| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
2.0 |
log10CFU/g |
10.1016/j.bmcl.2022.129113 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
3.5 |
log10CFU/ml |
10.1128/aac.00367-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
4.5 |
log10CFU/ml |
10.1128/aac.00367-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
5.1 |
log10CFU/ml |
10.1128/aac.00367-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
6.0 |
log10CFU/g |
10.1016/j.bmcl.2022.129113 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
78.6 |
% |
10.1128/aac.00367-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
nan |
None |
10.1128/aac.00367-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Activity |
nan |
None |
10.1128/aac.01099-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
EC50 |
470.0 |
nM |
10.1016/j.bmcl.2016.04.089 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
EC50 |
1300.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
FICI |
0.105 |
None |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
FICI |
0.126 |
None |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
FICI |
0.131 |
None |
10.1128/aac.01439-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Inhibition |
10.0 |
% |
10.1128/aac.00471-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Inhibition |
nan |
% |
10.1128/aac.00471-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
log10cfu |
8.15 |
None |
10.1128/aac.00471-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MBC |
3.13 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MBC |
4.0 |
mg/L |
10.1128/aac.00367-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MBC |
8.0 |
mg/L |
10.1128/aac.00367-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MBC |
nan |
None |
10.1021/acs.jnatprod.2c00065 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.006 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00471-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jnatprod.1c00578 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00621 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.031 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00876 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.047 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.094 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.094 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.070 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00065 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.00732-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.01037-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01742 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00876 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jnatprod.1c00578 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00621 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00072-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00732-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00748-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01037-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.01037-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.01121-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
3.1 |
ug.mL-1 |
10.1021/acs.jnatprod.0c01212 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.070 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00367-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00732-07 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01037-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01259-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00367-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01259-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01663-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01037-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01259-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01037-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01259-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01259-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01663-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
256.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01742 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01259-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.9b00288 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
3800.0 |
nM |
10.1021/acs.jnatprod.1c00232 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
nan |
None |
10.1016/j.ejmech.2019.04.067 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC100 |
2.35 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.01099-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC80 |
1.0 |
ug.mL-1 |
10.1021/np401094h |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01099-06 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Ratio |
1.0 |
None |
10.1128/aac.00748-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Ratio |
16.0 |
None |
10.1128/aac.01439-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Ratio |
21.0 |
None |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Ratio |
24.0 |
None |
10.1128/aac.00405-08 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Survival |
50.0 |
% |
10.1016/j.bmcl.2022.129113 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Survival |
71.4 |
% |
10.1128/aac.00367-09 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Survival |
90.0 |
% |
10.1016/j.bmcl.2022.129113 |
| Acinetobacter pittii |
Acinetobacter pittii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00072-08 |
| Actinomyces naeslundii |
Actinomyces naeslundii |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Bacillus anthracis |
Bacillus anthracis |
Activity |
nan |
None |
10.1128/aac.00067-10 |
| Bacillus anthracis |
Bacillus anthracis |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jnatprod.0c01309 |
| Bacillus anthracis |
Bacillus anthracis |
MIC |
31.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.043 |
| Bacillus cereus |
Bacillus cereus |
MBC |
nan |
None |
10.1021/acs.jnatprod.2c00065 |
| Bacillus cereus |
Bacillus cereus |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00360-08 |
| Bacillus cereus |
Bacillus cereus |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00065 |
| Bacillus cereus |
Bacillus cereus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00360-08 |
| Bacillus cereus |
Bacillus cereus |
MIC |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Bacillus cereus |
Bacillus cereus |
MIC |
nan |
None |
10.1016/j.bmc.2013.10.011 |
| Bacillus cereus |
Bacillus cereus |
Ratio |
8.0 |
None |
10.1128/aac.00360-08 |
| Bacillus licheniformis |
Bacillus licheniformis |
IZ |
24.0 |
mm |
10.1016/j.bmcl.2016.04.038 |
| Bacillus pumilus |
Bacillus pumilus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00389-08 |
| Bacillus spizizenii |
Bacillus spizizenii |
IZ |
13.0 |
mm |
10.1016/j.bmc.2018.02.049 |
| Bacillus spizizenii |
Bacillus spizizenii |
IZ |
25.0 |
mm |
10.1021/ml300350p |
| Bacillus spizizenii |
Bacillus spizizenii |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmc.2018.02.049 |
| Bacillus spizizenii |
Bacillus spizizenii |
MIC |
0.125 |
ug.mL-1 |
10.1021/ml300350p |
| Bacillus subtilis |
Bacillus subtilis |
Activity |
25.0 |
% |
10.1021/np020380x |
| Bacillus subtilis |
Bacillus subtilis |
Activity |
29.0 |
% |
10.1021/np020380x |
| Bacillus subtilis |
Bacillus subtilis |
Activity |
90.0 |
% |
10.1021/np020380x |
| Bacillus subtilis |
Bacillus subtilis |
Activity |
94.0 |
% |
10.1021/np020380x |
| Bacillus subtilis |
Bacillus subtilis |
Activity |
108.0 |
% |
10.1021/np020380x |
| Bacillus subtilis |
Bacillus subtilis |
Activity |
143.0 |
% |
10.1021/np020380x |
| Bacillus subtilis |
Bacillus subtilis |
Activity |
nan |
None |
10.1021/acs.jnatprod.7b00477 |
| Bacillus subtilis |
Bacillus subtilis |
FC |
2.0 |
None |
10.1016/j.bmc.2016.05.021 |
| Bacillus subtilis |
Bacillus subtilis |
GI |
100.0 |
% |
10.1016/j.bmc.2016.01.040 |
| Bacillus subtilis |
Bacillus subtilis |
Inhibition |
100.0 |
% |
10.1021/jm0703901 |
| Bacillus subtilis |
Bacillus subtilis |
Inhibition |
nan |
% |
10.1021/acs.jmedchem.7b00355 |
| Bacillus subtilis |
Bacillus subtilis |
Inhibition |
nan |
% |
10.1128/aac.01709-08 |
| Bacillus subtilis |
Bacillus subtilis |
IZ |
20.0 |
mm |
10.1016/j.bmc.2007.09.025 |
| Bacillus subtilis |
Bacillus subtilis |
IZ |
51.0 |
mm |
10.1016/j.ejmech.2008.09.035 |
| Bacillus subtilis |
Bacillus subtilis |
log(1/C) |
6.59 |
None |
10.1021/jm00210a025 |
| Bacillus subtilis |
Bacillus subtilis |
MBC |
0.4 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.01 |
ug.mL-1 |
10.1128/aac.00873-08 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.078 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00174 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.1 |
ug.mL-1 |
10.1128/aac.00873-08 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.ejmech.2007.12.019 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2020.127146 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.19 |
ug.mL-1 |
10.1007/s00044-011-9918-4 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.21 |
ug.mL-1 |
10.1021/jm00210a025 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.25 |
ug.mL-1 |
10.1021/acsmedchemlett.0c00381 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
3.125 |
ug.mL-1 |
10.1007/s00044-011-9918-4 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
3.9 |
ug.mL-1 |
10.1016/j.ejmech.2007.12.019 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
5.0 |
ug.mL-1 |
10.1021/jm400485e |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.09.035 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmc.2006.12.035 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
21.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.05.032 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
62.5 |
nM |
10.1016/j.bmc.2016.05.021 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.04.001 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
125.0 |
nM |
10.1016/j.bmc.2016.05.021 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
250.0 |
nM |
10.1016/j.bmc.2016.05.021 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.bmc.2006.12.035 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.04.001 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2019.111636 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.2c01076 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1000.0 |
nM |
10.1021/jm030003x |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1500.0 |
nM |
10.1021/jm061349l |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
4000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
nan |
None |
10.1016/j.bmc.2016.04.058 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Bacillus subtilis |
Bacillus subtilis |
MIC100 |
0.3 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Bacillus subtilis (strain 168) |
NH(3)-dependent NAD(+) synthetase |
IC50 |
1000.0 |
nM |
10.1021/jm030003x |
| Bacteria |
Cell membrane |
Activity |
3.45 |
% |
10.1021/acs.jmedchem.2c01076 |
| Bacteria |
Cell membrane |
Activity |
17.4 |
% |
10.1021/acs.jmedchem.2c01076 |
| Bacteria |
Cell membrane |
Activity |
nan |
None |
10.1021/acs.jmedchem.2c01076 |
| Bacteria |
Cell membrane |
Activity |
nan |
None |
10.1021/acs.jmedchem.8b00777 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
nan |
None |
10.1021/np050424c |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC |
nan |
None |
10.1021/np050424c |
| Bacteroides uniformis |
Bacteroides uniformis |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Bifidobacterium breve |
Bifidobacterium breve |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Bifidobacterium longum |
Bifidobacterium longum |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Bos taurus |
Progesterone receptor |
IC50 |
nan |
None |
None |
| Bos taurus |
Progesterone receptor |
Ki |
nan |
None |
None |
| Burkholderia cepacia |
Burkholderia cepacia |
Activity |
1.0 |
% |
10.1128/aac.00954-06 |
| Candida albicans |
Candida albicans |
IC50 |
nan |
None |
10.1021/jm900672t |
| Candida albicans |
Candida albicans |
IC50 |
nan |
None |
10.1021/np000436s |
| Candida albicans |
Candida albicans |
IZ |
0.0 |
mm |
10.1021/np900382x |
| Candida albicans |
Candida albicans |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.066 |
| Candida albicans |
Candida albicans |
MIC |
3.9 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.024 |
| Candida albicans |
Candida albicans |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2020.127146 |
| Candida albicans |
Candida albicans |
MIC |
256.0 |
ug.mL-1 |
10.1021/ml300350p |
| Candida albicans |
Candida albicans |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Candida albicans |
Candida albicans |
MIC |
nan |
None |
10.1016/j.bmcl.2012.09.041 |
| Candida albicans |
Candida albicans |
MIC |
nan |
None |
10.1016/j.bmcl.2013.11.024 |
| Candida albicans |
Candida albicans |
MIC |
nan |
None |
10.1016/j.bmcl.2015.01.026 |
| Candida albicans |
Candida albicans |
MIC |
nan |
None |
10.1021/acs.jnatprod.5b01129 |
| Candida albicans |
Candida albicans |
MIC |
nan |
None |
10.1021/np000436s |
| Canis lupus familiaris |
Brain |
Fu |
0.259 |
None |
10.1124/dmd.111.038778 |
| Cavia porcellus |
Cavia porcellus |
AUC |
6.22 |
None |
10.1128/aac.00196-08 |
| Cavia porcellus |
Cavia porcellus |
Cmax |
741.24 |
nM |
10.1128/aac.00120-07 |
| Cavia porcellus |
Cavia porcellus |
Cmax |
1190.84 |
nM |
10.1128/aac.00120-07 |
| Cavia porcellus |
Cavia porcellus |
Cmin |
0.14 |
ug ml-1 |
10.1128/aac.00120-07 |
| Cavia porcellus |
Cavia porcellus |
Cmin |
0.22 |
ug ml-1 |
10.1128/aac.00120-07 |
| Cavia porcellus |
Cavia porcellus |
T1/2 |
3.0 |
hr |
10.1128/aac.01533-06 |
| Cavia porcellus |
Cavia porcellus |
T1/2 |
5.8 |
hr |
10.1128/aac.00120-07 |
| Cavia porcellus |
Histamine H1 receptor |
pKb |
nan |
None |
10.1016/j.bmc.2008.10.042 |
| Cavia porcellus |
Leukotriene C4 synthase |
IC50 |
nan |
None |
None |
| Cavia porcellus |
Leukotriene C4 synthase |
Ki |
nan |
None |
None |
| Cavia porcellus |
Serotonin 4 (5-HT4) receptor |
IC50 |
nan |
None |
None |
| Cavia porcellus |
Serotonin 4 (5-HT4) receptor |
Ki |
nan |
None |
None |
| Chlamydia trachomatis |
Chlamydia trachomatis |
MIC |
0.004 |
ug.mL-1 |
10.1128/aac.00477-09 |
| Chlamydia trachomatis |
Chlamydia trachomatis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00477-09 |
| Chlamydia trachomatis |
Chlamydia trachomatis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00477-09 |
| Chlamydia trachomatis |
Chlamydia trachomatis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00477-09 |
| Chlamydia trachomatis |
Chlamydia trachomatis |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00477-09 |
| Chlorocebus sabaeus |
Vero |
Activity |
nan |
None |
10.1021/np020592u |
| Chlorocebus sabaeus |
Vero |
Activity |
nan |
None |
10.1021/np0400095 |
| Chlorocebus sabaeus |
Vero |
CC50 |
7.8 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.080 |
| Chlorocebus sabaeus |
Vero |
CC50 |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.06.055 |
| Chlorocebus sabaeus |
Vero |
CC50 |
50.0 |
ug.mL-1 |
10.1021/jm300123s |
| Chlorocebus sabaeus |
Vero |
CC50 |
128.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.041 |
| Chlorocebus sabaeus |
Vero |
CC50 |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.07.057 |
| Chlorocebus sabaeus |
Vero |
CC50 |
150.0 |
ug.mL-1 |
10.1016/j.ejmech.2015.10.024 |
| Chlorocebus sabaeus |
Vero |
CC50 |
500.0 |
ug.mL-1 |
10.1016/j.bmc.2012.09.019 |
| Chlorocebus sabaeus |
Vero |
CC50 |
500.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.07.023 |
| Chlorocebus sabaeus |
Vero |
CC50 |
500.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.05.057 |
| Chlorocebus sabaeus |
Vero |
CC50 |
512.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.090 |
| Chlorocebus sabaeus |
Vero |
CC50 |
512.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.07.025 |
| Chlorocebus sabaeus |
Vero |
CC50 |
512.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.01.042 |
| Chlorocebus sabaeus |
Vero |
CC50 |
75900.0 |
nM |
10.1007/s00044-011-9638-9 |
| Chlorocebus sabaeus |
Vero |
CC50 |
75940.0 |
nM |
10.1016/j.bmcl.2010.06.096 |
| Chlorocebus sabaeus |
Vero |
CC50 |
180000.0 |
nM |
10.1016/j.ejmech.2010.11.023 |
| Chlorocebus sabaeus |
Vero |
CC50 |
512000.0 |
nM |
10.1016/j.bmc.2019.04.017 |
| Chlorocebus sabaeus |
Vero |
CC50 |
512000.0 |
nM |
10.1016/j.ejmech.2018.09.049 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.bmc.2019.01.022 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.bmc.2022.116777 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.ejmech.2017.05.044 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.ejmech.2019.111595 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.ejmech.2021.113398 |
| Chlorocebus sabaeus |
Vero |
CD50 |
500.0 |
ug ml-1 |
10.1016/j.bmc.2013.07.003 |
| Chlorocebus sabaeus |
Vero |
GI |
44.78 |
% |
10.1016/j.bmcl.2016.06.089 |
| Chlorocebus sabaeus |
Vero |
IC50 |
10.0 |
ug.mL-1 |
10.1007/s00044-012-0074-2 |
| Chlorocebus sabaeus |
Vero |
IC50 |
58.0 |
ug.mL-1 |
10.1016/j.bmc.2013.06.027 |
| Chlorocebus sabaeus |
Vero |
IC50 |
62.5 |
ug.mL-1 |
10.1016/j.bmcl.2009.12.045 |
| Chlorocebus sabaeus |
Vero |
IC50 |
62.5 |
ug.mL-1 |
10.1016/j.bmcl.2012.12.069 |
| Chlorocebus sabaeus |
Vero |
IC50 |
62.5 |
ug.mL-1 |
10.1016/j.ejmech.2014.03.085 |
| Chlorocebus sabaeus |
Vero |
IC50 |
62.5 |
ug.mL-1 |
10.1021/jm060339h |
| Chlorocebus sabaeus |
Vero |
IC50 |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2022.117006 |
| Chlorocebus sabaeus |
Vero |
IC50 |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113603 |
| Chlorocebus sabaeus |
Vero |
IC50 |
89.3 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.029 |
| Chlorocebus sabaeus |
Vero |
IC50 |
97.4 |
ug.mL-1 |
10.1021/acs.jnatprod.8b00567 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100.0 |
ug.mL-1 |
10.1016/j.bmc.2007.05.063 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100.0 |
ug.mL-1 |
10.1016/j.bmc.2008.10.086 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100.0 |
ug.mL-1 |
10.1016/j.bmc.2010.02.024 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.06.010 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.10.050 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100.0 |
ug.mL-1 |
10.1021/acsmedchemlett.8b00410 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100.0 |
ug.mL-1 |
10.1021/np400497f |
| Chlorocebus sabaeus |
Vero |
IC50 |
110.67 |
ug.mL-1 |
10.1021/jm020891g |
| Chlorocebus sabaeus |
Vero |
IC50 |
137.6 |
ug.mL-1 |
10.1016/j.ejmech.2020.112045 |
| Chlorocebus sabaeus |
Vero |
IC50 |
142.9 |
ug.mL-1 |
10.1021/np400145u |
| Chlorocebus sabaeus |
Vero |
IC50 |
147.0 |
ug.mL-1 |
10.1016/s0960-894x(00)00058-5 |
| Chlorocebus sabaeus |
Vero |
IC50 |
158.0 |
ug.mL-1 |
10.1021/np980066w |
| Chlorocebus sabaeus |
Vero |
IC50 |
200.0 |
ug.mL-1 |
10.1016/j.bmc.2018.07.034 |
| Chlorocebus sabaeus |
Vero |
IC50 |
256.0 |
ug.mL-1 |
10.1021/acs.jmedchem.7b00582 |
| Chlorocebus sabaeus |
Vero |
IC50 |
1000.0 |
ug.mL-1 |
10.1016/s0960-894x(01)00266-9 |
| Chlorocebus sabaeus |
Vero |
IC50 |
50000.0 |
nM |
10.1016/j.bmc.2016.12.038 |
| Chlorocebus sabaeus |
Vero |
IC50 |
74500.0 |
nM |
10.1016/j.ejmech.2010.05.035 |
| Chlorocebus sabaeus |
Vero |
IC50 |
75900.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Chlorocebus sabaeus |
Vero |
IC50 |
75940.0 |
nM |
10.1016/j.bmcl.2007.01.037 |
| Chlorocebus sabaeus |
Vero |
IC50 |
75940.0 |
nM |
10.1016/j.ejmech.2009.09.033 |
| Chlorocebus sabaeus |
Vero |
IC50 |
77400.0 |
nM |
10.1007/s00044-010-9322-5 |
| Chlorocebus sabaeus |
Vero |
IC50 |
97900.0 |
nM |
10.1021/np800751j |
| Chlorocebus sabaeus |
Vero |
IC50 |
100000.0 |
nM |
10.1016/j.bmc.2007.05.053 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100000.0 |
nM |
10.1016/j.bmcl.2012.06.095 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100000.0 |
nM |
10.1016/j.bmcl.2015.12.080 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100000.0 |
nM |
10.1016/j.bmcl.2016.06.089 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100000.0 |
nM |
10.1016/j.ejmech.2013.01.017 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100000.0 |
nM |
10.1021/acsmedchemlett.7b00356 |
| Chlorocebus sabaeus |
Vero |
IC50 |
105000.0 |
nM |
10.1007/s00044-007-9073-0 |
| Chlorocebus sabaeus |
Vero |
IC50 |
108000.0 |
nM |
10.1016/j.bmcl.2013.09.013 |
| Chlorocebus sabaeus |
Vero |
IC50 |
113000.0 |
nM |
10.1016/j.bmc.2012.02.025 |
| Chlorocebus sabaeus |
Vero |
IC50 |
113000.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Chlorocebus sabaeus |
Vero |
IC50 |
113000.0 |
nM |
10.1021/ml200036r |
| Chlorocebus sabaeus |
Vero |
IC50 |
122000.0 |
nM |
10.1016/j.bmcl.2009.11.105 |
| Chlorocebus sabaeus |
Vero |
IC50 |
122000.0 |
nM |
10.1021/acs.jnatprod.9b01095 |
| Chlorocebus sabaeus |
Vero |
IC50 |
122000.0 |
nM |
10.1021/jm900340a |
| Chlorocebus sabaeus |
Vero |
IC50 |
122000.0 |
nM |
10.1021/jm901235p |
| Chlorocebus sabaeus |
Vero |
IC50 |
125000.0 |
nM |
10.1016/j.ejmech.2009.12.074 |
| Chlorocebus sabaeus |
Vero |
IC50 |
127000.0 |
nM |
10.1021/jm900003c |
| Chlorocebus sabaeus |
Vero |
IC50 |
127000.0 |
nM |
10.1021/jm900513a |
| Chlorocebus sabaeus |
Vero |
IC50 |
132500.0 |
nM |
10.1021/np400391p |
| Chlorocebus sabaeus |
Vero |
IC50 |
134480.0 |
nM |
10.1021/jm020891g |
| Chlorocebus sabaeus |
Vero |
IC50 |
138300.0 |
nM |
10.1016/j.bmc.2008.12.006 |
| Chlorocebus sabaeus |
Vero |
IC50 |
182000.0 |
nM |
10.1016/j.bmcl.2013.11.024 |
| Chlorocebus sabaeus |
Vero |
IC50 |
nan |
None |
10.1016/j.bmcl.2012.05.096 |
| Chlorocebus sabaeus |
Vero |
IC50 |
nan |
None |
10.1021/acs.jmedchem.5b01542 |
| Chlorocebus sabaeus |
Vero |
IC50 |
nan |
None |
10.1021/acsmedchemlett.5b00176 |
| Chlorocebus sabaeus |
Vero |
IC50 |
nan |
None |
10.1021/np0601399 |
| Chlorocebus sabaeus |
Vero |
Maximal non-toxic dose 50 |
64.0 |
ug ml-1 |
10.1021/jm0602662 |
| Chlorocebus sabaeus |
Vero |
MIC |
127000.0 |
nM |
10.1021/jm901112f |
| Chlorocebus sabaeus |
Vero |
MIC |
127000.0 |
nM |
10.1021/jm901273n |
| Chlorocebus sabaeus |
Vero |
MNTD |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2009.06.005 |
| Chlorocebus sabaeus |
Vero |
MNTD50 |
64.0 |
ug ml-1 |
10.1021/jm701560p |
| Chlorocebus sabaeus |
Vero |
MTD50 |
64.0 |
ug ml-1 |
10.1016/s0960-894x(99)00510-7 |
| Chlorocebus sabaeus |
Vero |
PI |
213.0 |
None |
10.1021/jm0602662 |
| Chlorocebus sabaeus |
Vero |
Ratio IC50 |
1080.0 |
None |
10.1016/j.bmc.2010.03.018 |
| Chlorocebus sabaeus |
Vero |
Selectivity |
400.0 |
None |
10.1016/j.bmcl.2005.06.010 |
| Citrobacter freundii |
Citrobacter freundii |
MIC |
0.023 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Citrobacter freundii |
Citrobacter freundii |
Ratio |
500.0 |
None |
10.1128/aac.00405-08 |
| Clostridioides difficile |
Clostridioides difficile |
MBC |
0.78 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.00342-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
9e-05 |
ug.mL-1 |
10.1128/aac.00342-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.0004 |
ug.mL-1 |
10.1128/aac.00342-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.0009 |
ug.mL-1 |
10.1128/aac.00342-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.001 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.0019 |
ug.mL-1 |
10.1128/aac.00342-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.002 |
ug.mL-1 |
10.1128/aac.00342-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.003 |
ug.mL-1 |
10.1128/aac.00342-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.004 |
ug.mL-1 |
10.1128/aac.00342-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00476-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.015 |
ug.mL-1 |
10.1021/acsmedchemlett.0c00381 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00342-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.06 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
16.0 |
ug.mL-1 |
10.1021/acsmedchemlett.0c00381 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00342-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00342-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00342-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.00476-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC90 |
0.015 |
ug.mL-1 |
10.1128/aac.00476-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC90 |
128.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Clostridium perfringens |
Clostridium perfringens |
log(1/C) |
8.44 |
None |
10.1021/jm00210a025 |
| Clostridium perfringens |
Clostridium perfringens |
MIC |
0.003 |
ug.mL-1 |
10.1021/jm00210a025 |
| Clostridium sporogenes |
Clostridium sporogenes |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Cricetulus griseus |
CHO |
CC50 |
512000.0 |
nM |
10.1016/j.ejmech.2019.111678 |
| Cricetulus griseus |
CHO |
IC50 |
nan |
None |
10.1021/acs.jmedchem.1c00707 |
| Cryptococcus neoformans |
Cryptococcus neoformans |
IC50 |
nan |
None |
10.1021/jm900672t |
| Cryptococcus neoformans |
Cryptococcus neoformans |
IC50 |
nan |
None |
10.1021/np000436s |
| Cryptococcus neoformans |
Cryptococcus neoformans |
MIC |
nan |
None |
10.1021/np000436s |
| Dialister invisus |
Dialister invisus |
Activity |
2.0 |
ug ml-1 |
10.1128/aac.00538-07 |
| Dialister invisus |
Dialister invisus |
Activity |
nan |
None |
10.1128/aac.00538-07 |
| Dialister invisus |
Dialister invisus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Dialister micraerophilus |
Dialister micraerophilus |
Activity |
2.0 |
ug ml-1 |
10.1128/aac.00538-07 |
| Dialister micraerophilus |
Dialister micraerophilus |
Activity |
nan |
None |
10.1128/aac.00538-07 |
| Dialister micraerophilus |
Dialister micraerophilus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Dialister micraerophilus |
Dialister micraerophilus |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Dialister micraerophilus |
Dialister micraerophilus |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Dialister pneumosintes |
Dialister pneumosintes |
Activity |
2.0 |
ug ml-1 |
10.1128/aac.00538-07 |
| Dialister pneumosintes |
Dialister pneumosintes |
Activity |
nan |
None |
10.1128/aac.00538-07 |
| Dialister pneumosintes |
Dialister pneumosintes |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Dialister pneumosintes |
Dialister pneumosintes |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Dialister pneumosintes |
Dialister pneumosintes |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Dialister propionicifaciens |
Dialister propionicifaciens |
Activity |
2.0 |
ug ml-1 |
10.1128/aac.00538-07 |
| Dialister propionicifaciens |
Dialister propionicifaciens |
Activity |
nan |
None |
10.1128/aac.00538-07 |
| Dialister propionicifaciens |
Dialister propionicifaciens |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00538-07 |
| Electrophorus electricus |
Acetylcholinesterase |
Inhibition |
16.23 |
% |
10.1016/j.bmc.2012.09.040 |
| Enterobacter cloacae |
Enterobacter cloacae |
EC50 |
6200.0 |
nM |
10.1016/j.bmcl.2016.04.089 |
| Enterobacter cloacae |
Enterobacter cloacae |
EC50 |
8800.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| Enterobacter cloacae |
Enterobacter cloacae |
FICI |
0.126 |
None |
10.1128/aac.01439-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
IZ |
0.0 |
mm |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
IZ |
8.0 |
mm |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
IZ |
10.0 |
mm |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
IZ |
13.0 |
mm |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
IZ |
26.0 |
mm |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
IZ |
28.0 |
mm |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MBC |
nan |
None |
10.1021/acs.jnatprod.2c00065 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.26 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01742 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00065 |
| Enterobacter cloacae |
Enterobacter cloacae |
Ratio |
260.0 |
None |
10.1128/aac.01439-09 |
| Enterobacter cloacae |
Enterobacter cloacae |
Ratio |
500.0 |
None |
10.1128/aac.00405-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
Ratio |
750.0 |
None |
10.1128/aac.00405-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
Ratio |
1400.0 |
None |
10.1128/aac.00405-08 |
| Enterococcus avium |
Enterococcus avium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00908-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
IC50 |
10000.0 |
nM |
10.1021/acs.jnatprod.2c00444 |
| Enterococcus faecalis |
Enterococcus faecalis |
IZ |
20.0 |
mm |
10.1016/j.bmc.2007.09.025 |
| Enterococcus faecalis |
Enterococcus faecalis |
IZ |
21.0 |
mm |
10.1016/j.bmc.2019.115097 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
1.56 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.008 |
ug.mL-1 |
10.1021/np050176k |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jnatprod.9b00062 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2020.127146 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm501082n |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00576-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.077 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.066 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1021/ml300350p |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00576-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00908-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.077 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00576-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00908-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.077 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00520 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.02.009 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1016/j.bmc.2019.04.032 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1021/np050424c |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC100 |
0.78 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC100 |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC>90 |
0.2 |
ug ml-1 |
10.1021/np400145u |
| Enterococcus faecium |
Enterococcus faecium |
EC50 |
130.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| Enterococcus faecium |
Enterococcus faecium |
EC50 |
1200.0 |
nM |
10.1016/j.bmcl.2016.04.089 |
| Enterococcus faecium |
Enterococcus faecium |
IC50 |
8.75 |
ug.mL-1 |
10.1021/np2006555 |
| Enterococcus faecium |
Enterococcus faecium |
IZ |
9.0 |
mm |
10.1016/j.bmc.2019.115097 |
| Enterococcus faecium |
Enterococcus faecium |
IZ |
nan |
None |
10.1021/np900382x |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
nan |
None |
10.1021/acs.jnatprod.2c00065 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.04 |
ug.mL-1 |
10.1021/np050176k |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
3.1 |
ug.mL-1 |
10.1021/acs.jnatprod.0c01212 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00576-06 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00065 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
21000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Equus caballus |
Cholinesterase |
Inhibition |
1.88 |
% |
10.1016/j.bmc.2012.09.040 |
| Escherichia coli |
DNA repair protein RecN |
Activity |
nan |
None |
10.1021/acs.jmedchem.0c00328 |
| Escherichia coli |
Escherichia coli |
AC50 |
32271.0 |
nM |
None |
| Escherichia coli |
Escherichia coli |
Activity |
0.0 |
% |
10.1128/aac.00375-07 |
| Escherichia coli |
Escherichia coli |
Activity |
1.17 |
% |
10.1021/np010076o |
| Escherichia coli |
Escherichia coli |
Activity |
27.82 |
% |
10.1021/np010076o |
| Escherichia coli |
Escherichia coli |
Activity |
32.6 |
% |
10.1128/aac.00375-07 |
| Escherichia coli |
Escherichia coli |
Activity |
32.8 |
% |
10.1128/aac.00375-07 |
| Escherichia coli |
Escherichia coli |
Activity |
35.8 |
% |
10.1128/aac.00375-07 |
| Escherichia coli |
Escherichia coli |
Activity |
64.0 |
mg/L |
10.1021/jm501082n |
| Escherichia coli |
Escherichia coli |
Activity |
80.2 |
% |
10.1128/aac.00375-07 |
| Escherichia coli |
Escherichia coli |
Activity |
85.1 |
% |
10.1128/aac.00375-07 |
| Escherichia coli |
Escherichia coli |
Activity |
89.56 |
% |
10.1021/np010076o |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1016/j.bmcl.2013.02.005 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1016/j.ejmech.2019.111636 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1021/acs.jmedchem.2c01076 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1021/jm400485e |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1128/aac.00043-09 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1128/aac.00375-07 |
| Escherichia coli |
Escherichia coli |
Antibiotic resistance |
nan |
None |
10.1016/s0960-894x(98)00536-8 |
| Escherichia coli |
Escherichia coli |
FC |
16.0 |
None |
10.1021/acs.jmedchem.2c01076 |
| Escherichia coli |
Escherichia coli |
FICI |
0.071 |
None |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
FICI |
0.111 |
None |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
FICI |
0.126 |
None |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
FICI |
0.128 |
None |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
GI |
98.0 |
% |
10.1016/j.bmc.2016.01.040 |
| Escherichia coli |
Escherichia coli |
IC90 |
0.5 |
ug.mL-1 |
10.1021/np400002p |
| Escherichia coli |
Escherichia coli |
Inhibition |
10.0 |
% |
10.1128/aac.00471-08 |
| Escherichia coli |
Escherichia coli |
Inhibition |
100.0 |
% |
10.1021/jm0703901 |
| Escherichia coli |
Escherichia coli |
Inhibition |
nan |
% |
10.1016/j.bmc.2018.07.034 |
| Escherichia coli |
Escherichia coli |
Inhibition |
nan |
% |
10.1128/aac.00471-08 |
| Escherichia coli |
Escherichia coli |
Inhibition |
nan |
% |
10.1128/aac.00691-09 |
| Escherichia coli |
Escherichia coli |
IZ |
6.0 |
mm |
10.1021/np900382x |
| Escherichia coli |
Escherichia coli |
IZ |
11.0 |
mm |
10.1016/j.bmc.2018.02.049 |
| Escherichia coli |
Escherichia coli |
IZ |
14.0 |
mm |
10.1016/j.bmc.2007.09.025 |
| Escherichia coli |
Escherichia coli |
IZ |
20.0 |
mm |
10.1021/np900382x |
| Escherichia coli |
Escherichia coli |
IZ |
27.0 |
mm |
10.1016/j.bmcl.2016.04.038 |
| Escherichia coli |
Escherichia coli |
IZ |
48.0 |
mm |
10.1016/j.ejmech.2008.09.035 |
| Escherichia coli |
Escherichia coli |
log10cfu |
8.58 |
None |
10.1128/aac.00471-08 |
| Escherichia coli |
Escherichia coli |
MBC |
3.0 |
ug ml-1 |
10.1128/aac.00375-07 |
| Escherichia coli |
Escherichia coli |
MBC |
8.0 |
ug ml-1 |
10.1016/j.bmcl.2023.129320 |
| Escherichia coli |
Escherichia coli |
MBC |
8.0 |
ug ml-1 |
10.1021/acs.jnatprod.5b00770 |
| Escherichia coli |
Escherichia coli |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Escherichia coli |
Escherichia coli |
MIC |
0.006 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00471-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.01333 |
ug.mL-1 |
10.1016/j.ejmech.2022.114108 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.02 |
ug.mL-1 |
10.1021/np050176k |
| Escherichia coli |
Escherichia coli |
MIC |
0.023 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.031 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.031 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.047 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.055 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1021/acs.jnatprod.1c00578 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00621 |
| Escherichia coli |
Escherichia coli |
MIC |
0.06 |
ug.mL-1 |
10.1021/jm501082n |
| Escherichia coli |
Escherichia coli |
MIC |
0.063 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.070 |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1021/jm301499r |
| Escherichia coli |
Escherichia coli |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.24 |
ug.mL-1 |
10.1016/j.bmcl.2006.10.016 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2008.09.035 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2018.02.049 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm501082n |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.64 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.066 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.024 |
ug.mL-1 |
10.1016/j.ejmech.2022.114108 |
| Escherichia coli |
Escherichia coli |
MIC |
1.9 |
ug.mL-1 |
10.1016/j.ejmech.2007.12.019 |
| Escherichia coli |
Escherichia coli |
MIC |
1.9 |
ug.mL-1 |
10.1128/aac.00580-10 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.077 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.03.061 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm020183v |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00375-07 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00748-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01783-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2.1 |
ug.mL-1 |
10.1128/aac.00580-10 |
| Escherichia coli |
Escherichia coli |
MIC |
2.5 |
ug.mL-1 |
10.1021/acs.jmedchem.7b00204 |
| Escherichia coli |
Escherichia coli |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.00375-07 |
| Escherichia coli |
Escherichia coli |
MIC |
3.9 |
ug.mL-1 |
10.1016/j.ejmech.2007.12.019 |
| Escherichia coli |
Escherichia coli |
MIC |
3.9 |
ug.mL-1 |
10.1128/aac.00580-10 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2023.129320 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.070 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jnatprod.0c01309 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00310-09 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00375-07 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01783-09 |
| Escherichia coli |
Escherichia coli |
MIC |
5.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.04.060 |
| Escherichia coli |
Escherichia coli |
MIC |
6.0 |
ug.mL-1 |
10.1021/jm00143a010 |
| Escherichia coli |
Escherichia coli |
MIC |
6.0 |
ug.mL-1 |
10.1021/jm00145a020 |
| Escherichia coli |
Escherichia coli |
MIC |
6.0 |
ug.mL-1 |
10.1021/jm00220a012 |
| Escherichia coli |
Escherichia coli |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.00375-07 |
| Escherichia coli |
Escherichia coli |
MIC |
6.25 |
ug.mL-1 |
10.1128/aac.00475-08 |
| Escherichia coli |
Escherichia coli |
MIC |
6.3 |
ug.mL-1 |
10.1021/acs.jnatprod.0c01212 |
| Escherichia coli |
Escherichia coli |
MIC |
7.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.04.060 |
| Escherichia coli |
Escherichia coli |
MIC |
7.0 |
ug.mL-1 |
10.1021/jm400485e |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.10.016 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2020.127146 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.04.001 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.02.009 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jnatprod.1c00578 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00621 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jnatprod.5b00770 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm301499r |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm501082n |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1021/ml300350p |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1039/d2md00041e |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00017-08 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00638-08 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01052-07 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01783-09 |
| Escherichia coli |
Escherichia coli |
MIC |
10.0 |
ug.mL-1 |
10.1021/jm400485e |
| Escherichia coli |
Escherichia coli |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.113049 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00043-09 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00638-08 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01052-07 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01053-06 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01128-06 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01783-09 |
| Escherichia coli |
Escherichia coli |
MIC |
20.0 |
ug.mL-1 |
10.1021/jm970791o |
| Escherichia coli |
Escherichia coli |
MIC |
22.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.05.032 |
| Escherichia coli |
Escherichia coli |
MIC |
24.0 |
ug.mL-1 |
10.1128/aac.01128-06 |
| Escherichia coli |
Escherichia coli |
MIC |
31.0 |
ug.mL-1 |
10.1021/jm501082n |
| Escherichia coli |
Escherichia coli |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| Escherichia coli |
Escherichia coli |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| Escherichia coli |
Escherichia coli |
MIC |
62.5 |
ug.mL-1 |
10.1016/j.bmc.2006.12.035 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.01.026 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.04.001 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Escherichia coli |
Escherichia coli |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Escherichia coli |
Escherichia coli |
MIC |
250.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.10.016 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1016/j.bmc.2006.12.035 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00310-09 |
| Escherichia coli |
Escherichia coli |
MIC |
2000.0 |
nM |
10.1016/j.ejmech.2019.111636 |
| Escherichia coli |
Escherichia coli |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2019.111636 |
| Escherichia coli |
Escherichia coli |
MIC |
4000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Escherichia coli |
Escherichia coli |
MIC |
4000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Escherichia coli |
Escherichia coli |
MIC |
4000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Escherichia coli |
Escherichia coli |
MIC |
4000.0 |
nM |
10.1021/acs.jmedchem.2c01076 |
| Escherichia coli |
Escherichia coli |
MIC |
4000.0 |
nM |
10.1021/acs.jmedchem.9b00288 |
| Escherichia coli |
Escherichia coli |
MIC |
8000.0 |
nM |
10.1021/acs.jmedchem.9b00288 |
| Escherichia coli |
Escherichia coli |
MIC |
10000.0 |
nM |
10.1021/acs.jnatprod.5b01129 |
| Escherichia coli |
Escherichia coli |
MIC |
16000.0 |
nM |
10.1016/j.bmc.2016.04.058 |
| Escherichia coli |
Escherichia coli |
MIC |
55000.0 |
nM |
10.1016/j.bmc.2016.04.058 |
| Escherichia coli |
Escherichia coli |
MIC |
25922000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.bmc.2013.10.011 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.bmc.2019.04.032 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.bmcl.2013.11.024 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.ejmech.2019.04.067 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1021/np050424c |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1021/np200320u |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
MIC100 |
3.13 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Escherichia coli |
Escherichia coli |
MIC90 |
100.0 |
nM |
10.1016/j.bmcl.2011.08.054 |
| Escherichia coli |
Escherichia coli |
MIC90 |
128.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.11.042 |
| Escherichia coli |
Escherichia coli |
MIC90 |
12500.0 |
nM |
10.1016/j.bmcl.2011.08.054 |
| Escherichia coli |
Escherichia coli |
MIC99 |
nan |
None |
10.1016/j.ejmech.2013.10.055 |
| Escherichia coli |
Escherichia coli |
Ratio |
1.0 |
None |
10.1128/aac.00748-09 |
| Escherichia coli |
Escherichia coli |
Ratio |
8.0 |
None |
10.1021/jm501082n |
| Escherichia coli |
Escherichia coli |
Ratio |
32.0 |
None |
10.1016/j.bmcl.2006.10.016 |
| Escherichia coli |
Escherichia coli |
Ratio |
32.0 |
None |
10.1016/j.ejmech.2019.111636 |
| Escherichia coli |
Escherichia coli |
Ratio |
85.0 |
None |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
Ratio |
85.0 |
None |
10.1128/aac.01439-09 |
| Escherichia coli |
Escherichia coli |
Ratio |
125.0 |
None |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
Ratio |
170.0 |
None |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
Ratio |
250.0 |
None |
10.1128/aac.00405-08 |
| Escherichia coli |
Escherichia coli |
Ratio |
250.0 |
None |
10.1128/aac.01439-09 |
| Escherichia coli |
GroEL/GroES |
IC50 |
100000.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| Escherichia coli |
LexA repressor |
Activity |
nan |
None |
10.1021/acs.jmedchem.0c00328 |
| Escherichia coli K-12 |
Beta-lactamase AmpC |
Potency |
707.9 |
nM |
None |
| Escherichia coli K-12 |
Cell division inhibitor sulA |
Activity |
nan |
None |
10.1021/acs.jmedchem.0c00328 |
| Escherichia coli K-12 |
DNA-directed RNA polymerase beta chain |
Inhibition |
57.0 |
% |
10.1021/jm00125a022 |
| Escherichia coli K-12 |
Phospho-N-acetylmuramoyl-pentapeptide-transferase |
IC50 |
nan |
ug.mL-1 |
10.1016/s0960-894x(03)00597-3 |
| Escherichia coli K-12 |
Recombinase A |
Activity |
nan |
None |
10.1021/acs.jmedchem.0c00328 |
| Escherichia coli O127:H6 (strain E2348/69 / EPEC) |
DNA-directed RNA polymerase subunit beta |
IC50 |
171000.0 |
nM |
10.1021/jm4004889 |
| Escherichia coli O127:H6 (strain E2348/69 / EPEC) |
DNA-directed RNA polymerase subunit beta |
IC50 |
233000.0 |
nM |
10.1021/jm4004889 |
| Escherichia coli O127:H6 (strain E2348/69 / EPEC) |
DNA-directed RNA polymerase subunit beta |
IC50 |
1130000.0 |
nM |
10.1021/jm4004889 |
| Fannyhessea vaginae |
Fannyhessea vaginae |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Fusobacterium nucleatum |
Fusobacterium nucleatum |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Gardnerella vaginalis |
Gardnerella vaginalis |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Haemophilus influenzae |
Haemophilus influenzae |
Inhibition |
10.0 |
% |
10.1128/aac.00471-08 |
| Haemophilus influenzae |
Haemophilus influenzae |
Inhibition |
nan |
% |
10.1128/aac.00471-08 |
| Haemophilus influenzae |
Haemophilus influenzae |
log10cfu |
8.14 |
None |
10.1128/aac.00471-08 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.0008 |
ug.mL-1 |
10.1128/aac.00471-08 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.125 |
ug.mL-1 |
10.1021/jm00167a029 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01545-06 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01545-06 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
25.0 |
nM |
10.1021/acs.jmedchem.5b00050 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01545-06 |
| Helicobacter pylori |
Helicobacter pylori |
MIC |
