6-{2-[(4-ethyl-2,3-dioxopiperazine-1-carbonyl)amino]-2-phenylacetamido}-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid

AlkaPlorer ID: AK013680

Synonym: None

IUPAC Name: (2S,5R,6R)-6-[[(2R)-2-[(4-ethyl-2,3-dioxopiperazine-1-carbonyl)amino]-2-phenylacetyl]amino]-3,3-dimethyl-7-oxo-4-thia-1-azabicyclo[3.2.0]heptane-2-carboxylic acid

Structure

SMILES: CCN1CCN(C(=O)N[C@@H](C(=O)N[C@@H]2C(=O)N3[C@@H]2SC(C)(C)[C@@H]3C(=O)O)C2=CC=CC=C2)C(=O)C1=O

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InChI: InChI=1S/C23H27N5O7S/c1-4-26-10-11-27(19(32)18(26)31)22(35)25-13(12-8-6-5-7-9-12)16(29)24-14-17(30)28-15(21(33)34)23(2,3)36-20(14)28/h5-9,13-15,20H,4,10-11H2,1-3H3,(H,24,29)(H,25,35)(H,33,34)/t13-,14-,15+,20-/m1/s1

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InChIKey: IVBHGBMCVLDMKU-GXNBUGAJSA-N

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Properties Information

Molecule Weight: 517.5640000000003

TPSA: 156.43

MolLogP: -0.2402999999999968

Number of H-Donors: 3

Number of H-Acceptors: 7

RingCount: 4

Activities Information

Organism Target Name Standard Type Standard Value Standard Units doi
Acinetobacter Acinetobacter Activity 0.0 % 10.1128/aac.00149-08
Acinetobacter Acinetobacter Activity 0.0 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter Activity 3.9 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter Activity 18.1 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter Activity 21.3 % 10.1128/aac.00149-08
Acinetobacter Acinetobacter Activity 29.8 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter Activity 52.1 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter Activity 68.1 % 10.1128/aac.00149-08
Acinetobacter Acinetobacter Activity 87.5 % 10.1128/aac.00149-08
Acinetobacter Acinetobacter Activity 96.1 % 10.1128/aac.00381-08
Acinetobacter Acinetobacter MIC 0.25 ug.mL-1 10.1128/aac.00381-08
Acinetobacter Acinetobacter MIC 0.5 ug.mL-1 10.1128/aac.00149-08
Acinetobacter Acinetobacter MIC 32.0 ug.mL-1 10.1128/aac.00149-08
Acinetobacter Acinetobacter MIC 64.0 ug.mL-1 10.1128/aac.00381-08
Acinetobacter Acinetobacter MIC50 8.0 ug.mL-1 10.1128/aac.00149-08
Acinetobacter Acinetobacter MIC50 16.0 ug.mL-1 10.1128/aac.00381-08
Acinetobacter Acinetobacter MIC50 64.0 ug.mL-1 10.1128/aac.00149-08
Acinetobacter Acinetobacter MIC50 128.0 ug.mL-1 10.1128/aac.00381-08
Acinetobacter Acinetobacter MIC90 64.0 ug.mL-1 10.1128/aac.00149-08
Acinetobacter Acinetobacter MIC90 128.0 ug.mL-1 10.1128/aac.00381-08
Acinetobacter baumannii Acinetobacter baumannii Activity 9.0 % 10.1128/aac.01581-07
Acinetobacter baumannii Acinetobacter baumannii Activity 10.0 % 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii Activity 12.0 % 10.1128/aac.00400-09
Acinetobacter baumannii Acinetobacter baumannii Activity 17.2 % 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii Activity 71.4 % 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii Activity 76.0 % 10.1128/aac.00400-09
Acinetobacter baumannii Acinetobacter baumannii Activity 82.9 % 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii Activity nan None 10.1128/aac.00764-10
Acinetobacter baumannii Acinetobacter baumannii MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1128/aac.00400-09
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter baumannii Acinetobacter baumannii MIC 3.0 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.00050-10
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.00856-09
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.01164-08
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.01407-08
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.01581-07
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1039/C5MD00377F
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.00856-09
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 12.0 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.00050-10
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.00856-09
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.01164-08
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.01197-09
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.01398-09
Acinetobacter baumannii Acinetobacter baumannii MIC 24.0 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.00838-06
Acinetobacter baumannii Acinetobacter baumannii MIC 48.0 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 64.0 ug.mL-1 10.1039/C5MD00377F
Acinetobacter baumannii Acinetobacter baumannii MIC 64.0 ug.mL-1 10.1128/aac.00267-07
Acinetobacter baumannii Acinetobacter baumannii MIC 125.0 ug.mL-1 10.1128/aac.00366-08
Acinetobacter baumannii Acinetobacter baumannii MIC 128.0 ug.mL-1 10.1128/aac.00050-10
Acinetobacter baumannii Acinetobacter baumannii MIC 128.0 ug.mL-1 10.1128/aac.00414-10
Acinetobacter baumannii Acinetobacter baumannii MIC 128.0 ug.mL-1 10.1128/aac.00838-06
Acinetobacter baumannii Acinetobacter baumannii MIC 128.0 ug.mL-1 10.1128/aac.01139-06
Acinetobacter baumannii Acinetobacter baumannii MIC 128.0 ug.mL-1 10.1128/aac.01164-08
Acinetobacter baumannii Acinetobacter baumannii MIC 128.0 ug.mL-1 10.1128/aac.01398-09
Acinetobacter baumannii Acinetobacter baumannii MIC 256.0 ug.mL-1 10.1128/aac.00050-10
Acinetobacter baumannii Acinetobacter baumannii MIC 256.0 ug.mL-1 10.1128/aac.00267-07
Acinetobacter baumannii Acinetobacter baumannii MIC 256.0 ug.mL-1 10.1128/aac.00856-09
Acinetobacter baumannii Acinetobacter baumannii MIC 256.0 ug.mL-1 10.1128/aac.00861-09
Acinetobacter baumannii Acinetobacter baumannii MIC 256.0 ug.mL-1 10.1128/aac.01164-08
Acinetobacter baumannii Acinetobacter baumannii MIC 256.0 ug.mL-1 10.1128/aac.01198-06
Acinetobacter baumannii Acinetobacter baumannii MIC 256.0 ug.mL-1 10.1128/aac.01512-06
Acinetobacter baumannii Acinetobacter baumannii MIC 512.0 ug.mL-1 10.1128/aac.00072-08
Acinetobacter baumannii Acinetobacter baumannii MIC50 4.0 ug.mL-1 10.1128/aac.00400-09
Acinetobacter baumannii Acinetobacter baumannii MIC50 125.0 ug.mL-1 10.1128/aac.00366-08
Acinetobacter baumannii Acinetobacter baumannii MIC50 128.0 ug.mL-1 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter baumannii Acinetobacter baumannii MIC50 128.0 ug.mL-1 10.1128/aac.01197-09
Acinetobacter baumannii Acinetobacter baumannii MIC50 128.0 ug.mL-1 10.1128/aac.01581-07
Acinetobacter baumannii Acinetobacter baumannii MIC90 128.0 ug.mL-1 10.1128/aac.00264-10
Acinetobacter baumannii Acinetobacter baumannii MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter baumannii Acinetobacter baumannii MIC90 128.0 ug.mL-1 10.1128/aac.01197-09
Acinetobacter baumannii Acinetobacter baumannii MIC90 128.0 ug.mL-1 10.1128/aac.01581-07
Acinetobacter baumannii Acinetobacter baumannii MIC90 250.0 ug.mL-1 10.1128/aac.00366-08
Acinetobacter baumannii Acinetobacter baumannii MIC90 512.0 ug.mL-1 10.1128/aac.00400-09
Acinetobacter baumannii ADC-11 Kcat 5.0 /s 10.1128/aac.00050-10
Acinetobacter baumannii ADC-11 Kcat/Km 0.2 /uM/s 10.1128/aac.00050-10
Acinetobacter baumannii ADC-11 Km 25000.0 nM 10.1128/aac.00050-10
Acinetobacter baumannii Beta-lactamase ADC-33 Kcat 4.0 /s 10.1128/aac.00050-10
Acinetobacter baumannii Beta-lactamase ADC-33 Kcat/Km 0.25 /uM/s 10.1128/aac.00050-10
Acinetobacter baumannii Beta-lactamase ADC-33 Km 16000.0 nM 10.1128/aac.00050-10
Acinetobacter calcoaceticus Acinetobacter calcoaceticus MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Acinetobacter calcoaceticus Acinetobacter calcoaceticus MIC 2.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter calcoaceticus Acinetobacter calcoaceticus MIC 8.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter calcoaceticus Acinetobacter calcoaceticus MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter calcoaceticus Acinetobacter calcoaceticus MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter haemolyticus Acinetobacter haemolyticus MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Acinetobacter haemolyticus Acinetobacter haemolyticus MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Acinetobacter haemolyticus Acinetobacter haemolyticus MIC 256.0 ug.mL-1 10.1128/aac.00267-07
Acinetobacter haemolyticus Acinetobacter haemolyticus MIC50 0.12 ug.mL-1 10.1128/aac.01047-08
Acinetobacter haemolyticus Acinetobacter haemolyticus MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter haemolyticus Acinetobacter haemolyticus MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter haemolyticus Acinetobacter haemolyticus MIC90 32.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter haemolyticus Acinetobacter haemolyticus MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter lwoffii Acinetobacter lwoffii MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Acinetobacter lwoffii Acinetobacter lwoffii MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Acinetobacter lwoffii Acinetobacter lwoffii MIC nan None 10.1128/aac.00598-10
Acinetobacter lwoffii Acinetobacter lwoffii MIC50 0.12 ug.mL-1 10.1128/aac.01047-08
Acinetobacter lwoffii Acinetobacter lwoffii MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter lwoffii Acinetobacter lwoffii MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter lwoffii Acinetobacter lwoffii MIC90 32.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter lwoffii Acinetobacter lwoffii MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Acinetobacter pittii Acinetobacter pittii Activity 63.2 % 10.1128/aac.01624-09
Acinetobacter pittii Acinetobacter pittii MIC 8.0 ug.mL-1 10.1128/aac.01624-09
Acinetobacter pittii Acinetobacter pittii MIC 12.0 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 16.0 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 24.0 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 32.0 ug.mL-1 10.1128/aac.00485-08
Acinetobacter pittii Acinetobacter pittii MIC 32.0 ug.mL-1 10.1128/aac.01624-09
Acinetobacter pittii Acinetobacter pittii MIC 64.0 ug.mL-1 10.1128/aac.01624-09
Acinetobacter pittii Acinetobacter pittii MIC 512.0 ug.mL-1 10.1128/aac.00072-08
Acinetobacter pittii Acinetobacter pittii MIC50 128.0 ug.mL-1 10.1128/aac.01624-09
Acinetobacter pittii Acinetobacter pittii MIC90 128.0 ug.mL-1 10.1128/aac.01624-09
Acinetobacter radioresistens Acinetobacter radioresistens MIC 1.0 ug.mL-1 10.1128/aac.00999-08
Acinetobacter radioresistens Acinetobacter radioresistens MIC 64.0 ug.mL-1 10.1128/aac.00999-08
Acinetobacter sp. Acinetobacter sp. Activity 23.0 % 10.1128/aac.01808-09
Acinetobacter sp. Acinetobacter sp. MIC 128.0 ug.mL-1 10.1128/aac.00838-06
Actinomyces israelii Actinomyces israelii Activity 0.0 % 10.1128/aac.00481-10
Actinomyces israelii Actinomyces israelii Activity 92.0 % 10.1128/aac.00481-10
Actinomyces israelii Actinomyces israelii MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Actinomyces israelii Actinomyces israelii MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Actinomyces israelii Actinomyces israelii MIC50 0.5 ug.mL-1 10.1128/aac.00481-10
Actinomyces israelii Actinomyces israelii MIC50 1.0 ug.mL-1 10.1128/aac.00481-10
Actinomyces israelii Actinomyces israelii MIC90 8.0 ug.mL-1 10.1128/aac.00481-10
Actinomyces naeslundii Actinomyces naeslundii Activity 0.0 % 10.1128/aac.00481-10
Actinomyces naeslundii Actinomyces naeslundii Activity 92.0 % 10.1128/aac.00481-10
Actinomyces naeslundii Actinomyces naeslundii MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Actinomyces naeslundii Actinomyces naeslundii MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Actinomyces naeslundii Actinomyces naeslundii MIC50 0.5 ug.mL-1 10.1128/aac.00481-10
Actinomyces naeslundii Actinomyces naeslundii MIC50 1.0 ug.mL-1 10.1128/aac.00481-10
Actinomyces naeslundii Actinomyces naeslundii MIC90 8.0 ug.mL-1 10.1128/aac.00481-10
Aeromonas allosaccharophila Extended-spectrum beta-lactamase PER-6 Kcat 0.1 /s 10.1128/aac.01585-09
Aeromonas allosaccharophila Extended-spectrum beta-lactamase PER-6 Kcat/Km 25.0 /uM/s 10.1128/aac.01585-09
Aeromonas allosaccharophila Extended-spectrum beta-lactamase PER-6 Km 4000.0 nM 10.1128/aac.01585-09
Aeromonas caviae Aeromonas caviae MIC 256.0 ug.mL-1 10.1128/aac.01462-06
Aeromonas caviae IMP-19 Kcat 41.2 /s 10.1128/aac.01462-06
Aeromonas caviae IMP-19 Kcat/Km 0.28 None 10.1128/aac.01462-06
Aeromonas caviae IMP-19 Km 148000.0 nM 10.1128/aac.01462-06
Aeromonas sobria Aeromonas sobria MIC 64.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Anaerococcus prevotii Anaerococcus prevotii Activity 0.0 % 10.1128/aac.00481-10
Anaerococcus prevotii Anaerococcus prevotii Activity 0.0 % 10.1128/aac.00696-08
Anaerococcus prevotii Anaerococcus prevotii Activity 100.0 % 10.1128/aac.00481-10
Anaerococcus prevotii Anaerococcus prevotii MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Anaerococcus prevotii Anaerococcus prevotii MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Anaerococcus prevotii Anaerococcus prevotii MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Anaerococcus prevotii Anaerococcus prevotii MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Anaerococcus prevotii Anaerococcus prevotii MIC50 0.125 ug.mL-1 10.1128/aac.00481-10
Anaerococcus prevotii Anaerococcus prevotii MIC90 0.125 ug.mL-1 10.1128/aac.00481-10
Anaerococcus prevotii Anaerococcus prevotii MIC90 0.25 ug.mL-1 10.1128/aac.00481-10
Anaerococcus tetradius Anaerococcus tetradius MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Anaerococcus tetradius Anaerococcus tetradius MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Anaerococcus tetradius Anaerococcus tetradius MIC90 0.25 ug.mL-1 10.1128/aac.01557-08
Bacillus anthracis Bacillus anthracis Inhibition nan % 10.1128/aac.01594-07
Bacillus anthracis Bacillus anthracis MIC 1.0 ug.mL-1 10.1016/j.bmc.2007.08.035
Bacillus cereus Bacillus cereus MIC 1.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Bacillus clausii Beta-lactamase Activity 23.0 None 10.1128/aac.00537-07
Bacillus clausii Beta-lactamase Kcat 38.0 /s 10.1128/aac.00537-07
Bacillus clausii Beta-lactamase Kcat/Km 2.0 /uM/s 10.1128/aac.00537-07
Bacillus clausii Beta-lactamase Km 21000.0 nM 10.1128/aac.00537-07
Bacillus subtilis Bacillus subtilis MIC 0.5 ug.mL-1 10.1016/j.bmc.2007.07.048
Bacteroides caccae Bacteroides caccae Activity 0.0 % 10.1128/aac.00696-08
Bacteroides caccae Bacteroides caccae Activity 2.2 % 10.1128/aac.00081-08
Bacteroides caccae Bacteroides caccae Activity 4.0 % 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae Activity 7.0 % 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae Activity 35.0 % 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae Activity 42.0 % 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae Activity 51.0 % 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae Activity 65.0 % 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae Activity 89.0 % 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae Activity 96.0 % 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae MIC 0.06 ug.mL-1 10.1128/aac.00081-08
Bacteroides caccae Bacteroides caccae MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Bacteroides caccae Bacteroides caccae MIC 1.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae MIC 1.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides caccae Bacteroides caccae MIC 8.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae MIC 8.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae MIC 8.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides caccae Bacteroides caccae MIC50 8.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides caccae Bacteroides caccae MIC50 8.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae MIC50 8.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae MIC50 128.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae MIC50 128.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae MIC90 16.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae MIC90 32.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides caccae Bacteroides caccae MIC90 64.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides caccae Bacteroides caccae MIC90 128.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides caccae Bacteroides caccae MIC90 256.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis Activity 0.5 % 10.1128/aac.00081-08
Bacteroides fragilis Bacteroides fragilis Activity 1.0 % 10.1128/aac.00696-08
Bacteroides fragilis Bacteroides fragilis Activity 2.0 % 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis Activity 2.0 % 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis Activity 27.0 % 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis Activity 35.0 % 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis Activity 62.0 % 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis Activity 67.0 % 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis Activity 95.0 % 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis Activity 97.0 % 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis MIC 0.015 ug.mL-1 10.1128/aac.01047-08
Bacteroides fragilis Bacteroides fragilis MIC 0.06 ug.mL-1 10.1128/aac.00081-08
Bacteroides fragilis Bacteroides fragilis MIC 0.06 ug.mL-1 10.1128/aac.01047-08
Bacteroides fragilis Bacteroides fragilis MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Bacteroides fragilis Bacteroides fragilis MIC 0.25 ug.mL-1 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis MIC 0.25 ug.mL-1 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis MIC 0.25 ug.mL-1 10.1128/aac.00696-08
Bacteroides fragilis Bacteroides fragilis MIC 1.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides fragilis Bacteroides fragilis MIC 2.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis MIC 4.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis MIC 4.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides fragilis Bacteroides fragilis MIC 16.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides fragilis Bacteroides fragilis MIC50 0.06 ug.mL-1 10.1128/aac.01047-08
Bacteroides fragilis Bacteroides fragilis MIC50 0.25 ug.mL-1 10.1128/aac.01047-08
Bacteroides fragilis Bacteroides fragilis MIC50 0.5 ug.mL-1 10.1128/aac.01557-08
Bacteroides fragilis Bacteroides fragilis MIC50 1.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides fragilis Bacteroides fragilis MIC50 1.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis MIC50 1.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis MIC50 8.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis MIC50 8.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis MIC50 8.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides fragilis Bacteroides fragilis MIC90 0.25 ug.mL-1 10.1128/aac.01047-08
Bacteroides fragilis Bacteroides fragilis MIC90 0.5 ug.mL-1 10.1128/aac.01047-08
Bacteroides fragilis Bacteroides fragilis MIC90 2.0 ug.mL-1 10.1128/aac.01557-08
Bacteroides fragilis Bacteroides fragilis MIC90 4.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides fragilis Bacteroides fragilis MIC90 8.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides fragilis Bacteroides fragilis MIC90 8.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis MIC90 128.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides fragilis Bacteroides fragilis MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides fragilis Bacteroides fragilis MIC90 256.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus Activity 0.0 % 10.1128/aac.00081-08
Bacteroides ovatus Bacteroides ovatus Activity 0.0 % 10.1128/aac.00696-08
Bacteroides ovatus Bacteroides ovatus Activity 7.0 % 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus Activity 42.0 % 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus Activity 51.0 % 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus Activity 89.0 % 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus MIC 0.06 ug.mL-1 10.1128/aac.00081-08
Bacteroides ovatus Bacteroides ovatus MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Bacteroides ovatus Bacteroides ovatus MIC 1.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus MIC 1.0 ug.mL-1 10.1128/aac.01557-08
Bacteroides ovatus Bacteroides ovatus MIC 4.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides ovatus Bacteroides ovatus MIC 8.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus MIC 8.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides ovatus Bacteroides ovatus MIC50 2.0 ug.mL-1 10.1128/aac.01557-08
Bacteroides ovatus Bacteroides ovatus MIC50 8.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides ovatus Bacteroides ovatus MIC50 8.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus MIC50 128.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus MIC90 4.0 ug.mL-1 10.1128/aac.01557-08
Bacteroides ovatus Bacteroides ovatus MIC90 16.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides ovatus Bacteroides ovatus MIC90 64.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides ovatus Bacteroides ovatus MIC90 256.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides sp. Bacteroides sp. Activity 0.0 % 10.1128/aac.00081-08
Bacteroides sp. Bacteroides sp. MIC 0.06 ug.mL-1 10.1128/aac.00081-08
Bacteroides sp. Bacteroides sp. MIC50 8.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides sp. Bacteroides sp. MIC90 32.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides stercoris Bacteroides stercoris Activity 0.0 % 10.1128/aac.00081-08
Bacteroides stercoris Bacteroides stercoris MIC 0.06 ug.mL-1 10.1128/aac.00081-08
Bacteroides stercoris Bacteroides stercoris MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Bacteroides stercoris Bacteroides stercoris MIC50 1.0 ug.mL-1 10.1128/aac.01557-08
Bacteroides stercoris Bacteroides stercoris MIC50 8.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides stercoris Bacteroides stercoris MIC90 32.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 0.0 % 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 1.3 % 10.1128/aac.00696-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 3.3 % 10.1128/aac.00081-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 7.0 % 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 37.0 % 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 42.0 % 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 51.0 % 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 63.0 % 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 89.0 % 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron Activity 93.0 % 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 0.06 ug.mL-1 10.1128/aac.00081-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 0.5 ug.mL-1 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 1.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 1.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 1.3 ug.mL-1 10.1128/aac.00696-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 4.0 ug.mL-1 10.1128/aac.01557-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 8.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 8.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 8.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 8.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 32.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 32.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 8.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 8.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 8.0 ug.mL-1 10.1128/aac.01557-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 16.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 16.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 32.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 32.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC50 128.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 16.0 ug.mL-1 10.1128/aac.01557-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 32.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 32.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 64.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 128.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC90 256.0 ug.mL-1 10.1128/aac.00481-10
Bacteroides uniformis Bacteroides uniformis Activity 0.0 % 10.1128/aac.00081-08
