
Trichomonas vaginalis |
Inhibition |
14.0 |
% |
10.1016/j.bmcl.2010.06.133 |
| Trichomonas vaginalis |
Trichomonas vaginalis |
Inhibition |
17.0 |
% |
10.1016/j.bmcl.2010.06.133 |
| Trypanosoma brucei |
Trypanosoma brucei |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Trypanosoma brucei brucei |
Trypanosoma brucei brucei |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Trypanosoma brucei rhodesiense |
Trypanosoma brucei rhodesiense |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Trypanosoma cruzi |
Trypanosoma cruzi |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| None |
ADMET |
Activity |
nan |
None |
10.1016/j.ejmech.2020.112600 |
| None |
ADMET |
Activity |
nan |
None |
10.1016/j.ejmech.2020.113042 |
| None |
ADMET |
Activity |
nan |
None |
10.1124/dmd.112.050054 |
| None |
ADMET |
CL |
0.198 |
uL/min |
10.1124/dmd.111.039180 |
| None |
ADMET |
CL |
3.0 |
mL.min-1.g-1 |
10.6019/CHEMBL3301361 |
| None |
ADMET |
CL |
5.0 |
mL.min-1.kg-1 |
10.1124/dmd.108.020479 |
| None |
ADMET |
CL |
6.31 |
uL.min-1.(10^6cells)-1 |
10.6019/CHEMBL3301361 |
| None |
ADMET |
CL |
10.8 |
uL.min-1.(10^6cells)-1 |
10.6019/CHEMBL3301361 |
| None |
ADMET |
CL |
12.2 |
mL.min-1.kg-1 |
10.1021/acs.jmedchem.5b01448 |
| None |
ADMET |
CL |
nan |
None |
10.1124/dmd.111.039180 |
| None |
ADMET |
Concentration |
0.69 |
mM |
10.1021/jm00177a019 |
| None |
ADMET |
Concentration |
0.7 |
mM |
10.1021/jm00177a019 |
| None |
ADMET |
Concentration |
0.72 |
mM |
10.1021/jm00177a019 |
| None |
ADMET |
Concentration |
0.74 |
mM |
10.1021/jm00177a019 |
| None |
ADMET |
Concentration |
0.75 |
mM |
10.1021/jm00177a019 |
| None |
ADMET |
delta logD |
0.0 |
None |
10.1021/jm0000564 |
| None |
ADMET |
Drugexcretion |
2.0 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| None |
ADMET |
Drugexcretion |
4.0 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| None |
ADMET |
Drugexcretion |
30.0 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| None |
ADMET |
Drugexcretion |
55.0 |
% |
10.1111/j.1365-2125.1980.tb01812.x |
| None |
ADMET |
Drug metabolism |
nan |
None |
10.1016/j.ejmech.2020.112600 |
| None |
ADMET |
eLog D |
0.38 |
None |
10.1021/jm0200409 |
| None |
ADMET |
F |
79.0 |
% |
10.1021/jm0000564 |
| None |
ADMET |
Fraction ionised |
0.0 |
None |
10.1021/jm0200409 |
| None |
ADMET |
Fu |
0.503 |
None |
10.1021/jm0200409 |
| None |
ADMET |
Fu |
1.0 |
None |
10.1021/jm0200409 |
| None |
ADMET |
Fu |
1.0 |
None |
10.1021/jm030408h |
| None |
ADMET |
IC50 |
500000.0 |
nM |
10.1124/dmd.112.050054 |
| None |
ADMET |
LD50 |
338.0 |
mg.kg-1 |
10.1021/acs.jnatprod.9b00577 |
| None |
ADMET |
LD50 |
500.0 |
mg.kg-1 |
10.1021/jm00350a001 |
| None |
ADMET |
log10(%HIA +10) |
1.978 |
None |
10.1016/j.ejmech.2010.11.005 |
| None |
ADMET |
Log K'w |
-0.02 |
None |
10.1021/jm0000822 |
| None |
ADMET |
LogP app |
-6.04 |
None |
10.1016/j.bmc.2007.03.040 |
| None |
ADMET |
LogP app |
-5.65 |
None |
10.1016/j.bmc.2007.03.040 |
| None |
ADMET |
MRT |
3.3 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
Papp |
0.3 |
10'6cm/s |
10.1016/j.ejmech.2009.03.039 |
| None |
ADMET |
Papp |
2.22 |
10^-6 cm/s |
10.1016/j.bmc.2007.03.040 |
| None |
ADMET |
Papp |
23.1 |
10'-2 cm/s |
10.1016/j.ejmech.2008.03.043 |
| None |
ADMET |
permeability |
1.76 |
10'-4 cm/s |
10.1021/jm901846t |
| None |
ADMET |
PPB |
26.64 |
% |
10.6019/CHEMBL3301361 |
| None |
ADMET |
Survival |
30.0 |
% |
10.1016/j.ejmech.2020.112600 |
| None |
ADMET |
T1/2 |
2.5 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
Tlag |
1.55 |
min |
10.1016/j.ejmech.2008.03.043 |
| None |
ADMET |
Total excretion |
0.0 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
0.6 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
0.7 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
1.5 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
2.9 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
3.3 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
3.5 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
3.8 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
10.4 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
11.9 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
12.1 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
13.3 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
13.8 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
58.4 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Total excretion |
64.0 |
% |
10.1021/jm00140a014 |
| None |
ADMET |
Vdss |
0.95 |
L.kg-1 |
10.1021/jm0200409 |
| None |
ADMET |
Vdss |
0.95 |
L.kg-1 |
10.1021/jm030408h |
| None |
ADMET |
