Molecule

Staurosporine

AlkaPlorer ID: AK004056

Synonym: None

IUPAC Name: (2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-16-one

Structure

SMILES: CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)N1C3=CC=CC=C3C3=C4CNC(=O)C4=C4C5=CC=CC=C5N2C4=C31

InChI: InChI=1S/C28H26N4O3/c1-28-26(34-3)17(29-2)12-20(35-28)31-18-10-6-4-8-14(18)22-23-16(13-30-27(23)33)21-15-9-5-7-11-19(15)32(28)25(21)24(22)31/h4-11,17,20,26,29H,12-13H2,1-3H3,(H,30,33)/t17-,20-,26-,28+/m1/s1

InChIKey: HKSZLNNOFSGOKW-FYTWVXJKSA-N

Reference

Further Metabolic Studies of Indole and Sugar Derivatives Using the Staurosporine Producer<i>Streptomyces staurosporeus</i>

PubChem CID: 44259

LOTUS: LTS0171945

SuperNatural Ⅲ: SN0128352-02

NPASS: NPC98371

{

NPAtlas: NPA014588

Source

Species	Genus	Family	Order	Class	Phylum	Kingdom	Domain
Coniella fragariae	Coniella	Schizoparmaceae	Diaporthales	Sordariomycetes	Ascomycota	Fungi	Eukaryota
None	Streptomyces	Streptomycetaceae	Kitasatosporales	Actinomycetes	Actinomycetota	None	Bacteria
Lyngbya majuscula	Lyngbya	Oscillatoriaceae	Oscillatoriales	Cyanophyceae	Cyanobacteriota	None	Bacteria
Preussia similis	Preussia	Sporormiaceae	Pleosporales	Dothideomycetes	Ascomycota	Fungi	Eukaryota
Streptomyces sp. HNA39	Streptomyces	Streptomycetaceae	Kitasatosporales	Actinomycetes	Actinomycetota	None	Bacteria
Callicarpa bodinieri	Callicarpa	Lamiaceae	Lamiales	Magnoliopsida	Streptophyta	Viridiplantae	Eukaryota
Streptocaulon juventas	Streptocaulon	Apocynaceae	Gentianales	Magnoliopsida	Streptophyta	Viridiplantae	Eukaryota
None	Tubifera	Reticulariaceae	Liceales	Eumycetozoa	Evosea	None	Eukaryota
Tricholoma terreum	Tricholoma	Tricholomataceae	Agaricales	Agaricomycetes	Basidiomycota	Fungi	Eukaryota
Streptomyces sp. H7667	Streptomyces	Streptomycetaceae	Kitasatosporales	Actinomycetes	Actinomycetota	None	Bacteria
Cupaniopsis macropetala	Cupaniopsis	Sapindaceae	Sapindales	Magnoliopsida	Streptophyta	Viridiplantae	Eukaryota