Bacteroides uniformis Bacteroides uniformis Activity 0.0 % 10.1128/aac.00696-08
Bacteroides uniformis Bacteroides uniformis Activity 4.0 % 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis Activity 35.0 % 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis Activity 65.0 % 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis Activity 96.0 % 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis MIC 0.06 ug.mL-1 10.1128/aac.00081-08
Bacteroides uniformis Bacteroides uniformis MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Bacteroides uniformis Bacteroides uniformis MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Bacteroides uniformis Bacteroides uniformis MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Bacteroides uniformis Bacteroides uniformis MIC 0.5 ug.mL-1 10.1128/aac.01557-08
Bacteroides uniformis Bacteroides uniformis MIC 2.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides uniformis Bacteroides uniformis MIC 8.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis MIC 8.0 ug.mL-1 10.1128/aac.00696-08
Bacteroides uniformis Bacteroides uniformis MIC 8.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides uniformis Bacteroides uniformis MIC50 0.5 ug.mL-1 10.1128/aac.01047-08
Bacteroides uniformis Bacteroides uniformis MIC50 1.0 ug.mL-1 10.1128/aac.01557-08
Bacteroides uniformis Bacteroides uniformis MIC50 4.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides uniformis Bacteroides uniformis MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides uniformis Bacteroides uniformis MIC50 8.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis MIC50 16.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides uniformis Bacteroides uniformis MIC50 128.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis MIC90 4.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides uniformis Bacteroides uniformis MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides uniformis Bacteroides uniformis MIC90 16.0 ug.mL-1 10.1128/aac.00081-08
Bacteroides uniformis Bacteroides uniformis MIC90 16.0 ug.mL-1 10.1128/aac.00355-08
Bacteroides uniformis Bacteroides uniformis MIC90 32.0 ug.mL-1 10.1128/aac.01047-08
Bacteroides uniformis Bacteroides uniformis MIC90 128.0 ug.mL-1 10.1128/aac.00355-08
Bos taurus Monoamine oxidase A Activity nan None 10.1021/jm800656v
Bos taurus Progesterone receptor IC50 nan None None
Bos taurus Progesterone receptor Ki nan None None
Brachyspira pilosicoli Class D beta-lactamase Activity 6.5 % 10.1128/aac.00684-07
Brachyspira pilosicoli Class D beta-lactamase Kcat 2.1 /s 10.1128/aac.00684-07
Brachyspira pilosicoli Class D beta-lactamase Kcat/Km 6.4 10'4/M/s 10.1128/aac.00684-07
Brachyspira pilosicoli Class D beta-lactamase Km 33000.0 nM 10.1128/aac.00684-07
Burkholderia cenocepacia Burkholderia cenocepacia MIC 4.0 ug.mL-1 10.1128/aac.00946-08
Burkholderia cenocepacia Burkholderia cenocepacia MIC 128.0 ug.mL-1 10.1128/aac.00946-08
Burkholderia cenocepacia Burkholderia cenocepacia MIC 256.0 ug.mL-1 10.1128/aac.00946-08
Burkholderia cenocepacia Burkholderia cenocepacia MIC 512.0 ug.mL-1 10.1128/aac.00946-08
Burkholderia cenocepacia PenB class A beta-lactamase Kcat 5.0 /s 10.1128/aac.00946-08
Burkholderia cenocepacia PenB class A beta-lactamase Kcat/Km 500.0 /uM/s 10.1128/aac.00946-08
Burkholderia cenocepacia PenB class A beta-lactamase Km 10000.0 nM 10.1128/aac.00946-08
Burkholderia cepacia Burkholderia cepacia Activity 11.0 % 10.1128/aac.00954-06
Burkholderia cepacia Burkholderia cepacia Activity 80.0 % 10.1128/aac.00954-06
Burkholderia cepacia Burkholderia cepacia MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Burkholderia cepacia Burkholderia cepacia MIC 2.0 ug.mL-1 10.1128/aac.01047-08
Burkholderia cepacia Burkholderia cepacia MIC50 1.0 ug.mL-1 10.1128/aac.01047-08
Burkholderia cepacia Burkholderia cepacia MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Burkholderia cepacia Burkholderia cepacia MIC50 32.0 ug.mL-1 10.1128/aac.01047-08
Burkholderia cepacia Burkholderia cepacia MIC50 256.0 ug.mL-1 10.1128/aac.00954-06
Burkholderia cepacia Burkholderia cepacia MIC90 2.0 ug.mL-1 10.1128/aac.01047-08
Burkholderia cepacia Burkholderia cepacia MIC90 64.0 ug.mL-1 10.1128/aac.01047-08
Burkholderia cepacia Burkholderia cepacia MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Burkholderia cepacia Burkholderia cepacia MIC90 256.0 ug.mL-1 10.1128/aac.00954-06
Campylobacter coli Campylobacter coli MIC 256.0 ug.mL-1 10.1128/aac.01655-08
Campylobacter coli Campylobacter coli MIC 512.0 ug.mL-1 10.1128/aac.01655-08
Campylobacter coli Campylobacter coli MIC50 512.0 ug.mL-1 10.1128/aac.01655-08
Campylobacter coli Campylobacter coli MIC90 512.0 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC 8.0 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC 16.0 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC 128.0 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC 256.0 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC 512.0 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC50 512.0 ug.mL-1 10.1128/aac.01655-08
Campylobacter jejuni Campylobacter jejuni MIC90 512.0 ug.mL-1 10.1128/aac.01655-08
Carnobacterium divergens Carnobacterium divergens MIC 12.0 ug.mL-1 10.1128/aac.01145-07
Carnobacterium divergens Carnobacterium divergens MIC 32.0 ug.mL-1 10.1128/aac.01145-07
Carnobacterium divergens Carnobacterium divergens MIC 64.0 ug.mL-1 10.1128/aac.01145-07
Carnobacterium divergens Carnobacterium divergens MIC 128.0 ug.mL-1 10.1128/aac.01145-07
Carnobacterium divergens Carnobacterium divergens MIC nan None 10.1128/aac.01145-07
Caulobacter vibrioides Metallo-beta-lactamase Kcat/Km 5.7 10'5/M/s 10.1128/aac.01062-07
Cavia porcellus Leukotriene C4 synthase IC50 nan None None
Cavia porcellus Leukotriene C4 synthase Ki nan None None
Cavia porcellus Serotonin 4 (5-HT4) receptor IC50 nan None None
Cavia porcellus Serotonin 4 (5-HT4) receptor Ki nan None None
Chryseobacterium indologenes Chryseobacterium indologenes Activity 16.0 ug ml-1 10.1128/aac.00083-07
Chryseobacterium indologenes Chryseobacterium indologenes MIC 4.0 ug.mL-1 10.1128/aac.01607-08
Citrobacter Citrobacter Activity 2.6 % 10.1128/aac.00381-08
Citrobacter Citrobacter Activity 3.6 % 10.1128/aac.00381-08
Citrobacter Citrobacter Activity 3.7 % 10.1128/aac.00381-08
Citrobacter Citrobacter Activity 29.1 % 10.1128/aac.00381-08
Citrobacter Citrobacter Activity 67.3 % 10.1128/aac.00381-08
Citrobacter Citrobacter Activity 937.0 % 10.1128/aac.00381-08
Citrobacter Citrobacter MIC 0.25 ug.mL-1 10.1128/aac.00381-08
Citrobacter Citrobacter MIC 16.0 ug.mL-1 10.1128/aac.00381-08
Citrobacter Citrobacter MIC50 4.0 ug.mL-1 10.1128/aac.00381-08
Citrobacter Citrobacter MIC50 128.0 ug.mL-1 10.1128/aac.00381-08
Citrobacter Citrobacter MIC90 16.0 ug.mL-1 10.1128/aac.00381-08
Citrobacter Citrobacter MIC90 128.0 ug.mL-1 10.1128/aac.00381-08
Citrobacter freundii Citrobacter freundii Activity 0.0 % 10.1128/aac.00149-08
Citrobacter freundii Citrobacter freundii Activity 24.2 % 10.1128/aac.00149-08
Citrobacter freundii Citrobacter freundii Activity 39.4 % 10.1128/aac.00149-08
Citrobacter freundii Citrobacter freundii Activity 71.0 % 10.1128/aac.00426-09
Citrobacter freundii Citrobacter freundii Activity 72.0 % 10.1128/aac.01808-09
Citrobacter freundii Citrobacter freundii Activity 100.0 % 10.1128/aac.00149-08
Citrobacter freundii Citrobacter freundii MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Citrobacter freundii Citrobacter freundii MIC 1.0 ug.mL-1 10.1128/aac.00149-08
Citrobacter freundii Citrobacter freundii MIC 1.0 ug.mL-1 10.1128/aac.00830-08
Citrobacter freundii Citrobacter freundii MIC 1.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter freundii Citrobacter freundii MIC 2.0 ug.mL-1 10.1128/aac.00149-08
Citrobacter freundii Citrobacter freundii MIC 2.0 ug.mL-1 10.1128/aac.00830-08
Citrobacter freundii Citrobacter freundii MIC 2.0 ug.mL-1 10.1128/aac.01197-09
Citrobacter freundii Citrobacter freundii MIC 4.0 ug.mL-1 10.1128/aac.00830-08
Citrobacter freundii Citrobacter freundii MIC 4.0 ug.mL-1 10.1128/aac.01337-07
Citrobacter freundii Citrobacter freundii MIC 8.0 ug.mL-1 10.1128/aac.00830-08
Citrobacter freundii Citrobacter freundii MIC 8.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter freundii Citrobacter freundii MIC 16.0 ug.mL-1 10.1128/aac.00830-08
Citrobacter freundii Citrobacter freundii MIC 32.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter freundii Citrobacter freundii MIC 64.0 ug.mL-1 10.1128/aac.00830-08
Citrobacter freundii Citrobacter freundii MIC 200.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Citrobacter freundii Citrobacter freundii MIC 256.0 ug.mL-1 10.1128/aac.00830-08
Citrobacter freundii Citrobacter freundii MIC 256.0 ug.mL-1 10.1128/aac.01395-06
Citrobacter freundii Citrobacter freundii MIC 256.0 ug.mL-1 10.1128/aac.01405-06
Citrobacter freundii Citrobacter freundii MIC 400.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Citrobacter freundii Citrobacter freundii MIC 512.0 ug.mL-1 10.1128/aac.01312-09
Citrobacter freundii Citrobacter freundii MIC50 2.0 ug.mL-1 10.1128/aac.00149-08
Citrobacter freundii Citrobacter freundii MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter freundii Citrobacter freundii MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter freundii Citrobacter freundii MIC50 8.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter freundii Citrobacter freundii MIC50 16.0 ug.mL-1 10.1128/aac.01197-09
Citrobacter freundii Citrobacter freundii MIC50 32.0 ug.mL-1 10.1128/aac.00149-08
Citrobacter freundii Citrobacter freundii MIC50 64.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter freundii Citrobacter freundii MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter freundii Citrobacter freundii MIC90 4.0 ug.mL-1 10.1128/aac.00149-08
Citrobacter freundii Citrobacter freundii MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter freundii Citrobacter freundii MIC90 64.0 ug.mL-1 10.1128/aac.00149-08
Citrobacter freundii Citrobacter freundii MIC90 64.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter freundii Citrobacter freundii MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter freundii Citrobacter freundii MIC90 128.0 ug.mL-1 10.1128/aac.01197-09
Citrobacter freundii PER-2 beta-lactamase Activity 30.0 % 10.1128/aac.01395-06
Citrobacter freundii PER-2 beta-lactamase Kcat 0.04 /s 10.1128/aac.01395-06
Citrobacter freundii PER-2 beta-lactamase Kcat/Km 0.2 /uM/s 10.1128/aac.01395-06
Citrobacter freundii PER-2 beta-lactamase Ki 200.0 nM 10.1128/aac.01395-06
Citrobacter gillenii Gil1 Kcat 306.0 /s 10.1128/aac.01152-06
Citrobacter gillenii Gil1 Kcat/Km 3400.0 /mM/s 10.1128/aac.01152-06
Citrobacter gillenii Gil1 Km 90000.0 nM 10.1128/aac.01152-06
Citrobacter gillenii Gil1 Ratio 61.0 None 10.1128/aac.01152-06
Citrobacter koseri Citrobacter koseri MIC 1.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter koseri Citrobacter koseri MIC 4.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter koseri Citrobacter koseri MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter koseri Citrobacter koseri MIC50 32.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter koseri Citrobacter koseri MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter koseri Citrobacter koseri MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Citrobacter koseri Citrobacter koseri MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Clostridioides difficile Clostridioides difficile Activity 0.0 % 10.1128/aac.00481-10
Clostridioides difficile Clostridioides difficile Activity 100.0 % 10.1128/aac.00481-10
Clostridioides difficile Clostridioides difficile Activity nan None 10.1128/aac.00696-08
Clostridioides difficile Clostridioides difficile MIC 1.0 ug.mL-1 10.1128/aac.00481-10
Clostridioides difficile Clostridioides difficile MIC 2.0 ug.mL-1 10.1128/aac.00481-10
Clostridioides difficile Clostridioides difficile MIC 2.0 ug.mL-1 10.1128/aac.00696-08
Clostridioides difficile Clostridioides difficile MIC 4.0 ug.mL-1 10.1128/aac.00476-08
Clostridioides difficile Clostridioides difficile MIC 8.0 ug.mL-1 10.1128/aac.01557-08
Clostridioides difficile Clostridioides difficile MIC50 4.0 ug.mL-1 10.1128/aac.00481-10
Clostridioides difficile Clostridioides difficile MIC50 8.0 ug.mL-1 10.1128/aac.00476-08
Clostridioides difficile Clostridioides difficile MIC50 8.0 ug.mL-1 10.1128/aac.01557-08
Clostridioides difficile Clostridioides difficile MIC90 8.0 ug.mL-1 10.1128/aac.00476-08
Clostridioides difficile Clostridioides difficile MIC90 8.0 ug.mL-1 10.1128/aac.00481-10
Clostridioides difficile Clostridioides difficile MIC90 16.0 ug.mL-1 10.1128/aac.01557-08
Clostridium butyricum Clostridium butyricum MIC 0.5 ug.mL-1 10.1128/aac.01557-08
Clostridium cadaveris Clostridium cadaveris MIC 0.125 ug.mL-1 10.1128/aac.01557-08
[Clostridium] innocuum [Clostridium] innocuum Activity 5.6 % 10.1128/aac.00696-08
[Clostridium] innocuum [Clostridium] innocuum MIC 0.125 ug.mL-1 10.1128/aac.01557-08
[Clostridium] innocuum [Clostridium] innocuum MIC 0.5 ug.mL-1 10.1128/aac.00696-08
[Clostridium] innocuum [Clostridium] innocuum MIC 2.0 ug.mL-1 10.1128/aac.00696-08
[Clostridium] innocuum [Clostridium] innocuum MIC 16.0 ug.mL-1 10.1128/aac.00696-08
Clostridium paraputrificum Clostridium paraputrificum Activity 0.0 % 10.1128/aac.00355-08
Clostridium paraputrificum Clostridium paraputrificum Activity 5.6 % 10.1128/aac.00696-08
Clostridium paraputrificum Clostridium paraputrificum Activity 100.0 % 10.1128/aac.00355-08
Clostridium paraputrificum Clostridium paraputrificum MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Clostridium paraputrificum Clostridium paraputrificum MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Clostridium paraputrificum Clostridium paraputrificum MIC 2.0 ug.mL-1 10.1128/aac.00696-08
Clostridium paraputrificum Clostridium paraputrificum MIC 16.0 ug.mL-1 10.1128/aac.00696-08
Clostridium paraputrificum Clostridium paraputrificum MIC50 0.25 ug.mL-1 10.1128/aac.00355-08
Clostridium paraputrificum Clostridium paraputrificum MIC50 0.5 ug.mL-1 10.1128/aac.00355-08
Clostridium paraputrificum Clostridium paraputrificum MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Clostridium perfringens Clostridium perfringens Activity 0.0 % 10.1128/aac.00355-08
Clostridium perfringens Clostridium perfringens Activity 0.0 % 10.1128/aac.00481-10
Clostridium perfringens Clostridium perfringens Activity 0.0 % 10.1128/aac.00696-08
Clostridium perfringens Clostridium perfringens Activity 100.0 % 10.1128/aac.00355-08
Clostridium perfringens Clostridium perfringens Activity 100.0 % 10.1128/aac.00481-10
Clostridium perfringens Clostridium perfringens MIC 0.015 ug.mL-1 10.1128/aac.01047-08
Clostridium perfringens Clostridium perfringens MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Clostridium perfringens Clostridium perfringens MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Clostridium perfringens Clostridium perfringens MIC 0.03 ug.mL-1 10.1128/aac.01047-08
Clostridium perfringens Clostridium perfringens MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Clostridium perfringens Clostridium perfringens MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Clostridium perfringens Clostridium perfringens MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Clostridium perfringens Clostridium perfringens MIC 4.0 ug.mL-1 10.1128/aac.00696-08
Clostridium perfringens Clostridium perfringens MIC50 0.015 ug.mL-1 10.1128/aac.01047-08
Clostridium perfringens Clostridium perfringens MIC50 0.06 ug.mL-1 10.1128/aac.01047-08
Clostridium perfringens Clostridium perfringens MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Clostridium perfringens Clostridium perfringens MIC50 0.25 ug.mL-1 10.1128/aac.00355-08
Clostridium perfringens Clostridium perfringens MIC50 0.25 ug.mL-1 10.1128/aac.00481-10
Clostridium perfringens Clostridium perfringens MIC50 0.5 ug.mL-1 10.1128/aac.00355-08
Clostridium perfringens Clostridium perfringens MIC90 0.015 ug.mL-1 10.1128/aac.01047-08
Clostridium perfringens Clostridium perfringens MIC90 0.03 ug.mL-1 10.1128/aac.01047-08
Clostridium perfringens Clostridium perfringens MIC90 0.25 ug.mL-1 10.1128/aac.01047-08
Clostridium perfringens Clostridium perfringens MIC90 0.5 ug.mL-1 10.1128/aac.00481-10
Clostridium perfringens Clostridium perfringens MIC90 0.5 ug.mL-1 10.1128/aac.01557-08
Clostridium perfringens Clostridium perfringens MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Clostridium septicum Clostridium septicum Activity 0.0 % 10.1128/aac.00355-08
Clostridium septicum Clostridium septicum Activity 100.0 % 10.1128/aac.00355-08
Clostridium septicum Clostridium septicum MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Clostridium septicum Clostridium septicum MIC50 0.25 ug.mL-1 10.1128/aac.00355-08
Clostridium septicum Clostridium septicum MIC50 0.5 ug.mL-1 10.1128/aac.00355-08
Clostridium septicum Clostridium septicum MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Clostridium tertium Clostridium tertium Activity 0.0 % 10.1128/aac.00355-08
Clostridium tertium Clostridium tertium Activity 5.6 % 10.1128/aac.00696-08
Clostridium tertium Clostridium tertium Activity 100.0 % 10.1128/aac.00355-08
Clostridium tertium Clostridium tertium MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Clostridium tertium Clostridium tertium MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Clostridium tertium Clostridium tertium MIC 2.0 ug.mL-1 10.1128/aac.00696-08
Clostridium tertium Clostridium tertium MIC 4.0 ug.mL-1 10.1128/aac.01557-08
Clostridium tertium Clostridium tertium MIC 16.0 ug.mL-1 10.1128/aac.00696-08
Clostridium tertium Clostridium tertium MIC50 0.25 ug.mL-1 10.1128/aac.00355-08
Clostridium tertium Clostridium tertium MIC50 0.5 ug.mL-1 10.1128/aac.00355-08
Clostridium tertium Clostridium tertium MIC50 8.0 ug.mL-1 10.1128/aac.01557-08
Clostridium tertium Clostridium tertium MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Cutibacterium acnes Cutibacterium acnes Activity 0.0 % 10.1128/aac.00696-08
Cutibacterium acnes Cutibacterium acnes MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Cutibacterium acnes Cutibacterium acnes MIC 0.25 ug.mL-1 10.1128/aac.00696-08
Cutibacterium acnes Cutibacterium acnes MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Cutibacterium acnes Cutibacterium acnes MIC50 0.25 ug.mL-1 10.1128/aac.01557-08
Cutibacterium acnes Cutibacterium acnes MIC90 1.0 ug.mL-1 10.1128/aac.01557-08
Dialister invisus Dialister invisus Activity 8.0 ug ml-1 10.1128/aac.00538-07
Dialister invisus Dialister invisus Activity 32.0 ug ml-1 10.1128/aac.00538-07
Dialister invisus Dialister invisus MIC 0.125 ug.mL-1 10.1128/aac.00538-07
Dialister micraerophilus Dialister micraerophilus Activity 8.0 ug ml-1 10.1128/aac.00538-07
Dialister micraerophilus Dialister micraerophilus Activity 32.0 ug ml-1 10.1128/aac.00538-07
Dialister micraerophilus Dialister micraerophilus MIC 0.125 ug.mL-1 10.1128/aac.00538-07
Dialister micraerophilus Dialister micraerophilus MIC50 0.125 ug.mL-1 10.1128/aac.00538-07
Dialister micraerophilus Dialister micraerophilus MIC90 1.0 ug.mL-1 10.1128/aac.00538-07
Dialister pneumosintes Dialister pneumosintes Activity 8.0 ug ml-1 10.1128/aac.00538-07
Dialister pneumosintes Dialister pneumosintes Activity 32.0 ug ml-1 10.1128/aac.00538-07
Dialister pneumosintes Dialister pneumosintes MIC 0.125 ug.mL-1 10.1128/aac.00538-07
Dialister pneumosintes Dialister pneumosintes MIC50 1.0 ug.mL-1 10.1128/aac.00538-07
Dialister pneumosintes Dialister pneumosintes MIC90 16.0 ug.mL-1 10.1128/aac.00538-07
Dialister propionicifaciens Dialister propionicifaciens Activity 8.0 ug ml-1 10.1128/aac.00538-07
Dialister propionicifaciens Dialister propionicifaciens Activity 32.0 ug ml-1 10.1128/aac.00538-07
Dialister propionicifaciens Dialister propionicifaciens MIC 0.125 ug.mL-1 10.1128/aac.00538-07
Eggerthella lenta Eggerthella lenta Activity 0.0 % 10.1128/aac.00481-10
Eggerthella lenta Eggerthella lenta Activity 92.0 % 10.1128/aac.00481-10
Eggerthella lenta Eggerthella lenta MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Eggerthella lenta Eggerthella lenta MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Eggerthella lenta Eggerthella lenta MIC 8.0 ug.mL-1 10.1128/aac.01557-08
Eggerthella lenta Eggerthella lenta MIC50 0.5 ug.mL-1 10.1128/aac.00481-10
Eggerthella lenta Eggerthella lenta MIC50 1.0 ug.mL-1 10.1128/aac.00481-10
Eggerthella lenta Eggerthella lenta MIC50 16.0 ug.mL-1 10.1128/aac.01557-08
Eggerthella lenta Eggerthella lenta MIC90 8.0 ug.mL-1 10.1128/aac.00481-10
Eggerthella lenta Eggerthella lenta MIC90 16.0 ug.mL-1 10.1128/aac.01557-08
Elizabethkingia meningoseptica GOB-1 metallo-beta-lactamase Kcat/Km 1.7 10'6/M/s 10.1128/aac.01062-07
Enterobacter Enterobacter MIC 32.0 ug.mL-1 10.1128/aac.01614-06
Enterobacter Enterobacter MIC 64.0 ug.mL-1 10.1128/aac.01614-06
Enterobacter Enterobacter MIC 128.0 ug.mL-1 10.1128/aac.01614-06
Enterobacter Enterobacter MIC 256.0 ug.mL-1 10.1128/aac.01614-06
Enterobacter cloacae Beta-lactamase MIC 32.0 ug.mL-1 10.1021/jm034056q
Enterobacter cloacae Beta-lactamase MIC 64.0 ug.mL-1 10.1021/jm034056q
Enterobacter cloacae Enterobacter cloacae Activity 0.0 % 10.1128/aac.01538-07
Enterobacter cloacae Enterobacter cloacae Activity 2.0 % 10.1128/aac.00149-08
Enterobacter cloacae Enterobacter cloacae Activity 3.2 % 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae Activity 3.5 % 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae Activity 4.2 % 10.1128/aac.01538-07
Enterobacter cloacae Enterobacter cloacae Activity 4.6 % 10.1128/aac.01538-07
Enterobacter cloacae Enterobacter cloacae Activity 4.9 % 10.1128/aac.01538-07
Enterobacter cloacae Enterobacter cloacae Activity 5.8 % 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae Activity 8.4 % 10.1128/aac.00400-09
Enterobacter cloacae Enterobacter cloacae Activity 9.0 % 10.1128/aac.00400-09
Enterobacter cloacae Enterobacter cloacae Activity 11.7 % 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae Activity 12.5 % 10.1128/aac.01538-07
Enterobacter cloacae Enterobacter cloacae Activity 25.7 % 10.1128/aac.00149-08
Enterobacter cloacae Enterobacter cloacae Activity 54.3 % 10.1128/aac.00149-08
Enterobacter cloacae Enterobacter cloacae Activity 69.0 % 10.1128/aac.01808-09
Enterobacter cloacae Enterobacter cloacae Activity 71.0 % 10.1128/aac.00426-09
Enterobacter cloacae Enterobacter cloacae Activity 82.5 % 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae Activity 82.6 % 10.1128/aac.00400-09
Enterobacter cloacae Enterobacter cloacae Activity 93.3 % 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae Activity 98.0 % 10.1128/aac.00149-08
Enterobacter cloacae Enterobacter cloacae ED50 30.0 mg.kg-1 10.1128/aac.01549-08
Enterobacter cloacae Enterobacter cloacae ED50 31.0 mg.kg-1 10.1128/aac.01549-08
Enterobacter cloacae Enterobacter cloacae ED50 32.0 mg.kg-1 10.1128/aac.01549-08
Enterobacter cloacae Enterobacter cloacae ED50 47.0 mg.kg-1 10.1128/aac.01549-08
Enterobacter cloacae Enterobacter cloacae ED50 60.0 mg.kg-1 10.1128/aac.01549-08
Enterobacter cloacae Enterobacter cloacae ED50 69.0 mg.kg-1 10.1128/aac.01549-08
Enterobacter cloacae Enterobacter cloacae ED50 71.0 mg.kg-1 10.1128/aac.01549-08
Enterobacter cloacae Enterobacter cloacae ED50 282.0 mg.kg-1 10.1128/aac.01549-08
Enterobacter cloacae Enterobacter cloacae MIC 0.25 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC 0.5 ug.mL-1 10.1128/aac.00149-08
Enterobacter cloacae Enterobacter cloacae MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Enterobacter cloacae Enterobacter cloacae MIC 1.0 ug.mL-1 10.1128/aac.00149-08
Enterobacter cloacae Enterobacter cloacae MIC 1.0 ug.mL-1 10.1128/aac.00400-09
Enterobacter cloacae Enterobacter cloacae MIC 1.0 ug.mL-1 10.1128/aac.00830-08
Enterobacter cloacae Enterobacter cloacae MIC 1.0 ug.mL-1 10.1128/aac.01047-08
Enterobacter cloacae Enterobacter cloacae MIC 2.0 ug.mL-1 10.1128/aac.00830-08
Enterobacter cloacae Enterobacter cloacae MIC 4.0 ug.mL-1 10.1128/aac.00830-08
Enterobacter cloacae Enterobacter cloacae MIC 4.0 ug.mL-1 10.1128/aac.01197-09
