Rifampicin

AlkaPlorer ID: AK017872

Synonym: None

IUPAC Name: [(7S,9E,11S,12R,13S,14R,15R,16R,17S,18S,19E,21Z)-2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-[(Z)-(4-methylpiperazin-1-yl)iminomethyl]-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate

Structure

SMILES: CO[C@H]1/C=C/O[C@@]2(C)OC3=C(C)C(O)=C4C(O)=C(N=C(O)/C(C)=C\C=C\[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C)C(/C=N/N1CCN(C)CC1)=C(O)C4=C3C2=O

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InChI: InChI=1S/C43H58N4O12/c1-21-12-11-13-22(2)42(55)45-33-28(20-44-47-17-15-46(9)16-18-47)37(52)30-31(38(33)53)36(51)26(6)40-32(30)41(54)43(8,59-40)57-19-14-29(56-10)23(3)39(58-27(7)48)25(5)35(50)24(4)34(21)49/h11-14,19-21,23-25,29,34-35,39,49-53H,15-18H2,1-10H3,(H,45,55)/b12-11+,19-14+,22-13-,44-20+/t21-,23+,24+,25+,29-,34-,35+,39+,43-/m0/s1

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InChIKey: JQXXHWHPUNPDRT-WLSIYKJHSA-N

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Properties Information

Molecule Weight: 822.9529999999996

TPSA: 223.64

MolLogP: 4.984920000000005

Number of H-Donors: 6

Number of H-Acceptors: 15

RingCount: 6

Activities Information

Organism Target Name Standard Type Standard Value Standard Units doi
Acinetobacter baumannii Acinetobacter baumannii Activity 2.0 log10CFU/g 10.1016/j.bmcl.2022.129113
Acinetobacter baumannii Acinetobacter baumannii Activity 3.5 log10CFU/ml 10.1128/aac.00367-09
Acinetobacter baumannii Acinetobacter baumannii Activity 4.5 log10CFU/ml 10.1128/aac.00367-09
Acinetobacter baumannii Acinetobacter baumannii Activity 5.1 log10CFU/ml 10.1128/aac.00367-09
Acinetobacter baumannii Acinetobacter baumannii Activity 6.0 log10CFU/g 10.1016/j.bmcl.2022.129113
Acinetobacter baumannii Acinetobacter baumannii Activity 78.6 % 10.1128/aac.00367-09
Acinetobacter baumannii Acinetobacter baumannii Activity nan None 10.1128/aac.00367-09
Acinetobacter baumannii Acinetobacter baumannii Activity nan None 10.1128/aac.01099-06
Acinetobacter baumannii Acinetobacter baumannii EC50 470.0 nM 10.1016/j.bmcl.2016.04.089
Acinetobacter baumannii Acinetobacter baumannii EC50 1300.0 nM 10.1021/acs.jmedchem.8b01293
Acinetobacter baumannii Acinetobacter baumannii FICI 0.105 None 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii FICI 0.126 None 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii FICI 0.131 None 10.1128/aac.01439-09
Acinetobacter baumannii Acinetobacter baumannii Inhibition 10.0 % 10.1128/aac.00471-08
Acinetobacter baumannii Acinetobacter baumannii Inhibition nan % 10.1128/aac.00471-08
Acinetobacter baumannii Acinetobacter baumannii log10cfu 8.15 None 10.1128/aac.00471-08
Acinetobacter baumannii Acinetobacter baumannii MBC 3.13 ug ml-1 10.1016/j.bmc.2018.07.034
Acinetobacter baumannii Acinetobacter baumannii MBC 4.0 mg/L 10.1128/aac.00367-09
Acinetobacter baumannii Acinetobacter baumannii MBC 8.0 mg/L 10.1128/aac.00367-09
Acinetobacter baumannii Acinetobacter baumannii MBC nan None 10.1021/acs.jnatprod.2c00065
Acinetobacter baumannii Acinetobacter baumannii MIC 0.006 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.008 ug.mL-1 10.1128/aac.00471-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.016 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.03 ug.mL-1 10.1021/acs.jnatprod.1c00578
Acinetobacter baumannii Acinetobacter baumannii MIC 0.03 ug.mL-1 10.1021/acs.jnatprod.2c00621
Acinetobacter baumannii Acinetobacter baumannii MIC 0.031 ug.mL-1 10.1021/acs.jmedchem.9b00876
Acinetobacter baumannii Acinetobacter baumannii MIC 0.032 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.047 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.094 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.094 ug.mL-1 10.1128/aac.01439-09
Acinetobacter baumannii Acinetobacter baumannii MIC 0.125 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.19 ug.mL-1 10.1128/aac.01439-09
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1016/j.ejmech.2018.08.070
Acinetobacter baumannii Acinetobacter baumannii MIC 0.25 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.38 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 0.5 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 1.0 ug.mL-1 10.1021/acs.jnatprod.2c00065