Properties Information

Molecule Weight: 466.5410000000003

TPSA？: 69.45000000000002

MolLogP？: 4.354000000000003

Number of H-Donors: 2

Number of H-Acceptors: 6

RingCount: 8

Activities Information

Organism	Target Name	Standard Type	Standard Value	Standard Units	doi
Alternaria mali	Alternaria mali	MIC	100.0	ug.mL-1	10.1021/jf0532617
Bacillus anthracis	Bacillus anthracis	MIC	128000.0	nM	10.1016/j.bmc.2009.08.061
Bacillus subtilis	Bacillus subtilis	MIC	10.0	ug.mL-1	10.1021/jf0532617
Bos taurus	cAMP-dependent protein kinase alpha-catalytic subunit	IC50	40.0	nM	10.1016/S0960-894X(01)80995-1
Bos taurus	cGMP-dependent protein kinase 1 alpha	IC50	18.0	nM	10.1016/0960-894X(94)00458-R
Bos taurus	cGMP-dependent protein kinase 1 alpha	IC50	18.0	nM	10.1016/S0960-894X(01)80995-1
Botrytis cinerea	Botrytis cinerea	MIC	50.0	ug.mL-1	10.1021/jf0532617
Brugia malayi	Brugia malayi	Activity	nan	None	10.1016/j.ejmech.2016.08.042
Candida albicans	Candida albicans	MIC	100.0	ug.mL-1	10.1021/jf0532617
Capsicum annuum	Capsicum annuum	Activity	nan	None	10.1021/jf0532617
Cavia porcellus	Cavia porcellus	IC50	25.0	nM	10.1016/0960-894X(96)00343-5
Cavia porcellus	Cavia porcellus	IC50	7500.0	nM	10.1016/0960-894X(96)00343-5
Chlorocebus sabaeus	Vero	IC50	2.4	nM	10.1016/j.bmc.2017.09.037
Chlorocebus sabaeus	Vero	IC50	28.0	nM	10.1016/j.ejmech.2019.01.073
Chlorocebus sabaeus	Vero	TC50	0.0024	uM	10.1016/j.ejmech.2017.07.060
Cladosporium cucumerinum	Cladosporium cucumerinum	MIC	1.0	ug.mL-1	10.1021/jf0532617
Colletotrichum orbiculare	Colletotrichum orbiculare	MIC	1.0	ug.mL-1	10.1021/jf0532617
Cricetulus griseus	CHO-K1	GI50	130.0	nM	10.1021/np200041v
Electrophorus electricus	Acetylcholinesterase	IC50	nan	None	10.1016/j.ejmech.2021.114095
Equus caballus	Cholinesterase	IC50	nan	None	10.1016/j.ejmech.2021.114095
Equus caballus	Cholinesterase	Inhibition	nan	%	10.1016/j.ejmech.2021.114095
Equus caballus	Ferritin light chain	Potency	50118.7	nM	None
Fusarium oxysporum f. sp. lycopersici	Fusarium oxysporum f. sp. lycopersici	MIC	50.0	ug.mL-1	10.1021/jf0532617
Gallus gallus	Myosin light chain kinase, smooth muscle	IC50	10.0	nM	10.1016/S0960-894X(01)80995-1
Gallus gallus	Myosin light chain kinase, smooth muscle	Kd	140.0	nM	10.1038/nbt1358
Homo sapiens	3-phosphoinositide dependent protein kinase-1	IC50	5.2	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	3-phosphoinositide dependent protein kinase-1	IC50	10.0	nM	10.1021/acs.jnatprod.7b01082
Homo sapiens	3-phosphoinositide dependent protein kinase-1	Kd	1.7	nM	10.1038/nbt1358
Homo sapiens	3-phosphoinositide dependent protein kinase-1	Kd	1.7	nM	10.1038/nbt.1990
Homo sapiens	3-phosphoinositide dependent protein kinase-1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	3-phosphoinositide dependent protein kinase-1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	518A2	EC50	30.0	nM	10.1016/j.ejmech.2017.11.046
Homo sapiens	8505C	IC50	200.0	nM	10.1016/j.ejmech.2013.11.025
Homo sapiens	A2780	Activity	0.4	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	A2780	Activity	1.0	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	A2780	Activity	3.0	%	10.1016/j.ejmech.2013.12.031
Homo sapiens	A2780	Activity	3.4	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	A2780	Activity	3.7	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	A2780	Activity	4.3	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	A2780	Activity	5.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	A2780	Activity	5.4	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	A2780	Activity	8.5	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	A2780	Activity	32.8	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	A2780	Activity	33.0	%	10.1016/j.ejmech.2013.12.031
Homo sapiens	A2780	Activity	38.0	%	10.1016/j.ejmech.2013.12.031
Homo sapiens	A2780	Activity	51.0	%	10.1016/j.ejmech.2013.12.031
Homo sapiens	A2780	Activity	52.0	%	10.1016/j.ejmech.2013.12.031
Homo sapiens	A2780	Activity	57.0	%	10.1016/j.ejmech.2013.12.031
Homo sapiens	A2780	Activity	57.8	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	A2780	Activity	68.0	%	10.1016/j.ejmech.2013.12.031
Homo sapiens	A2780	Activity	79.0	%	10.1016/j.ejmech.2013.12.031
Homo sapiens	A2780	Activity	87.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	A2780	Activity	90.5	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	A2780	Activity	nan	None	10.1016/j.ejmech.2013.12.031
Homo sapiens	A2780	EC50	100.0	nM	10.1016/j.ejmech.2019.02.057
Homo sapiens	A2780	EC50	100.0	nM	10.1016/j.ejmech.2020.112920
Homo sapiens	A2780	EC50	120.0	nM	10.1016/j.ejmech.2017.11.046
Homo sapiens	A2780	IC50	100.0	nM	10.1016/j.ejmech.2020.112425
Homo sapiens	A2780	IC50	200.0	nM	10.1016/j.ejmech.2013.11.025
Homo sapiens	A-375	Activity	46.95	%	10.1021/acs.jmedchem.6b00547
Homo sapiens	A-375	EC50	nan	None	10.1016/j.ejmech.2020.112920
Homo sapiens	A-375	IC50	2100.0	nM	10.1021/acs.jnatprod.1c01211
Homo sapiens	A-375	IC50	nan	None	10.1016/j.ejmech.2020.112425
Homo sapiens	A-375	Inhibition	102.0	%	10.1016/j.ejmech.2013.10.049
Homo sapiens	A-431	Activity	72.9	%	10.1016/j.bmc.2006.09.063
Homo sapiens	A-431	Activity	84.9	%	10.1016/j.bmc.2006.09.063
Homo sapiens	A-431	IC50	70.0	nM	10.1016/j.bmc.2012.03.061
Homo sapiens	A549	Activity	9.1	%	10.1021/jm701042w
Homo sapiens	A549	Activity	16.4	%	10.1021/jm701042w
Homo sapiens	A549	Activity	74.6	%	10.1021/jm701042w
Homo sapiens	A549	Activity	nan	None	10.1021/jm701042w
Homo sapiens	A549	EC50	40.0	nM	10.1016/j.ejmech.2017.11.046
Homo sapiens	A549	GI50	2.4	nM	10.1021/np700748h
Homo sapiens	A549	IC50	0.1399	ug.mL-1	10.1016/j.bmc.2008.12.030
Homo sapiens	A549	IC50	20.0	nM	10.1021/jm501942m
Homo sapiens	A549	IC50	20.0	nM	10.1039/C2MD20098H
Homo sapiens	A549	IC50	600.0	nM	10.1016/j.ejmech.2013.11.025
Homo sapiens	A549	IC50	3050.0	nM	10.1016/j.bmc.2014.04.005
Homo sapiens	A549	IC50	7470.0	nM	10.1021/acs.jmedchem.9b01669
Homo sapiens	A549	IC50	9100.0	nM	10.1021/acs.jnatprod.1c01211
Homo sapiens	A549	IC50	9500.0	nM	10.1016/j.bmcl.2021.128258
Homo sapiens	A549	IC50	13220.0	nM	10.1021/acs.jmedchem.9b01669
Homo sapiens	A549	IC50	nan	nM	10.1016/j.bmcl.2004.05.040
Homo sapiens	Activin receptor type-1	IC50	10005.0	nM	10.1021/jm500115w
Homo sapiens	Activin receptor type-1	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Activin receptor type-1	Kd	470.0	nM	10.1038/nbt1358
Homo sapiens	Activin receptor type-1	Kd	470.0	nM	10.1038/nbt.1990
Homo sapiens	Activin receptor type-1B	IC50	9118.0	nM	10.1021/jm500115w
Homo sapiens	Activin receptor type-1B	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Activin receptor type-1B	Kd	680.0	nM	10.1038/nbt1358
Homo sapiens	Activin receptor type-1B	Kd	680.0	nM	10.1038/nbt.1990
Homo sapiens	Activin receptor type-1B	Residual Activity	11.0	%	10.1042/bj20121418
Homo sapiens	Activin receptor type-1B	Residual Activity	70.0	%	10.1042/bj20121418
Homo sapiens	Activin receptor type-2A	Kd	8900.0	nM	10.1038/nbt.1990
Homo sapiens	Activin receptor type-2A	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Activin receptor type-2B	Kd	4600.0	nM	10.1038/nbt1358
Homo sapiens	Activin receptor type-2B	Kd	4600.0	nM	10.1038/nbt.1990
Homo sapiens	Adaptor-associated kinase	Kd	1.2	nM	10.1038/nbt1358
Homo sapiens	Adaptor-associated kinase	Kd	1.2	nM	10.1038/nbt.1990
Homo sapiens	Adaptor-associated kinase	Kd	1.3	nM	10.1038/nbt1068
Homo sapiens	Aldehyde dehydrogenase 1A1	Potency	39810.7	nM	None
Homo sapiens	ALK tyrosine kinase receptor	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	ALK tyrosine kinase receptor	IC50	0.67	nM	10.1021/acs.jmedchem.7b01039
Homo sapiens	ALK tyrosine kinase receptor	IC50	0.74	nM	10.1021/acs.jmedchem.7b01039
Homo sapiens	ALK tyrosine kinase receptor	IC50	1.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	ALK tyrosine kinase receptor	IC50	1.0	nM	10.1016/j.ejmech.2021.113511
Homo sapiens	ALK tyrosine kinase receptor	IC50	1.09	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	ALK tyrosine kinase receptor	IC50	1.6	nM	10.1021/acs.jmedchem.7b01039
Homo sapiens	ALK tyrosine kinase receptor	IC50	1.7	nM	10.1021/acs.jmedchem.7b01039
Homo sapiens	ALK tyrosine kinase receptor	IC50	2.3	nM	None
Homo sapiens	ALK tyrosine kinase receptor	IC50	2.36	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	ALK tyrosine kinase receptor	IC50	2.9	nM	10.1021/acs.jmedchem.7b01039
Homo sapiens	ALK tyrosine kinase receptor	IC50	2.98	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	ALK tyrosine kinase receptor	IC50	3.0	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	ALK tyrosine kinase receptor	IC50	3.8	nM	10.1021/acs.jmedchem.7b01039
Homo sapiens	ALK tyrosine kinase receptor	IC50	6.45	nM	10.1016/j.bmc.2023.117241
Homo sapiens	ALK tyrosine kinase receptor	IC50	6.7	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	ALK tyrosine kinase receptor	IC50	7.1	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	ALK tyrosine kinase receptor	IC50	7.1	nM	10.1021/acs.jnatprod.7b01082
Homo sapiens	ALK tyrosine kinase receptor	IC50	30.0	nM	10.1021/np4005745
Homo sapiens	ALK tyrosine kinase receptor	Inhibition	97.89	%	10.1016/j.ejmech.2013.03.043
Homo sapiens	ALK tyrosine kinase receptor	Inhibition	97.89	%	10.1016/j.ejmech.2013.07.056
Homo sapiens	ALK tyrosine kinase receptor	Kd	32.0	nM	10.1038/nbt1358
Homo sapiens	ALK tyrosine kinase receptor	Kd	32.0	nM	10.1038/nbt.1990
Homo sapiens	ALK tyrosine kinase receptor	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	ALK tyrosine kinase receptor	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	3.7	nM	10.1038/nbt1358
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	3.7	nM	10.1038/nbt.1990
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	9.0	nM	10.1038/nbt1068
Homo sapiens	AMP-activated protein kinase, alpha-2 subunit	Kd	12.0	nM	10.1038/nbt1358
Homo sapiens	AMP-activated protein kinase, alpha-2 subunit	Kd	12.0	nM	10.1038/nbt.1990
Homo sapiens	AMP-activated protein kinase, AMPK	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	AMP-activated protein kinase, AMPK	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	AMP-activated protein kinase (AMPK) alpha-1/beta-1/gamma-1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	AMP-activated protein kinase (AMPK) alpha-1/beta-1/gamma-1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Ankyrin repeat and protein kinase domain-containing protein 1	Kd	270.0	nM	10.1038/nbt1358
Homo sapiens	Ankyrin repeat and protein kinase domain-containing protein 1	Kd	270.0	nM	10.1038/nbt.1990
Homo sapiens	ATP-dependent DNA helicase Q1	Potency	35481.3	nM	None
Homo sapiens	Bcr/Abl fusion protein	IC50	55.7	nM	10.1016/j.ejmech.2020.112710
Homo sapiens	Bcr/Abl fusion protein	IC50	78.7	nM	10.1016/j.ejmech.2020.112710
Homo sapiens	Bcr/Abl fusion protein	IC50	121.8	nM	10.1016/j.bmc.2015.04.083
Homo sapiens	Bcr/Abl fusion protein	IC50	121.8	nM	10.1016/j.bmcl.2016.10.007
Homo sapiens	Beta-adrenergic receptor kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Beta-adrenergic receptor kinase 2	IC50	850.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Beta-adrenergic receptor kinase 2	IC50	862.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Beta-secretase 1	Kd	nan	None	10.1016/j.ejmech.2017.06.020
Homo sapiens	BGC-823	EC50	26.83	ug.mL-1	10.1016/j.bmcl.2011.08.039
Homo sapiens	BGC-823	IC50	6830.0	nM	10.1016/j.bmc.2012.08.059
Homo sapiens	Bile salt export pump	IC50	18700.0	nM	10.1093/toxsci/kfq269
Homo sapiens	Bile salt export pump	IC50	18700.0	nM	10.1093/toxsci/kft176
Homo sapiens	BJ	Activity	nan	None	10.1038/nature05859
Homo sapiens	BJ	EC50	2000.0	nM	10.1016/j.bmcl.2014.09.061
Homo sapiens	BJ	EC50	40000.0	nM	10.1021/acs.jnatprod.8b00884
Homo sapiens	BJ	IC50	2.0	nM	10.1016/j.bmcl.2012.08.005
Homo sapiens	Blood	IC50	100.0	nM	10.1016/j.bmc.2008.06.017
Homo sapiens	Blood	IC50	100.0	nM	10.1016/j.bmc.2008.09.015
Homo sapiens	BMP-2-inducible protein kinase	Kd	1.0	nM	10.1021/acsmedchemlett.3c00127
Homo sapiens	BMP-2-inducible protein kinase	Kd	3.7	nM	10.1038/nbt1068
Homo sapiens	BMP-2-inducible protein kinase	Kd	5.6	nM	10.1038/nbt1358
Homo sapiens	BMP-2-inducible protein kinase	Kd	5.6	nM	10.1038/nbt.1990
Homo sapiens	Bone morphogenetic protein receptor type-1A	IC50	4288.0	nM	10.1021/jm500115w
Homo sapiens	Bone morphogenetic protein receptor type-1A	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Bone morphogenetic protein receptor type-1A	Kd	3700.0	nM	10.1038/nbt1358
Homo sapiens	Bone morphogenetic protein receptor type-1A	Kd	3700.0	nM	10.1038/nbt.1990
Homo sapiens	Bone morphogenetic protein receptor type-1B	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Bone morphogenetic protein receptor type-1B	Kd	170.0	nM	10.1038/nbt.1990
Homo sapiens	Bone morphogenetic protein receptor type-2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Bone morphogenetic protein receptor type-2	IC50	1100.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Bone morphogenetic protein receptor type-2	IC50	2780.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Bone morphogenetic protein receptor type-2	Kd	2300.0	nM	10.1038/nbt.1990
Homo sapiens	Bone morphogenetic protein receptor type-2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Bromodomain-containing protein 4	Delta TM	-1.38	C	None
Homo sapiens	BR serine/threonine-protein kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	BR serine/threonine-protein kinase 1	IC50	0.498	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	BR serine/threonine-protein kinase 1	IC50	0.856	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	BR serine/threonine-protein kinase 1	Kd	26.0	nM	10.1038/nbt1358
Homo sapiens	BR serine/threonine-protein kinase 1	Kd	26.0	nM	10.1038/nbt.1990
Homo sapiens	BR serine/threonine-protein kinase 1	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	BR serine/threonine-protein kinase 1	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	BR serine/threonine-protein kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	BR serine/threonine-protein kinase 2	IC50	2.33	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	BR serine/threonine-protein kinase 2	IC50	3.29	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	BR serine/threonine-protein kinase 2	Kd	3.5	nM	10.1038/nbt1358
Homo sapiens	BR serine/threonine-protein kinase 2	Kd	3.5	nM	10.1038/nbt.1990
Homo sapiens	BR serine/threonine-protein kinase 2	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	BR serine/threonine-protein kinase 2	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	BT-549	IC50	80.0	nM	10.1016/j.bmc.2017.06.036
Homo sapiens	Caco-2	Activity	nan	None	10.1016/j.bmc.2010.04.074
Homo sapiens	Caco-2	NT	nan	None	10.1021/jm0102856
Homo sapiens	Caco-2	Papp	nan	None	10.1016/j.bmc.2008.09.015
Homo sapiens	Calcium/calmodulin-dependent protein kinase type 1B	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Calcium/calmodulin-dependent protein kinase type 1B	IC50	3.78	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Calcium/calmodulin-dependent protein kinase type 1B	IC50	4.99	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase I alpha	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase I alpha	IC50	3.02	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase I alpha	IC50	3.33	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CaM kinase I alpha	Kd	27.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase I alpha	Kd	27.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase I alpha	Kd	30.0	nM	10.1038/nbt1068
Homo sapiens	CaM kinase I alpha	Residual Activity	-6.0	%	10.1042/bj20121418
Homo sapiens	CaM kinase I alpha	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	CaM kinase I delta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase I delta	IC50	0.206	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CaM kinase I delta	IC50	0.298	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase I delta	Kd	1.1	nM	10.1038/nbt1358
Homo sapiens	CaM kinase I delta	Kd	1.1	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase I delta	Kd	2.0	nM	10.1038/nbt1068
Homo sapiens	CaM kinase I delta	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	CaM kinase I delta	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	CaM kinase I gamma	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase I gamma	IC50	3.96	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CaM kinase I gamma	IC50	5.34	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase I gamma	Kd	23.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase I gamma	Kd	23.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase I gamma	Kd	53.0	nM	10.1038/nbt1068
Homo sapiens	CaM kinase II	IC50	2.0	nM	10.1016/s0960-894x(03)00791-1
Homo sapiens	CaM kinase II	IC50	4.0	nM	10.1016/s0960-894x(03)00286-5
Homo sapiens	CaM kinase II	IC50	6.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	CaM kinase II alpha	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase II alpha	IC50	0.0307	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CaM kinase II alpha	IC50	0.0635	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase II alpha	IC50	1.0	nM	10.1016/j.bmcl.2006.05.092
Homo sapiens	CaM kinase II alpha	Kd	0.1	nM	10.1038/nbt1068
Homo sapiens	CaM kinase II alpha	Kd	0.16	nM	10.1038/nbt1358
Homo sapiens	CaM kinase II alpha	Kd	0.16	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase II beta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase II beta	IC50	0.0642	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CaM kinase II beta	IC50	0.07	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	CaM kinase II beta	IC50	0.0945	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase II beta	IC50	0.1	nM	10.1021/jm800861c
Homo sapiens	CaM kinase II beta	Kd	1.3	nM	10.1038/nbt1358
Homo sapiens	CaM kinase II beta	Kd	1.3	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase II beta	Kd	3.0	nM	10.1038/nbt1068
Homo sapiens	CaM kinase II beta	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	CaM kinase II beta	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	CaM kinase II delta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase II delta	IC50	0.0311	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase II delta	IC50	0.0645	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CaM kinase II delta	Kd	0.32	nM	10.1038/nbt1358
Homo sapiens	CaM kinase II delta	Kd	0.32	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase II delta	Kd	0.5	nM	10.1038/nbt1068
Homo sapiens	CaM kinase II delta	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	CaM kinase II delta	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	CaM kinase II gamma	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase II gamma	IC50	0.387	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase II gamma	IC50	0.656	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CaM kinase II gamma	Kd	0.5	nM	10.1038/nbt1068
Homo sapiens	CaM kinase II gamma	Kd	0.55	nM	10.1038/nbt1358
Homo sapiens	CaM kinase II gamma	Kd	0.55	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase II gamma	Residual Activity	-8.0	%	10.1042/bj20121418
Homo sapiens	CaM kinase II gamma	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	CaM kinase IV	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase IV	IC50	138.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CaM kinase IV	IC50	157.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM kinase IV	Inhibition	88.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	CaM kinase IV	Kd	41.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase IV	Kd	41.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase IV	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	CaM kinase IV	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	CaM-kinase kinase alpha	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM-kinase kinase alpha	IC50	29.8	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CaM-kinase kinase alpha	IC50	42.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM-kinase kinase alpha	Kd	0.039	nM	10.1038/nbt1358
Homo sapiens	CaM-kinase kinase alpha	Kd	0.039	nM	10.1038/nbt.1990
Homo sapiens	CaM-kinase kinase alpha	Kd	0.05	nM	10.1038/nbt1068
Homo sapiens	CaM-kinase kinase beta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM-kinase kinase beta	IC50	15.7	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CaM-kinase kinase beta	IC50	33.6	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CaM-kinase kinase beta	Kd	0.05	nM	10.1038/nbt1068
Homo sapiens	CaM-kinase kinase beta	Kd	0.16	nM	10.1038/nbt1358
Homo sapiens	CaM-kinase kinase beta	Kd	0.16	nM	10.1038/nbt.1990
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	IC50	0.935	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	IC50	1.5	nM	10.1016/j.bmcl.2013.11.020
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	IC50	1.58	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	IC50	2.3	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Kd	19.0	nM	10.1038/nbt1358
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Kd	19.0	nM	10.1038/nbt.1990
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	IC50	0.603	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	IC50	1.2	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	IC50	33.0	nM	10.1016/j.bmc.2011.02.036
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	Kd	29.0	nM	10.1038/nbt1358
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	Kd	29.0	nM	10.1038/nbt.1990
Homo sapiens	cAMP-dependent protein kinase, gamma catalytic subunit	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	cAMP-dependent protein kinase, gamma catalytic subunit	IC50	1.29	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	cAMP-dependent protein kinase, gamma catalytic subunit	IC50	6.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	0.7	nM	10.1016/j.ejmech.2018.06.016
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	0.9	nM	10.1016/j.bmcl.2006.05.092
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	1.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	3.6	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	3.6	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	4.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	6.5	nM	10.1016/0960-894X(95)00497-H
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	8.2	nM	10.1016/S0960-894X(00)80167-5
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	15.0	nM	10.1016/0960-894X(94)80004-9
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	15.0	nM	10.1016/j.ejmech.2021.113318
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	16.0	nM	10.1016/s0960-894x(03)00791-1
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	19.0	nM	10.1021/jm00053a003
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	80.0	nM	10.1021/jm020143r
Homo sapiens	cAMP-dependent protein kinase (PKA)	IC50	nan	nM	10.1016/s0960-894x(03)00461-x
Homo sapiens	Canalicular multispecific organic anion transporter 1	IC50	133000.0	nM	10.1093/toxsci/kft176
Homo sapiens	Canalicular multispecific organic anion transporter 2	IC50	133000.0	nM	10.1093/toxsci/kft176
Homo sapiens	CAPAN-1	IC50	12.3	nM	10.1016/j.ejmech.2020.113003
Homo sapiens	CAPAN-1	IC50	30.0	nM	10.1021/acsmedchemlett.0c00269
Homo sapiens	CAPAN-1	IC50	48.0	nM	10.1016/j.bmcl.2019.04.023
Homo sapiens	CAPAN-1	IC50	54.6	nM	10.1016/j.ejmech.2021.113727
Homo sapiens	CAPAN-1	IC50	660.0	nM	10.1016/j.bmc.2019.02.005
Homo sapiens	Casein kinase I	IC50	1400.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Casein kinase I alpha	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase I alpha	IC50	3850.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase I alpha	IC50	4188.0	nM	10.1016/j.ejmech.2010.04.026
Homo sapiens	Casein kinase I alpha	IC50	4210.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Casein kinase I alpha	Inhibition	51.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Casein kinase I alpha	Kd	970.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I delta	Delta TM	2.15	C	None
Homo sapiens	Casein kinase I delta	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase I delta	Kd	2400.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I delta	Kd	2400.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I delta	Residual Activity	46.0	%	10.1042/bj20121418
Homo sapiens	Casein kinase I delta	Residual Activity	77.0	%	10.1042/bj20121418
Homo sapiens	Casein kinase I epsilon	deltaTm	2.3	K	10.1021/acs.jmedchem.1c00845
Homo sapiens	Casein kinase I epsilon	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase I epsilon	Kd	73.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I epsilon	Kd	73.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I epsilon	Kd	690.0	nM	10.1038/nbt1068
Homo sapiens	Casein kinase I gamma 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase I gamma 1	IC50	7170.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Casein kinase I gamma 1	IC50	7440.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase I gamma 1	Inhibition	38.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Casein kinase I gamma 1	Kd	3500.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I gamma 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I gamma 1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Casein kinase I gamma 1	Residual Activity	56.0	%	10.1042/bj20121418
Homo sapiens	Casein kinase I gamma 1	Residual Activity	90.0	%	10.1042/bj20121418
Homo sapiens	Casein kinase I gamma 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase I gamma 2	IC50	1370.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Casein kinase I gamma 2	IC50	3070.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase I gamma 2	Kd	780.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I gamma 2	Kd	780.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I gamma 2	Kd	1400.0	nM	10.1038/nbt1068
Homo sapiens	Casein kinase I gamma 2	Residual Activity	35.0	%	10.1042/bj20121418
Homo sapiens	Casein kinase I gamma 2	Residual Activity	73.0	%	10.1042/bj20121418
Homo sapiens	Casein kinase II	IC50	3400.0	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	Casein kinase II	IC50	3400.0	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Casein kinase II	IC50	100000.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Casein kinase II	Residual Activity	81.0	%	10.1042/bj20121418
Homo sapiens	Casein kinase II	Residual Activity	85.0	%	10.1042/bj20121418
Homo sapiens	Casein kinase II alpha	IC50	3617.0	nM	10.1016/j.ejmech.2010.04.026
Homo sapiens	Casein kinase II alpha	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase II alpha	Inhibition	64.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Casein kinase II alpha	Kd	36.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase II alpha	Kd	940.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase II alpha (prime)	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase II alpha (prime)	IC50	442.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Casein kinase II alpha (prime)	IC50	844.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase II alpha (prime)	Kd	6.5	nM	10.1038/nbt1358
Homo sapiens	Casein kinase II alpha (prime)	Kd	230.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase II alpha (prime)	Residual Activity	83.0	%	10.1042/bj20121418
Homo sapiens	Casein kinase II alpha (prime)	Residual Activity	85.0	%	10.1042/bj20121418
Homo sapiens	Casein kinase I isoform alpha-like	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase I isoform alpha-like	IC50	1270.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Casein kinase I isoform alpha-like	IC50	2410.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase I isoform alpha-like	Kd	250.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I isoform alpha-like	Kd	250.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I isoform gamma-3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase I isoform gamma-3	IC50	1980.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Casein kinase I isoform gamma-3	IC50	3370.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Casein kinase I isoform gamma-3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I isoform gamma-3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I isoform gamma-3	Residual Activity	58.0	%	10.1042/bj20121418
Homo sapiens	Casein kinase I isoform gamma-3	Residual Activity	91.0	%	10.1042/bj20121418
Homo sapiens	Ca-Ski	IC50	11.44	nM	10.1016/j.ejmech.2021.113880
Homo sapiens	Caspase-3	Activity	nan	None	10.1016/j.ejmech.2012.05.032
Homo sapiens	Caspase-3/Caspase-7	Activity	100.0	%	10.1021/acs.jmedchem.5b00413
Homo sapiens	Caspase-3/Caspase-7	Activity	nan	None	10.1021/acsmedchemlett.2c00403
Homo sapiens	CCRF-CEM	IC50	23.0	nM	10.1016/j.bmcl.2012.08.005
Homo sapiens	CDC7/DBF4 (Cell division cycle 7-related protein kinase/Activator of S phase kinase)	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDC7/DBF4 (Cell division cycle 7-related protein kinase/Activator of S phase kinase)	IC50	46.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDC7/DBF4 (Cell division cycle 7-related protein kinase/Activator of S phase kinase)	IC50	63.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK12/Cyclin K	IC50	53.0	nM	10.1021/acs.jmedchem.8b00683
Homo sapiens	CDK17/Cyclin-Y	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK17/Cyclin-Y	IC50	10.7	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK17/Cyclin-Y	IC50	16.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK18/Cyclin Y	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK18/Cyclin Y	IC50	51.1	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK18/Cyclin Y	IC50	66.3	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK1/Cyclin A	IC50	1.7	nM	10.1021/jm301234k
Homo sapiens	CDK1/Cyclin A	IC50	1.93	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK1/Cyclin E	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK1/Cyclin E	IC50	2.17	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	CDK1/Cyclin E	IC50	4.53	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK1/Cyclin E	IC50	6.81	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK2/Cyclin A1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK2/Cyclin A1	IC50	0.5	nM	10.1021/jm301234k
Homo sapiens	CDK2/Cyclin A1	IC50	1.4	nM	10.1016/j.ejmech.2021.113232
Homo sapiens	CDK2/Cyclin A1	IC50	1.51	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK2/Cyclin A1	IC50	1.77	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK2/Cyclin A2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK2/Cyclin A2	IC50	0.4	nM	10.1021/jm301234k
Homo sapiens	CDK2/Cyclin A2	IC50	0.6	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK2/Cyclin A2	IC50	0.72	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	CDK2/Cyclin A2	IC50	0.727	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK2/Cyclin A2	IC50	1.0	nM	10.1021/acs.jmedchem.9b00113
Homo sapiens	CDK2/Cyclin A2	IC50	1.7	nM	10.1016/j.ejmech.2014.06.033
Homo sapiens	CDK2/Cyclin A2	IC50	3.2	nM	10.1016/j.bmc.2014.12.026
Homo sapiens	CDK2/Cyclin A2	IC50	5.8	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	CDK2/Cyclin A2	IC50	20.0	nM	10.1021/jm301234k
Homo sapiens	CDK2/Cyclin A2	IC50	62.0	nM	10.1016/j.ejmech.2020.112277
Homo sapiens	CDK2/Cyclin A2	IC50	50000.0	nM	10.1016/j.ejmech.2021.113232
Homo sapiens	CDK2/Cyclin O	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK2/Cyclin O	IC50	1.46	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	CDK2/Cyclin O	IC50	1.48	nM	10.1016/j.ejmech.2021.113232
Homo sapiens	CDK2/Cyclin O	IC50	1.54	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK2/Cyclin O	IC50	1.72	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK3/cyclin E	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	CDK3/cyclin E	Residual Activity	4.0	%	10.1042/bj20121418
Homo sapiens	CDK3/Cyclin E	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK3/Cyclin E	IC50	1.69	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK3/Cyclin E	IC50	2.08	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	CDK3/Cyclin E	IC50	2.89	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK3/Cyclin E	IC50	4.0	nM	10.1021/jm301234k
Homo sapiens	CDK3/Cyclin E	IC50	53.5	nM	10.1016/j.ejmech.2020.112277
Homo sapiens	CDK4/Cyclin D3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK4/Cyclin D3	IC50	27.0	nM	10.1021/acs.jmedchem.9b00113
Homo sapiens	CDK4/Cyclin D3	IC50	28.1	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK4/Cyclin D3	IC50	37.1	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK4/Cyclin D3	IC50	43.0	nM	10.1016/j.ejmech.2021.113327
Homo sapiens	CDK6/cyclin D1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK6/cyclin D1	IC50	2.9	nM	10.1021/jm301234k
Homo sapiens	CDK6/cyclin D1	IC50	9.18	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK6/cyclin D1	IC50	11.6	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK6/cyclin D1	IC50	31.0	nM	10.1016/j.bmcl.2022.128991
Homo sapiens	CDK6/cyclin D1	Inhibition	-90.0	%	10.1016/j.ejmech.2014.06.027
Homo sapiens	CDK6/cyclin D3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK6/cyclin D3	IC50	15.4	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK6/cyclin D3	IC50	50.0	nM	10.1016/j.bmcl.2023.129284
Homo sapiens	CDK6/cyclin D3	IC50	90.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK6/cyclin D3	IC50	116.0	nM	10.1021/jm801317h
Homo sapiens	CDK6/cyclin D3	IC50	133.0	nM	10.1021/acs.jmedchem.9b00113
Homo sapiens	CDK6/cyclin D3	Residual Activity	9.0	%	10.1042/bj20121418
Homo sapiens	CDK6/cyclin D3	Residual Activity	39.0	%	10.1042/bj20121418
Homo sapiens	CDK7/Cyclin H/MNAT1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK7/Cyclin H/MNAT1	IC50	72.0	nM	10.1021/acs.jmedchem.9b00113
Homo sapiens	CDK7/Cyclin H/MNAT1	IC50	76.6	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK7/Cyclin H/MNAT1	IC50	107.0	nM	10.1016/j.bmcl.2022.128991
Homo sapiens	CDK7/Cyclin H/MNAT1	IC50	120.0	nM	10.1021/acs.jmedchem.8b00683
Homo sapiens	CDK7/Cyclin H/MNAT1	IC50	183.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK8/Cyclin C	IC50	6.0	nM	10.1016/j.ejmech.2017.02.020
Homo sapiens	CDK8/Cyclin C	IC50	15.0	nM	10.1021/acs.jmedchem.8b00683
Homo sapiens	CDK8/Cyclin C	Inhibition	99.0	%	10.1016/j.ejmech.2017.02.020
Homo sapiens	CDK8/Cyclin C	Inhibition	100.0	%	10.1016/j.bmcl.2018.12.065
Homo sapiens	CDK8/Cyclin C	Inhibition	100.0	%	10.1016/j.ejmech.2017.02.020
Homo sapiens	CDK9/Cyclin K	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK9/Cyclin K	IC50	13.0	nM	10.1021/jm301234k
Homo sapiens	CDK9/Cyclin K	IC50	137.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK9/Cyclin K	IC50	214.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK9/cyclin T1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK9/cyclin T1	Delta Tm	3.6	degrees C	10.1021/jm301495v
Homo sapiens	CDK9/cyclin T1	IC50	3.3	nM	10.1021/jm801317h
Homo sapiens	CDK9/cyclin T1	IC50	4.78	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	CDK9/cyclin T1	IC50	13.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK9/cyclin T1	IC50	14.0	nM	10.1021/acs.jmedchem.8b00683
Homo sapiens	CDK9/cyclin T1	IC50	17.0	nM	10.1021/acs.jmedchem.9b00113
Homo sapiens	CDK9/cyclin T1	IC50	23.0	nM	10.1016/j.bmcl.2022.128991
Homo sapiens	CDK9/cyclin T1	Ki	7.0	nM	10.1021/jm301495v
Homo sapiens	CDK9/cyclin T1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	CDK9/cyclin T1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	CDK9/Cyclin-T2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	CDK9/Cyclin-T2	IC50	3.77	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cell division cycle 2-like protein kinase 6	Kd	190.0	nM	10.1038/nbt1358
Homo sapiens	Cell division cycle 2-like protein kinase 6	Kd	190.0	nM	10.1038/nbt.1990
Homo sapiens	Cell division protein kinase 8	Kd	510.0	nM	10.1038/nbt1358
Homo sapiens	Cell division protein kinase 8	Kd	510.0	nM	10.1038/nbt.1990
Homo sapiens	cGMP-dependent protein kinase 1 beta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	cGMP-dependent protein kinase 1 beta	IC50	1.12	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	cGMP-dependent protein kinase 1 beta	IC50	1.23	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	cGMP-dependent protein kinase 1 beta	IC50	2.84	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	cGMP-dependent protein kinase 1 beta	IC50	3.34	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	cGMP-dependent protein kinase 1 beta	IC50	5.0	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	cGMP-dependent protein kinase 1 beta	Kd	32.0	nM	10.1038/nbt1358
Homo sapiens	cGMP-dependent protein kinase 1 beta	Kd	32.0	nM	10.1038/nbt.1990
Homo sapiens	cGMP-dependent protein kinase 1 beta	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	cGMP-dependent protein kinase 1 beta	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	cGMP-dependent protein kinase 1 beta	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	cGMP-dependent protein kinase 1 beta	Residual Activity	6.0	%	10.1042/bj20121418
Homo sapiens	cGMP-dependent protein kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	cGMP-dependent protein kinase 2	IC50	5.77	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	cGMP-dependent protein kinase 2	IC50	26.5	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	cGMP-dependent protein kinase 2	Kd	16.0	nM	10.1038/nbt1358
Homo sapiens	cGMP-dependent protein kinase 2	Kd	16.0	nM	10.1038/nbt.1990
Homo sapiens	Chaperone activity of bc1 complex-like, mitochondrial	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Chaperone activity of bc1 complex-like, mitochondrial	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Citron Rho-interacting kinase	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Citron Rho-interacting kinase	IC50	458.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Citron Rho-interacting kinase	IC50	1040.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Citron Rho-interacting kinase	Kd	340.0	nM	10.1038/nbt1358
Homo sapiens	Citron Rho-interacting kinase	Kd	340.0	nM	10.1038/nbt.1990
Homo sapiens	c-Jun N-terminal kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	c-Jun N-terminal kinase 1	IC50	198.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	c-Jun N-terminal kinase 1	IC50	361.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	c-Jun N-terminal kinase 1	IC50	570.0	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	c-Jun N-terminal kinase 1	IC50	581.0	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	c-Jun N-terminal kinase 1	IC50	1746.0	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	c-Jun N-terminal kinase 1	IC50	3184.0	nM	10.1016/j.ejmech.2010.04.026
Homo sapiens	c-Jun N-terminal kinase 1	Inhibition	95.99	%	10.1016/j.bmc.2012.04.006
Homo sapiens	c-Jun N-terminal kinase 1	Kd	220.0	nM	10.1038/nbt1358
Homo sapiens	c-Jun N-terminal kinase 1	Kd	220.0	nM	10.1038/nbt.1990
Homo sapiens	c-Jun N-terminal kinase 1	Kd	520.0	nM	10.1038/nbt1068
Homo sapiens	c-Jun N-terminal kinase 1	Residual Activity	9.0	%	10.1042/bj20121418
Homo sapiens	c-Jun N-terminal kinase 1	Residual Activity	64.0	%	10.1042/bj20121418
Homo sapiens	c-Jun N-terminal kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	c-Jun N-terminal kinase 2	IC50	742.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	c-Jun N-terminal kinase 2	IC50	1850.0	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	c-Jun N-terminal kinase 2	IC50	2270.0	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	c-Jun N-terminal kinase 2	IC50	3360.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	c-Jun N-terminal kinase 2	Kd	910.0	nM	10.1038/nbt.1990
Homo sapiens	c-Jun N-terminal kinase 2	Kd	1100.0	nM	10.1038/nbt1068
Homo sapiens	c-Jun N-terminal kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	c-Jun N-terminal kinase 2	Residual Activity	35.0	%	10.1042/bj20121418
Homo sapiens	c-Jun N-terminal kinase 2	Residual Activity	67.0	%	10.1042/bj20121418
Homo sapiens	c-Jun N-terminal kinase 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	c-Jun N-terminal kinase 3	IC50	73.1	nM	10.1016/j.ejmech.2021.113674
Homo sapiens	c-Jun N-terminal kinase 3	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	c-Jun N-terminal kinase 3	Kd	110.0	nM	10.1038/nbt1358
Homo sapiens	c-Jun N-terminal kinase 3	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	c-Jun N-terminal kinase 3	Kd	340.0	nM	10.1038/nbt1068
Homo sapiens	c-Jun N-terminal kinase 3	Residual Activity	-5.0	%	10.1042/bj20121418
Homo sapiens	c-Jun N-terminal kinase 3	Residual Activity	12.0	%	10.1042/bj20121418
Homo sapiens	Coiled-coil domain-containing protein 6/Tyrosine-protein kinase receptor RET	IC50	2.22	nM	10.1016/j.ejmech.2020.112755
Homo sapiens	COLO 205	IC50	100.0	nM	10.1016/j.bmcl.2019.126807
Homo sapiens	CWR22R	EC50	251.19	nM	10.1021/acs.jmedchem.1c01532
Homo sapiens	Cyclin-dependent kinase 1	IC50	0.4	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Cyclin-dependent kinase 1	IC50	4.9	nM	10.1016/j.ejmech.2015.08.027
Homo sapiens	Cyclin-dependent kinase 1	IC50	8.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Cyclin-dependent kinase 1	IC50	18.0	nM	10.1021/jm900314j
Homo sapiens	Cyclin-dependent kinase 13	Kd	70.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 13/Cyclin-K	IC50	57.0	nM	10.1021/acs.jmedchem.8b00683
Homo sapiens	Cyclin-dependent kinase 14/Cyclin-Y	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cyclin-dependent kinase 14/Cyclin-Y	IC50	101.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cyclin-dependent kinase 14/Cyclin-Y	IC50	128.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Cyclin-dependent kinase 1/cyclin B	IC50	2.4	nM	10.1021/acs.jmedchem.9b00113
Homo sapiens	Cyclin-dependent kinase 1/cyclin B	IC50	2.52	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Cyclin-dependent kinase 1/cyclin B	IC50	3.2	nM	10.1208/aapsj080125
Homo sapiens	Cyclin-dependent kinase 1/cyclin B	IC50	6.0	nM	10.1016/j.tips.2004.07.006
Homo sapiens	Cyclin-dependent kinase 1/cyclin B	IC50	12.0	nM	10.1016/s0960-894x(03)00791-1
Homo sapiens	Cyclin-dependent kinase 1/cyclin B	IC50	30.0	nM	10.1021/jm020455u
Homo sapiens	Cyclin-dependent kinase 1/cyclin B1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cyclin-dependent kinase 1/cyclin B1	IC50	1.3	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Cyclin-dependent kinase 1/cyclin B1	IC50	1.38	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Cyclin-dependent kinase 1/cyclin B1	IC50	1.42	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cyclin-dependent kinase 1/cyclin B1	IC50	1.6	nM	10.1021/jm800861c
Homo sapiens	Cyclin-dependent kinase 1/cyclin B1	IC50	1.63	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Cyclin-dependent kinase 1/cyclin B1	IC50	2.16	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	Cyclin-dependent kinase 1/cyclin B1	IC50	3.3	nM	10.1021/jm801317h
Homo sapiens	Cyclin-dependent kinase 1/cyclin B1	IC50	25.0	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Cyclin-dependent kinase 1/cyclin B1	IC50	32.0	nM	10.1016/j.ejmech.2018.03.013
Homo sapiens	Cyclin-dependent kinase 1/cyclin B1	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Cyclin-dependent kinase 1/cyclin B1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Cyclin-dependent kinase 2	Delta TM	15.42	C	None
Homo sapiens	Cyclin-dependent kinase 2	IC50	0.1	nM	10.1007/s00044-009-9233-5
Homo sapiens	Cyclin-dependent kinase 2	IC50	0.36	nM	10.1021/jm800861c
Homo sapiens	Cyclin-dependent kinase 2	IC50	1.4	nM	10.1021/jm801317h
Homo sapiens	Cyclin-dependent kinase 2	IC50	2.6	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Cyclin-dependent kinase 2	IC50	3.8	nM	10.1021/jm801317h
Homo sapiens	Cyclin-dependent kinase 2	IC50	11.76	ug.mL-1	10.1016/j.bmc.2012.10.014
Homo sapiens	Cyclin-dependent kinase 2	Inhibition	-100.0	%	10.1016/j.ejmech.2015.07.030
Homo sapiens	Cyclin-dependent kinase 2	Inhibition	58.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Cyclin-dependent kinase 2	Kd	1.3	nM	10.1021/acsmedchemlett.3c00127
Homo sapiens	Cyclin-dependent kinase 2	Kd	7.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 2	Kd	7.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 2	Kd	8.1	nM	10.1038/nbt1068
Homo sapiens	Cyclin-dependent kinase 2/cyclin A	Delta Tm	6.22	degrees C	10.1021/jm301495v
Homo sapiens	Cyclin-dependent kinase 2/cyclin A	Ki	4.0	nM	10.1021/jm301495v
Homo sapiens	Cyclin-dependent kinase 2/cyclin A	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Cyclin-dependent kinase 2/cyclin E	IC50	1.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Cyclin-dependent kinase 2/cyclin E	IC50	12.0	nM	10.1016/s0960-894x(03)00791-1
Homo sapiens	Cyclin-dependent kinase 2/cyclin E	IC50	20.0	nM	10.1021/jm020455u
Homo sapiens	Cyclin-dependent kinase 2/cyclin E	IC50	nan	nM	10.1016/s0960-894x(03)00461-x
Homo sapiens	Cyclin-dependent kinase 2/cyclin E	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Cyclin-dependent kinase 2/cyclin E	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Cyclin-dependent kinase 2/cyclin E1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cyclin-dependent kinase 2/cyclin E1	IC50	1.43	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Cyclin-dependent kinase 2/cyclin E1	IC50	1.64	nM	10.1016/j.ejmech.2021.113232
Homo sapiens	Cyclin-dependent kinase 2/cyclin E1	IC50	1.67	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cyclin-dependent kinase 2/cyclin E1	IC50	1.88	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Cyclin-dependent kinase 2/cyclin E1	IC50	7.0	nM	10.1016/j.bmcl.2022.128991
Homo sapiens	Cyclin-dependent kinase 3	IC50	6.9	nM	10.1021/jm801317h
Homo sapiens	Cyclin-dependent kinase 3	Kd	30.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 3	Kd	30.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 4	Kd	20.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 4	Kd	50.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 4/cyclin D1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cyclin-dependent kinase 4/cyclin D1	IC50	6.6	nM	10.1021/jm301234k
Homo sapiens	Cyclin-dependent kinase 4/cyclin D1	IC50	18.3	nM	10.1021/jm801317h
Homo sapiens	Cyclin-dependent kinase 4/cyclin D1	IC50	20.3	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Cyclin-dependent kinase 4/cyclin D1	IC50	21.1	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cyclin-dependent kinase 4/cyclin D1	IC50	23.3	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Cyclin-dependent kinase 4/cyclin D1	IC50	30.0	nM	10.1016/j.bmcl.2023.129284
Homo sapiens	Cyclin-dependent kinase 4/cyclin D1	IC50	59.0	nM	10.1016/s0960-894x(03)00461-x
Homo sapiens	Cyclin-dependent kinase 4/cyclin D1	IC50	59.0	nM	10.1016/s0960-894x(03)00791-1
Homo sapiens	Cyclin-dependent kinase 4/cyclin D1	IC50	140.0	nM	10.1016/j.bmcl.2022.128991
Homo sapiens	Cyclin-dependent kinase 4/cyclin D1	IC50	nan	nM	10.1016/s0960-894x(03)00461-x
Homo sapiens	Cyclin-dependent kinase 4/cyclin D1	Inhibition	-93.0	%	10.1016/j.ejmech.2014.06.027
Homo sapiens	Cyclin-dependent kinase 5	Kd	84.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 5	Kd	84.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 5	Kd	89.0	nM	10.1038/nbt1068
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	Activity	98.4	%	10.1016/j.ejmech.2010.04.026
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	IC50	1.2	nM	10.1021/jm301234k
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	IC50	1.28	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	IC50	1.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	IC50	2.05	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	IC50	2.67	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	IC50	3.8	nM	10.1021/jm801317h
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	IC50	4.0	nM	10.1021/jm801317h
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	IC50	10.0	nM	10.1016/j.ejmech.2010.04.026
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	IC50	100.0	nM	10.1016/j.bmcl.2013.07.020
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Cyclin-dependent kinase 5/CDK5 activator 1	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Cyclin-dependent kinase 7	Kd	45.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 7	Kd	45.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 7/ cyclin H	IC50	910.0	nM	10.1021/jm301234k
Homo sapiens	Cyclin-dependent kinase 7/ cyclin H	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Cyclin-dependent kinase 7/ cyclin H	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Cyclin-dependent kinase 9	Kd	100.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 9	Kd	100.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase-like 1	Kd	330.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase-like 2	Kd	510.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase-like 3	IC50	1100.0	nM	10.1016/j.ejmech.2021.113299
Homo sapiens	Cyclin-dependent kinase-like 3	Kd	5100.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase-like 5	Kd	340.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-Y/Cyclin-dependent kinase 16	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cyclin-Y/Cyclin-dependent kinase 16	IC50	17.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Cyclin-Y/Cyclin-dependent kinase 16	IC50	24.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Cytochrome P450 11B2	IC50	11.0	nM	10.1021/jm401430e
Homo sapiens	Death-associated protein kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Death-associated protein kinase 1	IC50	0.5	nM	10.1021/jm800861c
Homo sapiens	Death-associated protein kinase 1	IC50	8.88	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Death-associated protein kinase 1	IC50	9.4	nM	10.1016/j.bmcl.2017.02.068
Homo sapiens	Death-associated protein kinase 1	IC50	13.08	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Death-associated protein kinase 1	IC50	13.1	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	Death-associated protein kinase 1	IC50	15.7	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Death-associated protein kinase 1	Inhibition	86.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Death-associated protein kinase 1	Kd	1.4	nM	10.1038/nbt1358
Homo sapiens	Death-associated protein kinase 1	Kd	1.4	nM	10.1038/nbt.1990
Homo sapiens	Death-associated protein kinase 1	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Death-associated protein kinase 1	Residual Activity	6.0	%	10.1042/bj20121418
Homo sapiens	Death-associated protein kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Death-associated protein kinase 2	IC50	5.56	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Death-associated protein kinase 2	IC50	7.25	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Death-associated protein kinase 2	Kd	1.6	nM	10.1038/nbt1358
Homo sapiens	Death-associated protein kinase 2	Kd	1.6	nM	10.1038/nbt.1990
Homo sapiens	Death-associated protein kinase 2	Kd	3.0	nM	10.1038/nbt1068
Homo sapiens	Death-associated protein kinase 2	Residual Activity	4.0	%	10.1042/bj20121418
Homo sapiens	Death-associated protein kinase 2	Residual Activity	6.0	%	10.1042/bj20121418
Homo sapiens	Death-associated protein kinase 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Death-associated protein kinase 3	IC50	1.84	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Death-associated protein kinase 3	IC50	3.45	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Death-associated protein kinase 3	Kd	1.0	nM	10.1038/nbt1068
Homo sapiens	Death-associated protein kinase 3	Kd	1.0	nM	10.1038/nbt1358
Homo sapiens	Death-associated protein kinase 3	Kd	1.0	nM	10.1038/nbt.1990
Homo sapiens	Death-associated protein kinase 3	Kd	1500.0	nM	10.1038/nbt1358
Homo sapiens	Death-associated protein kinase 3	Residual Activity	-3.0	%	10.1042/bj20121418
Homo sapiens	Death-associated protein kinase 3	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Discoidin domain-containing receptor 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Discoidin domain-containing receptor 2	IC50	0.367	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Discoidin domain-containing receptor 2	IC50	1.19	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Discoidin domain-containing receptor 2	Kd	42.0	nM	10.1038/nbt1358
Homo sapiens	Discoidin domain-containing receptor 2	Kd	42.0	nM	10.1038/nbt.1990
Homo sapiens	Discoidin domain-containing receptor 2	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Discoidin domain-containing receptor 2	Residual Activity	6.0	%	10.1042/bj20121418
Homo sapiens	DLD-1	IC50	9.0	nM	10.1016/j.ejmech.2011.11.040
Homo sapiens	DLD-1	IC50	9.0	nM	10.1016/s0960-894x(01)00535-2
Homo sapiens	DNA-(apurinic or apyrimidinic site) lyase	Potency	39810.7	nM	None
Homo sapiens	DOV13	EC50	nan	None	10.1016/j.bmcl.2006.05.092
Homo sapiens	DU-145	IC50	500.0	nM	10.1021/acs.jnatprod.9b00140
Homo sapiens	Dual serine/threonine and tyrosine protein kinase	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual serine/threonine and tyrosine protein kinase	IC50	31.3	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual serine/threonine and tyrosine protein kinase	IC50	65.2	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual serine/threonine and tyrosine protein kinase	IC50	69.0	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	Dual serine/threonine and tyrosine protein kinase	Kd	11.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	IC50	2.5	nM	10.1021/jm0102856
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	IC50	8.07	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	IC50	12.1	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	IC50	17.9	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	IC50	23.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	IC50	24.0	nM	10.1016/j.ejmech.2015.08.027
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	IC50	45.8	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	IC50	300.0	nM	10.1021/np4005745
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	IC50	670.0	nM	10.1016/j.bmc.2009.05.031
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	IC50	670.0	nM	10.1016/j.ejmech.2013.07.046
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	IC50	1000.0	nM	10.1021/jm020143r
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Kd	21.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Kd	21.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Potency	100.0	nM	None
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Residual Activity	6.0	%	10.1042/bj20121418