Enterobacter cloacae Enterobacter cloacae MIC 4.0 ug.mL-1 10.1128/aac.01549-08
Enterobacter cloacae Enterobacter cloacae MIC 6.0 ug.mL-1 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae MIC 8.0 ug.mL-1 10.1128/aac.00830-08
Enterobacter cloacae Enterobacter cloacae MIC 8.0 ug.mL-1 10.1128/aac.01047-08
Enterobacter cloacae Enterobacter cloacae MIC 8.0 ug.mL-1 10.1128/aac.01549-08
Enterobacter cloacae Enterobacter cloacae MIC 16.0 ug.mL-1 10.1016/0960-894X(95)00249-S
Enterobacter cloacae Enterobacter cloacae MIC 16.0 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC 16.0 ug.mL-1 10.1128/aac.01082-06
Enterobacter cloacae Enterobacter cloacae MIC 32.0 ug.mL-1 10.1128/aac.01047-08
Enterobacter cloacae Enterobacter cloacae MIC 50.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Enterobacter cloacae Enterobacter cloacae MIC 64.0 ug.mL-1 10.1016/s0960-894x(00)00444-3
Enterobacter cloacae Enterobacter cloacae MIC 64.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Enterobacter cloacae Enterobacter cloacae MIC 64.0 ug.mL-1 10.1128/aac.00830-08
Enterobacter cloacae Enterobacter cloacae MIC 64.0 ug.mL-1 10.1128/aac.01341-07
Enterobacter cloacae Enterobacter cloacae MIC 64.0 ug.mL-1 10.1128/aac.01549-08
Enterobacter cloacae Enterobacter cloacae MIC 96.0 ug.mL-1 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae MIC 100.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Enterobacter cloacae Enterobacter cloacae MIC 128.0 ug.mL-1 10.1016/0960-894X(95)00249-S
Enterobacter cloacae Enterobacter cloacae MIC 128.0 ug.mL-1 10.1128/aac.00707-08
Enterobacter cloacae Enterobacter cloacae MIC 128.0 ug.mL-1 10.1128/aac.00931-08
Enterobacter cloacae Enterobacter cloacae MIC 128.0 ug.mL-1 10.1128/aac.01341-07
Enterobacter cloacae Enterobacter cloacae MIC 192.0 ug.mL-1 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae MIC 256.0 ug.mL-1 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae MIC 256.0 ug.mL-1 10.1128/aac.00163-08
Enterobacter cloacae Enterobacter cloacae MIC 256.0 ug.mL-1 10.1128/aac.00260-09
Enterobacter cloacae Enterobacter cloacae MIC 256.0 ug.mL-1 10.1128/aac.00830-08
Enterobacter cloacae Enterobacter cloacae MIC 512.0 ug.mL-1 10.1128/aac.01312-09
Enterobacter cloacae Enterobacter cloacae MIC50 2.0 ug.mL-1 10.1128/aac.00149-08
Enterobacter cloacae Enterobacter cloacae MIC50 2.0 ug.mL-1 10.1128/aac.00400-09
Enterobacter cloacae Enterobacter cloacae MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Enterobacter cloacae Enterobacter cloacae MIC50 4.0 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Enterobacter cloacae Enterobacter cloacae MIC50 8.0 ug.mL-1 10.1128/aac.01047-08
Enterobacter cloacae Enterobacter cloacae MIC50 64.0 ug.mL-1 10.1128/aac.00149-08
Enterobacter cloacae Enterobacter cloacae MIC50 128.0 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Enterobacter cloacae Enterobacter cloacae MIC50 128.0 ug.mL-1 10.1128/aac.01197-09
Enterobacter cloacae Enterobacter cloacae MIC90 4.0 ug.mL-1 10.1128/aac.00149-08
Enterobacter cloacae Enterobacter cloacae MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Enterobacter cloacae Enterobacter cloacae MIC90 16.0 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Enterobacter cloacae Enterobacter cloacae MIC90 32.0 ug.mL-1 10.1128/aac.01047-08
Enterobacter cloacae Enterobacter cloacae MIC90 64.0 ug.mL-1 10.1128/aac.00149-08
Enterobacter cloacae Enterobacter cloacae MIC90 64.0 ug.mL-1 10.1128/aac.00400-09
Enterobacter cloacae Enterobacter cloacae MIC90 128.0 ug.mL-1 10.1128/aac.00381-08
Enterobacter cloacae Enterobacter cloacae MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Enterobacter cloacae Enterobacter cloacae MIC90 128.0 ug.mL-1 10.1128/aac.01197-09
Enterobacter cloacae IMI-1 Kcat 6.1 /s 10.1128/aac.00491-07
Enterobacter cloacae IMI-1 Kcat/Km 470.0 /mM/s 10.1128/aac.00491-07
Enterobacter cloacae IMI-1 Km 13000.0 nM 10.1128/aac.00491-07
Enterobacteriaceae Enterobacteriaceae Activity 1.6 % 10.1128/aac.00149-08
Enterobacteriaceae Enterobacteriaceae Activity 1.9 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 2.3 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 15.6 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 20.6 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 32.1 % 10.1128/aac.00044-07
Enterobacteriaceae Enterobacteriaceae Activity 38.6 % 10.1128/aac.00149-08
Enterobacteriaceae Enterobacteriaceae Activity 43.2 % 10.1128/aac.00149-08
Enterobacteriaceae Enterobacteriaceae Activity 63.8 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 90.2 % 10.1128/aac.00044-07
Enterobacteriaceae Enterobacteriaceae Activity 95.8 % 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae Activity 97.0 % 10.1128/aac.00149-08
Enterobacteriaceae Enterobacteriaceae MIC 0.25 ug.mL-1 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae MIC 0.5 ug.mL-1 10.1128/aac.00149-08
Enterobacteriaceae Enterobacteriaceae MIC 0.5 ug.mL-1 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae MIC50 2.0 ug.mL-1 10.1128/aac.00149-08
Enterobacteriaceae Enterobacteriaceae MIC50 4.0 ug.mL-1 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae MIC50 32.0 ug.mL-1 10.1128/aac.00149-08
Enterobacteriaceae Enterobacteriaceae MIC50 128.0 ug.mL-1 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae MIC90 4.0 ug.mL-1 10.1128/aac.00149-08
Enterobacteriaceae Enterobacteriaceae MIC90 8.0 ug.mL-1 10.1128/aac.00381-08
Enterobacteriaceae Enterobacteriaceae MIC90 64.0 ug.mL-1 10.1128/aac.00149-08
Enterobacteriaceae Enterobacteriaceae MIC90 128.0 ug.mL-1 10.1128/aac.00381-08
Enterocloster clostridioformis Enterocloster clostridioformis MIC 8.0 ug.mL-1 10.1128/aac.01557-08
Enterococcus avium Enterococcus avium MIC 1.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus avium Enterococcus avium MIC 4.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus avium Enterococcus avium MIC50 8.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus avium Enterococcus avium MIC50 16.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus avium Enterococcus avium MIC90 32.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus avium Enterococcus avium MIC90 64.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus casseliflavus Enterococcus casseliflavus MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Enterococcus casseliflavus Enterococcus casseliflavus MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Enterococcus casseliflavus Enterococcus casseliflavus MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus casseliflavus Enterococcus casseliflavus MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus casseliflavus Enterococcus casseliflavus MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus casseliflavus Enterococcus casseliflavus MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus durans Enterococcus durans MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Enterococcus durans Enterococcus durans MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Enterococcus durans Enterococcus durans MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus durans Enterococcus durans MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus durans Enterococcus durans MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus durans Enterococcus durans MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecalis Enterococcus faecalis MIC 1.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Enterococcus faecalis Enterococcus faecalis MIC 1.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecalis Enterococcus faecalis MIC 2.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Enterococcus faecalis Enterococcus faecalis MIC 2.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecalis Enterococcus faecalis MIC 64.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Enterococcus faecalis Enterococcus faecalis MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecalis Enterococcus faecalis MIC90 4.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecalis Enterococcus faecalis MIC90 64.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecalis Enterococcus faecalis MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecium Enterococcus faecium MIC 0.12 ug.mL-1 10.1016/s0960-894x(03)00512-2
Enterococcus faecium Enterococcus faecium MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecium Enterococcus faecium MIC 1.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Enterococcus faecium Enterococcus faecium MIC 1.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecium Enterococcus faecium MIC 32.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecium Enterococcus faecium MIC 64.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Enterococcus faecium Enterococcus faecium MIC 128.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecium Enterococcus faecium MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecium Enterococcus faecium MIC50 32.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecium Enterococcus faecium MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus faecium Enterococcus faecium MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus gallinarum Enterococcus gallinarum MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Enterococcus gallinarum Enterococcus gallinarum MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Enterococcus gallinarum Enterococcus gallinarum MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus gallinarum Enterococcus gallinarum MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus gallinarum Enterococcus gallinarum MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus gallinarum Enterococcus gallinarum MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus hirae Enterococcus hirae MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Enterococcus hirae Enterococcus hirae MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Enterococcus hirae Enterococcus hirae MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus hirae Enterococcus hirae MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus hirae Enterococcus hirae MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus hirae Enterococcus hirae MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Enterococcus sp. Enterococcus sp. Activity 0.0 % 10.1128/aac.01538-07
Enterococcus sp. Enterococcus sp. Activity 13.3 % 10.1128/aac.01538-07
Enterococcus sp. Enterococcus sp. Activity 17.3 % 10.1128/aac.01538-07
Enterococcus sp. Enterococcus sp. Activity 21.1 % 10.1128/aac.01538-07
Enterococcus sp. Enterococcus sp. Activity 22.2 % 10.1128/aac.01538-07
Enterococcus sp. Enterococcus sp. Activity 27.0 % 10.1128/aac.01538-07
Enterococcus sp. Enterococcus sp. MIC 0.25 ug.mL-1 10.1016/s0960-894x(03)00512-2
Enterococcus sp. Enterococcus sp. MIC 0.25 ug.mL-1 10.1016/s0960-894x(03)00542-0
Escherichia coli Beta-lactamase ACC-4 Kcat 0.13 /s 10.1128/aac.00389-07
Escherichia coli Beta-lactamase ACC-4 Kcat/Km 0.12 /s/microM 10.1128/aac.00389-07
Escherichia coli Beta-lactamase ACC-4 Km 1100.0 nM 10.1128/aac.00389-07
Escherichia coli Beta-lactamase OXA-7 Km 34000.0 nM 10.1128/aac.01714-09
Escherichia coli Beta-lactamase OXA-7 Vmax 3.5 nmol/sec 10.1128/aac.01714-09
Escherichia coli Beta-lactamase SHV-1 Kcat 1490.0 /s 10.1128/aac.01442-09
Escherichia coli Beta-lactamase SHV-1 Kcat/Km 62.1 /uM/s 10.1128/aac.01442-09
Escherichia coli Beta-lactamase SHV-1 Km 24000.0 nM 10.1128/aac.01442-09
Escherichia coli Beta-lactamase SHV-11 Kcat 30.0 /s 10.1128/aac.00387-08
Escherichia coli Beta-lactamase SHV-11 Kcat/Km 750.0 /uM/s 10.1128/aac.00387-08
Escherichia coli Beta-lactamase SHV-11 Km 40000.0 nM 10.1128/aac.00387-08
Escherichia coli Beta-lactamase TEM Kcat 1250.0 /s 10.1128/aac.00614-07
Escherichia coli Beta-lactamase TEM Kcat/Km 23.0 None 10.1128/aac.00614-07
Escherichia coli Beta-lactamase TEM Km 55.0 /s/microM 10.1128/aac.00614-07
Escherichia coli Beta-lactamase TEM MIC 128.0 ug.mL-1 10.1016/j.bmcl.2003.12.037
Escherichia coli BlaVIM-1 Kcat 1860.0 /s 10.1128/aac.00017-09
Escherichia coli BlaVIM-1 Kcat 1860.0 /s 10.1128/aac.00458-09
Escherichia coli BlaVIM-1 Kcat/Km 0.5 /uM/s 10.1128/aac.00458-09
Escherichia coli BlaVIM-1 Kcat/Km 0.53 /s/microM 10.1128/aac.00017-09
Escherichia coli BlaVIM-1 Km 3500000.0 nM 10.1128/aac.00458-09
Escherichia coli CMT-type beta lactamase Kcat 17.1 /s 10.1128/aac.00614-07
Escherichia coli CMT-type beta lactamase Kcat/Km 0.37 None 10.1128/aac.00614-07
Escherichia coli CMT-type beta lactamase Km 46.0 /s/microM 10.1128/aac.00614-07
Escherichia coli Escherichia coli Activity 0.0 % 10.1128/aac.01538-07
Escherichia coli Escherichia coli Activity 1.0 % 10.1128/aac.00400-09
Escherichia coli Escherichia coli Activity 1.0 ug ml-1 10.1128/aac.00083-07
Escherichia coli Escherichia coli Activity 1.1 % 10.1128/aac.01538-07
Escherichia coli Escherichia coli Activity 1.2 uM 10.1128/aac.01714-09
Escherichia coli Escherichia coli Activity 1.4 % 10.1128/aac.00400-09
Escherichia coli Escherichia coli Activity 1.6 % 10.1128/aac.01538-07
Escherichia coli Escherichia coli Activity 1.9 % 10.1128/aac.01538-07
Escherichia coli Escherichia coli Activity 2.3 % 10.1128/aac.00149-08
Escherichia coli Escherichia coli Activity 3.2 % 10.1128/aac.00381-08
Escherichia coli Escherichia coli Activity 5.6 % 10.1128/aac.01176-07
Escherichia coli Escherichia coli Activity 6.9 % 10.1128/aac.01538-07
Escherichia coli Escherichia coli Activity 16.7 % 10.1128/aac.00381-08
Escherichia coli Escherichia coli Activity 17.5 % 10.1128/aac.00149-08
Escherichia coli Escherichia coli Activity 30.0 % 10.1128/aac.00381-08
Escherichia coli Escherichia coli Activity 32.0 ug ml-1 10.1128/aac.00083-07
Escherichia coli Escherichia coli Activity 47.0 % 10.1128/aac.00061-09
Escherichia coli Escherichia coli Activity 53.3 % 10.1128/aac.00381-08
Escherichia coli Escherichia coli Activity 62.0 % 10.1128/aac.01808-09
Escherichia coli Escherichia coli Activity 68.3 % 10.1128/aac.00149-08
Escherichia coli Escherichia coli Activity 83.0 % 10.1128/aac.00426-09
Escherichia coli Escherichia coli Activity 93.6 % 10.1128/aac.00381-08
Escherichia coli Escherichia coli Activity 94.0 % 10.1128/aac.00426-09
Escherichia coli Escherichia coli Activity 94.4 % 10.1128/aac.01176-07
Escherichia coli Escherichia coli Activity 96.0 % 10.1128/aac.01808-09
Escherichia coli Escherichia coli Activity 96.5 % 10.1128/aac.00149-08
Escherichia coli Escherichia coli Activity 97.6 % 10.1128/aac.00400-09
Escherichia coli Escherichia coli Activity 98.0 % 10.1128/aac.01808-09
Escherichia coli Escherichia coli Activity 100.0 % 10.1128/aac.01176-07
Escherichia coli Escherichia coli Activity 100.0 % 10.1128/aac.01412-06
Escherichia coli Escherichia coli Activity nan None 10.1128/aac.00220-10
Escherichia coli Escherichia coli Activity nan None 10.1128/aac.00614-07
Escherichia coli Escherichia coli Activity nan None 10.1128/aac.01831-09
Escherichia coli Escherichia coli ED50 8.5 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 11.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 12.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 13.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 16.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 25.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 40.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 45.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 86.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 103.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 128.0 mg.kg-1 10.1016/j.bmc.2007.11.006
Escherichia coli Escherichia coli ED50 165.0 mg.kg-1 10.1021/jm060021p
Escherichia coli Escherichia coli ED50 176.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 256.0 mg.kg-1 10.1016/s0960-894x(99)00107-9
Escherichia coli Escherichia coli ED50 270.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 301.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli ED50 980.0 mg.kg-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli FC 2.0 None 10.1128/aac.01831-09
Escherichia coli Escherichia coli MBC 2.0 mg/L 10.1128/aac.01831-09
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1016/s0960-894x(99)00325-x
Escherichia coli Escherichia coli MIC 0.063 ug.mL-1 10.1128/aac.01395-06
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00381-08
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.01337-07
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli MIC 0.38 ug.mL-1 10.1128/aac.00163-08
Escherichia coli Escherichia coli MIC 0.38 ug.mL-1 10.1128/aac.00485-08
Escherichia coli Escherichia coli MIC 0.38 ug.mL-1 10.1128/aac.01145-07
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00149-08
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00219-09
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00389-07
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00774-09
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00856-09
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.01155-08
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.01284-08
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.01336-09
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.01561-09
Escherichia coli Escherichia coli MIC 0.75 ug.mL-1 10.1128/aac.00163-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1021/jm301490d
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00050-10
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00175-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00387-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00400-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00427-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00436-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00458-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00461-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00465-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00543-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00608-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00638-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00734-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00768-10
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00771-10
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00774-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00791-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00830-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00856-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00858-10
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00859-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00878-10
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00909-06
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00912-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.00961-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01028-07
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01062-07
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01082-06
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01152-06
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01155-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01164-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01176-07
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01180-07
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01252-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01284-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01359-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01442-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01456-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01462-06
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01463-07
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01539-07
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01561-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01581-08
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01585-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01600-06
Escherichia coli Escherichia coli MIC 1.024 ug.mL-1 10.1016/j.ejmech.2021.113975
Escherichia coli Escherichia coli MIC 1.5 ug.mL-1 10.1128/aac.00436-09
Escherichia coli Escherichia coli MIC 1.5 ug.mL-1 10.1128/aac.00465-08
Escherichia coli Escherichia coli MIC 1.5 ug.mL-1 10.1128/aac.00547-09
Escherichia coli Escherichia coli MIC 1.5 ug.mL-1 10.1128/aac.00684-07
Escherichia coli Escherichia coli MIC 1.5 ug.mL-1 10.1128/aac.01451-07
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00017-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00111-10
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00133-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00137-10
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00149-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00381-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00387-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00461-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00608-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00614-07
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00638-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00642-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00693-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00771-10
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00830-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00856-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00912-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00946-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01011-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01058-06
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01062-07
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01155-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01197-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01337-07
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01381-07
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01412-06
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01439-06
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01442-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01462-06
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01472-06
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01561-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01581-08
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01831-09
Escherichia coli Escherichia coli MIC 3.0 ug.mL-1 10.1128/aac.00485-08
Escherichia coli Escherichia coli MIC 3.13 ug.mL-1 10.1016/S0960-894X(96)00575-6
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1016/j.bmc.2007.07.048
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1016/j.bmc.2007.08.035
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1016/j.ejmech.2012.03.008
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1021/jm301490d
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1021/np500775e
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00158-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00175-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00299-07
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00485-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00608-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00638-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00688-09
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00746-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00771-10
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00912-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00946-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01011-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01082-06
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01337-07
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01341-07
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01381-07
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01442-09
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01463-07
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01581-08
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01672-07
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01818-09