0.007 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Helicobacter pylori |
Helicobacter pylori |
MIC |
0.06 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Helicobacter pylori |
Helicobacter pylori |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Helicobacter pylori |
Helicobacter pylori |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Helicobacter pylori |
Helicobacter pylori |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Helicobacter pylori |
Helicobacter pylori |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Helicobacter pylori |
Helicobacter pylori |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Helicobacter pylori |
Helicobacter pylori |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Helicobacter pylori |
Helicobacter pylori |
MIC90 |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Helicobacter pylori |
Helicobacter pylori |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Homo sapiens |
A549 |
Activity |
34.0 |
% |
10.1128/aac.00985-07 |
| Homo sapiens |
A549 |
Activity |
45.0 |
% |
10.1128/aac.00985-07 |
| Homo sapiens |
A549 |
Activity |
47.0 |
% |
10.1128/aac.00985-07 |
| Homo sapiens |
A549 |
Activity |
53.0 |
% |
10.1128/aac.00985-07 |
| Homo sapiens |
A549 |
Activity |
59.0 |
% |
10.1128/aac.00985-07 |
| Homo sapiens |
A549 |
Activity |
79.0 |
% |
10.1128/aac.00985-07 |
| Homo sapiens |
A549 |
Activity |
95.0 |
% |
10.1128/aac.00985-07 |
| Homo sapiens |
A549 |
Activity |
178.0 |
ug ml-1 |
10.1016/j.bmcl.2009.09.095 |
| Homo sapiens |
A549 |
Activity |
nan |
None |
10.1128/aac.00961-08 |
| Homo sapiens |
A549 |
Activity |
nan |
None |
10.1128/aac.00985-07 |
| Homo sapiens |
A549 |
CD50 |
nan |
None |
10.1016/j.bmc.2013.07.003 |
| Homo sapiens |
A549 |
FC |
1.9 |
None |
10.1128/aac.00961-08 |
| Homo sapiens |
A549 |
FC |
2.1 |
None |
10.1128/aac.00961-08 |
| Homo sapiens |
A549 |
FC |
4.0 |
None |
10.1128/aac.00961-08 |
| Homo sapiens |
A549 |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.045 |
| Homo sapiens |
A549 |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.01.004 |
| Homo sapiens |
A549 |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.03.020 |
| Homo sapiens |
A549 |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.03.065 |
| Homo sapiens |
A549 |
GI50 |
100.0 |
ug.mL-1 |
10.1039/C5MD00404G |
| Homo sapiens |
A549 |
GI50 |
121510000.0 |
nM |
10.1039/C6MD00278A |
| Homo sapiens |
A549 |
GI90 |
100.0 |
ug ml-1 |
10.1016/j.bmcl.2017.01.004 |
| Homo sapiens |
A549 |
GI90 |
100.0 |
ug ml-1 |
10.1016/j.bmcl.2019.03.020 |
| Homo sapiens |
A549 |
GI90 |
100.0 |
ug ml-1 |
10.1016/j.ejmech.2017.03.065 |
| Homo sapiens |
A549 |
Inhibition |
5.5 |
% |
10.1128/aac.00985-07 |
| Homo sapiens |
A549 |
Inhibition |
8.3 |
% |
10.1128/aac.00985-07 |
| Homo sapiens |
A549 |
Inhibition |
nan |
% |
10.1128/aac.00985-07 |
| Homo sapiens |
Acetylcholinesterase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Acetylcholinesterase |
Inhibition |
12.2 |
% |
10.1016/j.ejmech.2018.04.058 |
| Homo sapiens |
Acetylcholinesterase |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A1 receptor |
AC50 |
18808.1 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A2a receptor |
AC50 |
12966.1 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A2a receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A2a receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A3 receptor |
AC50 |
26999.8 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A3 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A3 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
2331.5 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1d adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-1d adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2b adrenergic receptor |
AC50 |
12000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2b adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2b adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2c adrenergic receptor |
AC50 |
10999.9 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2c adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2c adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-synuclein |
IC50 |
7100.0 |
nM |
10.1016/j.ejmech.2019.01.045 |
| Homo sapiens |
Alpha-synuclein |
IC50 |
46200.0 |
nM |
10.1016/j.ejmech.2019.01.045 |
| Homo sapiens |
Amyloid-beta A4 protein |
Activity |
48.4 |
% |
10.1039/C9MD00030E |
| Homo sapiens |
Amyloid-beta A4 protein |
Inhibition |
27.5 |
% |
10.1016/j.ejmech.2018.04.058 |
| Homo sapiens |
Angiotensin II type 2 (AT-2) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Angiotensin II type 2 (AT-2) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Arylacetamide deacetylase |
Drug metabolism |
41.77 |
pmol/min/mg |
10.1124/dmd.112.044537 |
| Homo sapiens |
Arylacetamide deacetylase |
Ki |
200000.0 |
nM |
10.1124/dmd.111.043067 |
| Homo sapiens |
Arylacetamide deacetylase |
Ki |
300000.0 |
nM |
10.1124/dmd.111.043067 |
| Homo sapiens |
Arylacetamide deacetylase |
Ki |
700000.0 |
nM |
10.1124/dmd.111.043067 |
| Homo sapiens |
Arylacetamide deacetylase |
Km |
200000.0 |
nM |
10.1124/dmd.111.043067 |
| Homo sapiens |
Arylacetamide deacetylase |
Km |
300000.0 |
nM |
10.1124/dmd.111.043067 |
| Homo sapiens |
Arylacetamide deacetylase |
Km |
400000.0 |
nM |
10.1124/dmd.111.043067 |
| Homo sapiens |
Arylacetamide deacetylase |
Vmax |
149.0 |
pmol/min/U |
10.1124/dmd.111.043067 |
| Homo sapiens |
Arylacetamide deacetylase |
Vmax |
211.8 |
pmol/min/mg |
10.1124/dmd.111.043067 |
| Homo sapiens |
Arylacetamide deacetylase |
Vmax |
272.6 |
pmol/min/mg |
10.1124/dmd.111.043067 |
| Homo sapiens |
Arylacetamide deacetylase |
Vmax/Km |
0.9 |
uL/min/U |
10.1124/dmd.111.043067 |
| Homo sapiens |
ATP-binding cassette sub-family G member 2 |
IC50 |
56000.0 |
nM |
10.1016/j.ejmech.2022.114346 |
| Homo sapiens |
Beta-1 adrenergic receptor |
AC50 |
28000.1 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-1 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-1 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
AC50 |
29000.1 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-2 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-3 adrenergic receptor |
AC50 |
32600.2 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-3 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-3 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Bile acid receptor FXR |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bile acid receptor FXR |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bile salt export pump |
AC50 |
9600.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bile salt export pump |
Activity |
nan |
None |
10.1038/nrd3028 |
| Homo sapiens |
Bile salt export pump |
IC50 |
11300.0 |
nM |
10.1124/dmd.111.040758 |
| Homo sapiens |
Bile salt export pump |
IC50 |
18700.0 |
nM |
10.1002/hep.27206 |
| Homo sapiens |
Bile salt export pump |
IC50 |
25300.0 |
nM |
10.1093/toxsci/kfq269 |
| Homo sapiens |
Bile salt export pump |
IC50 |
25300.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Bradykinin B1 receptor |
AC50 |
14249.8 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bradykinin B2 receptor |
AC50 |
18577.4 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bradykinin B2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Bradykinin B2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Brain |
Drug uptake |
0.29 |
ug ml-1 |
10.1021/jm901858n |
| Homo sapiens |
Bromodomain adjacent to zinc finger domain protein 2B |
Potency |
50118.7 |
nM |
None |
| Homo sapiens |
Calcitonin receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Calcitonin receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Canalicular multispecific organic anion transporter 1 |
Activity |
18.0 |
% |
10.1021/jm7015683 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 1 |
Activity |
nan |
None |
10.1016/s0002-9440(10)64794-3 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 1 |
Activity |
nan |
None |
10.1016/s0300-483x(01)00570-4 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 1 |
IC50 |
53000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 2 |
IC50 |
69000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Cannabinoid CB1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cannabinoid CB1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cannabinoid CB1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cannabinoid CB1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase II |
IC50 |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase II |
Ki |
nan |
None |
None |
| Homo sapiens |
Carboxylesterase 2 |
Drug metabolism |
2.99 |
pmol/min/mg |
10.1124/dmd.112.044537 |
| Homo sapiens |
Caspase-1 |
IC50 |
8319.0 |
nM |
None |
| Homo sapiens |
Caspase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cathepsin G |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cathepsin G |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 2 |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 4 |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin A receptor |
AC50 |
17080.1 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cholecystokinin A receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin A receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin B receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Chromobox protein homolog 1 |
Potency |
39810.7 |
nM |
None |
| Homo sapiens |
Corticotropin releasing factor receptor 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Corticotropin releasing factor receptor 2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-2 |
AC50 |
6400.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cysteinyl leukotriene receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cysteinyl leukotriene receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 |
Activity |
65.0 |
% |
10.1021/acs.jmedchem.0c02245 |
| Homo sapiens |
Cytochrome P450 1A2 |
FC |
1.37 |
None |
10.1128/aac.00660-09 |
| Homo sapiens |
Cytochrome P450 1A2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 1A2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2A6 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2A6 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2B6 |
Activity |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2B6 |
EC50 |
1300.0 |
nM |
10.1124/dmd.112.047118 |
| Homo sapiens |
Cytochrome P450 2B6 |
Emax |
16.9 |
None |
10.1124/dmd.112.047118 |
| Homo sapiens |
Cytochrome P450 2B6 |
FC |
3.6 |
None |
10.1128/aac.00660-09 |
| Homo sapiens |
Cytochrome P450 2B6 |
FC |
13.9 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Cytochrome P450 2C19 |
Activity |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2C19 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C8 |
Activity |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
Activity |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
FC |
1.0 |
None |
10.1016/j.bmcl.2016.06.088 |
| Homo sapiens |
Cytochrome P450 2C9 |
FC |
2.96 |
None |
10.1124/dmd.112.047928 |
| Homo sapiens |
Cytochrome P450 2C9 |
FC |
3.6 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Cytochrome P450 2C9 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2C9 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
FC |
1.0 |
None |
10.1016/j.bmcl.2016.06.088 |
| Homo sapiens |
Cytochrome P450 2D6 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2D6 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2E1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2E1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A |
Activity |
98.0 |
% |
10.1021/acs.jmedchem.0c02245 |
| Homo sapiens |
Cytochrome P450 3A |
Activity |
99.7 |
% |
10.1021/acs.jmedchem.0c02245 |
| Homo sapiens |
Cytochrome P450 3A4 |
Activity |
6.0 |
% |
10.1021/jm300601d |
| Homo sapiens |
Cytochrome P450 3A4 |
Activity |
20.0 |
% |
10.1016/j.bmcl.2022.128843 |
| Homo sapiens |
Cytochrome P450 3A4 |
Activity |
46.0 |
% |
10.1021/acs.jmedchem.0c02245 |
| Homo sapiens |
Cytochrome P450 3A4 |
Activity |
86.0 |
% |
10.1021/acs.jmedchem.0c02245 |
| Homo sapiens |
Cytochrome P450 3A4 |
Activity |
92.0 |
% |
10.1021/acs.jmedchem.0c02245 |
| Homo sapiens |
Cytochrome P450 3A4 |
Activity |
100.0 |
% |
10.1021/jm801073z |
| Homo sapiens |
Cytochrome P450 3A4 |
Activity |
nan |
None |
10.1021/acs.jmedchem.5b01078 |
| Homo sapiens |
Cytochrome P450 3A4 |
Activity |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
Emax |
5.0 |
% |
10.1021/acs.jmedchem.1c01887 |
| Homo sapiens |
Cytochrome P450 3A4 |
FC |
1.0 |
None |
10.1016/j.bmcl.2016.06.088 |
| Homo sapiens |
Cytochrome P450 3A4 |
FC |
6.63 |
None |
10.1128/aac.00660-09 |
| Homo sapiens |
Cytochrome P450 3A4 |
FC |
12.5 |
None |
10.1124/dmd.112.047928 |
| Homo sapiens |
Cytochrome P450 3A4 |
FC |
24.4 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Cytochrome P450 3A4 |
FC |
30.0 |
None |
10.1124/dmd.110.035840 |
| Homo sapiens |
Cytochrome P450 3A4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 3A4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
Ratio |
4.3 |
None |
10.1016/j.bmcl.2014.10.032 |
| Homo sapiens |
Cytochrome P450 3A5 |
Activity |
nan |
None |
10.1021/acs.jmedchem.5b01078 |
| Homo sapiens |
Cytochrome P450 51 |
IC50 |
30000.0 |
nM |
10.1124/dmd.106.013888 |
| Homo sapiens |
Delta opioid receptor |
AC50 |
17000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Delta opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Delta opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
DLD-1 |
Activity |
nan |
None |
10.1128/aac.00961-08 |
| Homo sapiens |
DNA polymerase iota |
Potency |
89125.1 |
nM |
None |
| Homo sapiens |
Dopamine D1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D2 receptor |
AC50 |
9200.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D3 receptor |
AC50 |
10999.9 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D3 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D3 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D4 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D4 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D4 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine transporter |
AC50 |
20000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Endothelin receptor ET-A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-A |
Ki |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-B |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Equilibrative nucleoside transporter 1 |
AC50 |
12445.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor beta |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor beta |
IC50 |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor beta |
Ki |
nan |
None |
None |
| Homo sapiens |
Galactocerebrosidase |
Potency |
631.0 |
nM |
None |
| Homo sapiens |
Gastric inhibitory polypeptide receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Geminin |
Potency |
29092.9 |
nM |
None |
| Homo sapiens |
Ghrelin receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucagon receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Glucocorticoid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Glutathione transferase omega 1 |
IC50 |
75000.0 |
nM |
10.1021/acs.jmedchem.8b00318 |
| Homo sapiens |
Guanine nucleotide-binding protein G(s), subunit alpha |
Potency |
39810.7 |
nM |
None |
| Homo sapiens |
HaCaT |
Survival |
55.0 |
% |
10.1021/acs.jnatprod.5b01033 |
| Homo sapiens |
HCT-116 |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.01.004 |
| Homo sapiens |
HCT-116 |
GI50 |
121510000.0 |
nM |
10.1039/C6MD00278A |
| Homo sapiens |
HCT-116 |
GI90 |
100.0 |
ug ml-1 |
10.1016/j.bmcl.2017.01.004 |
| Homo sapiens |
HEK293 |
CC50 |
100000.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| Homo sapiens |
HEK293 |
IC50 |
nan |
None |
10.1016/j.bmcl.2012.12.096 |
| Homo sapiens |
HEK293 |
Inhibition |
nan |
% |
10.1016/j.ejmech.2018.07.047 |
| Homo sapiens |
HEK293 |
LC50 |
200.0 |
ug.mL-1 |
10.1016/j.bmc.2008.10.042 |
| Homo sapiens |
HEK293 |
LC50 |
100000.0 |
nM |
10.1021/jm400240r |
| Homo sapiens |
HEK-293T |
Activity |
nan |
None |
10.1016/j.bmcl.2012.10.060 |
| Homo sapiens |
HeLa |
Activity |
100.4 |
% |
10.1021/acs.jmedchem.5b00608 |
| Homo sapiens |
HeLa |
Activity |
101.7 |
% |
10.1021/acs.jmedchem.5b00608 |
| Homo sapiens |
HeLa |
CC50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.093 |
| Homo sapiens |
HeLa |
CD50 |
190.0 |
uM |
10.1016/j.bmcl.2008.03.025 |
| Homo sapiens |
HeLa |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.045 |
| Homo sapiens |
HeLa |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.03.020 |
| Homo sapiens |
HeLa |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.03.065 |
| Homo sapiens |
HeLa |
GI90 |
100.0 |
ug ml-1 |
10.1016/j.bmcl.2019.03.020 |
| Homo sapiens |
HeLa |
GI90 |
100.0 |
ug ml-1 |
10.1016/j.ejmech.2017.03.065 |
| Homo sapiens |
HeLa |
IC20 |
180.0 |
ug ml-1 |
10.1128/aac.00729-05 |
| Homo sapiens |
HeLa |
IC20 |
nan |
None |
10.1128/aac.00729-05 |
| Homo sapiens |
HeLa |
IC50 |
270.0 |
ug.mL-1 |
10.1128/aac.00729-05 |
| Homo sapiens |
HeLa |
IC50 |
20000.0 |
nM |
10.1021/acs.jmedchem.5b00608 |
| Homo sapiens |
HeLa |
IC50 |
nan |
None |
10.1128/aac.00729-05 |
| Homo sapiens |
Hepatocyte |
Activity |
50.0 |
uM |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
Activity |
100.0 |
% |
10.1021/jm801073z |
| Homo sapiens |
Hepatocyte |
Activity |
123.2 |
% |
10.1021/acs.jmedchem.5b00608 |
| Homo sapiens |
Hepatocyte |
Activity |
nan |
None |
10.1016/j.bmcl.2014.10.032 |
| Homo sapiens |
Hepatocyte |
Activity |
nan |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
EC50 |
980.0 |
nM |
10.1124/dmd.112.047118 |
| Homo sapiens |
Hepatocyte |
Emax |
16.9 |
None |
10.1124/dmd.112.047118 |
| Homo sapiens |
Hepatocyte |
FC |
0.7 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
0.8 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
1.0 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
1.1 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
1.2 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
1.3 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
1.4 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
2.3 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
2.5 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
2.6 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
4.3 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
8.4 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
20.2 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
FC |
60.0 |
None |
10.1124/dmd.110.035840 |
| Homo sapiens |
Hepatocyte |
FC |
74.8 |
None |
10.1124/dmd.112.045765 |
| Homo sapiens |
Hepatocyte |
IC50 |
20000.0 |
nM |
10.1021/acs.jmedchem.5b00608 |
| Homo sapiens |
HepG2 |
Activity |
114.66 |
% |
10.1007/s00044-010-9405-3 |
| Homo sapiens |
HepG2 |
Activity |
116.03 |
% |
10.1007/s00044-010-9405-3 |
| Homo sapiens |
HepG2 |
Activity |
192.41 |
% |
10.1007/s00044-010-9405-3 |
| Homo sapiens |
HepG2 |
Activity |
nan |
None |
10.1016/j.bmc.2014.11.043 |
| Homo sapiens |
HepG2 |
CC50 |
175.9 |
ug.mL-1 |
10.1016/j.ejmech.2021.113472 |
| Homo sapiens |
HepG2 |
IC50 |
145330.0 |
nM |
10.1016/j.bmcl.2020.127146 |
| Homo sapiens |
HERG |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
HERG |
IC50 |
nan |
None |
None |
| Homo sapiens |
HERG |
Inhibition |
nan |
% |
10.1016/j.bmc.2019.01.022 |
| Homo sapiens |
HERG |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H1 receptor |
AC50 |
8700.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Histamine H1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H2 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Histamine H2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H3 receptor |
AC50 |
25000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
HMG-CoA reductase |
IC50 |
nan |
None |
None |
| Homo sapiens |
HMG-CoA reductase |
Ki |
nan |
None |
None |
| Homo sapiens |
Homo sapiens |
Activity |
5.8 |
% |
10.1128/aac.00247-07 |
| Homo sapiens |
Homo sapiens |
Activity |
99.0 |
% |
10.1128/aac.00579-07 |
| Homo sapiens |
Homo sapiens |
Activity |
nan |
None |
10.1002/hep.27206 |
| Homo sapiens |
Homo sapiens |
Activity |
nan |
None |
10.1128/aac.00247-07 |
| Homo sapiens |
Homo sapiens |
AUC |
13.1 |
ug ml-1 |
10.1128/aac.01474-06 |
| Homo sapiens |
Homo sapiens |
AUC |
24.5 |
ug ml-1 |
10.1128/aac.01474-06 |
| Homo sapiens |
Homo sapiens |
AUC |
100.0 |
ug ml-1 |
10.1128/aac.01474-06 |
| Homo sapiens |
Homo sapiens |
AUC |
171.0 |
ug ml-1 |
10.1128/aac.01474-06 |
| Homo sapiens |
Homo sapiens |
AUC |
6400.0 |
ng.hr.mL-1 |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
AUC |
13200.0 |
ng.hr.mL-1 |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
AUC |
19600.0 |
ng.hr.mL-1 |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
AUC |
21500.0 |
ng.hr.mL-1 |
10.1128/aac.00749-08 |
| Homo sapiens |
Homo sapiens |
AUC |
23100.0 |
ng.hr.mL-1 |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
AUC |
28200.0 |
ng.hr.mL-1 |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
AUC |
29700.0 |
ng.hr.mL-1 |
10.1371/journal.pmed.0030466 |
| Homo sapiens |
Homo sapiens |
AUC |
30100.0 |
ng.hr.mL-1 |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
AUC |
30700.0 |
ng.hr.mL-1 |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
AUC |
41700.0 |
ng.hr.mL-1 |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
AUC |
44000.0 |
ng.hr.mL-1 |
10.1128/aac.01621-06 |
| Homo sapiens |
Homo sapiens |
AUC |
44600.0 |
ng.hr.mL-1 |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
AUC |
45700.0 |
ng.hr.mL-1 |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
AUC |
48500.0 |
ng.hr.mL-1 |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
AUC |
48500.0 |
ng.hr.mL-1 |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
AUC |
49000.0 |
ng.hr.mL-1 |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
AUC |
50600.0 |
ng.hr.mL-1 |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
AUC |
60300.0 |
ng.hr.mL-1 |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
AUC |
73604.65 |
ng.hr.mL-1 |
10.1093/toxsci/kft176 |
| Homo sapiens |
Homo sapiens |
AUC |
79700.0 |
ng.hr.mL-1 |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
AUC |
79700.0 |
ng.hr.mL-1 |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
AUC |
112000.0 |
ng.hr.mL-1 |
10.1128/aac.01533-06 |
| Homo sapiens |
Homo sapiens |
CL |
1.3 |
mL.min-1.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
CL |
1.5 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
CL |
1.5 |
mL.min-1.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
CL |
8.9 |
L/hr |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
CL/F |
7.5 |
L/hr |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
CL/F |
9.2 |
L/hr |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
CL/F |
9.2 |
L/hr |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
CL/F |
15.1 |
L/hr |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
CL/F |
16.5 |
L/hr |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
CL/F |
19.2 |
L/hr |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
CL/F |
19.4 |
L/hr |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
CL/F |
20.2 |
L/hr |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
CL_renal |
0.2 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
CL_renal |
0.2 |
mL.min-1.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Cmax |
1458.17 |
nM |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Cmax |
2673.31 |
nM |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Cmax |
3074.31 |
nM |
10.1128/aac.01474-06 |
| Homo sapiens |
Homo sapiens |
Cmax |
3876.3 |
nM |
10.1128/aac.01474-06 |
| Homo sapiens |
Homo sapiens |
Cmax |
4252.99 |
nM |
None |
| Homo sapiens |
Homo sapiens |
Cmax |
6683.27 |
nM |
10.1371/journal.pmed.0030466 |
| Homo sapiens |
Homo sapiens |
Cmax |
8000.0 |
nM |
10.1128/aac.00527-07 |
| Homo sapiens |
Homo sapiens |
Cmax |
8500.0 |
nM |
10.1002/hep.27206 |
| Homo sapiens |
Homo sapiens |
Cmax |
8505.98 |
nM |
None |
| Homo sapiens |
Homo sapiens |
Cmax |
9721.13 |
nM |
10.1128/aac.00749-08 |
| Homo sapiens |
Homo sapiens |
Cmax |
11531.68 |
nM |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
Cmax |
11665.35 |
nM |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
Cmax |
12151.41 |
nM |
10.1128/aac.01605-07 |
| Homo sapiens |
Homo sapiens |
Cmax |
12285.07 |
nM |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
Cmax |
12758.98 |
nM |
10.1128/aac.00375-07 |
| Homo sapiens |
Homo sapiens |
Cmax |
12758.98 |
nM |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
Cmax |
12758.98 |
nM |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Cmax |
13002.0 |
nM |
None |
| Homo sapiens |
Homo sapiens |
Cmax |
13974.12 |
nM |
None |
| Homo sapiens |
Homo sapiens |
Cmax |
15796.83 |
nM |
10.1128/aac.01474-06 |
| Homo sapiens |
Homo sapiens |
Cmax |
17011.97 |
nM |
10.1128/aac.01474-06 |
| Homo sapiens |
Homo sapiens |
Cmax |
18956.19 |
nM |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Cmin |
329.0 |
ng/ml |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
Cmin |
360.0 |
ng/ml |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
Cp |
9.9 |
ug ml-1 |
10.1128/aac.01621-06 |
| Homo sapiens |
Homo sapiens |
Css |
3.726 |
uM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Homo sapiens |
DILI_Concern |
nan |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
DILI_severity_class |
8.0 |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
F |
50.0 |
% |
10.1021/jm400887j |
| Homo sapiens |
Homo sapiens |
F |
68.0 |
% |
10.1128/aac.00749-08 |
| Homo sapiens |
Homo sapiens |
F |
69.0 |
% |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
F |
74.0 |
% |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
F |
88.8 |
% |
10.1016/j.bmc.2007.08.060 |
| Homo sapiens |
Homo sapiens |
Fa |
1.0 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
fAUC |
16000.0 |
ng.hr.mL-1 |
10.1128/aac.01533-06 |
| Homo sapiens |
Homo sapiens |
fAUC |
112000.0 |
ng.hr.mL-1 |
10.1128/aac.01533-06 |
| Homo sapiens |
Homo sapiens |
FC |
45.0 |
None |
10.1128/aac.00579-07 |
| Homo sapiens |
Homo sapiens |
FC |
178.0 |
None |
10.1128/aac.00579-07 |
| Homo sapiens |
Homo sapiens |
FC |
422.0 |
None |
10.1128/aac.00579-07 |
| Homo sapiens |
Homo sapiens |
fCmax |
2.0 |
mg/L |
10.1128/aac.01533-06 |
| Homo sapiens |
Homo sapiens |
fCmax |
2.0 |
ug ml-1 |
10.1128/aac.00766-08 |
| Homo sapiens |
Homo sapiens |
fCmax |
7.0 |
mg/L |
10.1128/aac.01533-06 |
| Homo sapiens |
Homo sapiens |
fCmax |
14.0 |
mg/L |
10.1128/aac.01533-06 |
| Homo sapiens |
Homo sapiens |
F_fraction |
0.93 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Fg |
0.99 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Fh |
0.94 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Ka |
1.15 |
L/hr |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
Ka |
1.23 |
L/hr |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
Ka |
1.61 |
L/hr |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
Ka |
1.64 |
L/hr |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
MTT |
0.424 |
hr |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
Ratio |
0.82 |
None |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Ratio |
0.92 |
None |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Ratio |
0.94 |
None |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
Ratio |
0.97 |
None |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
Ratio |
0.98 |
None |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
Ratio |
1.04 |
None |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
Ratio |
1.09 |
None |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
Ratio |
1.13 |
None |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Ratio |
70.8 |
None |
10.1128/aac.00749-08 |
| Homo sapiens |
Homo sapiens |
Ratio AUC |
1.49 |
None |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Ratio AUC |
1.65 |
None |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.4 |
hr |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.6 |
hr |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.9 |
hr |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.9 |
hr |
10.1128/aac.01621-06 |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.0 |
hr |
10.1128/aac.00749-08 |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.0 |
hr |
None |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.1 |
hr |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.2 |
hr |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.2 |
hr |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.5 |
hr |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.9 |
hr |
None |
| Homo sapiens |
Homo sapiens |
T1/2 |
3.0 |
hr |
10.1128/aac.01533-06 |
| Homo sapiens |
Homo sapiens |
T1/2 |
3.0 |
hr |
10.1128/aac.01605-07 |
| Homo sapiens |
Homo sapiens |
T1/2 |
3.2 |
hr |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
T1/2 |
3.35 |
hr |
None |
| Homo sapiens |
Homo sapiens |
T1/2 |
3.5 |
hr |
10.1128/aac.00527-07 |
| Homo sapiens |
Homo sapiens |
T1/2 |
3.6 |
hr |
None |
| Homo sapiens |
Homo sapiens |
T1/2 |
5.0 |
hr |
None |
| Homo sapiens |
Homo sapiens |
T1/2 |
5.08 |
hr |
None |
| Homo sapiens |
Homo sapiens |
T1/2 |
7.3 |
hr |
None |
| Homo sapiens |
Homo sapiens |
T1/2 |
11.0 |
hr |
None |
| Homo sapiens |
Homo sapiens |
TIME |
3.611e-06 |
hr |
10.1128/aac.01204-07 |
| Homo sapiens |
Homo sapiens |
Tmax |
1.0 |
hr |
10.1128/aac.00527-07 |
| Homo sapiens |
Homo sapiens |
Tmax |
1.0 |
hr |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Tmax |
1.0 |
hr |
None |
| Homo sapiens |
Homo sapiens |
Tmax |
1.5 |
hr |
10.1128/aac.00749-08 |
| Homo sapiens |
Homo sapiens |
Tmax |
2.0 |
hr |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
Tmax |
2.0 |
hr |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Tmax |
2.5 |
hr |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
Tmax |
2.5 |
hr |
10.1128/aac.01474-06 |
| Homo sapiens |
Homo sapiens |
Tmax |
2.7 |
hr |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
Tmax |
3.12 |
hr |
10.1128/aac.01474-06 |
| Homo sapiens |
Homo sapiens |
Tmax |
3.27 |
hr |
10.1128/aac.01474-06 |
| Homo sapiens |
Homo sapiens |
Tmax |
3.67 |
hr |
10.1128/aac.01474-06 |
| Homo sapiens |
Homo sapiens |
Tmax |
4.0 |
hr |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Vbeta |
32.0 |
l |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
Vbeta |
33.0 |
l |
10.1128/aac.00341-07 |
| Homo sapiens |
Homo sapiens |
Vc/F |
23.3 |
l |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Vc/F |
25.3 |
l |
10.1128/aac.01550-06 |
| Homo sapiens |
Homo sapiens |
Vc/F |
27.4 |
l |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
Vc/F |
27.6 |
l |
10.1128/aac.00447-09 |
| Homo sapiens |
Homo sapiens |
Vd |
8.05 |
l |
10.1128/aac.01520-08 |
| Homo sapiens |
Homo sapiens |
Vd |
10.16 |
l |
10.1128/aac.01520-08 |
| Homo sapiens |
Homo sapiens |
Vd |
11.56 |
l |
10.1128/aac.01520-08 |
| Homo sapiens |
Homo sapiens |
Vdss |
0.97 |
L.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Vz |
51.5 |
l |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
Vz |
52.8 |
l |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
Vz |
53.2 |
l |
10.1128/aac.00461-07 |
| Homo sapiens |
Homo sapiens |
Vz |
53.4 |
l |
10.1128/aac.00461-07 |
| Homo sapiens |
HSP60/HSP10 |
IC50 |
100000.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| Homo sapiens |
HT-29 |
Activity |
nan |
None |
10.1128/aac.00961-08 |
| Homo sapiens |
Interleukin-8 receptor A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor A |
Ki |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor B |
IC50 |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor B |
Ki |
nan |
None |
None |
| Homo sapiens |
Jurkat |
CD50 |
nan |
None |
10.1016/j.bmc.2013.07.003 |
| Homo sapiens |
Kappa opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Kappa opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Kappa opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Leukocyte common antigen |
IC50 |
nan |
None |
None |
| Homo sapiens |
Leukocyte common antigen |
Ki |
nan |
None |
None |
| Homo sapiens |
Leukocyte elastase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Leukocyte elastase |
Ki |
nan |
None |
None |
| Homo sapiens |
Liver microsome |
CL |
0.7 |
mL.min-1.g-1 |
10.1124/dmd.111.043067 |
| Homo sapiens |
Liver microsome |
Stability |
nan |
% |
10.1021/acs.jmedchem.5b01542 |
| Homo sapiens |
Liver microsomes |
Activity |
nan |
None |
10.1021/tx300075j |
| Homo sapiens |
Liver microsomes |
Stability |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
LS180 |
Activity |
nan |
None |
10.1039/C6MD00300A |
| Homo sapiens |
LXR-alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
LXR-beta |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
MAP kinase ERK1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK1 |
Ki |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK2 |
Ki |
nan |
None |
None |
| Homo sapiens |
MAP kinase p38 alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase p38 alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase 9 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase 9 |
Ki |
nan |
None |
None |
| Homo sapiens |
MCF7 |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.01.004 |
| Homo sapiens |
MCF7 |
GI50 |
100.0 |
ug.mL-1 |
10.1039/C5MD00404G |
| Homo sapiens |
MCF7 |
GI50 |
121510000.0 |
nM |
10.1039/C6MD00278A |
| Homo sapiens |
MCF7 |
GI90 |
100.0 |
ug ml-1 |
10.1016/j.bmcl.2017.01.004 |
| Homo sapiens |
Melanocortin receptor 3 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Melanocortin receptor 3 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 3 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 4 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Melanocortin receptor 4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 5 |
Ki |
nan |
None |
None |
| Homo sapiens |
MG-63 |
IC20 |
120.0 |
ug ml-1 |
10.1128/aac.00729-05 |
| Homo sapiens |
MG-63 |
IC20 |
nan |
None |
10.1128/aac.00729-05 |
| Homo sapiens |
MG-63 |
IC50 |
240.0 |
ug.mL-1 |
10.1128/aac.00729-05 |
| Homo sapiens |
MG-63 |
IC50 |
nan |
None |
10.1128/aac.00729-05 |
| Homo sapiens |
Monoamine oxidase A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Monoamine oxidase A |
Activity |
nan |
None |
10.1021/jm800656v |
| Homo sapiens |
Monoamine oxidase A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Monoamine oxidase A |
Ki |
nan |
None |
None |
| Homo sapiens |
Motilin receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
MRC5 |
Activity |
65.0 |
ug ml-1 |
10.1016/j.bmcl.2009.09.095 |
| Homo sapiens |
MRC5 |
CC50 |
nan |
None |
10.1016/j.ejmech.2017.06.061 |
| Homo sapiens |
MRC5 |
IC50 |
100000.0 |
nM |
10.1021/acs.jnatprod.5b00266 |
| Homo sapiens |
MRC5 |
IC50 |
nan |
None |
10.1016/j.bmcl.2019.02.019 |
| Homo sapiens |
MRC5 |
IC50 |
nan |
None |
10.1016/j.ejmech.2022.114831 |
| Homo sapiens |
MRC5 |
IC50 |
nan |
None |
10.1021/acs.jmedchem.7b01332 |
| Homo sapiens |
MRC5 |
IC90 |
100000.0 |
nM |
10.1021/acs.jnatprod.5b00266 |
| Homo sapiens |
MRC5 |
Survival |
53.0 |
% |
10.1021/acs.jnatprod.5b01033 |
| Homo sapiens |
Multidrug resistance-associated protein 1 |
Activity |
110.0 |
% |
10.1016/s0304-3835(99)00024-5 |
| Homo sapiens |
Multidrug resistance-associated protein 4 |
IC50 |
41900.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Multidrug resistance-associated protein 5 |
Activity |
nan |
None |
10.1016/s0378-4274(01)00306-x |
| Homo sapiens |
Mu opioid receptor |
AC50 |
8000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Mu opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Mu opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Mu opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
AC50 |
7100.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurokinin 1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neurokinin 1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurokinin 2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neurokinin 2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Neuronal acetylcholine receptor protein alpha-4 subunit |
AC50 |
21999.9 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
AC50 |
22539.8 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
AC50 |
21579.9 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurotensin receptor 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Nitric oxide synthase, inducible |
Activity |
nan |
None |
10.1128/aac.00961-08 |
| Homo sapiens |
Norepinephrine transporter |
AC50 |
20000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Norepinephrine transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Norepinephrine transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Nuclear factor erythroid 2-related factor 2 |
Potency |
4109.5 |
nM |
None |
| Homo sapiens |
Nuclear factor erythroid 2-related factor 2 |
Potency |
4610.9 |
nM |
None |
| Homo sapiens |
Nuclear receptor subfamily 1 group I member 3 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Nuclear receptor subfamily 1 group I member 3 |
Activity |
nan |
None |
10.1016/j.ejmech.2019.06.031 |
| Homo sapiens |
PANC-1 |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.03.020 |
| Homo sapiens |
PANC-1 |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.03.065 |
| Homo sapiens |
PANC-1 |
GI90 |
100.0 |
ug ml-1 |
10.1016/j.bmcl.2019.03.020 |
| Homo sapiens |
PANC-1 |
GI90 |
100.0 |
ug ml-1 |
10.1016/j.ejmech.2017.03.065 |
| Homo sapiens |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
Potency |
50118.7 |
nM |
None |
| Homo sapiens |
Peroxisome proliferator-activated receptor alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
nan |
None |
10.1016/0006-2952(95)00045-2 |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
nan |
None |
10.1023/b:pham.0000026434.82855.69 |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
nan |
None |
10.1074/jbc.m010173200 |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
nan |
None |
10.1172/jci6663 |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
nan |
None |
None |
| Homo sapiens |
Phosphodiesterase 3A |
AC50 |
18330.3 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 4D |
AC50 |
12999.9 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 5A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Phosphodiesterase 5A |
Ki |
nan |
None |
None |
| Homo sapiens |
Plasma |
Cmax |
21872.53 |
nM |
10.1128/aac.01145-08 |
| Homo sapiens |
Plasma |
Drug uptake |
0.001 |
ug ml-1 |
10.1126/science.1106753 |
| Homo sapiens |
Plasma |
fCmax |
2.43 |
uM |
10.1124/dmd.111.040758 |
| Homo sapiens |
Plasma |
Fu |
0.15 |
None |
10.1128/aac.01145-08 |
| Homo sapiens |
Plasma |
Fu |
0.165 |
None |
10.1021/acs.jmedchem.5b00050 |
| Homo sapiens |
Plasma |
K(p,uu,CSF) |
2.2 |
None |
10.1021/jm901036q |
| Homo sapiens |
Plasma |
PPB |
85.0 |
% |
10.1128/aac.00749-08 |
| Homo sapiens |
Platelet activating factor receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Platelet activating factor receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Pregnane X receptor |
AC50 |
19899.6 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Pregnane X receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Pregnane X receptor |
Activity |
70.0 |
% |
10.1021/acs.jmedchem.9b01032 |
| Homo sapiens |
Pregnane X receptor |
Activity |
77.3 |
% |
10.1039/C6MD00300A |
| Homo sapiens |
Pregnane X receptor |
Activity |
100.0 |
% |
10.1021/acs.jmedchem.0c02201 |
| Homo sapiens |
Pregnane X receptor |
Activity |
100.0 |
% |
10.1021/acs.jmedchem.2c01640 |
| Homo sapiens |
Pregnane X receptor |
Activity |
107.0 |
% |
10.1016/j.bmcl.2008.06.018 |
| Homo sapiens |
Pregnane X receptor |
Activity |
114.0 |
% |
10.1021/acs.jmedchem.0c02245 |
| Homo sapiens |
Pregnane X receptor |
Activity |
nan |
None |
10.1016/j.bmc.2014.11.043 |
| Homo sapiens |
Pregnane X receptor |
Activity |
nan |
None |
10.1021/acs.jmedchem.6b00415 |
| Homo sapiens |
Pregnane X receptor |
Activity |
nan |
None |
10.1021/acsmedchemlett.1c00277 |
| Homo sapiens |
Pregnane X receptor |
Activity |
nan |
None |
10.1021/acsmedchemlett.9b00079 |
| Homo sapiens |
Pregnane X receptor |
Activity |
nan |
None |
10.1021/jm200025f |
| Homo sapiens |
Pregnane X receptor |
Activity |
nan |
None |
None |
| Homo sapiens |
Pregnane X receptor |
EC50 |
190.0 |
nM |
10.1021/acs.jmedchem.5b01891 |
| Homo sapiens |
Pregnane X receptor |
EC50 |
200.0 |
nM |
10.1124/dmd.110.035105 |
| Homo sapiens |
Pregnane X receptor |
EC50 |
226.0 |
nM |
10.1039/C6MD00300A |
| Homo sapiens |
Pregnane X receptor |
EC50 |
1100.0 |
nM |
10.1016/j.bmcl.2016.02.031 |
| Homo sapiens |
Pregnane X receptor |
EC50 |
1170.0 |
nM |
10.1021/acs.jmedchem.2c01640 |
| Homo sapiens |
Pregnane X receptor |
EC50 |
1190.0 |
nM |
10.1021/acs.jmedchem.0c02245 |
| Homo sapiens |
Pregnane X receptor |
EC50 |
1400.0 |
nM |
10.1021/acs.jmedchem.0c02201 |
| Homo sapiens |
Pregnane X receptor |
EC50 |
2000.0 |
nM |
10.1016/j.bmc.2018.07.038 |
| Homo sapiens |
Pregnane X receptor |
EC50 |
2300.0 |
nM |
10.1021/jm201716n |
| Homo sapiens |
Pregnane X receptor |
EC50 |
3200.0 |
nM |
10.1124/dmd.110.035105 |
| Homo sapiens |
Pregnane X receptor |
EC50 |
3500.0 |
nM |
10.1124/dmd.110.035105 |
| Homo sapiens |
Pregnane X receptor |
EC50 |
5600.0 |
nM |
10.1016/j.bmcl.2011.08.054 |
| Homo sapiens |
Pregnane X receptor |
Efficacy |
43.9 |
% |
10.1124/dmd.110.035105 |
| Homo sapiens |
Pregnane X receptor |
Efficacy |
75.0 |
% |
10.1016/j.bmcl.2016.02.031 |
| Homo sapiens |
Pregnane X receptor |
FC |
2.9 |
None |
10.1021/acsmedchemlett.1c00277 |
| Homo sapiens |
Pregnane X receptor |
FC |
9.5 |
None |
10.1016/j.bmcl.2011.08.054 |
| Homo sapiens |
Pregnane X receptor |
FC |
11.0 |
None |
10.1124/dmd.111.042879 |
| Homo sapiens |
Pregnane X receptor |
FC |
12.0 |
None |
10.1124/dmd.111.042879 |
| Homo sapiens |
Pregnane X receptor |
FC |
12.6 |
None |
10.1021/jm201716n |
| Homo sapiens |
Pregnane X receptor |
FC |
38.0 |
None |
10.1124/dmd.111.042879 |
| Homo sapiens |
Pregnane X receptor |
FC |
43.0 |
None |
10.1124/dmd.111.042879 |
| Homo sapiens |
Pregnane X receptor |
FC |
50.0 |
None |
10.1124/dmd.111.042879 |
| Homo sapiens |
Pregnane X receptor |
FC |
53.0 |
None |
10.1124/dmd.111.042879 |
| Homo sapiens |
Pregnane X receptor |
IC50 |
nan |
None |
10.1021/acs.jmedchem.0c02201 |
| Homo sapiens |
Pregnane X receptor |
Imax |
117.0 |
% |
10.1021/acs.jmedchem.5b01891 |
| Homo sapiens |
Pregnane X receptor |
Inhibition |
18.0 |
% |
10.1016/j.bmcl.2008.06.018 |
| Homo sapiens |
Pregnane X receptor |
Inhibition |
nan |
% |
10.1021/acs.jmedchem.2c01640 |
| Homo sapiens |
Progesterone receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Protein kinase C alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
Protein kinase C alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Retinoic acid receptor alpha |
AC50 |
3000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Retinoic acid receptor alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Retinoic acid receptor beta |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Retinoic acid receptor beta |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Retinoic acid receptor gamma |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 1a (5-HT1a) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 1a (5-HT1a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
AC50 |
12000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 3a (5-HT3a) receptor |
AC50 |
5200.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 7 (5-HT7) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
AC50 |
15000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Serum |
Activity |
80.0 |
% |
10.1128/aac.01605-07 |
| Homo sapiens |
Serum |
Cmax |
2430.28 |
nM |
10.1128/aac.00922-07 |
| Homo sapiens |
Serum |
Cmax |
18227.11 |
nM |
10.1128/aac.00961-08 |
| Homo sapiens |
Serum |
Drug uptake |
5.3 |
mg/L |
10.1128/aac.01081-09 |
| Homo sapiens |
Serum |
Drug uptake |
8.9 |
mg/L |
10.1128/aac.01081-09 |
| Homo sapiens |
Serum |
T1/2 |
2.0 |
hr |
10.1128/aac.00922-07 |
| Homo sapiens |
Serum |
Tmax |
1.2 |
hr |
10.1128/aac.00922-07 |
| Homo sapiens |
Serum albumin |
Binding |
73.3 |
% |
10.1021/jm991174y |
| Homo sapiens |
Serum albumin |
Kd |
12000.0 |
nM |
10.1128/aac.00971-08 |
| Homo sapiens |
Serum albumin |
Ratio |
0.5 |
None |
10.1128/aac.00971-08 |
| Homo sapiens |
Serum albumin |
Ratio |
1.0 |
None |
10.1128/aac.00971-08 |
| Homo sapiens |
Serum albumin |
Ratio |
1.5 |
None |
10.1128/aac.00971-08 |
| Homo sapiens |
Sigma opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Sigma opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Solute carrier family 22 member 1 |
Inhibition |
26.2 |
% |
10.1021/jm8003152 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1A2 |
Activity |
nan |
None |
10.1038/nrd3028 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1A2 |
Activity |
nan |
None |
10.1053/jhep.2002.34133 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1A2 |
Ki |
51000.0 |
nM |
10.1053/jhep.2002.34133 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Activity |
nan |
None |
10.1038/nrd3028 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Activity |
nan |
None |
10.1074/jbc.m004968200 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Activity |
nan |
None |
10.1124/jpet.102.043026 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
IC50 |
300.0 |
nM |
10.1124/dmd.111.042382 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
IC50 |
1200.0 |
nM |
10.1021/jm300212s |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
IC50 |
2200.0 |
nM |
10.1124/dmd.111.042382 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
IC50 |
2300.0 |
nM |
10.1124/dmd.111.042382 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Inhibition |
33.63 |
% |
10.1124/mol.112.084152 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Inhibition |
88.3 |
% |
10.1021/jm300212s |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Inhibition |
98.4 |
% |
10.1124/dmd.112.048470 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Ki |
1100.0 |
nM |
10.1021/jm300212s |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Ki |
17000.0 |
nM |
10.1053/jhep.2002.34133 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Km |
1500.0 |
nM |