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	IC50	14.6	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	IC50	37.4	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Kd	28.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Kd	28.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 3	IC50	2.54	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 3	IC50	17.2	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 3	Kd	5.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 3	Kd	5.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 4	IC50	1.0	nM	10.1021/jm020143r
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 4	IC50	988.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 4	IC50	1600.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 4	Kd	70.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 4	Kd	70.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 5	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 5	Activity	78.0	%	10.1016/j.bmc.2010.09.017
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 5	IC50	10.1	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 5	IC50	40.4	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 5	Inhibition	22.0	%	10.1016/j.bmc.2010.09.017
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 5	Kd	2.9	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	IC50	1.0	nM	10.1021/jm020143r
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	IC50	1.44	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	IC50	8.34	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Kd	3.4	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Kd	3.4	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Residual Activity	-3.0	%	10.1042/bj20121418
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 7	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 7	IC50	571.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 7	IC50	1280.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 7	Kd	30.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 7	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 7	Residual Activity	12.0	%	10.1042/bj20121418
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase; MEK1/2	Activity	18.0	%	10.1016/j.bmc.2010.09.017
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase; MEK1/2	Inhibition	82.0	%	10.1016/j.bmc.2010.09.017
Homo sapiens	Dual specificity protein kinase CLK2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity protein kinase CLK2	IC50	2.86	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity protein kinase CLK2	IC50	5.52	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity protein kinase CLK2	IC50	5.6	nM	10.1021/acs.jmedchem.0c01579
Homo sapiens	Dual specificity protein kinase CLK2	Kd	8.2	nM	10.1038/nbt1358
Homo sapiens	Dual specificity protein kinase CLK2	Kd	8.2	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase CLK2	Kd	12.0	nM	10.1038/nbt1068
Homo sapiens	Dual specificity protein kinase CLK2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Dual specificity protein kinase CLK2	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Dual specificity protein kinase CLK3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity protein kinase CLK3	IC50	530.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity protein kinase CLK3	IC50	1310.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity protein kinase CLK3	Kd	910.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity protein kinase CLK3	Kd	910.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase CLK3	Kd	3500.0	nM	10.1038/nbt1068
Homo sapiens	Dual specificity protein kinase CLK3	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Dual specificity protein kinase CLK3	Residual Activity	56.0	%	10.1042/bj20121418
Homo sapiens	Dual specificity protein kinase CLK4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity protein kinase CLK4	IC50	33.6	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity protein kinase CLK4	IC50	111.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity protein kinase CLK4	Kd	9.6	nM	10.1038/nbt1358
Homo sapiens	Dual specificity protein kinase CLK4	Kd	9.6	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase CLK4	Kd	15.0	nM	10.1038/nbt1068
Homo sapiens	Dual specificity protein kinase TTK	Kd	61.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity protein kinase TTK	Kd	61.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase TTK	Kd	100.0	nM	10.1038/nbt1068
Homo sapiens	Dual specificity testis-specific protein kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity testis-specific protein kinase 1	IC50	138.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity testis-specific protein kinase 1	IC50	261.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity testis-specific protein kinase 1	Kd	320.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity testis-specific protein kinase 1	Kd	320.0	nM	10.1038/nbt.1990
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	IC50	3.13	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	IC50	4.93	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	IC50	5.4	nM	10.1016/j.ejmech.2018.08.093
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	IC50	11.0	nM	10.1016/j.bmcl.2021.128226
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	IC50	19.0	nM	10.1021/acs.jmedchem.8b00185
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	Kd	4.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	IC50	0.967	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	IC50	1.14	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	IC50	3.0	nM	10.1016/j.bmcl.2021.128226
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Kd	28.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Kd	28.0	nM	10.1038/nbt.1990
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 2	IC50	112.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 2	IC50	248.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 2	Kd	250.0	nM	10.1038/nbt.1990
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 2	Residual Activity	17.0	%	10.1042/bj20121418
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 2	Residual Activity	65.0	%	10.1042/bj20121418
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 3	IC50	11.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 3	IC50	34.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 4	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificty protein kinase CLK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificty protein kinase CLK1	IC50	7.45	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificty protein kinase CLK1	IC50	14.2	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Dual specificty protein kinase CLK1	Kd	27.0	nM	10.1038/nbt1068
Homo sapiens	Dual specificty protein kinase CLK1	Kd	32.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificty protein kinase CLK1	Kd	32.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 1	IC50	49.8	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Ephrin type-A receptor 1	IC50	95.3	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-A receptor 1	IC50	139.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 1	Kd	300.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 1	Kd	300.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 1	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 1	Residual Activity	5.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 2	Delta Tm	7.0	degrees C	10.1016/j.ejmech.2020.112721
Homo sapiens	Ephrin type-A receptor 2	IC50	39.9	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-A receptor 2	IC50	74.5	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 2	IC50	262.6	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Ephrin type-A receptor 2	Inhibition	92.6	%	10.1021/jm070342g
Homo sapiens	Ephrin type-A receptor 2	Kd	870.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 2	Kd	1200.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 2	Kd	1200.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 2	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 2	Residual Activity	32.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 3	IC50	19.72	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Ephrin type-A receptor 3	IC50	31.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 3	IC50	39.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-A receptor 3	IC50	48.0	nM	10.1021/jm800861c
Homo sapiens	Ephrin type-A receptor 3	Kd	27.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 3	Kd	27.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 3	Kd	55.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 3	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 3	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 4	IC50	8.5	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-A receptor 4	IC50	12.5	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 4	Kd	290.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 4	Kd	290.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 4	Kd	710.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 4	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 4	Residual Activity	15.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 5	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 5	IC50	10.3	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-A receptor 5	IC50	21.5	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 5	Kd	95.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 5	Kd	95.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 5	Kd	150.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 5	Residual Activity	4.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 5	Residual Activity	7.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 6	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 6	IC50	11.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 6	IC50	20.3	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-A receptor 6	Kd	240.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 6	Kd	290.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 6	Kd	290.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 7	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 7	IC50	39.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-A receptor 7	IC50	56.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 7	Kd	630.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 7	Kd	630.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 7	Kd	690.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 7	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 7	Residual Activity	22.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 8	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 8	IC50	75.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-A receptor 8	IC50	137.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-A receptor 8	Kd	190.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 8	Kd	190.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 8	Kd	300.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 8	Residual Activity	10.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-A receptor 8	Residual Activity	33.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-B receptor 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-B receptor 1	IC50	20.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-B receptor 1	IC50	60.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-B receptor 1	IC50	127.9	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Ephrin type-B receptor 1	Kd	240.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-B receptor 1	Kd	240.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 1	Kd	590.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-B receptor 1	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-B receptor 1	Residual Activity	21.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-B receptor 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-B receptor 2	IC50	42.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-B receptor 2	IC50	116.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-B receptor 2	IC50	198.8	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Ephrin type-B receptor 2	Kd	2100.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-B receptor 2	Kd	2100.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-B receptor 2	Residual Activity	20.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-B receptor 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-B receptor 3	IC50	741.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-B receptor 3	IC50	1830.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-B receptor 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-B receptor 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 3	Residual Activity	119.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-B receptor 3	Residual Activity	131.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-B receptor 4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-B receptor 4	IC50	126.4	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Ephrin type-B receptor 4	IC50	150.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-B receptor 4	IC50	233.0	nM	10.1021/jm800861c
Homo sapiens	Ephrin type-B receptor 4	IC50	238.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ephrin type-B receptor 4	Inhibition	94.1	%	10.1021/jm070342g
Homo sapiens	Ephrin type-B receptor 4	Kd	2200.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-B receptor 4	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ephrin type-B receptor 4	Residual Activity	15.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-B receptor 4	Residual Activity	79.0	%	10.1042/bj20121418
Homo sapiens	Ephrin type-B receptor 6	Kd	210.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor	IC50	10.6	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Epidermal growth factor receptor erbB1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.29	nM	10.1021/acs.jmedchem.7b00178
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.38	nM	10.1021/acs.jmedchem.7b00178
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.6	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.1	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.2	nM	10.1021/acsmedchemlett.8b00373
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	2.3	nM	10.1016/j.bmcl.2020.127288
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	11.4	nM	10.1021/acs.jmedchem.7b00178
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	12.6	nM	10.1016/j.bmcl.2020.127288
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	16.5	nM	10.1021/acsmedchemlett.8b00373
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	26.7	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	37.0	nM	10.1021/acs.jmedchem.7b00178
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	39.8	nM	10.1016/j.ejmech.2021.113674
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	41.0	nM	10.1016/j.bmcl.2020.127288
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	44.0	nM	10.1016/j.bmc.2017.04.003
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	47.0	nM	10.1016/j.ejmech.2018.06.011
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	48.0	nM	10.1016/j.bmc.2016.02.017
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	49.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	50.5	nM	10.1016/j.bmcl.2020.127288
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	58.7	nM	10.1016/j.bmcl.2020.127288
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	68.0	nM	10.1016/j.ejmech.2016.12.055
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	74.2	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	78.0	nM	10.1016/j.ejmech.2021.113327
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	100.0	nM	10.1016/0960-894X(94)80004-9
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	102.4	nM	10.1016/j.ejmech.2010.04.026
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	125.0	nM	10.1016/j.bmcl.2020.127288
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	132.0	nM	10.1021/jm800861c
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	155.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	188.3	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	238.0	nM	10.1016/j.bmc.2017.04.001
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	283.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	283.0	nM	10.1016/j.ejmech.2021.113511
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	430.57	nM	10.1016/j.ejmech.2021.113495
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	178000.0	nM	10.1016/j.bmcl.2017.04.014
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	nan	None	10.1016/j.bmc.2017.09.003
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	59.0	%	10.1016/j.ejmech.2012.10.017
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	70.0	%	10.1016/j.bmc.2016.03.008
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	82.4	%	10.1021/jm070342g
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	86.0	%	10.1016/j.ejmech.2018.06.011
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	90.0	%	10.1016/j.ejmech.2012.09.039
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	94.0	%	10.1016/j.ejmech.2017.12.022
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	96.0	%	10.1016/j.ejmech.2012.10.017
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	96.8	%	10.1016/j.ejmech.2015.04.018
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	97.6	%	10.1016/j.ejmech.2013.03.043
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	97.6	%	10.1016/j.ejmech.2013.07.056
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	99.1	%	10.1016/j.bmc.2011.06.022
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	100.0	%	10.1016/j.bmc.2011.06.022
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	100.0	%	10.1016/j.ejmech.2018.06.011
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1021/acsmedchemlett.8b00373
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	0.35	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	0.77	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	70.0	nM	10.1038/nbt1068
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	96.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	96.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	120.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	120.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	210.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	210.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	270.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	270.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	290.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	290.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	300.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	300.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	370.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	370.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	600.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	600.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	1100.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	1100.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Potency	5.6	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	Potency	39.8	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	Potency	354.8	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	Potency	398.1	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	Residual Activity	19.0	%	10.1042/bj20121418
Homo sapiens	Epidermal growth factor receptor erbB1	Residual Activity	53.0	%	10.1042/bj20121418
Homo sapiens	Epithelial discoidin domain-containing receptor 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Epithelial discoidin domain-containing receptor 1	IC50	2.09	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Epithelial discoidin domain-containing receptor 1	IC50	4.28	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Epithelial discoidin domain-containing receptor 1	IC50	2890.0	nM	10.1016/j.ejmech.2020.112756
Homo sapiens	Epithelial discoidin domain-containing receptor 1	Kd	19.0	nM	10.1038/nbt1358
Homo sapiens	Epithelial discoidin domain-containing receptor 1	Kd	19.0	nM	10.1038/nbt.1990
Homo sapiens	Eukaryotic translation initiation factor 2-alpha kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Eukaryotic translation initiation factor 2-alpha kinase 4	Kd	16.0	nM	10.1038/nbt1358
Homo sapiens	Eukaryotic translation initiation factor 2-alpha kinase 4	Kd	16.0	nM	10.1038/nbt.1990
Homo sapiens	FaDu	EC50	100.0	nM	10.1016/j.ejmech.2020.112920
Homo sapiens	FaDu	EC50	200.0	nM	10.1016/j.ejmech.2019.02.057
Homo sapiens	FaDu	IC50	100.0	nM	10.1016/j.ejmech.2020.112425
Homo sapiens	Fibroblast	Control DMSO Apoptotic Cells (%)	49.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Apoptotic Cells (%)	50.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Apoptotic Cells (%)	52.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Apoptotic Cells (%)	53.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Apoptotic Cells (%)	55.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Apoptotic Cells (%)	63.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Apoptotic Cells (%)	65.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Apoptotic Cells (%)	66.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Apoptotic Cells (%)	68.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Apoptotic Cells (%)	69.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Apoptotic Cells (%)	80.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	11.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	12.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	15.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	18.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	21.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	22.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	24.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	25.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	32.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	55.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	58.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Fragmented Nuclei %	59.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Growth Rate	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Growth Rate	1.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Growth Rate	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Growth Rate	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Growth Rate	231110.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	31.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	34.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	44.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	51.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	53.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	59.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	60.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	61.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	62.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	64.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	66.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	67.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	68.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	69.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	70.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	72.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	75.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Healthy Nuclei (%)	83.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	1.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	4.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	5.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Membrane Permeable-Phenotype Cells (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	1.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	1.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	15.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	24.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitochondria Different-Phenotype Cells (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	19.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	30.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	31.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	31.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	34.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	36.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	37.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	44.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	46.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	47.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	49.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	49.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	50.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	56.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	59.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	61.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Mitotic Cells (%)	62.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	15.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	16.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	20.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	20.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	21.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	22.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Pyknosed Nuclei (%)	36.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Total Cells	80.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Total Cells	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Total Cells	99.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Total Cells	101.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Total Cells	106.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Total Cells	107.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Total Cells	108.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Total Cells	110.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Total Cells	125.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Total Cells	127.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Total Cells	131.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Total Cells	198.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Total Cells	199.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Total Cells	205.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Total Cells	208.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Total Cells	211.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Total Cells	212.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Total Cells	216.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Total Cells	230.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Total Cells	242.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	4.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	5.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	7.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	8.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	9.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	11.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	20.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	30.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	31.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Control DMSO Tubulin Phenotype Different Cells (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Growth Rate	-0.7	None	10.6019/CHEMBL5058564
Homo sapiens	Fibroblast	Growth Rate	-0.13	None	10.6019/CHEMBL5058564
Homo sapiens	Fibroblast	Growth Rate	0.0	None	10.6019/CHEMBL5058564
Homo sapiens	Fibroblast	Growth Rate	0.05	None	10.6019/CHEMBL5058564
Homo sapiens	Fibroblast	Growth Rate	0.35	None	10.6019/CHEMBL5058564
Homo sapiens	Fibroblast	Growth Rate	0.41	None	10.6019/CHEMBL5058564
Homo sapiens	Fibroblast	Growth Rate	0.61	None	10.6019/CHEMBL5058564
Homo sapiens	Fibroblast	Population Apoptotic (%)	31.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	35.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	44.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	50.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	56.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	60.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	63.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	70.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	71.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	71.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	72.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	72.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	73.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	73.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	74.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	75.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	76.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	77.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	83.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	85.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	86.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	87.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	87.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	88.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	88.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	91.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	91.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	92.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Apoptotic (%)	92.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	93.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	95.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	99.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Apoptotic (%)	100.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	13.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	15.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	16.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	17.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	18.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	20.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	21.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	22.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	22.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	23.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	24.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	27.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	28.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	30.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	31.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	32.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	36.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	41.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	42.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	47.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	48.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	51.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	52.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	58.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	59.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	60.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	61.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	64.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	79.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Fragmented Nuclei (%)	82.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	2.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	3.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	4.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	5.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	6.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	7.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	9.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	14.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	19.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	20.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	21.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	30.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	31.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	37.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	38.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	43.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	46.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	52.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	54.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	55.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	57.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	58.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	58.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	62.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Healthy Nuclei (%)	64.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	1.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	20.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	21.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	22.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	25.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	31.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	34.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	36.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	38.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	41.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	43.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	44.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Hoechst High Intensity Objects (%)	46.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	1.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	1.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	2.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	3.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	7.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	15.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	20.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	21.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	25.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	25.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	28.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	30.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	30.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	31.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	36.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	37.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	40.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	47.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	50.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	58.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	63.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	66.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	88.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	92.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Membrane Permeable-Phenotype (%)	100.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	2.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	17.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	17.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	20.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	21.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	30.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	31.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	43.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	75.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	92.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitochondria Different-Phenotype (%)	95.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	4.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	6.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	7.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	8.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	11.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	12.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	22.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	23.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	24.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	25.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	26.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	27.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	28.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	28.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	36.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	40.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	43.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	50.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	55.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	65.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Mitotic Cells (%)	68.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Normal (%)	53.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	55.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	56.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	58.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	61.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	63.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	65.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	66.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	68.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	70.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	72.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	73.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	74.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	77.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	78.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	79.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	81.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	85.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	86.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	87.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	88.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Normal (%)	98.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Normal (%)	99.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Normal (%)	100.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	17.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	17.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	19.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	20.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	25.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	30.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	32.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	33.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	34.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	35.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	36.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	37.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	38.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	41.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	43.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	45.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	46.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	52.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	57.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	59.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	66.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	69.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	71.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	72.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	74.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	78.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	82.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Pyknosed Nuclei (%)	84.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	4.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	7.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	13.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	14.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	17.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	20.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	25.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	28.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	40.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	42.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	45.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	50.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	53.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	54.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	54.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	55.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	55.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	58.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	60.0	%	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	66.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	91.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	92.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Population Tubulin-Different-Phenotype (%)	95.0	%	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	58.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	64.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	85.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	91.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	95.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	117.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	121.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	121.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	134.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	135.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	137.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	143.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	146.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	155.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	160.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	160.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	161.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	164.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	166.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	168.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	171.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	173.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	174.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	178.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	180.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	184.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	189.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	190.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	194.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	197.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	206.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	208.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	209.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	231.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	269.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	273.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	274.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	283.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	294.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	323.0	None	10.6019/CHEMBL5303300
Homo sapiens	Fibroblast	Total Cell Count	389.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	475.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Total Cell Count	882.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast growth factor receptor	IC50	27.0	nM	10.1016/j.bmcl.2021.128258
Homo sapiens	Fibroblast growth factor receptor	IC50	420.0	nM	10.1021/jm020143r
Homo sapiens	Fibroblast growth factor receptor 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Fibroblast growth factor receptor 1	IC50	2.42	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Fibroblast growth factor receptor 1	IC50	3.89	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Fibroblast growth factor receptor 1	IC50	6.3	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Fibroblast growth factor receptor 1	IC50	9.0	nM	10.1021/jm800861c
Homo sapiens	Fibroblast growth factor receptor 1	IC50	21.0	nM	10.1016/j.ejmech.2021.113219
Homo sapiens	Fibroblast growth factor receptor 1	Inhibition	86.5	%	10.1021/jm070342g
Homo sapiens	Fibroblast growth factor receptor 1	Kd	60.0	nM	10.1038/nbt1068
Homo sapiens	Fibroblast growth factor receptor 1	Kd	90.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 1	Kd	90.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 1	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Fibroblast growth factor receptor 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Fibroblast growth factor receptor 2	IC50	0.757	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Fibroblast growth factor receptor 2	IC50	1.77	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Fibroblast growth factor receptor 2	IC50	1.77	nM	10.1016/j.ejmech.2021.113511
Homo sapiens	Fibroblast growth factor receptor 2	IC50	2.09	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Fibroblast growth factor receptor 2	IC50	3.36	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Fibroblast growth factor receptor 2	IC50	5.8	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Fibroblast growth factor receptor 2	IC50	7.4	nM	10.1016/j.ejmech.2021.113219
Homo sapiens	Fibroblast growth factor receptor 2	IC50	34.0	nM	10.1021/jm800861c
Homo sapiens	Fibroblast growth factor receptor 2	Kd	100.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 2	Kd	100.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 2	Kd	160.0	nM	10.1038/nbt1068
Homo sapiens	Fibroblast growth factor receptor 2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Fibroblast growth factor receptor 2	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Fibroblast growth factor receptor 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Fibroblast growth factor receptor 3	Delta TM	13.02	C	None
Homo sapiens	Fibroblast growth factor receptor 3	IC50	6.42	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Fibroblast growth factor receptor 3	IC50	9.25	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Fibroblast growth factor receptor 3	IC50	10.3	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Fibroblast growth factor receptor 3	IC50	14.71	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Fibroblast growth factor receptor 3	IC50	15.6	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Fibroblast growth factor receptor 3	IC50	16.0	nM	10.1016/j.ejmech.2021.113219
Homo sapiens	Fibroblast growth factor receptor 3	IC50	16.7	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Fibroblast growth factor receptor 3	IC50	18.0	nM	10.1021/jm800861c
Homo sapiens	Fibroblast growth factor receptor 3	Kd	88.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 3	Kd	88.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 3	Kd	110.0	nM	10.1038/nbt1068
Homo sapiens	Fibroblast growth factor receptor 3	Kd	310.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 3	Kd	310.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 3	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Fibroblast growth factor receptor 3	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Fibroblast growth factor receptor 4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Fibroblast growth factor receptor 4	IC50	77.9	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Fibroblast growth factor receptor 4	IC50	107.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Fibroblast growth factor receptor 4	IC50	148.3	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Fibroblast growth factor receptor 4	IC50	240.0	nM	10.1016/j.ejmech.2021.113219
Homo sapiens	Fibroblast growth factor receptor 4	IC50	97300000.0	nM	10.1016/j.bmc.2018.10.004
Homo sapiens	Fibroblast growth factor receptor 4	Kd	250.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 4	Kd	250.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 4	Residual Activity	14.0	%	10.1042/bj20121418
Homo sapiens	Fibroblast growth factor receptor 4	Residual Activity	49.0	%	10.1042/bj20121418
Homo sapiens	Focal adhesion kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Focal adhesion kinase 1	EC50	11.32	ug.mL-1	10.1016/j.bmcl.2011.08.039
Homo sapiens	Focal adhesion kinase 1	IC50	9.12	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Focal adhesion kinase 1	IC50	11.0	nM	10.1021/acs.jnatprod.7b01082
Homo sapiens	Focal adhesion kinase 1	IC50	13.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Focal adhesion kinase 1	IC50	13.2	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Focal adhesion kinase 1	IC50	17.15	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Focal adhesion kinase 1	IC50	20.0	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Focal adhesion kinase 1	IC50	55.0	nM	10.1016/j.ejmech.2015.08.027
Homo sapiens	Focal adhesion kinase 1	IC50	62.0	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Focal adhesion kinase 1	IC50	80.0	nM	10.1021/np4005745
Homo sapiens	Focal adhesion kinase 1	IC50	500.0	nM	10.1016/j.bmc.2014.04.005
Homo sapiens	Focal adhesion kinase 1	IC50	3120.0	nM	10.1007/s00044-012-0306-5
Homo sapiens	Focal adhesion kinase 1	Inhibition	81.7	%	10.1021/jm070342g
Homo sapiens	Focal adhesion kinase 1	Kd	64.0	nM	10.1038/nbt1358
Homo sapiens	Focal adhesion kinase 1	Kd	64.0	nM	10.1038/nbt.1990
Homo sapiens	Focal adhesion kinase 1	Kd	68.0	nM	10.1038/nbt1068
Homo sapiens	Focal adhesion kinase 1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Focal adhesion kinase 1	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	G-361	IC50	nan	None	10.1016/j.bmcl.2012.08.005
Homo sapiens	Gamma-secretase	IC50	nan	None	10.1016/j.bmcl.2012.10.016
Homo sapiens	Glycogen synthase kinase-3	IC50	12.0	nM	10.1016/j.bmcl.2006.05.092
Homo sapiens	Glycogen synthase kinase-3 alpha	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Glycogen synthase kinase-3 alpha	IC50	2.4	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Glycogen synthase kinase-3 alpha	IC50	3.97	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Glycogen synthase kinase-3 alpha	IC50	5.1	nM	10.1021/acs.jmedchem.0c01579
Homo sapiens	Glycogen synthase kinase-3 alpha	IC50	28.0	nM	10.1016/j.bmcl.2014.08.049
Homo sapiens	Glycogen synthase kinase-3 alpha	Kd	140.0	nM	10.1038/nbt1358
Homo sapiens	Glycogen synthase kinase-3 alpha	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	Glycogen synthase kinase-3 alpha	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	Glycogen synthase kinase-3 alpha	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Glycogen synthase kinase-3 beta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Glycogen synthase kinase-3 beta	Activity	99.9	%	10.1016/j.ejmech.2010.04.026
Homo sapiens	Glycogen synthase kinase-3 beta	Delta TM	10.75	C	None
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	2.62	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	4.0	nM	10.1016/j.ejmech.2015.10.018
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	4.21	nM	10.1021/acs.jmedchem.6b00944
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	5.0	nM	10.1016/j.ejmech.2010.04.026
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	5.1	nM	10.1021/acs.jmedchem.0c01579
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	5.2	nM	10.1021/jm800861c
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	5.28	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	5.38	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	5.53	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	9.23	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	10.1	nM	10.1016/j.bmcl.2023.129263
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	11.0	nM	10.1016/j.bmcl.2011.10.076
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	15.0	nM	10.1016/j.bmcl.2017.11.036
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	15.0	nM	10.1016/j.ejmech.2008.08.012
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	15.0	nM	10.1021/jm301234k
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	18.6	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	24.0	nM	10.1016/j.ejmech.2019.02.001
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	24.0	nM	10.1021/acs.jnatprod.7b01082
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	30.0	nM	10.1016/j.ejmech.2021.113554
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	30.0	nM	10.1016/j.ejmech.2021.114095
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	33.0	nM	10.1016/j.bmcl.2014.05.085
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	38.0	nM	10.1016/j.bmc.2014.12.026
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	40.0	nM	10.1016/j.ejmech.2018.12.073
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	50.0	nM	10.1016/j.bmcl.2014.08.049
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	51.6	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	53.0	nM	10.1021/acsmedchemlett.9b00633
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	54.0	nM	10.1016/j.bmcl.2016.06.084
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	54.0	nM	10.1016/j.ejmech.2018.12.073
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	56.0	nM	10.1016/j.bmc.2009.05.031
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	56.0	nM	10.1021/jm049768a
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	63.8	nM	10.1016/j.ejmech.2020.112277
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	72.0	nM	10.1016/j.ejmech.2013.11.036