Escherichia coli Escherichia coli MIC 6.0 ug.mL-1 10.1128/aac.00465-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1016/j.ejmech.2019.02.024
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1021/jm301490d
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00050-10
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00175-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00227-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00427-09
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00465-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00608-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00771-10
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00856-09
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00896-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00946-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.01011-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.01252-09
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.01336-09
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.01462-06
Escherichia coli Escherichia coli MIC 12.0 ug.mL-1 10.1128/aac.00133-09
Escherichia coli Escherichia coli MIC 12.0 ug.mL-1 10.1128/aac.00771-10
Escherichia coli Escherichia coli MIC 12.0 ug.mL-1 10.1128/aac.00912-08
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00050-10
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00219-09
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00274-09
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00461-09
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00642-08
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00688-09
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00791-09
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00912-08
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.01337-07
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.01561-09
Escherichia coli Escherichia coli MIC 24.0 ug.mL-1 10.1128/aac.00912-08
Escherichia coli Escherichia coli MIC 25.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.00050-10
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.00133-09
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.00274-09
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.00389-07
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.00436-09
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.00642-08
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.00859-09
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.01028-07
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.01152-06
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.01164-08
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.01284-08
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.01439-06
Escherichia coli Escherichia coli MIC 32.0 ug.mL-1 10.1128/aac.01585-09
Escherichia coli Escherichia coli MIC 46.0 ug.mL-1 10.1128/aac.01714-09
Escherichia coli Escherichia coli MIC 48.0 ug.mL-1 10.1128/aac.00436-09
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/0960-894X(95)00249-S
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/j.bmcl.2018.01.006
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/s0960-894x(00)00444-3
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/s0960-894x(01)00148-2
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/s0960-894x(99)00106-7
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/s0960-894x(99)00107-9
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1021/jm034056q
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.00133-09
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.00219-09
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.00227-08
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.00387-08
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.00389-07
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.00642-08
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.00688-09
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.00746-08
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.00896-08
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.00909-06
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.01155-08
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.01284-08
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.01341-07
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.01359-09
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.01381-07
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.01439-06
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.01442-09
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.01561-09
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1128/aac.01672-07
Escherichia coli Escherichia coli MIC 96.0 ug.mL-1 10.1128/aac.00436-09
Escherichia coli Escherichia coli MIC 96.0 ug.mL-1 10.1128/aac.00684-07
Escherichia coli Escherichia coli MIC 125.0 nM 10.1016/j.bmc.2015.03.016
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1016/0960-894X(95)00249-S
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.00050-10
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.00111-10
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.00133-09
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.00158-08
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.00219-09
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.00389-07
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.00543-08
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.00642-08
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.00734-08
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.00859-09
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01155-08
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01180-07
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01284-08
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01341-07
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01359-09
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01439-06
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01442-09
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01451-07
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli MIC 128.0 ug.mL-1 10.1128/aac.01600-06
Escherichia coli Escherichia coli MIC 200.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1016/j.ejmech.2019.02.024
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00050-10
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00133-09
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00137-10
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00163-08
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00389-07
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00458-09
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00461-09
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00547-09
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00638-08
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00642-08
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00734-08
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00774-09
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.00961-09
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01028-07
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01058-06
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01145-07
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01164-08
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01284-08
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01395-06
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01412-06
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01451-07
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01539-07
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01549-08
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01581-08
Escherichia coli Escherichia coli MIC 256.0 ug.mL-1 10.1128/aac.01585-09
Escherichia coli Escherichia coli MIC 400.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Escherichia coli Escherichia coli MIC 500.0 ug.mL-1 10.1128/aac.00537-07
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1021/np500775e
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.00017-09
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.00387-08
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.00458-09
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.00614-07
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.00642-08
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.00878-10
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.01058-06
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.01312-09
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.01412-06
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.01456-09
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.01672-07
Escherichia coli Escherichia coli MIC 1000.0 ug.mL-1 10.1128/aac.00537-07
Escherichia coli Escherichia coli MIC 1024.0 ug.mL-1 10.1128/aac.00017-09
Escherichia coli Escherichia coli MIC 1024.0 ug.mL-1 10.1128/aac.00197-10
Escherichia coli Escherichia coli MIC 1024.0 ug.mL-1 10.1128/aac.00693-09
Escherichia coli Escherichia coli MIC 1024.0 ug.mL-1 10.1128/aac.01058-06
Escherichia coli Escherichia coli MIC 1024.0 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 1282.0 ug.mL-1 10.1128/aac.01431-08
Escherichia coli Escherichia coli MIC 2000.0 nM 10.1128/aac.01381-07
Escherichia coli Escherichia coli MIC 2000.0 ug.mL-1 10.1128/aac.00537-07
Escherichia coli Escherichia coli MIC 2048.0 ug.mL-1 10.1021/jm301490d
Escherichia coli Escherichia coli MIC 2048.0 ug.mL-1 10.1128/aac.00017-09
Escherichia coli Escherichia coli MIC 2048.0 ug.mL-1 10.1128/aac.00614-07
Escherichia coli Escherichia coli MIC 2048.0 ug.mL-1 10.1128/aac.01058-06
Escherichia coli Escherichia coli MIC 4000.0 nM 10.1016/j.bmc.2015.03.016
Escherichia coli Escherichia coli MIC 4000.0 ug.mL-1 10.1128/aac.00537-07
Escherichia coli Escherichia coli MIC 4096.0 ug.mL-1 10.1021/jm301490d
Escherichia coli Escherichia coli MIC 8000.0 ug.mL-1 10.1128/aac.00537-07
Escherichia coli Escherichia coli MIC 32000.0 ug.mL-1 10.1128/aac.00537-07
Escherichia coli Escherichia coli MIC nan None 10.1128/aac.00736-08
Escherichia coli Escherichia coli MIC nan None 10.1128/aac.01607-08
Escherichia coli Escherichia coli MIC50 1.0 ug.mL-1 10.1128/aac.00149-08
Escherichia coli Escherichia coli MIC50 1.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC50 2.0 ug.mL-1 10.1128/aac.00400-09
Escherichia coli Escherichia coli MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC50 2.0 ug.mL-1 10.1128/aac.01176-07
Escherichia coli Escherichia coli MIC50 4.0 ug.mL-1 10.1128/aac.00381-08
Escherichia coli Escherichia coli MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC50 16.0 ug.mL-1 10.1128/aac.00149-08
Escherichia coli Escherichia coli MIC50 16.0 ug.mL-1 10.1128/aac.00381-08
Escherichia coli Escherichia coli MIC50 16.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC50 50.0 ug.mL-1 10.1021/jm00391a032
Escherichia coli Escherichia coli MIC50 64.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC50 64.0 ug.mL-1 10.1128/aac.01412-06
Escherichia coli Escherichia coli MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC50 128.0 ug.mL-1 10.1128/aac.01197-09
Escherichia coli Escherichia coli MIC70 200.0 ug.mL-1 10.1021/jm00391a032
Escherichia coli Escherichia coli MIC90 0.5 ug.mL-1 10.1128/aac.01197-09
Escherichia coli Escherichia coli MIC90 2.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC90 4.0 ug.mL-1 10.1128/aac.00149-08
Escherichia coli Escherichia coli MIC90 4.0 ug.mL-1 10.1128/aac.00400-09
Escherichia coli Escherichia coli MIC90 8.0 ug.mL-1 10.1128/aac.00381-08
Escherichia coli Escherichia coli MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC90 8.0 ug.mL-1 10.1128/aac.01176-07
Escherichia coli Escherichia coli MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC90 32.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC90 64.0 ug.mL-1 10.1128/aac.00149-08
Escherichia coli Escherichia coli MIC90 64.0 ug.mL-1 10.1128/aac.01412-06
Escherichia coli Escherichia coli MIC90 128.0 ug.mL-1 10.1128/aac.00381-08
Escherichia coli Escherichia coli MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Escherichia coli Escherichia coli MIC90 128.0 ug.mL-1 10.1128/aac.01197-09
Escherichia coli Escherichia coli permeability 0.3 um/s 10.1128/aac.01714-09
Escherichia coli Escherichia coli Ratio 4.0 None 10.1128/aac.00734-08
Escherichia coli Escherichia coli Ratio 16.0 None 10.1016/j.ejmech.2012.03.008
Escherichia coli Escherichia coli Ratio 16.0 None 10.1128/aac.00734-08
Escherichia coli Metallo-beta-lactamase Kcat 32.7 /s 10.1128/aac.00017-09
Escherichia coli Metallo-beta-lactamase Kcat/Km 0.45 /s/microM 10.1128/aac.00017-09
Escherichia coli Metallo-beta-lactamase VIM-19 Kcat 860.0 /s 10.1128/aac.00458-09
Escherichia coli Metallo-beta-lactamase VIM-19 Kcat/Km 4.0 /uM/s 10.1128/aac.00458-09
Escherichia coli Metallo-beta-lactamase VIM-19 Km 250000.0 nM 10.1128/aac.00458-09
Escherichia coli K-12 Beta-lactamase AmpC MIC 4.0 ug.mL-1 10.1016/j.bmcl.2003.12.037
Eubacterium sp. Eubacterium sp. Activity 0.0 % 10.1128/aac.00481-10
Eubacterium sp. Eubacterium sp. Activity 92.0 % 10.1128/aac.00481-10
Eubacterium sp. Eubacterium sp. MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Eubacterium sp. Eubacterium sp. MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Eubacterium sp. Eubacterium sp. MIC50 0.5 ug.mL-1 10.1128/aac.00481-10
Eubacterium sp. Eubacterium sp. MIC50 1.0 ug.mL-1 10.1128/aac.00481-10
Eubacterium sp. Eubacterium sp. MIC90 8.0 ug.mL-1 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna Activity 0.0 % 10.1128/aac.00355-08
Finegoldia magna Finegoldia magna Activity 0.0 % 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna Activity 0.0 % 10.1128/aac.00696-08
Finegoldia magna Finegoldia magna Activity 3.0 % 10.1128/aac.00355-08
Finegoldia magna Finegoldia magna Activity 97.0 % 10.1128/aac.00355-08
Finegoldia magna Finegoldia magna Activity 100.0 % 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Finegoldia magna Finegoldia magna MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Finegoldia magna Finegoldia magna MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Finegoldia magna Finegoldia magna MIC50 0.03 ug.mL-1 10.1128/aac.00355-08
Finegoldia magna Finegoldia magna MIC50 0.06 ug.mL-1 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna MIC50 0.12 ug.mL-1 10.1128/aac.00355-08
Finegoldia magna Finegoldia magna MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Finegoldia magna Finegoldia magna MIC90 0.125 ug.mL-1 10.1128/aac.00481-10
Finegoldia magna Finegoldia magna MIC90 0.25 ug.mL-1 10.1128/aac.01557-08
Finegoldia magna Finegoldia magna MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Finegoldia magna Finegoldia magna MIC90 8.0 ug.mL-1 10.1128/aac.00355-08
Fluoribacter gormanii FEZ-1 protein Kcat/Km 1.2 10'4/M/s 10.1128/aac.01062-07
Fusobacterium mortiferum Fusobacterium mortiferum Activity 0.0 % 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum Activity 10.0 % 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum Activity 90.0 % 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum Activity 100.0 % 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Fusobacterium mortiferum Fusobacterium mortiferum MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Fusobacterium mortiferum Fusobacterium mortiferum MIC 0.25 ug.mL-1 10.1128/aac.01557-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC50 0.25 ug.mL-1 10.1128/aac.01557-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC50 0.5 ug.mL-1 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC50 2.0 ug.mL-1 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC90 1.0 ug.mL-1 10.1128/aac.01557-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Fusobacterium mortiferum Fusobacterium mortiferum MIC90 8.0 ug.mL-1 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum Activity 0.0 % 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum Activity 10.0 % 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum Activity 90.0 % 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum Activity 100.0 % 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC50 0.5 ug.mL-1 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC50 2.0 ug.mL-1 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Fusobacterium necrophorum Fusobacterium necrophorum MIC90 8.0 ug.mL-1 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum Activity 0.0 % 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum Activity 10.0 % 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum Activity 90.0 % 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum Activity 100.0 % 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Fusobacterium nucleatum Fusobacterium nucleatum MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Fusobacterium nucleatum Fusobacterium nucleatum MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC50 0.5 ug.mL-1 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC50 2.0 ug.mL-1 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC90 0.125 ug.mL-1 10.1128/aac.01557-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Fusobacterium nucleatum Fusobacterium nucleatum MIC90 8.0 ug.mL-1 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium Activity 0.0 % 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium Activity 10.0 % 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium Activity 90.0 % 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium Activity 100.0 % 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Fusobacterium varium Fusobacterium varium MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Fusobacterium varium Fusobacterium varium MIC 1.0 ug.mL-1 10.1128/aac.01557-08
Fusobacterium varium Fusobacterium varium MIC50 0.5 ug.mL-1 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium MIC50 2.0 ug.mL-1 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium MIC50 4.0 ug.mL-1 10.1128/aac.01557-08
Fusobacterium varium Fusobacterium varium MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium MIC90 8.0 ug.mL-1 10.1128/aac.00355-08
Fusobacterium varium Fusobacterium varium MIC90 8.0 ug.mL-1 10.1128/aac.01557-08
Haemophilus influenzae Haemophilus influenzae Activity 0.0 % 10.1128/aac.00149-08
Haemophilus influenzae Haemophilus influenzae Activity 0.0 % 10.1128/aac.01538-07
Haemophilus influenzae Haemophilus influenzae Activity 0.3 % 10.1128/aac.01538-07
Haemophilus influenzae Haemophilus influenzae Activity 1.0 % 10.1128/aac.00149-08
Haemophilus influenzae Haemophilus influenzae Activity 99.0 % 10.1128/aac.00149-08
Haemophilus influenzae Haemophilus influenzae Activity 100.0 % 10.1128/aac.00149-08
Haemophilus influenzae Haemophilus influenzae Activity 100.0 % 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae IZ 21.0 mm 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC 0.004 ug.mL-1 10.1128/aac.01047-08
Haemophilus influenzae Haemophilus influenzae MIC 0.03 ug.mL-1 10.1128/aac.00149-08
Haemophilus influenzae Haemophilus influenzae MIC 0.03 ug.mL-1 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Haemophilus influenzae Haemophilus influenzae MIC 4.0 ug.mL-1 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC50 0.004 ug.mL-1 10.1128/aac.01047-08
Haemophilus influenzae Haemophilus influenzae MIC50 0.008 ug.mL-1 10.1128/aac.01047-08
Haemophilus influenzae Haemophilus influenzae MIC50 0.015 ug.mL-1 10.1128/aac.01047-08
Haemophilus influenzae Haemophilus influenzae MIC50 0.03 ug.mL-1 10.1128/aac.00149-08
Haemophilus influenzae Haemophilus influenzae MIC50 0.03 ug.mL-1 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC50 0.06 ug.mL-1 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC50 0.12 ug.mL-1 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC50 8.0 ug.mL-1 10.1128/aac.01047-08
Haemophilus influenzae Haemophilus influenzae MIC50 32.0 ug.mL-1 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC90 0.004 ug.mL-1 10.1128/aac.01047-08
Haemophilus influenzae Haemophilus influenzae MIC90 0.015 ug.mL-1 10.1128/aac.01047-08
Haemophilus influenzae Haemophilus influenzae MIC90 0.03 ug.mL-1 10.1128/aac.01047-08
Haemophilus influenzae Haemophilus influenzae MIC90 0.06 ug.mL-1 10.1128/aac.00149-08
Haemophilus influenzae Haemophilus influenzae MIC90 0.06 ug.mL-1 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC90 0.12 ug.mL-1 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC90 0.25 ug.mL-1 10.1128/aac.00192-09
Haemophilus influenzae Haemophilus influenzae MIC90 32.0 ug.mL-1 10.1128/aac.01047-08
Haemophilus influenzae Haemophilus influenzae MIC90 64.0 ug.mL-1 10.1128/aac.00192-09
Haemophilus parainfluenzae Haemophilus parainfluenzae MIC 0.004 ug.mL-1 10.1128/aac.01047-08
Haemophilus parainfluenzae Haemophilus parainfluenzae MIC50 0.004 ug.mL-1 10.1128/aac.01047-08
Haemophilus parainfluenzae Haemophilus parainfluenzae MIC50 0.06 ug.mL-1 10.1128/aac.01047-08
Haemophilus parainfluenzae Haemophilus parainfluenzae MIC90 0.004 ug.mL-1 10.1128/aac.01047-08
Haemophilus parainfluenzae Haemophilus parainfluenzae MIC90 0.25 ug.mL-1 10.1128/aac.01047-08
Haemophilus parainfluenzae Haemophilus parainfluenzae MIC90 0.5 ug.mL-1 10.1128/aac.01047-08
Homo sapiens Acetylcholinesterase IC50 nan None None
Homo sapiens Acetylcholinesterase Ki nan None None
Homo sapiens Adenosine A1 receptor IC50 nan None None
Homo sapiens Adenosine A1 receptor Ki nan None None
Homo sapiens Adenosine A2a receptor IC50 nan None None
Homo sapiens Adenosine A2a receptor Ki nan None None
Homo sapiens Adenosine A3 receptor IC50 nan None None
Homo sapiens Adenosine A3 receptor Ki nan None None
Homo sapiens Alpha-1d adrenergic receptor IC50 nan None None
Homo sapiens Alpha-1d adrenergic receptor Ki nan None None
Homo sapiens Alpha-2a adrenergic receptor IC50 nan None None
Homo sapiens Alpha-2a adrenergic receptor Ki nan None None
Homo sapiens Alpha-2b adrenergic receptor IC50 nan None None
Homo sapiens Alpha-2b adrenergic receptor Ki nan None None
Homo sapiens Alpha-2c adrenergic receptor IC50 nan None None
Homo sapiens Alpha-2c adrenergic receptor Ki nan None None
Homo sapiens Angiotensin II type 2 (AT-2) receptor IC50 nan None None
Homo sapiens Angiotensin II type 2 (AT-2) receptor Ki nan None None
Homo sapiens Beta-1 adrenergic receptor IC50 nan None None
Homo sapiens Beta-1 adrenergic receptor Ki nan None None
Homo sapiens Beta-2 adrenergic receptor IC50 nan None None
Homo sapiens Beta-2 adrenergic receptor Ki nan None None
Homo sapiens Beta-3 adrenergic receptor IC50 nan None None
Homo sapiens Beta-3 adrenergic receptor Ki nan None None
Homo sapiens Bile salt export pump IC50 197400.0 nM 10.1124/dmd.112.047068
Homo sapiens Bradykinin B2 receptor IC50 nan None None
Homo sapiens Bradykinin B2 receptor Ki nan None None
Homo sapiens Caco-2 Papp 3.25 10^-8cm/s 10.1016/j.bmc.2007.07.048
Homo sapiens Calcitonin receptor IC50 nan None None
Homo sapiens Calcitonin receptor Ki nan None None
Homo sapiens Cannabinoid CB1 receptor IC50 nan None None
Homo sapiens Cannabinoid CB1 receptor Ki nan None None
Homo sapiens Carbonic anhydrase II IC50 nan None None
Homo sapiens Carbonic anhydrase II Ki nan None None
Homo sapiens Caspase-1 IC50 nan None None
Homo sapiens Caspase-1 Ki nan None None
Homo sapiens Cathepsin G IC50 nan None None
Homo sapiens Cathepsin G Ki nan None None
Homo sapiens C-C chemokine receptor type 2 IC50 nan None None
Homo sapiens C-C chemokine receptor type 2 Ki nan None None
Homo sapiens C-C chemokine receptor type 4 IC50 nan None None
Homo sapiens C-C chemokine receptor type 4 Ki nan None None
Homo sapiens C-C chemokine receptor type 5 IC50 nan None None
Homo sapiens C-C chemokine receptor type 5 Ki nan None None
Homo sapiens Cholecystokinin A receptor IC50 nan None None
Homo sapiens Cholecystokinin A receptor Ki nan None None
Homo sapiens Cyclooxygenase-1 IC50 nan None None
Homo sapiens Cyclooxygenase-1 Ki nan None None
Homo sapiens Cyclooxygenase-2 IC50 nan None None
Homo sapiens Cyclooxygenase-2 Ki nan None None