10.1124/jpet.102.043026 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Km |
13000.0 |
nM |
10.1053/jhep.2002.34133 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
Activity |
nan |
None |
10.1038/nrd3028 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
Activity |
nan |
None |
10.1074/jbc.m004968200 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
IC50 |
1500.0 |
nM |
10.1021/jm300212s |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
Inhibition |
22.01 |
% |
10.1124/mol.112.084152 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
Inhibition |
97.4 |
% |
10.1124/dmd.112.048470 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
Inhibition |
101.7 |
% |
10.1021/jm300212s |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
Ki |
1400.0 |
nM |
10.1021/jm300212s |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
Ki |
5000.0 |
nM |
10.1053/jhep.2002.34133 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
Km |
2300.0 |
nM |
10.1053/jhep.2002.34133 |
| Homo sapiens |
Solute carrier organic anion transporter family member 2B1 |
Activity |
nan |
None |
10.1038/nrd3028 |
| Homo sapiens |
Solute carrier organic anion transporter family member 2B1 |
Activity |
nan |
None |
10.1053/jhep.2002.34133 |
| Homo sapiens |
Solute carrier organic anion transporter family member 2B1 |
IC50 |
65000.0 |
nM |
10.1021/jm300212s |
| Homo sapiens |
Solute carrier organic anion transporter family member 2B1 |
Inhibition |
21.2 |
% |
10.1021/jm300212s |
| Homo sapiens |
Solute carrier organic anion transporter family member 2B1 |
Ki |
63000.0 |
nM |
10.1021/jm300212s |
| Homo sapiens |
TAR DNA-binding protein 43 |
Potency |
501.2 |
nM |
None |
| Homo sapiens |
Thiosulfate sulfurtransferase |
IC50 |
100000.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| Homo sapiens |
THP-1 |
Activity |
65.0 |
ug ml-1 |
10.1016/j.bmcl.2009.09.095 |
| Homo sapiens |
THP-1 |
GI50 |
0.14 |
ug.mL-1 |
10.1016/j.ejmech.2017.01.009 |
| Homo sapiens |
THP-1 |
IC50 |
100000.0 |
nM |
10.1021/acs.jnatprod.5b00266 |
| Homo sapiens |
THP-1 |
IC90 |
100000.0 |
nM |
10.1021/acs.jnatprod.5b00266 |
| Homo sapiens |
Thromboxane A2 receptor |
AC50 |
17364.6 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Thromboxane-A synthase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Thromboxane-A synthase |
Ki |
nan |
None |
None |
| Homo sapiens |
Type-1 angiotensin II receptor |
AC50 |
19395.9 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Tyrosine-protein kinase FYN |
IC50 |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase FYN |
Ki |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase LCK |
IC50 |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase LCK |
Ki |
nan |
None |
None |
| Homo sapiens |
Tyrosyl-DNA phosphodiesterase 1 |
Potency |
5173.5 |
nM |
None |
| Homo sapiens |
Tyrosyl-DNA phosphodiesterase 1 |
Potency |
18837.5 |
nM |
None |
| Homo sapiens |
Tyrosyl-DNA phosphodiesterase 1 |
Potency |
23715.0 |
nM |
None |
| Homo sapiens |
UDP-glucuronosyltransferase 1-1 |
Activity |
0.0 |
pm/min/mg |
10.1146/annurev.pharmtox.40.1.581 |
| Homo sapiens |
UDP-glucuronosyltransferase 1-6 |
Activity |
0.0 |
pm/min/mg |
10.1146/annurev.pharmtox.40.1.581 |
| Homo sapiens |
UDP-glucuronosyltransferase 1-9 |
Activity |
0.0 |
pm/min/mg |
10.1146/annurev.pharmtox.40.1.581 |
| Homo sapiens |
Vascular endothelial growth factor receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vascular endothelial growth factor receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasoactive intestinal polypeptide receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vasoactive intestinal polypeptide receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasopressin V1a receptor |
AC50 |
26699.9 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vasopressin V1a receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vasopressin V1a receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasopressin V2 receptor |
AC50 |
29999.9 |
nM |
10.1038/s41467-023-40064-9 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
Inhibition |
100.0 |
% |
10.1021/jm0703901 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
8000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MBC |
nan |
None |
10.1021/acs.jnatprod.2c00065 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
0.012 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00065 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
Ratio |
680.0 |
None |
10.1128/aac.00405-08 |
| Klebsiella oxytoca |
Klebsiella oxytoca |
Ratio |
700.0 |
None |
10.1128/aac.00405-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
EC50 |
11000.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
FICI |
0.125 |
None |
10.1128/aac.01439-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Inhibition |
10.0 |
% |
10.1128/aac.00471-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Inhibition |
nan |
% |
10.1128/aac.00471-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
IZ |
7.0 |
mm |
10.1016/j.bmc.2018.02.049 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
IZ |
27.0 |
mm |
10.1016/j.bmcl.2016.04.038 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
IZ |
45.0 |
mm |
10.1016/j.ejmech.2008.09.035 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
IZ |
nan |
None |
10.1016/j.bmc.2007.09.025 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
log10cfu |
8.5 |
None |
10.1128/aac.00471-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MBC |
3.13 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00471-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.064 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.073 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2018.02.049 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2008.09.035 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.9 |
ug.mL-1 |
10.1016/j.ejmech.2007.12.019 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.00017-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
7.8 |
ug.mL-1 |
10.1016/j.ejmech.2007.12.019 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00017-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.01439-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.04.001 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01053-06 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
22.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.05.032 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
25.0 |
ug.mL-1 |
10.1021/acs.jnatprod.0c01212 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
25.0 |
ug.mL-1 |
10.1021/jm00143a010 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
25.0 |
ug.mL-1 |
10.1021/jm00145a020 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
25.0 |
ug.mL-1 |
10.1021/jm00220a012 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b01287 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00017-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01247-10 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.bmc.2006.12.035 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.04.001 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1024.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01742 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4096.0 |
ug.mL-1 |
10.1016/j.bmc.2006.12.035 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32000.0 |
nM |
10.1016/j.ejmech.2019.111636 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32000.0 |
nM |
10.1021/acs.jmedchem.2c01076 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
nan |
None |
10.1016/j.bmc.2019.04.032 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
nan |
None |
10.1016/j.ejmech.2019.04.067 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC100 |
1.56 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Ratio |
10.0 |
None |
10.1128/aac.00405-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Ratio |
24.0 |
None |
10.1128/aac.01439-09 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Ratio |
43.0 |
None |
10.1128/aac.00405-08 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Ratio |
250.0 |
None |
10.1128/aac.00405-08 |
| Klebsiella pneumoniae subsp. pneumoniae |
Klebsiella pneumoniae subsp. pneumoniae |
EC50 |
5400.0 |
nM |
10.1016/j.bmcl.2016.04.089 |
| Leishmania donovani |
Leishmania donovani |
IC50 |
nan |
None |
10.1021/np020592u |
| Leishmania donovani |
Leishmania donovani |
IC50 |
nan |
None |
10.1021/np0400095 |
| Leishmania donovani |
Leishmania donovani |
IC50 |
nan |
None |
10.1021/np0601399 |
| Leishmania donovani |
Leishmania donovani |
IC90 |
nan |
None |
10.1021/np020592u |
| Leishmania donovani |
Leishmania donovani |
IC90 |
nan |
None |
10.1021/np0400095 |
| Leishmania donovani |
Leishmania donovani |
IC90 |
nan |
None |
10.1021/np0601399 |
| Listeria monocytogenes |
Listeria monocytogenes |
Inhibition |
100.0 |
% |
10.1021/jm0703901 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
nan |
None |
10.1016/j.bmc.2019.04.032 |
| Macaca fascicularis |
Brain |
Fu |
0.162 |
None |
10.1124/dmd.111.038778 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
Activity |
0.0 |
% |
10.1128/aac.00426-10 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
Activity |
11.1 |
% |
10.1128/aac.00426-10 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
Activity |
15.4 |
% |
10.1128/aac.00426-10 |
| Micrococcus luteus |
Micrococcus luteus |
IZ |
49.0 |
mm |
10.1016/j.bmc.2007.09.025 |
| Micrococcus luteus |
Micrococcus luteus |
MIC |
0.125 |
ug.mL-1 |
10.1021/ml300350p |
| Mobiluncus curtisii subsp. curtisii |
Mobiluncus curtisii subsp. curtisii |
MIC |
0.004 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Morganella morganii |
Morganella morganii |
MIC |
10.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00174 |
| Morganella morganii |
Morganella morganii |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Mus musculus |
Brain |
Drug uptake |
10.25 |
ug ml-1 |
10.1021/jm901858n |
| Mus musculus |
Brain |
Fu |
0.121 |
None |
10.1124/dmd.111.038778 |
| Mus musculus |
Canalicular multispecific organic anion transporter 2 |
Activity |
nan |
None |
10.1124/dmd.31.11.1296 |
| Mus musculus |
Integrin alpha M |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mus musculus |
Integrin alpha M |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mus musculus |
J774 |
Activity |
73.0 |
% |
10.1016/j.bmc.2016.01.028 |
| Mus musculus |
J774 |
Activity |
78.0 |
% |
10.1016/j.ejmech.2013.12.013 |
| Mus musculus |
J774 |
Activity |
80.0 |
% |
10.1016/j.bmcl.2016.03.066 |
| Mus musculus |
J774 |
Activity |
82.0 |
% |
10.1016/j.ejmech.2013.12.013 |
| Mus musculus |
J774 |
Activity |
85.0 |
% |
10.1016/j.bmc.2016.01.028 |
| Mus musculus |
J774 |
Activity |
86.0 |
% |
10.1016/j.ejmech.2013.12.013 |
| Mus musculus |
J774 |
Activity |
87.0 |
% |
10.1016/j.bmcl.2016.03.066 |
| Mus musculus |
J774 |
Activity |
93.0 |
% |
10.1016/j.bmcl.2016.03.066 |
| Mus musculus |
J774 |
Activity |
95.0 |
% |
10.1016/j.bmc.2016.01.028 |
| Mus musculus |
J774.A1 |
Activity |
1.03 |
deltalog10CFU |
10.1016/j.ejmech.2022.114145 |
| Mus musculus |
J774.A1 |
Activity |
90.0 |
% |
10.1128/aac.00375-07 |
| Mus musculus |
J774.A1 |
Activity |
94.4 |
None |
10.1128/aac.00375-07 |
| Mus musculus |
J774.A1 |
CC50 |
207.03 |
ug.mL-1 |
10.1016/j.bmc.2010.09.006 |
| Mus musculus |
J774.A1 |
IC50 |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2022.117006 |
| Mus musculus |
J774.A1 |
IC50 |
nan |
None |
10.1016/j.bmc.2019.07.045 |
| Mus musculus |
J774.A1 |
IC50 |
nan |
None |
10.1016/j.bmcl.2019.02.019 |
| Mus musculus |
Mus musculus |
Activity |
85.0 |
% |
10.1021/np50025a010 |
| Mus musculus |
Mus musculus |
Activity |
174.0 |
% |
10.1021/np50025a010 |
| Mus musculus |
Mus musculus |
AUC |
24760.0 |
ng.hr.mL-1 |
10.1128/aac.00367-09 |
| Mus musculus |
Mus musculus |
AUC |
48200.0 |
ng.hr.mL-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cmax |
6197.22 |
nM |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cmax |
19138.47 |
nM |
10.1128/aac.00367-09 |
| Mus musculus |
Mus musculus |
Cp |
0.66 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cp |
3.18 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cp |
3.33 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cp |
3.82 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cp |
4.49 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cp |
4.52 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cp |
5.1 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
EC90 |
0.007 |
None |
10.1016/s0960-894x(01)00283-9 |
| Mus musculus |
Mus musculus |
EC99 |
0.451 |
None |
10.1016/s0960-894x(01)00283-9 |
| Mus musculus |
Mus musculus |
FC |
1.3 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
FC |
1.5 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
FC |
1.8 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
FC |
1.9 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
FC |
2.0 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
FC |
2.1 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
FC |
2.5 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
FC |
2.7 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
FC |
3.7 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
FC |
4.5 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
FC |
8.4 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
FC |
16.5 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
FC |
171.9 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Mus musculus |
IC50 |
nan |
None |
10.1016/j.ejmech.2016.07.039 |
| Mus musculus |
Mus musculus |
Inhibition |
9.56 |
% |
10.1016/j.bmc.2016.09.012 |
| Mus musculus |
Mus musculus |
Inhibition |
nan |
% |
10.1016/j.ejmech.2016.08.034 |
| Mus musculus |
Mus musculus |
T1/2 |
2.86 |
hr |
10.1128/aac.00367-09 |
| Mus musculus |
Mus musculus |
T1/2 |
3.4 |
hr |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Tmax |
6.0 |
hr |
10.1371/journal.pmed.0030466 |
| Mus musculus |
NIH3T3 |
Survival |
62.0 |
% |
10.1021/acs.jnatprod.5b01033 |
| Mus musculus |
Nitric oxide synthase, inducible |
IC50 |
nan |
None |
None |
| Mus musculus |
Nitric oxide synthase, inducible |
Ki |
nan |
None |
None |
| Mus musculus |
Nuclear receptor subfamily 1 group I member 2 |
FC |
1.6 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
Nuclear receptor subfamily 1 group I member 2 |
FC |
1.7 |
None |
10.1124/dmd.112.048009 |
| Mus musculus |
RAW264.7 |
Activity |
nan |
None |
10.1016/j.ejmech.2017.12.088 |
| Mus musculus |
RAW264.7 |
CC50 |
80.39 |
ug.mL-1 |
10.1016/j.ejmech.2021.113472 |
| Mus musculus |
RAW264.7 |
CC50 |
24000.0 |
nM |
10.1016/j.ejmech.2020.112908 |
| Mus musculus |
RAW264.7 |
GI |
23.48 |
% |
10.1016/j.bmc.2017.03.053 |
| Mus musculus |
RAW264.7 |
GI |
nan |
None |
10.1016/j.bmc.2015.03.004 |
| Mus musculus |
RAW264.7 |
GI |
nan |
None |
10.1016/j.bmc.2017.11.031 |
| Mus musculus |
RAW264.7 |
GI |
nan |
None |
10.1016/j.ejmech.2018.07.046 |
| Mus musculus |
RAW264.7 |
GI50 |
700.0 |
ug.mL-1 |
10.1016/j.bmc.2015.04.001 |
| Mus musculus |
RAW264.7 |
GI50 |
850000.0 |
nM |
10.1039/C3MD00251A |
| Mus musculus |
RAW264.7 |
GI50 |
nan |
None |
10.1016/j.ejmech.2018.07.046 |
| Mus musculus |
RAW264.7 |
IC50 |
nan |
None |
10.1016/j.ejmech.2022.114831 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.bmc.2014.10.016 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.bmc.2015.02.032 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.bmc.2016.01.011 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.ejmech.2014.09.028 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.ejmech.2014.12.046 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.ejmech.2015.06.032 |
| Mycobacterium avium |
Mycobacterium avium |
Activity |
0.0 |
% |
10.1016/j.bmcl.2006.08.090 |
| Mycobacterium avium |
Mycobacterium avium |
GI |
90.0 |
% |
10.1016/j.bmc.2012.05.004 |
| Mycobacterium avium |
Mycobacterium avium |
GI |
90.0 |
% |
10.1016/j.bmc.2016.09.008 |
| Mycobacterium avium |
Mycobacterium avium |
GI |
90.0 |
% |
10.1016/j.bmcl.2011.11.114 |
| Mycobacterium avium |
Mycobacterium avium |
Inhibition |
90.0 |
% |
10.1016/j.bmc.2006.12.032 |
| Mycobacterium avium |
Mycobacterium avium |
Inhibition |
90.0 |
% |
10.1021/jm058167w |
| Mycobacterium avium |
Mycobacterium avium |
Inhibition |
90.0 |
% |
10.1021/jm0703901 |
| Mycobacterium avium |
Mycobacterium avium |
Inhibition |
90.0 |
% |
10.1021/jm070391t |
| Mycobacterium avium |
Mycobacterium avium |
Inhibition |
100.0 |
% |
10.1016/j.bmc.2006.12.032 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.bmcl.2007.02.024 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.125 |
ug.mL-1 |
10.1016/s0960-894x(03)00596-1 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.125 |
ug.mL-1 |
10.1016/s0960-894x(03)00597-3 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.15 |
ug.mL-1 |
10.1128/aac.00749-08 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2009.06.005 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm701560p |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.3 |
ug.mL-1 |
10.1016/s0960-894x(99)00510-7 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.3 |
ug.mL-1 |
10.1021/jm0602662 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.78 |
ug.mL-1 |
10.1039/C8MD00056E |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2013.10.011 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
3.1 |
ug.mL-1 |
10.1021/jm070638m |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00972 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
90.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.083 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
100.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
780.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
16000.0 |
nM |
10.1016/j.ejmech.2010.02.037 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
65000.0 |
nM |
10.1016/j.ejmech.2010.02.037 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
nan |
ug.mL-1 |
10.1016/s0960-894x(00)00159-1 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Mycobacterium avium |
Mycobacterium avium |
MIC50 |
16.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium avium |
Mycobacterium avium |
MIC50 |
32.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium avium |
Mycobacterium avium |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2016.03.003 |
| Mycobacterium avium |
Mycobacterium avium |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm058167w |
| Mycobacterium avium |
Mycobacterium avium |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Mycobacterium avium |
Mycobacterium avium |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm070391t |
| Mycobacterium avium |
Mycobacterium avium |
MIC90 |
128.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium avium |
Mycobacterium avium |
MIC90 |
780.0 |
nM |
10.1021/ml200036r |
| Mycobacterium avium |
Mycobacterium avium |
MIC>99 |
32.0 |
uM |
10.1016/j.bmc.2017.08.010 |
| Mycobacterium avium |
Mycobacterium avium |
MIC>99 |
32.0 |
uM |
10.1016/j.ejmech.2017.02.058 |
| Mycobacterium avium |
Mycobacterium avium |
MIC>99 |
32.0 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium avium |
Mycobacterium avium |
MIC>99 |
62.0 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium avium complex sp. |
Mycobacterium avium complex sp. |
MIC |
30.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.083 |
| Mycobacterium avium complex sp. |
Mycobacterium avium complex sp. |
MIC=>90 |
10.0 |
uM |
10.1016/j.bmc.2015.03.018 |
| Mycobacterium avium complex sp. |
Mycobacterium avium complex sp. |
MIC>90 |
10.0 |
uM |
10.1016/j.bmc.2015.06.047 |
| Mycobacterium avium subsp. paratuberculosis |
Mycobacterium avium subsp. paratuberculosis |
Activity |
2.0 |
ug ml-1 |
10.1128/aac.00678-07 |
| Mycobacterium avium subsp. paratuberculosis |
Mycobacterium avium subsp. paratuberculosis |
Activity |
64.0 |
ug ml-1 |
10.1128/aac.00678-07 |
| Mycobacterium avium subsp. paratuberculosis |
Mycobacterium avium subsp. paratuberculosis |
Activity |
nan |
None |
10.1128/aac.00678-07 |
| Mycobacterium avium subsp. paratuberculosis |
Mycobacterium avium subsp. paratuberculosis |
MIC=>90 |
109.0 |
uM |
10.1016/j.bmc.2015.03.018 |
| Mycobacterium avium subsp. paratuberculosis |
Mycobacterium avium subsp. paratuberculosis |
MIC>90 |
109.0 |
uM |
10.1016/j.bmc.2015.06.047 |
| Mycobacterium gordonae |
Mycobacterium gordonae |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium gordonae |
Mycobacterium gordonae |
MIC |
0.6 |
ug.mL-1 |
10.1016/s0960-894x(99)00510-7 |
| Mycobacterium gordonae |
Mycobacterium gordonae |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
Activity |
nan |
None |
10.1021/acs.jnatprod.7b00903 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
IC50 |
nan |
None |
10.1021/jm900672t |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
IC50 |
nan |
None |
10.1021/np900281r |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
0.125 |
ug.mL-1 |
10.1016/s0960-894x(03)00596-1 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
0.125 |
ug.mL-1 |
10.1016/s0960-894x(03)00597-3 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
0.2 |
ug.mL-1 |
10.1021/jm00150a006 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
0.3 |
ug.mL-1 |
10.1021/np9901940 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.06.010 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
0.78 |
ug.mL-1 |
10.1021/jm00100a012 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2013.10.011 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
3.1 |
ug.mL-1 |
10.1021/jm070638m |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
nan |
None |
10.1021/np900281r |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
Activity |
100.0 |
% |
10.1016/j.bmcl.2006.08.090 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
0.05 |
ug.mL-1 |
10.1021/jm00150a006 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
0.125 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
0.25 |
ug.mL-1 |
10.1016/s0960-894x(03)00596-1 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
0.25 |
ug.mL-1 |
10.1016/s0960-894x(03)00597-3 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2013.10.011 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
0.78 |
ug.mL-1 |
10.1039/C8MD00056E |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
30.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
100.0 |
nM |
10.1021/ml5003458 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
125.0 |
nM |
10.1016/j.ejmech.2010.02.037 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250.0 |
nM |
10.1016/j.ejmech.2010.02.037 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
7590.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC90 |
780.0 |
nM |
10.1021/ml200036r |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
0.125 |
uM |
10.1016/j.bmc.2017.08.010 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
0.125 |
uM |
10.1016/j.ejmech.2017.02.058 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
0.125 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
0.25 |
uM |
10.1016/j.bmc.2017.08.010 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
0.25 |
uM |
10.1016/j.ejmech.2017.02.058 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
0.25 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium leprae |
Mycobacterium leprae |
Activity |
0.0 |
pg |
10.1016/j.bmc.2019.04.032 |
| Mycobacterium leprae |
Mycobacterium leprae |
Activity |
0.0 |
pmol |
10.1016/j.bmc.2019.04.032 |
| Mycobacterium leprae |
Mycobacterium leprae |
Activity |
0.7 |
pmol |
10.1016/j.bmc.2019.04.032 |
| Mycobacterium leprae |
Mycobacterium leprae |
Activity |
0.73 |
pmol |
10.1016/j.bmc.2019.04.032 |
| Mycobacterium leprae |
Mycobacterium leprae |
Activity |
211.0 |
pg |
10.1016/j.bmc.2019.04.032 |
| Mycobacterium leprae |
Mycobacterium leprae |
Activity |
215.0 |
pg |
10.1016/j.bmc.2019.04.032 |
| Mycobacterium leprae |
Mycobacterium leprae |
Inhibition |
86.0 |
% |
10.1016/j.bmc.2019.04.032 |
| Mycobacterium marinum |
Mycobacterium marinum |
Activity |
1.9 |
deltalog10CFU/ml |
10.1016/j.bmc.2016.01.059 |
| Mycobacterium marinum |
Mycobacterium marinum |
Activity |
27.0 |
% |
10.1021/acs.jmedchem.1c02122 |
| Mycobacterium marinum |
Mycobacterium marinum |
Activity |
nan |
None |
10.1016/j.ejmech.2015.01.020 |
| Mycobacterium marinum |
Mycobacterium marinum |
Activity |
nan |
None |
10.1021/acs.jmedchem.1c01407 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm701560p |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
0.6 |
ug.mL-1 |
10.1016/s0960-894x(99)00510-7 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
0.6 |
ug.mL-1 |
10.1021/jm0602662 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
230.0 |
nM |
10.1021/ml5003458 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
1200.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC90 |
780.0 |
nM |
10.1021/ml200036r |
| Mycobacterium scrofulaceum |
Mycobacterium scrofulaceum |
MIC |
0.063 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium scrofulaceum |
Mycobacterium scrofulaceum |
MIC |
0.125 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium scrofulaceum |
Mycobacterium scrofulaceum |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycobacterium scrofulaceum |
Mycobacterium scrofulaceum |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium smegmatis |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.bmc.2014.10.016 |
| Mycobacterium smegmatis |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.bmc.2015.02.032 |
| Mycobacterium smegmatis |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.bmc.2015.03.004 |
| Mycobacterium smegmatis |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.ejmech.2015.06.032 |
| Mycobacterium smegmatis |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.ejmech.2016.08.034 |
| Mycobacterium smegmatis (strain ATCC 700084 / mc(2)155) |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.ejmech.2016.06.042 |
| Mycobacterium szulgai |
Mycobacterium szulgai |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycobacterium tuberculosis |
ATP-dependent Clp protease ATP-binding subunit ClpC1 |
Kd |
nan |
None |
10.1021/acs.jnatprod.9b01095 |
| Mycobacterium tuberculosis |
DNA-directed RNA polymerase beta chain |
IC50 |
10.0 |
nM |
10.1016/j.bmcl.2011.08.054 |
| Mycobacterium tuberculosis |
DNA-directed RNA polymerase beta chain |
logIC50 |
-2.399 |
None |
10.1016/j.bmcl.2011.08.054 |
| Mycobacterium tuberculosis |
Enoyl-[acyl-carrier-protein] reductase |
IC50 |
30.0 |
nM |
10.1021/jm500833f |
| Mycobacterium tuberculosis |
Enoyl-[acyl-carrier-protein] reductase |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2018.07.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
0.5 |
None |
10.1021/jm060957y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.0 |
log10CFU |
10.1021/acs.jmedchem.2c01493 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.0 |
log10CFU/ml |
10.1021/acs.jmedchem.1c02122 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.03 |
deltalog10CFU |
10.1021/acs.jmedchem.1c00263 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.06 |
deltalog10CFU |
10.1016/j.bmc.2016.01.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.1 |
log10CFU |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.58 |
log10CFU |
10.1021/acsmedchemlett.5b00324 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.76 |
log10CFU |
10.1039/C4MD00288A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.93 |
log10CFU |
10.1039/C4MD00288A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.0 |
log10CFU |
10.1021/acs.jmedchem.0c01727 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.1 |
deltalog10CFU/ml |
10.1016/j.bmc.2016.01.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.39 |
deltalog10CFU |
10.1016/j.bmc.2016.01.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.44 |
log10CFU |
10.1016/j.ejmech.2016.11.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.8 |
log10CFU |
10.1039/C4MD00288A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.86 |
deltalog10CFU |
10.1016/j.bmc.2016.01.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
3.0 |
log10CFU/ml |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
3.3 |
10'5CFU |
10.1016/j.bmc.2017.03.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
3.31 |
log10CFU |
10.1039/C4MD00288A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
3.9 |
log10CFU |
10.1016/j.bmcl.2016.09.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
4.49 |
log10CFU |
10.1021/acs.jmedchem.1c00263 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
5.2 |
None |
10.1016/j.bmcl.2016.09.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
5.6 |
% |
10.1128/aac.00897-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
9.2 |
% |
10.1128/aac.01124-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
29.19 |
% |
10.1016/j.bmcl.2012.10.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
61.2 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
79.8 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
82.58 |
% |
10.1016/j.bmcl.2012.10.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
87.0 |
% |
10.1016/j.ejmech.2016.08.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
87.0 |
% |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
87.2 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
90.9 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
93.8 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
94.2 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
94.5 |
% |
10.1128/aac.01124-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
95.0 |
% |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
95.79 |
% |
10.1021/jm701560p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
95.9 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
96.3 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
96.59 |
% |
10.1016/j.bmc.2010.09.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
98.0 |
% |
10.1021/jm100165w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
98.0 |
% |
10.1039/C5MD00131E |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
98.42 |
% |
10.1021/jm701560p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
99.4 |
% |
10.1128/aac.01124-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
99.79 |
% |
10.1021/jm701560p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
99.83 |
% |
10.1016/j.bmc.2010.09.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
99.93 |
% |
10.1016/j.bmc.2010.09.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
99.97 |
% |
10.1016/j.bmc.2010.09.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
100.0 |
% |
10.1021/np0703702 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
391.0 |
mg |
10.1126/science.1106753 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
466.0 |
mg |
10.1126/science.1106753 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmc.2009.04.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmc.2016.03.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmc.2022.116777 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmcl.2012.10.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmcl.2022.128824 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmcl.2022.128871 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.ejmech.2012.04.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.ejmech.2020.112772 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acs.jmedchem.0c01374 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acs.jmedchem.2c01493 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acs.jmedchem.5b01699 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acs.jmedchem.5b01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acs.jnatprod.7b00903 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acsmedchemlett.7b00287 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/jm0703901 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/ml200157f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1039/C4MD00288A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1039/d1md00387a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1128/aac.00661-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1128/aac.00898-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1128/aac.01468-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1128/aac.01486-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
C50g |
2.019 |
mg/L |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
C50g |
1932.0 |
mg/L |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
C50k |
7.652 |
mg/L |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
C50k |
22.41 |
mg/L |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
0.0 |
/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
1.95 |
/ml |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
39.0 |
None |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
2000.0 |
None |
10.1016/j.ejmech.2015.03.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
DIZ |
nan |
None |
10.1007/s00044-013-0487-6 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Drug uptake |
nan |
None |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC50 |
20.0 |
nM |
10.1016/j.bmcl.2012.12.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC90 |
0.02 |
uM |
10.1016/j.bmcl.2012.12.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC90 |
0.03 |
uM |
10.1016/j.bmcl.2012.12.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC90 |
0.1 |
ug ml-1 |
10.1016/j.bmcl.2004.09.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC90/MIC |
1.67 |
None |
10.1016/j.bmcl.2004.09.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC99 |
1.5 |
ug ml-1 |
10.1016/j.bmcl.2004.09.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
ED99 |
9.8 |
mg kg-1 |
10.1128/aac.01423-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Emax |
4.2 |
log10CFU/ml |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Emax |
6.2 |
log10CFU/ml |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Emax |
6.3 |
log10CFU/ml |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Emax |
30.0 |
mg kg-1 |
10.1128/aac.01423-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
0.46 |
None |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
0.48 |
None |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
0.81 |
None |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
0.98 |
None |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.34 |
log10RLU |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.42 |
log10RLU |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.49 |
None |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.5 |
None |
10.1016/j.ejmech.2019.112010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.6 |
None |
10.1016/j.ejmech.2020.112035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.6 |
None |
10.1016/j.ejmech.2020.112402 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.73 |
None |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.8 |
None |
10.1021/acs.jnatprod.9b00475 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.83 |
None |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.85 |
None |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
2.0 |
None |
10.1016/j.bmc.2016.09.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
2.0 |
None |
10.1016/j.ejmech.2009.12.074 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
2.0 |
None |
10.1016/j.ejmech.2014.12.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
2.2 |
None |
10.1016/j.bmc.2016.07.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
2.68 |
None |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
0.0 |
% |
10.1016/j.bmc.2012.09.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
46.21 |
% |
10.1016/j.bmc.2016.09.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
53.0 |
% |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
55.0 |
% |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
62.27 |
% |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
63.0 |
% |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
65.0 |
% |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
66.33 |
% |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
68.0 |
% |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
71.0 |
% |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
72.0 |
% |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
73.67 |
% |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
74.0 |
% |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
76.33 |
% |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
84.0 |
% |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
86.0 |
% |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
91.0 |
% |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
94.6 |
% |
10.1016/j.ejmech.2017.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
95.0 |
% |
10.1007/s00044-012-0451-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
95.0 |
% |
10.1016/j.bmcl.2013.06.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
95.0 |
% |
10.1016/j.ejmech.2011.07.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
95.0 |
% |
10.1016/j.ejmech.2011.07.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
95.0 |
% |
10.1016/j.ejmech.2012.01.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
96.0 |
% |
10.1016/j.ejmech.2008.12.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
96.4 |
% |
10.1016/j.ejmech.2017.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
96.8 |
% |
10.1016/j.ejmech.2017.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
97.0 |
% |
10.1016/j.bmc.2007.05.063 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
97.0 |
% |
10.1016/j.bmcl.2013.06.076 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
97.0 |
% |
10.1016/j.ejmech.2006.12.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
97.6 |
% |
10.1021/np9000569 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
98.0 |
% |
10.1007/s00044-011-9808-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
98.0 |
% |
10.1007/s00044-011-9857-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
98.0 |
% |
10.1007/s00044-012-0322-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
98.0 |
% |
10.1007/s00044-013-0803-1 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
98.0 |
% |
10.1016/j.bmc.2013.06.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
98.0 |
% |
10.1016/j.ejmech.2011.09.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
98.0 |
% |
10.1016/j.ejmech.2013.03.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
98.0 |
% |
10.1016/j.ejmech.2013.05.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
98.0 |
% |
10.1016/j.ejmech.2017.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1007/s00044-012-0026-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1007/s00044-012-0041-y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1007/s00044-012-0073-3 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1007/s00044-012-0129-4 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1016/j.ejmech.2012.12.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1016/j.ejmech.2013.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1016/j.ejmech.2014.02.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1016/j.ejmech.2017.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.5 |
% |
10.1016/j.ejmech.2017.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.bmc.2012.05.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.bmc.2012.09.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.bmc.2013.07.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.bmc.2016.09.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.bmcl.2011.11.114 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.bmcl.2020.127351 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.ejmech.2013.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
nan |
None |
10.1007/s00044-012-0255-z |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
nan |
None |
10.1016/j.bmc.2012.05.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
nan |
None |
10.1016/j.bmc.2013.07.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
nan |
None |
10.1016/j.bmc.2016.02.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
nan |
None |
10.1021/acs.jmedchem.5b00608 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
nan |
None |
10.1039/C7MD00146K |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI50 |
30.0 |
nM |
10.1016/j.ejmech.2013.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Hg |
0.361 |
None |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Hg |
4.542 |
None |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Hk |
1.388 |
None |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Hk |
45.33 |
None |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0014 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0014 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0016 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0017 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0017 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.093 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0018 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0018 |
ug.mL-1 |
10.1016/j.bmcl.2015.11.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0018 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.056 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0019 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0019 |
ug.mL-1 |
10.1039/C8MD00055G |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.002 |
ug.mL-1 |
10.1039/C5MD00057B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0021 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0021 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0024 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.093 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.004 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.004 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0043 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0047 |
ug.mL-1 |
10.1021/np9000703 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.02 |
ug.mL-1 |
10.1039/C8MD00055G |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.08 |
ug.mL-1 |
10.1021/acs.jnatprod.0c01104 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.72 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.72 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
2.0 |
ug.mL-1 |
10.1021/ml5001933 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
2.4 |
nM |
10.1016/j.bmcl.2019.03.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
2.4 |
nM |
10.1016/j.ejmech.2017.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
2.9 |
ug.mL-1 |
10.1021/ml5001933 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
4.1 |
nM |
10.1021/acsmedchemlett.5b00176 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
4.6 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
4.6 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
4.7 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
8.4 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
10.0 |
nM |
10.1016/j.bmc.2020.115797 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
13.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
20.0 |
nM |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
20.0 |
nM |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
20.0 |
nM |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
30.0 |
nM |
10.1016/j.bmcl.2017.07.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
40.0 |
nM |
10.1016/j.ejmech.2017.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
60.0 |
nM |
10.1016/j.bmc.2020.115797 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
91.0 |
nM |
10.1021/acs.jmedchem.2c01493 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
147.0 |
ug.mL-1 |
10.1016/s0960-894x(01)00283-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
152.0 |
nM |
10.1021/np500617u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
550.0 |
nM |
10.1016/j.ejmech.2019.01.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
1200.0 |
nM |
10.1016/j.bmc.2021.116506 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
1200.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
1220.0 |
nM |
10.1016/j.ejmech.2019.01.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
50000.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
nan |
None |
10.1021/ml5001933 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
nan |
None |
10.1021/np900281r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.015 |
ug.mL-1 |
10.1016/j.ejmech.2010.06.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.0151 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.0173 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.028 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.043 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.043 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.056 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.048 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.051 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.53 |
ug.mL-1 |
10.1039/C8MD00055G |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.72 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.8 |
ug.mL-1 |
10.1039/C8MD00055G |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
3.7 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
3.7 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
4.9 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
4.9 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
6.9 |
nM |
10.1021/acsmedchemlett.5b00176 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
12.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
20.0 |
nM |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
22.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
30.0 |
nM |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
30.0 |
nM |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
39.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
2300.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
50000.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Imax |
54.0 |
% |
10.1016/j.bmcl.2019.04.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
INH |
0.13 |