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	72.2	nM	10.1039/C7MD00449D
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	89.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	160.0	nM	10.1021/jm021095d
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	200.0	nM	10.1016/j.bmc.2009.05.031
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	200.0	nM	10.1016/j.ejmech.2013.07.046
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	nan	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Glycogen synthase kinase-3 beta	IC50	nan	nM	10.1021/jm049768a
Homo sapiens	Glycogen synthase kinase-3 beta	Inhibition	8.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Glycogen synthase kinase-3 beta	Inhibition	99.9	%	10.1016/j.ejmech.2021.113554
Homo sapiens	Glycogen synthase kinase-3 beta	IZ	13.0	mm	10.1021/np900163f
Homo sapiens	Glycogen synthase kinase-3 beta	IZ	nan	None	10.1021/np900163f
Homo sapiens	Glycogen synthase kinase-3 beta	Kd	4.3	nM	10.1021/acsmedchemlett.3c00127
Homo sapiens	Glycogen synthase kinase-3 beta	Kd	69.0	nM	10.1038/nbt1358
Homo sapiens	Glycogen synthase kinase-3 beta	Kd	69.0	nM	10.1038/nbt.1990
Homo sapiens	Glycogen synthase kinase-3 beta	Ki	22.0	nM	10.1016/j.bmcl.2010.01.072
Homo sapiens	Glycogen synthase kinase-3 beta	Residual Activity	4.0	%	10.1042/bj20121418
Homo sapiens	Glycogen synthase kinase-3 beta	Residual Activity	13.0	%	10.1042/bj20121418
Homo sapiens	G-protein coupled receptor kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	G-protein coupled receptor kinase 2	IC50	879.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	G-protein coupled receptor kinase 2	IC50	1440.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	G protein-coupled receptor kinase 4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	G protein-coupled receptor kinase 4	IC50	69.9	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	G protein-coupled receptor kinase 4	IC50	113.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	G protein-coupled receptor kinase 4	Kd	37.0	nM	10.1038/nbt.1990
Homo sapiens	G protein-coupled receptor kinase 5	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	G protein-coupled receptor kinase 5	IC50	24.6	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	G protein-coupled receptor kinase 5	IC50	73.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	G protein-coupled receptor kinase 5	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	G protein-coupled receptor kinase 5	Residual Activity	10.0	%	10.1042/bj20121418
Homo sapiens	G protein-coupled receptor kinase 6	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	G protein-coupled receptor kinase 6	IC50	32.9	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	G protein-coupled receptor kinase 6	IC50	61.7	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	G protein-coupled receptor kinase 6	IC50	34000.0	nM	None
Homo sapiens	G protein-coupled receptor kinase 6	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	G protein-coupled receptor kinase 6	Residual Activity	17.0	%	10.1042/bj20121418
Homo sapiens	G protein-coupled receptor kinase 7	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	G protein-coupled receptor kinase 7	IC50	4.56	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	G protein-coupled receptor kinase 7	IC50	5.96	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	G protein-coupled receptor kinase 7	Kd	0.86	nM	10.1038/nbt.1990
Homo sapiens	G protein-coupled receptor kinase 7	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	HaCaT	IC50	1600.0	nM	10.1021/acs.jnatprod.1c01211
Homo sapiens	HCT-116	Activity	3.0	%	10.1016/j.ejmech.2018.11.034
Homo sapiens	HCT-116	Activity	8.4	%	10.1016/j.ejmech.2018.11.034
Homo sapiens	HCT-116	Activity	25.6	%	10.1016/j.ejmech.2018.11.034
Homo sapiens	HCT-116	Activity	27.0	%	10.1016/j.ejmech.2019.01.052
Homo sapiens	HCT-116	Activity	63.1	%	10.1016/j.ejmech.2018.11.034
Homo sapiens	HCT-116	Activity	nan	None	10.1016/j.ejmech.2018.11.034
Homo sapiens	HCT-116	IC50	6.0	nM	10.1021/jm020455u
Homo sapiens	HCT-116	IC50	28.1	nM	10.1016/j.ejmech.2020.113003
Homo sapiens	HCT-116	IC50	30.0	nM	10.1021/acs.jnatprod.8b00103
Homo sapiens	HCT-116	IC50	37.0	nM	10.1016/j.bmcl.2019.04.023
Homo sapiens	HCT-116	IC50	40.0	nM	10.1021/acsmedchemlett.0c00269
Homo sapiens	HCT-116	IC50	48.1	nM	10.1016/j.ejmech.2021.113727
Homo sapiens	HCT-116	IC50	55.0	nM	10.1021/acs.jnatprod.7b01055
Homo sapiens	HCT-116	IC50	100.0	nM	10.1016/j.bmcl.2019.126807
Homo sapiens	HCT-116	IC50	6940.0	nM	10.1039/d2md00076h
Homo sapiens	HCT-116	IC50	8860.0	nM	10.1021/acs.jmedchem.9b01669
Homo sapiens	HCT-116	IC50	13200.0	nM	10.1007/s00044-012-0306-5
Homo sapiens	HCT-116	IC50	16150.0	nM	10.1021/acs.jmedchem.9b01669
Homo sapiens	HCT-116	IC50	nan	nM	10.1016/s0960-894x(03)00461-x
Homo sapiens	HCT-116	Inhibition	nan	%	10.1016/j.ejmech.2013.10.049
Homo sapiens	HEK293	Activity	45.0	%	10.1021/acs.jmedchem.8b00542
Homo sapiens	HEK293	Activity	60.0	%	10.1021/acs.jmedchem.8b00542
Homo sapiens	HEK293	CC50	3.54	nM	10.1016/j.ejmech.2017.06.020
Homo sapiens	HEK293	EC50	794.33	nM	10.1021/acs.jmedchem.1c01532
Homo sapiens	HEK293	EC50	2000.0	nM	10.1016/j.bmcl.2014.09.061
Homo sapiens	HEK293	EC50	nan	None	10.1016/j.ejmech.2020.112920
Homo sapiens	HEK293	IC50	3.7	nM	10.1016/j.ejmech.2019.06.027
Homo sapiens	HEK293	IC50	56.0	nM	10.1016/j.ejmech.2014.04.025
Homo sapiens	HEK293	IC50	410.0	nM	10.1021/acs.jmedchem.1c01411
Homo sapiens	HEK293	IC50	34330.0	nM	10.1016/j.ejmech.2022.114190
Homo sapiens	HEK-293T	Control DMSO Apoptotic Cells (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Apoptotic Cells (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Apoptotic Cells (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Apoptotic Cells (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Apoptotic Cells (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Apoptotic Cells (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Apoptotic Cells (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Apoptotic Cells (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Apoptotic Cells (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Apoptotic Cells (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Apoptotic Cells (%)	39.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Apoptotic Cells (%)	42.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	3.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	6.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	12.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	14.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	19.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Fragmented Nuclei %	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Growth Rate	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Growth Rate	1.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	21.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	24.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	37.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	39.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	42.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	45.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	49.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	65.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	69.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	69.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	70.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	73.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	77.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	79.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	82.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	82.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	84.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	85.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	86.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Healthy Nuclei (%)	86.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Membrane Permeable-Phenotype Cells (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Membrane Permeable-Phenotype Cells (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Membrane Permeable-Phenotype Cells (%)	1.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Membrane Permeable-Phenotype Cells (%)	1.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Membrane Permeable-Phenotype Cells (%)	2.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Membrane Permeable-Phenotype Cells (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Membrane Permeable-Phenotype Cells (%)	3.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Membrane Permeable-Phenotype Cells (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Membrane Permeable-Phenotype Cells (%)	4.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Membrane Permeable-Phenotype Cells (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Membrane Permeable-Phenotype Cells (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Membrane Permeable-Phenotype Cells (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	4.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	5.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	6.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	7.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	13.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	14.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	17.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	22.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	32.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	51.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	68.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitochondria Different-Phenotype Cells (%)	77.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	49.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	54.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	57.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	57.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	60.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	60.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	62.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	66.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	81.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	81.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	83.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	85.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	85.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	86.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	87.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	88.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	90.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Mitotic Cells (%)	91.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	3.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	7.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	8.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	11.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	26.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	37.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	45.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	48.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	49.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	67.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Pyknosed Nuclei (%)	69.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	233.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	256.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	274.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	293.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	322.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	351.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	364.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Total Cells	370.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Total Cells	594.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	680.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Total Cells	681.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Total Cells	691.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	838.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	865.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	1046.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Total Cells	1069.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Total Cells	1080.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	1765.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Total Cells	2439.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Total Cells	2812.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Total Cells	3025.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	1.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	11.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	12.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	13.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	25.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	27.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	31.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	32.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	45.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	47.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Control DMSO Tubulin Phenotype Different Cells (%)	48.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Growth Rate	-0.75	None	10.6019/CHEMBL5058564
Homo sapiens	HEK-293T	Growth Rate	-0.46	None	10.6019/CHEMBL5058564
Homo sapiens	HEK-293T	Growth Rate	0.09	None	10.6019/CHEMBL5058564
Homo sapiens	HEK-293T	Growth Rate	0.11	None	10.6019/CHEMBL5058564
Homo sapiens	HEK-293T	Growth Rate	0.33	None	10.6019/CHEMBL5058564
Homo sapiens	HEK-293T	Growth Rate	0.42	None	10.6019/CHEMBL5058564
Homo sapiens	HEK-293T	Population Apoptotic (%)	6.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	17.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	25.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	26.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	28.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	29.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	31.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	41.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	48.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	55.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	56.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	58.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	63.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	68.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	70.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	76.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	81.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	82.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	83.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	85.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	86.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	87.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	87.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	89.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	89.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	90.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Apoptotic (%)	91.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	92.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	93.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	95.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	96.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Apoptotic (%)	97.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	2.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	3.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	11.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	13.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	14.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	16.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	20.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	21.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	21.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	22.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	30.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	32.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	35.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	36.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	37.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Fragmented Nuclei (%)	41.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	1.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	17.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	17.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	18.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	19.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	20.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	22.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	23.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	29.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	30.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	34.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	35.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	37.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	37.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	38.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	40.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	50.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	51.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	66.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	72.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	73.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	76.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	82.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Healthy Nuclei (%)	88.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	2.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	3.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	4.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	5.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	6.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	7.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	8.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	9.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	11.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	12.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	14.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	17.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	19.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	20.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	21.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	22.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	24.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Hoechst High Intensity Objects (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	1.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	2.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	5.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	6.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	7.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	11.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	12.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	20.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	28.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Membrane Permeable-Phenotype (%)	35.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	6.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	9.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	12.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	25.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	35.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	45.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	46.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	47.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	51.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	52.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	57.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	60.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	62.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	62.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	63.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	64.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	65.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	66.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	68.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	73.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	75.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	80.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	82.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	83.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitochondria Different-Phenotype (%)	100.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	9.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	12.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	13.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	14.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	16.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	17.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	18.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	31.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	36.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	41.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	43.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	44.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	51.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	58.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	66.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	68.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	70.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	71.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	72.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	73.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	74.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	81.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	82.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	87.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	88.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	89.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	90.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Mitotic Cells (%)	93.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Normal (%)	70.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	73.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	75.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	76.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	77.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	78.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	79.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	80.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	82.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	85.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	85.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Normal (%)	86.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	87.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Normal (%)	88.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	88.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Normal (%)	89.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	89.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Normal (%)	90.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Normal (%)	91.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Normal (%)	92.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Normal (%)	93.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	93.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Normal (%)	94.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	94.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Normal (%)	95.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Normal (%)	96.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Normal (%)	96.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Normal (%)	97.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	8.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	23.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	24.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	29.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	35.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	37.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	41.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	46.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	48.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	50.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	51.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	52.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	55.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	55.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	57.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	58.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	61.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	62.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	63.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	64.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	65.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	65.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	66.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	66.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	70.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	71.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Pyknosed Nuclei (%)	75.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	1.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	16.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	20.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	25.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	32.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	34.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	35.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	44.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	57.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	58.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	59.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	60.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	61.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	68.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	72.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	72.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	73.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	74.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	75.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	76.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	77.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	79.0	%	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	86.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	87.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	89.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Population Tubulin-Different-Phenotype (%)	100.0	%	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	146.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	165.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	213.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	219.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	224.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	241.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	318.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	323.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	325.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	332.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	345.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	355.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	361.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	396.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	410.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	457.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	467.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	472.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	489.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	517.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	520.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	548.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	557.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	562.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	595.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	612.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	654.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	669.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	695.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	728.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	759.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	791.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	806.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	809.0	None	10.6019/CHEMBL5303300
Homo sapiens	HEK-293T	Total Cell Count	855.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	929.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	1044.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	1085.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	1445.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	1593.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	1847.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	2008.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEK-293T	Total Cell Count	2237.0	None	10.6019/CHEMBL4689842
Homo sapiens	HeLa	Activity	33.0	%	10.1016/j.ejmech.2018.07.050
Homo sapiens	HeLa	Activity	33.0	%	10.1016/j.ejmech.2018.08.097
Homo sapiens	HeLa	Activity	nan	None	10.1016/j.bmc.2014.06.032
Homo sapiens	HeLa	Activity	nan	None	10.1016/j.bmcl.2022.128588
Homo sapiens	HeLa	Activity	nan	None	10.1016/j.ejmech.2012.05.032
Homo sapiens	HeLa	Activity	nan	None	10.1038/nchembio809
Homo sapiens	HeLa	Activity	nan	None	10.1039/C2MD20098H
Homo sapiens	HeLa	Concentration	20.0	nM ml-1	10.1016/s0960-894x(03)00592-4
Homo sapiens	HeLa	Concentration	200.0	nM ml-1	10.1016/s0960-894x(03)00592-4
Homo sapiens	HeLa	EC50	29.12	ug.mL-1	10.1016/j.bmcl.2011.08.039
Homo sapiens	HeLa	IC50	0.004	nM	10.1021/np100727h
Homo sapiens	HeLa	IC50	0.004	nM	10.1021/np200035m
Homo sapiens	HeLa	IC50	25.0	nM	10.1021/jm501942m
Homo sapiens	HeLa	IC50	25.0	nM	10.1039/C2MD20098H
Homo sapiens	HeLa	IC50	175.0	nM	10.1016/j.bmcl.2012.08.005
Homo sapiens	HeLa	IC50	2720.0	nM	10.1016/j.bmc.2014.04.005
Homo sapiens	HeLa	IC50	9120.0	nM	10.1016/j.bmc.2012.08.059
Homo sapiens	HeLa S3	IC50	0.004	nM	10.1016/j.ejmech.2020.112506
Homo sapiens	Hepatocyte growth factor receptor	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Hepatocyte growth factor receptor	IC50	33.7	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Hepatocyte growth factor receptor	IC50	57.0	nM	10.1016/j.bmcl.2020.127076
Homo sapiens	Hepatocyte growth factor receptor	IC50	57.0	nM	10.1016/j.bmcl.2020.127740
Homo sapiens	Hepatocyte growth factor receptor	IC50	69.2	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Hepatocyte growth factor receptor	IC50	75.0	nM	None
Homo sapiens	Hepatocyte growth factor receptor	IC50	90.0	nM	10.1016/j.bmc.2017.04.003
Homo sapiens	Hepatocyte growth factor receptor	IC50	90.45	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Hepatocyte growth factor receptor	IC50	103.0	nM	10.1021/jm800861c
Homo sapiens	Hepatocyte growth factor receptor	IC50	128.0	nM	10.1016/j.ejmech.2018.01.061
Homo sapiens	Hepatocyte growth factor receptor	IC50	130.0	nM	10.1016/j.bmcl.2006.05.092
Homo sapiens	Hepatocyte growth factor receptor	IC50	144.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Hepatocyte growth factor receptor	IC50	153.0	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Hepatocyte growth factor receptor	IC50	179.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Hepatocyte growth factor receptor	IC50	179.0	nM	10.1016/j.ejmech.2021.113511
Homo sapiens	Hepatocyte growth factor receptor	IC50	190.0	nM	10.1016/j.bmcl.2016.05.007
Homo sapiens	Hepatocyte growth factor receptor	IC50	310.0	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Hepatocyte growth factor receptor	IC50	404.9	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Hepatocyte growth factor receptor	IC50	940.0	nM	10.1021/np4005745
Homo sapiens	Hepatocyte growth factor receptor	IC50	nan	None	10.1016/j.bmc.2017.09.003
Homo sapiens	Hepatocyte growth factor receptor	Inhibition	87.0	%	10.1016/j.ejmech.2012.09.039
Homo sapiens	Hepatocyte growth factor receptor	Inhibition	90.0	%	10.1021/jm070342g
Homo sapiens	Hepatocyte growth factor receptor	Kd	130.0	nM	10.1038/nbt.1990
Homo sapiens	Hepatocyte growth factor receptor	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	Hepatocyte growth factor receptor	Kd	190.0	nM	10.1038/nbt1358
Homo sapiens	Hepatocyte growth factor receptor	Kd	190.0	nM	10.1038/nbt.1990
Homo sapiens	Hepatocyte growth factor receptor	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Hepatocyte growth factor receptor	Residual Activity	5.0	%	10.1042/bj20121418
Homo sapiens	HepG2	Activity	21.1	%	10.1021/np400653p
Homo sapiens	HepG2	EC50	21.74	ug.mL-1	10.1016/j.bmcl.2011.08.039
Homo sapiens	HepG2	EC50	2000.0	nM	10.1016/j.bmcl.2014.09.061
Homo sapiens	HepG2	IC50	18.0	nM	10.1016/j.bmc.2017.09.037
Homo sapiens	HepG2	IC50	6730.0	nM	10.1016/j.bmc.2012.08.059
Homo sapiens	HepG2	IC50	9040.0	nM	10.1007/s00044-012-0306-5
Homo sapiens	HepG2	IC50 relative	100.0	nM	10.6019/EOS300108
Homo sapiens	HepG2	Inhibition	100.0	%	10.1016/j.ejmech.2013.10.049
Homo sapiens	HERG	IC50	90400.0	nM	10.1016/j.ejmech.2020.112517
Homo sapiens	HERG	Ki	nan	nM	10.1021/jm049478u
Homo sapiens	Hexokinase type IV	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Hexokinase type IV	IC50	0.488	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Hexokinase type IV	IC50	0.81	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Histone acetyltransferase GCN5	Potency	28183.8	nM	None
Homo sapiens	HL-60	Activity	10.5	%	10.1016/j.bmcl.2014.07.033
Homo sapiens	HL-60	Activity	17.4	%	10.1016/j.bmcl.2014.07.033
Homo sapiens	HL-60	IC50	7.6	nM	10.1016/j.ejmech.2020.113003
Homo sapiens	HL-60	IC50	19.0	nM	10.1016/j.bmcl.2019.04.023
Homo sapiens	HL-60	IC50	40.0	nM	10.1021/acsmedchemlett.0c00269
Homo sapiens	HL-60	IC50	41.0	nM	10.1016/j.ejmech.2021.113727
Homo sapiens	HL-60	IC50	9240.0	nM	10.1016/j.bmc.2019.02.005
Homo sapiens	Homeodomain-interacting protein kinase 1	IC50	2639.0	nM	10.1021/jm800861c
Homo sapiens	Homeodomain-interacting protein kinase 1	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Homeodomain-interacting protein kinase 1	Kd	2700.0	nM	10.1038/nbt.1990
Homo sapiens	Homeodomain-interacting protein kinase 1	Residual Activity	59.0	%	10.1042/bj20121418
Homo sapiens	Homeodomain-interacting protein kinase 1	Residual Activity	87.0	%	10.1042/bj20121418
Homo sapiens	Homeodomain-interacting protein kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Homeodomain-interacting protein kinase 2	IC50	146.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Homeodomain-interacting protein kinase 2	IC50	585.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Homeodomain-interacting protein kinase 2	Kd	190.0	nM	10.1038/nbt.1990
Homo sapiens	Homeodomain-interacting protein kinase 2	Residual Activity	12.0	%	10.1042/bj20121418
Homo sapiens	Homeodomain-interacting protein kinase 2	Residual Activity	47.0	%	10.1042/bj20121418
Homo sapiens	Homeodomain-interacting protein kinase 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Homeodomain-interacting protein kinase 3	IC50	202.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Homeodomain-interacting protein kinase 3	IC50	710.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Homeodomain-interacting protein kinase 3	Kd	75.0	nM	10.1038/nbt.1990
Homo sapiens	Homeodomain-interacting protein kinase 3	Residual Activity	27.0	%	10.1042/bj20121418
Homo sapiens	Homeodomain-interacting protein kinase 3	Residual Activity	74.0	%	10.1042/bj20121418
Homo sapiens	Homeodomain-interacting protein kinase 4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Homeodomain-interacting protein kinase 4	IC50	138.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Homeodomain-interacting protein kinase 4	IC50	314.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Homeodomain-interacting protein kinase 4	Kd	390.0	nM	10.1038/nbt.1990
Homo sapiens	Hormonally up-regulated neu tumor-associated kinase	Kd	620.0	nM	10.1038/nbt.1990
Homo sapiens	HT-1080	Activity	61.5	%	10.1007/s00044-012-0428-9
Homo sapiens	HT-29	EC50	150.0	nM	10.1016/j.ejmech.2017.11.046
Homo sapiens	HT-29	EC50	200.0	nM	10.1016/j.ejmech.2019.02.057
Homo sapiens	HT-29	EC50	200.0	nM	10.1016/j.ejmech.2020.112920
Homo sapiens	HT-29	ED50	0.0026	uM	10.1021/np200557e
Homo sapiens	HT-29	ED50	2.6	nM	10.1021/np9001724
Homo sapiens	HT-29	ED50	20.0	uM	10.1021/np200557e
Homo sapiens	HT-29	GI50	10.9	nM	10.1021/np700748h
Homo sapiens	HT-29	GI50	3600.0	nM	10.1021/np200041v
Homo sapiens	HT-29	IC50	2.0	nM	10.1021/np200051j
Homo sapiens	HT-29	IC50	2.5	nM	10.1021/np200062x
Homo sapiens	HT-29	IC50	10.0	nM	10.1016/j.bmcl.2020.127109
Homo sapiens	HT-29	IC50	20.0	nM	10.1016/j.bmc.2018.07.025
Homo sapiens	HT-29	IC50	200.0	nM	10.1016/j.ejmech.2013.11.025
Homo sapiens	HT-29	IC50	200.0	nM	10.1016/j.ejmech.2020.112425
Homo sapiens	HT-29	Inhibition	92.6	%	10.1016/j.ejmech.2013.10.049
Homo sapiens	Huh-7	IC50	230.0	nM	10.1021/np400838a
Homo sapiens	HUVEC	Activity	nan	None	10.1021/acs.jnatprod.1c00008
Homo sapiens	HUVEC	IC50	4.0	nM	10.1016/j.ejmech.2011.11.040
Homo sapiens	HUVEC	IC50	4.0	nM	10.1016/s0960-894x(01)00535-2
Homo sapiens	HUVEC	IC50	500.0	nM	10.1039/D1MD00125F
Homo sapiens	HUVEC	Inhibition	nan	%	10.1039/D1MD00125F
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	IC50	39.0	nM	10.1016/j.ejmech.2011.01.045
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	IC50	62.6	nM	10.1016/j.ejmech.2021.113475
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	IC50	70.7	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	IC50	227.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	IC50	233.0	nM	10.1021/jm801317h
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	Kd	5.8	nM	10.1038/nbt.1990
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	Residual Activity	6.0	%	10.1042/bj20121418
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	IC50	0.9	nM	10.1016/j.bmc.2014.12.026
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	IC50	1.0	nM	10.1016/j.ejmech.2013.11.036
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	IC50	207.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	IC50	250.0	nM	10.1016/j.bmcl.2004.05.040
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	IC50	465.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	IC50	490.0	nM	10.1016/j.ejmech.2011.01.045
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	IC50	771.0	nM	10.1021/jm801317h
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	IC50	1410.0	nM	10.1016/j.bmc.2009.05.031
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	IC50	1410.0	nM	10.1016/j.ejmech.2013.07.046
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	Inhibition	64.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	Kd	31.0	nM	10.1038/nbt.1990
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	Residual Activity	10.0	%	10.1042/bj20121418
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	Residual Activity	35.0	%	10.1042/bj20121418
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	IC50	0.199	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	IC50	0.439	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	Kd	5.1	nM	10.1038/nbt1358
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	Kd	5.1	nM	10.1038/nbt.1990
Homo sapiens	Insulin-like growth factor I receptor	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Insulin-like growth factor I receptor	IC50	27.5	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Insulin-like growth factor I receptor	IC50	35.03	nM	10.1016/j.ejmech.2010.04.026
Homo sapiens	Insulin-like growth factor I receptor	IC50	43.3	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Insulin-like growth factor I receptor	IC50	47.4	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Insulin-like growth factor I receptor	IC50	85.33	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Insulin-like growth factor I receptor	IC50	160.0	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Insulin-like growth factor I receptor	IC50	190.0	nM	10.1021/np4005745
Homo sapiens	Insulin-like growth factor I receptor	IC50	200.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Insulin-like growth factor I receptor	IC50	200.7	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Insulin-like growth factor I receptor	IC50	1325.0	nM	10.1016/j.bmcl.2011.03.003
Homo sapiens	Insulin-like growth factor I receptor	IC50	1533.0	nM	10.1016/j.bmcl.2011.03.003
Homo sapiens	Insulin-like growth factor I receptor	IC50	1646.0	nM	10.1016/j.bmcl.2011.03.003
Homo sapiens	Insulin-like growth factor I receptor	IC50	1701.0	nM	10.1016/j.bmcl.2011.03.003
Homo sapiens	Insulin-like growth factor I receptor	Inhibition	50.0	%	10.1021/acs.jmedchem.7b00324
Homo sapiens	Insulin-like growth factor I receptor	Inhibition	96.9	%	10.1021/jm070342g
Homo sapiens	Insulin-like growth factor I receptor	Kd	210.0	nM	10.1038/nbt1358
Homo sapiens	Insulin-like growth factor I receptor	Kd	210.0	nM	10.1038/nbt.1990
Homo sapiens	Insulin-like growth factor I receptor	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Insulin-like growth factor I receptor	Residual Activity	14.0	%	10.1042/bj20121418
Homo sapiens	Insulin-like growth factor I receptor	Residual Activity	112.0	%	10.1042/bj20121418
Homo sapiens	Insulin receptor	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Insulin receptor	IC50	8.5	nM	10.1021/jm800861c
Homo sapiens	Insulin receptor	IC50	8.81	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Insulin receptor	IC50	14.73	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Insulin receptor	IC50	17.7	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Insulin receptor	IC50	73.6	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Insulin receptor	IC50	300.0	nM	10.1021/jm020143r
Homo sapiens	Insulin receptor	Kd	73.0	nM	10.1038/nbt1068
Homo sapiens	Insulin receptor	Kd	110.0	nM	10.1038/nbt1358
Homo sapiens	Insulin receptor	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	Insulin receptor	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Insulin receptor	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Insulin receptor	Residual Activity	5.0	%	10.1042/bj20121418
Homo sapiens	Insulin receptor	Residual Activity	13.0	%	10.1042/bj20121418
Homo sapiens	Insulin receptor-related protein	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Insulin receptor-related protein	IC50	7.59	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Insulin receptor-related protein	IC50	15.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Insulin receptor-related protein	Kd	81.0	nM	10.1038/nbt1358
Homo sapiens	Insulin receptor-related protein	Kd	81.0	nM	10.1038/nbt.1990
Homo sapiens	Insulin receptor-related protein	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Insulin receptor-related protein	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Interferon-induced, double-stranded RNA-activated protein kinase	IC50	100.0	nM	10.1016/j.bmcl.2011.04.149
Homo sapiens	Interferon-induced, double-stranded RNA-activated protein kinase	Kd	360.0	nM	10.1038/nbt1358
Homo sapiens	Interferon-induced, double-stranded RNA-activated protein kinase	Kd	360.0	nM	10.1038/nbt.1990
Homo sapiens	Interleukin-1 receptor-associated kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Interleukin-1 receptor-associated kinase 1	IC50	16.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Interleukin-1 receptor-associated kinase 1	IC50	59.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Interleukin-1 receptor-associated kinase 1	Inhibition	85.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Interleukin-1 receptor-associated kinase 1	Kd	40.0	nM	10.1038/nbt.1990
Homo sapiens	Interleukin-1 receptor-associated kinase 1	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Interleukin-1 receptor-associated kinase 1	Residual Activity	5.0	%	10.1042/bj20121418
Homo sapiens	Interleukin-1 receptor-associated kinase 3	Kd	13.0	nM	10.1038/nbt1358
Homo sapiens	Interleukin-1 receptor-associated kinase 3	Kd	13.0	nM	10.1038/nbt.1990
Homo sapiens	Interleukin-1 receptor-associated kinase 4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Interleukin-1 receptor-associated kinase 4	IC50	4.21	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Interleukin-1 receptor-associated kinase 4	IC50	4.51	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Interleukin-1 receptor-associated kinase 4	IC50	6.19	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Interleukin-1 receptor-associated kinase 4	IC50	34.0	nM	10.1021/jm800861c
Homo sapiens	Interleukin-1 receptor-associated kinase 4	Kd	1.7	nM	10.1038/nbt.1990
Homo sapiens	Interleukin-1 receptor-associated kinase 4	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Jurkat	Activity	15.87	%	10.1021/acs.jnatprod.0c00261
Homo sapiens	Jurkat	Activity	30.37	%	10.1021/acs.jnatprod.0c00261
Homo sapiens	Jurkat	Activity	53.44	%	10.1021/acs.jnatprod.0c00261
Homo sapiens	Jurkat	Activity	nan	None	10.1021/acs.jnatprod.0c00261
Homo sapiens	Jurkat	Activity	nan	None	10.1021/jm049640t
Homo sapiens	Jurkat	IC50	39.3	nM	10.1016/j.ejmech.2021.113727
Homo sapiens	Jurkat	IC50	71.0	nM	10.1016/j.bmcl.2009.04.039
Homo sapiens	Jurkat	IC50	140.0	nM	10.1021/np400838a
Homo sapiens	Jurkat	IC50	311.0	nM	10.1016/j.bmcl.2009.04.039
Homo sapiens	Jurkat	IC50	3200.0	nM	10.1021/acs.jnatprod.1c01211
Homo sapiens	Jurkat	Selectivity Index	4.0	None	10.1016/j.bmcl.2009.04.039
Homo sapiens	K562	IC50	40.0	nM	10.1021/acsmedchemlett.0c00269
Homo sapiens	K562	IC50	76.8	nM	10.1016/j.ejmech.2020.113003
Homo sapiens	K562	IC50	83.0	nM	10.1016/j.bmcl.2019.04.023
Homo sapiens	K562	IC50	100.0	nM	10.1016/j.ejmech.2021.113727
Homo sapiens	K562	IC50	1700.0	nM	10.1021/acs.jnatprod.8b00103
Homo sapiens	K562	IC50	23100.0	nM	10.1016/j.bmc.2019.02.005
Homo sapiens	K562	IC50	153000.0	nM	10.1016/j.bmc.2015.04.083
Homo sapiens	K562	IC50	nan	None	10.1016/j.bmcl.2012.08.005
Homo sapiens	K562	IC50	nan	None	10.1021/acs.jmedchem.6b00374
Homo sapiens	K562	Inhibition	100.0	%	10.1016/j.ejmech.2013.10.049
Homo sapiens	KB	ED50	0.0024	ug ml-1	10.1021/np50059a012
Homo sapiens	KB 3-1	IC50	200.0	nM	10.1021/acs.jnatprod.7b00236
Homo sapiens	KB-V1	Activity	50.0	%	10.1016/j.ejmech.2017.06.047
Homo sapiens	Kinase suppressor of Ras 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Kinase suppressor of Ras 1	IC50	4590.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Kinase suppressor of Ras 1	IC50	7940.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Kinase suppressor of Ras 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Kinase suppressor of Ras 2	IC50	3980.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Kinase suppressor of Ras 2	IC50	6820.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Kinesin-1 heavy chain/ Tyrosine-protein kinase receptor RET	IC50	1.51	nM	10.1016/j.ejmech.2020.112755
Homo sapiens	KOPN-8	Activity	0.1	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	KOPN-8	Activity	0.2	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	KOPN-8	Activity	0.3	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	KOPN-8	Activity	20.08	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	KOPN-8	Activity	30.37	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	KOPN-8	Activity	45.2	%	10.1016/j.ejmech.2018.12.059
Homo sapiens	KOPN-8	Activity	49.55	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	KOPN-8	Activity	53.2	%	10.1016/j.ejmech.2018.12.059
Homo sapiens	KOPN-8	Activity	74.4	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	KOPN-8	Activity	nan	None	10.1021/acs.jnatprod.8b01087
Homo sapiens	KOPN-8	EC50	710.0	nM	10.1021/acs.jnatprod.8b00884
Homo sapiens	KOPN-8	FC	0.4	None	10.1016/j.ejmech.2018.01.004
Homo sapiens	KOPN-8	FC	0.5	None	10.1016/j.ejmech.2018.01.004
Homo sapiens	KOPN-8	FC	0.6	None	10.1016/j.ejmech.2018.01.004
Homo sapiens	KOPN-8	FC	0.7	None	10.1016/j.ejmech.2018.01.004
Homo sapiens	L02	IC50	9500.0	nM	10.1021/acs.jnatprod.8b00103
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	Activity	2.0	%	10.1016/j.bmcl.2014.08.049
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	Activity	5.0	%	10.1016/j.bmcl.2014.08.049
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	IC50	1.0	nM	10.1016/j.bmcl.2013.04.086
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	IC50	4.85	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	IC50	17.1	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	Kd	0.39	nM	10.1038/nbt.1990
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	Kd	3.1	nM	10.1038/nbt.1990
Homo sapiens	Leukocyte tyrosine kinase receptor	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Leukocyte tyrosine kinase receptor	IC50	3.6	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Leukocyte tyrosine kinase receptor	IC50	19.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Leukocyte tyrosine kinase receptor	IC50	29.2	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Leukocyte tyrosine kinase receptor	Kd	37.0	nM	10.1038/nbt1358
Homo sapiens	Leukocyte tyrosine kinase receptor	Kd	37.0	nM	10.1038/nbt.1990
Homo sapiens	LIM domain kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	LIM domain kinase 1	IC50	2.44	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	LIM domain kinase 1	IC50	2.71	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	LIM domain kinase 1	IC50	48.0	nM	10.1016/j.ejmech.2018.06.016
Homo sapiens	LIM domain kinase 1	Kd	480.0	nM	10.1038/nbt1358
Homo sapiens	LIM domain kinase 1	Kd	480.0	nM	10.1038/nbt.1990
Homo sapiens	LIM domain kinase 1	Kd	690.0	nM	10.1038/nbt1068
Homo sapiens	LIM domain kinase 1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	LIM domain kinase 1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	LIM domain kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	LIM domain kinase 2	IC50	89.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	LIM domain kinase 2	IC50	102.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	LIM domain kinase 2	Kd	9200.0	nM	10.1038/nbt1358
Homo sapiens	LIM domain kinase 2	Kd	9200.0	nM	10.1038/nbt.1990
Homo sapiens	LN-229	IC50	3.0	nM	10.1021/acsmedchemlett.0c00269
Homo sapiens	LN-229	IC50	9.7	nM	10.1016/j.ejmech.2021.113727
Homo sapiens	LoVo	IC50	1.0	nM	10.1016/j.ejmech.2011.11.040
Homo sapiens	LoVo	IC50	1.0	nM	10.1016/s0960-894x(01)00535-2
Homo sapiens	LoVo	NT	nan	None	10.1021/jm0102856
Homo sapiens	LOX IMVI	IC50	7150.0	nM	10.1016/j.ejmech.2021.113277
Homo sapiens	Lysyl-tRNA synthetase	IC50	0.86	nM	10.1021/acs.jnatprod.7b01082
Homo sapiens	Lysyl-tRNA synthetase	IC50	9.0	nM	10.1016/j.bmc.2008.06.017
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	0.31	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	0.46	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	1.11	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	1.54	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	1.92	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	5.94	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	18.03	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	58.47	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	89.91	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	93.41	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Macrophage colony stimulating factor receptor	IC50	1.14	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Macrophage colony stimulating factor receptor	IC50	1.24	nM	10.1016/j.ejmech.2020.112710
Homo sapiens	Macrophage colony stimulating factor receptor	IC50	1.3	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Macrophage colony stimulating factor receptor	IC50	2.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Macrophage colony stimulating factor receptor	IC50	3.13	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Macrophage colony stimulating factor receptor	IC50	970.0	nM	10.1016/j.bmcl.2017.04.014
Homo sapiens	Macrophage colony stimulating factor receptor	Kd	12.0	nM	10.1038/nbt1358
Homo sapiens	Macrophage colony stimulating factor receptor	Kd	12.0	nM	10.1038/nbt.1990
Homo sapiens	Macrophage colony stimulating factor receptor	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Macrophage colony stimulating factor receptor	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Macrophage-stimulating protein receptor	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Macrophage-stimulating protein receptor	IC50	77.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Macrophage-stimulating protein receptor	IC50	102.7	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Macrophage-stimulating protein receptor	IC50	149.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Macrophage-stimulating protein receptor	IC50	326.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Macrophage-stimulating protein receptor	IC50	442.5	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Macrophage-stimulating protein receptor	Kd	400.0	nM	10.1038/nbt.1990
Homo sapiens	Macrophage-stimulating protein receptor	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Macrophage-stimulating protein receptor	Residual Activity	13.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase-activated protein kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase-activated protein kinase 2	IC50	36.25	nM	10.1016/j.ejmech.2010.04.026