Homo sapiens Cysteinyl leukotriene receptor 1 IC50 nan None None
Homo sapiens Cysteinyl leukotriene receptor 1 Ki nan None None
Homo sapiens Cytochrome P450 1A2 IC50 nan None None
Homo sapiens Cytochrome P450 1A2 Ki nan None None
Homo sapiens Cytochrome P450 2A6 IC50 nan None None
Homo sapiens Cytochrome P450 2A6 Ki nan None None
Homo sapiens Cytochrome P450 2C19 IC50 nan None None
Homo sapiens Cytochrome P450 2C19 Ki nan None None
Homo sapiens Cytochrome P450 2C9 IC50 nan None None
Homo sapiens Cytochrome P450 2C9 Ki nan None None
Homo sapiens Cytochrome P450 2D6 IC50 nan None None
Homo sapiens Cytochrome P450 2D6 Ki nan None None
Homo sapiens Cytochrome P450 2E1 IC50 nan None None
Homo sapiens Cytochrome P450 2E1 Ki nan None None
Homo sapiens Cytochrome P450 3A4 IC50 nan None None
Homo sapiens Cytochrome P450 3A4 Ki nan None None
Homo sapiens Delta opioid receptor IC50 nan None None
Homo sapiens Delta opioid receptor Ki nan None None
Homo sapiens Dopamine D1 receptor IC50 nan None None
Homo sapiens Dopamine D1 receptor Ki nan None None
Homo sapiens Dopamine D2 receptor IC50 nan None None
Homo sapiens Dopamine D2 receptor Ki nan None None
Homo sapiens Dopamine D3 receptor IC50 nan None None
Homo sapiens Dopamine D3 receptor Ki nan None None
Homo sapiens Dopamine D4 receptor IC50 nan None None
Homo sapiens Dopamine D4 receptor Ki nan None None
Homo sapiens Dopamine transporter IC50 nan None None
Homo sapiens Dopamine transporter Ki nan None None
Homo sapiens Endothelin receptor ET-A IC50 nan None None
Homo sapiens Endothelin receptor ET-A Ki nan None None
Homo sapiens Epidermal growth factor receptor erbB1 IC50 nan None None
Homo sapiens Epidermal growth factor receptor erbB1 Ki nan None None
Homo sapiens Estrogen receptor alpha IC50 nan None None
Homo sapiens Estrogen receptor alpha Ki nan None None
Homo sapiens Estrogen receptor beta IC50 nan None None
Homo sapiens Estrogen receptor beta Ki nan None None
Homo sapiens Glucocorticoid receptor IC50 nan None None
Homo sapiens Glucocorticoid receptor Ki nan None None
Homo sapiens HERG IC50 nan None None
Homo sapiens HERG Ki nan None None
Homo sapiens Histamine H1 receptor IC50 nan None None
Homo sapiens Histamine H1 receptor Ki nan None None
Homo sapiens Histamine H2 receptor IC50 nan None None
Homo sapiens Histamine H2 receptor Ki nan None None
Homo sapiens HMG-CoA reductase IC50 nan None None
Homo sapiens HMG-CoA reductase Ki nan None None
Homo sapiens Homo sapiens CL 4.0 mL.min-1.kg-1 10.1021/jm900403j
Homo sapiens Homo sapiens CL 8.78 L/hr 10.1128/aac.01477-06
Homo sapiens Homo sapiens CL 11.3 L/hr 10.1128/aac.01477-06
Homo sapiens Homo sapiens CL 11.7 L/hr 10.1128/aac.01477-06
Homo sapiens Homo sapiens CL_renal 3.2 mL.min-1.kg-1 10.1021/jm900403j
Homo sapiens Homo sapiens DILI_Concern nan None 10.1016/j.drudis.2016.02.015
Homo sapiens Homo sapiens DILI_severity_class 3.0 None 10.1016/j.drudis.2016.02.015
Homo sapiens Homo sapiens Drug uptake 446.0 mg/L 10.1128/aac.01477-06
Homo sapiens Homo sapiens Drug uptake 767.0 mg/L 10.1128/aac.01477-06
Homo sapiens Homo sapiens MRT 0.85 hr 10.1128/aac.01477-06
Homo sapiens Homo sapiens MRT 1.02 hr 10.1128/aac.01477-06
Homo sapiens Homo sapiens T1/2 0.69 hr 10.1128/aac.01477-06
Homo sapiens Homo sapiens T1/2 1.05 hr 10.1128/aac.01477-06
Homo sapiens Homo sapiens Vc 6.49 l 10.1128/aac.01477-06
Homo sapiens Homo sapiens Vc 7.01 l 10.1128/aac.01477-06
Homo sapiens Homo sapiens Vc/F 3.37 l 10.1128/aac.01477-06
Homo sapiens Homo sapiens Vdss 8.13 l 10.1128/aac.01477-06
Homo sapiens Homo sapiens Vdss 9.61 l 10.1128/aac.01477-06
Homo sapiens Homo sapiens Vdss 10.4 l 10.1128/aac.01477-06
Homo sapiens Homo sapiens Vdss 11.8 l 10.1128/aac.01477-06
Homo sapiens Homo sapiens Vp/F 3.12 l 10.1128/aac.01477-06
Homo sapiens Interleukin-8 receptor A IC50 nan None None
Homo sapiens Interleukin-8 receptor A Ki nan None None
Homo sapiens Interleukin-8 receptor B IC50 nan None None
Homo sapiens Interleukin-8 receptor B Ki nan None None
Homo sapiens Kappa opioid receptor IC50 nan None None
Homo sapiens Kappa opioid receptor Ki nan None None
Homo sapiens Leukocyte common antigen IC50 nan None None
Homo sapiens Leukocyte common antigen Ki nan None None
Homo sapiens Leukocyte elastase IC50 nan None None
Homo sapiens Leukocyte elastase Ki nan None None
Homo sapiens MAP kinase ERK1 IC50 nan None None
Homo sapiens MAP kinase ERK1 Ki nan None None
Homo sapiens MAP kinase ERK2 IC50 nan None None
Homo sapiens MAP kinase ERK2 Ki nan None None
Homo sapiens MAP kinase p38 alpha IC50 nan None None
Homo sapiens MAP kinase p38 alpha Ki nan None None
Homo sapiens Matrix metalloproteinase-1 IC50 nan None None
Homo sapiens Matrix metalloproteinase-1 Ki nan None None
Homo sapiens Matrix metalloproteinase 9 IC50 nan None None
Homo sapiens Matrix metalloproteinase 9 Ki nan None None
Homo sapiens Melanocortin receptor 3 IC50 nan None None
Homo sapiens Melanocortin receptor 3 Ki nan None None
Homo sapiens Melanocortin receptor 4 IC50 nan None None
Homo sapiens Melanocortin receptor 4 Ki nan None None
Homo sapiens Melanocortin receptor 5 IC50 nan None None
Homo sapiens Melanocortin receptor 5 Ki nan None None
Homo sapiens Monoamine oxidase A IC50 nan None None
Homo sapiens Monoamine oxidase A Ki nan None None
Homo sapiens Mu opioid receptor IC50 nan None None
Homo sapiens Mu opioid receptor Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M1 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M1 Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M2 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M2 Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M3 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M3 Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M4 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M4 Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M5 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M5 Ki nan None None
Homo sapiens Neurokinin 1 receptor IC50 nan None None
Homo sapiens Neurokinin 1 receptor Ki nan None None
Homo sapiens Neurokinin 2 receptor IC50 nan None None
Homo sapiens Neurokinin 2 receptor Ki nan None None
Homo sapiens Neuropeptide Y receptor type 1 IC50 nan None None
Homo sapiens Neuropeptide Y receptor type 1 Ki nan None None
Homo sapiens Neuropeptide Y receptor type 2 IC50 nan None None
Homo sapiens Neuropeptide Y receptor type 2 Ki nan None None
Homo sapiens Norepinephrine transporter IC50 nan None None
Homo sapiens Norepinephrine transporter Ki nan None None
Homo sapiens Oligopeptide transporter small intestine isoform Ki 30000000.0 nM 10.1021/jm048982w
Homo sapiens Phosphodiesterase 5A IC50 nan None None
Homo sapiens Phosphodiesterase 5A Ki nan None None
Homo sapiens Platelet activating factor receptor IC50 nan None None
Homo sapiens Platelet activating factor receptor Ki nan None None
Homo sapiens Protein kinase C alpha IC50 nan None None
Homo sapiens Protein kinase C alpha Ki nan None None
Homo sapiens Receptor protein-tyrosine kinase erbB-2 IC50 nan None None
Homo sapiens Receptor protein-tyrosine kinase erbB-2 Ki nan None None
Homo sapiens Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform IC50 nan None None
Homo sapiens Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform Ki nan None None
Homo sapiens Serotonin 2a (5-HT2a) receptor IC50 nan None None
Homo sapiens Serotonin 2a (5-HT2a) receptor Ki nan None None
Homo sapiens Serotonin 2b (5-HT2b) receptor IC50 nan None None
Homo sapiens Serotonin 2b (5-HT2b) receptor Ki nan None None
Homo sapiens Serotonin 2c (5-HT2c) receptor IC50 nan None None
Homo sapiens Serotonin 2c (5-HT2c) receptor Ki nan None None
Homo sapiens Serotonin 6 (5-HT6) receptor IC50 nan None None
Homo sapiens Serotonin 6 (5-HT6) receptor Ki nan None None
Homo sapiens Serotonin transporter IC50 nan None None
Homo sapiens Serotonin transporter Ki nan None None
Homo sapiens Sigma opioid receptor IC50 nan None None
Homo sapiens Sigma opioid receptor Ki nan None None
Homo sapiens Solute carrier family 22 member 8 Inhibition nan % 10.1124/dmd.112.049569
Homo sapiens Thromboxane-A synthase IC50 nan None None
Homo sapiens Thromboxane-A synthase Ki nan None None
Homo sapiens Tyrosine-protein kinase FYN IC50 nan None None
Homo sapiens Tyrosine-protein kinase FYN Ki nan None None
Homo sapiens Tyrosine-protein kinase LCK IC50 nan None None
Homo sapiens Tyrosine-protein kinase LCK Ki nan None None
Homo sapiens Vascular endothelial growth factor receptor 1 IC50 nan None None
Homo sapiens Vascular endothelial growth factor receptor 1 Ki nan None None
Homo sapiens Vasoactive intestinal polypeptide receptor 1 IC50 nan None None
Homo sapiens Vasoactive intestinal polypeptide receptor 1 Ki nan None None
Homo sapiens Vasopressin V1a receptor IC50 nan None None
Homo sapiens Vasopressin V1a receptor Ki nan None None
Homo sapiens Voltage-gated L-type calcium channel IC50 1226000.0 nM 10.1038/srep02100
Hoylesella loescheii Hoylesella loescheii MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Hoylesella oralis Hoylesella oralis Activity 0.0 % 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis Activity 11.0 % 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis Activity 78.0 % 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis Activity 100.0 % 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Hoylesella oralis Hoylesella oralis MIC 0.5 ug.mL-1 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis MIC50 0.03 ug.mL-1 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis MIC50 16.0 ug.mL-1 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis MIC90 4.0 ug.mL-1 10.1128/aac.00481-10
Hoylesella oralis Hoylesella oralis MIC90 128.0 ug.mL-1 10.1128/aac.00481-10
Janthinobacterium lividum THIN-B proetin Kcat/Km 2.0 10'5/M/s 10.1128/aac.01062-07
Klebsiella aerogenes Klebsiella aerogenes Activity 69.0 % 10.1128/aac.00426-09
Klebsiella aerogenes Klebsiella aerogenes Activity 88.0 % 10.1128/aac.01808-09
Klebsiella aerogenes Klebsiella aerogenes ED50 421.0 mg.kg-1 10.1021/jm060021p
Klebsiella aerogenes Klebsiella aerogenes MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Klebsiella aerogenes Klebsiella aerogenes MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Klebsiella aerogenes Klebsiella aerogenes MIC 8.0 ug.mL-1 10.1016/j.bmc.2007.07.048
Klebsiella aerogenes Klebsiella aerogenes MIC 8.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella aerogenes Klebsiella aerogenes MIC 12.5 ug.mL-1 10.1016/S0960-894X(96)00575-6
Klebsiella aerogenes Klebsiella aerogenes MIC 32.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella aerogenes Klebsiella aerogenes MIC 64.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Klebsiella aerogenes Klebsiella aerogenes MIC 100.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Klebsiella aerogenes Klebsiella aerogenes MIC 256.0 ug.mL-1 10.1128/aac.01028-07
Klebsiella aerogenes Klebsiella aerogenes MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella aerogenes Klebsiella aerogenes MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella aerogenes Klebsiella aerogenes MIC50 64.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella aerogenes Klebsiella aerogenes MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella aerogenes Klebsiella aerogenes MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella aerogenes Klebsiella aerogenes MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella aerogenes Klebsiella aerogenes MIC90 64.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella aerogenes Klebsiella aerogenes MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella oxytoca Klebsiella oxytoca Activity 1.0 % 10.1128/aac.00400-09
Klebsiella oxytoca Klebsiella oxytoca Activity 9.0 % 10.1128/aac.00400-09
Klebsiella oxytoca Klebsiella oxytoca Activity 68.0 % 10.1128/aac.00426-09
Klebsiella oxytoca Klebsiella oxytoca Activity 89.0 % 10.1128/aac.01808-09
Klebsiella oxytoca Klebsiella oxytoca Activity 90.0 % 10.1128/aac.00400-09
Klebsiella oxytoca Klebsiella oxytoca Activity 100.0 % 10.1128/aac.00426-09
Klebsiella oxytoca Klebsiella oxytoca MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Klebsiella oxytoca Klebsiella oxytoca MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Klebsiella oxytoca Klebsiella oxytoca MIC 1.0 ug.mL-1 10.1128/aac.00400-09
Klebsiella oxytoca Klebsiella oxytoca MIC 256.0 ug.mL-1 10.1128/aac.00260-09
Klebsiella oxytoca Klebsiella oxytoca MIC50 2.0 ug.mL-1 10.1128/aac.00400-09
Klebsiella oxytoca Klebsiella oxytoca MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella oxytoca Klebsiella oxytoca MIC50 8.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella oxytoca Klebsiella oxytoca MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella oxytoca Klebsiella oxytoca MIC90 16.0 ug.mL-1 10.1128/aac.00400-09
Klebsiella oxytoca Klebsiella oxytoca MIC90 64.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Beta-lactamase NDM-1 Kcat 14.0 /s 10.1128/aac.00774-09
Klebsiella pneumoniae Beta-lactamase NDM-1 Kcat/Km 1.17 /s/microM 10.1128/aac.00774-09
Klebsiella pneumoniae Beta-lactamase NDM-1 Km 12000.0 nM 10.1128/aac.00774-09
Klebsiella pneumoniae Beta-lactamase SHV-1 Kcat 1490.0 /s 10.1128/aac.01381-07
Klebsiella pneumoniae Beta-lactamase SHV-1 Kcat 1490.0 /s 10.1128/aac.01525-07
Klebsiella pneumoniae Beta-lactamase SHV-1 Kcat/Km 62.1 /uM/s 10.1128/aac.01381-07
Klebsiella pneumoniae Beta-lactamase SHV-1 Kcat/Km 62.5 /uM/s 10.1128/aac.01525-07
Klebsiella pneumoniae Beta-lactamase SHV-1 Km 24000.0 nM 10.1128/aac.01381-07
Klebsiella pneumoniae Beta-lactamase SHV-1 Km 24000.0 nM 10.1128/aac.01525-07
Klebsiella pneumoniae Beta-lactamase SHV-55 Kcat 27.0 /s 10.1128/aac.01525-07
Klebsiella pneumoniae Beta-lactamase SHV-55 Kcat/Km 3.7 /uM/s 10.1128/aac.01525-07
Klebsiella pneumoniae Beta-lactamase SHV-55 Km 8000.0 nM 10.1128/aac.01525-07
Klebsiella pneumoniae Beta-lactamase SHV-72 Kcat 1918.0 /s 10.1128/aac.01381-07
Klebsiella pneumoniae Beta-lactamase SHV-72 Kcat/Km 44.6 /uM/s 10.1128/aac.01381-07
Klebsiella pneumoniae Beta-lactamase SHV-72 Km 43000.0 nM 10.1128/aac.01381-07
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Kcat 24.0 /s 10.1128/aac.00491-07
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Kcat 51.0 /s 10.1128/aac.00197-10
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Kcat/Km 3.4 /uM/s 10.1128/aac.00197-10
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Kcat/Km 1333.0 /mM/s 10.1128/aac.00491-07
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Km 15000.0 nM 10.1128/aac.00197-10
Klebsiella pneumoniae Carbepenem-hydrolyzing beta-lactamase KPC Km 18000.0 nM 10.1128/aac.00491-07
Klebsiella pneumoniae Extended spectrum beta-lactamase CTX-M-71 Kcat 27.0 /s 10.1128/aac.00461-09
Klebsiella pneumoniae Extended spectrum beta-lactamase CTX-M-71 Km 3200.0 nM 10.1128/aac.00461-09
Klebsiella pneumoniae Extended spectrum beta-lactamase CTX-M-71 Ratio 8.4 None 10.1128/aac.00461-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 0.0 % 10.1128/aac.00556-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 0.0 % 10.1128/aac.01821-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 0.5 % 10.1128/aac.00149-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 1.3 % 10.1128/aac.00400-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 1.7 % 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 2.0 % 10.1128/aac.00400-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 2.4 % 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 6.1 % 10.1128/aac.01538-07
Klebsiella pneumoniae Klebsiella pneumoniae Activity 7.3 % 10.1128/aac.01538-07
Klebsiella pneumoniae Klebsiella pneumoniae Activity 9.3 % 10.1128/aac.01538-07
Klebsiella pneumoniae Klebsiella pneumoniae Activity 11.4 % 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 13.3 % 10.1128/aac.01538-07
Klebsiella pneumoniae Klebsiella pneumoniae Activity 16.7 % 10.1128/aac.01821-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 18.9 % 10.1128/aac.01538-07
Klebsiella pneumoniae Klebsiella pneumoniae Activity 24.2 % 10.1128/aac.00149-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 28.0 % 10.1128/aac.01808-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 38.2 % 10.1128/aac.00556-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 57.0 % 10.1128/aac.00426-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 62.1 % 10.1128/aac.00149-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 77.3 % 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 85.0 % 10.1128/aac.01808-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 94.0 % 10.1128/aac.00426-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 95.9 % 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae Activity 96.7 % 10.1128/aac.00400-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 97.0 % 10.1128/aac.01808-09
Klebsiella pneumoniae Klebsiella pneumoniae Activity 97.1 % 10.1128/aac.00149-08
Klebsiella pneumoniae Klebsiella pneumoniae ED50 23.0 mg.kg-1 10.1128/aac.01549-08
Klebsiella pneumoniae Klebsiella pneumoniae ED50 24.0 mg.kg-1 10.1128/aac.01549-08
Klebsiella pneumoniae Klebsiella pneumoniae ED50 28.0 mg.kg-1 10.1128/aac.01549-08
Klebsiella pneumoniae Klebsiella pneumoniae ED50 58.0 mg.kg-1 10.1128/aac.01549-08
Klebsiella pneumoniae Klebsiella pneumoniae ED50 193.0 mg.kg-1 10.1128/aac.01549-08
Klebsiella pneumoniae Klebsiella pneumoniae ED50 245.0 mg.kg-1 10.1128/aac.01549-08
Klebsiella pneumoniae Klebsiella pneumoniae log10cfu -1.76 None 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae log10cfu -0.34 None 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae log10cfu -0.32 None 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae log10cfu 0.03 None 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae log10cfu 0.25 None 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae log10cfu 2.93 None 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.06 ug.mL-1 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.25 ug.mL-1 10.1128/aac.00083-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.25 ug.mL-1 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.5 ug.mL-1 10.1128/aac.00149-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.5 ug.mL-1 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.00400-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.00830-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.00746-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.00830-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.01549-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 3.0 ug.mL-1 10.1128/aac.00746-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 3.0 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00387-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00746-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.00830-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.0 ug.mL-1 10.1128/aac.01197-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4.096 ug.mL-1 10.1016/j.ejmech.2021.113975
Klebsiella pneumoniae Klebsiella pneumoniae MIC 6.0 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.00736-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.00830-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.01549-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 12.0 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.00736-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.00830-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.00746-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01284-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01381-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1128/aac.00197-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1128/aac.00690-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1128/aac.01549-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1128/aac.01818-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 96.0 ug.mL-1 10.1128/aac.01312-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1128/aac.00158-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1128/aac.00299-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1128/aac.00690-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1128/aac.00909-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1128/aac.01284-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 128.0 ug.mL-1 10.1128/aac.01818-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1016/j.ejmech.2019.02.024
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.00011-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.00137-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.00260-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.00436-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.00461-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.00543-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.00690-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.00774-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.00830-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.01180-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.01301-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.01312-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.01451-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1128/aac.01539-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 320.0 ug.mL-1 10.1128/aac.01818-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 400.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Klebsiella pneumoniae Klebsiella pneumoniae MIC 512.0 ug.mL-1 10.1128/aac.00387-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 512.0 ug.mL-1 10.1128/aac.00458-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 512.0 ug.mL-1 10.1128/aac.01198-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 512.0 ug.mL-1 10.1128/aac.01312-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 512.0 ug.mL-1 10.1128/aac.01672-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1024.0 ug.mL-1 10.1128/aac.00017-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1024.0 ug.mL-1 10.1128/aac.00197-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1024.0 ug.mL-1 10.1128/aac.00693-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2000.0 nM 10.1128/aac.01381-07
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2048.0 ug.mL-1 10.1128/aac.00017-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 2.0 ug.mL-1 10.1128/aac.00149-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 2.0 ug.mL-1 10.1128/aac.00400-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 3.0 ug.mL-1 10.1128/aac.00746-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 4.0 ug.mL-1 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 8.0 ug.mL-1 10.1128/aac.00083-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 8.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 12.0 ug.mL-1 10.1128/aac.00746-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 16.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 32.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 64.0 ug.mL-1 10.1128/aac.00149-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 64.0 ug.mL-1 10.1128/aac.00556-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 64.0 ug.mL-1 10.1128/aac.00746-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 64.0 ug.mL-1 10.1128/aac.01821-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 128.0 ug.mL-1 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 128.0 ug.mL-1 10.1128/aac.01197-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 256.0 ug.mL-1 10.1128/aac.00746-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC50 512.0 ug.mL-1 10.1128/aac.01821-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 8.0 ug.mL-1 10.1128/aac.00149-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 8.0 ug.mL-1 10.1128/aac.00400-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 12.0 ug.mL-1 10.1128/aac.00746-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 16.0 ug.mL-1 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 24.0 ug.mL-1 10.1128/aac.00746-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 32.0 ug.mL-1 10.1128/aac.00083-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 32.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 64.0 ug.mL-1 10.1128/aac.00083-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 64.0 ug.mL-1 10.1128/aac.00149-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 64.0 ug.mL-1 10.1128/aac.00556-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 64.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 128.0 ug.mL-1 10.1128/aac.00381-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 128.0 ug.mL-1 10.1128/aac.01197-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 128.0 ug.mL-1 10.1128/aac.01821-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 256.0 ug.mL-1 10.1128/aac.00746-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC90 512.0 ug.mL-1 10.1128/aac.01821-09