Vdss |
1.0 |
L.kg-1 |
10.1124/dmd.108.020479 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Index Value |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Active |
2.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Marginal |
3.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
DILI positive/negative |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
GGT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Index Value |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1021/tx1000865 |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1021/tx900326k |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1124/dmd.110.035113 |
| None |
Hepatotoxicity |
LDH Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LDH Increase - Index Value |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LDH Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Index Value |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Index Value |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
NON-PROTEIN TARGET |
Fu |
0.52 |
None |
10.1124/dmd.108.020479 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (acute) |
0.0 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (animal toxicity known) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (benign tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (granulomatous hepatitis) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (mechanism) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
5.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
50.0 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (time to onset) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| None |
NON-PROTEIN TARGET |
Potency |
667.8 |
nM |
None |
| None |
NON-PROTEIN TARGET |
Potency |
21117.7 |
nM |
None |
| None |
No relevant target |
CHI |
20.59 |
None |
10.1016/j.ejmech.2019.111770 |
| None |
No relevant target |
Daq |
10.2 |
10'-6cm2/s |
10.1021/jm901846t |
| None |
No relevant target |
LogD |
0.2 |
None |
10.1016/j.bmcl.2016.11.048 |
| None |
No relevant target |
LogD |
0.27 |
None |
10.1021/jm8005228 |
| None |
No relevant target |
LogD |
0.33 |
None |
10.1021/jm8005228 |
| None |
No relevant target |
LogD |
0.51 |
None |
10.1021/jf102525e |
| None |
No relevant target |
LogD |
0.51 |
None |
10.1021/jm0000564 |
| None |
No relevant target |
LogD |
0.51 |
None |
10.1021/jm0100990 |
| None |
No relevant target |
LogD7.4 |
0.25 |
None |
10.6019/CHEMBL3301361 |
| None |
No relevant target |
log K |
-1.72 |
None |
10.1016/j.bmcl.2006.03.061 |
| None |
No relevant target |
LogP |
0.11 |
None |
10.1021/jm0000822 |
| None |
No relevant target |
LogP |
0.29 |
None |
10.1016/j.bmcl.2010.08.145 |
| None |
No relevant target |
LogP |
0.33 |
None |
10.1016/j.bmcl.2010.08.145 |
| None |
No relevant target |
LogP |
0.34 |
None |
10.1021/jm901846t |
| None |
No relevant target |
LogP |
0.46 |
None |
10.1016/j.bmcl.2021.128318 |
| None |
No relevant target |
LogP |
0.51 |
None |
10.1016/j.bmc.2007.03.040 |
| None |
No relevant target |
LogP |
0.51 |
None |
10.1016/j.bmcl.2016.11.048 |
| None |
No relevant target |
LogP |
0.51 |
None |
10.1021/jf102525e |
| None |
No relevant target |
LogP |
0.51 |
None |
10.1021/jm0000822 |
| None |
No relevant target |
LogP |
1.43 |
None |
10.1016/j.ejmech.2009.06.029 |
| None |
No relevant target |
logPapp |
-6.04 |
None |
10.1021/jf102525e |
| None |
No relevant target |
Log S |
-1.02 |
None |
10.1016/s0960-894x(00)00172-4 |
| None |
No relevant target |
-log(solubility) |
2.7 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
-log(solubility) |
2.87 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
-log(solubility) |
2.91 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
-log(solubility) |
2.93 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
-log(solubility) |
3.0 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
-log(solubility) |
5.48 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
pKa |
0.0 |
None |
10.1021/jf102525e |
| None |
No relevant target |
pKa |
9.5 |
None |
10.1111/j.1365-2125.1980.tb01812.x |
| None |
No relevant target |
pKa |
9.63 |
None |
10.1021/jm901846t |
| None |
No relevant target |
pKa |
nan |
None |
10.1021/jm0000564 |
| None |
No relevant target |
pKa |
nan |
None |
10.1021/jm0200409 |
| None |
No relevant target |
pKa |
nan |
None |
10.1021/jm030408h |
| None |
No relevant target |
pKa_A1 |
9.48 |
None |
10.6019/CHEMBL3301361 |
| None |
No relevant target |
Retention_time |
7.45 |
min |
10.1016/j.ejmech.2019.111770 |
| None |
No relevant target |
Rm |
0.31 |
None |
10.1016/j.bmcl.2021.128318 |
| None |