Homo sapiens	MAP kinase-activated protein kinase 2	IC50	65.9	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	MAP kinase-activated protein kinase 2	IC50	110.0	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	MAP kinase-activated protein kinase 2	IC50	128.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase-activated protein kinase 2	IC50	150.0	nM	10.1021/np900246t
Homo sapiens	MAP kinase-activated protein kinase 2	IC50	400.0	nM	10.1021/jm300411k
Homo sapiens	MAP kinase-activated protein kinase 2	IC50	660.0	nM	10.1016/j.bmcl.2009.10.102
Homo sapiens	MAP kinase-activated protein kinase 2	IC50	700.0	nM	10.1016/j.bmcl.2009.10.102
Homo sapiens	MAP kinase-activated protein kinase 2	IC50	1700.0	nM	10.1016/j.bmcl.2009.10.102
Homo sapiens	MAP kinase-activated protein kinase 2	IC50	3400.0	nM	10.1016/j.bmcl.2009.10.102
Homo sapiens	MAP kinase-activated protein kinase 2	Inhibition	100.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	MAP kinase-activated protein kinase 2	Kd	880.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase-activated protein kinase 2	Kd	880.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase-activated protein kinase 2	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase-activated protein kinase 2	Residual Activity	14.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase-activated protein kinase 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase-activated protein kinase 3	IC50	2000.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	MAP kinase-activated protein kinase 3	IC50	3550.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase-activated protein kinase 3	Residual Activity	46.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase-activated protein kinase 3	Residual Activity	101.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase-activated protein kinase 5	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase-activated protein kinase 5	IC50	129.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	MAP kinase-activated protein kinase 5	IC50	295.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase-activated protein kinase 5	Kd	270.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase-activated protein kinase 5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase-activated protein kinase 5	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase-activated protein kinase 5	Residual Activity	29.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase ERK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase ERK1	IC50	1310.0	nM	10.1016/j.bmc.2009.05.031
Homo sapiens	MAP kinase ERK1	IC50	1310.0	nM	10.1016/j.ejmech.2013.07.046
Homo sapiens	MAP kinase ERK1	IC50	1400.0	nM	10.1016/j.ejmech.2015.08.027
Homo sapiens	MAP kinase ERK1	IC50	4130.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	MAP kinase ERK1	IC50	4900.0	nM	10.1016/j.bmcl.2006.05.092
Homo sapiens	MAP kinase ERK1	IC50	5089.0	nM	10.1016/j.ejmech.2010.04.026
Homo sapiens	MAP kinase ERK1	IC50	6540.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	MAP kinase ERK1	IC50	7791.0	nM	10.1021/jm800861c
Homo sapiens	MAP kinase ERK1	IC50	9582.0	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	MAP kinase ERK1	IC50	27370.0	nM	10.1021/jm801317h
Homo sapiens	MAP kinase ERK1	IC50	30100.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase ERK1	Inhibition	99.37	%	10.1016/j.bmc.2012.04.006
Homo sapiens	MAP kinase ERK1	Kd	8400.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase ERK1	Kd	8400.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase ERK1	Residual Activity	13.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase ERK1	Residual Activity	66.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase ERK2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase ERK2	Delta TM	1.22	C	None
Homo sapiens	MAP kinase ERK2	IC50	1.0	nM	10.1021/jm020143r
Homo sapiens	MAP kinase ERK2	IC50	2.5	nM	10.1021/jm0102856
Homo sapiens	MAP kinase ERK2	IC50	370.0	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	MAP kinase ERK2	IC50	370.0	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	MAP kinase ERK2	IC50	659.1	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	MAP kinase ERK2	IC50	1380.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	MAP kinase ERK2	IC50	3948.0	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	MAP kinase ERK2	IC50	4491.0	nM	10.1021/jm800861c
Homo sapiens	MAP kinase ERK2	IC50	7180.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	MAP kinase ERK2	IC50	8451.0	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	MAP kinase ERK2	IC50	34000.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase ERK2	Inhibition	100.3	%	10.1016/j.bmc.2012.04.006
Homo sapiens	MAP kinase ERK2	Inhibition	100.31	%	10.1016/j.bmc.2013.07.026
Homo sapiens	MAP kinase ERK2	Kd	7300.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase ERK2	Kd	7300.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase ERK2	Residual Activity	37.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase ERK2	Residual Activity	82.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	IC50	44.17	nM	10.1021/acsmedchemlett.2c00442
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	IC50	52.7	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	IC50	53.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	Kd	170.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	Kd	170.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38	IC50	1000.0	nM	10.1021/jm020143r
Homo sapiens	MAP kinase p38 alpha	Delta Tm	0.4	degrees C	10.1016/j.ejmech.2020.112721
Homo sapiens	MAP kinase p38 alpha	IC50	10.5	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	MAP kinase p38 alpha	IC50	6600.0	nM	10.1039/C6MD00351F
Homo sapiens	MAP kinase p38 alpha	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase p38 alpha	IC50	nan	None	10.1016/j.ejmech.2021.113277
Homo sapiens	MAP kinase p38 alpha	IC50	nan	None	10.1021/jm800861c
Homo sapiens	MAP kinase p38 alpha	IC50	nan	None	10.1021/jm901297e
Homo sapiens	MAP kinase p38 alpha	Inhibition	11.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	MAP kinase p38 alpha	Inhibition	nan	%	10.1016/j.bmc.2012.04.006
Homo sapiens	MAP kinase p38 alpha	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase p38 alpha	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 alpha	Kd	nan	None	10.1038/nbt1068
Homo sapiens	MAP kinase p38 alpha	Kd	nan	None	10.1038/nchembio.162
Homo sapiens	MAP kinase p38 alpha	Residual Activity	79.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase p38 alpha	Residual Activity	81.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase p38 beta	Delta Tm	0.4	degrees C	10.1016/j.ejmech.2020.112721
Homo sapiens	MAP kinase p38 beta	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase p38 beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase p38 beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 beta	Kd	nan	None	10.1038/nbt1068
Homo sapiens	MAP kinase p38 beta	Residual Activity	89.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase p38 beta	Residual Activity	97.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase p38 delta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase p38 delta	IC50	81.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	MAP kinase p38 delta	IC50	160.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase p38 delta	Kd	240.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 delta	Residual Activity	6.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase p38 delta	Residual Activity	25.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase p38 gamma	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase p38 gamma	IC50	78.7	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	MAP kinase p38 gamma	IC50	275.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase p38 gamma	Kd	42.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase p38 gamma	Kd	42.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 gamma	Kd	92.0	nM	10.1038/nbt1068
Homo sapiens	MAP kinase p38 gamma	Residual Activity	8.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase p38 gamma	Residual Activity	35.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase signal-integrating kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase signal-integrating kinase 2	IC50	8.85	nM	10.1021/acsmedchemlett.2c00442
Homo sapiens	MAP kinase signal-integrating kinase 2	IC50	19.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	MAP kinase signal-integrating kinase 2	IC50	20.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP kinase signal-integrating kinase 2	IC50	27.12	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	MAP kinase signal-integrating kinase 2	Kd	17.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase signal-integrating kinase 2	Kd	17.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase signal-integrating kinase 2	Kd	22.0	nM	10.1038/nbt1068
Homo sapiens	MAP kinase signal-integrating kinase 2	Residual Activity	4.0	%	10.1042/bj20121418
Homo sapiens	MAP kinase signal-integrating kinase 2	Residual Activity	8.0	%	10.1042/bj20121418
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	IC50	0.133	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	IC50	0.148	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Kd	0.1	nM	10.1038/nbt1068
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Kd	0.7	nM	10.1038/nbt1358
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Kd	0.7	nM	10.1038/nbt.1990
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	IC50	0.114	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	IC50	0.131	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	Kd	0.5	nM	10.1021/acsmedchemlett.3c00127
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	Kd	5.4	nM	10.1038/nbt1358
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	Kd	5.4	nM	10.1038/nbt.1990
Homo sapiens	Maternal embryonic leucine zipper kinase	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Maternal embryonic leucine zipper kinase	IC50	0.542	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Maternal embryonic leucine zipper kinase	IC50	0.687	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Maternal embryonic leucine zipper kinase	Kd	33.0	nM	10.1038/nbt1358
Homo sapiens	Maternal embryonic leucine zipper kinase	Kd	33.0	nM	10.1038/nbt.1990
Homo sapiens	Maternal embryonic leucine zipper kinase	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	Maternal embryonic leucine zipper kinase	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	MCF-10A	Activity	1.22	%	10.1016/j.ejmech.2018.11.034
Homo sapiens	MCF-10A	Activity	2.18	%	10.1016/j.ejmech.2018.11.034
Homo sapiens	MCF-10A	Activity	9.96	%	10.1016/j.ejmech.2018.11.034
Homo sapiens	MCF-10A	Activity	85.6	%	10.1016/j.ejmech.2018.11.034
Homo sapiens	MCF-10A	Activity	nan	None	10.1016/j.ejmech.2018.11.034
Homo sapiens	MCF-10A	IC50	nan	None	10.1021/acs.jmedchem.1c01411
Homo sapiens	MCF7	Activity	0.6	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MCF7	Activity	1.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MCF7	Activity	2.33	%	10.1016/j.bmc.2020.115328
Homo sapiens	MCF7	Activity	3.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MCF7	Activity	3.4	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MCF7	Activity	3.5	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MCF7	Activity	7.4	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MCF7	Activity	7.9	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MCF7	Activity	8.16	%	10.1016/j.bmc.2020.115328
Homo sapiens	MCF7	Activity	8.41	ng/ml	10.1016/j.bmc.2020.115328
Homo sapiens	MCF7	Activity	9.6	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MCF7	Activity	11.27	%	10.1016/j.bmc.2020.115328
Homo sapiens	MCF7	Activity	24.9	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MCF7	Activity	62.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MCF7	Activity	83.6	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MCF7	Activity	93.0	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MCF7	Activity	nan	None	10.1016/j.ejmech.2010.12.008
Homo sapiens	MCF7	EC50	100.0	nM	10.1016/j.ejmech.2017.11.046
Homo sapiens	MCF7	EC50	100.0	nM	10.1016/j.ejmech.2019.02.057
Homo sapiens	MCF7	EC50	100.0	nM	10.1016/j.ejmech.2020.112920
Homo sapiens	MCF7	GI50	11000.0	nM	10.1021/np200041v
Homo sapiens	MCF7	IC50	13.0	nM	10.1039/C2MD20098H
Homo sapiens	MCF7	IC50	20.0	nM	10.1016/j.bmcl.2020.127109
Homo sapiens	MCF7	IC50	50.0	nM	10.1021/np100727h
Homo sapiens	MCF7	IC50	50.0	nM	10.1021/np200035m
Homo sapiens	MCF7	IC50	64.0	nM	10.1016/j.bmcl.2012.08.005
Homo sapiens	MCF7	IC50	100.0	nM	10.1016/j.ejmech.2020.112425
Homo sapiens	MCF7	IC50	180.0	nM	10.1016/j.bmc.2012.03.061
Homo sapiens	MCF7	IC50	400.0	nM	10.1016/j.ejmech.2013.11.025
Homo sapiens	MCF7	IC50	520.0	nM	10.1021/np400838a
Homo sapiens	MCF7	IC50	1800.0	nM	10.1021/acs.jnatprod.7b00236
Homo sapiens	MCF7	IC50	3070.0	nM	10.1016/j.bmc.2012.03.040
Homo sapiens	MCF7	IC50	3390.0	nM	10.1016/j.ejmech.2019.112019
Homo sapiens	MCF7	IC50	3670.0	nM	10.1016/j.ejmech.2020.112745
Homo sapiens	MCF7	IC50	3670.0	nM	10.1016/j.ejmech.2021.113283
Homo sapiens	MCF7	IC50	4100.0	nM	10.1016/j.ejmech.2021.113800
Homo sapiens	MCF7	IC50	4100.0	nM	10.1016/j.ejmech.2021.114008
Homo sapiens	MCF7	IC50	6080.0	nM	10.1016/j.ejmech.2021.113964
Homo sapiens	MCF7	IC50	6300.0	nM	10.1021/acs.jnatprod.1c01211
Homo sapiens	MCF7	IC50	7250.0	nM	10.1039/d2md00076h
Homo sapiens	MCF7	IC50	7330.0	nM	10.1016/j.ejmech.2020.112745
Homo sapiens	MCF7	IC50	8810.0	nM	10.1016/j.bmc.2020.115328
Homo sapiens	MCF7	IC50	9200.0	nM	10.1016/j.ejmech.2019.112019
Homo sapiens	MCF7	IC50	16060.0	nM	10.1007/s00044-012-0306-5
Homo sapiens	MDA-MB-231	Activity	0.5	%	10.1016/j.ejmech.2015.07.034
Homo sapiens	MDA-MB-231	Activity	3.9	%	10.1016/j.ejmech.2019.01.052
Homo sapiens	MDA-MB-231	Activity	6.8	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	MDA-MB-231	Activity	10.9	%	10.1021/acs.jnatprod.8b00540
Homo sapiens	MDA-MB-231	Activity	18.8	%	10.1016/j.ejmech.2015.07.034
Homo sapiens	MDA-MB-231	Activity	23.28	%	10.1016/j.ejmech.2015.07.034
Homo sapiens	MDA-MB-231	Activity	25.0	%	10.1016/j.ejmech.2015.07.034
Homo sapiens	MDA-MB-231	Activity	33.22	%	10.1016/j.ejmech.2015.07.034
Homo sapiens	MDA-MB-231	Activity	42.21	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	MDA-MB-231	Activity	43.5	%	10.1016/j.ejmech.2015.07.034
Homo sapiens	MDA-MB-231	Activity	50.99	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	MDA-MB-231	Activity	55.7	%	10.1016/j.ejmech.2015.07.034
Homo sapiens	MDA-MB-231	Activity	nan	None	10.1016/j.ejmech.2015.07.034
Homo sapiens	MDA-MB-231	Activity	nan	None	10.1021/acs.jmedchem.8b00753
Homo sapiens	MDA-MB-231	GI50	7.1	nM	10.1021/np700748h
Homo sapiens	MDA-MB-231	IC50	0.8581	nM	10.1016/j.ejmech.2021.113880
Homo sapiens	MDA-MB-231	IC50	2.5	nM	10.1021/acsmedchemlett.0c00420
Homo sapiens	MDA-MB-231	IC50	10.0	nM	10.1016/j.ejmech.2020.112948
Homo sapiens	MDA-MB-231	IC50	240.0	nM	10.1016/j.bmc.2017.06.036
Homo sapiens	MDA-MB-231	IC50	4250.0	nM	10.1016/j.ejmech.2020.112112
Homo sapiens	MDA-MB-231	IC50	4310.0	nM	10.1016/j.ejmech.2020.112745
Homo sapiens	MDA-MB-231	IC50	6750.0	nM	10.1016/j.ejmech.2020.112745
Homo sapiens	MDA-MB-231	IC50	6750.0	nM	10.1016/j.ejmech.2021.113283
Homo sapiens	MDA-MB-231	Inhibition	93.0	%	10.1016/j.ejmech.2013.10.049
Homo sapiens	MDA-MB-453	IC50	23.51	nM	10.1016/j.ejmech.2021.113880
Homo sapiens	MDA-MB-468	IC50	150.0	nM	10.1016/j.bmc.2017.06.036
Homo sapiens	MDA-MB-468	IC50	4370.0	nM	10.1016/j.ejmech.2019.112019
Homo sapiens	MDA-MB-468	IC50	6460.0	nM	10.1016/j.ejmech.2019.112019
Homo sapiens	Menin/Histone-lysine N-methyltransferase MLL	Potency	3162.3	nM	None
Homo sapiens	MFE-280	Activity	0.9	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-280	Activity	1.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-280	Activity	3.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-280	Activity	17.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-280	Activity	18.9	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-280	Activity	23.2	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-280	Activity	24.7	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-280	Activity	25.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-280	Activity	30.5	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-280	Activity	47.5	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-280	Activity	51.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-280	Activity	57.0	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-296	Activity	2.4	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-296	Activity	4.4	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-296	Activity	6.6	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-296	Activity	6.8	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-296	Activity	7.5	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-296	Activity	11.6	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-296	Activity	15.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-296	Activity	20.2	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-296	Activity	24.4	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-296	Activity	57.2	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-296	Activity	60.3	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MFE-296	Activity	83.6	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	MG-63	Activity	nan	None	10.1016/j.ejmech.2018.08.044
Homo sapiens	MIA PaCa-2	IC50	370.0	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	MIA PaCa-2	IC50	370.0	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Microtubule-associated protein tau	Potency	1412.5	nM	None
Homo sapiens	Microtubule-associated protein tau	Potency	3162.3	nM	None
Homo sapiens	Microtubule-associated protein tau	Potency	4466.8	nM	None
Homo sapiens	Microtubule-associated protein tau	Potency	14125.4	nM	None
Homo sapiens	Microtubule-associated serine/threonine-protein kinase 1	Kd	150.0	nM	10.1038/nbt.1990
Homo sapiens	Misshapen-like kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Misshapen-like kinase 1	IC50	0.235	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Misshapen-like kinase 1	IC50	0.451	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Misshapen-like kinase 1	IC50	0.47	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Misshapen-like kinase 1	IC50	0.49	nM	10.1021/jm800861c
Homo sapiens	Misshapen-like kinase 1	Inhibition	98.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Misshapen-like kinase 1	Kd	1.0	nM	10.1038/nbt.1990
Homo sapiens	Misshapen-like kinase 1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Misshapen-like kinase 1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Mitogen-activated protein kinase 15	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase 15	IC50	7.3	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Mitogen-activated protein kinase 15	IC50	8.01	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase 15	IC50	9.1	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase 15	Kd	5.5	nM	10.1021/acsmedchemlett.3c00127
Homo sapiens	Mitogen-activated protein kinase 15	Kd	35.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase 15	Kd	35.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase 6	Kd	3100.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase 6	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase 7	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase 7	IC50	121.6	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Mitogen-activated protein kinase 7	IC50	5520.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase 7	IC50	6368.0	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Mitogen-activated protein kinase 7	IC50	11800.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase 7	Kd	1600.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase 7	Kd	1600.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 1	IC50	391.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase 1	IC50	485.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 1	Kd	350.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 10	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 10	IC50	2.69	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 10	IC50	2.84	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase 10	IC50	580.0	nM	10.1016/j.ejmech.2021.113299
Homo sapiens	Mitogen-activated protein kinase kinase kinase 10	Kd	52.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 10	Kd	52.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	IC50	4.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	IC50	5.06	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	IC50	39.0	nM	10.1016/j.ejmech.2021.113299
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	Kd	20.0	nM	10.1021/jm401094t
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	Kd	20.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	Kd	20.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 12	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 12	IC50	18.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase 12	IC50	180.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 12	Kd	1500.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 13	Kd	210.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 14	IC50	2300.0	nM	10.1016/j.bmcl.2010.06.027
Homo sapiens	Mitogen-activated protein kinase kinase kinase 15	Kd	2.5	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 2	IC50	23.5	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase 2	IC50	43.5	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 2	Kd	2.4	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 3	IC50	7.55	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase 3	IC50	10.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 3	Kd	2800.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 4	Kd	1200.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 4	Kd	1200.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 4	Kd	2200.0	nM	10.1038/nbt1068
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	IC50	0.69	nM	10.1021/acs.jnatprod.7b01058
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	IC50	17.6	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	IC50	19.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	IC50	37.0	nM	10.1016/j.bmcl.2008.05.040
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	IC50	1000.0	nM	10.1016/j.bmcl.2008.05.040
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	110.0	nM	10.1016/j.bmcl.2008.05.040
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	110.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	120.0	nM	10.1038/nbt1068
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Mitogen-activated protein kinase kinase kinase 6	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 6	IC50	90.8	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase 6	IC50	475.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 6	Kd	260.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7	IC50	35.0	nM	10.1021/jm800861c
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7	IC50	43.11	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7	IC50	66.2	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7	IC50	99.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7	Inhibition	81.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7	Kd	67.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7	Residual Activity	14.0	%	10.1042/bj20121418
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7-interacting protein 1	IC50	35.0	nM	10.1021/jm800861c
Homo sapiens	Mitogen-activated protein kinase kinase kinase 8	Activity	nan	None	10.1016/j.bmcl.2011.07.069
Homo sapiens	Mitogen-activated protein kinase kinase kinase 8	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	IC50	0.544	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	IC50	1.52	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	IC50	11.0	nM	10.1016/j.ejmech.2021.113299
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	Kd	10.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	Kd	10.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 1	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 1	Kd	4.3	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 1	Kd	4.3	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 2	Kd	8.8	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 2	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 3	IC50	0.0825	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 3	IC50	0.0833	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 3	Kd	8.2	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 3	Kd	8.2	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	IC50	0.348	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	IC50	0.57	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	Kd	24.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	Kd	24.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	IC50	0.177	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	IC50	0.309	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	18.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	18.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	26.0	nM	10.1038/nbt1068
Homo sapiens	Mitogen-activated protein kinase kinase kinase MLK4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mitogen-activated protein kinase kinase kinase MLK4	IC50	765.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Mitogen-activated protein kinase kinase kinase MLK4	IC50	1470.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mixed lineage kinase 7	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Mixed lineage kinase 7	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mixed lineage kinase 7	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MM1.S	IC50	44.2	nM	10.1016/j.ejmech.2020.113003
Homo sapiens	Monocyte	Activity	nan	None	10.1016/j.bmc.2014.06.032
Homo sapiens	Multidrug resistance-associated protein 4	IC50	37900.0	nM	10.1093/toxsci/kft176
Homo sapiens	Muscle, skeletal receptor tyrosine protein kinase	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Muscle, skeletal receptor tyrosine protein kinase	IC50	3.8	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Muscle, skeletal receptor tyrosine protein kinase	IC50	54.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Muscle, skeletal receptor tyrosine protein kinase	IC50	290.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Muscle, skeletal receptor tyrosine protein kinase	Kd	86.0	nM	10.1038/nbt1358
Homo sapiens	Muscle, skeletal receptor tyrosine protein kinase	Kd	86.0	nM	10.1038/nbt.1990
Homo sapiens	Muscle, skeletal receptor tyrosine protein kinase	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	MV4-11	EC50	6.31	nM	10.1021/acs.jmedchem.1c01532
Homo sapiens	MV4-11	IC50	50.0	nM	10.1016/j.ejmech.2021.113727
Homo sapiens	MV4-11	IC50	nan	None	10.1021/acs.jmedchem.6b00374
Homo sapiens	Myelin transcription factor 1	Activity	5.0	%	10.1016/j.ejmech.2012.06.007
Homo sapiens	Myosin IIIA	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Myosin IIIA	IC50	40.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Myosin IIIA	IC50	44.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Myosin IIIA	Kd	500.0	nM	10.1038/nbt1358
Homo sapiens	Myosin IIIA	Kd	500.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin-IIIB	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Myosin-IIIB	IC50	5.19	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Myosin-IIIB	IC50	6.4	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Myosin-IIIB	Kd	300.0	nM	10.1038/nbt1358
Homo sapiens	Myosin-IIIB	Kd	300.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin light chain kinase	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Myosin light chain kinase	IC50	129.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Myosin light chain kinase	IC50	188.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Myosin light chain kinase	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	myosin light chain kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	myosin light chain kinase 2	IC50	13.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	myosin light chain kinase 2	IC50	15.5	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	myosin light chain kinase 2	Kd	61.0	nM	10.1038/nbt1358
Homo sapiens	myosin light chain kinase 2	Kd	61.0	nM	10.1038/nbt.1990
Homo sapiens	myosin light chain kinase 2	Kd	110.0	nM	10.1038/nbt1068
Homo sapiens	Myosin light chain kinase family member 4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Myosin light chain kinase family member 4	IC50	52.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Myosin light chain kinase family member 4	IC50	54.5	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Myosin light chain kinase family member 4	Kd	470.0	nM	10.1038/nbt1358
Homo sapiens	Myosin light chain kinase family member 4	Kd	470.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin light chain kinase, smooth muscle	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Myosin light chain kinase, smooth muscle	IC50	10.0	nM	10.1016/0960-894X(94)00458-R
Homo sapiens	Myosin light chain kinase, smooth muscle	IC50	40.0	nM	10.1021/jm00053a003
Homo sapiens	Myosin light chain kinase, smooth muscle	IC50	43.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Myosin light chain kinase, smooth muscle	IC50	51.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Myosin light chain kinase, smooth muscle	Kd	15.0	nM	10.1038/nbt1358
Homo sapiens	Myosin light chain kinase, smooth muscle	Kd	15.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin light chain kinase, smooth muscle	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Myosin light chain kinase, smooth muscle	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Myotonin-protein kinase	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Myotonin-protein kinase	IC50	105.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Myotonin-protein kinase	IC50	242.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Myotonin-protein kinase	Kd	3.5	nM	10.1038/nbt1358
Homo sapiens	Myotonin-protein kinase	Kd	3.5	nM	10.1038/nbt.1990
Homo sapiens	Myotonin-protein kinase	Residual Activity	9.0	%	10.1042/bj20121418
Homo sapiens	Myotonin-protein kinase	Residual Activity	16.0	%	10.1042/bj20121418
Homo sapiens	NAD-dependent deacetylase sirtuin 1	IC50	nan	None	10.1021/jm060118b
Homo sapiens	NAD-dependent deacetylase sirtuin 2	Activity	nan	None	10.1021/jm060118b
Homo sapiens	NADPH oxidase 4	IC50	70.77	nM	10.1016/j.ejmech.2021.113475
Homo sapiens	NALM-6	Activity	0.0	%	10.1016/j.ejmech.2016.02.034
Homo sapiens	NALM-6	Activity	18.8	%	10.1016/j.ejmech.2016.02.034
Homo sapiens	NALM-6	Activity	25.0	%	10.1016/j.ejmech.2016.02.034
Homo sapiens	NALM-6	Activity	49.0	%	10.1016/j.ejmech.2016.02.034
Homo sapiens	NALM-6	Activity	nan	None	10.1016/j.ejmech.2016.02.034
Homo sapiens	NALM-6	EC50	1400.0	nM	10.1021/acs.jnatprod.8b00884
Homo sapiens	NCI-H460	GI50	3600.0	nM	10.1021/np200041v
Homo sapiens	NCI-H460	IC50	24.0	nM	10.1016/j.bmcl.2019.04.023
Homo sapiens	NCI-H460	IC50	59.7	nM	10.1016/j.ejmech.2020.113003
Homo sapiens	NCI-H460	IC50	60.0	nM	10.1021/acsmedchemlett.0c00269
Homo sapiens	NCI-H460	IC50	100.0	nM	10.1016/j.ejmech.2021.113727
Homo sapiens	NCI-H460	IC50	11500.0	nM	10.1016/j.bmc.2019.02.005
Homo sapiens	NCI-H460	IC50	nan	nM	10.1016/s0960-894x(03)00461-x
Homo sapiens	NCI-H69	Inhibition	95.4	%	10.1016/j.ejmech.2013.10.049
Homo sapiens	NCI-N87	Inhibition	95.1	%	10.1016/j.ejmech.2013.10.049
Homo sapiens	Nerve growth factor receptor Trk-A	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Nerve growth factor receptor Trk-A	Activity	nan	None	10.1039/C2MD00271J
Homo sapiens	Nerve growth factor receptor Trk-A	IC50	0.5	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Nerve growth factor receptor Trk-A	IC50	1.29	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Nerve growth factor receptor Trk-A	IC50	1.36	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Nerve growth factor receptor Trk-A	IC50	1.59	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Nerve growth factor receptor Trk-A	IC50	1.7	nM	10.1021/jm800861c
Homo sapiens	Nerve growth factor receptor Trk-A	IC50	3.1	nM	10.1039/C2MD00271J
Homo sapiens	Nerve growth factor receptor Trk-A	IC50	5.78	nM	10.1016/j.bmc.2021.116596
Homo sapiens	Nerve growth factor receptor Trk-A	IC50	8.3	nM	10.1039/C2MD00271J
Homo sapiens	Nerve growth factor receptor Trk-A	IC50	1670.0	nM	10.1016/j.ejmech.2020.112756
Homo sapiens	Nerve growth factor receptor Trk-A	IC50	1000000.0	nM	10.1016/j.bmc.2018.10.004
Homo sapiens	Nerve growth factor receptor Trk-A	Inhibition	94.0	%	10.1021/jm070342g
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	2.0	nM	10.1038/nbt1068
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	4.0	nM	10.1038/nbt1358
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	4.0	nM	10.1038/nbt.1990
Homo sapiens	Nerve growth factor receptor Trk-A	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	IC50	0.0636	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	IC50	0.093	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	IC50	0.96	nM	10.1039/C2MD00271J
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	IC50	1.0	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	IC50	4.5	nM	10.1039/C2MD00271J
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	Kd	3.8	nM	10.1038/nbt1358
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	Kd	3.8	nM	10.1038/nbt.1990
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	Residual Activity	-12.0	%	10.1042/bj20121418
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	Residual Activity	29.0	%	10.1042/bj20121418
Homo sapiens	Non-receptor tyrosine-protein kinase TNK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Non-receptor tyrosine-protein kinase TNK1	IC50	0.584	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Non-receptor tyrosine-protein kinase TNK1	IC50	1.84	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Non-receptor tyrosine-protein kinase TNK1	Kd	2.5	nM	10.1038/nbt1358
Homo sapiens	Non-receptor tyrosine-protein kinase TNK1	Kd	2.5	nM	10.1038/nbt.1990
Homo sapiens	NT-3 growth factor receptor	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	NT-3 growth factor receptor	IC50	0.123	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	NT-3 growth factor receptor	IC50	0.22	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	NT-3 growth factor receptor	Kd	17.0	nM	10.1038/nbt1358
Homo sapiens	NT-3 growth factor receptor	Kd	17.0	nM	10.1038/nbt.1990
Homo sapiens	NUAK family SNF1-like kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	NUAK family SNF1-like kinase 1	IC50	1.31	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	NUAK family SNF1-like kinase 1	IC50	1.35	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	NUAK family SNF1-like kinase 1	IC50	1.41	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	NUAK family SNF1-like kinase 1	IC50	8.0	nM	10.1021/np4005745
Homo sapiens	NUAK family SNF1-like kinase 1	Kd	4.4	nM	10.1038/nbt1358
Homo sapiens	NUAK family SNF1-like kinase 1	Kd	4.4	nM	10.1038/nbt.1990
Homo sapiens	NUAK family SNF1-like kinase 1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	NUAK family SNF1-like kinase 1	Residual Activity	8.0	%	10.1042/bj20121418
Homo sapiens	NUAK family SNF1-like kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	NUAK family SNF1-like kinase 2	IC50	1.67	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	NUAK family SNF1-like kinase 2	IC50	1.9	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	NUAK family SNF1-like kinase 2	Kd	0.086	nM	10.1038/nbt1358
Homo sapiens	NUAK family SNF1-like kinase 2	Kd	0.086	nM	10.1038/nbt.1990
Homo sapiens	PANC-1	IC50	20.0	nM	10.1016/j.bmcl.2020.127109
Homo sapiens	PAS domain-containing serine/threonine-protein kinase	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	PAS domain-containing serine/threonine-protein kinase	IC50	5.54	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	PAS domain-containing serine/threonine-protein kinase	IC50	15.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	PAS domain-containing serine/threonine-protein kinase	Residual Activity	-3.0	%	10.1042/bj20121418
Homo sapiens	PAS domain-containing serine/threonine-protein kinase	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	PBMC	IC50	16.0	nM	10.1016/j.bmc.2008.06.017
Homo sapiens	PBMC	IC50	16.0	nM	10.1016/j.bmc.2008.09.015
Homo sapiens	PC-3	Activity	0.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	PC-3	Activity	0.2	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	PC-3	Activity	0.7	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	PC-3	Activity	1.0	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	PC-3	Activity	1.2	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	PC-3	Activity	1.3	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	PC-3	Activity	4.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	6.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	8.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	9.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	10.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	24.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	31.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	46.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	47.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	60.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	68.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	84.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	87.0	%	10.1016/j.ejmech.2017.03.067
Homo sapiens	PC-3	Activity	97.3	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	PC-3	Activity	98.0	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	PC-3	Activity	98.6	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	PC-3	Activity	nan	None	10.1016/j.ejmech.2018.08.044
Homo sapiens	PC-3	IC50	17.0	nM	10.1021/acs.jnatprod.7b01055
Homo sapiens	PC-3	IC50	39.0	nM	10.1021/acs.jnatprod.7b01058
Homo sapiens	PC-3	IC50	4910.0	nM	10.1021/acs.jmedchem.9b01669
Homo sapiens	PC-3	IC50	5920.0	nM	10.1021/acs.jmedchem.9b01669
Homo sapiens	PC-3	Inhibition	97.1	%	10.1016/j.ejmech.2013.10.049
Homo sapiens	PDZ-binding kinase	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	PDZ-binding kinase	IC50	54.3	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	PDZ-binding kinase	IC50	83.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Peregrin	Delta TM	-0.73	C	None
Homo sapiens	Peripheral plasma membrane protein CASK	deltaTm	4.5	K	10.1021/acs.jmedchem.1c00845
Homo sapiens	Peripheral plasma membrane protein CASK	Kd	19.0	nM	10.1038/nbt.1990
Homo sapiens	P-glycoprotein 1	Activity	140.0	%	10.1038/bjc.1996.205
Homo sapiens	Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing beta polypeptide	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing subunit gamma	Kd	430.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha	Kd	43.0	nM	10.1038/nbt1358
Homo sapiens	Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha	Kd	43.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-4-phosphate 5-kinase type-1 gamma	Kd	2700.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 beta	Kd	77.0	nM	10.1038/nbt1358
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 beta	Kd	77.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 gamma	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphorylase kinase	IC50	0.5	nM	10.1021/jm00079a024
Homo sapiens	Phosphorylase kinase gamma subunit 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Phosphorylase kinase gamma subunit 1	IC50	1.92	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Phosphorylase kinase gamma subunit 1	IC50	2.58	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Phosphorylase kinase gamma subunit 1	Kd	0.5	nM	10.1038/nbt1068
Homo sapiens	Phosphorylase kinase gamma subunit 1	Kd	0.65	nM	10.1038/nbt1358
Homo sapiens	Phosphorylase kinase gamma subunit 1	Kd	0.65	nM	10.1038/nbt.1990
Homo sapiens	Phosphorylase kinase gamma subunit 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Phosphorylase kinase gamma subunit 2	IC50	0.1	nM	10.1021/jm800861c
Homo sapiens	Phosphorylase kinase gamma subunit 2	IC50	0.336	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Phosphorylase kinase gamma subunit 2	IC50	0.49	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Phosphorylase kinase gamma subunit 2	IC50	0.62	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	0.14	nM	10.1038/nbt1358
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	0.14	nM	10.1038/nbt.1990
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	1.0	nM	10.1038/nbt1068
Homo sapiens	Phosphorylase kinase gamma subunit 2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Phosphorylase kinase gamma subunit 2	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	PI3-kinase p110-alpha subunit	IC50	nan	None	10.1016/j.bmc.2017.02.030
Homo sapiens	PI3-kinase p110-alpha subunit	Inhibition	97.0	%	10.1016/j.bmc.2011.06.022
Homo sapiens	PI3-kinase p110-alpha subunit	Kd	400.0	nM	10.1038/nbt.1990
Homo sapiens	PI3-kinase p110-alpha subunit	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	PI3-kinase p110-alpha subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PI3-kinase p110-beta subunit	IC50	nan	None	10.1016/j.bmc.2017.02.030
Homo sapiens	PI3-kinase p110-beta subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PI3-kinase p110-delta subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PI3-kinase p110-gamma subunit	Kd	1800.0	nM	10.1038/nbt.1990
Homo sapiens	PI4-kinase beta subunit	Kd	460.0	nM	10.1038/nbt.1990
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Platelet-derived growth factor receptor	IC50	2.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Platelet-derived growth factor receptor alpha	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Platelet-derived growth factor receptor alpha	IC50	0.1	nM	10.1021/jm800861c
Homo sapiens	Platelet-derived growth factor receptor alpha	IC50	0.418	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Platelet-derived growth factor receptor alpha	IC50	0.43	nM	10.1016/j.bmc.2017.04.003
Homo sapiens	Platelet-derived growth factor receptor alpha	IC50	0.45	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Platelet-derived growth factor receptor alpha	IC50	0.58	nM	10.1016/j.ejmech.2021.113327
Homo sapiens	Platelet-derived growth factor receptor alpha	IC50	0.6	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Platelet-derived growth factor receptor alpha	IC50	0.793	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Platelet-derived growth factor receptor alpha	Inhibition	88.4	%	10.1021/jm070342g
Homo sapiens	Platelet-derived growth factor receptor alpha	Inhibition	92.6	%	10.1016/j.bmc.2011.06.022
Homo sapiens	Platelet-derived growth factor receptor alpha	Inhibition	97.5	%	10.1016/j.bmc.2011.06.022
Homo sapiens	Platelet-derived growth factor receptor alpha	Kd	10.0	nM	10.1038/nbt1358
Homo sapiens	Platelet-derived growth factor receptor alpha	Kd	10.0	nM	10.1038/nbt.1990
Homo sapiens	Platelet-derived growth factor receptor alpha	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Platelet-derived growth factor receptor alpha	Residual Activity	5.0	%	10.1042/bj20121418
Homo sapiens	Platelet-derived growth factor receptor beta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	0.6	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	0.76	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	2.34	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	3.56	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	4.3	nM	10.1016/j.ejmech.2015.08.027
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	4.7	nM	10.1016/j.ejmech.2018.03.013
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	55.0	nM	10.1016/j.bmcl.2021.128258
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	204.7	nM	10.1016/j.ejmech.2017.08.067
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	94.81	%	10.1016/j.bmc.2011.06.022
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	95.8	%	10.1016/j.bmc.2011.06.022
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	99.8	%	10.1016/j.ejmech.2015.04.018
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	1.8	nM	10.1038/nbt1358
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	1.8	nM	10.1038/nbt.1990
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	2.7	nM	10.1038/nbt1068
Homo sapiens	Platelet-derived growth factor receptor beta	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Platelet-derived growth factor receptor beta	Residual Activity	4.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C alpha	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C alpha	IC50	0.305	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase C alpha	IC50	0.37	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Protein kinase C alpha	IC50	0.474	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	Protein kinase C alpha	IC50	0.506	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C alpha	IC50	0.542	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Protein kinase C alpha	IC50	0.7	nM	10.1021/jm800861c
Homo sapiens	Protein kinase C alpha	IC50	1.0	nM	10.1016/j.bmcl.2006.05.092
Homo sapiens	Protein kinase C alpha	IC50	1.2	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Protein kinase C alpha	IC50	2.4	nM	10.1021/acs.jnatprod.7b01058
Homo sapiens	Protein kinase C alpha	IC50	3.0	nM	10.1016/j.bmc.2011.02.036
Homo sapiens	Protein kinase C alpha	IC50	4.0	nM	10.1016/0960-894X(95)00060-7
Homo sapiens	Protein kinase C alpha	IC50	28.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Protein kinase C alpha	IC50	28.0	nM	10.1021/jm049478u
Homo sapiens	Protein kinase C alpha	IC50	45.0	nM	10.1016/s0960-894x(03)00286-5
Homo sapiens	Protein kinase C alpha	IC50	45.0	nM	10.1021/jm950588y
Homo sapiens	Protein kinase C alpha	Kd	50.0	nM	10.1038/nbt1068
Homo sapiens	Protein kinase C alpha	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C alpha	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C beta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C beta	IC50	1.44	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	Protein kinase C beta	IC50	2.5	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase C beta	IC50	2.78	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C beta	IC50	4.0	nM	10.1016/j.bmc.2008.06.017
Homo sapiens	Protein kinase C beta	IC50	7.26	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase C beta	IC50	10.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Protein kinase C beta	IC50	10.0	nM	10.1021/jm049478u
Homo sapiens	Protein kinase C beta	IC50	12.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C beta	IC50	19.0	nM	10.1016/s0960-894x(03)00286-5
Homo sapiens	Protein kinase C beta	IC50	19.0	nM	10.1021/jm950588y
Homo sapiens	Protein kinase C beta	IC50	23.0	nM	10.1016/s0960-894x(03)00286-5
Homo sapiens	Protein kinase C beta	IC50	23.0	nM	10.1021/jm950588y
Homo sapiens	Protein kinase C beta	IC50	63.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Protein kinase C beta	IC50	63.0	nM	10.1021/jm049478u
Homo sapiens	Protein kinase C beta	IC50	77.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Protein kinase C beta	IC50	77.0	nM	10.1021/jm049478u
Homo sapiens	Protein kinase C beta	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C beta	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C delta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C delta	IC50	0.128	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C delta	IC50	0.129	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase C delta	IC50	5.5	nM	10.1021/acs.jnatprod.7b01082
Homo sapiens	Protein kinase C delta	IC50	28.0	nM	10.1016/s0960-894x(03)00286-5
Homo sapiens	Protein kinase C delta	IC50	28.0	nM	10.1021/jm950588y
Homo sapiens	Protein kinase C delta	IC50	41.0	nM	10.1074/jbc.m707233200
Homo sapiens	Protein kinase C delta	IC50	49.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Protein kinase C delta	IC50	49.0	nM	10.1021/jm049478u
Homo sapiens	Protein kinase C delta	IC50	570.0	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Protein kinase C delta	Kd	1.5	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C delta	Kd	1.5	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C delta	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C delta	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C epsilon	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C epsilon	IC50	0.143	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase C epsilon	IC50	0.198	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C epsilon	IC50	0.6	nM	10.1016/j.bmc.2014.12.026
Homo sapiens	Protein kinase C epsilon	IC50	1.0	nM	10.1074/jbc.m707233200
Homo sapiens	Protein kinase C epsilon	IC50	1.5	nM	10.1016/j.bmc.2009.05.031
Homo sapiens	Protein kinase C epsilon	IC50	1.5	nM	10.1016/j.ejmech.2013.07.046
Homo sapiens	Protein kinase C epsilon	IC50	12.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Protein kinase C epsilon	IC50	18.0	nM	10.1016/s0960-894x(03)00286-5
Homo sapiens	Protein kinase C epsilon	IC50	18.0	nM	10.1021/jm950588y
Homo sapiens	Protein kinase C epsilon	IC50	21.0	nM	10.1074/jbc.m707233200
Homo sapiens	Protein kinase C epsilon	Kd	0.25	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C epsilon	Kd	0.25	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C epsilon	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C epsilon	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C eta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C eta	IC50	0.251	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C eta	IC50	1.17	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase C eta	IC50	5.0	nM	10.1016/s0960-894x(03)00286-5
Homo sapiens	Protein kinase C eta	IC50	5.0	nM	10.1021/jm950588y
Homo sapiens	Protein kinase C eta	Kd	4.8	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C eta	Kd	4.8	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C eta	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C eta	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C eta	Selectivity	0.5017	None	10.1038/nbt1358
Homo sapiens	Protein kinase C gamma	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C gamma	IC50	0.542	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase C gamma	IC50	1.43	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C gamma	IC50	2.76	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Protein kinase C gamma	IC50	6.6	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Protein kinase C gamma	IC50	18.0	nM	10.1074/jbc.m707233200
Homo sapiens	Protein kinase C gamma	IC50	59.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Protein kinase C gamma	IC50	59.0	nM	10.1021/jm049478u
Homo sapiens	Protein kinase C gamma	IC50	110.0	nM	10.1016/s0960-894x(03)00286-5
Homo sapiens	Protein kinase C gamma	IC50	110.0	nM	10.1021/jm950588y
Homo sapiens	Protein kinase C gamma	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C gamma	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C iota	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C iota	IC50	16.7	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase C iota	IC50	31.6	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C iota	IC50	364.0	nM	10.1074/jbc.m707233200
Homo sapiens	Protein kinase C iota	Kd	26.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C iota	Residual Activity	10.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C iota	Residual Activity	50.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C mu	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C mu	IC50	1.35	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase C mu	IC50	3.6	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C mu	Kd	27.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C mu	Kd	27.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C mu	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C mu	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C nu	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C nu	IC50	1.52	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C nu	IC50	2.07	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase C nu	Kd	18.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C nu	Kd	18.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C (PKC)	IC50	0.08	nM	10.1021/jm020143r
Homo sapiens	Protein kinase C (PKC)	IC50	0.6	nM	10.1016/S0960-894X(01)80407-8
Homo sapiens	Protein kinase C (PKC)	IC50	1.0	nM	10.1016/j.ejmech.2013.11.036
Homo sapiens	Protein kinase C (PKC)	IC50	2.0	nM	10.1016/0960-894X(94)00460-W
Homo sapiens	Protein kinase C (PKC)	IC50	2.7	nM	10.1016/S0960-894X(00)80167-5
Homo sapiens	Protein kinase C (PKC)	IC50	3.0	nM	10.1016/0960-894X(95)00497-H
Homo sapiens	Protein kinase C (PKC)	IC50	6.0	nM	10.1016/0960-894X(94)80004-9
Homo sapiens	Protein kinase C (PKC)	IC50	7.0	nM	10.1016/s0960-894x(03)00791-1
Homo sapiens	Protein kinase C (PKC)	IC50	7.0	nM	10.1021/jm0000214
Homo sapiens	Protein kinase C (PKC)	IC50	8.0	nM	10.1016/0960-894X(94)80024-3
Homo sapiens	Protein kinase C (PKC)	IC50	23.0	nM	10.1016/0960-894X(96)00343-5
Homo sapiens	Protein kinase C (PKC)	IC50	38.0	nM	10.1016/j.bmcl.2014.05.085
Homo sapiens	Protein kinase C (PKC)	IC50	1100.0	nM	10.1021/jm020455u
Homo sapiens	Protein kinase C theta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C theta	IC50	1.44	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C theta	IC50	2.58	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase C theta	IC50	5.0	nM	10.1021/acs.jmedchem.0c01271
Homo sapiens	Protein kinase C theta	IC50	6.0	nM	10.1021/acs.jmedchem.0c01271
Homo sapiens	Protein kinase C theta	Inhibition	50.0	%	10.1021/acs.jmedchem.0c01271
Homo sapiens	Protein kinase C theta	Kd	8.5	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C theta	Kd	8.5	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C theta	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C zeta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C zeta	IC50	39.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase C zeta	IC50	76.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase C zeta	IC50	216.8	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Protein kinase C zeta	IC50	1500.0	nM	10.1016/s0960-894x(03)00286-5