Acinetobacter baumannii Acinetobacter baumannii MIC 1.5 ug.mL-1 10.1128/aac.00732-07
Acinetobacter baumannii Acinetobacter baumannii MIC 1.5 ug.mL-1 10.1128/aac.01037-09
Acinetobacter baumannii Acinetobacter baumannii MIC 1.5 ug.mL-1 10.1128/aac.01439-09
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1021/acs.jmedchem.6b01742
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1021/acs.jmedchem.9b00876
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1021/acs.jnatprod.1c00578
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1021/acs.jnatprod.2c00621
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.00072-08
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.00732-07
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.00748-09
Acinetobacter baumannii Acinetobacter baumannii MIC 2.0 ug.mL-1 10.1128/aac.01037-09
Acinetobacter baumannii Acinetobacter baumannii MIC 3.0 ug.mL-1 10.1128/aac.01037-09
Acinetobacter baumannii Acinetobacter baumannii MIC 3.0 ug.mL-1 10.1128/aac.01121-08
Acinetobacter baumannii Acinetobacter baumannii MIC 3.1 ug.mL-1 10.1021/acs.jnatprod.0c01212
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1016/j.ejmech.2018.08.070
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1016/j.ejmech.2019.05.090
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.00367-09
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.00732-07
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.01037-09
Acinetobacter baumannii Acinetobacter baumannii MIC 4.0 ug.mL-1 10.1128/aac.01259-06
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.00367-09
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.01259-06
Acinetobacter baumannii Acinetobacter baumannii MIC 8.0 ug.mL-1 10.1128/aac.01663-08
Acinetobacter baumannii Acinetobacter baumannii MIC 12.0 ug.mL-1 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.01037-09
Acinetobacter baumannii Acinetobacter baumannii MIC 16.0 ug.mL-1 10.1128/aac.01259-06
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.01037-09
Acinetobacter baumannii Acinetobacter baumannii MIC 32.0 ug.mL-1 10.1128/aac.01259-06
Acinetobacter baumannii Acinetobacter baumannii MIC 64.0 ug.mL-1 10.1016/j.ejmech.2022.114360
Acinetobacter baumannii Acinetobacter baumannii MIC 128.0 ug.mL-1 10.1128/aac.01259-06
Acinetobacter baumannii Acinetobacter baumannii MIC 128.0 ug.mL-1 10.1128/aac.01663-08
Acinetobacter baumannii Acinetobacter baumannii MIC 256.0 ug.mL-1 10.1021/acs.jmedchem.6b01742
Acinetobacter baumannii Acinetobacter baumannii MIC 256.0 ug.mL-1 10.1128/aac.01259-06
Acinetobacter baumannii Acinetobacter baumannii MIC 1000.0 nM 10.1021/acs.jmedchem.1c00614
Acinetobacter baumannii Acinetobacter baumannii MIC 1000.0 nM 10.1021/acs.jmedchem.1c02122
Acinetobacter baumannii Acinetobacter baumannii MIC 1000.0 nM 10.1021/acs.jmedchem.9b00288
Acinetobacter baumannii Acinetobacter baumannii MIC 3800.0 nM 10.1021/acs.jnatprod.1c00232
Acinetobacter baumannii Acinetobacter baumannii MIC nan None 10.1016/j.ejmech.2019.04.067
Acinetobacter baumannii Acinetobacter baumannii MIC100 2.35 ug ml-1 10.1016/j.bmc.2018.07.034
Acinetobacter baumannii Acinetobacter baumannii MIC50 4.0 ug.mL-1 10.1128/aac.01099-06
Acinetobacter baumannii Acinetobacter baumannii MIC80 1.0 ug.mL-1 10.1021/np401094h
Acinetobacter baumannii Acinetobacter baumannii MIC90 8.0 ug.mL-1 10.1128/aac.01099-06
Acinetobacter baumannii Acinetobacter baumannii Ratio 1.0 None 10.1128/aac.00748-09
Acinetobacter baumannii Acinetobacter baumannii Ratio 16.0 None 10.1128/aac.01439-09
Acinetobacter baumannii Acinetobacter baumannii Ratio 21.0 None 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii Ratio 24.0 None 10.1128/aac.00405-08
Acinetobacter baumannii Acinetobacter baumannii Survival 50.0 % 10.1016/j.bmcl.2022.129113
Acinetobacter baumannii Acinetobacter baumannii Survival 71.4 % 10.1128/aac.00367-09
Acinetobacter baumannii Acinetobacter baumannii Survival 90.0 % 10.1016/j.bmcl.2022.129113