Klebsiella pneumoniae Metallo-beta-lactamase VIM-2 Kcat 33.0 /s 10.1128/aac.00774-09
Klebsiella pneumoniae Metallo-beta-lactamase VIM-2 Kcat/Km 0.45 /s/microM 10.1128/aac.00774-09
Klebsiella pneumoniae Metallo-beta-lactamase VIM-2 Km 72000.0 nM 10.1128/aac.00774-09
Listeria monocytogenes Listeria monocytogenes IZ 30.7 mm 10.1128/aac.00503-10
Listeria monocytogenes Listeria monocytogenes IZ 35.3 mm 10.1128/aac.00503-10
Micrococcus luteus Micrococcus luteus MIC 0.06 ug.mL-1 10.1016/s0960-894x(03)00512-2
Moraxella catarrhalis Moraxella catarrhalis MIC 0.004 ug.mL-1 10.1128/aac.01047-08
Moraxella catarrhalis Moraxella catarrhalis MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Moraxella catarrhalis Moraxella catarrhalis MIC 1.0 ug.mL-1 10.1128/aac.00400-09
Moraxella catarrhalis Moraxella catarrhalis MIC50 0.004 ug.mL-1 10.1128/aac.01047-08
Moraxella catarrhalis Moraxella catarrhalis MIC50 0.25 ug.mL-1 10.1128/aac.01047-08
Moraxella catarrhalis Moraxella catarrhalis MIC50 1.0 ug.mL-1 10.1128/aac.00400-09
Moraxella catarrhalis Moraxella catarrhalis MIC90 0.008 ug.mL-1 10.1128/aac.01047-08
Moraxella catarrhalis Moraxella catarrhalis MIC90 0.015 ug.mL-1 10.1128/aac.01047-08
Moraxella catarrhalis Moraxella catarrhalis MIC90 1.0 ug.mL-1 10.1128/aac.00400-09
Moraxella catarrhalis Moraxella catarrhalis MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Morganella morganii Morganella morganii Activity 0.0 % 10.1128/aac.00149-08
Morganella morganii Morganella morganii Activity 100.0 % 10.1128/aac.00149-08
Morganella morganii Morganella morganii MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Morganella morganii Morganella morganii MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Morganella morganii Morganella morganii MIC 0.5 ug.mL-1 10.1128/aac.00149-08
Morganella morganii Morganella morganii MIC 50.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Morganella morganii Morganella morganii MIC50 0.25 ug.mL-1 10.1128/aac.01047-08
Morganella morganii Morganella morganii MIC50 0.5 ug.mL-1 10.1128/aac.00149-08
Morganella morganii Morganella morganii MIC50 0.5 ug.mL-1 10.1128/aac.01047-08
Morganella morganii Morganella morganii MIC50 8.0 ug.mL-1 10.1128/aac.01047-08
Morganella morganii Morganella morganii MIC90 1.0 ug.mL-1 10.1128/aac.00149-08
Morganella morganii Morganella morganii MIC90 1.0 ug.mL-1 10.1128/aac.01047-08
Morganella morganii Morganella morganii MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Mus musculus Mus musculus ED50 128.0 mg.kg-1 10.1016/s0960-894x(99)00106-7
Mus musculus Mus musculus ED50 256.0 mg.kg-1 10.1016/s0960-894x(99)00106-7
Mus musculus Nitric oxide synthase, inducible IC50 nan None None
Mus musculus Nitric oxide synthase, inducible Ki nan None None
Mus musculus Solute carrier family 22 member 6 Inhibition nan % 10.1124/dmd.112.049569
Mus musculus Solute carrier family 22 member 8 Inhibition nan % 10.1124/dmd.112.049569
Mus musculus Solute carrier family 22 member 8 PPB nan % 10.1124/dmd.112.049569
Oryctolagus cuniculus Angiotensin-converting enzyme IC50 nan None None
Oryctolagus cuniculus Angiotensin-converting enzyme Ki nan None None
Oryctolagus cuniculus Arachidonate 15-lipoxygenase IC50 nan None None
Oryctolagus cuniculus Arachidonate 15-lipoxygenase Ki nan None None
Paeniclostridium sordellii Paeniclostridium sordellii MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Parabacteroides distasonis Parabacteroides distasonis Activity 0.0 % 10.1128/aac.00081-08
Parabacteroides distasonis Parabacteroides distasonis Activity 0.0 % 10.1128/aac.00696-08
Parabacteroides distasonis Parabacteroides distasonis Activity 7.0 % 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis Activity 42.0 % 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis Activity 51.0 % 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis Activity 89.0 % 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis MIC 0.06 ug.mL-1 10.1128/aac.00081-08
Parabacteroides distasonis Parabacteroides distasonis MIC 0.25 ug.mL-1 10.1128/aac.00696-08
Parabacteroides distasonis Parabacteroides distasonis MIC 1.0 ug.mL-1 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis MIC 2.0 ug.mL-1 10.1128/aac.01557-08
Parabacteroides distasonis Parabacteroides distasonis MIC 8.0 ug.mL-1 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis MIC 8.0 ug.mL-1 10.1128/aac.00696-08
Parabacteroides distasonis Parabacteroides distasonis MIC 16.0 ug.mL-1 10.1128/aac.00696-08
Parabacteroides distasonis Parabacteroides distasonis MIC50 4.0 ug.mL-1 10.1128/aac.01557-08
Parabacteroides distasonis Parabacteroides distasonis MIC50 8.0 ug.mL-1 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis MIC50 16.0 ug.mL-1 10.1128/aac.00081-08
Parabacteroides distasonis Parabacteroides distasonis MIC50 128.0 ug.mL-1 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis MIC90 4.0 ug.mL-1 10.1128/aac.01557-08
Parabacteroides distasonis Parabacteroides distasonis MIC90 16.0 ug.mL-1 10.1128/aac.00081-08
Parabacteroides distasonis Parabacteroides distasonis MIC90 64.0 ug.mL-1 10.1128/aac.00481-10
Parabacteroides distasonis Parabacteroides distasonis MIC90 256.0 ug.mL-1 10.1128/aac.00481-10
Parabacteroides merdae Parabacteroides merdae Activity 0.0 % 10.1128/aac.00081-08
Parabacteroides merdae Parabacteroides merdae Activity 0.0 % 10.1128/aac.00696-08
Parabacteroides merdae Parabacteroides merdae MIC 0.06 ug.mL-1 10.1128/aac.00081-08
Parabacteroides merdae Parabacteroides merdae MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Parabacteroides merdae Parabacteroides merdae MIC 4.0 ug.mL-1 10.1128/aac.00696-08
Parabacteroides merdae Parabacteroides merdae MIC 8.0 ug.mL-1 10.1128/aac.00696-08
Parabacteroides merdae Parabacteroides merdae MIC50 8.0 ug.mL-1 10.1128/aac.00081-08
Parabacteroides merdae Parabacteroides merdae MIC90 32.0 ug.mL-1 10.1128/aac.00081-08
Paraclostridium bifermentans Paraclostridium bifermentans MIC 0.5 ug.mL-1 10.1128/aac.01557-08
Parvimonas micra Parvimonas micra Activity 0.0 % 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra Activity 0.0 % 10.1128/aac.00481-10
Parvimonas micra Parvimonas micra Activity 0.0 % 10.1128/aac.00696-08
Parvimonas micra Parvimonas micra Activity 3.0 % 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra Activity 97.0 % 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra MIC 0.015 ug.mL-1 10.1128/aac.01047-08
Parvimonas micra Parvimonas micra MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Parvimonas micra Parvimonas micra MIC 0.03 ug.mL-1 10.1128/aac.01047-08
Parvimonas micra Parvimonas micra MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Parvimonas micra Parvimonas micra MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Parvimonas micra Parvimonas micra MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Parvimonas micra Parvimonas micra MIC50 0.015 ug.mL-1 10.1128/aac.01047-08
Parvimonas micra Parvimonas micra MIC50 0.03 ug.mL-1 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra MIC50 0.03 ug.mL-1 10.1128/aac.01047-08
Parvimonas micra Parvimonas micra MIC50 0.12 ug.mL-1 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra MIC50 0.12 ug.mL-1 10.1128/aac.01047-08
Parvimonas micra Parvimonas micra MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Parvimonas micra Parvimonas micra MIC50 0.25 ug.mL-1 10.1128/aac.00481-10
Parvimonas micra Parvimonas micra MIC90 0.015 ug.mL-1 10.1128/aac.01047-08
Parvimonas micra Parvimonas micra MIC90 0.125 ug.mL-1 10.1128/aac.01557-08
Parvimonas micra Parvimonas micra MIC90 0.25 ug.mL-1 10.1128/aac.01047-08
Parvimonas micra Parvimonas micra MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra MIC90 8.0 ug.mL-1 10.1128/aac.00355-08
Parvimonas micra Parvimonas micra MIC90 16.0 ug.mL-1 10.1128/aac.00481-10
Pasteurella sp. Pasteurella sp. Activity 23.0 % 10.1128/aac.01808-09
Pectobacterium atrosepticum Pectobacterium atrosepticum MIC 64.0 ug.mL-1 10.1128/aac.01062-07
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus Activity 0.0 % 10.1128/aac.00355-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus Activity 0.0 % 10.1128/aac.00481-10
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus Activity 0.0 % 10.1128/aac.00696-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus Activity 3.0 % 10.1128/aac.00355-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus Activity 97.0 % 10.1128/aac.00355-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus Activity 100.0 % 10.1128/aac.00481-10
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC50 0.03 ug.mL-1 10.1128/aac.00355-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC50 0.03 ug.mL-1 10.1128/aac.00481-10
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC50 0.06 ug.mL-1 10.1128/aac.00481-10
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC50 0.12 ug.mL-1 10.1128/aac.00355-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC90 0.06 ug.mL-1 10.1128/aac.00481-10
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC90 8.0 ug.mL-1 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius Activity 0.0 % 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius Activity 3.0 % 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius Activity 97.0 % 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius Activity 100.0 % 10.1128/aac.00481-10
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC 0.015 ug.mL-1 10.1128/aac.01047-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC 0.25 ug.mL-1 10.1128/aac.01557-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC50 0.015 ug.mL-1 10.1128/aac.01047-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC50 0.03 ug.mL-1 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC50 0.06 ug.mL-1 10.1128/aac.01047-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC50 0.12 ug.mL-1 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC50 0.25 ug.mL-1 10.1128/aac.00481-10
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC50 0.25 ug.mL-1 10.1128/aac.01557-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC90 0.015 ug.mL-1 10.1128/aac.01047-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC90 0.06 ug.mL-1 10.1128/aac.01047-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC90 2.0 ug.mL-1 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC90 8.0 ug.mL-1 10.1128/aac.00355-08
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC90 16.0 ug.mL-1 10.1128/aac.00481-10
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC90 16.0 ug.mL-1 10.1128/aac.01557-08
Peptostreptococcus sp. Peptostreptococcus sp. Activity 0.0 % 10.1128/aac.00696-08
Peptostreptococcus sp. Peptostreptococcus sp. MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Phocaeicola vulgatus Phocaeicola vulgatus Activity 0.0 % 10.1128/aac.00081-08
Phocaeicola vulgatus Phocaeicola vulgatus Activity 0.0 % 10.1128/aac.00696-08
Phocaeicola vulgatus Phocaeicola vulgatus Activity 4.0 % 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus Activity 7.0 % 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus Activity 35.0 % 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus Activity 42.0 % 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus Activity 51.0 % 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus Activity 65.0 % 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus Activity 89.0 % 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus Activity 96.0 % 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC 0.06 ug.mL-1 10.1128/aac.00081-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC 1.0 ug.mL-1 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus MIC 1.0 ug.mL-1 10.1128/aac.01557-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC 2.0 ug.mL-1 10.1128/aac.00696-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC 8.0 ug.mL-1 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC 8.0 ug.mL-1 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus MIC 16.0 ug.mL-1 10.1128/aac.00696-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC50 2.0 ug.mL-1 10.1128/aac.01557-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC50 8.0 ug.mL-1 10.1128/aac.00081-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC50 8.0 ug.mL-1 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC50 8.0 ug.mL-1 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus MIC50 128.0 ug.mL-1 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC50 128.0 ug.mL-1 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 16.0 ug.mL-1 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 16.0 ug.mL-1 10.1128/aac.01557-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 32.0 ug.mL-1 10.1128/aac.00081-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 64.0 ug.mL-1 10.1128/aac.00481-10
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 128.0 ug.mL-1 10.1128/aac.00355-08
Phocaeicola vulgatus Phocaeicola vulgatus MIC90 256.0 ug.mL-1 10.1128/aac.00481-10
Porphyromonas asaccharolytica Porphyromonas asaccharolytica MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Porphyromonas asaccharolytica Porphyromonas asaccharolytica MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Porphyromonas asaccharolytica Porphyromonas asaccharolytica MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Porphyromonas gingivalis Porphyromonas gingivalis MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella bivia Prevotella bivia Activity 0.0 % 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia Activity 0.0 % 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia Activity 11.0 % 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia Activity 22.0 % 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia Activity 71.0 % 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia Activity 78.0 % 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia Activity 100.0 % 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia Activity 100.0 % 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia MIC 0.06 ug.mL-1 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella bivia Prevotella bivia MIC 0.5 ug.mL-1 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia MIC50 0.03 ug.mL-1 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia MIC50 0.03 ug.mL-1 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella bivia Prevotella bivia MIC50 16.0 ug.mL-1 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia MIC50 16.0 ug.mL-1 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia MIC90 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella bivia Prevotella bivia MIC90 1.0 ug.mL-1 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia MIC90 4.0 ug.mL-1 10.1128/aac.00481-10
Prevotella bivia Prevotella bivia MIC90 128.0 ug.mL-1 10.1128/aac.00355-08
Prevotella bivia Prevotella bivia MIC90 128.0 ug.mL-1 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae Activity 0.0 % 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae Activity 0.0 % 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae Activity 11.0 % 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae Activity 22.0 % 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae Activity 71.0 % 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae Activity 78.0 % 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae Activity 100.0 % 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae Activity 100.0 % 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae MIC 0.06 ug.mL-1 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella buccae Prevotella buccae MIC 0.5 ug.mL-1 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae MIC50 0.03 ug.mL-1 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae MIC50 0.03 ug.mL-1 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella buccae Prevotella buccae MIC50 16.0 ug.mL-1 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae MIC50 16.0 ug.mL-1 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae MIC90 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella buccae Prevotella buccae MIC90 1.0 ug.mL-1 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae MIC90 4.0 ug.mL-1 10.1128/aac.00481-10
Prevotella buccae Prevotella buccae MIC90 128.0 ug.mL-1 10.1128/aac.00355-08
Prevotella buccae Prevotella buccae MIC90 128.0 ug.mL-1 10.1128/aac.00481-10
Prevotella corporis Prevotella corporis MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella corporis Prevotella corporis MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella denticola Prevotella denticola MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella denticola Prevotella denticola MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella denticola Prevotella denticola MIC90 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella disiens Prevotella disiens MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella disiens Prevotella disiens MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella intermedia Prevotella intermedia Activity 0.0 % 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia Activity 0.0 % 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia Activity 22.0 % 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia Activity 71.0 % 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia Activity 100.0 % 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia Activity 100.0 % 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia MIC 0.06 ug.mL-1 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella intermedia Prevotella intermedia MIC 2.0 ug.mL-1 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia MIC50 0.03 ug.mL-1 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia MIC50 0.03 ug.mL-1 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella intermedia Prevotella intermedia MIC50 8.0 ug.mL-1 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia MIC50 16.0 ug.mL-1 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia MIC90 0.03 ug.mL-1 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia MIC90 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella intermedia Prevotella intermedia MIC90 1.0 ug.mL-1 10.1128/aac.00355-08
Prevotella intermedia Prevotella intermedia MIC90 16.0 ug.mL-1 10.1128/aac.00481-10
Prevotella intermedia Prevotella intermedia MIC90 128.0 ug.mL-1 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica Activity 0.0 % 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica Activity 22.0 % 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica Activity 71.0 % 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica Activity 100.0 % 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica MIC 0.06 ug.mL-1 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella melaninogenica Prevotella melaninogenica MIC50 0.03 ug.mL-1 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella melaninogenica Prevotella melaninogenica MIC50 16.0 ug.mL-1 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica MIC90 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella melaninogenica Prevotella melaninogenica MIC90 1.0 ug.mL-1 10.1128/aac.00355-08
Prevotella melaninogenica Prevotella melaninogenica MIC90 128.0 ug.mL-1 10.1128/aac.00355-08
Prevotella nigrescens Prevotella nigrescens MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella nigrescens Prevotella nigrescens MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
Prevotella nigrescens Prevotella nigrescens MIC90 0.125 ug.mL-1 10.1128/aac.01557-08
Propionibacterium Propionibacterium Activity 0.0 % 10.1128/aac.00696-08
Propionibacterium Propionibacterium MIC 0.25 ug.mL-1 10.1128/aac.00696-08
Propionibacterium Propionibacterium MIC 0.5 ug.mL-1 10.1128/aac.00696-08
Proteus mirabilis Proteus mirabilis Activity 0.0 % 10.1128/aac.00149-08
Proteus mirabilis Proteus mirabilis Activity 0.0 % 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis Activity 0.0 % 10.1128/aac.00400-09
Proteus mirabilis Proteus mirabilis Activity 0.3 % 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis Activity 97.0 % 10.1128/aac.00426-09
Proteus mirabilis Proteus mirabilis Activity 99.4 % 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis Activity 100.0 % 10.1128/aac.00149-08
Proteus mirabilis Proteus mirabilis Activity 100.0 % 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis Activity 100.0 % 10.1128/aac.00400-09
Proteus mirabilis Proteus mirabilis Activity 100.0 % 10.1128/aac.01808-09
Proteus mirabilis Proteus mirabilis MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Proteus mirabilis Proteus mirabilis MIC 0.25 ug.mL-1 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis MIC 0.5 ug.mL-1 10.1128/aac.00149-08
Proteus mirabilis Proteus mirabilis MIC 0.5 ug.mL-1 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis MIC 1.0 ug.mL-1 10.1128/aac.00400-09
Proteus mirabilis Proteus mirabilis MIC 1.0 ug.mL-1 10.1128/aac.01197-09
Proteus mirabilis Proteus mirabilis MIC 16.0 ug.mL-1 10.1128/aac.00111-10
Proteus mirabilis Proteus mirabilis MIC 128.0 ug.mL-1 10.1128/aac.00111-10
Proteus mirabilis Proteus mirabilis MIC50 0.25 ug.mL-1 10.1128/aac.01047-08
Proteus mirabilis Proteus mirabilis MIC50 0.5 ug.mL-1 10.1128/aac.00149-08
Proteus mirabilis Proteus mirabilis MIC50 0.5 ug.mL-1 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis MIC50 2.0 ug.mL-1 10.1128/aac.00400-09
Proteus mirabilis Proteus mirabilis MIC50 32.0 ug.mL-1 10.1128/aac.01197-09
Proteus mirabilis Proteus mirabilis MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Proteus mirabilis Proteus mirabilis MIC90 0.5 ug.mL-1 10.1128/aac.01047-08
Proteus mirabilis Proteus mirabilis MIC90 1.0 ug.mL-1 10.1128/aac.00149-08
Proteus mirabilis Proteus mirabilis MIC90 2.0 ug.mL-1 10.1128/aac.00381-08
Proteus mirabilis Proteus mirabilis MIC90 2.0 ug.mL-1 10.1128/aac.01047-08
Proteus mirabilis Proteus mirabilis MIC90 64.0 ug.mL-1 10.1128/aac.00400-09
Proteus mirabilis Proteus mirabilis MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Proteus mirabilis Proteus mirabilis MIC90 128.0 ug.mL-1 10.1128/aac.01197-09
Proteus vulgaris Proteus vulgaris MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Proteus vulgaris Proteus vulgaris MIC 16.0 ug.mL-1 10.1128/aac.00274-09
Proteus vulgaris Proteus vulgaris MIC 32.0 ug.mL-1 10.1128/aac.00274-09
Proteus vulgaris Proteus vulgaris MIC 200.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Proteus vulgaris Proteus vulgaris MIC50 0.5 ug.mL-1 10.1128/aac.01047-08
Proteus vulgaris Proteus vulgaris MIC50 64.0 ug.mL-1 10.1128/aac.01047-08
Proteus vulgaris Proteus vulgaris MIC90 1.0 ug.mL-1 10.1128/aac.01047-08
Proteus vulgaris Proteus vulgaris MIC90 2.0 ug.mL-1 10.1128/aac.01047-08
Proteus vulgaris Proteus vulgaris MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Providencia rettgeri Providencia rettgeri MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Providencia rettgeri Providencia rettgeri MIC 256.0 ug.mL-1 10.1128/aac.01312-09
Providencia rettgeri Providencia rettgeri MIC50 1.0 ug.mL-1 10.1128/aac.01047-08
Providencia rettgeri Providencia rettgeri MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Providencia rettgeri Providencia rettgeri MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Providencia rettgeri Providencia rettgeri MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Providencia rettgeri Providencia rettgeri MIC90 1285.0 ug.mL-1 10.1128/aac.01047-08
Providencia sp. Providencia sp. Activity 3.7 % 10.1128/aac.00149-08