Homo sapiens	Protein kinase C zeta	IC50	1500.0	nM	10.1021/jm950588y
Homo sapiens	Protein kinase C zeta	IC50	10000.0	nM	10.1021/jm049478u
Homo sapiens	Protein kinase C zeta	Inhibition	10.0	%	10.1016/s0960-894x(03)00644-9
Homo sapiens	Protein kinase C zeta	Inhibition	90.0	%	10.1021/jm2005892
Homo sapiens	Protein kinase C zeta	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase C zeta	Residual Activity	20.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase N1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase N1	IC50	1.0	nM	10.1021/np4005745
Homo sapiens	Protein kinase N1	IC50	1.2	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Protein kinase N1	IC50	3.78	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase N1	IC50	4.21	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase N1	Kd	1.3	nM	10.1038/nbt1358
Homo sapiens	Protein kinase N1	Kd	1.3	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase N2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase N2	IC50	1.97	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	Protein kinase N2	IC50	2.2	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Protein kinase N2	IC50	6.09	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein kinase N2	IC50	11.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein kinase N2	Kd	2.5	nM	10.1038/nbt1358
Homo sapiens	Protein kinase N2	Kd	2.5	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase N2	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Protein kinase N2	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Protein odd-skipped-related 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein odd-skipped-related 1	IC50	19.1	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein odd-skipped-related 1	IC50	61.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein tyrosine kinase 2 beta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein tyrosine kinase 2 beta	IC50	8.44	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Protein tyrosine kinase 2 beta	IC50	10.6	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Protein tyrosine kinase 2 beta	Kd	3.5	nM	10.1038/nbt1358
Homo sapiens	Protein tyrosine kinase 2 beta	Kd	3.5	nM	10.1038/nbt.1990
Homo sapiens	Protein tyrosine kinase 2 beta	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Protein tyrosine kinase 2 beta	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	deltaTm	4.8	K	10.1021/acs.jmedchem.1c00845
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	IC50	4.68	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	IC50	11.6	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	IC50	83.0	nM	10.1016/j.bmc.2016.05.025
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Kd	6.4	nM	10.1021/acsmedchemlett.3c00127
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Kd	6.4	nM	10.1038/nbt1358
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Kd	6.4	nM	10.1038/nbt.1990
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	IC50	0.07	nM	10.1016/j.bmcl.2009.06.066
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	IC50	0.145	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	IC50	0.149	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	IC50	0.2	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	IC50	1.0	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	IC50	1.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	Kd	30.0	nM	10.1038/nbt1358
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	Kd	30.0	nM	10.1038/nbt.1990
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Pseudopodium-enriched atypical kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Pseudopodium-enriched atypical kinase 1	IC50	2.03	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Pseudopodium-enriched atypical kinase 1	IC50	3.04	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Putative uncharacterized serine/threonine-protein kinase SgK110	Kd	25.0	nM	10.1038/nbt.1990
Homo sapiens	Pyruvate dehydrogenase kinase isoform 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Pyruvate dehydrogenase kinase isoform 1	IC50	0.506	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Pyruvate dehydrogenase kinase isoform 1	IC50	0.538	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Raji	EC50	2000.0	nM	10.1016/j.bmcl.2014.09.061
Homo sapiens	Ramos	Activity	nan	None	10.1016/j.bmc.2019.06.029
Homo sapiens	Rec1	IC50	25.5	nM	10.1016/j.ejmech.2021.113727
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 3	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 4	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	27.6	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	34.0	nM	10.1016/j.ejmech.2016.12.055
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	51.0	nM	10.1016/j.ejmech.2022.114661
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	60.8	nM	10.1016/j.ejmech.2018.06.011
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	104.0	nM	10.1016/j.bmcl.2020.127288
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	108.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	115.0	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	131.0	nM	10.1016/j.bmcl.2020.127288
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Inhibition	94.0	%	10.1016/j.ejmech.2018.06.011
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Inhibition	100.0	%	10.1016/j.ejmech.2017.12.022
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Inhibition	100.0	%	10.1016/j.ejmech.2018.06.011
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Kd	190.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	IC50	28.3	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	IC50	29.4	nM	10.1016/j.bmcl.2020.127288
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	IC50	112.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	IC50	138.0	nM	10.1016/j.ejmech.2021.113674
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	IC50	282.0	nM	10.1021/jm800861c
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	IC50	329.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	IC50	535.0	nM	10.1016/j.bmcl.2020.127288
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	Kd	770.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	Residual Activity	12.0	%	10.1042/bj20121418
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	Residual Activity	58.0	%	10.1042/bj20121418
Homo sapiens	Receptor tyrosine-protein kinase erbB-3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Regulator of G-protein signaling 4	Potency	10621.3	nM	None
Homo sapiens	Retinoblastoma-associated protein	FC	0.8	None	10.1016/j.ejmech.2018.01.004
Homo sapiens	Retinoblastoma-associated protein	FC	1.0	None	10.1016/j.ejmech.2018.01.004
Homo sapiens	Retinoblastoma-associated protein	IC50	66.0	nM	10.1016/j.ejmech.2017.02.062
Homo sapiens	Rho-associated protein kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Rho-associated protein kinase 1	IC50	0.444	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Rho-associated protein kinase 1	IC50	0.64	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Rho-associated protein kinase 1	IC50	0.68	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Rho-associated protein kinase 1	IC50	0.799	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Rho-associated protein kinase 1	IC50	1.1	nM	10.1021/jm800861c
Homo sapiens	Rho-associated protein kinase 1	IC50	19.0	nM	10.1016/j.ejmech.2015.08.027
Homo sapiens	Rho-associated protein kinase 1	Inhibition	85.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Rho-associated protein kinase 1	Kd	0.28	nM	10.1038/nbt.1990
Homo sapiens	Rho-associated protein kinase 1	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Rho-associated protein kinase 1	Residual Activity	5.0	%	10.1042/bj20121418
Homo sapiens	Rho-associated protein kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Rho-associated protein kinase 2	IC50	0.246	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Rho-associated protein kinase 2	IC50	0.933	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Rho-associated protein kinase 2	IC50	7.8	nM	10.1021/acs.jnatprod.7b01058
Homo sapiens	Rho-associated protein kinase 2	IC50	9.0	nM	10.1021/acs.jnatprod.7b01055
Homo sapiens	Rho-associated protein kinase 2	Kd	0.24	nM	10.1038/nbt.1990
Homo sapiens	Rho-associated protein kinase 2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Rho-associated protein kinase 2	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Rhodopsin kinase	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Rhodopsin kinase	IC50	57.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Rhodopsin kinase	IC50	78.1	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Rhodopsin kinase	Kd	0.97	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase 1	IC50	0.43	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ribosomal protein S6 kinase 1	IC50	0.553	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase 1	IC50	0.871	nM	10.1039/c9md00537d
Homo sapiens	Ribosomal protein S6 kinase 1	IC50	1.0	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Ribosomal protein S6 kinase 1	Kd	1.3	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase 1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase 1	Residual Activity	4.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase 2	IC50	0.726	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ribosomal protein S6 kinase 2	IC50	2.35	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 1	IC50	0.09	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Ribosomal protein S6 kinase alpha 1	IC50	0.1	nM	10.1021/jm800861c
Homo sapiens	Ribosomal protein S6 kinase alpha 1	IC50	0.126	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ribosomal protein S6 kinase alpha 1	IC50	0.126	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 1	IC50	0.5	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Ribosomal protein S6 kinase alpha 1	IC50	1.2	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	43.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	43.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	1200.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	1200.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 2	IC50	0.14	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ribosomal protein S6 kinase alpha 2	IC50	0.227	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	8.9	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	8.9	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	10.0	nM	10.1038/nbt1068
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	190.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	190.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 3	IC50	0.0795	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ribosomal protein S6 kinase alpha 3	IC50	0.124	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 3	IC50	0.5	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	60.0	nM	10.1038/nbt1068
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	69.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	69.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 4	IC50	2.98	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ribosomal protein S6 kinase alpha 4	IC50	11.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	120.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	120.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	2200.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	2200.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 5	IC50	0.426	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ribosomal protein S6 kinase alpha 5	IC50	1.4	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Ribosomal protein S6 kinase alpha 5	IC50	1.42	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	20.0	nM	10.1038/nbt1068
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	42.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	42.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	890.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	890.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 6	IC50	0.134	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Ribosomal protein S6 kinase alpha 6	IC50	0.159	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	18.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	18.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	3300.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	3300.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	RPMI-8226	Activity	0.245	ng/ml	10.1016/j.ejmech.2020.112062
Homo sapiens	RPMI-8226	Activity	0.4081	ng/ml	10.1016/j.ejmech.2020.112062
Homo sapiens	RPMI-8226	Activity	1.508	ng/ml	10.1016/j.ejmech.2020.112062
Homo sapiens	RPMI-8226	Activity	24.97	ng/ml	10.1016/j.ejmech.2020.112062
Homo sapiens	RPMI-8226	Activity	336.16	pg/ml	10.1016/j.ejmech.2020.112062
Homo sapiens	RPMI-8226	Activity	449.8	pg/ml	10.1016/j.ejmech.2020.112062
Homo sapiens	Scavenger mRNA-decapping enzyme DcpS	Inhibition	nan	%	None
Homo sapiens	SEM	Activity	0.0	%	10.1016/j.ejmech.2016.02.034
Homo sapiens	SEM	Activity	2.6	%	10.1016/j.ejmech.2016.02.034
Homo sapiens	SEM	Activity	5.5	%	10.1016/j.ejmech.2016.02.034
Homo sapiens	SEM	Activity	85.3	%	10.1016/j.ejmech.2016.02.034
Homo sapiens	SEM	Activity	100.0	%	10.1016/j.ejmech.2016.02.034
Homo sapiens	SEM	Activity	nan	None	10.1016/j.ejmech.2016.02.034
Homo sapiens	Serine/threonine-protein kinase 10	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 10	Delta Tm	22.9	degrees C	10.1016/j.ejmech.2020.112721
Homo sapiens	Serine/threonine-protein kinase 10	IC50	6.93	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 10	IC50	9.01	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 10	Kd	0.03	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 10	Kd	0.037	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 10	Kd	0.037	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 10	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase 11	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 11	IC50	48.7	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 11	IC50	70.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 11	Kd	61.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 11	Kd	61.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 11	Residual Activity	19.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase 11	Residual Activity	74.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase 16	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 16	IC50	235.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 16	IC50	242.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 16	Kd	200.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 16	Kd	270.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 16	Kd	270.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 17A	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 17A	IC50	30.4	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 17A	IC50	31.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 17A	IC50	54.0	nM	10.1021/acs.jmedchem.2c00173
Homo sapiens	Serine/threonine-protein kinase 17A	Kd	14.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 17A	Kd	14.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 17A	Kd	23.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 17A	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase 17A	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase 17B	Delta Tm	8.57	degrees C	10.1021/acs.jmedchem.1c01165
Homo sapiens	Serine/threonine-protein kinase 17B	IC50	25.8	nM	10.1016/j.bmc.2014.12.026
Homo sapiens	Serine/threonine-protein kinase 17B	Kd	21.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 17B	Kd	21.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 17B	Kd	26.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 2	Delta Tm	16.9	degrees C	10.1016/j.ejmech.2020.112721
Homo sapiens	Serine/threonine-protein kinase 2	IC50	9.04	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 2	IC50	14.6	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 2	IC50	19.0	nM	10.1021/acs.jmedchem.0c01579
Homo sapiens	Serine/threonine-protein kinase 2	Kd	0.02	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 2	Kd	0.024	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 2	Kd	0.024	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 24	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 24	Delta Tm	8.8	degrees C	10.1021/acs.jmedchem.0c02144
Homo sapiens	Serine/threonine-protein kinase 24	IC50	3.34	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	Serine/threonine-protein kinase 24	IC50	4.32	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 24	IC50	11.8	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 24	Kd	120.0	nM	10.1021/acsmedchemlett.3c00127
Homo sapiens	Serine/threonine-protein kinase 24	Kd	120.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 24	Kd	120.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 24	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase 25	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 25	IC50	1.9	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	Serine/threonine-protein kinase 25	IC50	2.71	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 25	IC50	3.98	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 25	Kd	110.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 25	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 32A	Kd	13.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 32B	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 32B	IC50	25.8	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 32B	IC50	49.1	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 32B	Kd	98.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 32B	Kd	98.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 32C	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 32C	IC50	139.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 32C	IC50	325.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 32C	Kd	310.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 32C	Kd	310.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 33	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 33	IC50	36.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 33	IC50	38.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 33	Kd	1.8	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 33	Kd	1.8	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 33	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase 33	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase 35	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 36	Kd	2900.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 36	Kd	6700.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 36	Kd	6700.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 38	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 38	IC50	0.628	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 38	IC50	6.87	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 38	Kd	56.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 38-like	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 38-like	IC50	0.831	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 38-like	IC50	1.47	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase 38-like	Kd	28.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 38-like	Kd	28.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 38-like	Kd	77.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase AKT	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase AKT	EC50	460.0	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	Serine/threonine-protein kinase AKT	EC50	460.0	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Serine/threonine-protein kinase AKT	EC50	nan	None	10.1016/j.bmcl.2006.05.092
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	1.5	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	1.5	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	3.8	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	4.57	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	4.62	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	4.62	nM	10.1016/j.ejmech.2021.113511
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	4.95	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	5.94	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	6.0	nM	10.1021/jm800861c
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	7.04	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	9.0	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	11.0	nM	10.1016/j.bmcl.2006.05.092
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	11.0	nM	10.1016/j.bmcl.2013.11.020
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	12.0	nM	10.1016/j.ejmech.2015.08.027
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	12.0	nM	10.1021/acs.jnatprod.7b01082
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	17.6	nM	10.1016/j.bmc.2014.12.026
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	17.6	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	30.0	nM	10.1021/np4005745
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	40.0	nM	10.1016/j.ejmech.2013.11.036
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	56.0	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	130.0	nM	10.1016/j.bmc.2013.11.052
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	290.0	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	290.0	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	4000.0	nM	10.1016/j.ejmech.2019.111875
Homo sapiens	Serine/threonine-protein kinase AKT	Inhibition	61.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Serine/threonine-protein kinase AKT	Inhibition	96.52	%	10.1016/j.ejmech.2013.03.043
Homo sapiens	Serine/threonine-protein kinase AKT	Inhibition	96.52	%	10.1016/j.ejmech.2013.07.056
Homo sapiens	Serine/threonine-protein kinase AKT	Inhibition	nan	%	10.1016/j.bmc.2016.05.031
Homo sapiens	Serine/threonine-protein kinase AKT	Kd	20.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase AKT	Kd	20.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase AKT	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase AKT	Residual Activity	13.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase AKT2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase AKT2	IC50	6.5	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	Serine/threonine-protein kinase AKT2	IC50	6.5	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Serine/threonine-protein kinase AKT2	IC50	9.0	nM	10.1016/j.bmcl.2006.05.092
Homo sapiens	Serine/threonine-protein kinase AKT2	IC50	16.0	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Serine/threonine-protein kinase AKT2	IC50	21.5	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase AKT2	IC50	41.5	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase AKT2	Kd	44.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase AKT2	Kd	44.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase AKT2	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase AKT2	Residual Activity	4.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase AKT3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase AKT3	IC50	0.64	nM	10.1021/jm801317h
Homo sapiens	Serine/threonine-protein kinase AKT3	IC50	3.75	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase AKT3	IC50	5.0	nM	10.1016/j.bmcl.2006.05.092
Homo sapiens	Serine/threonine-protein kinase AKT3	IC50	10.0	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	Serine/threonine-protein kinase AKT3	IC50	10.0	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Serine/threonine-protein kinase AKT3	IC50	10.0	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Serine/threonine-protein kinase AKT3	IC50	13.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase AKT3	Kd	170.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase AKT3	Kd	170.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase AKT3	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase AKT3	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase A-Raf	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Delta TM	16.68	C	None
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	0.46	nM	10.1016/j.ejmech.2021.113495
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	0.6	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	0.86	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	0.936	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	1.0	nM	10.1016/j.bmc.2014.06.047
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	1.0	nM	10.1016/j.bmc.2016.03.042
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	1.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	1.0	nM	10.1016/j.ejmech.2021.113511
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	1.38	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	2.0	nM	10.1016/j.bmc.2016.03.042
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	2.28	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	2.4	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	3.0	nM	10.1016/j.bmc.2020.115525
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	3.67	nM	10.1016/j.ejmech.2018.09.032
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	7.63	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	11.0	nM	10.1016/j.ejmech.2015.08.027
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	15.0	nM	10.1016/j.ejmech.2013.11.036
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	18.0	nM	10.1016/j.bmc.2009.05.031
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	18.0	nM	10.1016/j.ejmech.2013.07.046
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	18.09	nM	10.1016/j.ejmech.2020.112108
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	22.0	nM	10.1021/jm800861c
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	23.0	nM	10.1016/j.ejmech.2018.03.013
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	39.0	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Inhibition	84.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Kd	16.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Kd	17.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Kd	110.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Residual Activity	-9.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Delta Tm	9.9	degrees C	10.1016/j.ejmech.2020.112721
Homo sapiens	Serine/threonine-protein kinase Aurora-B	IC50	1.0	nM	10.1016/j.bmc.2014.06.047
Homo sapiens	Serine/threonine-protein kinase Aurora-B	IC50	1.0	nM	10.1016/j.bmc.2016.03.042
Homo sapiens	Serine/threonine-protein kinase Aurora-B	IC50	1.5	nM	10.1016/j.bmcl.2016.05.017
Homo sapiens	Serine/threonine-protein kinase Aurora-B	IC50	1.8	nM	10.1016/j.ejmech.2014.07.108
Homo sapiens	Serine/threonine-protein kinase Aurora-B	IC50	6.0	nM	10.1016/j.bmc.2020.115525
Homo sapiens	Serine/threonine-protein kinase Aurora-B	IC50	6.04	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Aurora-B	IC50	7.0	nM	10.1016/j.bmc.2016.03.042
Homo sapiens	Serine/threonine-protein kinase Aurora-B	IC50	7.8	nM	10.1016/j.ejmech.2018.09.032
Homo sapiens	Serine/threonine-protein kinase Aurora-B	IC50	8.0	nM	10.1021/np4005745
Homo sapiens	Serine/threonine-protein kinase Aurora-B	IC50	10.6	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Aurora-B	IC50	26.13	nM	10.1016/j.ejmech.2020.112108
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Kd	19.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Kd	19.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Aurora-C	IC50	1.92	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Aurora-C	IC50	2.42	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Kd	11.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Kd	23.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Kd	23.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase B-raf	Delta Tm	0.8	degrees C	10.1016/j.ejmech.2020.112721
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	4.5	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	4.5	nM	10.1016/j.ejmech.2021.113511
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	5.0	nM	10.1016/j.bmc.2014.12.026
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	5.03	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	8.7	nM	10.1021/acs.jnatprod.7b01082
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	8.8	nM	10.1016/j.ejmech.2021.113674
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	14.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	14.0	nM	10.1016/j.ejmech.2021.113511
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	31.6	nM	10.1016/j.ejmech.2021.113277
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	nan	None	10.1016/j.bmc.2017.09.003
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	nan	None	10.1016/j.bmcl.2016.10.029
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase B-raf	Inhibition	0.015	%	10.1016/j.ejmech.2013.11.036
Homo sapiens	Serine/threonine-protein kinase B-raf	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase B-raf	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Chk1	Activity	-1.28	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk1	Activity	-0.27	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk1	Activity	0.31	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk1	Activity	1.47	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk1	Activity	2.55	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk1	Activity	6.54	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk1	Activity	9.81	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk1	Activity	13.67	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk1	Activity	41.24	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk1	Activity	55.99	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	0.1	nM	10.1021/jm800861c
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	0.142	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	0.16	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	0.186	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	0.5	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	0.5	nM	10.1021/jm801317h
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	1.2	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	2.1	nM	10.1021/jm2007326
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	2.1	nM	10.1021/jm900314j
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	9.5	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	9.5	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	2100.0	nM	10.1016/j.bmc.2009.11.058
Homo sapiens	Serine/threonine-protein kinase Chk1	Inhibition	73.0	%	10.1021/jm900314j
Homo sapiens	Serine/threonine-protein kinase Chk1	Inhibition	86.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Serine/threonine-protein kinase Chk1	Kd	3.2	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Chk1	Kd	3.2	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Chk1	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Chk2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk2	IC50	3.34	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Serine/threonine-protein kinase Chk2	IC50	4.86	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Serine/threonine-protein kinase Chk2	IC50	5.72	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Chk2	IC50	6.7	nM	10.1021/jm800861c
Homo sapiens	Serine/threonine-protein kinase Chk2	IC50	9.21	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Chk2	IC50	27.0	nM	10.1016/j.ejmech.2011.01.045
Homo sapiens	Serine/threonine-protein kinase Chk2	IC50	27.0	nM	10.1021/jm2007326
Homo sapiens	Serine/threonine-protein kinase Chk2	IC50	27.0	nM	10.1021/jm900314j
Homo sapiens	Serine/threonine-protein kinase Chk2	IC50	27000.0	nM	10.1016/j.bmc.2009.11.058
Homo sapiens	Serine/threonine-protein kinase Chk2	Kd	74.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Chk2	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Chk2	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase c-TAK1	IC50	0.297	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase c-TAK1	IC50	0.438	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Kd	0.5	nM	10.1021/acsmedchemlett.3c00127
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Kd	3.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Kd	3.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase D2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase D2	IC50	1.33	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase D2	IC50	1.48	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase D2	Kd	72.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase D2	Kd	72.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase D2	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase D2	Residual Activity	5.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase DCLK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase DCLK1	IC50	173.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase DCLK1	IC50	361.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase DCLK1	Kd	110.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase DCLK1	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase DCLK2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase DCLK2	IC50	83.5	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase DCLK2	IC50	94.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase DCLK2	Kd	73.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase DCLK2	Kd	73.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase DCLK2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase DCLK2	Residual Activity	9.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase DCLK3	Kd	17.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase DCLK3	Kd	17.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase EEF2K	Residual Activity	74.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase EEF2K	Residual Activity	120.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE1	IC50	45.3	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE1	IC50	204.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE1	Kd	21.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE2	IC50	17.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE2	IC50	65.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase GAK	IC50	11.0	nM	10.1016/j.ejmech.2021.113158
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	17.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	17.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	68.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase haspin	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase haspin	IC50	19.0	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	Serine/threonine-protein kinase haspin	IC50	32.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase haspin	IC50	75.6	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase haspin	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase haspin	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase ICK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase ICK	IC50	38.6	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase ICK	IC50	41.06	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Serine/threonine-protein kinase ICK	IC50	53.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase ICK	Kd	16.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase LATS1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase LATS1	IC50	12.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase LATS1	IC50	13.3	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase LATS1	Kd	42.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase LATS1	Kd	42.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase LATS2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase LATS2	IC50	3.76	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase LATS2	IC50	8.62	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase LATS2	Kd	17.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase LATS2	Kd	17.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase LMTK3	IC50	0.002399	nM	None
Homo sapiens	Serine/threonine-protein kinase LMTK3	IC50	0.0024	nM	10.1016/j.bmcl.2020.127108
Homo sapiens	Serine/threonine-protein kinase LMTK3	Inhibition	108.86	%	None
Homo sapiens	Serine/threonine-protein kinase MAK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MAK	IC50	22.7	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase MAK	IC50	28.7	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MAK	Kd	2600.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MARK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MARK1	IC50	0.261	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase MARK1	IC50	0.417	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MARK1	Kd	4.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MARK1	Kd	4.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MARK1	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase MARK1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MRCK-A	IC50	0.998	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase MRCK-A	IC50	5.35	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Kd	57.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Kd	57.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase MRCK beta	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MRCK beta	IC50	0.727	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase MRCK beta	IC50	4.75	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MRCK beta	Kd	42.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MRCK beta	Kd	42.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MRCK beta	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase MRCK gamma	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MRCK gamma	IC50	0.19	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase MRCK gamma	IC50	0.848	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MRCK gamma	Kd	37.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MRCK gamma	Kd	37.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MST1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MST1	Delta Tm	13.8	degrees C	10.1021/acs.jmedchem.0c02144
Homo sapiens	Serine/threonine-protein kinase MST1	IC50	1.02	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase MST1	IC50	1.58	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	0.19	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	0.19	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	0.2	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	1.0	nM	10.1021/acsmedchemlett.3c00127
Homo sapiens	Serine/threonine-protein kinase MST1	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase MST1	Residual Activity	4.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase MST2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MST2	Delta Tm	12.4	degrees C	10.1021/acs.jmedchem.0c02144
Homo sapiens	Serine/threonine-protein kinase MST2	IC50	0.41	nM	10.1021/jm800861c
Homo sapiens	Serine/threonine-protein kinase MST2	IC50	2.83	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase MST2	IC50	4.72	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Serine/threonine-protein kinase MST2	IC50	5.49	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MST2	Kd	0.18	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MST2	Kd	0.18	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MST2	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase MST2	Residual Activity	5.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase MST4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MST4	Delta Tm	7.1	degrees C	10.1021/acs.jmedchem.0c02144
Homo sapiens	Serine/threonine-protein kinase MST4	IC50	2.87	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase MST4	IC50	21.9	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase MST4	Kd	140.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MST4	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase mTOR	IC50	nan	None	10.1016/j.bmc.2017.02.030
Homo sapiens	Serine/threonine-protein kinase mTOR	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase mTOR	Residual Activity	87.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase mTOR	Residual Activity	90.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase mTOR	Residual Activity	93.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase mTOR	Residual Activity	101.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase N3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase N3	IC50	7.8	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase N3	IC50	13.2	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek1	IC50	9.1	nM	10.1016/j.bmcl.2021.128418
Homo sapiens	Serine/threonine-protein kinase Nek1	IC50	9.22	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Nek1	IC50	18.4	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek1	Kd	860.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Nek1	Kd	860.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Nek11	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek11	IC50	290.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Nek11	IC50	752.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek11	Kd	3100.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Nek11	Residual Activity	5.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Nek11	Residual Activity	54.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase NEK2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase NEK2	IC50	170.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase NEK2	IC50	345.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase NEK2	IC50	4790.0	nM	10.1021/np4005745
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	740.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	750.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	750.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK2	Residual Activity	32.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase NEK2	Residual Activity	63.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Nek3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek3	IC50	24200.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek3	IC50	63700.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Nek3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Nek3	Residual Activity	67.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Nek3	Residual Activity	105.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Nek4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek4	IC50	74.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Nek4	IC50	96.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Nek5	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek5	IC50	76.3	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Nek5	IC50	96.5	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek5	Kd	810.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Nek5	Kd	810.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK6	IC50	10000.0	nM	10.1021/np4005745
Homo sapiens	Serine/threonine-protein kinase NEK6	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase NEK6	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase NEK6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK6	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase NEK6	Residual Activity	72.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase NEK6	Residual Activity	75.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase NEK7	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase NEK7	Kd	4500.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase NEK7	Kd	4500.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK7	Residual Activity	93.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase NEK7	Residual Activity	114.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Nek8	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek8	IC50	17.5	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Nek8	IC50	35.1	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase NEK9	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase NEK9	IC50	71.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase NEK9	IC50	131.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase NEK9	Kd	3100.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase NEK9	Kd	3100.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK9	Kd	6700.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase NIM1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase NIM1	IC50	91.5	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase NIM1	IC50	129.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase NIM1	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine protein kinase NLK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine protein kinase NLK	IC50	55.5	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine protein kinase NLK	IC50	77.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine protein kinase NLK	Kd	220.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine protein kinase NLK	Kd	220.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine protein kinase NLK	Residual Activity	6.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine protein kinase NLK	Residual Activity	30.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase OSR1	Kd	440.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PAK 1	Delta Tm	5.9	degrees C	10.1021/acs.jmedchem.0c02144
Homo sapiens	Serine/threonine-protein kinase PAK 1	IC50	0.212	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PAK 1	IC50	0.3	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Serine/threonine-protein kinase PAK 1	IC50	0.541	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PAK 1	Inhibition	84.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Serine/threonine-protein kinase PAK 1	Kd	0.57	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK 1	Kd	0.57	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 1	Kd	2.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PAK 2	IC50	1.0	nM	10.1021/jm800861c
Homo sapiens	Serine/threonine-protein kinase PAK 2	IC50	1.17	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PAK 2	IC50	2.59	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Serine/threonine-protein kinase PAK 2	IC50	3.46	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PAK 2	Kd	3.1	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK 2	Kd	3.1	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 2	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PAK 2	Residual Activity	5.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PAK 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PAK 3	IC50	0.235	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PAK 3	IC50	0.343	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PAK 3	Kd	0.5	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK 3	Kd	7.1	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK 3	Kd	7.1	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 3	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PAK 3	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PAK 4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PAK 4	IC50	1.0	nM	10.1016/j.bmcl.2019.126807
Homo sapiens	Serine/threonine-protein kinase PAK 4	IC50	1.9	nM	10.1016/j.ejmech.2017.02.063
Homo sapiens	Serine/threonine-protein kinase PAK 4	IC50	22.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PAK 4	IC50	27.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PAK 4	Inhibition	100.0	%	10.1016/j.ejmech.2019.111878
Homo sapiens	Serine/threonine-protein kinase PAK 4	Kd	6.3	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK 4	Kd	6.3	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 4	Kd	8.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK 4	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PAK6	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PAK6	IC50	31.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PAK6	IC50	34.5	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PAK6	Kd	0.4	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK6	Kd	0.57	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK6	Kd	0.57	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK6	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PAK6	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PAK7	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PAK7	IC50	2.53	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PAK7	IC50	5.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PAK7	Kd	1.2	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK7	Kd	1.2	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK7	Kd	3.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK7	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	24.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	24.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	25.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-2	Kd	96.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-2	Kd	96.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-3	Kd	270.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-3	Kd	270.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PFTAIRE-1	Kd	160.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PFTAIRE-1	Kd	160.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PFTAIRE-2	Kd	260.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PIM1	Activity	0.0	%	10.1021/jm0504858
Homo sapiens	Serine/threonine-protein kinase PIM1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	2.67	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	2.7	nM	10.1021/jm800861c
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	4.33	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	4.63	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	7.5	nM	10.1021/jm801242y
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	10.0	nM	10.1016/j.bmcl.2009.01.005
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	10.0	nM	10.1021/jm800937p
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	10.0	nM	10.1021/jm801242y
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	17.0	nM	10.1016/j.bmc.2020.115828
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	22.0	nM	10.1016/j.bmc.2016.03.016
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	24.6	nM	10.1021/jm801242y
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	31.0	nM	10.1016/j.ejmech.2018.04.056
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	58.0	nM	10.1021/acs.jnatprod.7b01082
Homo sapiens	Serine/threonine-protein kinase PIM1	IC50	110.0	nM	10.1021/np4005745
Homo sapiens	Serine/threonine-protein kinase PIM1	Kb	705.0	10^6/M	10.1021/jm0504858
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	1.4	nM	10.1021/jm0504858
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	3.2	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	3.2	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	15.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PIM1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PIM1	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PIM2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PIM2	IC50	4.73	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PIM2	IC50	7.0	nM	10.1021/jm801242y
Homo sapiens	Serine/threonine-protein kinase PIM2	IC50	21.7	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PIM2	IC50	28.0	nM	10.1021/np070431w
Homo sapiens	Serine/threonine-protein kinase PIM2	IC50	345.0	nM	10.1021/jm801242y
Homo sapiens	Serine/threonine-protein kinase PIM2	Kd	1.9	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PIM2	Kd	1.9	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PIM2	Kd	4.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PIM2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PIM2	Residual Activity	8.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PIM3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PIM3	IC50	0.0885	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PIM3	IC50	0.0979	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PIM3	IC50	0.1206	nM	10.1016/j.bmcl.2017.02.068
Homo sapiens	Serine/threonine-protein kinase PIM3	Kd	0.51	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PIM3	Kd	0.51	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PIM3	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PIM3	Residual Activity	5.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PLK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PLK1	IC50	0.92	ug.mL-1	10.1016/j.bmc.2012.10.014
Homo sapiens	Serine/threonine-protein kinase PLK1	IC50	76.9	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PLK1	IC50	192.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Serine/threonine-protein kinase PLK1	IC50	222.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PLK1	IC50	317.9	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Serine/threonine-protein kinase PLK1	IC50	540.0	nM	10.1021/np4005745
Homo sapiens	Serine/threonine-protein kinase PLK1	IC50	864.6	nM	10.1016/j.ejmech.2017.11.058
Homo sapiens	Serine/threonine-protein kinase PLK1	IC50	864.6	nM	10.1016/j.ejmech.2019.111769
Homo sapiens	Serine/threonine-protein kinase PLK1	IC50	22400.0	nM	10.1016/j.bmc.2012.11.054
Homo sapiens	Serine/threonine-protein kinase PLK1	IC50	129000.0	nM	10.1016/j.bmc.2012.11.054
Homo sapiens	Serine/threonine-protein kinase PLK1	Inhibition	58.0	%	10.1016/j.ejmech.2017.05.049
Homo sapiens	Serine/threonine-protein kinase PLK1	Inhibition	58.0	%	10.1016/j.ejmech.2018.02.070
Homo sapiens	Serine/threonine-protein kinase PLK1	Inhibition	95.0	%	10.1016/j.ejmech.2017.05.049
Homo sapiens	Serine/threonine-protein kinase PLK1	Inhibition	95.0	%	10.1016/j.ejmech.2018.02.070
Homo sapiens	Serine/threonine-protein kinase PLK1	Kd	190.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PLK1	Kd	190.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PLK1	Ratio IC50	5.0	None	10.1016/j.bmc.2012.11.054
Homo sapiens	Serine/threonine-protein kinase PLK1	Residual Activity	4.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PLK1	Residual Activity	53.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PLK2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PLK2	IC50	197.0	nM	10.1021/jm800861c