Acinetobacter pittii Acinetobacter pittii MIC 2.0 ug.mL-1 10.1128/aac.00072-08
Actinomyces naeslundii Actinomyces naeslundii MIC 0.03 ug.mL-1 10.1021/acs.jmedchem.1c02045
Bacillus anthracis Bacillus anthracis Activity nan None 10.1128/aac.00067-10
Bacillus anthracis Bacillus anthracis MIC 0.25 ug.mL-1 10.1021/acs.jnatprod.0c01309
Bacillus anthracis Bacillus anthracis MIC 31.0 ug.mL-1 10.1016/j.ejmech.2019.04.043
Bacillus cereus Bacillus cereus MBC nan None 10.1021/acs.jnatprod.2c00065
Bacillus cereus Bacillus cereus MIC 0.03 ug.mL-1 10.1128/aac.00360-08
Bacillus cereus Bacillus cereus MIC 0.25 ug.mL-1 10.1021/acs.jnatprod.2c00065
Bacillus cereus Bacillus cereus MIC 0.25 ug.mL-1 10.1128/aac.00360-08
Bacillus cereus Bacillus cereus MIC nan None 10.1016/j.bmc.2010.05.016
Bacillus cereus Bacillus cereus MIC nan None 10.1016/j.bmc.2013.10.011
Bacillus cereus Bacillus cereus Ratio 8.0 None 10.1128/aac.00360-08
Bacillus licheniformis Bacillus licheniformis IZ 24.0 mm 10.1016/j.bmcl.2016.04.038
Bacillus pumilus Bacillus pumilus MIC 128.0 ug.mL-1 10.1128/aac.00389-08
Bacillus spizizenii Bacillus spizizenii IZ 13.0 mm 10.1016/j.bmc.2018.02.049
Bacillus spizizenii Bacillus spizizenii IZ 25.0 mm 10.1021/ml300350p
Bacillus spizizenii Bacillus spizizenii MIC 0.125 ug.mL-1 10.1016/j.bmc.2018.02.049
Bacillus spizizenii Bacillus spizizenii MIC 0.125 ug.mL-1 10.1021/ml300350p
Bacillus subtilis Bacillus subtilis Activity 25.0 % 10.1021/np020380x
Bacillus subtilis Bacillus subtilis Activity 29.0 % 10.1021/np020380x
Bacillus subtilis Bacillus subtilis Activity 90.0 % 10.1021/np020380x
Bacillus subtilis Bacillus subtilis Activity 94.0 % 10.1021/np020380x
Bacillus subtilis Bacillus subtilis Activity 108.0 % 10.1021/np020380x
Bacillus subtilis Bacillus subtilis Activity 143.0 % 10.1021/np020380x
Bacillus subtilis Bacillus subtilis Activity nan None 10.1021/acs.jnatprod.7b00477
Bacillus subtilis Bacillus subtilis FC 2.0 None 10.1016/j.bmc.2016.05.021
Bacillus subtilis Bacillus subtilis GI 100.0 % 10.1016/j.bmc.2016.01.040
Bacillus subtilis Bacillus subtilis Inhibition 100.0 % 10.1021/jm0703901
Bacillus subtilis Bacillus subtilis Inhibition nan % 10.1021/acs.jmedchem.7b00355
Bacillus subtilis Bacillus subtilis Inhibition nan % 10.1128/aac.01709-08
Bacillus subtilis Bacillus subtilis IZ 20.0 mm 10.1016/j.bmc.2007.09.025
Bacillus subtilis Bacillus subtilis IZ 51.0 mm 10.1016/j.ejmech.2008.09.035
Bacillus subtilis Bacillus subtilis log(1/C) 6.59 None 10.1021/jm00210a025
Bacillus subtilis Bacillus subtilis MBC 0.4 ug ml-1 10.1016/j.bmc.2018.07.034
Bacillus subtilis Bacillus subtilis MIC 0.01 ug.mL-1 10.1128/aac.00873-08
Bacillus subtilis Bacillus subtilis MIC 0.078 ug.mL-1 10.1021/acs.jnatprod.2c00174
Bacillus subtilis Bacillus subtilis MIC 0.1 ug.mL-1 10.1128/aac.00873-08
Bacillus subtilis Bacillus subtilis MIC 0.12 ug.mL-1 10.1016/j.ejmech.2007.12.019
Bacillus subtilis Bacillus subtilis MIC 0.125 ug.mL-1 10.1016/j.bmcl.2020.127146
Bacillus subtilis Bacillus subtilis MIC 0.125 ug.mL-1 10.1016/j.ejmech.2022.114360
Bacillus subtilis Bacillus subtilis MIC 0.19 ug.mL-1 10.1007/s00044-011-9918-4
Bacillus subtilis Bacillus subtilis MIC 0.21 ug.mL-1 10.1021/jm00210a025
Bacillus subtilis Bacillus subtilis MIC 0.25 ug.mL-1 10.1021/acsmedchemlett.0c00381
Bacillus subtilis Bacillus subtilis MIC 3.125 ug.mL-1 10.1007/s00044-011-9918-4
Bacillus subtilis Bacillus subtilis MIC 3.9 ug.mL-1 10.1016/j.ejmech.2007.12.019
Bacillus subtilis Bacillus subtilis MIC 5.0 ug.mL-1 10.1021/jm400485e
Bacillus subtilis Bacillus subtilis MIC 10.0 ug.mL-1 10.1016/j.ejmech.2008.09.035
Bacillus subtilis Bacillus subtilis MIC 16.0 ug.mL-1 10.1016/j.bmc.2006.12.035
Bacillus subtilis Bacillus subtilis MIC 21.0 ug.mL-1 10.1016/j.bmcl.2017.05.032
Bacillus subtilis Bacillus subtilis MIC 62.5 nM 10.1016/j.bmc.2016.05.021
Bacillus subtilis Bacillus subtilis MIC 64.0 ug.mL-1 10.1016/j.ejmech.2008.04.001
Bacillus subtilis Bacillus subtilis MIC 125.0 nM 10.1016/j.bmc.2016.05.021
Bacillus subtilis Bacillus subtilis MIC 250.0 nM 10.1016/j.bmc.2016.05.021
Bacillus subtilis Bacillus subtilis MIC 256.0 ug.mL-1 10.1016/j.bmc.2006.12.035