ug ml-1 |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
0.0 |
% |
10.1021/jm100165w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
13.0 |
% |
10.1016/j.bmcl.2019.04.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
49.0 |
% |
10.1016/j.bmcl.2008.09.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
54.8 |
% |
10.1021/jm030479g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
56.0 |
% |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
61.0 |
% |
10.1021/acs.jmedchem.5b00608 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
61.2 |
% |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
63.0 |
% |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
68.0 |
% |
10.1021/acs.jmedchem.5b00608 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
73.0 |
% |
10.1016/j.bmcl.2008.09.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
80.0 |
% |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
90.0 |
% |
10.1016/j.bmc.2008.10.086 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
90.0 |
% |
10.1021/np050424c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
91.7 |
% |
10.1021/jm030479g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
91.9 |
% |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
93.0 |
% |
10.1021/jm061288r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
94.0 |
% |
10.1016/j.bmcl.2008.09.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
94.3 |
% |
10.1021/jm030479g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.0 |
% |
10.1016/j.bmc.2017.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.0 |
% |
10.1016/j.bmcl.2004.05.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.0 |
% |
10.1016/j.ejmech.2011.03.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.0 |
% |
10.1016/j.ejmech.2011.08.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.0 |
% |
10.1016/j.ejmech.2013.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
97.0 |
% |
10.1016/j.ejmech.2009.09.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
97.6 |
% |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1007/s00044-011-9952-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1016/j.bmc.2017.09.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1016/j.bmcl.2015.07.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1016/j.bmcl.2016.06.038 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1016/j.ejmech.2007.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1016/j.ejmech.2010.06.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1016/j.ejmech.2012.05.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1016/j.ejmech.2012.08.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1016/j.ejmech.2014.02.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1016/j.ejmech.2014.06.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1016/j.ejmech.2014.07.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1016/j.ejmech.2016.02.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1016/j.ejmech.2020.112886 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
98.0 |
% |
10.1039/d2md00076h |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1007/s00044-011-9950-4 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1007/s00044-013-0472-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1007/s00044-013-0839-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.bmc.2015.11.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.bmcl.2008.09.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2009.11.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2010.04.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2012.03.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2014.07.100 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2020.112358 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.5 |
% |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1007/s00044-012-9971-7 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1016/j.bmc.2006.12.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1016/j.bmc.2014.10.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1016/j.bmcl.2007.04.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1016/j.bmcl.2008.09.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1016/j.bmcl.2021.128261 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1016/j.ejmech.2012.08.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1016/j.ejmech.2022.114831 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1021/jm0703901 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1021/jm070391t |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1021/jm100165w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1021/jm100568q |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
nan |
% |
10.1007/s00044-013-0472-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
nan |
% |
10.1016/j.ejmech.2015.03.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
nan |
% |
10.1016/j.ejmech.2019.05.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IZ |
28.0 |
mm |
10.1016/j.bmc.2007.09.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Kgmax |
6.195 |
10'-3 log10CFU/ml/hr |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Kgmax |
9.756 |
10'-3 log10CFU/ml/hr |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Kkmax |
15.83 |
10'-3 log10CFU/ml/hr |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Kkmax |
29.38 |
10'-3 log10CFU/ml/hr |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
1.0 |
None |
10.1021/jm4019228 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
1.76 |
None |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
1.89 |
None |
10.1126/science.1106753 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
1.93 |
None |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
2.75 |
None |
10.1126/science.1106753 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
2.8 |
None |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.21 |
None |
10.1016/j.ejmech.2010.05.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.279 |
None |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.31 |
None |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.71 |
None |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.8 |
None |
10.1016/j.ejmech.2010.07.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.972 |
None |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.98 |
None |
10.1016/j.ejmech.2010.05.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.05 |
None |
10.1126/science.1106753 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.53 |
None |
10.1021/np3007167 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.72 |
None |
10.1126/science.1106753 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.231 |
None |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.634 |
None |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.75 |
None |
10.1021/np3007167 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
6.14 |
None |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
7.409 |
None |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
nan |
None |
10.1016/j.ejmech.2010.07.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
4.1 |
None |
10.1128/aac.00898-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
6.0 |
None |
10.1128/aac.00898-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-1.82 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-1.7 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-1.55 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-1.25 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-1.17 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-0.89 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-0.88 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-0.28 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
0.221 |
None |
10.1128/aac.01474-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
0.3 |
None |
10.1128/aac.01474-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
0.44 |
None |
10.1128/aac.01474-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
1.32 |
None |
10.1128/aac.00753-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
1.7 |
None |
10.1016/j.ejmech.2012.02.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
4.63 |
None |
10.1128/aac.00753-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
6.36 |
None |
10.1128/aac.00753-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(1/C) |
5.91 |
None |
10.1021/jm00210a025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
0.5 |
None |
10.1016/j.bmc.2017.11.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
0.8 |
None |
10.1016/j.ejmech.2017.12.088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
0.9 |
None |
10.1016/j.ejmech.2020.112178 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.2 |
None |
10.1016/j.bmc.2017.11.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.3 |
None |
10.1016/j.bmc.2017.03.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.5 |
None |
10.1016/j.ejmech.2017.12.088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.8 |
None |
10.1016/j.ejmech.2020.112178 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
2.0 |
None |
10.1016/j.bmc.2017.03.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
2.0 |
None |
10.1016/j.bmc.2017.12.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
2.7 |
None |
10.1021/acs.jmedchem.2c00972 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
-logMIC |
6.924 |
None |
10.1007/s00044-012-0385-3 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
0.01 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
0.12 |
uM |
10.1021/acs.jnatprod.9b01095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
0.24 |
uM |
10.1021/acs.jnatprod.9b01095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
0.39 |
uM |
10.1016/j.bmc.2008.12.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
100.0 |
ug ml-1 |
10.1016/j.bmc.2007.09.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
161.0 |
ng/ml |
10.1021/acs.jnatprod.5b00770 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
nan |
None |
10.1016/j.ejmech.2018.02.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC90 |
0.1 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC90 |
0.5 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC99.9 |
0.78 |
ug ml-1 |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC99.9 |
1.56 |
ug ml-1 |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC99.9 |
1.56 |
ug ml-1 |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MCC |
3.0 |
ug.mL-1 |
10.1021/jm0602662 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0008 |
ug.mL-1 |
10.1128/aac.00550-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.001 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0016 |
ug.mL-1 |
10.1128/aac.00550-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.002 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0021 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0025 |
ug.mL-1 |
10.1021/np800082e |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0025 |
ug.mL-1 |
10.1039/d2md00401a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.003 |
ug.mL-1 |
10.1007/s00044-012-0222-8 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.003 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.003 |
ug.mL-1 |
10.1039/C8MD00212F |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0032 |
ug.mL-1 |
10.1128/aac.00550-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.ejmech.2010.07.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.ejmech.2020.112045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.ejmech.2020.112440 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.004 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.005 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.005 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00972 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.006 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0063 |
ug.mL-1 |
10.1021/acs.jnatprod.5b00961 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.007 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.007 |
ug.mL-1 |
10.1021/jm4012033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.008 |
ug.mL-1 |
10.1016/j.bmcl.2007.02.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.008 |
ug.mL-1 |
10.1021/jm500432n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.bmcl.2014.09.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2020.112175 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.01 |
ug.mL-1 |
10.1021/jm4012033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0125 |
ug.mL-1 |
10.1016/j.bmcl.2018.12.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.013 |
ug.mL-1 |
10.1016/j.bmcl.2018.05.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.bmc.2007.04.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.bmc.2010.02.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.076 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.ejmech.2008.12.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.ejmech.2022.114145 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1021/jm500432n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.016 |
ug.mL-1 |
10.1016/j.bmcl.2006.12.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.016 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.016 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00972 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.017 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.019 |
ug.mL-1 |
10.1016/j.bmcl.2018.05.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.bmcl.2006.08.090 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.093 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2014.10.079 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2017.03.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.ejmech.2021.113603 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1021/jm00150a006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1021/np5005328 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmc.2010.05.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmc.2013.09.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmc.2013.10.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmc.2019.07.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmc.2022.116777 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.093 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2021.113580 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00500 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1021/jm201608g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1021/np049831z |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1039/d1md00387a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.037 |
ug.mL-1 |
10.1016/j.bmc.2022.117006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.037 |
ug.mL-1 |
10.1016/j.ejmech.2020.112409 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.038 |
ug.mL-1 |
10.1016/j.ejmech.2016.11.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0382 |
ug.mL-1 |
10.1016/j.ejmech.2021.113398 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00500 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1039/C5MD00057B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.041 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.042 |
ug.mL-1 |
10.1016/j.ejmech.2022.114502 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.043 |
ug.mL-1 |
10.1016/j.bmcl.2015.11.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.043 |
ug.mL-1 |
10.1016/j.ejmech.2017.06.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.043 |
ug.mL-1 |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.045 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.049 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmc.2015.04.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2014.09.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2017.06.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2019.06.038 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/jm00150a006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/jm500853v |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1128/aac.01288-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1128/aac.01486-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.057 |
ug.mL-1 |
10.1016/j.ejmech.2020.112075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmc.2008.10.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2008.04.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2010.11.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2011.10.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2014.02.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2019.07.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2020.112996 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2021.113580 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/s0960-894x(00)00058-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/s0960-894x(00)00648-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00515 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1021/np0303411 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1021/np2000667 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1039/d1md00387a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.062 |
ug.mL-1 |
10.1016/j.ejmech.2021.113472 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.062 |
ug.mL-1 |
10.1021/jm000413a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.bmcl.2012.08.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.ejmech.2012.03.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.ejmech.2021.113657 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.063 |
ug.mL-1 |
10.1016/j.bmc.2011.01.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.063 |
ug.mL-1 |
10.1016/j.bmc.2011.02.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.063 |
ug.mL-1 |
10.1021/np050554l |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.07 |
ug.mL-1 |
10.1016/j.bmc.2008.02.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.07 |
ug.mL-1 |
10.1021/jm201608g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.07 |
ug.mL-1 |
10.1021/np400391p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.074 |
ug.mL-1 |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.075 |
ug.mL-1 |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.078 |
ug.mL-1 |
10.1016/j.ejmech.2019.01.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.078 |
ug.mL-1 |
10.1039/C7MD00350A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.078 |
ug.mL-1 |
10.1039/C7MD00366H |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.08 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00972 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.08 |
ug.mL-1 |
10.1021/jm061288r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.09 |
ug.mL-1 |
10.1021/jm900672t |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.095 |
ug.mL-1 |
10.1016/j.bmcl.2018.07.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1007/s00044-013-0787-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmc.2016.01.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2005.08.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2007.10.083 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2009.04.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2011.05.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2015.07.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2019.06.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2010.09.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2019.112010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1021/acs.jnatprod.1c00812 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1021/acs.jnatprod.7b00300 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1021/acsmedchemlett.1c00431 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm060339h |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm060957y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1021/np400391p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.bmcl.2007.07.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.bmcl.2011.09.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.ejmech.2010.12.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.ejmech.2011.10.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.12 |
ug.mL-1 |
10.1021/jm020891g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.12 |
ug.mL-1 |
10.1021/np5001494 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1007/s00044-013-0781-3 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmc.2007.05.063 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmc.2008.10.086 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmc.2013.09.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.073 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2007.04.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2011.02.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2012.05.063 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2009.10.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2021.113472 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/s0960-894x(00)00188-8 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/s0960-894x(01)00266-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1021/jm049952w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1021/np049640w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1021/np980066w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00643-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.127 |
ug.mL-1 |
10.1016/j.bmc.2018.03.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.15 |
ug.mL-1 |
10.1016/j.ejmech.2011.04.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.15 |
ug.mL-1 |
10.1016/j.ejmech.2014.06.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.15 |
ug.mL-1 |
10.1021/np500538c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.15 |
ug.mL-1 |
10.1128/aac.00749-08 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.16 |
ug.mL-1 |
10.1021/np0002233 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.161 |
ug.mL-1 |
10.1021/acs.jnatprod.5b00770 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.195 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.195 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.197 |
ug.mL-1 |
10.1016/j.ejmech.2018.05.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1007/s00044-011-9948-y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2005.08.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2007.07.089 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2011.06.076 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2012.12.073 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2016.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2017.10.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2019.01.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.040 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2020.127434 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2011.06.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2013.10.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2017.07.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2018.07.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2020.112886 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1021/jm070638m |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1039/C7MD00350A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1039/C7MD00366H |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1128/aac.00643-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.23 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.24 |
nM |
10.1007/s00044-011-9662-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.24 |
nM |
10.1007/s00044-011-9705-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.24 |
ug.mL-1 |
10.1039/C6MD00085A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.24 |
ug.mL-1 |
10.1039/C6MD00593D |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-011-9950-4 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-012-0026-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-012-0041-y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-012-0073-3 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-013-0472-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-013-0839-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2007.03.086 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2010.08.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2010.09.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2016.10.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2005.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2007.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2009.06.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2010.07.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2012.03.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00360 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm0110284 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm701560p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1021/np010101q |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1021/np010216u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1021/np050424c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00643-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00661-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.29 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.3 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.3 |
ug.mL-1 |
10.1016/s0960-894x(99)00510-7 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.3 |
ug.mL-1 |
10.1021/jm0602662 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.37 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.39 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.39 |
ug.mL-1 |
10.1016/j.bmcl.2017.07.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.39 |
ug.mL-1 |
10.1016/j.ejmech.2017.06.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.39 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.090 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.39 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.39 |
ug.mL-1 |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2015.03.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2015.10.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2016.05.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2016.11.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.41 |
ug.mL-1 |
10.1016/j.ejmech.2017.01.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.42 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.48 |
ug.mL-1 |
10.1016/j.ejmech.2017.01.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
nM |
10.1016/j.ejmech.2019.111578 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1007/s00044-012-0451-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2015.11.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2019.04.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.073 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2005.11.087 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2009.12.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2023.129189 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2009.11.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2010.11.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.03.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.08.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2012.01.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1021/np020592u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1021/np0400095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1021/np0601399 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1021/np9700681 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.51 |
ug.mL-1 |
10.1016/j.ejmech.2017.01.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.51 |
ug.mL-1 |
10.1016/j.ejmech.2020.113102 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.6 |
ug.mL-1 |
10.1016/j.ejmech.2010.05.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.62 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.64 |
ug.mL-1 |
10.1021/acs.jnatprod.5b00975 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.65 |
ug.mL-1 |
10.1021/acsmedchemlett.1c00431 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.72 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.72 |
ug.mL-1 |
10.1016/j.bmcl.2019.06.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.75 |
ug.mL-1 |
10.1016/j.bmcl.2006.07.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.75 |
ug.mL-1 |
10.1016/j.ejmech.2017.01.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.75 |
ug.mL-1 |
10.1016/j.ejmech.2020.113102 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.75 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.bmcl.2012.01.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.78 |
ug.mL-1 |
10.1039/C8MD00056E |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.78 |
ug.mL-1 |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.8 |
ug.mL-1 |
10.1016/j.bmc.2010.09.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.8 |
ug.mL-1 |
10.1016/j.bmcl.2020.127655 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.84 |
ug.mL-1 |
10.1016/j.ejmech.2011.04.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.91 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
mg |
10.1016/j.bmc.2007.07.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
nM |
10.1016/j.bmcl.2019.04.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
nM |
10.1021/acs.jmedchem.1c00837 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1007/s00044-012-0074-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2007.08.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2009.04.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.07.073 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.09.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.01.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.08.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.06.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.03.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.07.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.09.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2015.10.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm00210a025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.2 |
ug.mL-1 |
10.1016/j.bmc.2011.11.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.2 |
ug.mL-1 |
10.1016/j.ejmech.2014.10.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.47 |
ug.mL-1 |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.47 |
ug.mL-1 |
10.1021/jm201608g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.6 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
nM |
10.1021/acs.jmedchem.1c00837 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1007/s00044-012-0268-7 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2011.01.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2013.09.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2019.04.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.11.107 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.05.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.02.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.12.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2010.06.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.03.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.10.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.10.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00202 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm000149l |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1021/np050554l |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1039/C9MD00057G |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.5 |
ug.mL-1 |
10.1016/j.bmc.2011.11.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.5 |
ug.mL-1 |
10.1016/j.ejmech.2014.10.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.5 |
ug.mL-1 |
10.1016/j.ejmech.2021.113266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.0 |
nM |
10.1021/acs.jmedchem.1c00837 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.0 |
nM |
10.1021/ml5001933 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.05.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.1 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.12 |
ug.mL-1 |
10.1021/jm060339h |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.13 |
ug.mL-1 |
10.1016/j.bmcl.2009.04.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.13 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.64 |
nM |
10.1021/acsmedchemlett.5b00176 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
nM |
10.1021/acs.jmedchem.1c00837 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
nM |
10.1021/jm5005978 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.01.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm201608g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1039/d2md00260d |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.2 |
ug.mL-1 |
10.1016/j.ejmech.2010.05.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
5.0 |
nM |
10.1021/acs.jmedchem.1c00837 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
5.0 |
nM |
10.1021/acsmedchemlett.9b00343 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
5.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.08.090 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.0 |
nM |
10.1016/j.bmcl.2011.06.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.0 |
nM |
10.1016/j.bmcl.2011.07.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.0 |
nM |
10.1021/acs.jnatprod.1c00232 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.25 |
nM |
10.1021/acs.jnatprod.0c00804 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.25 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.5 |
nM |
10.1021/acsmedchemlett.5b00176 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.5 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7.5 |
ug.mL-1 |
10.1007/s00044-013-0485-8 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
nM |
10.1021/ml5001728 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
nM |
10.1021/ml500531p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmc.2019.07.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2015.03.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.083 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1016/s0960-894x(01)00266-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00360 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
9.0 |
nM |
10.1021/acs.jmedchem.1c00707 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
9.24 |
ug.mL-1 |
10.1016/j.ejmech.2022.114145 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
nM |
10.1016/j.bmc.2010.07.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
nM |
10.1016/j.ejmech.2009.12.074 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
nM |
10.1021/acsmedchemlett.9b00343 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
nM |
10.1021/jm5005978 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112409 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113398 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113603 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114145 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00500 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
11.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
11.0 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.0 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
15.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
15.0 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
15.0 |
nM |
10.1021/jm401268f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
15.0 |
nM |
10.1021/ml5001728 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
15.0 |
nM |
10.1021/ml500531p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
15.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.12.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
nM |
10.1016/j.bmcl.2015.04.099 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmc.2011.02.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmc.2016.10.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116529 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.073 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.08.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00360 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00643-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00661-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
18.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
20.0 |
nM |
10.1016/j.bmc.2010.08.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
20.0 |
nM |
10.1016/j.ejmech.2018.02.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
20.0 |
nM |
10.1021/jm5002937 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
20.0 |
nM |
10.1021/jm5005978 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
20.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.09.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
22.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
22.0 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1007/s00044-012-0451-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.bmc.2019.04.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.08.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.01.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1021/acsmedchemlett.1c00431 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1021/jm070638m |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
27.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
30.0 |
nM |
10.1016/j.bmcl.2015.04.099 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
30.0 |
nM |
10.1021/acs.jnatprod.9b01095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
30.0 |
nM |
10.1021/jm401268f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
30.0 |
nM |
10.1021/jm5005978 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
30.0 |
ug.mL-1 |
10.1007/s00044-013-0485-8 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1007/s00044-011-9573-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116529 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.08.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.07.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.05.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.03.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.090 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.01.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
36.4 |
nM |
10.1021/acsmedchemlett.5b00176 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
36.89 |
ug.mL-1 |
10.1016/j.ejmech.2019.06.038 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
36.89 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00330 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
37.0 |
nM |
10.1016/j.bmc.2009.06.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
38.0 |
nM |
10.1016/j.bmcl.2013.11.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
38.65 |
ug.mL-1 |
10.1016/j.ejmech.2019.06.038 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
38.65 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00330 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1016/j.bmc.2010.08.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1016/j.bmcl.2012.12.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1016/j.bmcl.2016.02.076 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1021/acs.jnatprod.2c01003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1021/acsmedchemlett.5b00424 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1021/ml5003458 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1039/c5md00340g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1039/C6MD00231E |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1007/s00044-010-9399-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1007/s00044-011-9952-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1007/s00044-012-0060-8 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1007/s00044-012-0129-4 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1007/s00044-012-0322-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1007/s00044-013-0803-1 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.07.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.ejmech.2010.06.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.ejmech.2010.08.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.09.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.12.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.05.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.09.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.01.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
41.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45.7 |
ug.mL-1 |
10.1007/s00044-013-0485-8 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
49.0 |
nM |
10.1021/acsmedchemlett.7b00356 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
nM |
10.1016/j.bmcl.2009.12.062 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
nM |
10.1016/j.bmcl.2011.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
nM |
10.1016/j.bmcl.2016.02.076 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
nM |
10.1016/j.ejmech.2013.11.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
nM |
10.1021/acsmedchemlett.2c00254 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
nM |
10.1021/acsmedchemlett.5b00424 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
nM |
10.1021/jm900003c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
nM |
10.1021/ml5003458 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
nM |
10.1039/c5md00340g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.0 |
nM |
10.1016/j.bmcl.2013.11.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.0 |
nM |
10.1016/j.bmcl.2020.127074 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.0 |
nM |
10.1016/j.ejmech.2009.12.074 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.0 |
nM |
10.1016/j.ejmech.2013.11.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.0 |
nM |
10.1021/acs.jnatprod.0c00194 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.0 |
nM |
10.1021/jm401268f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.0 |
nM |
10.1021/jm900003c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.0 |
nM |
10.1021/jm901235p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.7 |
nM |
10.1039/C3MD00251A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2010.09.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2019.04.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2022.116777 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.03.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.01.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111678 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113580 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00360 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm701560p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1039/d1md00387a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1039/d2md00260d |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
70.0 |
nM |
10.1016/j.bmc.2007.05.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
70.0 |
nM |
10.1039/C3MD00366C |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
70.0 |
nM |
10.1039/C7MD00146K |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
80.0 |
nM |
10.1016/j.bmc.2013.11.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
80.0 |
nM |
10.1016/j.bmc.2014.10.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
80.0 |
nM |
10.1039/C7MD00146K |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
89.0 |
nM |
10.1016/j.bmcl.2013.11.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
90.0 |
nM |
10.1016/j.bmc.2011.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
90.0 |
nM |
10.1016/j.bmcl.2015.12.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
90.0 |
nM |
10.1016/j.bmcl.2015.12.083 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
90.0 |
nM |
10.1021/acs.jnatprod.2c01003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
90.0 |
nM |
10.1021/acs.jnatprod.6b00839 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1007/s00044-011-9770-6 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1007/s00044-013-0850-7 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.bmc.2009.08.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.bmc.2010.03.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.bmc.2012.08.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.bmcl.2009.10.107 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.bmcl.2009.11.105 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.bmcl.2010.10.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.bmcl.2011.03.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.bmcl.2011.12.119 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.ejmech.2011.07.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.ejmech.2011.07.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.ejmech.2011.09.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.ejmech.2013.11.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1021/jm900003c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1021/jm900340a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1021/jm901112f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1021/jm901273n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1021/np800751j |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.06.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
ug.mL-1 |
10.1021/np2000667 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
ug.mL-1 |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
110.0 |
nM |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
110.0 |
ug.mL-1 |
10.1016/j.bmc.2007.09.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
119.0 |
nM |