No relevant target |
Solubility |
19950.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
89070.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
140300.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
141200.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
144500.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
169700.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
173900.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
186700.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
188600.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
199800.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
208400.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
212100.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
217400.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
224800.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
235100.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
238100.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
246200.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
254000.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
266300.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
267900.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
279000.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
287000.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
316500.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
324000.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
352700.0 |
ug.mL-1 |
10.1039/C5MD00551E |
| None |
No relevant target |
Solubility |
1910000.0 |
nM |
10.1016/j.bmcl.2006.03.061 |
| None |
No relevant target |
Solubility |
100000000.0 |
nM |
10.1016/j.bmcl.2006.03.061 |
| None |
Phospholipidosis |
Maximum test concentration that did not exhibit cytotoxicity |
100.0 |
uM |
None |
| None |
Phospholipidosis |
Phospholipidosis |
nan |
None |
10.1021/ci6004542 |
| None |
Phospholipidosis |
Phospholipidosis |
nan |
None |
10.1021/mp100103e |
| None |
Phospholipidosis |
Phospholipidosis |
nan |
None |
10.1080/15376510701857262 |
| None |
Phospholipidosis |
Phospholipidosis as % of positive control |
0.3 |
% |
None |
| None |
Unchecked |
Ac50 |
7.079 |
uM |
None |
| None |
Unchecked |
AC50 |
7079.5 |
nM |
None |
| None |
Unchecked |
AC50 |
10710.0 |
nM |
None |
| None |
Unchecked |
AC50 |
14530.0 |
nM |
None |
| None |
Unchecked |
Activity |
8.0 |
% |
10.1016/j.ejmech.2020.113042 |
| None |
Unchecked |
Activity |
9.0 |
% |
10.1016/j.ejmech.2020.113042 |
| None |
Unchecked |
Activity |
10.0 |
% |
10.1016/j.ejmech.2020.113042 |
| None |
Unchecked |
Activity |
12.0 |
% |
10.1016/j.ejmech.2020.113042 |
| None |
Unchecked |
Activity |
15.0 |
% |
10.1016/j.ejmech.2020.113042 |
| None |
Unchecked |
Activity |
18.0 |
% |
10.1016/j.ejmech.2020.113042 |
| None |
Unchecked |
Activity |
19.0 |
% |
10.1016/j.ejmech.2020.113042 |
| None |
Unchecked |
Activity |
25.0 |
% |
10.1016/j.ejmech.2020.113042 |
| None |
Unchecked |
Activity |
nan |
None |
10.1016/j.bmc.2008.04.066 |
| None |
Unchecked |
Activity |
nan |
None |
10.1021/jm800197b |
| None |
Unchecked |
Hepatotoxicity (acute) |
100.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (association with vascular disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (choleostasis) |
5.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (chronic liver disease) |
7.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cirrhosis) |
5.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (comment) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cytolytic) |
98.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (malignant tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (severe hepatitis) |
57.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (steatosis) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (successful reintroduction) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
IC50 |
500000.0 |
nM |
10.1021/jm00385a031 |
| None |
Unchecked |
IC50 |
nan |
None |
None |
| None |
Unchecked |
Kd |
5790.0 |
nM |
10.1016/j.ejmech.2010.07.055 |
| None |
Unchecked |
Kd |
6640.0 |
nM |
10.1016/j.ejmech.2010.07.055 |
| None |
Unchecked |
Ki |
2500.0 |
nM |
10.1016/j.bmc.2017.03.026 |
| None |
Unchecked |
Ki |
14000000.0 |
nM |
10.1016/j.pharmthera.2004.10.013 |
| None |
Unchecked |
Ki |
nan |
None |
None |
| None |
Unchecked |
Potency |
6513.1 |
nM |
None |
| None |
Unchecked |
Ratio Ki |
2.48 |
None |
10.1016/j.bmc.2017.03.026 |
| None |
Unchecked |
Ratio Ki |
4.0 |
None |
10.1016/j.bmc.2017.03.026 |
| None |
Unchecked |
Selectivity Index |
1.52 |
None |
10.1039/C3MD00251A |