Bacillus subtilis Bacillus subtilis MIC 256.0 ug.mL-1 10.1016/j.ejmech.2008.04.001
Bacillus subtilis Bacillus subtilis MIC 1000.0 nM 10.1016/j.ejmech.2019.111636
Bacillus subtilis Bacillus subtilis MIC 1000.0 nM 10.1021/acs.jmedchem.1c00614
Bacillus subtilis Bacillus subtilis MIC 1000.0 nM 10.1021/acs.jmedchem.1c02140
Bacillus subtilis Bacillus subtilis MIC 1000.0 nM 10.1021/acs.jmedchem.2c01076
Bacillus subtilis Bacillus subtilis MIC 1000.0 nM 10.1021/jm030003x
Bacillus subtilis Bacillus subtilis MIC 1500.0 nM 10.1021/jm061349l
Bacillus subtilis Bacillus subtilis MIC 4000.0 nM 10.1021/acs.jmedchem.1c02122
Bacillus subtilis Bacillus subtilis MIC nan None 10.1016/j.bmc.2016.04.058
Bacillus subtilis Bacillus subtilis MIC nan None 10.1016/j.bmcl.2012.08.003
Bacillus subtilis Bacillus subtilis MIC100 0.3 ug ml-1 10.1016/j.bmc.2018.07.034
Bacillus subtilis (strain 168) NH(3)-dependent NAD(+) synthetase IC50 1000.0 nM 10.1021/jm030003x
Bacteria Cell membrane Activity 3.45 % 10.1021/acs.jmedchem.2c01076
Bacteria Cell membrane Activity 17.4 % 10.1021/acs.jmedchem.2c01076
Bacteria Cell membrane Activity nan None 10.1021/acs.jmedchem.2c01076
Bacteria Cell membrane Activity nan None 10.1021/acs.jmedchem.8b00777
Bacteroides fragilis Bacteroides fragilis MIC 0.25 ug.mL-1 10.1021/acs.jmedchem.1c02045
Bacteroides fragilis Bacteroides fragilis MIC nan None 10.1021/np050424c
Bacteroides ovatus Bacteroides ovatus MIC 1.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC 0.5 ug.mL-1 10.1021/acs.jmedchem.1c02045
Bacteroides thetaiotaomicron Bacteroides thetaiotaomicron MIC nan None 10.1021/np050424c
Bacteroides uniformis Bacteroides uniformis MIC 0.5 ug.mL-1 10.1021/acs.jmedchem.1c02045
Bifidobacterium breve Bifidobacterium breve MIC 0.25 ug.mL-1 10.1021/acs.jmedchem.1c02045
Bifidobacterium longum Bifidobacterium longum MIC 0.5 ug.mL-1 10.1021/acs.jmedchem.1c02045
Bos taurus Progesterone receptor IC50 nan None None
Bos taurus Progesterone receptor Ki nan None None
Burkholderia cepacia Burkholderia cepacia Activity 1.0 % 10.1128/aac.00954-06
Candida albicans Candida albicans IC50 nan None 10.1021/jm900672t
Candida albicans Candida albicans IC50 nan None 10.1021/np000436s
Candida albicans Candida albicans IZ 0.0 mm 10.1021/np900382x
Candida albicans Candida albicans MIC 1.0 ug.mL-1 10.1016/j.ejmech.2014.07.066
Candida albicans Candida albicans MIC 3.9 ug.mL-1 10.1016/j.bmcl.2016.02.024
Candida albicans Candida albicans MIC 64.0 ug.mL-1 10.1016/j.bmcl.2020.127146
Candida albicans Candida albicans MIC 256.0 ug.mL-1 10.1021/ml300350p
Candida albicans Candida albicans MIC nan None 10.1016/j.bmcl.2012.08.003
Candida albicans Candida albicans MIC nan None 10.1016/j.bmcl.2012.09.041
Candida albicans Candida albicans MIC nan None 10.1016/j.bmcl.2013.11.024
Candida albicans Candida albicans MIC nan None 10.1016/j.bmcl.2015.01.026
Candida albicans Candida albicans MIC nan None 10.1021/acs.jnatprod.5b01129
Candida albicans Candida albicans MIC nan None 10.1021/np000436s
Canis lupus familiaris Brain Fu 0.259 None 10.1124/dmd.111.038778
Cavia porcellus Cavia porcellus AUC 6.22 None 10.1128/aac.00196-08
Cavia porcellus Cavia porcellus Cmax 741.24 nM 10.1128/aac.00120-07
Cavia porcellus Cavia porcellus Cmax 1190.84 nM 10.1128/aac.00120-07
Cavia porcellus Cavia porcellus Cmin 0.14 ug ml-1 10.1128/aac.00120-07
Cavia porcellus Cavia porcellus Cmin 0.22 ug ml-1 10.1128/aac.00120-07
Cavia porcellus Cavia porcellus T1/2 3.0 hr 10.1128/aac.01533-06
Cavia porcellus Cavia porcellus T1/2 5.8 hr 10.1128/aac.00120-07
Cavia porcellus Histamine H1 receptor pKb nan None 10.1016/j.bmc.2008.10.042
Cavia porcellus Leukotriene C4 synthase IC50 nan None None
Cavia porcellus Leukotriene C4 synthase Ki nan None None
Cavia porcellus Serotonin 4 (5-HT4) receptor IC50 nan None None
Cavia porcellus Serotonin 4 (5-HT4) receptor Ki nan None None
Chlamydia trachomatis Chlamydia trachomatis MIC 0.004 ug.mL-1 10.1128/aac.00477-09
Chlamydia trachomatis Chlamydia trachomatis MIC 0.25 ug.mL-1 10.1128/aac.00477-09
Chlamydia trachomatis Chlamydia trachomatis MIC 8.0 ug.mL-1 10.1128/aac.00477-09