10.1007/s00044-012-0385-3 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.bmc.2011.04.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.bmc.2019.01.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.bmcl.2014.02.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.ejmech.2009.09.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.ejmech.2009.09.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.ejmech.2009.09.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.ejmech.2010.10.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.ejmech.2011.07.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.ejmech.2012.04.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.ejmech.2017.06.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.ejmech.2020.112035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.ejmech.2020.112402 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.01.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.07.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111678 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00202 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
140.0 |
nM |
10.1016/j.ejmech.2013.11.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
140.0 |
nM |
10.1021/np200022b |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
150.0 |
nM |
10.1016/j.bmc.2014.08.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
150.0 |
nM |
10.1016/j.bmc.2014.10.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
150.0 |
nM |
10.1016/j.bmc.2016.07.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
150.0 |
nM |
10.1016/j.bmc.2017.11.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
150.0 |
nM |
10.1016/j.ejmech.2014.09.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
150.0 |
nM |
10.1016/j.ejmech.2014.12.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
150.0 |
nM |
10.1021/jm020891g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
152.0 |
nM |
10.1016/j.bmcl.2009.07.147 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
160.0 |
nM |
10.1016/j.bmcl.2012.12.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
164.0 |
nM |
10.1016/j.ejmech.2019.06.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
190.0 |
nM |
10.1016/j.ejmech.2010.11.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
nM |
10.1016/j.bmcl.2009.11.105 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
nM |
10.1016/j.bmcl.2019.02.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
210.0 |
nM |
10.1016/j.bmcl.2013.11.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
210.0 |
nM |
10.1016/j.ejmech.2017.12.088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
210.0 |
nM |
10.1021/np900281r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
230.0 |
nM |
10.1007/s00044-011-9638-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
230.0 |
nM |
10.1016/j.bmc.2014.10.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
230.0 |
nM |
10.1016/j.bmc.2015.02.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
230.0 |
nM |
10.1016/j.bmc.2015.03.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
230.0 |
nM |
10.1016/j.bmc.2016.01.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
230.0 |
nM |
10.1016/j.bmc.2016.09.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
230.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
230.0 |
nM |
10.1016/j.bmcl.2020.127074 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
230.0 |
nM |
10.1016/j.ejmech.2015.06.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
230.0 |
nM |
10.1016/j.ejmech.2016.06.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
240.0 |
nM |
10.1016/j.bmc.2012.01.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
240.0 |
nM |
10.1016/j.bmc.2012.06.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
240.0 |
nM |
10.1016/j.bmc.2013.11.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
240.0 |
nM |
10.1016/j.bmcl.2007.01.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
240.0 |
nM |
10.1016/j.bmcl.2020.127037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
240.0 |
nM |
10.1016/j.ejmech.2016.03.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
240.0 |
nM |
10.1016/j.ejmech.2021.113266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
240.0 |
nM |
10.1021/np0580210 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
240.0 |
ug.mL-1 |
10.1128/aac.01486-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
243.0 |
nM |
10.1016/j.ejmech.2013.01.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
250.0 |
nM |
10.1016/j.bmc.2019.02.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
250.0 |
nM |
10.1016/j.ejmech.2010.02.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.128088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
256.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
256.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00202 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
280.0 |
ug.mL-1 |
10.1007/s00044-013-0487-6 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
290.0 |
nM |
10.1016/j.ejmech.2014.06.075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
300.0 |
nM |
10.1016/j.bmc.2014.10.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
300.0 |
nM |
10.1016/j.ejmech.2017.10.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
300.0 |
nM |
10.1016/j.ejmech.2020.112699 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
300.0 |
nM |
10.1021/acs.jnatprod.0c00151 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
300.0 |
nM |
10.1021/np000267b |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
350.0 |
nM |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
377.0 |
nM |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
480.0 |
nM |
10.1016/j.bmcl.2010.06.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
480.0 |
nM |
10.1016/j.bmcl.2012.10.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
490.0 |
nM |
10.1016/j.bmcl.2013.11.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.bmc.2017.03.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2010.02.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2010.04.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2020.112178 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1021/acs.jmedchem.6b00674 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1128/aac.00055-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
600.0 |
nM |
10.1021/acs.jnatprod.9b00475 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
610.0 |
nM |
10.1016/j.bmc.2014.10.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
610.0 |
nM |
10.1016/j.ejmech.2020.112898 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
610.0 |
nM |
10.1021/np0202226 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
640.0 |
nM |
10.1021/acsmedchemlett.7b00356 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
910.0 |
nM |
10.1016/j.ejmech.2018.04.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
940.0 |
nM |
10.1016/j.bmc.2007.05.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
950.0 |
nM |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
970.0 |
nM |
10.1016/j.bmc.2011.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
970.0 |
nM |
10.1016/j.ejmech.2018.04.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.bmc.2008.12.070 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2015.11.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1130.0 |
nM |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1210.0 |
nM |
10.1021/jm2003624 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1220.0 |
nM |
10.1016/j.ejmech.2018.01.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1400.0 |
nM |
10.1016/j.bmc.2015.03.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1410.0 |
nM |
10.1016/j.bmc.2008.12.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1500.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1800.0 |
nM |
10.1128/aac.00055-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1900.0 |
nM |
10.1016/j.bmc.2010.03.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1900.0 |
nM |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1900.0 |
nM |
10.1021/jm900003c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1900.0 |
nM |
10.1021/jm901273n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2000.0 |
nM |
10.1016/j.bmcl.2009.11.105 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2000.0 |
nM |
10.1016/j.bmcl.2013.08.101 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2000.0 |
nM |
10.1016/j.bmcl.2015.12.083 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2000.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2000.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2000.0 |
nM |
10.1021/jm900340a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2400.0 |
nM |
10.1016/j.bmcl.2009.12.062 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2400.0 |
nM |
10.1016/j.bmcl.2011.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2400.0 |
nM |
10.1016/j.ejmech.2020.112358 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2430.0 |
nM |
10.1016/j.bmcl.2009.07.147 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2430.0 |
nM |
10.1016/j.ejmech.2011.07.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2800.0 |
nM |
10.1016/j.bmc.2015.03.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3000.0 |
nM |
10.1016/j.bmc.2018.07.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3120.0 |
nM |
10.1016/j.bmcl.2011.06.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3120.0 |
nM |
10.1016/j.bmcl.2011.07.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3790.0 |
nM |
10.1007/s00044-011-9638-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3790.0 |
nM |
10.1016/j.bmc.2007.05.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3790.0 |
nM |
10.1016/j.ejmech.2009.09.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3800.0 |
nM |
10.1007/s00044-013-0850-7 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3800.0 |
nM |
10.1016/j.bmcl.2009.10.107 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3800.0 |
nM |
10.1016/j.ejmech.2009.09.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3800.0 |
nM |
10.1016/j.ejmech.2012.04.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3820.0 |
nM |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4000.0 |
nM |
10.1016/j.bmc.2010.08.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2013.11.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4800.0 |
nM |
10.1016/j.bmc.2012.08.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4800.0 |
nM |
10.1016/j.bmcl.2017.01.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
5000.0 |
nM |
10.1021/jm5002937 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6700.0 |
nM |
10.1016/j.ejmech.2015.03.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7200.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7200.0 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8000.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8000.0 |
nM |
10.1016/j.ejmech.2016.11.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12100.0 |
nM |
10.1016/j.ejmech.2018.04.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12200.0 |
nM |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12500.0 |
nM |
10.1021/ml5001933 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
15180.0 |
nM |
10.1016/j.bmcl.2010.06.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
15190.0 |
nM |
10.1016/j.ejmech.2010.10.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
15200.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16000.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
19000.0 |
nM |
10.1039/C7MD00146K |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
19400.0 |
nM |
10.1016/j.bmcl.2017.01.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
21000.0 |
nM |
10.1039/C6MD00278A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
24000.0 |
nM |
10.1039/C6MD00278A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25000.0 |
nM |
10.1016/j.ejmech.2010.04.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
30370.0 |
nM |
10.1016/j.bmc.2014.08.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
30370.0 |
nM |
10.1016/j.ejmech.2014.09.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
30400.0 |
nM |
10.1016/j.bmcl.2019.02.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32000.0 |
nM |
10.1021/jm900003c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32000.0 |
nM |
10.1021/jm901273n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40000.0 |
nM |
10.1016/j.bmc.2019.01.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40000.0 |
nM |
10.1016/j.ejmech.2019.06.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
48000.0 |
nM |
10.1016/j.ejmech.2016.02.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
48600.0 |
nM |
10.1021/acsmedchemlett.2c00254 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
48610.0 |
nM |
10.1016/j.ejmech.2020.112967 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50000.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50000.0 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50000.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64000.0 |
nM |
10.1039/C3MD00366C |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100000.0 |
nM |
10.1016/j.ejmech.2016.11.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
121510.0 |
nM |
10.1016/j.bmc.2007.05.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
151900.0 |
nM |
10.1016/j.ejmech.2018.02.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
250000.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.01.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
256000.0 |
nM |
10.1039/C3MD00366C |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
311000.0 |
nM |
10.1016/j.ejmech.2010.11.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
311080.0 |
nM |
10.1016/j.ejmech.2020.112898 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
ug.mL-1 |
10.1016/s0960-894x(00)00159-1 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1007/s00044-013-0472-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1016/j.bmc.2007.05.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1016/j.bmcl.2018.05.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1016/j.ejmech.2014.09.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1039/C3MD00366C |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1128/aac.01486-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC100 |
0.2 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC100 |
0.25 |
microg/ml |
10.1016/j.ejmech.2009.09.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC100 |
0.5 |
uM |
10.1021/acs.jnatprod.5b00266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.0019 |
ug.mL-1 |
10.1016/j.bmcl.2017.01.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.0043 |
ug.mL-1 |
10.1016/j.bmcl.2017.01.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.035 |
ug.mL-1 |
10.1016/j.bmcl.2022.128824 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.035 |
ug.mL-1 |
10.1016/j.bmcl.2022.128871 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.1 |
ug.mL-1 |
10.1021/jm030479g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.5 |
ug.mL-1 |
10.1007/s00044-010-9322-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2021.116560 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.5 |
ug.mL-1 |
10.1021/jm100165w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.7 |
ug.mL-1 |
10.1016/j.bmcl.2020.127351 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.7 |
ug.mL-1 |
10.1016/j.bmcl.2021.128261 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.8 |
ug.mL-1 |
10.1016/j.bmcl.2020.127351 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.8 |
ug.mL-1 |
10.1016/j.bmcl.2021.128261 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm100568q |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
4.21 |
ug.mL-1 |
10.1007/s00044-010-9322-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
21.0 |
nM |
10.1021/acs.jmedchem.2c00266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
40.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128824 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
40.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128871 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
128.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
200.0 |
nM |
10.1016/j.bmc.2021.116506 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
240.0 |
nM |
10.1021/acs.jmedchem.2c00266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC70 |
0.08 |
uM |
10.1016/j.bmcl.2017.07.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
0.003 |
ug ml-1 |
10.1021/jm500833f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
0.004 |
uM |
10.1021/acs.jmedchem.6b01358 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
0.007 |
ug ml-1 |
10.1021/jm500833f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
0.008 |
uM |
10.1021/acs.jmedchem.6b01358 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
0.016 |
uM |
10.1021/acs.jmedchem.6b01358 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
0.04 |
uM |
10.1039/C5MD00589B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
1.2 |
uM |
10.1039/C5MD00589B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
16.0 |
ug ml-1 |
10.1021/jm500833f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC80 |
26.6 |
nM |
10.1021/jm5003606 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC80 |
180.0 |
nM |
10.1021/jm5003606 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=<90 |
0.0625 |
ug ml-1 |
10.1016/j.ejmech.2021.113202 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=<90 |
0.125 |
ug ml-1 |
10.1021/acs.jmedchem.7b00582 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=<90 |
4.0 |
ug ml-1 |
10.1016/j.ejmech.2021.113202 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=<90 |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2021.113202 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.003 |
ug ml-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.008 |
ug ml-1 |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.05 |
ug ml-1 |
10.1016/j.bmcl.2015.10.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.05 |
ug ml-1 |
10.1016/j.ejmech.2015.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.05 |
uM |
10.1016/j.ejmech.2015.05.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.057 |
ug ml-1 |
10.1021/acsmedchemlett.7b00068 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.06 |
ug ml-1 |
10.1016/j.ejmech.2020.112420 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.06 |
uM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.071 |
uM |
10.1016/j.ejmech.2017.05.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.078 |
ug ml-1 |
10.1016/j.ejmech.2019.111595 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.084 |
ug ml-1 |
10.1016/j.ejmech.2018.03.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.096 |
ug ml-1 |
10.1016/j.ejmech.2018.09.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.11 |
uM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.13 |
uM |
10.1016/j.ejmech.2015.10.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.152 |
uM |
10.1016/j.ejmech.2019.01.073 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.5 |
mg/L |
10.1016/j.bmcl.2015.09.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
2.0 |
ug ml-1 |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
10.0 |
uM |
10.1016/j.bmc.2015.03.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
20.0 |
ug ml-1 |
10.1021/acsmedchemlett.7b00068 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
40.0 |
ug ml-1 |
10.1016/j.bmcl.2015.10.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
40.0 |
ug ml-1 |
10.1016/j.ejmech.2015.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
40.0 |
ug ml-1 |
10.1016/j.ejmech.2018.03.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
40.0 |
ug ml-1 |
10.1016/j.ejmech.2018.09.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
40.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111595 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
40.0 |
ug ml-1 |
10.1021/acsmedchemlett.7b00068 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
57.0 |
uM |
10.1016/j.ejmech.2017.05.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2020.112420 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
128.0 |
uM |
10.1016/j.ejmech.2019.01.073 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
256.0 |
mg/L |
10.1016/j.bmcl.2015.09.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.01 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.02 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.03 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.038 |
uM |
10.1016/j.ejmech.2018.12.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.04 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.05 |
ug ml-1 |
10.1021/acs.jnatprod.8b00567 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.05 |
ug ml-1 |
10.1021/acsmedchemlett.6b00330 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.059 |
ug ml-1 |
10.1016/j.bmcl.2018.07.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.0781 |
ug ml-1 |
10.1021/acsmedchemlett.8b00177 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.092 |
uM |
10.1021/acsmedchemlett.7b00106 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.1 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.2 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
3.3 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
10.0 |
uM |
10.1016/j.bmc.2015.06.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
27.24 |
uM |
10.1021/acsmedchemlett.7b00106 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
40.0 |
ug ml-1 |
10.1016/j.bmcl.2018.07.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
40.0 |
ug ml-1 |
10.1021/acsmedchemlett.8b00177 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
40.0 |
uM |
10.1016/j.ejmech.2018.12.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
48.6 |
uM |
10.1021/acsmedchemlett.7b00106 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.003 |
ug.mL-1 |
10.1021/jm300123s |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.004 |
ug.mL-1 |
10.1021/acsmedchemlett.0c00381 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.005 |
ug.mL-1 |
10.1021/acs.jmedchem.1c01349 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.0173 |
ug.mL-1 |
10.1016/j.bmcl.2017.01.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.02 |
ug.mL-1 |
10.1016/j.bmcl.2017.01.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.02 |
ug.mL-1 |
10.1021/np400497f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.02 |
ug.mL-1 |
10.1038/nchembio884 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.1c01349 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.04 |
ug.mL-1 |
10.1021/np400497f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.041 |
ug.mL-1 |
10.1021/jm300123s |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.043 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.048 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2012.05.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2022.114404 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.05 |
ug.mL-1 |
10.1021/np400497f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.057 |
ug.mL-1 |
10.1016/j.bmcl.2022.128824 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.06 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00202 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.0625 |
ug.mL-1 |
10.1016/j.bmcl.2012.09.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.064 |
ug.mL-1 |
10.1016/j.bmcl.2022.128871 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.08 |
ug.mL-1 |
10.1021/np400497f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.09 |
ug.mL-1 |
10.1021/np400497f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.125 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01064 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.13 |
ug.mL-1 |
10.1038/nchembio884 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2022.114404 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.25 |
ug.mL-1 |
10.1039/C8MD00389K |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.3 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.39 |
ug.mL-1 |
10.1016/j.ejmech.2017.05.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.39 |
ug.mL-1 |
10.1016/j.ejmech.2018.07.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2016.03.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.064 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.5 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.5 |
ug.mL-1 |
10.1021/jm0703901 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.5 |
ug.mL-1 |
10.1021/jm070391t |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.51 |
ug.mL-1 |
10.1039/C5MD00404G |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.7 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.064 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.75 |
ug.mL-1 |
10.1039/C5MD00404G |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.8 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.064 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.8 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2016.03.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1.47 |
ug.mL-1 |
10.1016/j.bmcl.2012.05.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1.5 |
nM |
10.1016/j.bmcl.2019.05.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1.6 |
nM |
10.1021/acs.jmedchem.5b01542 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
2.0 |
ug.mL-1 |
10.1007/s00044-010-9322-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm300123s |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
2.91 |
nM |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
2.95 |
ug.mL-1 |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
3.2 |
nM |
10.1021/acs.jmedchem.5b01542 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
3.29 |
ug.mL-1 |
10.1021/np400497f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.064 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
4.5 |
nM |
10.1016/j.ejmech.2021.113734 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
6.0 |
nM |
10.1039/d1md00063b |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
7.0 |
nM |
10.1016/j.bmcl.2019.126911 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
7.37 |
ug.mL-1 |
10.1007/s00044-010-9322-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
8.0 |
nM |
10.1016/j.bmcl.2008.03.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
9.0 |
nM |
10.1021/acs.jmedchem.5b01542 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
9.0 |
nM |
10.1039/C9MD00161A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
10.0 |
nM |
10.1016/j.bmcl.2021.127784 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
10.0 |
nM |
10.1016/j.ejmech.2021.113207 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
10.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
10.0 |
nM |
10.1021/ml200036r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
10.0 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
13.0 |
nM |
10.1016/j.ejmech.2022.114105 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
15.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
15.6 |
nM |
10.1016/j.ejmech.2019.06.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
18.0 |
nM |
10.1016/j.ejmech.2019.06.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
19.0 |
nM |
10.1016/j.bmcl.2019.126911 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
20.0 |
nM |
10.1016/j.bmc.2016.12.038 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
20.0 |
nM |
10.1016/j.ejmech.2021.113734 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
20.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
20.0 |
nM |
10.1021/ml200036r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
20.0 |
nM |
10.1039/C9MD00161A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
21.7 |
nM |
10.1016/j.ejmech.2019.06.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
23.0 |
nM |
10.1016/j.ejmech.2022.114105 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
25.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
25.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114404 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
28.0 |
nM |
10.1021/acs.jnatprod.1c00198 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
30.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.05.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.07.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
40.0 |
nM |
10.1016/j.bmc.2012.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
40.0 |
nM |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
40.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
40.0 |
ug.mL-1 |
10.1007/s00044-011-9718-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
40.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128824 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
40.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128871 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
50.0 |
nM |
10.1016/j.ejmech.2012.08.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
50.0 |
nM |
10.1016/j.ejmech.2017.05.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
50.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
50.0 |
nM |
10.1021/ml200036r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
60.0 |
nM |
10.1007/s00044-012-9971-7 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
60.0 |
nM |
10.1016/j.bmcl.2019.02.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
60.0 |
nM |
10.1039/C8MD00480C |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
70.0 |
nM |
10.1016/j.bmcl.2013.09.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
70.0 |
nM |
10.1016/j.ejmech.2015.05.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
70.0 |
nM |
10.1021/acsmedchemlett.5b00141 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
70.0 |
nM |
10.1021/ml200036r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
90.0 |
nM |
10.1007/s00044-007-9073-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
90.0 |
nM |
10.1016/j.bmc.2012.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
90.0 |
nM |
10.1016/j.bmcl.2012.06.095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
100.0 |
nM |
10.1016/j.ejmech.2017.06.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
100.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
100.0 |
nM |
10.1021/acs.jnatprod.5b00266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
100.0 |
nM |
10.1021/jm900513a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
120.0 |
nM |
10.1016/j.ejmech.2013.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
128.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
128.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
130.0 |
nM |
10.1016/j.bmcl.2011.08.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
130.0 |
nM |
10.1021/jm201716n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
150.0 |
nM |
10.1021/np900806j |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
190.0 |
nM |
10.1016/j.ejmech.2017.05.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
200.0 |
nM |
10.1016/j.bmc.2012.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
200.0 |
nM |
10.1021/ml200036r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
210.0 |
nM |
10.1016/j.ejmech.2015.05.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
210.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
300.0 |
nM |
10.1039/d2md00155a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
460.0 |
nM |
10.1021/jm201716n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
500.0 |
nM |
10.1016/j.ejmech.2016.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
610.0 |
nM |
10.1016/j.bmcl.2012.06.095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
610.0 |
nM |
10.1021/acs.jnatprod.5b01033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
760.0 |
nM |
10.1016/j.ejmech.2020.112821 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
780.0 |
nM |
10.1021/ml200036r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
800.0 |
nM |
10.1021/ml200036r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
910.0 |
nM |
10.1016/j.bmcl.2019.03.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
910.0 |
nM |
10.1016/j.ejmech.2017.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
980.0 |
nM |
10.1016/j.ejmech.2017.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1000.0 |
nM |
10.1016/j.ejmech.2017.05.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1000.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1000.0 |
nM |
10.1021/ml200036r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1900.0 |
nM |
10.1016/j.bmcl.2011.08.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1900.0 |
nM |
10.1021/jm900513a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1930.0 |
nM |
10.1016/j.ejmech.2012.08.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
2400.0 |
nM |
10.1021/acsmedchemlett.5b00141 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
2600.0 |
nM |
10.1016/j.bmc.2012.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
2600.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
2600.0 |
nM |
10.1021/ml200036r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
8000.0 |
nM |
10.1016/j.ejmech.2021.113734 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
38900.0 |
nM |
10.1016/j.ejmech.2015.05.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
155500.0 |
nM |
10.1021/acsmedchemlett.5b00141 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
311070.0 |
nM |
10.1021/acsmedchemlett.5b00141 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
311100.0 |
nM |
10.1016/j.ejmech.2015.05.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
nan |
None |
10.1016/j.ejmech.2016.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
nan |
None |
10.1021/acs.jmedchem.5b01542 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
nan |
None |
10.1021/acs.jnatprod.5b01033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC95 |
0.03 |
ug ml-1 |
10.1016/j.bmc.2017.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC95 |
0.25 |
ug ml-1 |
10.1016/j.bmcl.2011.06.074 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC97 |
0.015 |
ug ml-1 |
10.1016/j.bmcl.2011.06.074 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC98 |
40.0 |
ug ml-1 |
10.1016/j.ejmech.2017.06.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC98 |
40.0 |
ug ml-1 |
10.1016/j.ejmech.2018.03.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
0.012 |
uM |
10.1016/j.bmc.2015.10.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
0.25 |
uM |
10.1016/j.bmc.2017.08.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
0.25 |
uM |
10.1016/j.ejmech.2017.02.058 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
0.25 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
8.0 |
uM |
10.1016/j.bmc.2017.08.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
8.0 |
uM |
10.1021/acs.jmedchem.5b00608 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
8.0 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.00167 |
uM |
10.1016/j.bmcl.2019.05.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.003 |
uM |
10.1021/ml400088y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.004 |
uM |
10.1016/j.bmc.2014.10.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.00482 |
uM |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.005 |
uM |
10.1016/j.bmc.2020.115530 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.007 |
uM |
10.1016/j.ejmech.2020.112772 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.0083 |
uM |
10.1016/j.bmcl.2014.05.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.012 |
uM |
10.1021/acs.jmedchem.7b01347 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.013 |
uM |
10.1016/j.bmc.2014.10.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.02 |
ug ml-1 |
10.1016/j.bmcl.2013.10.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.02 |
ug ml-1 |
10.1016/j.ejmech.2014.01.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.037 |
uM |
10.1021/acs.jmedchem.2c00266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.041 |
uM |
10.1021/acs.jmedchem.2c00266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.125 |
ug ml-1 |
10.1016/j.bmc.2013.06.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.14 |
uM |
10.1016/j.ejmech.2013.10.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.19 |
uM |
10.1021/jm401735w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.197 |
ug ml-1 |
10.1016/j.bmcl.2016.04.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.197 |
ug ml-1 |
10.1016/j.bmcl.2016.10.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.197 |
ug ml-1 |
10.1039/C4MD00224E |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.2 |
ug ml-1 |
10.1016/j.ejmech.2014.07.100 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.2 |
ug ml-1 |
10.1016/j.ejmech.2015.01.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.2 |
ug ml-1 |
10.1016/j.ejmech.2015.02.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.25 |
ug ml-1 |
10.1016/j.ejmech.2014.03.085 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.25 |
ug ml-1 |
10.1016/j.ejmech.2019.07.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.5 |
uM |
10.1016/j.bmcl.2017.02.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
1.0 |
ug ml-1 |
10.1016/j.bmc.2012.09.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
1.0 |
ug ml-1 |
10.1016/j.bmc.2013.07.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
40.0 |
ug ml-1 |
10.1007/s00044-011-9942-4 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
40.0 |
ug ml-1 |
10.1007/s00044-012-0273-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
nan |
None |
10.1016/j.bmc.2013.07.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
PAE |
5.2 |
day |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
PAE |
12.0 |
day |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
PAE |
12.9 |
day |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
PAE |
19.3 |
day |
10.1128/aac.01533-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
0.5 |
None |
10.1021/jm500833f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
1.0 |
None |
10.1016/j.bmcl.2008.03.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
4.0 |
None |
10.1128/aac.00550-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
15.6 |
None |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
65.0 |
None |
10.1016/j.bmcl.2009.07.147 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
650.0 |
None |
10.1016/j.bmcl.2009.07.147 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
nan |
None |
10.1016/j.ejmech.2018.02.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Selectivity Index |
0.2 |
None |
10.1021/acs.jmedchem.1c01349 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Selectivity ratio |
4.0 |
None |
10.1021/acs.jmedchem.6b01358 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Selectivity ratio |
7.35 |
None |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis H37Rv |
Mycobacterium tuberculosis H37Rv |
MIC50 |
1.53 |
nM |
10.1021/acs.jmedchem.1c01407 |
| Mycobacterium tuberculosis H37Rv |
Mycobacterium tuberculosis H37Rv |
MIC50 |
10.0 |
nM |
10.1016/j.ejmech.2020.112908 |
| Mycobacterium tuberculosis H37Rv |
Mycobacterium tuberculosis H37Rv |
MIC50 |
2900.0 |
nM |
10.1016/j.ejmech.2020.112908 |
| Mycobacterium tuberculosis H37Rv |
Mycobacterium tuberculosis H37Rv |
MIC90 |
8000.0 |
nM |
10.1016/j.ejmech.2021.113734 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
Cytochrome bc1 complex cytochrome b subunit |
Inhibition |
nan |
% |
10.1021/acs.jmedchem.8b00172 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
50000.0 |
nM |
10.1016/j.bmc.2016.01.011 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.bmc.2014.10.016 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.bmc.2015.03.004 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.ejmech.2015.06.032 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.ejmech.2016.08.034 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
nan |
None |
10.1021/ml500531p |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
FAD-dependent decaprenylphosphoryl-beta-D-ribofuranose 2-oxidase |
MIC |
0.015 |
ug.mL-1 |
10.1021/acs.jmedchem.1c00263 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
Polyketide synthase Pks13 |
MIC=<90 |
0.0625 |
ug ml-1 |
10.1021/acs.jmedchem.9b00010 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
Polyketide synthase Pks13 |
MIC=<90 |
0.125 |
ug ml-1 |
10.1021/acs.jmedchem.9b00010 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
Polyketide synthase Pks13 |
MIC=<90 |
4.0 |
ug ml-1 |
10.1021/acs.jmedchem.9b00010 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
Polyketide synthase Pks13 |
MIC=<90 |
128.0 |
ug ml-1 |
10.1021/acs.jmedchem.9b00010 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
Activity |
3.0 |
log10CFU/ml |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
Activity |
nan |
None |
10.1016/j.ejmech.2016.07.068 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
IC50 |
10.0 |
nM |
None |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
IC50 |
910.0 |
nM |
10.1016/j.bmcl.2019.03.020 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
Inhibition |
100.0 |
% |
10.1016/j.ejmech.2022.114831 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
Inhibition |
100.0 |
% |
10.1021/jm058167w |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.01302-08 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.031 |
ug.mL-1 |
10.1128/aac.01302-08 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.063 |
ug.mL-1 |
10.1128/aac.01302-08 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.45 |
ug.mL-1 |
10.1016/j.ejmech.2020.113102 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.81 |
ug.mL-1 |
10.1016/j.ejmech.2020.113102 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
350.0 |
nM |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
nan |
None |
10.1016/j.bmcl.2019.06.055 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm058167w |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC90 |
20.0 |
nM |
10.1016/j.ejmech.2016.07.068 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC90 |
980.0 |
nM |
10.1016/j.bmcl.2019.03.020 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC90 |
2200.0 |
nM |
10.1016/j.bmcl.2019.126671 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC>99 |
0.25 |
ug ml-1 |
10.1016/j.ejmech.2014.07.066 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
Activity |
25.0 |
% |
10.1021/acs.jmedchem.8b00832 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
IC50 |
0.0012 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
IC50 |
0.0015 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
IC50 |
0.0016 |
ug.mL-1 |
10.1016/j.bmcl.2015.11.071 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
IC50 |
0.0027 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.093 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
IC50 |
0.003 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.093 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.0002 |
ug.mL-1 |
10.1128/aac.00550-09 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.0004 |
ug.mL-1 |
10.1128/aac.00550-09 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.0008 |
ug.mL-1 |
10.1128/aac.00550-09 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.0016 |
ug.mL-1 |
10.1128/aac.00550-09 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.0032 |
ug.mL-1 |
10.1128/aac.00550-09 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.017 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.041 |
ug.mL-1 |
10.1016/j.bmcl.2015.11.071 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.093 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.08 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.093 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm070638m |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
4.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
20.0 |
nM |
10.1021/ml5003458 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
60.7 |
nM |
10.1039/C3MD00251A |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC90 |
0.004 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC90 |
0.0042 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis variant microti |
Mycobacterium tuberculosis variant microti |
MIC |
30380.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
Activity |
nan |
None |
10.1128/aac.00730-07 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
log10cfu |
0.46 |
None |
10.1128/aac.00730-07 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
log10cfu |
1.52 |
None |
10.1128/aac.00730-07 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
Log10 cfu |
4.13 |
None |
10.1128/aac.00821-06 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00400-10 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00400-10 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00400-10 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
MIC |
0.13 |
ug.mL-1 |
10.1128/aac.00400-10 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00400-10 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00730-07 |
| Mycobacterium xenopi |
Mycobacterium xenopi |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
DIZ |
nan |
None |
10.1016/j.bmcl.2019.07.001 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
IZ |
0.0 |
mm |
10.1016/j.bmcl.2019.07.001 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
4000.0 |
nM |
10.1021/acs.jnatprod.9b01095 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
162000.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
nan |
None |
10.1016/j.bmc.2022.116777 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
nan |
None |
10.1016/j.ejmech.2020.112996 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC50 |
128.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC90 |
128.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC90 |
162300.0 |
nM |
10.1021/ml200036r |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
5.0 |
ug.mL-1 |
10.1128/aac.00590-09 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
25.0 |
ug.mL-1 |