Providencia sp. Providencia sp. Activity 92.6 % 10.1128/aac.00149-08
Providencia sp. Providencia sp. MIC 0.5 ug.mL-1 10.1128/aac.00149-08
Providencia sp. Providencia sp. MIC50 2.0 ug.mL-1 10.1128/aac.00149-08
Providencia sp. Providencia sp. MIC90 16.0 ug.mL-1 10.1128/aac.00149-08
Providencia stuartii Providencia stuartii MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Providencia stuartii Providencia stuartii MIC 32.0 ug.mL-1 10.1128/aac.00274-09
Providencia stuartii Providencia stuartii MIC 256.0 ug.mL-1 10.1128/aac.00017-09
Providencia stuartii Providencia stuartii MIC50 1.0 ug.mL-1 10.1128/aac.01047-08
Providencia stuartii Providencia stuartii MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Providencia stuartii Providencia stuartii MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Providencia stuartii Providencia stuartii MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Providencia stuartii Providencia stuartii MIC90 1285.0 ug.mL-1 10.1128/aac.01047-08
Pseudomonas aeruginosa Beta-lactamase Kcat 1.1 /s 10.1128/aac.00859-09
Pseudomonas aeruginosa Beta-lactamase Kcat 5.0 /s 10.1128/aac.01410-08
Pseudomonas aeruginosa Beta-lactamase Kcat/Km 125.0 /uM/s 10.1128/aac.01410-08
Pseudomonas aeruginosa Beta-lactamase Kcat/Km 300.0 /mM/s 10.1128/aac.00859-09
Pseudomonas aeruginosa Beta-lactamase Km 300.0 nM 10.1128/aac.00859-09
Pseudomonas aeruginosa Beta-lactamase Km 40000.0 nM 10.1128/aac.01410-08
Pseudomonas aeruginosa Beta-lactamase bla(BEL1) Kcat 2.0 /s 10.1128/aac.00859-09
Pseudomonas aeruginosa Beta-lactamase bla(BEL1) Kcat/Km 130.0 /mM/s 10.1128/aac.00859-09
Pseudomonas aeruginosa Beta-lactamase bla(BEL1) Km 15000.0 nM 10.1128/aac.00859-09
Pseudomonas aeruginosa Beta-lactamase VIM-1 Kcat 374.0 /s 10.1128/aac.00465-08
Pseudomonas aeruginosa Beta-lactamase VIM-1 Kcat/Km 2.7 /M/s 10.1128/aac.00465-08
Pseudomonas aeruginosa Beta-lactamase VIM-1 Km 1377000.0 nM 10.1128/aac.00465-08
Pseudomonas aeruginosa Beta-lactamase VIM-2 Kcat 300.0 /s 10.1128/aac.00166-08
Pseudomonas aeruginosa Beta-lactamase VIM-2 Kcat/Km 2.4 /uM/s 10.1128/aac.00166-08
Pseudomonas aeruginosa Beta-lactamase VIM-2 Km 125000.0 nM 10.1128/aac.00166-08
Pseudomonas aeruginosa Class B carbapenemase VIM-13 Kcat 362.0 /s 10.1128/aac.00465-08
Pseudomonas aeruginosa Class B carbapenemase VIM-13 Kcat/Km 4.9 /M/s 10.1128/aac.00465-08
Pseudomonas aeruginosa Class B carbapenemase VIM-13 Km 729000.0 nM 10.1128/aac.00465-08
Pseudomonas aeruginosa Metallo-b-lactamase Kcat 140.0 /s 10.1128/aac.00166-08
Pseudomonas aeruginosa Metallo-b-lactamase Kcat/Km 5.4 /uM/s 10.1128/aac.00166-08
Pseudomonas aeruginosa Metallo-b-lactamase Km 26000.0 nM 10.1128/aac.00166-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 0.0 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 0.0 % 10.1128/aac.00400-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 0.0 % 10.1128/aac.01538-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 1.3 % 10.1128/aac.01538-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 2.5 % 10.1128/aac.01538-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 3.7 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 7.3 % 10.1128/aac.00400-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 9.0 % 10.1128/aac.00810-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 9.4 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 13.0 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 14.0 % 10.1128/aac.00679-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 17.3 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 19.0 % 10.1128/aac.00679-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 21.0 % 10.1128/aac.01483-06
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 21.6 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 27.1 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 28.0 % 10.1128/aac.00810-07
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 28.4 % 10.1128/aac.00834-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 34.8 % 10.1128/aac.00453-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 39.0 % 10.1128/aac.00707-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 39.5 % 10.1128/aac.00453-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 72.9 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 78.4 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 81.0 % 10.1128/aac.00426-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 82.7 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 83.0 % 10.1128/aac.01808-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 87.0 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 90.6 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 92.7 % 10.1128/aac.00400-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 96.3 % 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity 256.0 ug ml-1 10.1128/aac.01043-06
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity nan None 10.1128/aac.00428-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity nan None 10.1128/aac.01278-06
Pseudomonas aeruginosa Pseudomonas aeruginosa ED50 103.0 mg.kg-1 10.1128/aac.01549-08
Pseudomonas aeruginosa Pseudomonas aeruginosa ED50 246.0 mg.kg-1 10.1128/aac.01549-08
Pseudomonas aeruginosa Pseudomonas aeruginosa ED50 980.0 mg.kg-1 10.1128/aac.01549-08
Pseudomonas aeruginosa Pseudomonas aeruginosa FICI nan None 10.1128/aac.01071-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.25 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.38 ug.mL-1 10.1128/aac.01451-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.5 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.00400-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.0 ug.mL-1 10.1128/aac.01617-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1.5 ug.mL-1 10.1128/aac.01617-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00428-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00810-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00822-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1128/aac.00900-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 3.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 3.0 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 3.0 ug.mL-1 10.1128/aac.00465-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 3.0 ug.mL-1 10.1128/aac.00900-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 3.1 ug.mL-1 10.1128/aac.00464-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1016/j.bmc.2007.07.048
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00341-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00834-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.01047-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.01104-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.01172-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.01197-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.01360-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.01549-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 6.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 7.5 ug.mL-1 10.1128/aac.01071-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1016/s0960-894x(00)00444-3
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.01172-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1128/aac.01573-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 12.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 12.0 ug.mL-1 10.1128/aac.01573-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 12.5 ug.mL-1 10.1128/aac.00464-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00110-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00453-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00707-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00810-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00822-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00834-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00859-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.01104-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.01573-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.01617-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 24.0 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 24.0 ug.mL-1 10.1128/aac.00707-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 24.0 ug.mL-1 10.1128/aac.00822-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 24.0 ug.mL-1 10.1128/aac.01617-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00110-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00707-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00822-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00834-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01104-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01172-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01549-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01573-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.01646-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 40.0 ug.mL-1 10.1128/aac.01071-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 48.0 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 48.0 ug.mL-1 10.1128/aac.00465-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 48.0 ug.mL-1 10.1128/aac.00707-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 48.0 ug.mL-1 10.1128/aac.00822-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1016/s0960-894x(00)00444-3
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1021/acs.jmedchem.9b01279
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.00080-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.00160-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.00341-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.00465-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.00679-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.00707-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.01011-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.01104-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.01172-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.01267-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.01483-06
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.01549-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1128/aac.01646-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 96.0 ug.mL-1 10.1128/aac.01267-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 100.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 100.0 ug.mL-1 10.1128/aac.00464-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.00080-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.00110-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.00175-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.00341-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.00707-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.00734-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.01104-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.01172-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.01561-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1128/aac.01646-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 192.0 ug.mL-1 10.1128/aac.00465-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 200.0 ug.mL-1 10.1128/aac.00464-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.00110-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.00282-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.00299-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.00341-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.00465-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.00734-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.00900-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.01104-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.01172-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.01360-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.01405-06
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.01451-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.01561-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.01617-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1128/aac.01646-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 384.0 ug.mL-1 10.1128/aac.00385-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 512.0 ug.mL-1 10.1128/aac.00110-10
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1024.0 ug.mL-1 10.1128/aac.00341-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 4.0 ug.mL-1 10.1128/aac.00400-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 8.0 ug.mL-1 10.1016/j.bmcl.2008.04.023
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 8.0 ug.mL-1 10.1128/aac.01047-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 16.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 16.0 ug.mL-1 10.1128/aac.01047-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 32.0 ug.mL-1 10.1021/acs.jmedchem.7b00377
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 128.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC50 128.0 ug.mL-1 10.1128/aac.01197-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC80 32.0 ug.mL-1 10.1016/j.bmcl.2008.04.023
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 64.0 ug.mL-1 10.1016/j.bmcl.2008.04.023
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 64.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 64.0 ug.mL-1 10.1128/aac.00400-09
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 64.0 ug.mL-1 10.1128/aac.01047-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 128.0 ug.mL-1 10.1021/acs.jmedchem.7b00377
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 128.0 ug.mL-1 10.1128/aac.00381-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC90 128.0 ug.mL-1 10.1128/aac.01197-09
Pseudomonas aeruginosa Pseudomonas aeruginosa Ratio 10.0 None 10.1128/aac.01617-08
Pseudomonas aeruginosa Pseudomonas aeruginosa TIME 0.4283 hr 10.1128/aac.00428-08
Pseudomonas aeruginosa Pseudomonas aeruginosa TIME 0.4333 hr 10.1128/aac.00428-08
Pseudomonas aeruginosa Pseudomonas aeruginosa TIME 0.455 hr 10.1128/aac.00428-08
Pseudomonas aeruginosa Pseudomonas aeruginosa TIME 0.4617 hr 10.1128/aac.00428-08
Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) Beta-lactamase Kcat 2.0 /s 10.1128/aac.01410-08
Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) Beta-lactamase Kcat/Km 50.0 /uM/s 10.1128/aac.01410-08
Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG12228) Beta-lactamase Km 100000.0 nM 10.1128/aac.01410-08
Pseudomonas fluorescens Beta-lactamase Kcat/Km 210.0 /mM/s 10.1128/aac.00961-09
Pseudomonas fluorescens Pseudomonas fluorescens Activity 23.0 % 10.1128/aac.01808-09
Pseudomonas fluorescens Pseudomonas fluorescens MIC 4.0 ug.mL-1 10.1128/aac.00961-09
Pseudomonas luteola Beta-lactamase Kcat 8.0 /s 10.1128/aac.00427-09
Pseudomonas luteola Beta-lactamase Kcat/Km 1.14 /s/microM 10.1128/aac.00427-09
Pseudomonas luteola Beta-lactamase Km 7000.0 nM 10.1128/aac.00427-09
Pseudomonas putida Pseudomonas putida MIC 64.0 ug.mL-1 10.1128/aac.00838-06
Pseudomonas putida Pseudomonas putida MIC 128.0 ug.mL-1 10.1128/aac.00707-08
Pseudomonas putida Pseudomonas putida MIC 128.0 ug.mL-1 10.1128/aac.00931-08
Rattus norvegicus Aldose reductase IC50 nan None None
Rattus norvegicus Aldose reductase Ki nan None None
Rattus norvegicus Alpha-1a adrenergic receptor IC50 nan None None
Rattus norvegicus Alpha-1a adrenergic receptor Ki nan None None
Rattus norvegicus Alpha-1b adrenergic receptor IC50 nan None None
Rattus norvegicus Alpha-1b adrenergic receptor Ki nan None None
Rattus norvegicus Androgen Receptor IC50 nan None None
Rattus norvegicus Androgen Receptor Ki nan None None
Rattus norvegicus Glycine receptor IC50 nan None None
Rattus norvegicus Glycine receptor Ki nan None None
Rattus norvegicus Insulin receptor IC50 nan None None
Rattus norvegicus Insulin receptor Ki nan None None
Rattus norvegicus Nitric-oxide synthase, brain IC50 nan None None
Rattus norvegicus Nitric-oxide synthase, brain Ki nan None None
Rattus norvegicus Serotonin 1a (5-HT1a) receptor IC50 nan None None
Rattus norvegicus Serotonin 1a (5-HT1a) receptor Ki nan None None
Rattus norvegicus Serotonin 1b (5-HT1b) receptor IC50 nan None None
Rattus norvegicus Serotonin 1b (5-HT1b) receptor Ki nan None None
Rattus norvegicus Solute carrier family 22 member 6 Activity nan None None
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium ED50 45.0 mg.kg-1 10.1128/aac.01549-08
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium ED50 152.0 mg.kg-1 10.1128/aac.01549-08
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium ED50 1121.0 mg.kg-1 10.1128/aac.01549-08
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 4.0 ug.mL-1 10.1128/aac.01472-06
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 8.0 ug.mL-1 10.1128/aac.01549-08
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 64.0 ug.mL-1 10.1128/aac.01549-08
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 256.0 ug.mL-1 10.1128/aac.00079-09
Salmonella enterica subsp. enterica serovar Westhampton Extended-spectrum beta-lactamase CTX-M-53 Kcat 90.0 /s 10.1128/aac.01581-08
Salmonella enterica subsp. enterica serovar Westhampton Extended-spectrum beta-lactamase CTX-M-53 Kcat/Km 7.5 /s/microM 10.1128/aac.01581-08
Salmonella enterica subsp. enterica serovar Westhampton Extended-spectrum beta-lactamase CTX-M-53 Km 12000.0 nM 10.1128/aac.01581-08
Schaalia meyeri Schaalia meyeri Activity 0.0 % 10.1128/aac.00481-10
Schaalia meyeri Schaalia meyeri Activity 92.0 % 10.1128/aac.00481-10
Schaalia meyeri Schaalia meyeri MIC 0.03 ug.mL-1 10.1128/aac.00481-10
Schaalia meyeri Schaalia meyeri MIC 0.06 ug.mL-1 10.1128/aac.00481-10
Schaalia meyeri Schaalia meyeri MIC50 0.5 ug.mL-1 10.1128/aac.00481-10
Schaalia meyeri Schaalia meyeri MIC50 1.0 ug.mL-1 10.1128/aac.00481-10
Schaalia meyeri Schaalia meyeri MIC90 8.0 ug.mL-1 10.1128/aac.00481-10
Serratia fonticola Carbapenem-hydrolizing beta-lactamase SFC-1 Kcat 44.7 /s 10.1128/aac.00491-07
Serratia fonticola Carbapenem-hydrolizing beta-lactamase SFC-1 Kcat/Km 1190.0 /mM/s 10.1128/aac.00491-07
Serratia fonticola Carbapenem-hydrolizing beta-lactamase SFC-1 Km 38000.0 nM 10.1128/aac.00491-07
Serratia marcescens Serratia marcescens Activity 0.9 % 10.1128/aac.00400-09
Serratia marcescens Serratia marcescens Activity 1.9 % 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens Activity 3.4 % 10.1128/aac.00149-08
Serratia marcescens Serratia marcescens Activity 4.4 % 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens Activity 4.7 % 10.1128/aac.00400-09
Serratia marcescens Serratia marcescens Activity 20.0 % 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens Activity 30.0 % 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens Activity 50.0 % 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens Activity 93.2 % 10.1128/aac.00149-08
Serratia marcescens Serratia marcescens Activity 93.6 % 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens Activity 94.4 % 10.1128/aac.00400-09
Serratia marcescens Serratia marcescens Activity 100.0 % 10.1128/aac.01808-09
Serratia marcescens Serratia marcescens ED50 128.0 mg.kg-1 10.1016/s0960-894x(99)00107-9
Serratia marcescens Serratia marcescens MIC 0.25 ug.mL-1 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens MIC 0.5 ug.mL-1 10.1128/aac.00149-08
Serratia marcescens Serratia marcescens MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC 1.0 ug.mL-1 10.1128/aac.00400-09
Serratia marcescens Serratia marcescens MIC 1.0 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC 2.0 ug.mL-1 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens MIC 8.0 ug.mL-1 10.1016/s0960-894x(00)00444-3
Serratia marcescens Serratia marcescens MIC 8.0 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC 32.0 ug.mL-1 10.1016/s0960-894x(99)00106-7
Serratia marcescens Serratia marcescens MIC 32.0 ug.mL-1 10.1016/s0960-894x(99)00107-9
Serratia marcescens Serratia marcescens MIC 32.0 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC 64.0 ug.mL-1 10.1016/s0960-894x(00)00444-3
Serratia marcescens Serratia marcescens MIC 64.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Serratia marcescens Serratia marcescens MIC 128.0 ug.mL-1 10.1128/aac.01539-07
Serratia marcescens Serratia marcescens MIC 200.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Serratia marcescens Serratia marcescens MIC 256.0 ug.mL-1 10.1128/aac.00768-10
Serratia marcescens Serratia marcescens MIC 256.0 ug.mL-1 10.1128/aac.01028-07
Serratia marcescens Serratia marcescens MIC 256.0 ug.mL-1 10.1128/aac.01539-07
Serratia marcescens Serratia marcescens MIC50 1.0 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC50 2.0 ug.mL-1 10.1128/aac.00149-08
Serratia marcescens Serratia marcescens MIC50 2.0 ug.mL-1 10.1128/aac.00400-09
Serratia marcescens Serratia marcescens MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC50 4.0 ug.mL-1 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC50 8.0 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC50 64.0 ug.mL-1 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC90 4.0 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC90 8.0 ug.mL-1 10.1128/aac.00400-09
Serratia marcescens Serratia marcescens MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC90 16.0 ug.mL-1 10.1128/aac.00149-08
Serratia marcescens Serratia marcescens MIC90 16.0 ug.mL-1 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC90 64.0 ug.mL-1 10.1128/aac.01047-08
Serratia marcescens Serratia marcescens MIC90 128.0 ug.mL-1 10.1128/aac.00381-08
Serratia marcescens Serratia marcescens MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Severe acute respiratory syndrome coronavirus 2 Replicase polyprotein 1ab Inhibition -6.84 % 10.6019/CHEMBL4495564
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Hit score 0.2065 None 10.1101/2020.04.21.054387
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Inhibition -0.05 % 10.6019/CHEMBL4495565
Shigella sonnei Shigella sonnei MIC 64.0 ug.mL-1 10.1128/aac.00227-08
Shouchella clausii Shouchella clausii MIC 8000.0 ug.mL-1 10.1128/aac.00537-07
Shouchella clausii Shouchella clausii MIC 16000.0 ug.mL-1 10.1128/aac.00537-07
Staphylococcus aureus Staphylococcus aureus Activity 0.0 % 10.1128/aac.01538-07
Staphylococcus aureus Staphylococcus aureus Activity 100.0 % 10.1128/aac.01538-07
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1021/jm0703183
Staphylococcus aureus Staphylococcus aureus ED50 12.0 mg.kg-1 10.1128/aac.01549-08
Staphylococcus aureus Staphylococcus aureus ED50 16.0 mg.kg-1 10.1128/aac.01549-08
Staphylococcus aureus Staphylococcus aureus ED50 418.0 mg.kg-1 10.1128/aac.01549-08
Staphylococcus aureus Staphylococcus aureus IC50 nan None 10.1021/np900499q
Staphylococcus aureus Staphylococcus aureus MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1016/s0960-894x(03)00512-2
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1016/s0960-894x(03)00542-0
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1128/aac.01472-06
Staphylococcus aureus Staphylococcus aureus MIC 1.0 ug.mL-1 10.1016/j.bmc.2007.07.048
Staphylococcus aureus Staphylococcus aureus MIC 1.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Staphylococcus aureus Staphylococcus aureus MIC 1.0 ug.mL-1 10.1128/aac.01549-08
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1016/j.bmc.2007.08.035
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1016/j.bmcl.2015.10.063
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1016/0960-894X(95)00249-S
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Staphylococcus aureus Staphylococcus aureus MIC 8.0 ug.mL-1 10.1016/j.bmcl.2003.12.037
Staphylococcus aureus Staphylococcus aureus MIC 8.0 ug.mL-1 10.1016/j.bmcl.2015.10.063
Staphylococcus aureus Staphylococcus aureus MIC 8.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Staphylococcus aureus Staphylococcus aureus MIC 16.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1128/aac.01472-06
Staphylococcus aureus Staphylococcus aureus MIC 50.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1128/aac.01549-08