Chlamydia trachomatis Chlamydia trachomatis MIC 32.0 ug.mL-1 10.1128/aac.00477-09
Chlamydia trachomatis Chlamydia trachomatis MIC 128.0 ug.mL-1 10.1128/aac.00477-09
Chlorocebus sabaeus Vero Activity nan None 10.1021/np020592u
Chlorocebus sabaeus Vero Activity nan None 10.1021/np0400095
Chlorocebus sabaeus Vero CC50 7.8 ug.mL-1 10.1016/j.ejmech.2018.01.080
Chlorocebus sabaeus Vero CC50 32.0 ug.mL-1 10.1016/j.bmcl.2019.06.055
Chlorocebus sabaeus Vero CC50 50.0 ug.mL-1 10.1021/jm300123s
Chlorocebus sabaeus Vero CC50 128.0 ug.mL-1 10.1016/j.bmcl.2019.07.041
Chlorocebus sabaeus Vero CC50 128.0 ug.mL-1 10.1016/j.ejmech.2019.07.057
Chlorocebus sabaeus Vero CC50 150.0 ug.mL-1 10.1016/j.ejmech.2015.10.024
Chlorocebus sabaeus Vero CC50 500.0 ug.mL-1 10.1016/j.bmc.2012.09.019
Chlorocebus sabaeus Vero CC50 500.0 ug.mL-1 10.1016/j.bmcl.2017.07.023
Chlorocebus sabaeus Vero CC50 500.0 ug.mL-1 10.1016/j.ejmech.2017.05.057
Chlorocebus sabaeus Vero CC50 512.0 ug.mL-1 10.1016/j.ejmech.2017.11.090
Chlorocebus sabaeus Vero CC50 512.0 ug.mL-1 10.1016/j.ejmech.2018.07.025
Chlorocebus sabaeus Vero CC50 512.0 ug.mL-1 10.1016/j.ejmech.2019.01.042
Chlorocebus sabaeus Vero CC50 75900.0 nM 10.1007/s00044-011-9638-9
Chlorocebus sabaeus Vero CC50 75940.0 nM 10.1016/j.bmcl.2010.06.096
Chlorocebus sabaeus Vero CC50 180000.0 nM 10.1016/j.ejmech.2010.11.023
Chlorocebus sabaeus Vero CC50 512000.0 nM 10.1016/j.bmc.2019.04.017
Chlorocebus sabaeus Vero CC50 512000.0 nM 10.1016/j.ejmech.2018.09.049
Chlorocebus sabaeus Vero CC50 nan None 10.1016/j.bmc.2019.01.022
Chlorocebus sabaeus Vero CC50 nan None 10.1016/j.bmc.2022.116777
Chlorocebus sabaeus Vero CC50 nan None 10.1016/j.ejmech.2017.05.044
Chlorocebus sabaeus Vero CC50 nan None 10.1016/j.ejmech.2019.111595
Chlorocebus sabaeus Vero CC50 nan None 10.1016/j.ejmech.2021.113398
Chlorocebus sabaeus Vero CD50 500.0 ug ml-1 10.1016/j.bmc.2013.07.003
Chlorocebus sabaeus Vero GI 44.78 % 10.1016/j.bmcl.2016.06.089
Chlorocebus sabaeus Vero IC50 10.0 ug.mL-1 10.1007/s00044-012-0074-2
Chlorocebus sabaeus Vero IC50 58.0 ug.mL-1 10.1016/j.bmc.2013.06.027
Chlorocebus sabaeus Vero IC50 62.5 ug.mL-1 10.1016/j.bmcl.2009.12.045
Chlorocebus sabaeus Vero IC50 62.5 ug.mL-1 10.1016/j.bmcl.2012.12.069
Chlorocebus sabaeus Vero IC50 62.5 ug.mL-1 10.1016/j.ejmech.2014.03.085
Chlorocebus sabaeus Vero IC50 62.5 ug.mL-1 10.1021/jm060339h
Chlorocebus sabaeus Vero IC50 64.0 ug.mL-1 10.1016/j.bmc.2022.117006
Chlorocebus sabaeus Vero IC50 64.0 ug.mL-1 10.1016/j.ejmech.2021.113603
Chlorocebus sabaeus Vero IC50 89.3 ug.mL-1 10.1016/j.bmcl.2008.09.029
Chlorocebus sabaeus Vero IC50 97.4 ug.mL-1 10.1021/acs.jnatprod.8b00567
Chlorocebus sabaeus Vero IC50 100.0 ug.mL-1 10.1016/j.bmc.2007.05.063
Chlorocebus sabaeus Vero IC50 100.0 ug.mL-1 10.1016/j.bmc.2008.10.086
Chlorocebus sabaeus Vero IC50 100.0 ug.mL-1 10.1016/j.bmc.2010.02.024
Chlorocebus sabaeus Vero IC50 100.0 ug.mL-1 10.1016/j.bmcl.2005.06.010
Chlorocebus sabaeus Vero IC50 100.0 ug.mL-1 10.1016/j.ejmech.2009.10.050
Chlorocebus sabaeus Vero IC50 100.0 ug.mL-1 10.1021/acsmedchemlett.8b00410
Chlorocebus sabaeus Vero IC50 100.0 ug.mL-1 10.1021/np400497f
Chlorocebus sabaeus Vero IC50 110.67 ug.mL-1 10.1021/jm020891g
Chlorocebus sabaeus Vero IC50 137.6 ug.mL-1 10.1016/j.ejmech.2020.112045
Chlorocebus sabaeus Vero IC50 142.9 ug.mL-1 10.1021/np400145u
Chlorocebus sabaeus Vero IC50 147.0 ug.mL-1 10.1016/s0960-894x(00)00058-5
Chlorocebus sabaeus Vero IC50 158.0 ug.mL-1 10.1021/np980066w
Chlorocebus sabaeus Vero IC50 200.0 ug.mL-1 10.1016/j.bmc.2018.07.034
Chlorocebus sabaeus Vero IC50 256.0 ug.mL-1 10.1021/acs.jmedchem.7b00582
Chlorocebus sabaeus Vero IC50 1000.0 ug.mL-1 10.1016/s0960-894x(01)00266-9
Chlorocebus sabaeus Vero IC50 50000.0 nM 10.1016/j.bmc.2016.12.038
Chlorocebus sabaeus Vero IC50 74500.0 nM 10.1016/j.ejmech.2010.05.035
Chlorocebus sabaeus Vero IC50 75900.0 nM 10.1016/j.bmcl.2008.12.088
Chlorocebus sabaeus Vero IC50 75940.0 nM 10.1016/j.bmcl.2007.01.037
Chlorocebus sabaeus Vero IC50 75940.0 nM 10.1016/j.ejmech.2009.09.033
Chlorocebus sabaeus Vero IC50 77400.0 nM 10.1007/s00044-010-9322-5