10.1128/aac.00590-09 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2013.10.011 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.001 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
100.0 |
ug.mL-1 |
10.1128/aac.00590-09 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
500.0 |
ug.mL-1 |
10.1128/aac.00590-09 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
100000.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
nan |
None |
10.1016/j.bmc.2022.116777 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
nan |
None |
10.1016/j.ejmech.2020.112996 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC50 |
128.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC90 |
128.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC90 |
150000.0 |
nM |
10.1021/ml200036r |
| Mycolicibacterium aurum |
Mycolicibacterium aurum |
MIC |
0.78 |
ug.mL-1 |
10.1021/jm070638m |
| Mycolicibacterium aurum |
Mycolicibacterium aurum |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jnatprod.9b01015 |
| Mycolicibacterium aurum |
Mycolicibacterium aurum |
MIC |
470.0 |
nM |
10.1016/j.ejmech.2019.111578 |
| Mycolicibacterium diernhoferi |
Mycolicibacterium diernhoferi |
MIC |
4.0 |
ug.mL-1 |
10.1021/np2006555 |
| Mycolicibacterium flavescens |
Mycolicibacterium flavescens |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycolicibacterium flavescens |
Mycolicibacterium flavescens |
MIC |
128.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
0.25 |
ug.mL-1 |
10.1016/s0960-894x(01)00283-9 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.5 |
ug.mL-1 |
10.1007/s00044-012-0451-x |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.bmcl.2009.12.045 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.072 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.03.039 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.033 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.049 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.08.014 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2012.01.008 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.11.002 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
25.0 |
ug.mL-1 |
10.1021/jm070638m |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2013.10.011 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.001 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
128.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1890.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
nan |
None |
10.1016/j.bmc.2022.116777 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
nan |
None |
10.1016/j.ejmech.2020.112996 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC50 |
32.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.01545-09 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
DIZ |
nan |
None |
10.1007/s00044-013-0487-6 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
IZ |
25.0 |
mm |
10.1016/j.bmc.2007.09.025 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
log(1/C) |
6.48 |
None |
10.1021/jm00210a025 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MBC |
0.06 |
ug ml-1 |
10.1021/acs.jnatprod.2c00065 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00065 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
0.032 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
0.27 |
ug.mL-1 |
10.1021/jm00210a025 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
40.0 |
ug.mL-1 |
10.1007/s00044-013-0487-6 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
30380.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Activity |
32.4 |
% |
10.1016/j.ejmech.2016.07.068 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Activity |
66.5 |
% |
10.1016/j.ejmech.2016.07.068 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Activity |
95.6 |
% |
10.1016/j.ejmech.2016.07.068 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Activity |
123.4 |
% |
10.1016/j.ejmech.2016.07.068 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Activity |
nan |
None |
10.1016/j.ejmech.2016.07.068 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Activity |
nan |
None |
10.1016/j.ejmech.2019.05.081 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
DIZ |
nan |
None |
10.1007/s00044-013-0487-6 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
FICI |
0.5 |
None |
10.1016/j.bmc.2014.06.012 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
FICI |
0.63 |
None |
10.1016/j.bmc.2014.06.012 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
FICI |
1.0 |
None |
10.1016/j.bmc.2014.06.012 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
GI50 |
1.04 |
ug.mL-1 |
10.1016/j.ejmech.2014.02.042 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
GI50 |
1220.0 |
nM |
10.1016/j.ejmech.2014.06.075 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
IC50 |
1870.0 |
nM |
10.1016/j.bmcl.2015.02.052 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
IC50 |
3110.0 |
nM |
10.1128/aac.00803-09 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
IC50 |
4360.0 |
nM |
10.1128/aac.00803-09 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
IC90 |
0.2 |
ug.mL-1 |
10.1021/np400002p |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
IZ |
30.0 |
mm |
10.1016/j.bmc.2007.09.025 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MBC |
8.0 |
ug ml-1 |
10.1021/acs.jnatprod.2c00065 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MBC |
130.0 |
ug ml-1 |
10.1016/j.bmc.2007.09.025 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
0.1 |
ug.mL-1 |
10.1021/acs.jnatprod.1c00812 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2006.10.016 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
0.5 |
ug.mL-1 |
10.1039/d2md00260d |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
0.5 |
ug.mL-1 |
10.1126/science.1106753 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
0.78 |
ug.mL-1 |
10.1039/C8MD00056E |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.08.066 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.5 |
ug.mL-1 |
10.1007/s00044-012-0451-x |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.bmcl.2009.12.045 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.072 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.03.039 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.033 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.049 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.08.014 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2012.01.008 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.11.002 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.75 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.058 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
2.15 |
ug.mL-1 |
10.1016/j.bmcl.2015.05.044 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00972 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1021/np2006555 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00012-09 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2010.11.020 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00065 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.111578 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.05.049 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
25.0 |
ug.mL-1 |
10.1021/jm070638m |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2012.02.039 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.10.016 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.001 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
32.0 |
ug.mL-1 |
10.1016/s0960-894x(99)00510-7 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm0602662 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm701560p |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00012-09 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
55.0 |
ug.mL-1 |
10.1016/j.ejmech.2010.05.017 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2010.05.016 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2013.10.011 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
100.0 |
ug.mL-1 |
10.1039/C7MD00350A |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
140.0 |
ug.mL-1 |
10.1016/j.bmc.2007.09.025 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
350.0 |
nM |
10.1016/j.ejmech.2021.113932 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
480.0 |
ug.mL-1 |
10.1007/s00044-013-0487-6 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1890.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
3790.0 |
nM |
10.1016/j.ejmech.2010.11.023 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
5000.0 |
nM |
10.1016/j.ejmech.2021.113212 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
6250.0 |
nM |
10.1128/aac.00803-09 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
10000.0 |
nM |
10.1016/j.ejmech.2021.113212 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
16700.0 |
nM |
10.1016/j.bmcl.2013.11.024 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
22600.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
100000.0 |
ug.mL-1 |
10.1039/C7MD00366H |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
nan |
ug.mL-1 |
10.1016/s0960-894x(03)00597-3 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
nan |
None |
10.1016/j.ejmech.2009.09.001 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
nan |
None |
10.1128/aac.00012-09 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC100 |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC50 |
0.57 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC50 |
0.63 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC50 |
0.76 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC50 |
2.08 |
ug.mL-1 |
10.1016/j.ejmech.2013.10.034 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC>90 |
0.3 |
ug ml-1 |
10.1021/np400145u |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
0.76 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
2.15 |
ug.mL-1 |
10.1016/j.ejmech.2013.10.034 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
2.4 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
2.83 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c01349 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
8.2 |
ug.mL-1 |
10.1038/nchembio884 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
2500.0 |
nM |
10.1016/j.ejmech.2016.07.068 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
10000.0 |
nM |
10.1016/j.ejmech.2017.05.026 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
162300.0 |
nM |
10.1021/ml200036r |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC99 |
0.2 |
uM |
10.1016/j.bmc.2014.06.012 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC99 |
0.32 |
uM |
10.1016/j.bmc.2014.06.012 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC99 |
0.63 |
uM |
10.1016/j.bmc.2014.06.012 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC99 |
1.26 |
uM |
10.1039/C3MD00387F |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC99 |
2.53 |
uM |
10.1016/j.bmc.2014.06.012 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Ratio |
0.126 |
None |
10.1016/j.bmc.2014.06.012 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Ratio |
0.254 |
None |
10.1016/j.bmc.2014.06.012 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Ratio |
0.5 |
None |
10.1016/j.bmc.2014.06.012 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Ratio |
64.0 |
None |
10.1016/j.bmcl.2006.10.016 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Selectivity Index |
1.0 |
None |
10.1021/acs.jmedchem.1c01349 |
| Mycolicibacterium vaccae |
Mycolicibacterium vaccae |
MIC |
3800.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Neisseria gonorrhoeae |
Neisseria gonorrhoeae |
MIC |
0.125 |
ug.mL-1 |
10.1021/jm00167a029 |
| Neisseria meningitidis |
Neisseria meningitidis |
Activity |
0.0 |
% |
10.1128/aac.00994-08 |
| Neisseria meningitidis |
Neisseria meningitidis |
Activity |
0.0 |
% |
10.1128/aac.01812-09 |
| Neisseria meningitidis |
Neisseria meningitidis |
Activity |
1.0 |
% |
10.1128/aac.00994-08 |
| Neisseria meningitidis |
Neisseria meningitidis |
Activity |
99.0 |
% |
10.1128/aac.00994-08 |
| Neisseria meningitidis |
Neisseria meningitidis |
Activity |
100.0 |
% |
10.1128/aac.01812-09 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
1.5e-05 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
2.4e-05 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
2.5e-05 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
2.9e-05 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
3.4e-05 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
5.7e-05 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
6.1e-05 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
6.5e-05 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
8.9e-05 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
0.000125 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
0.00015 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
0.000225 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
0.002 |
ug.mL-1 |
10.1128/aac.00994-08 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.01812-09 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
0.032 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
0.256 |
ug.mL-1 |
10.1128/aac.00315-10 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC50 |
0.015 |
ug.mL-1 |
10.1128/aac.01812-09 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC50 |
0.064 |
ug.mL-1 |
10.1128/aac.00994-08 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC90 |
0.03 |
ug.mL-1 |
10.1128/aac.01812-09 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC90 |
0.125 |
ug.mL-1 |
10.1128/aac.00994-08 |
| Oryctolagus cuniculus |
Angiotensin-converting enzyme |
IC50 |
nan |
None |
None |
| Oryctolagus cuniculus |
Angiotensin-converting enzyme |
Ki |
nan |
None |
None |
| Oryctolagus cuniculus |
Arachidonate 15-lipoxygenase |
IC50 |
2949.0 |
nM |
None |
| Oryctolagus cuniculus |
Arachidonate 15-lipoxygenase |
Ki |
nan |
None |
None |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Activity |
8.2 |
% |
10.1128/aac.00367-09 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Activity |
411.7 |
/uL |
10.1128/aac.00367-09 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Activity |
nan |
None |
10.1128/aac.00367-09 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
AUC |
40280.0 |
ng.hr.mL-1 |
10.1128/aac.00367-09 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Cmax |
20195.64 |
nM |
10.1128/aac.00367-09 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
T1/2 |
3.38 |
hr |
10.1128/aac.00367-09 |
| Papio hamadryas |
Plasma |
PPB |
27.32 |
% |
10.1021/jm901858n |
| Pasteurella multocida |
Pasteurella multocida |
MIC |
0.1 |
ug.mL-1 |
10.1128/aac.00245-08 |
| Pasteurella multocida |
Pasteurella multocida |
MIC |
0.2 |
ug.mL-1 |
10.1128/aac.00245-08 |
| Pasteurella multocida |
Pasteurella multocida |
MIC |
0.78 |
ug.mL-1 |
10.1128/aac.00245-08 |
| Pasteurella multocida |
Pasteurella multocida |
MIC |
50.0 |
ug.mL-1 |
10.1128/aac.00245-08 |
| Pasteurella multocida |
Pasteurella multocida |
Ratio |
64.0 |
None |
10.1128/aac.00245-08 |
| Pasteurella multocida |
Pasteurella multocida |
Ratio |
512.0 |
None |
10.1128/aac.00245-08 |
| Peptococcus niger |
Peptococcus niger |
MIC |
0.004 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC |
0.004 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC |
0.004 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Peptostreptococcus sp. |
Peptostreptococcus sp. |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
10.0 |
% |
10.1128/aac.00808-06 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
13.0 |
% |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
14.0 |
% |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
15.0 |
% |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
16.0 |
% |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
25.0 |
% |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
36.0 |
% |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
49.0 |
% |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
65.0 |
% |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
93.0 |
% |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
nan |
None |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
nan |
None |
10.1128/aac.00808-06 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
190.0 |
nM |
10.1128/aac.00808-06 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
274.0 |
nM |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
528.0 |
nM |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
1000.0 |
nM |
10.1016/j.bmc.2010.01.068 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
2830.0 |
nM |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
2990.0 |
nM |
10.1128/aac.00527-07 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
4200.0 |
nM |
10.1128/aac.00808-06 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
nan |
None |
10.1021/np020592u |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
nan |
None |
10.1021/np0400095 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
nan |
None |
10.1021/np0601399 |
| Plasmodium falciparum |
Plasmodium falciparum |
MIC |
0.0023 |
ug.mL-1 |
10.1021/np0602012 |
| Plasmodium falciparum |
Plasmodium falciparum |
MIC90 |
2000.0 |
nM |
10.1128/aac.00808-06 |
| Plasmodium falciparum |
Plasmodium falciparum |
MIC90 |
109600.0 |
nM |
10.1128/aac.00808-06 |
| Plasmodium falciparum |
Plasmodium falciparum |
Potency |
1168.9 |
nM |
None |
| Plasmodium falciparum |
Plasmodium falciparum |
Potency |
1852.6 |
nM |
None |
| Plasmodium yoelii |
Plasmodium yoelii |
IC50 |
22200.0 |
nM |
10.1021/jm201095h |
| Porphyromonas asaccharolytica |
Porphyromonas asaccharolytica |
MIC |
0.004 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Prevotella bivia |
Prevotella bivia |
MIC |
0.004 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Prevotella bivia |
Prevotella bivia |
MIC |
0.06 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Prevotella bivia |
Prevotella bivia |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Prevotella disiens |
Prevotella disiens |
MIC |
0.12 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Prevotella disiens |
Prevotella disiens |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Prevotella intermedia |
Prevotella intermedia |
MIC |
0.12 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Priestia megaterium |
Priestia megaterium |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.01.026 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Proteus mirabilis |
Proteus mirabilis |
Ratio |
2.0 |
None |
10.1128/aac.00405-08 |
| Proteus vulgaris |
Proteus vulgaris |
IZ |
10.0 |
mm |
10.1016/j.bmc.2018.02.049 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmc.2018.02.049 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Proteus vulgaris |
Proteus vulgaris |
Ratio |
2.0 |
None |
10.1128/aac.00405-08 |
| Providencia alcalifaciens |
Providencia alcalifaciens |
MIC |
8000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
nan |
None |
10.1021/acs.jmedchem.6b01742 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
nan |
None |
10.1021/acs.jnatprod.5b01129 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
EC50 |
5200.0 |
nM |
10.1016/j.bmcl.2016.04.089 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
EC50 |
7800.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
FC |
3.0 |
None |
10.1021/acs.jnatprod.5b01129 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
FC |
128.0 |
None |
10.1021/acs.jmedchem.1c00614 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
FC |
100000.0 |
None |
10.1128/aac.01071-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
FIC |
0.25 |
None |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
FIC |
0.5 |
None |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
FICI |
0.05 |
None |
10.1128/aac.01071-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
FICI |
1.25 |
None |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
FICI |
1.5 |
None |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Inhibition |
10.0 |
% |
10.1128/aac.00471-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Inhibition |
100.0 |
% |
10.1021/jm0703901 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Inhibition |
nan |
% |
10.1128/aac.00471-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
6.0 |
mm |
10.1016/j.bmc.2018.02.049 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
29.0 |
mm |
10.1016/j.bmcl.2016.04.038 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
log10cfu |
8.56 |
None |
10.1128/aac.00471-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MBC |
32.0 |
ug ml-1 |
10.1021/acs.jnatprod.2c00065 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00471-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.03.061 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01742 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm00167a029 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
10.0 |
ug.mL-1 |
10.1128/aac.01071-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
12.0 |
ug.mL-1 |
10.1021/jm00145a020 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
13.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.04.060 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
13.0 |
ug.mL-1 |
10.1021/jm400485e |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01742 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1039/d2md00041e |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
20.0 |
ug.mL-1 |
10.1128/aac.01071-07 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
31.0 |
ug.mL-1 |
10.1021/jm501082n |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2006.12.035 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.01.026 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.04.001 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00065 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1021/ml300350p |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00017-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
62.5 |
ug.mL-1 |
10.1021/acs.jnatprod.0c01309 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2020.127146 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.bmc.2006.12.035 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
500.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.12.019 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
512.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1024.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1024.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01742 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2048.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4096.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16000.0 |
nM |
10.1021/acs.jmedchem.9b00288 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
19000.0 |
nM |
10.1021/acs.jnatprod.5b01129 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
25000.0 |
nM |
10.1016/j.bmc.2016.04.058 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
27000.0 |
nM |
10.1021/acs.jnatprod.5b01129 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32000.0 |
nM |
10.1016/j.ejmech.2019.111636 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32000.0 |
nM |
10.1021/acs.jmedchem.2c01076 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
53000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2048000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1016/j.bmc.2018.02.049 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1016/j.bmc.2019.04.032 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1016/j.ejmech.2019.04.067 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1021/np050424c |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC>90 |
17.8 |
ug ml-1 |
10.1021/np400145u |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
mortality |
100.0 |
% |
10.1021/acs.jmedchem.6b01742 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Ratio |
2.0 |
None |
10.1128/aac.00405-08 |
| Rattus norvegicus |
Aldose reductase |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Aldose reductase |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1a adrenergic receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1a adrenergic receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1b adrenergic receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1b adrenergic receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Androgen Receptor |
AC50 |
3000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Androgen Receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Androgen Receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Androgen Receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Bile salt export pump |
IC50 |
34700.0 |
nM |
10.1124/dmd.111.040758 |
| Rattus norvegicus |
Bile salt export pump |
Ki |
11900.0 |
nM |
10.1016/s0016-5085(00)70224-1 |
| Rattus norvegicus |
Brain |
Fu |
0.068 |
None |
10.1124/dmd.111.038778 |
| Rattus norvegicus |
Brain |
Fu |
0.121 |
None |
10.1124/dmd.111.038778 |
| Rattus norvegicus |
Brain |
Fu |
0.13 |
None |
10.1124/dmd.110.035998 |
| Rattus norvegicus |
Brain |
Kp |
0.92 |
None |
10.1124/dmd.110.035998 |
| Rattus norvegicus |
Brain |
Vd |
6.9 |
L.kg-1 |
10.1124/dmd.110.035998 |
| Rattus norvegicus |
Brain |
Vdu |
6.9 |
ml |
10.1021/jm901036q |
| Rattus norvegicus |
Cyclooxygenase-1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
GABA receptor alpha-1 subunit |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Glutamate (NMDA) receptor subunit zeta 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Glycine receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Glycine receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Insulin receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Insulin receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Jejunum |
CL |
0.0 |
mL.min-1.g-1 |
10.1124/dmd.111.043067 |
| Rattus norvegicus |
Kidney |
CL |
0.0 |
mL.min-1.g-1 |
10.1124/dmd.111.043067 |
| Rattus norvegicus |
Liver |
IC50 |
nan |
None |
10.1002/hep.27206 |
| Rattus norvegicus |
Liver microsome |
CL |
0.0 |
mL.min-1.g-1 |
10.1124/dmd.111.043067 |
| Rattus norvegicus |
Liver microsome |
Stability |
nan |
% |
10.1021/acs.jmedchem.5b01542 |
| Rattus norvegicus |
Multidrug resistance protein 1a |
Activity |
nan |
None |
10.1016/0006-2952(95)00045-2 |
| Rattus norvegicus |
Nitric-oxide synthase, brain |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Nitric-oxide synthase, brain |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Nuclear receptor subfamily 1 group I member 2 |
Activity |
nan |
None |
10.1124/dmd.110.035105 |
| Rattus norvegicus |
Nuclear receptor subfamily 1 group I member 2 |
Activity |
nan |
None |
10.1124/dmd.111.042879 |
| Rattus norvegicus |
Plasma |
Cp(f) |
0.83 |
uM |
10.1021/jm901036q |
| Rattus norvegicus |
Plasma |
Fu |
0.12 |
None |
10.1021/jm901036q |
| Rattus norvegicus |
Plasma |
Fu |
0.2 |
None |
10.1021/jm901371v |
| Rattus norvegicus |
Plasma |
K(p,uu,CSF) |
0.34 |
None |
10.1021/jm901036q |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
-31.0 |
% |
10.1021/jm00164a013 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
-30.0 |
% |
10.1021/jm00164a013 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
-27.0 |
% |
10.1021/jm00164a013 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
34000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
35000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
36000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
36000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
37000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
37000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
38000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
38000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
39000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
40000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
41000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.6 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.7 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.8 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.9 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
2.0 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
274.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
325.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
360.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
384.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
548.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
557.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
610.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
668.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
712.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
755.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
771.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
779.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
780.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
781.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
787.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
799.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
806.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
813.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
827.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
830.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
835.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
841.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
851.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
864.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
871.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
897.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
906.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
907.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
922.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
943.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
955.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
966.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
974.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
976.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1040.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1084.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
26.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
27.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
28.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
30.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
32.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
33.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
33.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
36.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
36.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
36.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
37.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
41.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
41.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
42.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
46.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
14.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
14.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
14.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
17.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
17.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
17.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
17.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
54.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
55.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
55.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
56.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
56.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
56.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
58.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
58.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
59.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
60.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
60.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
60.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
60.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
61.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
61.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
62.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
62.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
62.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
63.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
63.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
64.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
64.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
65.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
65.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
66.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
66.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
68.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
68.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
68.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
69.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
69.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
70.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
74.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.02 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.04 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.14 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.16 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.18 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.2 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.28 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.32 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.34 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.38 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.4 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.42 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.44 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.5 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.66 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.78 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
1.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
3.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
4.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
5.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
3.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
3.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
3.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
3.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
4.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
5.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
6.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
9.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
10.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
90.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
96.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
100.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
105.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
106.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
106.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
110.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
112.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
113.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
122.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
128.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
132.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
136.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
146.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
158.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
160.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
164.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
168.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
172.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
174.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
178.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
182.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
184.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
186.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
190.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
192.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
202.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
98.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
100.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
101.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
102.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
103.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
104.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
105.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
106.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
107.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
108.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
109.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
106.67 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
107.33 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
108.0 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
108.33 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
540.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
600.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
632.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
633.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
670.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
680.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
686.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
716.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
730.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
734.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
736.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
746.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
748.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
750.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
760.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
766.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
768.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
774.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
776.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
782.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
783.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
784.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
796.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
804.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
806.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
810.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
816.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
822.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
830.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
836.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
838.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
848.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
866.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
936.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
115.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
139.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
142.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
143.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
106.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
106.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
106.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
106.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
106.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
107.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
107.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
107.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
107.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
108.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
108.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
108.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
109.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
3.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
4.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
4.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
5.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
5.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
5.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
6.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2032.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2034.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2036.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2052.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2074.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2078.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2102.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2114.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2126.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2136.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2144.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2146.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2180.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2208.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2210.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2212.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2224.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2250.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2264.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2266.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2268.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2272.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2290.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2318.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2326.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2336.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2356.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2366.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2390.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2394.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2396.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
0.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
2.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
2.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1663.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1703.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1776.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1798.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1803.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1812.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1822.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1824.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1836.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1842.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1850.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1854.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1858.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1866.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1878.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1880.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1884.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1888.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1890.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1902.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1916.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1932.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1934.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1936.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1942.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1948.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1986.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1992.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2028.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2030.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2104.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2120.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
34.87 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
35.03 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.5 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.73 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
42.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
42.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
42.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
42.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
42.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
43.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
43.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
44.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
44.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
45.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
46.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
47.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
130000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
134000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
135000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
136000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
137000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
137300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
138000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
139000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
139300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
140000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
141000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