Staphylococcus aureus Staphylococcus aureus MIC 128.0 ug.mL-1 10.1016/j.bmcl.2015.10.063
Staphylococcus aureus Staphylococcus aureus MIC 128.0 ug.mL-1 10.1128/aac.01472-06
Staphylococcus aureus Staphylococcus aureus MIC 200.0 ug.mL-1 10.1016/S0960-894X(96)00575-6
Staphylococcus aureus Staphylococcus aureus MIC 528.0 ug.mL-1 10.1016/j.ejmech.2021.113691
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1021/np900499q
Staphylococcus aureus Staphylococcus aureus MIC50 0.25 ug.mL-1 10.1128/aac.01047-08
Staphylococcus aureus Staphylococcus aureus MIC50 1.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus aureus Staphylococcus aureus MIC50 32.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus aureus Staphylococcus aureus MIC50 64.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus aureus Staphylococcus aureus MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus aureus Staphylococcus aureus MIC90 0.5 ug.mL-1 10.1128/aac.01047-08
Staphylococcus aureus Staphylococcus aureus MIC90 2.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus aureus Staphylococcus aureus MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis Activity 0.0 % 10.1128/aac.01538-07
Staphylococcus epidermidis Staphylococcus epidermidis Activity 1.2 % 10.1128/aac.01538-07
Staphylococcus epidermidis Staphylococcus epidermidis Activity 4.2 % 10.1128/aac.01538-07
Staphylococcus epidermidis Staphylococcus epidermidis Activity 100.0 % 10.1128/aac.01538-07
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.004 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC50 0.004 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC50 0.25 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC50 0.5 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC50 1.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC50 8.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC90 0.004 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC90 0.5 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC90 8.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC90 64.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus haemolyticus Staphylococcus haemolyticus MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Staphylococcus haemolyticus Staphylococcus haemolyticus MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Staphylococcus haemolyticus Staphylococcus haemolyticus MIC 2.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus haemolyticus Staphylococcus haemolyticus MIC 4.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Staphylococcus haemolyticus Staphylococcus haemolyticus MIC 16.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Staphylococcus haemolyticus Staphylococcus haemolyticus MIC 32.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Staphylococcus haemolyticus Staphylococcus haemolyticus MIC 64.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Staphylococcus haemolyticus Staphylococcus haemolyticus MIC50 32.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus haemolyticus Staphylococcus haemolyticus MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Staphylococcus haemolyticus Staphylococcus haemolyticus MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Stenotrophomonas maltophilia Beta-lactamase L1 Kcat/Km 7.0 10'6/M/s 10.1128/aac.01062-07
Stenotrophomonas maltophilia Stenotrophomonas maltophilia Activity 23.0 % 10.1128/aac.01808-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia Activity nan None 10.1128/aac.00682-07
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 16.0 ug.mL-1 10.1128/aac.00400-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 16.0 ug.mL-1 10.1128/aac.01283-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 32.0 ug.mL-1 10.1128/aac.01047-08
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 32.0 ug.mL-1 10.1128/aac.01283-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 32.0 ug.mL-1 10.1128/aac.01485-07
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 64.0 ug.mL-1 10.1016/s0960-894x(99)00325-x
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 128.0 ug.mL-1 10.1128/aac.01047-08
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 256.0 ug.mL-1 10.1128/aac.00682-07
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 512.0 ug.mL-1 10.1128/aac.00682-07
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 512.0 ug.mL-1 10.1128/aac.01283-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 1024.0 ug.mL-1 10.1128/aac.00682-07
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 1024.0 ug.mL-1 10.1128/aac.01283-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 1024.0 ug.mL-1 10.1128/aac.01513-08
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 2048.0 ug.mL-1 10.1128/aac.01485-07
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC50 128.0 ug.mL-1 10.1128/aac.01047-08
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC50 512.0 ug.mL-1 10.1128/aac.00400-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC90 512.0 ug.mL-1 10.1128/aac.00400-09
Stenotrophomonas maltophilia Stenotrophomonas maltophilia Ratio 1.7 None 10.1128/aac.00682-07
Streptococcus Streptococcus MIC 0.12 ug.mL-1 10.1016/s0960-894x(03)00512-2
Streptococcus agalactiae Streptococcus agalactiae MIC 0.0004 ug.mL-1 10.1128/aac.01047-08
Streptococcus agalactiae Streptococcus agalactiae MIC 0.06 ug.mL-1 10.1128/aac.01047-08
Streptococcus agalactiae Streptococcus agalactiae MIC 0.12 ug.mL-1 10.1016/s0960-894x(03)00512-2
Streptococcus agalactiae Streptococcus agalactiae MIC50 0.004 ug.mL-1 10.1128/aac.01047-08
Streptococcus agalactiae Streptococcus agalactiae MIC50 0.12 ug.mL-1 10.1128/aac.01047-08
Streptococcus agalactiae Streptococcus agalactiae MIC90 0.03 ug.mL-1 10.1128/aac.01047-08
Streptococcus agalactiae Streptococcus agalactiae MIC90 0.25 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.004 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.006 ug.mL-1 10.1016/s0960-894x(03)00512-2
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.04 ug.mL-1 10.1128/aac.01107-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.06 ug.mL-1 10.1016/s0960-894x(03)00512-2
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.06 ug.mL-1 10.1128/aac.01107-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.08 ug.mL-1 10.1128/aac.01107-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.09 ug.mL-1 10.1128/aac.01107-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.1 ug.mL-1 10.1128/aac.01107-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.11 ug.mL-1 10.1128/aac.01107-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.12 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.12 ug.mL-1 10.1128/aac.01107-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.25 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.5 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC 2.0 ug.mL-1 10.1016/s0960-894x(03)00512-2
Streptococcus pneumoniae Streptococcus pneumoniae MIC nan None 10.1016/j.bmc.2007.08.035
Streptococcus pneumoniae Streptococcus pneumoniae MIC nan None 10.1128/aac.01107-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.004 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.008 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.015 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.25 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.5 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 2.0 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.004 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.015 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.03 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 1.0 ug.mL-1 10.1128/aac.01047-08
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 4.0 ug.mL-1 10.1128/aac.01047-08
Streptococcus pyogenes Streptococcus pyogenes MIC 0.004 ug.mL-1 10.1128/aac.01047-08
Streptococcus pyogenes Streptococcus pyogenes MIC 0.006 ug.mL-1 10.1016/s0960-894x(03)00512-2
Streptococcus pyogenes Streptococcus pyogenes MIC 0.015 ug.mL-1 10.1128/aac.01047-08
Streptococcus pyogenes Streptococcus pyogenes MIC50 0.004 ug.mL-1 10.1128/aac.01047-08
Streptococcus pyogenes Streptococcus pyogenes MIC50 0.03 ug.mL-1 10.1128/aac.01047-08
Streptococcus pyogenes Streptococcus pyogenes MIC90 0.004 ug.mL-1 10.1128/aac.01047-08
Streptococcus pyogenes Streptococcus pyogenes MIC90 0.06 ug.mL-1 10.1128/aac.01047-08
Streptococcus sp. Streptococcus sp. MIC 0.06 ug.mL-1 10.1016/s0960-894x(03)00542-0
Stutzerimonas stutzeri Stutzerimonas stutzeri MIC 512.0 ug.mL-1 10.1128/aac.01456-09
Thomasclavelia ramosa Thomasclavelia ramosa MIC 0.125 ug.mL-1 10.1128/aac.01557-08
Veillonella parvula Veillonella parvula MIC 0.03 ug.mL-1 10.1128/aac.00355-08
Veillonella parvula Veillonella parvula MIC 1.0 ug.mL-1 10.1128/aac.00355-08
Yersinia enterocolitica Yersinia enterocolitica MIC 0.094 ug.mL-1 10.1128/aac.01754-09
Yersinia enterocolitica Yersinia enterocolitica MIC 0.19 ug.mL-1 10.1128/aac.01754-09
Yersinia enterocolitica Yersinia enterocolitica MIC 0.75 ug.mL-1 10.1128/aac.01754-09
None ADMET CL 4.0 mL.min-1.kg-1 10.1124/dmd.108.020479
None ADMET MRT 1.1 hr 10.1124/dmd.108.020479
None ADMET T1/2 0.96 hr 10.1124/dmd.108.020479
None ADMET Vdss 0.27 L.kg-1 10.1124/dmd.108.020479
None Hepatotoxicity Alkaline Phosphatase Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity Alkaline Phosphatase Increase - Index Value 0.3 None 10.2174/1570163043334794
None Hepatotoxicity Alkaline Phosphatase Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None Hepatotoxicity Composite Activity - Active 0.0 None 10.2174/1570163043334794
None Hepatotoxicity Composite Activity - Marginal 0.0 None 10.2174/1570163043334794
None Hepatotoxicity Composite Activity - Score nan None 10.2174/1570163043334794
None Hepatotoxicity GGT Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity GGT Increase - Index Value 0.0 None 10.2174/1570163043334794
None Hepatotoxicity GGT Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None Hepatotoxicity Hepatotoxicity nan None 10.1021/tx900326k
None Hepatotoxicity HepSE_bilirubinemia 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_cholecystitis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_cholelithiasis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_cirrhosis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_Combined Scores 3.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_elevated liver function tests 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatic failure 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatic necrosis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatitis 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatomegaly 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_jaundice 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_liver disease 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_liver fatty 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_liver function tests abnormal 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity LDH Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity LDH Increase - Index Value 0.0 None 10.2174/1570163043334794
None Hepatotoxicity LDH Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None Hepatotoxicity SGOT Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity SGOT Increase - Index Value 0.3 None 10.2174/1570163043334794
None Hepatotoxicity SGOT Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None Hepatotoxicity SGPT Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity SGPT Increase - Index Value 0.0 None 10.2174/1570163043334794
None Hepatotoxicity SGPT Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None NON-PROTEIN TARGET Activity 0.0 % 10.1128/aac.00081-08
None NON-PROTEIN TARGET Activity 0.0 % 10.1128/aac.00481-10
None NON-PROTEIN TARGET Activity 0.0 % 10.1128/aac.00696-08
None NON-PROTEIN TARGET Activity 5.6 % 10.1128/aac.00696-08
None NON-PROTEIN TARGET Activity 9.8 % 10.1128/aac.01173-09
None NON-PROTEIN TARGET Activity 92.0 % 10.1128/aac.00481-10
None NON-PROTEIN TARGET Fu 0.5 None 10.1124/dmd.108.020479
None NON-PROTEIN TARGET Hepatotoxicity (acute) 0.2 % 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (animal toxicity known) nan None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (benign tumour) 0.0 None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (granulomatous hepatitis) 0.0 None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (mechanism) nan None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (moderate) 14.0 None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (moderate) 25.6 % 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (time to onset) nan None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET MIC 0.0 ug.mL-1 10.1128/aac.00481-10
None NON-PROTEIN TARGET MIC 0.016 ug.mL-1 10.1128/aac.00684-07
None NON-PROTEIN TARGET MIC 0.03 ug.mL-1 10.1128/aac.00481-10
None NON-PROTEIN TARGET MIC 0.06 ug.mL-1 10.1128/aac.00081-08
None NON-PROTEIN TARGET MIC 0.06 ug.mL-1 10.1128/aac.00481-10
None NON-PROTEIN TARGET MIC 0.12 ug.mL-1 10.1128/aac.01047-08
None NON-PROTEIN TARGET MIC 0.125 ug.mL-1 10.1128/aac.01557-08
None NON-PROTEIN TARGET MIC 0.25 ug.mL-1 10.1128/aac.00791-09
None NON-PROTEIN TARGET MIC 0.25 ug.mL-1 10.1128/aac.01252-09
None NON-PROTEIN TARGET MIC 0.5 ug.mL-1 10.1128/aac.00696-08
None NON-PROTEIN TARGET MIC 0.5 ug.mL-1 10.1128/aac.00791-09
None NON-PROTEIN TARGET MIC 0.5 ug.mL-1 10.1128/aac.01047-08
None NON-PROTEIN TARGET MIC 0.5 ug.mL-1 10.1128/aac.01463-07
None NON-PROTEIN TARGET MIC 0.5 ug.mL-1 10.1128/aac.01557-08
None NON-PROTEIN TARGET MIC 1.0 ug.mL-1 10.1128/aac.00427-09
None NON-PROTEIN TARGET MIC 1.0 ug.mL-1 10.1128/aac.01463-07
None NON-PROTEIN TARGET MIC 1.0 ug.mL-1 10.1128/aac.01557-08
None NON-PROTEIN TARGET MIC 2.0 ug.mL-1 10.1128/aac.00427-09
None NON-PROTEIN TARGET MIC 2.0 ug.mL-1 10.1128/aac.00696-08
None NON-PROTEIN TARGET MIC 2.0 ug.mL-1 10.1128/aac.01152-06
None NON-PROTEIN TARGET MIC 2.0 ug.mL-1 10.1128/aac.01463-07
None NON-PROTEIN TARGET MIC 2.0 ug.mL-1 10.1128/aac.01557-08
None NON-PROTEIN TARGET MIC 4.0 ug.mL-1 10.1128/aac.00128-10
None NON-PROTEIN TARGET MIC 4.0 ug.mL-1 10.1128/aac.00696-08
None NON-PROTEIN TARGET MIC 4.0 ug.mL-1 10.1128/aac.01252-09
None NON-PROTEIN TARGET MIC 4.0 ug.mL-1 10.1128/aac.01463-07
None NON-PROTEIN TARGET MIC 4.0 ug.mL-1 10.1128/aac.01585-09
None NON-PROTEIN TARGET MIC 8.0 ug.mL-1 10.1128/aac.00696-08
None NON-PROTEIN TARGET MIC 16.0 ug.mL-1 10.1128/aac.00128-10
None NON-PROTEIN TARGET MIC 16.0 ug.mL-1 10.1128/aac.00630-09
None NON-PROTEIN TARGET MIC 16.0 ug.mL-1 10.1128/aac.00696-08
None NON-PROTEIN TARGET MIC 16.0 ug.mL-1 10.1128/aac.01284-08
None NON-PROTEIN TARGET MIC 16.0 ug.mL-1 10.1128/aac.01581-08
None NON-PROTEIN TARGET MIC 32.0 ug.mL-1 10.1128/aac.00128-10
None NON-PROTEIN TARGET MIC 32.0 ug.mL-1 10.1128/aac.00630-09
None NON-PROTEIN TARGET MIC 48.0 ug.mL-1 10.1128/aac.00684-07
None NON-PROTEIN TARGET MIC 64.0 ug.mL-1 10.1128/aac.00734-08
None NON-PROTEIN TARGET MIC 64.0 ug.mL-1 10.1128/aac.01284-08
None NON-PROTEIN TARGET MIC 64.0 ug.mL-1 10.1128/aac.01600-06
None NON-PROTEIN TARGET MIC 128.0 ug.mL-1 10.1128/aac.00128-10
None NON-PROTEIN TARGET MIC 256.0 ug.mL-1 10.1128/aac.00630-09
None NON-PROTEIN TARGET MIC 256.0 ug.mL-1 10.1128/aac.01581-08
None NON-PROTEIN TARGET MIC 512.0 ug.mL-1 10.1128/aac.00128-10
None NON-PROTEIN TARGET MIC 1024.0 ug.mL-1 10.1128/aac.00128-10
None NON-PROTEIN TARGET MIC50 0.12 ug.mL-1 10.1128/aac.01047-08
None NON-PROTEIN TARGET MIC50 0.125 ug.mL-1 10.1128/aac.01557-08
None NON-PROTEIN TARGET MIC50 0.5 ug.mL-1 10.1128/aac.00481-10
None NON-PROTEIN TARGET MIC50 1.0 ug.mL-1 10.1128/aac.00481-10
None NON-PROTEIN TARGET MIC50 1.0 ug.mL-1 10.1128/aac.01557-08
None NON-PROTEIN TARGET MIC50 2.0 ug.mL-1 10.1128/aac.01557-08
None NON-PROTEIN TARGET MIC50 4.0 ug.mL-1 10.1128/aac.01047-08
None NON-PROTEIN TARGET MIC50 8.0 ug.mL-1 10.1128/aac.00081-08
None NON-PROTEIN TARGET MIC50 256.0 ug.mL-1 10.1128/aac.00630-09
None NON-PROTEIN TARGET MIC90 0.25 ug.mL-1 10.1128/aac.01557-08
None NON-PROTEIN TARGET MIC90 2.0 ug.mL-1 10.1128/aac.01557-08
None NON-PROTEIN TARGET MIC90 8.0 ug.mL-1 10.1128/aac.00481-10
None NON-PROTEIN TARGET MIC90 16.0 ug.mL-1 10.1128/aac.01047-08
None NON-PROTEIN TARGET MIC90 32.0 ug.mL-1 10.1128/aac.00081-08
None NON-PROTEIN TARGET MIC90 32.0 ug.mL-1 10.1128/aac.01047-08
None NON-PROTEIN TARGET MIC90 128.0 ug.mL-1 10.1128/aac.01047-08
None NON-PROTEIN TARGET MIC90 256.0 ug.mL-1 10.1128/aac.00630-09
None No relevant target LogP 0.45 None 10.1128/aac.01714-09
None Unchecked Activity 4.6 % 10.1128/aac.00083-07
None Unchecked Activity 31.0 % 10.1128/aac.01164-08
None Unchecked Activity 35.0 % 10.1128/aac.01164-08
None Unchecked Activity nan None 10.1016/j.bmcl.2003.12.037
None Unchecked FC 2.7 None 10.1128/aac.00197-10
None Unchecked FC 10.0 None 10.1128/aac.00537-07
None Unchecked Hepatotoxicity (acute) 4.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (association with vascular disease) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (choleostasis) 3.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (chronic liver disease) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (cirrhosis) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (comment) nan None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (cytolytic) 1.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (malignant tumour) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (severe hepatitis) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (steatosis) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (successful reintroduction) nan None 10.1016/s0399-8320(04)95062-2
None Unchecked IC50 166.0 nM 10.1021/acs.jmedchem.5b00586
None Unchecked IC50 nan None None
None Unchecked Inhibition nan % 10.1128/aac.01821-09
None Unchecked K0.5 1.06 uM 10.1128/aac.01714-09
None Unchecked Kcat 0.4 /s 10.1128/aac.01600-06
None Unchecked Kcat 0.5 /s 10.1128/aac.01463-07
None Unchecked Kcat 0.54 /s 10.1128/aac.01252-09
None Unchecked Kcat 1.0 /s 10.1128/aac.00856-09
None Unchecked Kcat 2.7 /s 10.1128/aac.01028-07
None Unchecked Kcat 5.0 /s 10.1128/aac.01028-07
None Unchecked Kcat 5.0 /s 10.1128/aac.01164-08
None Unchecked Kcat 5.0 /s 10.1128/aac.01410-08
None Unchecked Kcat 5.5 /s 10.1128/aac.01410-08
None Unchecked Kcat 9.0 /s 10.1128/aac.01062-07
None Unchecked Kcat 10.0 /s 10.1128/aac.00858-10
None Unchecked Kcat 14.61 /s 10.1128/aac.00083-07
None Unchecked Kcat 17.0 /s 10.1128/aac.00693-09
None Unchecked Kcat 40.0 /s 10.1128/aac.00163-08
None Unchecked Kcat 40.0 /s 10.1128/aac.00961-09
None Unchecked Kcat 42.0 /s 10.1128/aac.00197-10
None Unchecked Kcat 50.0 /s 10.1128/aac.00387-08
None Unchecked Kcat 64.0 /s 10.1128/aac.01145-07
None Unchecked Kcat 89.0 /s 10.1128/aac.00614-07
None Unchecked Kcat 160.0 /s 10.1128/aac.00017-09
None Unchecked Kcat 172.0 /s 10.1128/aac.01058-06
None Unchecked Kcat 213.0 /s 10.1128/aac.01058-06
None Unchecked Kcat 306.0 /s 10.1128/aac.01058-06
None Unchecked Kcat 336.0 /s 10.1128/aac.01058-06
None Unchecked Kcat 406.0 /s 10.1128/aac.01442-09
None Unchecked Kcat 945.0 /s 10.1128/aac.00614-07
None Unchecked Kcat 1179.0 /s 10.1021/jm301490d
None Unchecked Kcat 1216.0 /s 10.1128/aac.01058-06
None Unchecked Kcat 1250.0 /s 10.1128/aac.01058-06
None Unchecked Kcat 1900.0 /s 10.1128/aac.00166-08
None Unchecked Kcat 2736.0 /s 10.1021/jm301490d
None Unchecked Kcat nan None 10.1128/aac.00774-09
None Unchecked Kcat nan None 10.1128/aac.01028-07
None Unchecked Kcat/Km 0.025 /s/microM 10.1128/aac.00856-09
None Unchecked Kcat/Km 0.039 /uM/s 10.1128/aac.00083-07
None Unchecked Kcat/Km 0.5 /uM/s 10.1128/aac.01164-08
None Unchecked Kcat/Km 0.54 /uM/s 10.1128/aac.00166-08
None Unchecked Kcat/Km 1.1 microM/s 10.1128/aac.00693-09
None Unchecked Kcat/Km 1.2 10'4/M/s 10.1128/aac.00409-10
None Unchecked Kcat/Km 1.2 /uM/s 10.1128/aac.00050-10
None Unchecked Kcat/Km 1.47 /uM/s 10.1128/aac.01028-07
None Unchecked Kcat/Km 1.7 10'6/M/s 10.1128/aac.00409-10
None Unchecked Kcat/Km 1.92 /uM/s 10.1128/aac.01028-07
None Unchecked Kcat/Km 2.3 /uM/s 10.1128/aac.01058-06
None Unchecked Kcat/Km 2.6 10'4/M/s 10.1128/aac.01062-07
None Unchecked Kcat/Km 2.7 10'6/M/s 10.1128/aac.01252-09
None Unchecked Kcat/Km 2.9 None 10.1128/aac.00614-07
None Unchecked Kcat/Km 3.5 /uM/s 10.1128/aac.00197-10
None Unchecked Kcat/Km 3.9 /uM/s 10.1128/aac.01058-06
None Unchecked Kcat/Km 4.3 /s/microM 10.1128/aac.00017-09
None Unchecked Kcat/Km 5.1 10'4/M/s 10.1128/aac.00858-10
None Unchecked Kcat/Km 6.0 /uM/s 10.1128/aac.01442-09
None Unchecked Kcat/Km 6.0 None 10.1128/aac.00614-07
None Unchecked Kcat/Km 6.12 /uM/s 10.1128/aac.01058-06
None Unchecked Kcat/Km 6.7 10'4/M/s 10.1128/aac.00409-10
None Unchecked Kcat/Km 6.7 10'4/M/s 10.1128/aac.01062-07
None Unchecked Kcat/Km 7.0 10'6/M/s 10.1128/aac.00409-10
None Unchecked Kcat/Km 7.0 /uM/s 10.1128/aac.00197-10
None Unchecked Kcat/Km 7.1 /uM/s 10.1128/aac.01058-06
None Unchecked Kcat/Km 7.2 10'5/M/s 10.1128/aac.00858-10
None Unchecked Kcat/Km 7.9 /uM/s 10.1128/aac.01058-06
None Unchecked Kcat/Km 8.6 /uM/s 10.1128/aac.01058-06
None Unchecked Kcat/Km 9.0 /uM/s 10.1021/jm301490d
None Unchecked Kcat/Km 14.0 None 10.1128/aac.01145-07
None Unchecked Kcat/Km 15.8 /uM/s 10.1021/jm301490d
None Unchecked Kcat/Km 125.0 /uM/s 10.1128/aac.01410-08
None Unchecked Kcat/Km 135.0 /uM/s 10.1128/aac.01410-08
None Unchecked Kcat/Km 200.0 /uM/s 10.1128/aac.01585-09
None Unchecked Kcat/Km 800.0 /mM/s 10.1128/aac.00961-09
None Unchecked Kcat/Km 800.0 /uM/s 10.1128/aac.00163-08
None Unchecked Kcat/Km 914.0 /mM/s 10.1128/aac.01145-07
None Unchecked Kcat/Km 1000.0 /uM/s 10.1128/aac.00387-08
None Unchecked Kcat/Km 1500.0 /mM/s 10.1128/aac.01082-06
None Unchecked Kcat/Km nan None 10.1128/aac.00774-09
None Unchecked Kcat/Km nan None 10.1128/aac.01028-07
None Unchecked Ki 200.0 nM 10.1128/aac.01252-09
None Unchecked Ki 1000.0 nM 10.1128/aac.01463-07
None Unchecked Ki 16000.0 nM 10.1128/aac.00693-09
None Unchecked Ki nan None None
None Unchecked Km 15.0 /s/microM 10.1128/aac.00614-07
None Unchecked Km 320.0 /s/microM 10.1128/aac.00614-07
None Unchecked Km 1400.0 nM 10.1128/aac.00389-07
None Unchecked Km 1400.0 nM 10.1128/aac.01028-07
None Unchecked Km 3400.0 nM 10.1128/aac.01028-07
None Unchecked Km 6000.0 nM 10.1128/aac.00197-10
None Unchecked Km 10000.0 nM 10.1128/aac.01164-08
None Unchecked Km 10000.0 nM 10.1128/aac.01600-06
None Unchecked Km 12000.0 nM 10.1128/aac.00197-10
None Unchecked Km 20000.0 nM 10.1128/aac.00409-10
None Unchecked Km 27000.0 nM 10.1128/aac.01058-06
None Unchecked Km 39000.0 nM 10.1128/aac.01058-06
None Unchecked Km 40000.0 nM 10.1128/aac.00856-09
None Unchecked Km 40000.0 nM 10.1128/aac.01410-08
None Unchecked Km 44000.0 nM 10.1128/aac.01058-06
None Unchecked Km 50000.0 nM 10.1128/aac.00387-08
None Unchecked Km 50000.0 nM 10.1128/aac.01058-06
None Unchecked Km 50000.0 nM 10.1128/aac.01082-06
None Unchecked Km 51000.0 nM 10.1128/aac.00163-08
None Unchecked Km 55000.0 nM 10.1128/aac.01058-06
None Unchecked Km 68000.0 nM 10.1128/aac.01442-09
None Unchecked Km 70000.0 nM 10.1128/aac.01145-07
None Unchecked Km 74600.0 nM 10.1021/jm301490d
None Unchecked Km 170000.0 nM 10.1128/aac.00409-10
None Unchecked Km 170000.0 nM 10.1128/aac.01058-06
None Unchecked Km 175000.0 nM 10.1128/aac.00961-09
None Unchecked Km 200000.0 nM 10.1128/aac.00858-10
None Unchecked Km 305000.0 nM 10.1021/jm301490d
None Unchecked Km 340000.0 nM 10.1128/aac.01062-07
None Unchecked Km 375000.0 nM 10.1128/aac.00083-07
None Unchecked Km 700000.0 nM 10.1128/aac.00409-10
None Unchecked Km 3500000.0 nM 10.1128/aac.00166-08
None Unchecked Km 4200000.0 nM 10.1128/aac.00409-10
None Unchecked Km nan None 10.1128/aac.00774-09
None Unchecked Km nan None 10.1128/aac.01028-07
None Unchecked MIC 128.0 ug.mL-1 10.1016/j.bmcl.2003.12.037
None Unchecked Ratio 8.0 None 10.1128/aac.00614-07
None Unchecked Ratio 40.0 /mM/s 10.1128/aac.01600-06
None Unchecked Ratio 100.0 None 10.1128/aac.01463-07
None Unchecked Vmax 0.17 nmol 10.1128/aac.00389-07
None Unchecked Vmax 0.35 nmol/sec 10.1128/aac.01714-09
None Unchecked Vmax/Km 0.12 None 10.1128/aac.00389-07

Metabolism Information