Chlorocebus sabaeus Vero IC50 97900.0 nM 10.1021/np800751j
Chlorocebus sabaeus Vero IC50 100000.0 nM 10.1016/j.bmc.2007.05.053
Chlorocebus sabaeus Vero IC50 100000.0 nM 10.1016/j.bmcl.2012.06.095
Chlorocebus sabaeus Vero IC50 100000.0 nM 10.1016/j.bmcl.2015.12.080
Chlorocebus sabaeus Vero IC50 100000.0 nM 10.1016/j.bmcl.2016.06.089
Chlorocebus sabaeus Vero IC50 100000.0 nM 10.1016/j.ejmech.2013.01.017
Chlorocebus sabaeus Vero IC50 100000.0 nM 10.1021/acsmedchemlett.7b00356
Chlorocebus sabaeus Vero IC50 105000.0 nM 10.1007/s00044-007-9073-0
Chlorocebus sabaeus Vero IC50 108000.0 nM 10.1016/j.bmcl.2013.09.013
Chlorocebus sabaeus Vero IC50 113000.0 nM 10.1016/j.bmc.2012.02.025
Chlorocebus sabaeus Vero IC50 113000.0 nM 10.1016/j.bmcl.2014.05.062
Chlorocebus sabaeus Vero IC50 113000.0 nM 10.1021/ml200036r
Chlorocebus sabaeus Vero IC50 122000.0 nM 10.1016/j.bmcl.2009.11.105
Chlorocebus sabaeus Vero IC50 122000.0 nM 10.1021/acs.jnatprod.9b01095
Chlorocebus sabaeus Vero IC50 122000.0 nM 10.1021/jm900340a
Chlorocebus sabaeus Vero IC50 122000.0 nM 10.1021/jm901235p
Chlorocebus sabaeus Vero IC50 125000.0 nM 10.1016/j.ejmech.2009.12.074
Chlorocebus sabaeus Vero IC50 127000.0 nM 10.1021/jm900003c
Chlorocebus sabaeus Vero IC50 127000.0 nM 10.1021/jm900513a
Chlorocebus sabaeus Vero IC50 132500.0 nM 10.1021/np400391p
Chlorocebus sabaeus Vero IC50 134480.0 nM 10.1021/jm020891g
Chlorocebus sabaeus Vero IC50 138300.0 nM 10.1016/j.bmc.2008.12.006
Chlorocebus sabaeus Vero IC50 182000.0 nM 10.1016/j.bmcl.2013.11.024
Chlorocebus sabaeus Vero IC50 nan None 10.1016/j.bmcl.2012.05.096
Chlorocebus sabaeus Vero IC50 nan None 10.1021/acs.jmedchem.5b01542
Chlorocebus sabaeus Vero IC50 nan None 10.1021/acsmedchemlett.5b00176
Chlorocebus sabaeus Vero IC50 nan None 10.1021/np0601399
Chlorocebus sabaeus Vero Maximal non-toxic dose 50 64.0 ug ml-1 10.1021/jm0602662
Chlorocebus sabaeus Vero MIC 127000.0 nM 10.1021/jm901112f
Chlorocebus sabaeus Vero MIC 127000.0 nM 10.1021/jm901273n
Chlorocebus sabaeus Vero MNTD 64.0 ug ml-1 10.1016/j.ejmech.2009.06.005
Chlorocebus sabaeus Vero MNTD50 64.0 ug ml-1 10.1021/jm701560p
Chlorocebus sabaeus Vero MTD50 64.0 ug ml-1 10.1016/s0960-894x(99)00510-7
Chlorocebus sabaeus Vero PI 213.0 None 10.1021/jm0602662
Chlorocebus sabaeus Vero Ratio IC50 1080.0 None 10.1016/j.bmc.2010.03.018
Chlorocebus sabaeus Vero Selectivity 400.0 None 10.1016/j.bmcl.2005.06.010
Citrobacter freundii Citrobacter freundii MIC 0.023 ug.mL-1 10.1128/aac.00405-08
Citrobacter freundii Citrobacter freundii Ratio 500.0 None 10.1128/aac.00405-08
Clostridioides difficile Clostridioides difficile MBC 0.78 ug ml-1 10.1016/j.bmc.2018.07.034
Clostridioides difficile Clostridioides difficile MIC 6e-05 ug.mL-1 10.1128/aac.00342-08
Clostridioides difficile Clostridioides difficile MIC 9e-05 ug.mL-1 10.1128/aac.00342-08
Clostridioides difficile Clostridioides difficile MIC 0.0004 ug.mL-1 10.1128/aac.00342-08
Clostridioides difficile Clostridioides difficile MIC 0.0009 ug.mL-1 10.1128/aac.00342-08
Clostridioides difficile Clostridioides difficile MIC 0.001 ug.mL-1 10.1021/acs.jmedchem.1c02045
Clostridioides difficile Clostridioides difficile MIC 0.0019 ug.mL-1 10.1128/aac.00342-08
Clostridioides difficile Clostridioides difficile MIC 0.002 ug.mL-1 10.1128/aac.00342-08
Clostridioides difficile Clostridioides difficile MIC 0.003 ug.mL-1 10.1128/aac.00342-08
Clostridioides difficile Clostridioides difficile MIC 0.004 ug.mL-1 10.1128/aac.00342-08
Clostridioides difficile Clostridioides difficile MIC 0.008 ug.mL-1 10.1128/aac.00476-08
Clostridioides difficile Clostridioides difficile MIC 0.015 ug.mL-1 10.1021/acsmedchemlett.0c00381
Clostridioides difficile Clostridioides difficile MIC 0.016 ug.mL-1 10.1128/aac.00342-08
Clostridioides difficile Clostridioides difficile MIC 0.03 ug.mL-1 10.1021/acs.jmedchem.1c02045
Clostridioides difficile Clostridioides difficile MIC 0.06 ug.mL-1 10.1021/acs.jmedchem.1c02045
Clostridioides difficile Clostridioides difficile MIC 0.25 ug.mL-1 10.1021/acs.jmedchem.1c02045