143000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
143300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
145700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
147000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
150000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
152000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
156000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
157000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
70.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
75.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
76.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
77.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
78.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
84.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
89.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
91.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
96.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
96.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
98.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
99.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
100.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
101.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
102.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
104.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
106.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
108.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
110.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
113.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
114.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
114.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
128.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
147.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
157.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
158.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
160.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
163.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
165.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
204.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
76.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
76.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
77.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
79.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
80.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
82.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
82.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
82.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
82.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
84.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
84.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
84.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
84.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
84.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
85.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
85.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
85.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
86.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
86.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
86.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
86.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
87.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
87.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
88.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
89.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
89.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
90.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
91.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
92.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
17.8 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
18.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
19.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
19.7 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
19.8 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.3 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.4 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.7 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.1 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.2 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.3 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.5 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.6 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.7 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.8 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
23.47 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
23.73 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
23.83 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.47 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
390300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
394000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
397700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
399300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
53.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
55.8 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
56.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
58.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
58.8 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
58.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
59.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.23 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.1 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.5 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.8 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.8 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
66.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
66.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
4.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
4.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
5.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
5.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
5.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
5.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
5.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
6.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
6.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
6.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
6.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
7.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
7.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
7.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
7.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
8.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
2.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
3.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
4.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
6.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
6.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
6.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
7.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
7.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
7.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
7.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
8.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
8.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
8.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
9.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
9.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
9.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
10.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
11.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
11.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
11.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
12.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
12.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
13.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
13.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
13.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
70.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
71.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
72.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
77.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
79.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
80.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
81.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
83.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
88.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
90.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
93.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
95.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
96.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
103.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
104.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
105.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
106.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
107.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
109.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
110.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
111.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
111.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
112.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
113.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
116.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1080.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1155.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1178.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1202.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1248.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1274.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1278.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1286.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1340.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1346.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1354.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1376.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1386.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1396.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1406.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1420.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1422.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1444.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1448.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1454.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1468.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1470.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1500.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1514.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1542.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1562.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1570.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1574.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1596.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1598.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1608.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1010670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1035000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1047330.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1053000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1065000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1070000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1072000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1077000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1082670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1103000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1105000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1110000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1111330.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1112000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1114000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1115000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1116000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1118000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1125000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1134000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1142000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1143000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1152000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1156000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1179000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1181000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1182000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1183000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1219000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1225000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1259000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1260000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.3 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.5 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.7 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.9 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.1 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.5 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.3 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.4 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.6 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.63 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
55000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
56000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
56700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
57000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
57300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
58000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
59000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
60000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
60300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
61000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
61000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
62000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
63000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5700000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5790000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5958000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6010000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6092000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6104000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6168000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6208000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6212000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6220000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6236000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6242000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6246000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6282000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6332000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6358000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6402000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6412000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6536000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6576000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6580000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6582000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6730000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6738000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6772000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6832000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6840000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7028000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7262000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7426000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7548000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7866000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7996000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
8036000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
8190000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
3.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
3.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
9.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
9.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
9.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
10.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
10.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
10.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
10.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
10.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
11.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
11.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
136.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
137.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
137.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
137.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
137.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
138.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
138.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
138.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
138.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
149.33 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
150.33 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
152.67 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
153.0 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
189.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
190.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
190.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
191.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
191.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
192.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
192.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
193.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
194.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
194.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
196.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
196.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
201.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
203.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
206.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
223.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
234.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
238.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
242.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
249.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
259.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
264.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
275.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
298.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
298.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
308.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
316.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
356.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
375.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
379.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
390.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Tissue Severity Score |
nan |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Tissue Severity Score |
nan |
None |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
228.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
230.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
332.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
358.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
394.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
396.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
452.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
460.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
482.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
506.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
528.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
546.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
556.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
624.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
660.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
664.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
682.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
710.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
730.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
754.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
758.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
906.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
968.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1128.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1166.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1204.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1214.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1320.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1326.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1650.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1682.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
2058.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9070.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9940.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10170.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10200.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10490.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10500.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10700.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11630.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11650.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11690.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11900.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11920.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11960.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
12040.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
12220.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
12330.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
12390.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
12470.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
12700.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
12700.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
12800.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
12910.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
12940.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
13090.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
13120.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
13160.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
13840.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
14230.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
14620.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
15360.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
16120.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
16520.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
17130.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
18560.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
0.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
0.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
7.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
7.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
7.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
7.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
13.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
13.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
16.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
16.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Serotonin 1a (5-HT1a) receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1a (5-HT1a) receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1b (5-HT1b) receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1b (5-HT1b) receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Serum |
AUC |
277000.0 |
ng.hr.mL-1 |
10.1128/aac.00458-08 |
| Rattus norvegicus |
Solute carrier family 22 member 7 |
Activity |
nan |
None |
10.1016/s0014-5793(98)00585-7 |
| Rattus norvegicus |
Solute carrier organic anion transporter family member 1A1 |
Activity |
nan |
None |
None |
| Rattus norvegicus |
Solute carrier organic anion transporter family member 1A1 |
Ki |
18200.0 |
nM |
10.1023/a:1014264614637 |
| Rattus norvegicus |
Solute carrier organic anion transporter family member 1A4 |
Ki |
1400.0 |
nM |
10.1053/jhep.2000.8539 |
| Rattus norvegicus |
Solute carrier organic anion transporter family member 1A4 |
Ki |
1460.0 |
nM |
10.1023/a:1014264614637 |
| Rattus norvegicus |
Voltage-gated L-type calcium channel alpha-1C subunit |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Voltage-gated N-type calcium channel alpha-1B subunit |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
IZ |
0.0 |
mm |
10.1016/j.ejmech.2010.07.050 |
| Salmonella enterica |
Salmonella enterica |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00310-09 |
| Salmonella enterica |
Salmonella enterica |
MIC |
2000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Salmonella enterica subsp. enterica serovar Abony |
Salmonella enterica subsp. enterica serovar Abony |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.066 |
| Salmonella enterica subsp. enterica serovar Paratyphi A |
Salmonella paratyphi |
IZ |
6.0 |
mm |
10.1016/j.bmc.2018.02.049 |
| Salmonella enterica subsp. enterica serovar Paratyphi A |
Salmonella paratyphi |
MIC |
12.0 |
ug.mL-1 |
10.1021/jm00143a010 |
| Salmonella enterica subsp. enterica serovar Paratyphi A |
Salmonella paratyphi |
MIC |
12.0 |
ug.mL-1 |
10.1021/jm00145a020 |
| Salmonella enterica subsp. enterica serovar Paratyphi A |
Salmonella paratyphi |
MIC |
nan |
None |
10.1016/j.bmc.2018.02.049 |
| Salmonella enterica subsp. enterica serovar Paratyphi B |
Salmonella enterica subsp. enterica serovar Paratyphi B |
MIC |
12.0 |
ug.mL-1 |
10.1021/jm00220a012 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
Activity |
nan |
None |
10.1016/j.ejmech.2017.06.061 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
Inhibition |
100.0 |
% |
10.1021/jm0703901 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00079-09 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00615-06 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
4000.0 |
nM |
10.1021/acs.jmedchem.9b00288 |
| Serratia marcescens |
Serratia marcescens |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00405-08 |
| Serratia marcescens |
Serratia marcescens |
MIC |
32.0 |
ug.mL-1 |
10.1021/ml300350p |
| Serratia marcescens |
Serratia marcescens |
Ratio |
2.0 |
None |
10.1128/aac.00405-08 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Hit score |
0.08736 |
None |
10.1101/2020.04.21.054387 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
19952.62 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
20000.0 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition index |
0.2558 |
None |
10.1101/2020.04.03.023846 |
| Shigella dysenteriae |
Shigella dysenteriae |
IZ |
8.0 |
mm |
10.1016/j.bmc.2018.02.049 |
| Shigella dysenteriae |
Shigella dysenteriae |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2018.02.049 |
| Shigella sonnei |
Shigella sonnei |
MIC |
1700.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.01244-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
2.0 |
% |
10.1128/aac.00846-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
2.3 |
% |
10.1128/aac.00090-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
4.0 |
% |
10.1128/aac.00846-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
18.8 |
% |
10.1128/aac.00090-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
20.0 |
% |
10.1016/j.bmc.2006.12.027 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
46.0 |
% |
10.1128/aac.00120-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
50.0 |
% |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
92.0 |
% |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
94.0 |
% |
10.1128/aac.00470-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
94.0 |
% |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
96.0 |
% |
10.1128/aac.00470-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
99.9 |
% |
10.1016/j.bmcl.2023.129320 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00470-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.bmc.2016.11.056 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.bmcl.2023.129320 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.ejmech.2018.04.049 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.ejmech.2019.112026 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.ejmech.2021.113691 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/acs.jmedchem.2c01076 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/jm0703183 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/jm3012728 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/jm900519b |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00064-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00350-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00458-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00596-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00766-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00804-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01302-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01395-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01480-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01605-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01649-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Antibiotic resistance |
nan |
None |
10.1016/s0960-894x(98)00536-8 |
| Staphylococcus aureus |
Staphylococcus aureus |
AUC |
19650.0 |
ng.hr.mL-1 |
10.1128/aac.00455-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
50.0 |
nM |
10.1016/j.bmcl.2016.04.089 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
50.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
150.0 |
nM |
10.1016/j.bmcl.2016.04.089 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
230.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
0.09 |
mg.kg-1 |
10.1021/jm00167a029 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
0.14 |
mg.kg-1 |
10.1021/jm00145a020 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
0.28 |
mg.kg-1 |
10.1021/jm00167a029 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
0.98 |
None |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
0.99 |
None |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
1.19 |
None |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
1.2 |
None |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
1.9 |
None |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
2.0 |
None |
10.1128/aac.01605-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
2.5 |
None |
10.1128/aac.01605-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
4.0 |
None |
10.1039/d2md00351a |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
8.0 |
None |
10.1016/j.ejmech.2021.113723 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
15.0 |
None |
10.1039/d2md00351a |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
128.0 |
None |
10.1016/j.bmcl.2023.129320 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
500.0 |
None |
10.1021/jm3012728 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
1024.0 |
None |
10.1016/j.bmcl.2023.129320 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
4096.0 |
None |
10.1021/acs.jmedchem.2c01076 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
16000.0 |
None |
10.1016/j.ejmech.2021.113723 |
| Staphylococcus aureus |
Staphylococcus aureus |
fCmax |
3.82 |
ug ml-1 |
10.1128/aac.00455-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
FIC |
1.0 |
None |
10.1021/acs.jnatprod.2c00621 |
| Staphylococcus aureus |
Staphylococcus aureus |
GI |
nan |
None |
10.1016/j.bmc.2015.04.069 |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
0.0025 |
ug.mL-1 |
10.1021/np000436s |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
0.01 |
ug.mL-1 |
10.1021/np000436s |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
250.0 |
ug.mL-1 |
10.1021/np050176k |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
10000.0 |
nM |
10.1021/acs.jnatprod.2c00444 |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
nan |
None |
10.1021/np2006555 |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
nan |
None |
10.1021/np900281r |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
10.0 |
% |
10.1128/aac.00471-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
76.3 |
% |
10.1016/j.ejmech.2021.113402 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
76.3 |
% |
10.1039/D1MD00230A |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
100.0 |
% |
10.1021/jm0703901 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
nan |
% |
10.1128/aac.00471-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
nan |
% |
10.1128/aac.01302-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
10.0 |
mm |
10.1016/j.bmc.2018.02.049 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
23.0 |
mm |
10.1016/j.bmcl.2017.05.032 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
25.0 |
mm |
10.1016/j.bmcl.2016.04.038 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
27.0 |
mm |
10.1016/j.bmcl.2017.05.032 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
30.0 |
mm |
10.1016/j.bmcl.2017.05.032 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
31.0 |
mm |
10.1016/j.bmc.2007.09.025 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
33.0 |
mm |
10.1016/j.bmcl.2017.05.032 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
49.0 |
mm |
10.1016/j.ejmech.2008.09.035 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
nan |
None |
10.1021/np900382x |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
-1.72 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
0.86 |
None |
10.1128/aac.00237-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
1.0 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
1.1 |
None |
10.1128/aac.00208-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
1.36 |
None |
10.1128/aac.00208-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
1.78 |
None |
10.1128/aac.00237-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
2.0 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
3.0 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
7.5 |
None |
10.1128/aac.00471-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
42.6 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-3.02 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
0.5 |
None |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
1.43 |
None |
10.1128/aac.00120-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.0 |
None |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.1 |
None |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.68 |
None |
10.1128/aac.00120-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
6.9 |
None |
10.1128/aac.00458-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
43.35 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log(1/C) |
8.07 |
None |
10.1021/jm00210a025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.08 |
ug ml-1 |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.12 |
ug ml-1 |
10.1128/aac.00458-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.2 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.4 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.5 |
ug ml-1 |
10.1128/aac.00208-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.8 |
ug ml-1 |
10.1128/aac.00120-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
1.0 |
ug ml-1 |
10.1016/j.bmcl.2023.129320 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
2.0 |
mg/ml |
10.1021/acs.jmedchem.6b00485 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
2.0 |
ug ml-1 |
10.1016/j.bmcl.2023.129320 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
2.0 |
uM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
2.0 |
uM |
10.1021/acs.jmedchem.7b01903 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
2.5 |
ug ml-1 |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
3.6 |
ug ml-1 |
10.1128/aac.00120-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
4.0 |
ug ml-1 |
10.1128/aac.00458-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
8.0 |
ng/ml |
10.1021/acs.jnatprod.5b00770 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
8.0 |
ug ml-1 |
10.1128/aac.00208-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
nan |
None |
10.1021/acs.jnatprod.2c00065 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC |
0.25 |
ug ml-1 |
10.1128/aac.00766-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC |
4.0 |
ug ml-1 |
10.1128/aac.00766-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC |
6.25 |
ug ml-1 |
10.1128/aac.00457-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC |
25.0 |
ug ml-1 |
10.1128/aac.00457-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC |
46.9 |
uM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC |
46.9 |
uM |
10.1021/acs.jmedchem.7b01903 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBIC |
0.0625 |
ug ml-1 |
10.1128/aac.00455-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBIC |
0.2 |
ug ml-1 |
10.1128/aac.00457-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBIC |
nan |
None |
10.1128/aac.00455-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6e-06 |
ug.mL-1 |
10.1128/aac.00437-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.0002 |
ug.mL-1 |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.00025 |
ug.mL-1 |
10.1128/aac.00471-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.0005 |
ug.mL-1 |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.002 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.002 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.002 |
ug.mL-1 |
10.1021/np050176k |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.002 |
ug.mL-1 |
10.1021/np200320u |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.002 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.002 |
ug.mL-1 |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.003 |
ug.mL-1 |
10.1021/jm00164a013 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.bmcl.2007.02.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.004 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00065 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.004 |
ug.mL-1 |
10.1021/acs.jnatprod.5b00770 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.004 |
ug.mL-1 |
10.1021/np200320u |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.004 |
ug.mL-1 |
10.1128/aac.00064-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.004 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.004 |
ug.mL-1 |
10.1128/aac.00834-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.004 |
ug.mL-1 |
10.1128/aac.01455-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.004 |
ug.mL-1 |
10.1128/aac.01544-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.004 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.005 |
ug.mL-1 |
10.1021/jm00145a020 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.005 |
ug.mL-1 |
10.1021/np010173h |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.006 |
ug.mL-1 |
10.1016/j.ejmech.2017.10.048 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.006 |
ug.mL-1 |
10.1128/aac.00457-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.006 |
ug.mL-1 |
10.1128/aac.00834-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.007 |
ug.mL-1 |
10.1021/jm00210a025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.0078 |
ug.mL-1 |
10.1021/acs.jnatprod.1c00578 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.0078 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00621 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1016/j.bmcl.2006.10.016 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1016/j.bmcl.2007.08.048 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.077 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1016/j.ejmech.2012.09.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.066 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1016/j.ejmech.2016.03.061 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1021/acsmedchemlett.0c00381 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.01455-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.01649-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.01 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00520 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.01 |
ug.mL-1 |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.012 |
ug.mL-1 |
10.1128/aac.00457-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.01221 |
ug.mL-1 |
10.1016/j.bmc.2010.02.005 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.0125 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.ejmech.2012.09.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.0156 |
ug.mL-1 |
10.1016/j.ejmech.2019.02.009 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.016 |
ug.mL-1 |
10.1016/j.bmcl.2015.07.043 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.016 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.066 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.016 |
ug.mL-1 |
10.1016/j.ejmech.2016.03.061 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.016 |
ug.mL-1 |
10.1021/jm00167a029 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00120-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.01455-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.01605-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2013.04.060 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.02 |
ug.mL-1 |
10.1021/jm400485e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.02 |
ug.mL-1 |
10.1021/np000436s |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.02 |
ug.mL-1 |
10.1128/aac.00766-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.0225 |
ug.mL-1 |
10.1007/s00044-011-9918-4 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.025 |
ug.mL-1 |
10.1021/jm00143a010 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.025 |
ug.mL-1 |
10.1021/jm00220a012 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00520 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jnatprod.9b00062 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.03 |
ug.mL-1 |
10.1021/jm501082n |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00208-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00766-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.03125 |
ug.mL-1 |
10.1016/j.ejmech.2019.02.009 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.049 |
ug.mL-1 |
10.1128/aac.00971-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.05 |
ug.mL-1 |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2007.12.019 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00350-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00915-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01480-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.bmcl.2020.127146 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.0625 |
ug.mL-1 |
10.1128/aac.00455-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.07 |
ug.mL-1 |
10.1016/j.ejmech.2012.09.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.078 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00174 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmc.2021.116580 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2020.127146 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.060 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01480-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.21 |
ug.mL-1 |
10.1016/j.bmc.2021.116580 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2018.02.049 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2023.129320 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2008.09.035 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jnatprod.0c01309 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1021/np050438i |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01649-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.3 |
ug.mL-1 |
10.1016/j.ejmech.2012.09.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.3125 |
ug.mL-1 |
10.1021/np000436s |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2020.127146 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2008.04.001 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/ml300350p |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.6 |
ug.mL-1 |
10.1016/j.ejmech.2012.09.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.625 |
ug.mL-1 |
10.1128/aac.00247-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.9 |
ug.mL-1 |
10.1016/j.ejmech.2007.12.019 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00458-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00971-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01649-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.25 |
ug.mL-1 |
10.1016/j.ejmech.2012.09.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.562 |
ug.mL-1 |
10.1007/s00044-011-9918-4 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.6 |