Homo sapiens	Serine/threonine-protein kinase PLK2	IC50	328.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PLK2	IC50	365.9	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Serine/threonine-protein kinase PLK2	IC50	471.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PLK2	IC50	957.2	nM	10.1016/j.ejmech.2017.11.058
Homo sapiens	Serine/threonine-protein kinase PLK2	IC50	957.2	nM	10.1016/j.ejmech.2019.111769
Homo sapiens	Serine/threonine-protein kinase PLK2	Kd	200.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PLK2	Residual Activity	28.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PLK2	Residual Activity	69.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PLK3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PLK3	IC50	182.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PLK3	IC50	224.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PLK3	IC50	10000.0	nM	10.1016/j.ejmech.2017.11.058
Homo sapiens	Serine/threonine-protein kinase PLK3	IC50	10000.0	nM	10.1016/j.ejmech.2019.111769
Homo sapiens	Serine/threonine-protein kinase PLK3	Kd	910.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PLK3	Kd	910.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PLK3	Residual Activity	50.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PLK3	Residual Activity	81.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PLK4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PLK4	IC50	7.17	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PLK4	IC50	9.49	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	0.75	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	0.77	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	0.77	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PRKX	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PRKX	IC50	1.39	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase PRKX	IC50	1.49	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase PRKX	Kd	13.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PRKX	Kd	13.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PRKX	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase PRP4 homolog	Kd	220.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RAF	IC50	130.0	nM	10.1016/j.ejmech.2015.08.027
Homo sapiens	Serine/threonine-protein kinase RAF	IC50	140.0	nM	10.1016/j.bmcl.2006.05.092
Homo sapiens	Serine/threonine-protein kinase RAF	IC50	240.0	nM	10.1016/j.ejmech.2018.03.013
Homo sapiens	Serine/threonine-protein kinase RAF	IC50	10000.0	nM	10.1021/jm801317h
Homo sapiens	Serine/threonine-protein kinase RAF	IC50	nan	None	10.1016/j.bmc.2017.09.003
Homo sapiens	Serine/threonine-protein kinase RAF	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase RAF	Inhibition	nan	%	10.1016/j.bmc.2012.04.006
Homo sapiens	Serine/threonine-protein kinase RAF	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase RAF	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RAF	Potency	177.8	nM	None
Homo sapiens	Serine/threonine-protein kinase RAF	Residual Activity	99.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase RAF	Residual Activity	109.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase RAF and Dual specificity mitogen-activated protein kinase kinase 1 (Raf/MEK)	IC50	2.5	nM	10.1021/jm0102856
Homo sapiens	Serine/threonine-protein kinase receptor R3	IC50	850.0	nM	10.1021/jm500115w
Homo sapiens	Serine/threonine-protein kinase receptor R3	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase receptor R3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase receptor R3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIO1	Kd	130.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase RIO1	Kd	130.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIO2	Kd	390.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIO3	Kd	76.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase RIO3	Kd	76.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIO3	Kd	76.0	nM	None
Homo sapiens	Serine/threonine-protein kinase RIO3	Kd	79.43	nM	None
Homo sapiens	Serine/threonine-protein kinase RIPK2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase RIPK2	IC50	317.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase RIPK2	IC50	395.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase RIPK2	Kd	5100.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase RIPK2	Kd	5200.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase RIPK2	Kd	5200.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIPK2	Residual Activity	12.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase RIPK2	Residual Activity	49.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase SBK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SBK1	IC50	99.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SBK1	IC50	193.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase SBK1	Kd	3.2	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Sgk1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Sgk1	IC50	6.75	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Sgk1	IC50	9.28	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Sgk1	IC50	14.0	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Serine/threonine-protein kinase Sgk1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Sgk1	Residual Activity	8.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Sgk2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Sgk2	IC50	15.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Sgk2	IC50	16.5	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Sgk2	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Sgk2	Residual Activity	11.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Sgk3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Sgk3	IC50	69.6	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase Sgk3	IC50	76.5	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase Sgk3	Kd	3.4	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Sgk3	Residual Activity	8.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase Sgk3	Residual Activity	42.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase SIK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SIK1	IC50	0.458	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase SIK1	IC50	1.34	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SIK1	Kd	2.2	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase SIK1	Kd	2.2	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SIK1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase SIK1	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase SIK2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SIK2	IC50	0.345	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase SIK2	IC50	0.37	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SIK2	IC50	1100.0	nM	10.1021/acs.jmedchem.0c02144
Homo sapiens	Serine/threonine-protein kinase SIK2	Kd	1.1	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase SIK2	Kd	1.1	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SIK3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SIK3	IC50	0.972	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase SIK3	IC50	1.24	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SIK3	IC50	460.0	nM	10.1021/acs.jmedchem.0c02144
Homo sapiens	Serine/threonine-protein kinase SIK3	Kd	0.46	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SRPK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SRPK1	IC50	24.5	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SRPK1	IC50	42.8	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase SRPK1	Kd	5.5	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase SRPK1	Kd	5.5	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SRPK1	Residual Activity	-3.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase SRPK1	Residual Activity	11.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase SRPK2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SRPK2	IC50	185.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase SRPK2	IC50	227.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SRPK2	Kd	67.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase SRPK2	Kd	67.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SRPK2	Residual Activity	12.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase SRPK2	Residual Activity	49.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase SRPK3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SRPK3	IC50	1580.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase SRPK3	IC50	1960.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase SRPK3	Kd	73.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SRPK3	Residual Activity	40.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase SRPK3	Residual Activity	92.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase TAO1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase TAO1	IC50	0.469	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase TAO1	IC50	1.21	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase TAO1	Kd	0.45	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TAO1	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase TAO1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase TAO2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase TAO2	IC50	3.54	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase TAO2	IC50	11.7	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase TAO2	Kd	12.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TAO2	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase TAO2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase TAO3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase TAO3	IC50	1.25	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase TAO3	IC50	2.11	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase TAO3	Kd	0.22	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TAO3	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase TBK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase TBK1	IC50	2.18	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase TBK1	IC50	3.86	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase TBK1	Kd	0.89	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TBK1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase TBK1	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase TNNI3K	Kd	1000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase TNNI3K	Kd	1000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase tousled-like 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase tousled-like 1	IC50	21.7	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase tousled-like 1	IC50	30.4	nM	10.1016/j.ejmech.2018.11.037
Homo sapiens	Serine/threonine-protein kinase tousled-like 1	IC50	36.4	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase tousled-like 1	Kd	27.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase tousled-like 1	Kd	27.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase tousled-like 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase tousled-like 2	IC50	3.37	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase tousled-like 2	IC50	3.66	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase tousled-like 2	Inhibition	nan	%	10.1016/j.ejmech.2021.113904
Homo sapiens	Serine/threonine-protein kinase tousled-like 2	Kd	16.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase tousled-like 2	Kd	16.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase tousled-like 2	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase ULK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase ULK1	IC50	8.95	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase ULK1	IC50	10.3	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase ULK1	Kd	9.9	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase ULK2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase ULK2	IC50	2.67	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase ULK2	IC50	3.66	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase ULK2	Kd	0.79	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase ULK2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase ULK2	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase ULK3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase ULK3	IC50	1.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase ULK3	IC50	4.2	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase ULK3	Kd	1.2	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase ULK3	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase ULK3	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase VRK1	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase VRK2	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase VRK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase VRK2	Residual Activity	90.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase VRK2	Residual Activity	108.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase WEE1	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase WEE1	Kd	1600.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase WEE1	Kd	1600.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase WNK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase WNK1	IC50	12100.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase WNK1	IC50	17500.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase WNK2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase WNK2	IC50	1450.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase WNK2	IC50	1460.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase WNK2	Residual Activity	30.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase WNK2	Residual Activity	92.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase WNK3	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Serine/threonine-protein kinase WNK3	Residual Activity	42.0	%	10.1042/bj20121418
Homo sapiens	Serine/threonine-protein kinase WNK3	Residual Activity	88.0	%	10.1042/bj20121418
Homo sapiens	SF-268	GI50	44.0	nM	10.1021/np200041v
Homo sapiens	SH-SY5Y	Activity	2.63	%	10.1016/j.bmc.2015.12.007
Homo sapiens	SH-SY5Y	Activity	6.19	%	10.1016/j.bmc.2015.12.007
Homo sapiens	SH-SY5Y	Activity	9.4	%	10.1016/j.ejmech.2019.01.052
Homo sapiens	SH-SY5Y	Activity	14.49	%	10.1016/j.bmc.2015.12.007
Homo sapiens	SH-SY5Y	Activity	nan	None	10.1021/acs.jnatprod.7b00751
Homo sapiens	SNF-related serine/threonine-protein kinase	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	SNF-related serine/threonine-protein kinase	IC50	3.79	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	SNF-related serine/threonine-protein kinase	IC50	8.01	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	SNF-related serine/threonine-protein kinase	Kd	90.0	nM	10.1038/nbt.1990
Homo sapiens	SPS1/STE20-related protein kinase YSK4	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	SPS1/STE20-related protein kinase YSK4	IC50	1.85	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	SPS1/STE20-related protein kinase YSK4	IC50	15.6	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	SPS1/STE20-related protein kinase YSK4	Kd	0.86	nM	10.1038/nbt.1990
Homo sapiens	ST486	IC50	7.0	nM	10.1016/j.ejmech.2011.11.040
Homo sapiens	STE20/SPS1-related proline-alanine-rich protein kinase	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	STE20/SPS1-related proline-alanine-rich protein kinase	IC50	14.4	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	STE20/SPS1-related proline-alanine-rich protein kinase	IC50	17.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	STE20/SPS1-related proline-alanine-rich protein kinase	Kd	130.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Stem cell growth factor receptor	IC50	1.0	nM	10.1016/j.bmcl.2006.05.092
Homo sapiens	Stem cell growth factor receptor	IC50	3.6	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Stem cell growth factor receptor	IC50	4.1	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Stem cell growth factor receptor	IC50	4.5	nM	10.1016/j.bmc.2017.04.003
Homo sapiens	Stem cell growth factor receptor	IC50	23.0	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	Stem cell growth factor receptor	IC50	23.0	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Stem cell growth factor receptor	IC50	47.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Stem cell growth factor receptor	IC50	65.19	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Stem cell growth factor receptor	IC50	72.7	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Stem cell growth factor receptor	IC50	84.2	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Stem cell growth factor receptor	IC50	84.2	nM	10.1016/j.ejmech.2021.113511
Homo sapiens	Stem cell growth factor receptor	Inhibition	96.7	%	10.1021/jm070342g
Homo sapiens	Stem cell growth factor receptor	Inhibition	99.8	%	10.1016/j.ejmech.2015.04.018
Homo sapiens	Stem cell growth factor receptor	Kd	0.43	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	0.6	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	0.64	nM	10.1016/j.ejmech.2011.02.057
Homo sapiens	Stem cell growth factor receptor	Kd	0.64	nM	10.1038/nbt1358
Homo sapiens	Stem cell growth factor receptor	Kd	0.64	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	9.5	nM	10.1038/nbt1358
Homo sapiens	Stem cell growth factor receptor	Kd	9.5	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	15.0	nM	10.1038/nbt1358
Homo sapiens	Stem cell growth factor receptor	Kd	15.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	19.0	nM	10.1016/j.ejmech.2011.02.057
Homo sapiens	Stem cell growth factor receptor	Kd	19.0	nM	10.1038/nbt1358
Homo sapiens	Stem cell growth factor receptor	Kd	19.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	22.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	38.0	nM	10.1038/nbt1358
Homo sapiens	Stem cell growth factor receptor	Kd	38.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	100.0	nM	10.1038/nbt1068
Homo sapiens	Stem cell growth factor receptor	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Stem cell growth factor receptor	Residual Activity	10.0	%	10.1042/bj20121418
Homo sapiens	SUP-B15	Activity	0.2	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	SUP-B15	Activity	9.8	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	SUP-B15	Activity	10.0	%	10.1016/j.ejmech.2018.12.059
Homo sapiens	SUP-B15	Activity	39.4	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	SUP-B15	Activity	44.2	%	10.1016/j.ejmech.2018.01.004
Homo sapiens	SUP-B15	Activity	52.3	%	10.1016/j.ejmech.2018.12.059
Homo sapiens	SUP-B15	EC50	550.0	nM	10.1021/acs.jnatprod.8b00884
Homo sapiens	SW-1736	EC50	200.0	nM	10.1016/j.ejmech.2019.02.057
Homo sapiens	SW480	IC50	100.0	nM	10.1016/j.bmcl.2019.126807
Homo sapiens	T47D	Activity	0.1	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	T47D	Activity	0.4	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	T47D	Activity	0.6	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	T47D	Activity	2.4	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	T47D	Activity	2.5	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	T47D	Activity	3.5	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	T47D	Activity	4.8	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	T47D	Activity	5.5	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	T47D	Activity	6.2	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	T47D	Activity	88.4	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	T47D	Activity	90.6	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	T47D	Activity	95.0	%	10.1016/j.bmcl.2017.07.063
Homo sapiens	T47D	IC50	4520.0	nM	10.1016/j.ejmech.2020.112112
Homo sapiens	T47D	IC50	11700.0	nM	10.1016/j.bmc.2021.116168
Homo sapiens	TAK1/TAB1	IC50	39.0	nM	10.1021/acsmedchemlett.0c00547
Homo sapiens	Tau-tubulin kinase 1	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tau-tubulin kinase 2	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	Telomerase reverse transcriptase	IC50	3310.0	nM	10.1016/j.ejmech.2020.112994
Homo sapiens	Telomerase reverse transcriptase	IC50	4140.0	nM	10.1016/j.bmc.2012.08.059
Homo sapiens	Telomerase reverse transcriptase	IC50	8300.0	nM	10.1016/j.ejmech.2012.11.039
Homo sapiens	Telomerase reverse transcriptase	IC50	8320.0	nM	10.1016/j.bmc.2011.08.013
Homo sapiens	Telomerase reverse transcriptase	IC50	8500.0	nM	10.1016/j.ejmech.2016.09.011
Homo sapiens	Telomerase reverse transcriptase	IC50	8670.0	nM	10.1016/j.ejmech.2022.114255
Homo sapiens	Telomerase reverse transcriptase	IC50	8970.0	nM	10.1016/j.ejmech.2016.02.009
Homo sapiens	Telomerase reverse transcriptase	Inhibition	10.7	%	10.1016/j.ejmech.2014.11.027
Homo sapiens	Telomerase reverse transcriptase	Inhibition	11.3	%	10.1016/j.ejmech.2014.11.027
Homo sapiens	Telomerase reverse transcriptase	Inhibition	12.7	%	10.1016/j.ejmech.2014.11.027
Homo sapiens	Telomerase reverse transcriptase	Inhibition	15.4	%	10.1016/j.ejmech.2014.11.027
Homo sapiens	Telomerase reverse transcriptase	Inhibition	18.9	%	10.1016/j.ejmech.2014.11.027
Homo sapiens	Telomerase reverse transcriptase	Inhibition	28.7	%	10.1016/j.ejmech.2014.11.027
Homo sapiens	Telomerase reverse transcriptase	Inhibition	30.1	%	10.1016/j.ejmech.2014.11.027
Homo sapiens	Telomerase reverse transcriptase	Inhibition	40.1	%	10.1016/j.ejmech.2014.11.027
Homo sapiens	Telomerase reverse transcriptase	Inhibition	56.5	%	10.1016/j.ejmech.2014.11.027
Homo sapiens	Telomerase reverse transcriptase	Inhibition	nan	%	10.1016/j.ejmech.2014.11.027
Homo sapiens	TERT-RPE1	Activity	9.1	%	10.1016/j.ejmech.2019.01.052
Homo sapiens	TERT-RPE1	IC50	5.5	nM	10.1016/j.ejmech.2020.113003
Homo sapiens	TERT-RPE1	IC50	250.0	nM	10.1016/j.bmc.2019.02.005
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	IC50	0.0473	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	IC50	0.052	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	Kd	24.0	nM	10.1038/nbt1358
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	Kd	24.0	nM	10.1038/nbt.1990
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Testis-specific serine/threonine-protein kinase 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Testis-specific serine/threonine-protein kinase 2	IC50	3.32	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Testis-specific serine/threonine-protein kinase 2	IC50	4.32	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Testis-specific serine/threonine-protein kinase 2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Testis-specific serine/threonine-protein kinase 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Testis-specific serine/threonine-protein kinase 3	IC50	3.21	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Testis-specific serine/threonine-protein kinase 3	IC50	7.01	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Testis-specific serine/threonine-protein kinase 6	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Testis-specific serine/threonine-protein kinase 6	IC50	112.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Testis-specific serine/threonine-protein kinase 6	IC50	193.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	TGF-beta receptor type I	IC50	6870.0	nM	10.1016/j.bmcl.2012.12.008
Homo sapiens	TGF-beta receptor type I	IC50	18500.0	nM	10.1021/jm500115w
Homo sapiens	TGF-beta receptor type I	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	TGF-beta receptor type I	Kd	2000.0	nM	10.1038/nbt1358
Homo sapiens	TGF-beta receptor type I	Kd	2000.0	nM	10.1038/nbt.1990
Homo sapiens	TGF-beta receptor type I	Residual Activity	30.0	%	10.1042/bj20121418
Homo sapiens	TGF-beta receptor type I	Residual Activity	79.0	%	10.1042/bj20121418
Homo sapiens	TGF-beta receptor type II	IC50	nan	None	10.1016/j.ejmech.2018.10.052
Homo sapiens	TGF-beta receptor type II	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	TGF-beta receptor type II	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Thioredoxin reductase 1	IC50	43.18	nM	10.1016/j.ejmech.2021.113475
Homo sapiens	TRAF2- and NCK-interacting kinase	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	TRAF2- and NCK-interacting kinase	IC50	0.314	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	TRAF2- and NCK-interacting kinase	IC50	0.551	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	TRAF2- and NCK-interacting kinase	IC50	1.4	nM	10.1016/j.bmcl.2012.11.013
Homo sapiens	TRAF2- and NCK-interacting kinase	IC50	39.0	nM	10.1016/j.bmcl.2012.11.013
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	4.7	nM	10.1038/nbt1358
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	4.7	nM	10.1038/nbt.1990
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	6.0	nM	10.1038/nbt1068
Homo sapiens	TRAF2- and NCK-interacting kinase	Ratio IC50	28.0	None	10.1016/j.bmcl.2012.11.013
Homo sapiens	Transcription intermediary factor 1-alpha	Delta TM	-0.4	C	None
Homo sapiens	Transient receptor potential cation channel subfamily M member 6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Inhibition	nan	%	10.1016/j.bmcl.2011.11.064
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine kinase non-receptor protein 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine kinase non-receptor protein 2	IC50	24.9	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine kinase non-receptor protein 2	IC50	34.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine kinase non-receptor protein 2	Inhibition	96.4	%	10.1021/jm070342g
Homo sapiens	Tyrosine kinase non-receptor protein 2	Kd	16.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine kinase non-receptor protein 2	Kd	16.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine kinase non-receptor protein 2	Kd	17.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine kinase non-receptor protein 2	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine kinase non-receptor protein 2	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase ABL	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase ABL	Delta TM	9.51	C	None
Homo sapiens	Tyrosine-protein kinase ABL	IC50	21.7	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase ABL	IC50	30.0	nM	10.1021/jm020455u
Homo sapiens	Tyrosine-protein kinase ABL	IC50	35.18	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase ABL	IC50	54.1	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase ABL	IC50	76.0	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Tyrosine-protein kinase ABL	IC50	100.0	nM	10.1021/jm020143r
Homo sapiens	Tyrosine-protein kinase ABL	IC50	105.9	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Tyrosine-protein kinase ABL	IC50	136.0	nM	10.1021/jm800861c
Homo sapiens	Tyrosine-protein kinase ABL	IC50	196.2	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase ABL	IC50	210.0	nM	10.1016/j.bmc.2013.11.052
Homo sapiens	Tyrosine-protein kinase ABL	IC50	290.0	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Tyrosine-protein kinase ABL	IC50	339.0	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Tyrosine-protein kinase ABL	Inhibition	87.2	%	10.1021/jm070342g
Homo sapiens	Tyrosine-protein kinase ABL	Inhibition	94.6	%	10.1016/j.bmc.2011.06.022
Homo sapiens	Tyrosine-protein kinase ABL	Inhibition	94.87	%	10.1016/j.ejmech.2013.03.043
Homo sapiens	Tyrosine-protein kinase ABL	Inhibition	94.87	%	10.1016/j.ejmech.2013.07.056
Homo sapiens	Tyrosine-protein kinase ABL	Inhibition	96.9	%	10.1016/j.ejmech.2011.01.020
Homo sapiens	Tyrosine-protein kinase ABL	Inhibition	102.0	%	10.1016/j.bmc.2013.07.026
Homo sapiens	Tyrosine-protein kinase ABL	Kd	2.9	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	8.4	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	11.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	18.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	21.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	22.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	23.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	27.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	36.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	37.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	38.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Kd	46.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	52.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	91.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	130.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	170.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Kd	170.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	210.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	220.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	270.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	290.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	340.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Kd	400.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Kd	410.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Kd	500.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Kd	550.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	1000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	2800.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase ABL	Residual Activity	18.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase ABL2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase ABL2	IC50	10.1	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase ABL2	IC50	15.8	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase ABL2	IC50	75.9	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase ABL2	Inhibition	90.2	%	10.1016/j.ejmech.2011.01.020
Homo sapiens	Tyrosine-protein kinase ABL2	Kd	110.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL2	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL2	Kd	160.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL2	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase ABL2	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase BLK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase BLK	IC50	1.07	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase BLK	IC50	1.09	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase BLK	Inhibition	nan	%	10.1016/j.ejmech.2021.114051
Homo sapiens	Tyrosine-protein kinase BLK	Kd	15.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase BLK	Kd	15.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase BLK	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase BMX	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase BMX	IC50	2.99	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase BMX	IC50	6.16	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase BMX	Kd	170.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase BMX	Kd	170.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase BMX	Kd	410.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase BMX	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase BMX	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase BRK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase BRK	IC50	162.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase BRK	IC50	247.0	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase BRK	IC50	277.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase BRK	IC50	1250.0	nM	10.1016/j.ejmech.2013.11.039
Homo sapiens	Tyrosine-protein kinase BRK	Kd	2300.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase BRK	Kd	2300.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase BRK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase BRK	Residual Activity	6.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase BRK	Residual Activity	38.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase BTK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase BTK	IC50	13.38	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase BTK	IC50	17.2	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase BTK	IC50	18.1	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Tyrosine-protein kinase BTK	IC50	22.07	nM	None
Homo sapiens	Tyrosine-protein kinase BTK	IC50	23.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase BTK	IC50	36.0	nM	10.1021/jm800861c
Homo sapiens	Tyrosine-protein kinase BTK	IC50	65.0	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase BTK	IC50	100.0	nM	10.1021/acs.jmedchem.9b00113
Homo sapiens	Tyrosine-protein kinase BTK	IC50	15000.0	nM	10.1016/j.bmcl.2017.04.014
Homo sapiens	Tyrosine-protein kinase BTK	Inhibition	nan	%	10.1016/j.bmc.2016.05.031
Homo sapiens	Tyrosine-protein kinase BTK	Inhibition	nan	%	10.1021/acs.jmedchem.9b01916
Homo sapiens	Tyrosine-protein kinase BTK	Kd	210.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase BTK	Kd	210.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase BTK	Kd	710.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase BTK	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase BTK	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase CSK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase CSK	IC50	7.12	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase CSK	IC50	14.3	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase CSK	Inhibition	89.3	%	10.1021/jm070342g
Homo sapiens	Tyrosine-protein kinase CSK	Kd	330.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase CSK	Kd	330.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase CSK	Kd	440.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase CSK	Residual Activity	4.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase CSK	Residual Activity	29.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase CTK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase CTK	IC50	392.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase CTK	IC50	492.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase CTK	Kd	260.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FER	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase FER	IC50	0.203	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase FER	IC50	0.365	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase FER	IC50	1.8	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase FER	Kd	24.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FER	Kd	24.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FER	Kd	30.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase FER	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase FER	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase FES	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase FES	IC50	1.52	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase FES	IC50	2.08	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase FES	IC50	8.1	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase FES	Kd	23.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FES	Kd	23.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FES	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase FGR	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase FGR	IC50	0.658	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase FGR	IC50	1.15	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase FGR	Kd	17.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FGR	Kd	17.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FGR	Kd	30.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase FGR	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase FRK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase FRK	IC50	4.56	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase FRK	IC50	17.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase FRK	Kd	45.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FRK	Kd	45.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FRK	Kd	260.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase FRK	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase FRK	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase FYN	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase FYN	IC50	1.1	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase FYN	IC50	2.0	nM	10.1016/j.bmcl.2009.10.038
Homo sapiens	Tyrosine-protein kinase FYN	IC50	2.06	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase FYN	IC50	4.4	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase FYN	IC50	5.0	nM	10.1021/jm0607202
Homo sapiens	Tyrosine-protein kinase FYN	IC50	15.0	nM	10.1021/jm0607202
Homo sapiens	Tyrosine-protein kinase FYN	IC50	36.0	nM	10.1021/jm0607202
Homo sapiens	Tyrosine-protein kinase FYN	IC50	83.0	nM	10.1021/jm0607202
Homo sapiens	Tyrosine-protein kinase FYN	IC50	270.0	nM	10.1021/jm0607202
Homo sapiens	Tyrosine-protein kinase FYN	IC50	510.0	nM	10.1021/jm0607202
Homo sapiens	Tyrosine-protein kinase FYN	Kd	33.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FYN	Kd	33.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FYN	Kd	51.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase FYN	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase HCK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase HCK	IC50	1.9	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase HCK	IC50	3.03	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase HCK	Kd	12.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase HCK	Kd	20.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase HCK	Kd	20.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase HCK	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase HCK	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase HCK	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase ITK/TSK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase ITK/TSK	IC50	3.59	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase ITK/TSK	IC50	4.02	nM	None
Homo sapiens	Tyrosine-protein kinase ITK/TSK	IC50	10.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase ITK/TSK	IC50	12.02	nM	None
Homo sapiens	Tyrosine-protein kinase ITK/TSK	IC50	12.81	nM	None
Homo sapiens	Tyrosine-protein kinase ITK/TSK	IC50	16000.0	nM	10.1016/j.bmcl.2017.04.014
Homo sapiens	Tyrosine-protein kinase ITK/TSK	Kd	19.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ITK/TSK	Kd	19.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ITK/TSK	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase ITK/TSK	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase JAK1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase JAK1	IC50	0.627	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase JAK1	IC50	0.631	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase JAK1	IC50	1.0	nM	None
Homo sapiens	Tyrosine-protein kinase JAK1	IC50	1.01	nM	None
Homo sapiens	Tyrosine-protein kinase JAK1	IC50	3.0	nM	10.1016/j.bmc.2016.04.030
Homo sapiens	Tyrosine-protein kinase JAK1	IC50	3.0	nM	10.1021/acsmedchemlett.6b00247
Homo sapiens	Tyrosine-protein kinase JAK1	IC50	12.5	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase JAK1	Inhibition	97.0	%	10.1016/j.bmc.2016.04.030
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	6.1	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase JAK2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase JAK2	IC50	0.115	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase JAK2	IC50	0.189	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase JAK2	IC50	0.31	nM	10.1016/j.ejmech.2016.03.074
Homo sapiens	Tyrosine-protein kinase JAK2	IC50	0.4	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase JAK2	IC50	1.0	nM	None
Homo sapiens	Tyrosine-protein kinase JAK2	IC50	2.0	nM	10.1016/j.bmc.2016.04.030
Homo sapiens	Tyrosine-protein kinase JAK2	IC50	2.0	nM	10.1016/j.ejmech.2013.11.036
Homo sapiens	Tyrosine-protein kinase JAK2	IC50	2.0	nM	10.1021/acsmedchemlett.6b00247
Homo sapiens	Tyrosine-protein kinase JAK2	IC50	2.3	nM	10.1016/j.bmc.2014.12.026
Homo sapiens	Tyrosine-protein kinase JAK2	IC50	4.7	nM	10.1021/jm800861c
Homo sapiens	Tyrosine-protein kinase JAK2	Inhibition	95.0	%	10.1016/j.bmc.2016.04.030
Homo sapiens	Tyrosine-protein kinase JAK2	Kd	9.8	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase JAK2	Kd	11.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase JAK2	Kd	11.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase JAK2	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase JAK2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	0.0913	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	0.1	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	0.12	nM	10.1021/acs.jnatprod.7b01082
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	0.138	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	0.15	nM	10.1021/jm800861c
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	0.184	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	0.5	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	1.0	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	1.0	nM	10.1016/j.bmc.2016.04.030
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	1.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	1.0	nM	10.1021/acsmedchemlett.6b00247
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	1.0	nM	None
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	6.0	nM	10.1016/j.bmcl.2006.10.062
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	6.0	nM	10.1016/j.bmcl.2009.04.039
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	8.0	nM	10.1016/j.ejmech.2021.113674
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	100.0	nM	10.1016/j.bmcl.2017.04.014
Homo sapiens	Tyrosine-protein kinase JAK3	Inhibition	95.3	%	10.1021/jm070342g
Homo sapiens	Tyrosine-protein kinase JAK3	Inhibition	98.0	%	10.1016/j.bmc.2016.04.030
Homo sapiens	Tyrosine-protein kinase JAK3	Kd	10.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase JAK3	Kd	12.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase JAK3	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase LCK	Activity	0.77	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase LCK	Activity	0.9	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase LCK	Activity	1.71	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase LCK	Activity	4.02	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase LCK	Activity	4.17	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase LCK	Activity	14.7	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase LCK	Activity	27.22	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase LCK	Activity	56.02	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase LCK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase LCK	Activity	70.13	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase LCK	Activity	87.83	%	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase LCK	IC50	1.01	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase LCK	IC50	1.33	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Tyrosine-protein kinase LCK	IC50	1.4	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase LCK	IC50	1.5	nM	10.1016/j.bmcl.2009.10.038
Homo sapiens	Tyrosine-protein kinase LCK	IC50	1.57	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase LCK	IC50	1.8	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase LCK	IC50	2.65	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase LCK	IC50	2.68	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Tyrosine-protein kinase LCK	IC50	3.73	ug.mL-1	10.1016/j.bmc.2012.10.014
Homo sapiens	Tyrosine-protein kinase LCK	IC50	4.0	nM	10.1021/jm800861c
Homo sapiens	Tyrosine-protein kinase LCK	IC50	4.49	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Tyrosine-protein kinase LCK	IC50	18.0	nM	10.1016/j.bmc.2008.06.017
Homo sapiens	Tyrosine-protein kinase LCK	IC50	2100.0	nM	10.1021/jm00053a003
Homo sapiens	Tyrosine-protein kinase LCK	Inhibition	89.0	%	10.1016/j.bmcl.2017.11.040
Homo sapiens	Tyrosine-protein kinase LCK	Kd	20.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase LCK	Kd	30.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase LCK	Kd	30.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase LCK	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase LCK	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase LCK	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase LCK	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase Lyn	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase Lyn	IC50	0.473	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase Lyn	IC50	0.49	nM	10.1021/jm800861c
Homo sapiens	Tyrosine-protein kinase Lyn	IC50	0.728	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase Lyn	IC50	0.805	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase Lyn	IC50	0.964	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase Lyn	IC50	1.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Tyrosine-protein kinase Lyn	IC50	1.0	nM	10.1016/j.ejmech.2021.113511
Homo sapiens	Tyrosine-protein kinase Lyn	IC50	1.3	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Tyrosine-protein kinase Lyn	IC50	1.3	nM	10.1016/j.bmcl.2009.10.038
Homo sapiens	Tyrosine-protein kinase Lyn	IC50	1.39	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Tyrosine-protein kinase Lyn	IC50	2.1	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase Lyn	IC50	2.68	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase Lyn	Inhibition	nan	%	10.1016/j.bmcl.2019.01.019
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	40.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	40.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	210.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase Lyn	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase Lyn	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	0.18	nM	10.1016/j.bmcl.2011.10.076
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	0.2	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	0.2	nM	10.1021/acs.jmedchem.6b00374
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	0.254	nM	10.1016/j.bmc.2021.116596
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	0.259	nM	10.1016/j.bmc.2021.116596
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	0.52	nM	10.1016/j.bmc.2017.04.003
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	0.71	nM	10.1016/j.ejmech.2018.06.010
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	0.755	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	0.83	nM	10.1016/j.ejmech.2018.06.010
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	1.0	nM	10.1016/j.ejmech.2014.07.108
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	1.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	1.0	nM	10.1016/j.ejmech.2021.113511
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	1.0	nM	10.1021/jm800861c
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	1.01	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	1.15	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	1.52	nM	10.1016/j.ejmech.2018.06.010
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	1.74	nM	10.1016/j.ejmech.2018.06.010
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	1.78	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	1.96	nM	10.1016/j.ejmech.2018.06.010
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	2.03	nM	10.1016/j.ejmech.2018.06.010
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	3.44	nM	10.1016/j.ejmech.2020.112710
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	4.95	nM	10.1016/j.ejmech.2018.06.010
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	5.49	nM	10.1016/j.ejmech.2018.06.010
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	nan	None	10.1016/j.bmc.2017.09.003
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	96.4	%	10.1021/jm070342g
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	99.9	%	10.1016/j.ejmech.2015.04.018
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	100.0	%	10.1016/j.bmcl.2012.10.016
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.22	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	1.8	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.1	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.1	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.4	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.4	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.5	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.5	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.9	nM	10.1021/jm401094t
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.9	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.9	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	3.3	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	nan	None	10.1016/j.ejmech.2018.06.010
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase receptor RET	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	0.46	nM	10.1021/jm800861c
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	0.82	nM	10.1016/j.ejmech.2020.112755
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	1.27	nM	10.1016/j.ejmech.2020.112755
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	1.29	nM	10.1016/j.ejmech.2020.112755
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	1.39	nM	10.1016/j.ejmech.2020.112755
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	1.69	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	2.03	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	3.43	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	4.6	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	4.7	nM	10.1016/j.bmc.2017.04.003
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	12.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	15.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	15.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	28.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	28.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor RET	Residual Activity	3.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase receptor RET	Residual Activity	9.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase receptor Tie-1	Kd	65.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor Tie-1	Kd	65.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	IC50	1.45	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	IC50	2.75	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	IC50	48.99	nM	10.1016/j.ejmech.2010.04.026
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Inhibition	95.3	%	10.1021/jm070342g
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Kd	280.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Kd	280.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase receptor UFO	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase receptor UFO	IC50	3.0	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase receptor UFO	IC50	3.9	nM	10.1016/j.bmcl.2018.10.013
Homo sapiens	Tyrosine-protein kinase receptor UFO	IC50	7.65	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase receptor UFO	IC50	11.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase receptor UFO	IC50	40.0	nM	10.1021/np4005745
Homo sapiens	Tyrosine-protein kinase receptor UFO	Kd	6.8	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor UFO	Kd	6.8	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor UFO	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase receptor UFO	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase SRC	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase SRC	IC50	0.83	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Tyrosine-protein kinase SRC	IC50	1.0	nM	10.1016/s0960-894x(03)00286-5
Homo sapiens	Tyrosine-protein kinase SRC	IC50	1.0	nM	10.1021/jm950588y
Homo sapiens	Tyrosine-protein kinase SRC	IC50	1.3	nM	10.1021/jm800861c
Homo sapiens	Tyrosine-protein kinase SRC	IC50	2.2	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase SRC	IC50	2.59	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase SRC	IC50	2.6	nM	10.1021/acs.jnatprod.7b01082
Homo sapiens	Tyrosine-protein kinase SRC	IC50	2.91	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase SRC	IC50	3.12	nM	10.1016/j.ejmech.2020.112710
Homo sapiens	Tyrosine-protein kinase SRC	IC50	3.78	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Tyrosine-protein kinase SRC	IC50	4.7	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase SRC	IC50	5.0	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Tyrosine-protein kinase SRC	IC50	6.3	nM	10.1038/nchembio.162
Homo sapiens	Tyrosine-protein kinase SRC	IC50	8.8	nM	10.1016/j.ejmech.2018.03.013
Homo sapiens	Tyrosine-protein kinase SRC	IC50	9.7	nM	10.1016/j.ejmech.2015.08.027
Homo sapiens	Tyrosine-protein kinase SRC	IC50	40.0	nM	10.1021/np4005745
Homo sapiens	Tyrosine-protein kinase SRC	IC50	70.0	nM	10.1021/jm020143r
Homo sapiens	Tyrosine-protein kinase SRC	IC50	300.0	nM	10.1016/j.bmc.2012.09.057
Homo sapiens	Tyrosine-protein kinase SRC	IC50	300.0	nM	10.1016/j.bmcl.2010.10.121
Homo sapiens	Tyrosine-protein kinase SRC	IC50	300.0	nM	10.1016/j.bmcl.2011.01.047
Homo sapiens	Tyrosine-protein kinase SRC	IC50	350.0	nM	10.1016/0960-894X(94)80004-9
Homo sapiens	Tyrosine-protein kinase SRC	IC50	600.0	nM	10.1016/j.bmcl.2011.10.124
Homo sapiens	Tyrosine-protein kinase SRC	IC50	600.0	nM	10.1016/j.bmcl.2013.03.124
Homo sapiens	Tyrosine-protein kinase SRC	IC50	1920.0	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	Tyrosine-protein kinase SRC	IC50	1920.0	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Tyrosine-protein kinase SRC	IC50	3000.0	nM	10.1021/jm00053a003
Homo sapiens	Tyrosine-protein kinase SRC	Inhibition	89.8	%	10.1021/jm070342g
Homo sapiens	Tyrosine-protein kinase SRC	Inhibition	99.36	%	10.1016/j.bmc.2011.04.053
Homo sapiens	Tyrosine-protein kinase SRC	Kd	8.0	nM	10.1038/nchembio.162
Homo sapiens	Tyrosine-protein kinase SRC	Kd	86.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase SRC	Kd	86.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase SRC	Kd	100.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase SRC	Residual Activity	-2.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase SRC	Residual Activity	8.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase Srms	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase Srms	IC50	4230.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase Srms	IC50	8770.0	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase Srms	Kd	740.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase Srms	Kd	740.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase SYK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase SYK	IC50	0.1	nM	10.1021/jm800861c