Clostridioides difficile Clostridioides difficile MIC 2.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Clostridioides difficile Clostridioides difficile MIC 8.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Clostridioides difficile Clostridioides difficile MIC 16.0 ug.mL-1 10.1021/acsmedchemlett.0c00381
Clostridioides difficile Clostridioides difficile MIC 32.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Clostridioides difficile Clostridioides difficile MIC 32.0 ug.mL-1 10.1128/aac.00342-08
Clostridioides difficile Clostridioides difficile MIC 128.0 ug.mL-1 10.1128/aac.00342-08
Clostridioides difficile Clostridioides difficile MIC 256.0 ug.mL-1 10.1128/aac.00342-08
Clostridioides difficile Clostridioides difficile MIC50 0.015 ug.mL-1 10.1128/aac.00476-08
Clostridioides difficile Clostridioides difficile MIC90 0.015 ug.mL-1 10.1128/aac.00476-08
Clostridioides difficile Clostridioides difficile MIC90 128.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Clostridium perfringens Clostridium perfringens log(1/C) 8.44 None 10.1021/jm00210a025
Clostridium perfringens Clostridium perfringens MIC 0.003 ug.mL-1 10.1021/jm00210a025
Clostridium sporogenes Clostridium sporogenes MIC 1.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Cricetulus griseus CHO CC50 512000.0 nM 10.1016/j.ejmech.2019.111678
Cricetulus griseus CHO IC50 nan None 10.1021/acs.jmedchem.1c00707
Cryptococcus neoformans Cryptococcus neoformans IC50 nan None 10.1021/jm900672t
Cryptococcus neoformans Cryptococcus neoformans IC50 nan None 10.1021/np000436s
Cryptococcus neoformans Cryptococcus neoformans MIC nan None 10.1021/np000436s
Dialister invisus Dialister invisus Activity 2.0 ug ml-1 10.1128/aac.00538-07
Dialister invisus Dialister invisus Activity nan None 10.1128/aac.00538-07
Dialister invisus Dialister invisus MIC 0.06 ug.mL-1 10.1128/aac.00538-07
Dialister micraerophilus Dialister micraerophilus Activity 2.0 ug ml-1 10.1128/aac.00538-07
Dialister micraerophilus Dialister micraerophilus Activity nan None 10.1128/aac.00538-07
Dialister micraerophilus Dialister micraerophilus MIC 0.06 ug.mL-1 10.1128/aac.00538-07
Dialister micraerophilus Dialister micraerophilus MIC50 0.06 ug.mL-1 10.1128/aac.00538-07
Dialister micraerophilus Dialister micraerophilus MIC90 0.06 ug.mL-1 10.1128/aac.00538-07
Dialister pneumosintes Dialister pneumosintes Activity 2.0 ug ml-1 10.1128/aac.00538-07
Dialister pneumosintes Dialister pneumosintes Activity nan None 10.1128/aac.00538-07
Dialister pneumosintes Dialister pneumosintes MIC 0.06 ug.mL-1 10.1128/aac.00538-07
Dialister pneumosintes Dialister pneumosintes MIC50 2.0 ug.mL-1 10.1128/aac.00538-07
Dialister pneumosintes Dialister pneumosintes MIC90 4.0 ug.mL-1 10.1128/aac.00538-07
Dialister propionicifaciens Dialister propionicifaciens Activity 2.0 ug ml-1 10.1128/aac.00538-07
Dialister propionicifaciens Dialister propionicifaciens Activity nan None 10.1128/aac.00538-07
Dialister propionicifaciens Dialister propionicifaciens MIC 0.06 ug.mL-1 10.1128/aac.00538-07
Electrophorus electricus Acetylcholinesterase Inhibition 16.23 % 10.1016/j.bmc.2012.09.040
Enterobacter cloacae Enterobacter cloacae EC50 6200.0 nM 10.1016/j.bmcl.2016.04.089
Enterobacter cloacae Enterobacter cloacae EC50 8800.0 nM 10.1021/acs.jmedchem.8b01293
Enterobacter cloacae Enterobacter cloacae FICI 0.126 None 10.1128/aac.01439-09
Enterobacter cloacae Enterobacter cloacae IZ 0.0 mm 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae IZ 8.0 mm 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae IZ 10.0 mm 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae IZ 13.0 mm 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae IZ 26.0 mm 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae IZ 28.0 mm 10.1128/aac.00072-07
Enterobacter cloacae Enterobacter cloacae MBC nan None 10.1021/acs.jnatprod.2c00065
Enterobacter cloacae Enterobacter cloacae MIC 0.008 ug.mL-1 10.1128/aac.00405-08
Enterobacter cloacae Enterobacter cloacae MIC 0.016 ug.mL-1 10.1128/aac.00405-08
Enterobacter cloacae Enterobacter cloacae MIC 0.016 ug.mL-1 10.1128/aac.01439-09
Enterobacter cloacae Enterobacter cloacae MIC 0.032 ug.mL-1 10.1128/aac.00405-08