ug.mL-1 |
10.1016/j.ejmech.2017.10.048 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00237-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00971-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01649-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.02.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/np200320u |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00846-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00971-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
7.8 |
nM |
10.1021/acs.jmedchem.9b00288 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.04.001 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01649-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
10.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
10.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00174 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.08.048 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01649-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
18.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
20.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
21.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.05.032 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
22.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.05.032 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
31.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.043 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2006.12.035 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00350-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00834-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01649-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
63.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.10.016 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.08.048 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2020.127146 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00915-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01649-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
100.0 |
nM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
100.0 |
nM |
10.1021/acs.jmedchem.7b01903 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
100.0 |
nM |
10.1021/acs.jnatprod.5b01129 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
125.0 |
ug.mL-1 |
10.1128/aac.01649-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.077 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00350-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01081-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
250.0 |
nM |
10.1021/acs.jmedchem.9b00288 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
250.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
250.0 |
ug.mL-1 |
10.1128/aac.01649-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00846-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2019.111636 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.2c01076 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1000.0 |
nM |
10.1021/acs.jnatprod.2c00481 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1000.0 |
ug.mL-1 |
10.1016/j.bmc.2015.09.027 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1024.0 |
ug.mL-1 |
10.1128/aac.00209-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1250.0 |
nM |
10.1021/acs.jmedchem.1c01809 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1900.0 |
nM |
10.1021/acs.jnatprod.1c00232 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2048.0 |
ug.mL-1 |
10.1128/aac.01544-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4096.0 |
ug.mL-1 |
10.1016/j.bmc.2006.12.035 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
15400.0 |
nM |
10.1021/acs.jnatprod.2c00481 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
25923000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmc.2013.10.011 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmc.2019.04.032 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmcl.2013.11.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1021/np050424c |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1021/np200320u |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1021/np900281r |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1128/aac.00455-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC100 |
0.15 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC100 |
0.2 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC100 |
6.25 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC100 |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.004 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.008 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.015 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.016 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.015 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.016 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00846-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC99 |
nan |
None |
10.1016/j.ejmech.2013.10.055 |
| Staphylococcus aureus |
Staphylococcus aureus |
PAE |
1.8 |
hr |
10.1016/j.bmcl.2023.129320 |
| Staphylococcus aureus |
Staphylococcus aureus |
PAE |
3.45 |
hr |
10.1016/j.bmcl.2023.129320 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
4.5 |
None |
10.1128/aac.00120-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
7.0 |
None |
10.1021/acs.jmedchem.9b00720 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
23.0 |
None |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
29.0 |
None |
10.1016/j.ejmech.2018.03.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
29.0 |
None |
10.1016/j.ejmech.2019.04.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
533.0 |
None |
10.1128/aac.00458-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
2000.0 |
None |
10.1016/j.bmc.2019.02.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
40000.0 |
None |
10.1016/j.ejmech.2017.10.048 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
500000.0 |
None |
10.1016/j.ejmech.2018.03.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
500000.0 |
None |
10.1016/j.ejmech.2019.04.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
500000.0 |
None |
10.1021/acs.jmedchem.9b00720 |
| Staphylococcus aureus |
Staphylococcus aureus |
T1/2 |
3.56 |
hr |
10.1128/aac.00455-10 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
nan |
None |
10.1128/aac.00343-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Inhibition |
100.0 |
% |
10.1021/jm0703901 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
IZ |
40.0 |
mm |
10.1016/j.bmc.2018.02.049 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
log10cfu |
0.17 |
None |
10.1128/aac.00237-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
log10cfu |
2.5 |
None |
10.1128/aac.00237-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
0.006 |
ug ml-1 |
10.1128/aac.00343-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.01011-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
3.0 |
uM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
3.0 |
uM |
10.1021/acs.jmedchem.7b01903 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBEC |
15.6 |
uM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBEC |
15.6 |
uM |
10.1021/acs.jmedchem.7b01903 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBEC |
50.0 |
ug ml-1 |
10.1128/aac.00457-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBIC |
0.2 |
ug ml-1 |
10.1128/aac.00457-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.066 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.ejmech.2016.03.061 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.004 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.006 |
ug.mL-1 |
10.1128/aac.00343-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.008 |
ug.mL-1 |
10.1016/j.bmcl.2015.07.043 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.008 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.077 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.008 |
ug.mL-1 |
10.1016/j.ejmech.2016.03.061 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.008 |
ug.mL-1 |
10.1021/jm00167a029 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.01011-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.012 |
ug.mL-1 |
10.1128/aac.00457-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.0156 |
ug.mL-1 |
10.1016/j.ejmech.2019.02.009 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.016 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00520 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.03 |
ug.mL-1 |
10.1021/jm501082n |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.078 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00174 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00237-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2018.02.049 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114360 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
20.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
100.0 |
nM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
100.0 |
nM |
10.1021/acs.jmedchem.7b01903 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
100.0 |
nM |
10.1021/acs.jnatprod.5b01129 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
250.0 |
nM |
10.1021/acs.jmedchem.9b00288 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c00614 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1000.0 |
nM |
10.1021/acs.jmedchem.1c02140 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
0.015 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
0.015 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Ratio |
1.0 |
None |
10.1128/aac.00343-07 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
Activity |
0.0 |
% |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
Activity |
7.0 |
% |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
Activity |
93.0 |
% |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
BBC |
0.125 |
ug ml-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
BBC |
0.25 |
ug ml-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
BBC |
8.0 |
ug ml-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
BBC |
32.0 |
ug ml-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
BBC |
64.0 |
ug ml-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MBC50 |
8.0 |
ug ml-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MBC90 |
32.0 |
ug ml-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC90 |
0.03 |
ug.mL-1 |
10.1128/aac.01052-06 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00520 |
| Stenotrophomonas maltophilia |
Stenotrophomonas maltophilia |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00520 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
0.12 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
0.12 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
0.8 |
% |
10.1128/aac.01384-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
98.8 |
% |
10.1128/aac.01384-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
nan |
None |
10.1021/acs.jmedchem.0c00520 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
IZ |
25.0 |
mm |
10.1016/j.bmcl.2016.04.038 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.004 |
ug.mL-1 |
10.1021/np050176k |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.0625 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00520 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.063 |
ug.mL-1 |
10.1021/jm00167a029 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.12 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.034 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
10.0 |
nM |
10.1021/acs.jnatprod.2c00481 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
20.0 |
nM |
10.1021/acs.jnatprod.2c00481 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
110.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC100 |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.01384-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC>90 |
0.01 |
ug ml-1 |
10.1021/np400145u |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
0.03 |
ug.mL-1 |
10.1128/aac.01384-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
ED50 |
0.35 |
mg.kg-1 |
10.1021/jm00167a029 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
ED50 |
0.47 |
mg.kg-1 |
10.1021/jm00167a029 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
Inhibition |
10.0 |
% |
10.1128/aac.00471-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
Inhibition |
100.0 |
% |
10.1021/jm0703901 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
Inhibition |
nan |
% |
10.1128/aac.00471-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
log10cfu |
6.44 |
None |
10.1128/aac.00471-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.00025 |
ug.mL-1 |
10.1128/aac.00471-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.008 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00520 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.063 |
ug.mL-1 |
10.1021/jm00167a029 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
nan |
None |
10.1021/np050424c |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
0.06 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
0.12 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00485 |
| Streptococcus salivarius |
Streptococcus salivarius |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Streptococcus salivarius |
Streptococcus salivarius |
MIC100 |
0.2 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Streptomyces albus |
Streptomyces albus |
MIC |
5.0 |
ug.mL-1 |
10.1128/aac.01406-09 |
| Streptomyces albus |
Streptomyces albus |
MIC |
20.0 |
ug.mL-1 |
10.1128/aac.01406-09 |
| Streptomyces albus |
Streptomyces albus |
MIC |
40.0 |
ug.mL-1 |
10.1128/aac.01406-09 |
| Treponema denticola |
Treponema denticola |
MIC |
0.004 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Trichophyton rubrum |
Trichophyton rubrum |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.066 |
| Veillonella parvula |
Veillonella parvula |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| Vibrio cholerae |
Vibrio cholerae |
MIC |
128000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| Xanthomonas campestris |
Xanthomonas campestris |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.01.026 |
| Yersinia pseudotuberculosis |
Yersinia pseudotuberculosis |
MIC |
11000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| None |
ADMET |
Activity |
0.0 |
% |
10.1021/np50025a010 |
| None |
ADMET |
Activity |
1.0 |
% |
10.1021/np50025a010 |
| None |
ADMET |
Activity |
4.0 |
% |
10.1021/np50025a010 |
| None |
ADMET |
Activity |
48.0 |
% |
10.1021/np50025a010 |
| None |
ADMET |
Activity |
52.7 |
% |
10.1021/acs.jmedchem.5b00608 |
| None |
ADMET |
Activity |
58.0 |
% |
10.1021/np50025a010 |
| None |
ADMET |
Activity |
66.0 |
% |
10.1021/np50025a010 |
| None |
ADMET |
Activity |
82.0 |
% |
10.1021/np50025a010 |
| None |
ADMET |
Activity |
85.0 |
% |
10.1016/j.ejmech.2013.09.061 |
| None |
ADMET |
Activity |
93.0 |
% |
10.1016/j.ejmech.2013.09.061 |
| None |
ADMET |
Activity |
94.0 |
% |
10.1016/j.ejmech.2013.09.061 |
| None |
ADMET |
Activity |
98.3 |
% |
10.1021/acs.jmedchem.5b00608 |
| None |
ADMET |
Activity |
103.1 |
% |
10.1021/acs.jmedchem.5b00608 |
| None |
ADMET |
Activity |
105.6 |
% |
10.1021/acs.jmedchem.5b00608 |
| None |
ADMET |
Activity |
nan |
None |
10.1016/j.ejmech.2015.10.049 |
| None |
ADMET |
AUC |
0.0 |
ng.hr.mL-1 |
10.1128/aac.01533-06 |
| None |
ADMET |
AUC |
4600.0 |
ng.hr.mL-1 |
10.1128/aac.00775-08 |
| None |
ADMET |
AUC |
7000.0 |
ng.hr.mL-1 |
10.1128/aac.01533-06 |
| None |
ADMET |
AUC |
14000.0 |
ng.hr.mL-1 |
10.1128/aac.01533-06 |
| None |
ADMET |
AUC |
64400.0 |
ng.hr.mL-1 |
10.1128/aac.01544-08 |
| None |
ADMET |
AUC |
122000.0 |
ng.hr.mL-1 |
10.1128/aac.01533-06 |
| None |
ADMET |
AUC |
304000.0 |
ng.hr.mL-1 |
10.1128/aac.00458-08 |
| None |
ADMET |
BPR |
0.03 |
None |
10.1021/jm901036q |
| None |
ADMET |
CC50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.093 |
| None |
ADMET |
CL |
0.0 |
mL.min-1.g-1 |
10.1124/dmd.111.043067 |
| None |
ADMET |
CL |
0.2 |
mL.min-1.g-1 |
10.1124/dmd.111.043067 |
| None |
ADMET |
CL |
0.7 |
mL.min-1.g-1 |
10.1124/dmd.111.043067 |
| None |
ADMET |
CL |
3.5 |
mL.min-1.kg-1 |
10.1124/dmd.108.020479 |
| None |
ADMET |
CL |
32.0 |
mL.min-1.kg-1 |
10.1021/jm000407e |
| None |
ADMET |
CL |
99.0 |
L/hr |
10.1128/aac.01533-06 |
| None |
ADMET |
Cmax |
1215.14 |
nM |
10.1128/aac.00775-08 |
| None |
ADMET |
Cmax |
5954.19 |
nM |
10.1128/aac.01544-08 |
| None |
ADMET |
Cmax |
8019.93 |
nM |
10.1128/aac.00458-08 |
| None |
ADMET |
Cmax |
13000.0 |
nM |
10.1021/acs.jmedchem.9b01071 |
| None |
ADMET |
Cmin |
0.1 |
ug ml-1 |
10.1128/aac.00775-08 |
| None |
ADMET |
Cmin |
1.3 |
ug ml-1 |
10.1128/aac.01544-08 |
| None |
ADMET |
Cmin |
3.8 |
mg/L |
10.1128/aac.00458-08 |
| None |
ADMET |
Drug metabolism |
90.0 |
% |
10.1016/j.bmcl.2019.07.001 |
| None |
ADMET |
Drug metabolism |
nan |
None |
10.1016/j.bmcl.2019.07.001 |
| None |
ADMET |
Drug uptake |
10.0 |
ug ml-1 |
10.1128/aac.00985-07 |
| None |
ADMET |
Fu |
0.118 |
None |
10.1124/dmd.111.038778 |
| None |
ADMET |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.045 |
| None |
ADMET |
GI50 |
100.0 |
ug.mL-1 |
10.1039/C5MD00404G |
| None |
ADMET |
IC50 |
20000.0 |
nM |
10.1021/acs.jmedchem.5b00608 |
| None |
ADMET |
IC50 |
100000.0 |
nM |
10.1016/j.ejmech.2013.01.017 |
| None |
ADMET |
IC50 |
100000.0 |
nM |
10.1021/jm401735w |
| None |
ADMET |
IC50 |
nan |
None |
10.1016/j.ejmech.2013.06.010 |
| None |
ADMET |
Inhibition |
nan |
% |
10.1016/j.bmcl.2016.04.012 |
| None |
ADMET |
Ki |
50000.0 |
nM |
10.1021/np50025a010 |
| None |
ADMET |
Ki |
100000.0 |
nM |
10.1021/np50025a010 |
| None |
ADMET |
Ki |
140000.0 |
nM |
10.1021/np50025a010 |
| None |
ADMET |
K(p,uu,brain) |
0.035 |
None |
10.1021/jm901036q |
| None |
ADMET |
MRT |
4.6 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
PPB |
64.0 |
% |
10.1128/aac.00971-08 |
| None |
ADMET |
Ratio |
1.0 |
None |
10.1128/aac.00971-08 |
| None |
ADMET |
Selectivity Index |
643.12 |
None |
10.1016/j.ejmech.2021.113472 |
| None |
ADMET |
Selectivity Index |
1407.2 |
None |
10.1016/j.ejmech.2021.113472 |
| None |
ADMET |
Selectivity Index |
nan |
None |
10.1016/j.bmc.2022.116777 |
| None |
ADMET |
Stability |
nan |
% |
10.1021/acs.jmedchem.2c01076 |
| None |
ADMET |
Stability |
nan |
% |
10.1021/acs.jmedchem.5b01542 |
| None |
ADMET |
Survival |
nan |
None |
10.1016/j.ejmech.2019.06.038 |
| None |
ADMET |
T1/2 |
2.5 |
hr |
10.1128/aac.00775-08 |
| None |
ADMET |
T1/2 |
3.5 |
hr |
10.1021/jm000407e |
| None |
ADMET |
T1/2 |
3.8 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
T1/2 |
4.1 |
hr |
10.1128/aac.01544-08 |
| None |
ADMET |
T1/2 |
4.7 |
hr |
10.1016/j.bmc.2016.11.008 |
| None |
ADMET |
T1/2 |
9.3 |
hr |
10.1016/j.bmc.2016.11.008 |
| None |
ADMET |
TI |
nan |
None |
10.1016/j.ejmech.2013.06.010 |
| None |
ADMET |
TI |
nan |
None |
10.1016/j.ejmech.2017.06.061 |
| None |
ADMET |
Tmax |
1.5 |
hr |
10.1021/acs.jmedchem.9b01071 |
| None |
ADMET |
Tmax |
2.1 |
hr |
10.1128/aac.00775-08 |
| None |
ADMET |
Vc |
430.89 |
l |
10.1128/aac.01533-06 |
| None |
ADMET |
Vd |
8.8 |
L.kg-1 |
10.1021/jm000407e |
| None |
ADMET |
Vd |
33.65 |
l |
10.1128/aac.01520-08 |
| None |
ADMET |
Vd |
43.66 |
l |
10.1128/aac.01520-08 |
| None |
ADMET |
Vd |
49.94 |
l |
10.1128/aac.01520-08 |
| None |
ADMET |
Vd |
52.1 |
l |
10.1128/aac.01520-08 |
| None |
ADMET |
Vd |
102.6 |
l |
10.1128/aac.01520-08 |
| None |
ADMET |
Vd |
102.8 |
l |
10.1128/aac.01520-08 |
| None |
ADMET |
Vdss |
0.97 |
L.kg-1 |
10.1124/dmd.108.020479 |
| None |
Erythrocyte |
LC50 |
nan |
None |
10.1021/acs.jnatprod.5b01129 |
| None |
Erythrocyte |
MHC10 |
nan |
None |
10.1021/acs.jmedchem.2c01076 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Index Value |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Active |
1.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Marginal |
3.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Index Value |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Number of Reports |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1021/tx1000865 |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1021/tx900326k |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1124/dmd.110.035113 |
| None |
Hepatotoxicity |
HepSE_bilirubinemia |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholecystitis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholelithiasis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cirrhosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_Combined Scores |
3.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_elevated liver function tests |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic failure |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic necrosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatitis |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatomegaly |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_jaundice |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver disease |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver fatty |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver function tests abnormal |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
LDH Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LDH Increase - Index Value |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LDH Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LTKB_BD DILI severity score |
8.0 |
None |
10.1016/j.drudis.2011.05.007 |
| None |
Hepatotoxicity |
SGOT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Index Value |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Index Value |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Lipid bilayer |
Activity |
nan |
None |
10.1016/j.ejmech.2016.07.068 |
| None |
Molecular identity unknown |
PPB |
91.0 |
% |
10.1021/jm501661f |
| None |
NON-PROTEIN TARGET |
Activity |
nan |
None |
10.1016/j.ejmech.2016.07.005 |
| None |
NON-PROTEIN TARGET |
Activity |
nan |
None |
10.1021/acs.jmedchem.6b00624 |
| None |
NON-PROTEIN TARGET |
fAUC/MIC |
300.0 |
None |
10.1016/j.bmcl.2013.07.006 |
| None |
NON-PROTEIN TARGET |
fCmax/MIC |
20.0 |
None |
10.1016/j.bmcl.2013.07.006 |
| None |
NON-PROTEIN TARGET |
fT>MIC |
100.0 |
% |
10.1016/j.bmcl.2013.07.006 |
| None |
NON-PROTEIN TARGET |
Fu |
0.119 |
None |
10.1124/dmd.111.038778 |
| None |
NON-PROTEIN TARGET |
Fu |
0.2 |
None |
10.1124/dmd.108.020479 |
| None |
NON-PROTEIN TARGET |
Fu |
0.62 |
None |
10.1021/jm401963n |
| None |
NON-PROTEIN TARGET |
GI |
nan |
None |
10.1016/j.ejmech.2016.06.042 |
| None |
NON-PROTEIN TARGET |
GI50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.056 |
| None |
NON-PROTEIN TARGET |
GI90 |
100.0 |
ug ml-1 |
10.1016/j.bmcl.2016.11.056 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (acute) |
7.3 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (animal toxicity known) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (benign tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (granulomatous hepatitis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (mechanism) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
22.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
23.0 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (time to onset) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
IC20 |
30.0 |
ug ml-1 |
10.1128/aac.00729-05 |
| None |
NON-PROTEIN TARGET |
IC50 |
0.0016 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.056 |
| None |
NON-PROTEIN TARGET |
IC50 |
0.45 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.056 |
| None |
NON-PROTEIN TARGET |
IC50 |
0.51 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.056 |
| None |
NON-PROTEIN TARGET |
IC50 |
0.75 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.056 |
| None |
NON-PROTEIN TARGET |
IC50 |
0.81 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.056 |
| None |
NON-PROTEIN TARGET |
IC50 |
130.0 |
ug.mL-1 |
10.1128/aac.00729-05 |
| None |
NON-PROTEIN TARGET |
IC50 |
96000.0 |
nM |
10.1128/aac.00126-08 |
| None |
NON-PROTEIN TARGET |
IC50 |
nan |
None |
10.1016/j.bmcl.2016.11.003 |
| None |
NON-PROTEIN TARGET |
IC50 |
nan |
None |
10.1016/j.ejmech.2016.07.039 |
| None |
NON-PROTEIN TARGET |
IC90 |
0.041 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.056 |
| None |
NON-PROTEIN TARGET |
IC90 |
0.061 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.045 |
| None |
NON-PROTEIN TARGET |
IC90 |
0.89 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.045 |
| None |
NON-PROTEIN TARGET |
Inhibition |
75.0 |
% |
10.1128/aac.00126-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| None |
NON-PROTEIN TARGET |
MIC |
0.004 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| None |
NON-PROTEIN TARGET |
MIC |
0.004 |
ug.mL-1 |
10.1128/aac.00477-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00477-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01052-07 |
| None |
NON-PROTEIN TARGET |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01052-07 |
| None |
NON-PROTEIN TARGET |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01052-07 |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00477-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.89 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.045 |
| None |
NON-PROTEIN TARGET |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01052-07 |
| None |
NON-PROTEIN TARGET |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01052-07 |
| None |
NON-PROTEIN TARGET |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01052-07 |
| None |
NON-PROTEIN TARGET |
MIC |
4.8 |
ug.mL-1 |
10.1016/j.ejmech.2013.04.060 |
| None |
NON-PROTEIN TARGET |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00477-09 |
| None |
NON-PROTEIN TARGET |
MIC |
40.0 |
ug.mL-1 |
10.1128/aac.01406-09 |
| None |
NON-PROTEIN TARGET |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00477-09 |
| None |
NON-PROTEIN TARGET |
MIC |
1890.0 |
nM |
10.1016/j.bmcl.2010.06.096 |
| None |
NON-PROTEIN TARGET |
MIC |
15180.0 |
nM |
10.1016/j.bmcl.2010.06.096 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.45 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.056 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.45 |
ug.mL-1 |
10.1039/C5MD00404G |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.056 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.51 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.056 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.7 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.056 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.75 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.056 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.81 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.056 |
| None |
NON-PROTEIN TARGET |
MIC90 |
0.81 |
ug.mL-1 |
10.1039/C5MD00404G |
| None |
NON-PROTEIN TARGET |
MIC95 |
0.24 |
uM |
10.1016/j.bmc.2011.05.028 |
| None |
NON-PROTEIN TARGET |
RatioAUC/MIC |
271.0 |
None |
10.1128/aac.01520-08 |
| None |
NON-PROTEIN TARGET |
RatioAUC/MIC |
665.0 |
None |
10.1128/aac.01520-08 |
| None |
NON-PROTEIN TARGET |
RatioAUC/MIC |
1500.0 |
None |
10.1016/j.bmcl.2013.07.006 |
| None |
NON-PROTEIN TARGET |
%T>MIC |
100.0 |
% |
10.1016/j.bmcl.2013.07.006 |
| None |
NON-PROTEIN TARGET |
T>MIC |
6.54 |
hr |
10.1128/aac.00367-09 |
| None |
NON-PROTEIN TARGET |
T>MIC |
7.5 |
hr |
10.1128/aac.00367-09 |
| None |
No relevant target |
Activity |
0.0 |
mol/mol |
10.1016/j.ejmech.2016.07.039 |
| None |
No relevant target |
IC50 |
nan |
None |
10.1016/j.bmcl.2015.11.071 |
| None |
No relevant target |
Kinetic_solubility |
nan |
None |
10.1016/j.ejmech.2012.08.047 |
| None |
No relevant target |
Kinetic_solubility |
nan |
None |
10.1021/acs.jmedchem.1c00707 |
| None |
No relevant target |
Kinetic_solubility |
nan |
None |
10.1021/acs.jmedchem.5b01542 |
| None |
No relevant target |
LogD |
1.3 |
None |
10.1021/acs.jmedchem.5b00050 |
| None |
No relevant target |
LogD |
1.31 |
None |
10.1016/j.ejmech.2022.114434 |
| None |
No relevant target |
LogD |
1.67 |
None |
10.1021/jm901858n |
| None |
No relevant target |
LogP |
1.66 |
None |
10.1016/j.bmcl.2015.07.043 |
| None |
No relevant target |
LogP |
1.66 |
None |
10.1016/j.ejmech.2014.07.066 |
| None |
No relevant target |
LogP |
1.66 |
None |
10.1016/j.ejmech.2016.03.061 |
| None |
No relevant target |
LogP |
1.66 |
None |
10.1016/j.ejmech.2019.02.009 |
| None |
No relevant target |
LogP |
3.72 |
None |
10.1016/j.bmc.2018.07.049 |
| None |
No relevant target |
LogP |
nan |
None |
10.1016/j.ejmech.2016.07.039 |
| None |
No relevant target |
LogP |
nan |
None |
10.1021/acs.jmedchem.7b01332 |
| None |
No relevant target |
-log(solubility) |
4.01 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
-log(solubility) |
4.02 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
-log(solubility) |
4.14 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
-log(solubility) |
4.21 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
-log(solubility) |
4.31 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
pKa |
2.2 |
None |
10.1124/dmd.110.035998 |
| None |
No relevant target |
pKa |
7.6 |
None |
10.1124/dmd.110.035998 |
| None |
No relevant target |
solubility |
nan |
None |
10.1016/j.bmc.2017.09.037 |
| None |
No relevant target |
Solubility |
1400.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.07.043 |
| None |
No relevant target |
Solubility |
1400.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.066 |
| None |
No relevant target |
Solubility |
1400.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.03.061 |
| None |
No relevant target |
Solubility |
1400.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.02.009 |
| None |
No relevant target |
Solubility |
174900.0 |
nM |
10.1016/j.ejmech.2022.114434 |
| None |
No relevant target |
Solubility |
183300.0 |
nM |
10.1016/j.ejmech.2020.112497 |
| None |
No relevant target |
Solubility |
751000.0 |
nM |
10.1021/acs.jmedchem.5b00050 |
| None |
Osteoblast |
Activity |
40.0 |
% |
10.1128/aac.00729-05 |
| None |
Osteoblast |
IC20 |
nan |
None |
10.1128/aac.00729-05 |
| None |
Osteoblast |
IC50 |
nan |
None |
10.1128/aac.00729-05 |
| None |
Phospholipidosis |
Phospholipidosis |
nan |
None |
10.1021/ci6004542 |
| None |
Phospholipidosis |
Phospholipidosis |
nan |
None |
10.1021/mp100103e |
| None |
Unchecked |
AbsAC90 |
6.43 |
uM |
None |
| None |
Unchecked |
Ac50 |
0.5623 |
uM |
None |
| None |
Unchecked |
Ac50 |
14.13 |
uM |
None |
| None |
Unchecked |
Ac50 |
19.95 |
uM |
None |
| None |
Unchecked |
Ac50 |
22.39 |
uM |
None |
| None |
Unchecked |
Ac50 |
28.18 |
uM |
None |
| None |
Unchecked |
Ac50 |
44.67 |
uM |
None |
| None |
Unchecked |
AC50 |
562.3 |
nM |
None |
| None |
Unchecked |
AC50 |
14130.0 |
nM |
None |
| None |
Unchecked |
AC50 |
19952.6 |
nM |
None |
| None |
Unchecked |
AC50 |
22387.2 |
nM |
None |
| None |
Unchecked |
AC50 |
28183.8 |
nM |
None |
| None |
Unchecked |
AC50 |
44668.4 |
nM |
None |
| None |
Unchecked |
Activity |
0.0 |
% |
10.1128/aac.00126-08 |
| None |
Unchecked |
Activity |
2.43 |
% |
10.1128/aac.00126-08 |
| None |
Unchecked |
Activity |
66.9 |
% |
10.1016/j.ejmech.2016.07.005 |
| None |
Unchecked |
Activity |
67.1 |
% |
10.1016/j.ejmech.2015.10.049 |
| None |
Unchecked |
Activity |
97.57 |
% |
10.1128/aac.00126-08 |
| None |
Unchecked |
Activity |
nan |
None |
10.1016/j.ejmech.2010.07.050 |
| None |
Unchecked |
Activity |
nan |
None |
10.1021/acs.jmedchem.1c02140 |
| None |
Unchecked |
Activity |
nan |
None |
10.1021/jm200201k |
| None |
Unchecked |
Activity |
nan |
None |
10.1124/mol.60.5.934 |
| None |
Unchecked |
CC50 |
72000.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| None |
Unchecked |
CC50 |
nan |
None |
10.1021/acs.jmedchem.2c01076 |
| None |
Unchecked |
FC |
8.0 |
None |
10.1016/j.ejmech.2022.114204 |
| None |
Unchecked |
FC |
64.0 |
None |
10.1021/acs.jmedchem.1c02140 |
| None |
Unchecked |
FC |
4096.0 |
None |
10.1016/j.ejmech.2022.114360 |
| None |
Unchecked |
FC |
500000.0 |
None |
10.1016/j.ejmech.2022.114204 |
| None |
Unchecked |
Hepatotoxicity (acute) |
38.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (association with vascular disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (choleostasis) |
19.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (chronic liver disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cirrhosis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (comment) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cytolytic) |
14.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (malignant tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (severe hepatitis) |
6.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (steatosis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (successful reintroduction) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
IC50 |
0.04 |
ug.mL-1 |
10.1128/aac.00343-07 |
| None |
Unchecked |
IC50 |
11.5 |
nM |
10.1128/aac.00753-10 |
| None |
Unchecked |
IC50 |
12.0 |
nM |
10.1021/jm4004889 |
| None |
Unchecked |
IC50 |
14.0 |
nM |
10.1021/acs.jmedchem.5b00050 |
| None |
Unchecked |
IC50 |
15.0 |
nM |
10.1021/acs.jmedchem.6b00485 |
| None |
Unchecked |
IC50 |
15.0 |
nM |
10.1128/aac.01649-07 |
| None |
Unchecked |
IC50 |
16.0 |
nM |
10.1021/jm400485e |
| None |
Unchecked |
IC50 |
17.0 |
nM |
10.1021/jm4004889 |
| None |
Unchecked |
IC50 |
27.0 |
nM |
10.1021/jm400485e |
| None |
Unchecked |
IC50 |
30.0 |
nM |
10.1016/j.ejmech.2013.04.060 |
| None |
Unchecked |
IC50 |
30.0 |
nM |
10.1021/jm400485e |
| None |
Unchecked |
IC50 |
30.0 |
nM |
10.1021/ml5001933 |
| None |
Unchecked |
IC50 |
62.92 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| None |
Unchecked |
IC50 |
80.0 |
nM |
10.1021/ml300350p |
| None |
Unchecked |
IC50 |
140.0 |
nM |
10.1016/j.bmcl.2020.127146 |
| None |
Unchecked |
IC50 |
6410.0 |
nM |
None |
| None |
Unchecked |
IC50 |
7420.0 |
nM |
None |
| None |
Unchecked |
IC50 |
8940.0 |
nM |
None |
| None |
Unchecked |
IC50 |
9700.0 |
nM |
None |
| None |
Unchecked |
IC50 |
10350.0 |
nM |
None |
| None |
Unchecked |
IC50 |
25000.0 |
nM |
10.1016/j.bmc.2016.09.012 |
| None |
Unchecked |
IC50 |
25000.0 |
nM |
10.1016/j.bmc.2017.11.031 |
| None |
Unchecked |
IC50 |
25000.0 |
nM |
10.1016/j.ejmech.2017.12.088 |
| None |
Unchecked |
IC50 |
25000.0 |
nM |
10.1021/acs.jmedchem.6b00485 |
| None |
Unchecked |
IC50 |
25000.0 |
nM |
10.1128/aac.01649-07 |
| None |
Unchecked |
IC50 |
32559.0 |
nM |
None |
| None |
Unchecked |
IC50 |
52100.0 |
nM |
10.1016/j.bmcl.2011.08.054 |
| None |
Unchecked |
IC50 |
63000.0 |
nM |
10.1021/acs.jmedchem.8b01293 |
| None |
Unchecked |
IC50 |
109000.0 |
nM |
10.1021/jm4004889 |
| None |
Unchecked |
IC50 |
126000.0 |
nM |
10.1021/jm201716n |
| None |
Unchecked |
IC50 |
313000.0 |
nM |
10.1021/jm201716n |
| None |
Unchecked |
IC50 |
465000.0 |
nM |
10.1021/jm4004889 |
| None |
Unchecked |
IC50 |
500000.0 |
nM |
10.1016/j.ejmech.2021.113568 |
| None |
Unchecked |
IC50 |
610000.0 |
nM |
10.1021/jm4004889 |
| None |
Unchecked |
IC50 |
830000.0 |
nM |
10.1021/jm201716n |
| None |
Unchecked |
IC50 |
nan |
None |
10.1016/j.bmc.2015.02.032 |
| None |
Unchecked |
IC50 |
nan |
None |
10.1016/j.ejmech.2014.12.046 |
| None |
Unchecked |
IC50 |
nan |
None |
10.1016/j.ejmech.2016.06.042 |
| None |
Unchecked |
IC50 |
nan |
None |
10.1021/ml5001728 |
| None |
Unchecked |
IC50 |
nan |
None |
None |
| None |
Unchecked |
Inhibition |
5.0 |
% |
10.1021/jm400485e |
| None |
Unchecked |
Inhibition |
7.8 |
% |
10.1128/aac.00753-10 |
| None |
Unchecked |
Inhibition |
8.3 |
% |
10.1128/aac.00753-10 |
| None |
Unchecked |
Inhibition |
69.6 |
% |
10.1016/j.bmc.2014.12.060 |
| None |
Unchecked |
Inhibition |
95.0 |
% |
10.1016/j.bmcl.2009.12.045 |
| None |
Unchecked |
Inhibition |
nan |
% |
10.1016/j.ejmech.2020.112671 |
| None |
Unchecked |
Kd |
195000.0 |
nM |
10.1021/jm991174y |
| None |
Unchecked |
Ki |
nan |
None |
None |
| None |
Unchecked |
logIC50 |
1.717 |
None |
10.1016/j.bmcl.2011.08.054 |
| None |
Unchecked |
MIC |
0.004 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| None |
Unchecked |
MIC |
0.1 |
ug.mL-1 |
10.1021/acs.jnatprod.1c00812 |
| None |
Unchecked |
MIC |
9.24 |
ug.mL-1 |
10.1021/acs.jmedchem.1c00263 |
| None |
Unchecked |
MIC |
10.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c00263 |
| None |
Unchecked |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c02045 |
| None |
Unchecked |
MIC |
50.0 |
nM |
10.1016/j.ejmech.2020.112179 |
| None |
Unchecked |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.001 |
| None |
Unchecked |
MIC |
190.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| None |
Unchecked |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| None |
Unchecked |
MIC |
4000.0 |
nM |
10.1021/acs.jmedchem.1c02122 |
| None |
Unchecked |
MIC |
12200.0 |
nM |
10.1016/j.ejmech.2020.112179 |
| None |
Unchecked |
MIC |
48600.0 |
nM |
10.1016/j.ejmech.2020.112179 |
| None |
Unchecked |
MIC100 |
0.01 |
ug ml-1 |
10.1016/j.ejmech.2020.112420 |
| None |
Unchecked |
MIC=>90 |
0.015 |
ug ml-1 |
10.1016/j.ejmech.2020.112538 |
| None |
Unchecked |
MIC=>90 |
9.317 |
ug ml-1 |
10.1016/j.ejmech.2020.112538 |
| None |
Unchecked |
MIC=>90 |
10.0 |
ug ml-1 |
10.1016/j.ejmech.2020.112538 |
| None |
Unchecked |
PI |
256.0 |
None |
10.1016/j.ejmech.2009.06.005 |
| None |
Unchecked |
PI |
828.12 |
None |
10.1016/j.bmc.2010.09.006 |
| None |
Unchecked |
Potency |
1778.3 |
nM |
None |
| None |
Unchecked |
Potency |
10322.5 |
nM |
None |
| None |
Unchecked |
Potency |
15848.9 |
nM |
None |
| None |
Unchecked |
Potency |
18356.4 |
nM |
None |
| None |
Unchecked |
Potency |
25929.0 |
nM |
None |
| None |
Unchecked |
Ratio |
0.054 |
None |
10.1093/toxsci/kft176 |
| None |
Unchecked |
Ratio |
0.07 |
None |
10.1093/toxsci/kft176 |
| None |
Unchecked |
Ratio |
0.089 |
None |
10.1093/toxsci/kft176 |
| None |
Unchecked |
Ratio |
0.147 |
None |
10.1093/toxsci/kft176 |
| None |
Unchecked |
Ratio |
0.27 |
None |
10.1128/aac.00120-07 |
| None |
Unchecked |
Ratio |
0.75 |
None |
10.1016/j.bmcl.2022.128692 |
| None |
Unchecked |
Ratio |
0.83 |
None |
10.1016/j.bmcl.2022.128692 |
| None |
Unchecked |
Ratio |
0.93 |
None |
10.1016/j.bmcl.2022.128692 |
| None |
Unchecked |
Ratio |
1.09 |
None |
10.1016/j.bmcl.2022.128692 |
| None |
Unchecked |
Ratio |
2.0 |
None |
10.1021/acs.jmedchem.9b00288 |
| None |
Unchecked |
Ratio |
3.94 |
None |
10.1128/aac.00367-09 |
| None |
Unchecked |
Ratio |
4.16 |
None |
10.1128/aac.00367-09 |
| None |
Unchecked |
Ratio |
6.19 |
None |
10.1128/aac.00367-09 |
| None |
Unchecked |
Ratio |
10.07 |
None |
10.1128/aac.00367-09 |
| None |
Unchecked |
Ratio |
61.2 |
None |
10.1128/aac.00120-07 |
| None |
Unchecked |
Ratio |
64.1 |
None |
10.1128/aac.01533-06 |
| None |
Unchecked |
Ratio |
100.0 |
None |
10.1016/j.bmcl.2013.07.006 |
| None |
Unchecked |
Ratio |
100.0 |
None |
10.1128/aac.00775-08 |
| None |
Unchecked |
Ratio |
224.36 |
None |
10.1128/aac.01533-06 |
| None |
Unchecked |
Ratio |
256.0 |
None |
10.1021/jm701560p |
| None |
Unchecked |
Ratio |
440.0 |
None |
10.1128/aac.00458-08 |
| None |
Unchecked |
Ratio |
448.72 |
None |
10.1128/aac.01533-06 |
| None |
Unchecked |
Ratio |
460.0 |
None |
10.1128/aac.00775-08 |
| None |
Unchecked |
Ratio |
465.0 |
None |
10.1128/aac.01533-06 |
| None |
Unchecked |
Ratio |
800.0 |
None |
10.1016/j.bmc.2008.10.086 |
| None |
Unchecked |
Ratio |
16250.0 |
None |
10.1016/j.bmcl.2009.09.095 |
| None |
Unchecked |
Ratio |
16256.0 |
None |
10.1016/j.bmcl.2009.09.095 |
| None |
Unchecked |
Ratio |
20260.0 |
None |
10.1128/aac.00458-08 |
| None |
Unchecked |
Ratio |
44510.0 |
None |
10.1016/j.bmcl.2009.09.095 |
| None |
Unchecked |
RatioAUC/MIC |
24.14 |
None |
10.1128/aac.01533-06 |
| None |
Unchecked |
RatioAUC/MIC |
169.0 |
None |
10.1128/aac.01533-06 |
| None |
Unchecked |
RatioAUC/MIC |
224.36 |
None |
10.1128/aac.01533-06 |
| None |
Unchecked |
RatioAUC/MIC |
448.72 |
None |
10.1128/aac.01533-06 |
| None |
Unchecked |
Ratio IC50 |
1.0 |
None |
10.1021/jm400485e |
| None |
Unchecked |
Ratio IC50 |
61.0 |
None |
10.1021/jm900340a |
| None |
Unchecked |
Ratio IC50 |
1080.0 |
None |
10.1016/j.bmc.2010.03.018 |
| None |
Unchecked |
Ratio IC50 |
1220.0 |
None |
10.1021/jm900340a |
| None |
Unchecked |
Ratio IC50 |
2033.0 |
None |
10.1021/jm901235p |
| None |
Unchecked |
Selectivity index |
8000.0 |
SI |
10.1016/s0960-894x(01)00266-9 |
| None |
Unchecked |
Selectivity Index |
8.0 |
None |
10.1016/j.ejmech.2019.111678 |
| None |
Unchecked |
Selectivity Index |
10.0 |
None |
10.1007/s00044-012-0074-2 |
| None |
Unchecked |
Selectivity Index |
61.0 |
None |
10.1016/j.bmcl.2009.11.105 |
| None |
Unchecked |
Selectivity Index |
112.35 |
None |
10.1016/j.bmcl.2016.03.045 |
| None |
Unchecked |
Selectivity Index |
123.0 |
None |
10.1016/j.bmcl.2016.11.056 |
| None |
Unchecked |
Selectivity Index |
123.0 |
None |
10.1016/j.bmcl.2017.01.004 |
| None |
Unchecked |
Selectivity Index |
123.0 |
None |
10.1016/j.ejmech.2017.03.065 |
| None |
Unchecked |
Selectivity Index |
133.0 |
None |
10.1016/j.bmcl.2016.11.056 |
| None |
Unchecked |
Selectivity Index |
133.0 |
None |
10.1016/j.bmcl.2017.01.004 |
| None |
Unchecked |
Selectivity Index |
133.0 |
None |
10.1016/j.ejmech.2017.01.009 |
| None |
Unchecked |
Selectivity Index |
133.0 |
None |
10.1016/j.ejmech.2017.03.065 |
| None |
Unchecked |
Selectivity Index |
138.88 |
None |
10.1016/j.bmcl.2016.03.045 |
| None |
Unchecked |
Selectivity Index |
196.0 |
None |
10.1016/j.bmcl.2016.11.056 |
| None |
Unchecked |
Selectivity Index |
196.0 |
None |
10.1016/j.ejmech.2017.01.009 |
| None |
Unchecked |
Selectivity Index |
196.0 |
None |
10.1039/C5MD00404G |
| None |
Unchecked |
Selectivity Index |
208.0 |
None |
10.1016/j.ejmech.2017.01.009 |
| None |
Unchecked |
Selectivity Index |
222.0 |
None |
10.1016/j.bmcl.2016.11.056 |
| None |
Unchecked |
Selectivity Index |
222.0 |
None |
10.1039/C5MD00404G |
| None |
Unchecked |
Selectivity Index |
244.0 |
None |
10.1016/j.ejmech.2017.01.009 |
| None |
Unchecked |
Selectivity Index |
400.0 |
None |
10.1016/j.ejmech.2009.10.050 |
| None |
Unchecked |
Selectivity Index |
512.0 |
None |
10.1016/j.bmcl.2019.07.041 |
| None |
Unchecked |
Selectivity Index |
512.0 |
None |
10.1016/j.ejmech.2019.07.057 |
| None |
Unchecked |
Selectivity Index |
526.31 |
None |
10.1021/jm401735w |
| None |
Unchecked |
Selectivity Index |
714.0 |
None |
10.1016/j.bmcl.2016.05.093 |
| None |
Unchecked |
Selectivity Index |
800.0 |
None |
10.1016/j.bmc.2008.08.050 |
| None |
Unchecked |
Selectivity Index |
800.0 |
None |
10.1016/j.ejmech.2010.06.036 |
| None |
Unchecked |
Selectivity Index |
909.0 |
None |
10.1016/j.bmcl.2012.06.095 |
| None |
Unchecked |
Selectivity Index |
947.0 |
None |
10.1016/j.ejmech.2010.11.023 |
| None |
Unchecked |
Selectivity Index |
1000.0 |
None |
10.1016/j.bmc.2018.07.034 |
| None |
Unchecked |
Selectivity Index |
1024.0 |
None |
10.1016/j.bmc.2019.04.017 |
| None |
Unchecked |
Selectivity Index |
1024.0 |
None |
10.1016/j.ejmech.2018.09.049 |
| None |
Unchecked |
Selectivity Index |
1100.0 |
None |
10.1016/j.bmcl.2015.12.080 |
| None |
Unchecked |
Selectivity Index |
1167.0 |
None |
10.1007/s00044-007-9073-0 |
| None |
Unchecked |
Selectivity Index |
1220.0 |
None |
10.1016/j.bmcl.2009.11.105 |
| None |
Unchecked |
Selectivity Index |
1250.0 |
None |
10.1016/j.bmcl.2016.05.093 |
| None |
Unchecked |
Selectivity Index |
1250.0 |
None |
10.1021/np400497f |
| None |
Unchecked |
Selectivity Index |
1312.0 |
None |
10.1016/j.ejmech.2017.11.090 |
| None |
Unchecked |
Selectivity Index |
1363.4 |
None |
10.1016/j.ejmech.2015.10.024 |
| None |
Unchecked |
Selectivity Index |
1488.0 |
None |
10.1016/j.bmcl.2008.09.029 |
| None |
Unchecked |
Selectivity Index |
1543.0 |
None |
10.1016/j.bmcl.2013.09.013 |
| None |
Unchecked |
Selectivity Index |
1754.4 |
None |
10.1039/C6MD00278A |
| None |
Unchecked |
Selectivity Index |
2000.0 |
None |
10.1016/j.ejmech.2017.05.026 |
| None |
Unchecked |
Selectivity Index |
2050.0 |
None |
10.1021/acs.jmedchem.7b00582 |
| None |
Unchecked |
Selectivity Index |
2325.5 |
None |
10.1016/j.bmcl.2015.11.071 |
| None |
Unchecked |
Selectivity Index |
2439.0 |
None |
10.1016/j.bmcl.2015.11.071 |
| None |
Unchecked |
Selectivity Index |
2500.0 |
None |
10.1016/j.bmc.2016.12.038 |
| None |
Unchecked |
Selectivity Index |
2500.0 |
None |
10.1016/j.ejmech.2016.09.059 |
| None |
Unchecked |
Selectivity Index |
2702.7 |
None |
10.1016/j.bmcl.2016.02.043 |
| None |
Unchecked |
Selectivity Index |
2857.1 |
None |
10.1016/j.bmcl.2016.02.043 |
| None |
Unchecked |
Selectivity Index |
2857.14 |
None |
10.1016/j.bmcl.2016.02.043 |
| None |
Unchecked |
Selectivity Index |
4066.0 |
None |
10.1021/acs.jnatprod.9b01095 |
| None |
Unchecked |
Selectivity Index |
5000.0 |
None |
10.1039/C6MD00278A |
| None |
Unchecked |
Selectivity Index |
6564.0 |
None |
10.1016/j.ejmech.2019.01.042 |
| None |
Unchecked |
Selectivity Index |
12500.0 |
None |
10.1021/acsmedchemlett.8b00410 |
| None |
Unchecked |
Selectivity Index |
14000.0 |
None |
10.1016/j.bmc.2015.04.001 |
| None |
Unchecked |
Selectivity Index |
14000.0 |
None |
10.1039/C3MD00251A |
| None |
Unchecked |
Selectivity Index |
15000.0 |
None |
10.1021/jm300123s |
| None |
Unchecked |
Selectivity Index |
34400.0 |
None |
10.1016/j.ejmech.2020.112045 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.bmc.2019.07.045 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.bmcl.2019.02.019 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.ejmech.2016.07.039 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1021/acs.jmedchem.7b01332 |
| None |
Unchecked |
Selectivity ratio |
1.1 |
None |
10.1021/acs.jmedchem.2c00266 |
| None |
Unchecked |
Selectivity ratio |
1.3 |
None |
10.1021/acs.jmedchem.2c00266 |
| None |
Unchecked |
Selectivity ratio |
98.0 |
None |
10.1016/j.bmc.2008.12.006 |
| None |
Unchecked |
Selectivity ratio |
500.0 |
None |
10.1039/C7MD00350A |
| None |
Unchecked |
Selectivity ratio |
500.0 |
None |
10.1039/C7MD00366H |
| None |
Unchecked |
Selectivity ratio |
800.0 |
None |
10.1016/j.bmc.2010.02.024 |
| None |
Unchecked |
Time |
nan |
None |
10.1128/aac.00620-10 |
| None |
Unchecked |
TIME |
0.005556 |
hr |
10.1128/aac.00620-10 |