Homo sapiens	Tyrosine-protein kinase SYK	IC50	0.133	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase SYK	IC50	0.217	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase SYK	IC50	0.45	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase SYK	IC50	1.0	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Tyrosine-protein kinase SYK	IC50	1.0	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Tyrosine-protein kinase SYK	IC50	1.0	nM	10.1016/j.ejmech.2021.113511
Homo sapiens	Tyrosine-protein kinase SYK	IC50	1.08	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Tyrosine-protein kinase SYK	IC50	1.3	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase SYK	IC50	1.3	nM	10.1016/j.ejmech.2021.113393
Homo sapiens	Tyrosine-protein kinase SYK	IC50	3.0	nM	10.1016/j.bmc.2008.09.015
Homo sapiens	Tyrosine-protein kinase SYK	IC50	3.0	nM	10.1016/j.bmcl.2009.02.049
Homo sapiens	Tyrosine-protein kinase SYK	IC50	60.0	nM	10.1016/j.ejmech.2013.11.036
Homo sapiens	Tyrosine-protein kinase SYK	Inhibition	90.2	%	10.1021/jm070342g
Homo sapiens	Tyrosine-protein kinase SYK	Inhibition	97.3	%	10.1016/j.ejmech.2021.113393
Homo sapiens	Tyrosine-protein kinase SYK	Kd	7.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase SYK	Kd	14.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase SYK	Kd	14.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase SYK	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase SYK	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase TEC	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase TEC	IC50	24.6	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase TEC	IC50	43.1	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase TEC	IC50	128000.0	nM	10.1016/j.bmcl.2017.04.014
Homo sapiens	Tyrosine-protein kinase TEC	Inhibition	92.5	%	10.1021/jm070342g
Homo sapiens	Tyrosine-protein kinase TEC	Kd	1300.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase TEC	Kd	1300.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TEC	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase TEC	Residual Activity	19.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase TIE-2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase TIE-2	IC50	29.9	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase TIE-2	IC50	50.9	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Tyrosine-protein kinase TIE-2	IC50	52.0	nM	10.1021/jm800861c
Homo sapiens	Tyrosine-protein kinase TIE-2	IC50	65.5	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase TIE-2	IC50	213.2	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase TIE-2	IC50	59500000.0	nM	10.1016/j.bmc.2018.10.004
Homo sapiens	Tyrosine-protein kinase TIE-2	Inhibition	90.9	%	10.1021/jm070342g
Homo sapiens	Tyrosine-protein kinase TIE-2	Kd	140.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase TIE-2	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TIE-2	Kd	240.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase TIE-2	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase TIE-2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase TXK	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase TXK	IC50	19.1	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase TXK	IC50	21.6	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase TXK	Kd	230.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase TXK	Kd	230.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TXK	Residual Activity	4.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase TXK	Residual Activity	21.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase TYK2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase TYK2	IC50	0.205	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase TYK2	IC50	0.234	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase TYK2	IC50	0.351	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Tyrosine-protein kinase TYK2	IC50	0.6	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase TYK2	IC50	66.9	nM	10.1016/j.ejmech.2020.112277
Homo sapiens	Tyrosine-protein kinase TYK2	Kd	56.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase TYK2	Kd	56.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TYK2	Kd	3100.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase YES	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase YES	IC50	2.35	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Tyrosine-protein kinase YES	IC50	2.39	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase YES	IC50	2.56	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase YES	IC50	4.4	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Tyrosine-protein kinase YES	Kd	49.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase YES	Kd	52.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase YES	Kd	52.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase YES	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase ZAP-70	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase ZAP-70	IC50	1.1	nM	10.1016/j.ejmech.2021.113393
Homo sapiens	Tyrosine-protein kinase ZAP-70	IC50	1.3	nM	10.1021/acs.jnatprod.7b01082
Homo sapiens	Tyrosine-protein kinase ZAP-70	IC50	3.29	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase ZAP-70	IC50	7.35	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Tyrosine-protein kinase ZAP-70	IC50	8.63	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Tyrosine-protein kinase ZAP-70	IC50	12.4	nM	10.1016/j.bmc.2017.02.030
Homo sapiens	Tyrosine-protein kinase ZAP-70	IC50	53.0	nM	10.1016/j.bmc.2008.06.017
Homo sapiens	Tyrosine-protein kinase ZAP-70	IC50	53.0	nM	10.1016/j.bmc.2008.09.015
Homo sapiens	Tyrosine-protein kinase ZAP-70	Inhibition	102.1	%	10.1016/j.ejmech.2021.113393
Homo sapiens	Tyrosine-protein kinase ZAP-70	Kd	44.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ZAP-70	Kd	44.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ZAP-70	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Tyrosine-protein kinase ZAP-70	Residual Activity	6.0	%	10.1042/bj20121418
Homo sapiens	U-251	Activity	nan	None	10.1021/acs.jmedchem.5b00686
Homo sapiens	U2OS	Activity	0.4	%	10.1016/j.ejmech.2019.01.052
Homo sapiens	U2OS	Activity	22.6	%	10.1021/acs.jnatprod.7b00064
Homo sapiens	U2OS	Control DMSO Apoptotic Cells (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Apoptotic Cells (%)	24.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Apoptotic Cells (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Apoptotic Cells (%)	31.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Apoptotic Cells (%)	35.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Apoptotic Cells (%)	36.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Apoptotic Cells (%)	37.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Apoptotic Cells (%)	43.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Apoptotic Cells (%)	50.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Apoptotic Cells (%)	52.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Apoptotic Cells (%)	59.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	3.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	4.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	6.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	11.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	13.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	17.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Fragmented Nuclei %	39.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Growth Rate	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Growth Rate	1.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	54.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	70.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	70.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	73.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	77.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	78.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	81.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	81.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	82.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	83.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	86.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	87.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	87.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	88.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	89.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	90.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Healthy Nuclei (%)	91.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	1.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	2.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	3.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	9.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Membrane Permeable-Phenotype Cells (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	1.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	21.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	24.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitochondria Different-Phenotype Cells (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	32.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	39.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	40.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	42.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	47.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	48.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	49.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	50.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	52.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	56.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	60.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	62.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	62.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	63.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	64.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	68.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	73.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Mitotic Cells (%)	75.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	6.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	7.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	8.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	11.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	12.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	13.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Pyknosed Nuclei (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	33.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Total Cells	43.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Total Cells	54.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Total Cells	70.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	78.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	92.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Total Cells	99.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	102.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	139.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	149.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Total Cells	152.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	153.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	156.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	165.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	178.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	199.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	212.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	255.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Total Cells	276.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	330.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Total Cells	361.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Total Cells	732.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	1.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	7.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	19.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	28.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	31.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	64.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	69.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	70.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	91.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	92.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Control DMSO Tubulin Phenotype Different Cells (%)	93.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Growth Rate	0.49	None	10.6019/CHEMBL5058564
Homo sapiens	U2OS	Growth Rate	0.65	None	10.6019/CHEMBL5058564
Homo sapiens	U2OS	Growth Rate	0.69	None	10.6019/CHEMBL5058564
Homo sapiens	U2OS	Growth Rate	0.79	None	10.6019/CHEMBL5058564
Homo sapiens	U2OS	Population Apoptotic (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	25.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	30.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	38.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	38.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	40.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	43.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	45.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	50.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	51.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	53.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	56.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	58.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	59.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	62.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	70.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	71.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	72.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	73.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	77.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	83.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	85.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	86.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	86.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	87.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	87.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	88.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	88.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	89.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	89.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	90.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	91.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Apoptotic (%)	93.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	94.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	95.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	96.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Apoptotic (%)	100.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	1.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	9.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	13.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	17.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	21.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	22.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	24.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	26.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	27.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	30.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	34.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	34.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	38.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	40.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	40.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	41.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	42.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	43.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	45.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	45.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	46.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	47.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	48.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	50.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	51.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	53.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	55.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	58.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	64.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	65.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Fragmented Nuclei (%)	67.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	1.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	3.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Healthy Nuclei (%)	4.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Healthy Nuclei (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	5.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Healthy Nuclei (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	6.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Healthy Nuclei (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	8.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Healthy Nuclei (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	11.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Healthy Nuclei (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	19.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Healthy Nuclei (%)	22.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	37.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	38.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Healthy Nuclei (%)	46.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	49.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	56.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	56.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Healthy Nuclei (%)	71.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	77.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	81.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Healthy Nuclei (%)	83.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Healthy Nuclei (%)	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	86.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	87.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	88.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Healthy Nuclei (%)	91.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	1.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	3.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	14.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	15.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	25.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Hoechst High Intensity Objects (%)	27.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	2.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	17.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	20.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	33.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	43.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	53.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	62.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	66.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	71.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	85.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	87.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	89.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	90.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	92.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	94.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	95.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	96.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	97.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	100.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Membrane Permeable-Phenotype (%)	100.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	1.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	17.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	45.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	50.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	51.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	53.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	56.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	57.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	57.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	60.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	66.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	66.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	68.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	69.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	71.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	71.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	75.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	75.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	80.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	83.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	85.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	92.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	95.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	96.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	100.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitochondria Different-Phenotype (%)	100.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	0.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	3.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	5.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	8.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	10.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	12.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	12.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	13.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	13.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	14.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	16.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	22.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	26.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	27.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	28.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	30.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	37.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	40.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	41.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	43.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	46.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	48.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	50.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	54.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	56.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	60.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	61.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	61.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Mitotic Cells (%)	66.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	69.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	75.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	83.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Mitotic Cells (%)	100.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Normal (%)	72.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	73.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	74.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	81.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	84.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	85.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	86.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	88.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	91.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	92.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	93.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	94.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	95.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	96.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	96.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Normal (%)	97.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Normal (%)	98.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Normal (%)	99.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Normal (%)	100.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	2.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	4.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	4.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	5.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	6.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	7.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	7.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	8.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	9.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	11.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	18.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	23.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	28.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	29.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	30.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	31.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	36.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	38.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	38.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	40.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	42.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	43.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	45.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	46.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	47.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	48.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	50.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	50.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	52.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	57.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	58.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	60.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	61.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	63.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	68.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	70.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	73.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Pyknosed Nuclei (%)	80.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	0.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	2.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	9.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	10.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	17.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	20.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	25.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	33.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	36.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	40.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	43.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	44.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	49.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	50.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	68.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	73.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	85.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	89.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	91.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	92.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	93.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	94.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	95.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	96.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	100.0	%	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Population Tubulin-Different-Phenotype (%)	100.0	%	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	16.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	20.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	26.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	27.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	50.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	57.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	58.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	58.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	64.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	72.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	78.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	81.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	82.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	86.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	92.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	93.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	95.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	101.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	121.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	131.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	133.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	138.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	141.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	148.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	164.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	167.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	176.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	177.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	184.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	186.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	232.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	234.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	264.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	264.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	265.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	339.0	None	10.6019/CHEMBL5303300
Homo sapiens	U2OS	Total Cell Count	342.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	351.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	363.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	379.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Total Cell Count	434.0	None	10.6019/CHEMBL4689842
Homo sapiens	U-87 MG	IC50	20.0	nM	10.1016/j.bmcl.2020.127109
Homo sapiens	U-937	IC50	2000.0	nM	10.1016/j.bmc.2006.10.035
Homo sapiens	Uncharacterized aarF domain-containing protein kinase 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Uncharacterized aarF domain-containing protein kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	UoC-B1	EC50	2000.0	nM	10.1021/acs.jnatprod.8b00884
Homo sapiens	Vascular endothelial growth factor receptor 1	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Vascular endothelial growth factor receptor 1	IC50	5.4	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Vascular endothelial growth factor receptor 1	IC50	6.31	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Vascular endothelial growth factor receptor 1	IC50	8.19	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Vascular endothelial growth factor receptor 1	IC50	14.7	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Vascular endothelial growth factor receptor 1	IC50	15.97	nM	10.1016/j.ejmech.2018.06.010
Homo sapiens	Vascular endothelial growth factor receptor 1	IC50	19.0	nM	10.1021/jm800861c
Homo sapiens	Vascular endothelial growth factor receptor 1	IC50	35.0	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	93.4	%	10.1016/j.bmc.2011.06.022
Homo sapiens	Vascular endothelial growth factor receptor 1	Kd	11.0	nM	10.1021/acsmedchemlett.3c00127
Homo sapiens	Vascular endothelial growth factor receptor 1	Kd	150.0	nM	10.1038/nbt1358
Homo sapiens	Vascular endothelial growth factor receptor 1	Kd	150.0	nM	10.1038/nbt.1990
Homo sapiens	Vascular endothelial growth factor receptor 1	Residual Activity	-1.0	%	10.1042/bj20121418
Homo sapiens	Vascular endothelial growth factor receptor 1	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Vascular endothelial growth factor receptor 2	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	1.2	nM	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	1.67	nM	10.1016/j.ejmech.2018.06.010
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	2.1	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	3.4	nM	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	3.5	nM	10.1016/j.ejmech.2015.06.029
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	3.5	nM	10.1021/jm800861c
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	3.8	nM	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	3.85	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	4.1	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	4.8	nM	10.1016/j.bmc.2017.04.003
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	6.0	nM	10.1016/j.bmc.2015.08.010
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	8.0	nM	10.1021/jm300576q
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	10.0	nM	10.1021/np4005745
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	10.36	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	10.7	nM	10.1016/j.ejmech.2015.08.031
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	11.0	nM	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	11.7	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	13.73	nM	10.1016/j.bmc.2011.09.042
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	14.0	nM	10.1016/s0960-894x(03)00644-9
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	15.97	nM	10.1021/acs.jmedchem.7b01091
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	32.2	nM	10.1016/j.bmc.2021.116454
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	70.0	nM	10.1021/jm901388c
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	72.0	nM	10.1016/j.bmc.2016.09.021
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	72.0	nM	10.1016/j.bmc.2017.09.003
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	72.0	nM	10.1016/j.bmcl.2016.10.029
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	80.0	nM	10.1021/jm020143r
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	88.0	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	88.0	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	330.0	nM	10.1016/j.bmc.2020.115328
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	500.0	nM	10.1039/D1MD00125F
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	19000.0	nM	10.1016/j.bmcl.2017.04.014
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	78.1	%	10.1016/j.ejmech.2015.04.018
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	82.0	%	10.1016/j.bmc.2016.03.008
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	85.0	%	10.1016/j.ejmech.2012.09.039
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	87.85	%	10.1039/D1MD00125F
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	91.8	%	10.1021/jm070342g
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	92.9	%	10.1016/j.bmc.2011.06.022
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	96.44	%	10.1016/j.bmc.2011.06.022
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	99.24	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	99.58	%	10.1016/j.bmc.2011.04.053
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	100.26	%	10.1016/j.bmc.2013.07.026
Homo sapiens	Vascular endothelial growth factor receptor 2	Kd	220.0	nM	10.1038/nbt1358
Homo sapiens	Vascular endothelial growth factor receptor 2	Kd	220.0	nM	10.1038/nbt.1990
Homo sapiens	Vascular endothelial growth factor receptor 2	Kd	270.0	nM	10.1038/nbt1068
Homo sapiens	Vascular endothelial growth factor receptor 2	Ki	1.7	nM	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	Ki	nan	None	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Vascular endothelial growth factor receptor 2	Residual Activity	2.0	%	10.1042/bj20121418
Homo sapiens	Vascular endothelial growth factor receptor 2	T1/2	0.08333	hr	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 3	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
Homo sapiens	Vascular endothelial growth factor receptor 3	IC50	0.7	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Vascular endothelial growth factor receptor 3	IC50	0.9	nM	10.1016/j.bmc.2016.05.057
Homo sapiens	Vascular endothelial growth factor receptor 3	IC50	1.9	nM	10.1021/jm800861c
Homo sapiens	Vascular endothelial growth factor receptor 3	IC50	2.29	nM	10.1016/j.ejmech.2017.10.003
Homo sapiens	Vascular endothelial growth factor receptor 3	IC50	2.69	nM	10.1016/j.ejmech.2018.10.052
Homo sapiens	Vascular endothelial growth factor receptor 3	IC50	3.27	nM	10.1016/j.ejmech.2018.06.010
Homo sapiens	Vascular endothelial growth factor receptor 3	IC50	3.8	nM	10.1016/j.ejmech.2018.02.080
Homo sapiens	Vascular endothelial growth factor receptor 3	IC50	58.0	nM	10.1016/j.bmcl.2005.12.017
Homo sapiens	Vascular endothelial growth factor receptor 3	IC50	58.0	nM	10.1016/j.bmcl.2005.12.065
Homo sapiens	Vascular endothelial growth factor receptor 3	Kd	28.0	nM	10.1038/nbt1358
Homo sapiens	Vascular endothelial growth factor receptor 3	Kd	28.0	nM	10.1038/nbt.1990
Homo sapiens	Vascular endothelial growth factor receptor 3	Kd	31.0	nM	10.1038/nbt1068
Homo sapiens	Vascular endothelial growth factor receptor 3	Residual Activity	0.0	%	10.1042/bj20121418
Homo sapiens	Vascular endothelial growth factor receptor 3	Residual Activity	1.0	%	10.1042/bj20121418
Homo sapiens	Wee1-like protein kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	WI-38	IC50	24410.0	nM	10.1016/j.bmcl.2021.128258
Homo sapiens	WI-38	IC50	nan	None	10.1021/acs.jmedchem.6b00374
Homo sapiens	Z-138	IC50	6.7	nM	10.1016/j.ejmech.2020.113003
Homo sapiens	Z-138	IC50	18.0	nM	10.1016/j.bmcl.2019.04.023
Homo sapiens	Z-138	IC50	20.0	nM	10.1021/acsmedchemlett.0c00269
Homo sapiens	Z-138	IC50	41.8	nM	10.1016/j.ejmech.2021.113727
Homo sapiens	Z-138	IC50	21500.0	nM	10.1016/j.bmc.2019.02.005
Ilyonectria destructans	Ilyonectria destructans	MIC	100.0	ug.mL-1	10.1021/jf0532617
Mus musculus	B16-F10	Activity	0.461	%	10.1016/j.ejmech.2016.01.003
Mus musculus	B16-F10	Activity	22.2	%	10.1016/j.ejmech.2016.01.003
Mus musculus	B16-F10	Activity	33.9	%	10.1016/j.ejmech.2016.01.003
Mus musculus	B16-F10	Activity	43.5	%	10.1016/j.ejmech.2016.01.003
Mus musculus	B16-F10	FC	21.0	None	10.1016/j.ejmech.2016.01.003
Mus musculus	B16-F10	IC50	2820.0	nM	10.1016/j.bmc.2012.03.040
Mus musculus	Casein kinase 2	IC50	10000.0	nM	10.1021/jm049478u
Mus musculus	Cyclin-dependent kinase 1	IC50	8.0	nM	10.1021/jm049478u
Mus musculus	Epidermal growth factor receptor erbB1	IC50	0.35	ug.mL-1	10.1021/np50066a009
Mus musculus	Epidermal growth factor receptor erbB1	IC50	10000.0	nM	10.1021/jm049478u
Mus musculus	Insulin receptor	IC50	200.0	nM	10.1021/jm049478u
Mus musculus	L929	Activity	nan	None	10.1021/np960581z
Mus musculus	L929	IC50	200.0	nM	10.1021/acs.jnatprod.7b00236
Mus musculus	MAP kinase ERK2	IC50	10000.0	nM	10.1021/jm049478u
Mus musculus	MEF	Activity	nan	None	10.1016/j.ejmech.2012.09.012
Mus musculus	Mus musculus	Activity	-2.0	g	10.1016/j.bmc.2006.09.063
Mus musculus	Mus musculus	Activity	-1.0	g	10.1016/j.bmc.2006.09.063
Mus musculus	Mus musculus	Activity	-0.6	g	10.1016/j.bmc.2006.09.063
Mus musculus	N2a	Activity	1.3	%	10.1016/j.ejmech.2016.12.057
Mus musculus	N2a	IC50	11.3	nM	10.1016/j.ejmech.2016.12.057
Mus musculus	NIH3T3	EC50	8.0	nM	10.1016/j.ejmech.2017.11.046
Mus musculus	NIH3T3	EC50	8.0	nM	10.1016/j.ejmech.2019.02.057
Mus musculus	NIH3T3	EC50	8.0	nM	10.1016/j.ejmech.2020.112920
Mus musculus	NIH3T3	IC50	8.0	nM	10.1016/j.ejmech.2020.112425
Mus musculus	NIH3T3	IC50	200.0	nM	10.1016/j.ejmech.2013.11.025
Mus musculus	NIH3T3	IC50	140120.0	nM	10.1016/j.bmc.2013.11.004
Mus musculus	P388	ED50	0.08	ug ml-1	10.1021/np50059a012
Mus musculus	Platelet-derived growth factor receptor	IC50	2.0	nM	10.1021/jm049478u
Mus musculus	Serine/threonine-protein kinase MST2	Kd	0.15	nM	10.1038/nbt1068
Mus musculus	Splenocyte	IC50	400.0	nM	10.1016/S0960-894X(01)80995-1
Mus musculus	Testis-specific serine/threonine-protein kinase 1	IC50	0.33	nM	10.1016/j.ejmech.2016.03.074
Mus musculus	Tyrosine-protein kinase BLK	IC50	400.0	nM	10.1016/0960-894X(94)00458-R
Mus musculus	ULK3 kinase	Kd	3.0	nM	10.1038/nbt1068
Mycobacterium tuberculosis	Mycobacterium tuberculosis	MIC	14700.0	nM	10.1016/j.bmc.2009.08.061
Mycobacterium tuberculosis	Serine/threonine-protein kinase pknB	Kd	88.0	nM	10.1038/nbt.1990
Pectobacterium carotovorum	Pectobacterium carotovorum	MIC	100.0	ug.mL-1	10.1021/jf0532617
Phytophthora capsici	Phytophthora capsici	Activity	nan	None	10.1021/jf0532617
Phytophthora capsici	Phytophthora capsici	MIC	1.0	ug.mL-1	10.1021/jf0532617
Plasmodium falciparum	Calcium-dependent protein kinase 1	Kd	0.25	nM	10.1038/nbt.1990
Plasmodium falciparum	Plasmodium falciparum	EC50	nan	None	10.1016/j.bmcl.2014.09.061
Plasmodium falciparum	Plasmodium falciparum	IC50	0.0	nM	10.1016/j.bmc.2010.01.068
Plasmodium falciparum	Plasmodium falciparum	IC50	150.0	nM	10.1021/jm0300983
Plasmodium falciparum	Plasmodium falciparum	IC50	190.0	nM	10.1021/jm0300983
Plasmodium falciparum	Plasmodium falciparum	IC50	nan	None	10.1038/nchembio.87
Plasmodium falciparum	Protein kinase Pfmrk	IC50	4000.0	nM	10.1021/jm0300983
Plasmodium falciparum	Protein kinase Pfmrk	IC50	4000.0	nM	10.1021/jm040108f
Plasmodium falciparum (isolate 3D7)	Cell division control protein 2 homolog	Kd	800.0	nM	10.1038/nbt.1990
Pyricularia grisea	Pyricularia grisea	MIC	100.0	ug.mL-1	10.1021/jf0532617
Ralstonia solanacearum	Ralstonia solanacearum	MIC	100.0	ug.mL-1	10.1021/jf0532617
Rattus norvegicus	cAMP-dependent protein kinase alpha-catalytic subunit	IC50	18.0	nM	10.1021/jm00079a024
Rattus norvegicus	cAMP-dependent protein kinase alpha-catalytic subunit	IC50	27.0	nM	10.1021/jm00113a038
Rattus norvegicus	cAMP-dependent protein kinase alpha-catalytic subunit	IC50	120.0	nM	10.1021/jm00079a024
Rattus norvegicus	Dual specificity tyrosine-phosphorylation-regulated kinase 1A	IC50	12.0	nM	10.1016/j.ejmech.2021.113554
Rattus norvegicus	Glycogen synthase kinase-3 beta	IC50	15.0	nM	10.1016/j.ejmech.2021.113445
Rattus norvegicus	PC-12	Activity	100.0	%	10.1021/jm200982p
Rattus norvegicus	PC-12	RFU	6000.0	None	10.1016/j.bmc.2013.06.037
Rattus norvegicus	PC-12	RFU	30000.0	None	10.1016/j.bmc.2013.06.037
Rattus norvegicus	Protein kinase C gamma	IC50	9.0	nM	10.1021/jm00079a024
Rattus norvegicus	Protein kinase C (PKC)	IC50	3.0	nM	10.1021/jm00079a024
Rattus norvegicus	Protein kinase C (PKC)	IC50	3.0	nM	10.1021/jm9702037
Rattus norvegicus	Protein kinase C (PKC)	IC50	6.0	nM	10.1016/S0960-894X(01)80356-5
Rattus norvegicus	Protein kinase C (PKC)	IC50	8.0	nM	10.1016/S0960-894X(00)80013-X
Rattus norvegicus	Protein kinase C (PKC)	IC50	9.0	nM	10.1016/0960-894X(94)00458-R
Rattus norvegicus	Protein kinase C (PKC)	IC50	9.0	nM	10.1016/S0960-894X(01)80995-1
Rattus norvegicus	Protein kinase C (PKC)	IC50	9.0	nM	10.1021/jm00053a003
Rattus norvegicus	Protein kinase C (PKC)	IC50	9.0	nM	10.1021/jm00079a024
Rattus norvegicus	Protein kinase C (PKC)	IC50	10.0	nM	10.1016/s0960-894x(99)00375-3
Rattus norvegicus	Protein kinase C (PKC)	IC50	190.0	nM	10.1016/s0960-894x(03)00286-5
Rattus norvegicus	Protein kinase C (PKC)	IC50	190.0	nM	10.1021/jm950588y
Rattus norvegicus	Protein kinase C (PKC)	IC50	300.0	nM	10.1016/j.bmcl.2019.126886
Rattus norvegicus	Protein kinase C (PKC)	IC50	500.0	nM	10.1016/j.bmcl.2019.126886
Rattus norvegicus	Protein kinase C (PKC)	IC50	800.0	nM	10.1016/j.bmcl.2019.126886
Rattus norvegicus	Protein kinase C (PKC)	IC50	1000.0	nM	10.1016/j.bmcl.2019.126886
Rattus norvegicus	Protein kinase C, PKC; classical	IC50	2.7	nM	10.1021/jm00113a038
Rattus norvegicus	Protein kinase C, PKC; classical	IC50	9.0	nM	10.1021/jm00053a003
Rattus norvegicus	Rattus norvegicus	Inhibition	45.0	%	10.1016/S0960-894X(01)80408-X
Rattus norvegicus	RBL-2H3	IC50	200.0	nM	10.1016/j.bmcl.2019.01.019
Rattus norvegicus	RBL-2H3	IC50	300.0	nM	10.1016/j.bmcl.2019.01.019
Rattus norvegicus	RBL-2H3	IC50	700.0	nM	10.1016/j.bmcl.2019.01.019
Rattus norvegicus	RBL-2H3	IC50	1000.0	nM	10.1016/j.bmcl.2019.01.019
Rattus norvegicus	RBL-2H3	Inhibition	nan	%	10.1016/j.bmcl.2019.01.019
Rattus norvegicus	Tubulin alpha-1 chain	Kd	770.0	nM	10.1038/nbt1358
Rhizoctonia solani	Rhizoctonia solani	MIC	1.0	ug.mL-1	10.1021/jf0532617
Saccharomyces cerevisiae	Saccharomyces cerevisiae	MIC	1.0	ug.mL-1	10.1021/jf0532617
Schistosoma mansoni	Schistosoma mansoni	EC50	203.0	nM	10.6019/CHEMBL5096127
Schistosoma mansoni	Schistosoma mansoni	In vitro activity	nan	None	10.6019/CHEMBL5096127
Schistosoma mansoni	Schistosoma mansoni	Worm movement inhibition	99.77	%	10.6019/CHEMBL5096127
Sclerotinia sclerotiorum	Sclerotinia sclerotiorum	MIC	100.0	ug.mL-1	10.1021/jf0532617
Stagonosporopsis cucurbitacearum	Stagonosporopsis cucurbitacearum	MIC	10.0	ug.mL-1	10.1021/jf0532617
Streptomyces	Streptomyces	IZ	13.0	mm	10.1021/np0603424
Sus scrofa	Tubulin	Activity	nan	None	10.1021/np50059a012
Xanthomonas vesicatoria	Xanthomonas vesicatoria	MIC	50.0	ug.mL-1	10.1021/jf0532617
None	ADMET	Activity	nan	None	10.1016/j.bmcl.2009.01.025
None	ADMET	Activity	nan	None	10.1016/j.ejmech.2016.02.034
None	ADMET	Inhibition	16.0	%	10.1016/j.ejmech.2014.07.064
None	ADMET	Inhibition	80.0	%	10.1016/j.ejmech.2014.07.064
None	ADMET	Inhibition	90.0	%	10.1016/j.ejmech.2014.07.064
None	ADMET	Selectivity Index	nan	None	10.1021/acs.jmedchem.1c01411
None	ADMET	Tox50	0.02	uM	10.1021/jm950588y
None	NON-PROTEIN TARGET	AC50	7790.0	nM	None
None	NON-PROTEIN TARGET	AC50	17430.0	nM	None
None	NON-PROTEIN TARGET	AC50	26770.0	nM	None
None	NON-PROTEIN TARGET	Activity	nan	None	10.1016/j.bmc.2014.06.032
None	NON-PROTEIN TARGET	Activity	nan	None	10.1016/j.bmcl.2012.06.077
None	NON-PROTEIN TARGET	Activity	nan	None	10.1038/nchembio809
None	NON-PROTEIN TARGET	EC50	24.92	ug.mL-1	10.1016/j.bmcl.2011.08.039
None	NON-PROTEIN TARGET	IC50	7.0	nM	10.1016/s0960-894x(01)00535-2
None	NON-PROTEIN TARGET	IC50	31.0	nM	10.1021/jm501942m
None	NON-PROTEIN TARGET	IC50	130.0	nM	10.1021/np400838a
None	NON-PROTEIN TARGET	IC50	200.0	nM	10.1016/j.ejmech.2013.11.025
None	NON-PROTEIN TARGET	IC50	380.0	nM	10.1021/np400838a
None	NON-PROTEIN TARGET	IC50	4950.0	nM	10.1016/j.bmc.2012.08.059
None	NON-PROTEIN TARGET	Inhibition	100.0	%	10.1016/j.ejmech.2013.10.049
None	NON-PROTEIN TARGET	Inhibition	101.0	%	10.1016/j.ejmech.2013.10.049
None	NON-PROTEIN TARGET	Inhibition	106.0	%	10.1016/j.ejmech.2013.10.049
None	NON-PROTEIN TARGET	Ratio EC50	nan	None	10.1016/j.bmcl.2014.09.061
None	No relevant target	LogP	nan	None	10.1016/j.ejmech.2012.09.039
None	No relevant target	permeability	nan	None	10.1016/j.ejmech.2017.06.020
None	No relevant target	solubility	nan	None	10.1016/j.bmc.2008.09.015
None	Unchecked	AbsAC40_uM	0.0107	uM	None
None	Unchecked	AbsAC40_uM	0.243	uM	None
None	Unchecked	AbsAC40_uM	0.809	uM	None
None	Unchecked	AbsAC40_uM	1.45	uM	None
None	Unchecked	AC50	11.4	nM	None
None	Unchecked	AC50	70000.0	nM	None
None	Unchecked	Activity	0.08	%	10.1128/aac.00126-08
None	Unchecked	Activity	14.54	%	10.1128/aac.00126-08
None	Unchecked	Activity	23.83	%	10.1128/aac.00126-08
None	Unchecked	Activity	61.57	%	10.1128/aac.00126-08
None	Unchecked	Activity	63.9	%	10.1021/jm8001185
None	Unchecked	Activity	65.0	%	10.1016/j.ejmech.2018.10.052
None	Unchecked	Activity	nan	None	10.1021/acs.jmedchem.1c00874
None	Unchecked	Activity	nan	None	10.1021/acs.jmedchem.2c01471
None	Unchecked	Activity	nan	None	10.1021/acsmedchemlett.9b00530
None	Unchecked	Activity	nan	None	10.1021/acsmedchemlett.9b00614
None	Unchecked	Activity	nan	None	10.1021/np50059a012
None	Unchecked	Activity	nan	None	10.1074/jbc.m609885200
None	Unchecked	deltaTm	4.5	K	10.1021/acs.jmedchem.1c00845
None	Unchecked	Delta Tm	4.0	degrees C	10.1021/acs.jmedchem.0c00898
None	Unchecked	EC50	20.0	nM	10.1021/jm950588y
None	Unchecked	EC50	350.0	nM	10.1021/acs.jnatprod.8b00884
None	Unchecked	EC50	nan	nM	10.1016/s0960-894x(03)00644-9
None	Unchecked	ED50	7.5	uM	10.1021/jm950588y
None	Unchecked	FC	0.6	None	10.1016/j.ejmech.2018.01.004
None	Unchecked	FC	0.7	None	10.1016/j.ejmech.2018.01.004
None	Unchecked	IC50	0.00047	ug.mL-1	10.1021/np50089a001
None	Unchecked	IC50	0.0011	ug.mL-1	10.1021/np50066a009
None	Unchecked	IC50	0.0024	ug.mL-1	10.1021/np50089a001
None	Unchecked	IC50	0.0031	ug.mL-1	10.1021/np50089a001
None	Unchecked	IC50	0.01	ug.mL-1	10.1021/np50066a009
None	Unchecked	IC50	0.2	nM	10.1016/j.ejmech.2020.113003
None	Unchecked	IC50	0.31	nM	10.1021/jm800861c
None	Unchecked	IC50	0.386	nM	10.1016/j.bmc.2018.02.022
None	Unchecked	IC50	0.5	nM	10.1021/jm00053a003
None	Unchecked	IC50	0.66	nM	10.1016/j.ejmech.2017.10.003
None	Unchecked	IC50	0.7	nM	10.1073/pnas.0708800104
None	Unchecked	IC50	1.0	nM	10.1208/aapsj080125
None	Unchecked	IC50	2.2	nM	10.1021/acs.jnatprod.7b01082
None	Unchecked	IC50	2.5	nM	10.1021/jm00053a003
None	Unchecked	IC50	2.52	nM	10.1016/j.ejmech.2021.113511
None	Unchecked	IC50	2.6	nM	10.1016/j.bmc.2009.07.056
None	Unchecked	IC50	2.93	nM	10.1016/j.ejmech.2018.10.052
None	Unchecked	IC50	3.0	nM	10.1016/0960-894X(94)80004-9
None	Unchecked	IC50	3.0	nM	10.1016/S0960-894X(01)80408-X
None	Unchecked	IC50	4.0	nM	10.1021/jm049478u
None	Unchecked	IC50	4.0	nM	10.1021/jm950588y
None	Unchecked	IC50	4.9	nM	10.1021/acsmedchemlett.0c00420
None	Unchecked	IC50	5.0	nM	10.1016/0960-894X(94)80004-9
None	Unchecked	IC50	5.0	nM	10.1016/j.ejmech.2021.113318
None	Unchecked	IC50	5.0	ug.mL-1	10.1021/np990171l
None	Unchecked	IC50	6.0	nM	10.1016/j.ejmech.2021.113318
None	Unchecked	IC50	6.0	nM	10.1021/jm049478u
None	Unchecked	IC50	6.6	nM	10.1016/j.bmcl.2022.128991
None	Unchecked	IC50	7.0	nM	10.1073/pnas.0708800104
None	Unchecked	IC50	8.2	nM	10.1016/j.ejmech.2016.03.074
None	Unchecked	IC50	8.5	nM	10.1073/pnas.0708800104
None	Unchecked	IC50	10.0	nM	10.1016/j.bmc.2014.12.026
None	Unchecked	IC50	10.0	nM	10.1016/j.ejmech.2021.113445
None	Unchecked	IC50	12.0	nM	10.1016/j.ejmech.2018.02.080
None	Unchecked	IC50	12.0	nM	10.1021/jm049478u
None	Unchecked	IC50	14.0	nM	10.1021/jm049478u
None	Unchecked	IC50	15.0	nM	10.1016/j.tips.2004.07.006
None	Unchecked	IC50	16.0	nM	10.1016/j.ejmech.2020.113003
None	Unchecked	IC50	20.0	nM	10.1016/j.ejmech.2021.113318
None	Unchecked	IC50	20.0	nM	10.1016/s0960-894x(98)00468-5
None	Unchecked	IC50	23.0	nM	10.1016/j.bmcl.2019.04.023
None	Unchecked	IC50	26.0	nM	10.1016/j.ejmech.2013.11.036
None	Unchecked	IC50	26.0	ug.mL-1	10.1021/np50066a009
None	Unchecked	IC50	30.0	nM	10.1016/j.bmc.2012.03.061
None	Unchecked	IC50	30.0	nM	10.1021/acsmedchemlett.0c00269
None	Unchecked	IC50	30.8	nM	10.1016/j.ejmech.2021.113727
None	Unchecked	IC50	39.0	nM	10.1016/j.bmcl.2019.04.023
None	Unchecked	IC50	40.0	nM	10.1016/0960-894X(94)00458-R
None	Unchecked	IC50	40.0	nM	10.1021/jm00079a024
None	Unchecked	IC50	46.0	nM	10.1021/jm701575k
None	Unchecked	IC50	49.1	nM	10.1016/j.ejmech.2021.113727
None	Unchecked	IC50	60.1	nM	10.1016/j.ejmech.2020.112277
None	Unchecked	IC50	80.0	nM	10.1021/jm020455u
None	Unchecked	IC50	100.0	nM	10.1016/s0960-894x(03)00286-5
None	Unchecked	IC50	100.0	nM	10.1021/jm950588y
None	Unchecked	IC50	121.0	nM	10.1021/jm00053a003
None	Unchecked	IC50	240.0	nM	10.1038/nchembio.87
None	Unchecked	IC50	600.0	nM	10.1021/acs.jnatprod.8b00103
None	Unchecked	IC50	1400.0	nM	10.1021/jm049478u
None	Unchecked	IC50	2000.0	nM	10.1016/j.bmc.2008.07.007
None	Unchecked	IC50	2800.0	nM	10.1021/acs.jnatprod.7b00236
None	Unchecked	IC50	3550.0	nM	10.1016/j.bmc.2019.02.005
None	Unchecked	IC50	4180.0	nM	10.1016/j.bmc.2013.11.004
None	Unchecked	IC50	7000.0	nM	10.1021/jm00053a003
None	Unchecked	IC50	7620.0	nM	10.1042/bj20030674
None	Unchecked	IC50	11320.0	nM	10.1016/j.bmc.2012.03.040
None	Unchecked	IC50	14000.0	nM	10.1016/s0960-894x(03)00286-5
None	Unchecked	IC50	14000.0	nM	10.1021/jm950588y
None	Unchecked	IC50	14220.0	nM	10.1042/bj20030674
None	Unchecked	IC50	21500.0	nM	10.1016/j.bmc.2019.02.005
None	Unchecked	IC50	28230.0	nM	10.1042/bj20030674
None	Unchecked	IC50	nan	nM	10.1021/jm00053a003
None	Unchecked	Inhibition	nan	%	10.1021/acs.jmedchem.9b01658
None	Unchecked	Inhibition	nan	%	10.1021/jm3001532
None	Unchecked	Inhibition	nan	%	10.1038/nchembio.87
None	Unchecked	Inhibition	nan	%	10.1039/D1MD00125F
None	Unchecked	Ki	5.0	nM	10.1016/j.bmc.2008.07.007
None	Unchecked	Potency	1000.0	nM	None
None	Unchecked	Potency	28183.8	nM	None
None	Unchecked	Ratio	0.5	None	10.1042/bj20030674
None	Unchecked	Ratio	1.9	None	10.1042/bj20030674
None	Unchecked	Ratio IC50	0.04	None	10.1016/j.ejmech.2020.112425
None	Unchecked	Ratio IC50	0.08	None	10.1016/j.ejmech.2020.112425
None	Unchecked	Ratio IC50	0.4	None	10.1021/jm801317h
None	Unchecked	Ratio IC50	0.8	None	10.1021/jm801317h
None	Unchecked	Ratio IC50	0.87	None	10.1016/j.bmcl.2014.05.085
None	Unchecked	Ratio IC50	0.9	None	10.1016/j.ejmech.2017.11.058
None	Unchecked	Ratio IC50	1.0	None	10.1021/jm801317h
None	Unchecked	Ratio IC50	1.1	None	10.1021/jm801317h
None	Unchecked	Ratio IC50	1.107	None	10.1016/j.ejmech.2019.111769
None	Unchecked	Ratio IC50	1.2	None	10.1021/jm801317h
None	Unchecked	Ratio IC50	2.0	None	10.1021/jm801317h
None	Unchecked	Ratio IC50	4.3	None	10.1016/j.bmcl.2020.127288
None	Unchecked	Ratio IC50	5.4	None	10.1021/jm801317h
None	Unchecked	Ratio IC50	10.0	None	10.1021/jm801242y
None	Unchecked	Ratio IC50	10.45	None	10.1016/j.ejmech.2017.11.058
None	Unchecked	Ratio IC50	11.0	None	10.1016/j.bmc.2011.02.036
None	Unchecked	Ratio IC50	11.57	None	10.1016/j.ejmech.2019.111769
None	Unchecked	Ratio IC50	30.0	None	10.1021/jm801317h

Metabolism Information

AKRT ID	Reaction	Reaction Link ID
AKRT010864	CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1O)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4.C[SAH]>>CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4	2.1.1.139-RXN