Enterobacter cloacae Enterobacter cloacae MIC 0.125 ug.mL-1 10.1128/aac.00405-08
Enterobacter cloacae Enterobacter cloacae MIC 0.26 ug.mL-1 10.1128/aac.00405-08
Enterobacter cloacae Enterobacter cloacae MIC 1.5 ug.mL-1 10.1128/aac.01439-09
Enterobacter cloacae Enterobacter cloacae MIC 6.0 ug.mL-1 10.1128/aac.01439-09
Enterobacter cloacae Enterobacter cloacae MIC 8.0 ug.mL-1 10.1128/aac.00405-08
Enterobacter cloacae Enterobacter cloacae MIC 12.0 ug.mL-1 10.1128/aac.00405-08
Enterobacter cloacae Enterobacter cloacae MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.6b01742
Enterobacter cloacae Enterobacter cloacae MIC 16.0 ug.mL-1 10.1021/acs.jnatprod.2c00065
Enterobacter cloacae Enterobacter cloacae Ratio 260.0 None 10.1128/aac.01439-09
Enterobacter cloacae Enterobacter cloacae Ratio 500.0 None 10.1128/aac.00405-08
Enterobacter cloacae Enterobacter cloacae Ratio 750.0 None 10.1128/aac.00405-08
Enterobacter cloacae Enterobacter cloacae Ratio 1400.0 None 10.1128/aac.00405-08
Enterococcus avium Enterococcus avium MIC 1.0 ug.mL-1 10.1128/aac.00908-07
Enterococcus faecalis Enterococcus faecalis IC50 10000.0 nM 10.1021/acs.jnatprod.2c00444
Enterococcus faecalis Enterococcus faecalis IZ 20.0 mm 10.1016/j.bmc.2007.09.025
Enterococcus faecalis Enterococcus faecalis IZ 21.0 mm 10.1016/j.bmc.2019.115097
Enterococcus faecalis Enterococcus faecalis MBC 1.56 ug ml-1 10.1016/j.bmc.2018.07.034
Enterococcus faecalis Enterococcus faecalis MBC 25.0 ug ml-1 10.1016/j.bmc.2018.07.034
Enterococcus faecalis Enterococcus faecalis MIC 0.008 ug.mL-1 10.1021/np050176k
Enterococcus faecalis Enterococcus faecalis MIC 0.03 ug.mL-1 10.1021/acs.jnatprod.9b00062
Enterococcus faecalis Enterococcus faecalis MIC 0.125 ug.mL-1 10.1016/j.ejmech.2022.114360
Enterococcus faecalis Enterococcus faecalis MIC 0.19 ug.mL-1 10.1128/aac.01710-09
Enterococcus faecalis Enterococcus faecalis MIC 0.25 ug.mL-1 10.1128/aac.01710-09
Enterococcus faecalis Enterococcus faecalis MIC 0.5 ug.mL-1 10.1016/j.bmcl.2020.127146
Enterococcus faecalis Enterococcus faecalis MIC 0.5 ug.mL-1 10.1021/jm501082n
Enterococcus faecalis Enterococcus faecalis MIC 0.5 ug.mL-1 10.1128/aac.00576-06
Enterococcus faecalis Enterococcus faecalis MIC 1.0 ug.mL-1 10.1016/j.bmcl.2016.05.077
Enterococcus faecalis Enterococcus faecalis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2014.07.066
Enterococcus faecalis Enterococcus faecalis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Enterococcus faecalis Enterococcus faecalis MIC 1.0 ug.mL-1 10.1021/jm00167a029
Enterococcus faecalis Enterococcus faecalis MIC 1.0 ug.mL-1 10.1021/ml300350p
Enterococcus faecalis Enterococcus faecalis MIC 1.0 ug.mL-1 10.1128/aac.00576-06
Enterococcus faecalis Enterococcus faecalis MIC 1.0 ug.mL-1 10.1128/aac.00908-07
Enterococcus faecalis Enterococcus faecalis MIC 2.0 ug.mL-1 10.1016/j.bmcl.2016.05.077
Enterococcus faecalis Enterococcus faecalis MIC 2.0 ug.mL-1 10.1128/aac.00576-06
Enterococcus faecalis Enterococcus faecalis MIC 2.0 ug.mL-1 10.1128/aac.00908-07
Enterococcus faecalis Enterococcus faecalis MIC 3.0 ug.mL-1 10.1128/aac.01710-09
Enterococcus faecalis Enterococcus faecalis MIC 4.0 ug.mL-1 10.1016/j.bmcl.2016.05.077
Enterococcus faecalis Enterococcus faecalis MIC 4.0 ug.mL-1 10.1021/acs.jmedchem.0c00520
Enterococcus faecalis Enterococcus faecalis MIC 4.0 ug.mL-1 10.1128/aac.01710-09
Enterococcus faecalis Enterococcus faecalis MIC 8.0 ug.mL-1 10.1016/j.ejmech.2019.02.009
Enterococcus faecalis Enterococcus faecalis MIC 8.0 ug.mL-1 10.1128/aac.01710-09
Enterococcus faecalis Enterococcus faecalis MIC 16.0 ug.mL-1 10.1128/aac.01710-09
Enterococcus faecalis Enterococcus faecalis MIC 32.0 ug.mL-1 10.1128/aac.01710-09
Enterococcus faecalis Enterococcus faecalis MIC 1000.0 nM 10.1021/acs.jmedchem.1c00614
Enterococcus faecalis Enterococcus faecalis MIC 1000.0 nM 10.1021/acs.jmedchem.1c02122
Enterococcus faecalis Enterococcus faecalis MIC 1000.0 nM 10.1021/acs.jmedchem.1c02140
Enterococcus faecalis Enterococcus faecalis MIC nan None 10.1016/j.bmc.2019.04.032
Enterococcus faecalis Enterococcus faecalis MIC nan None 10.1016/j.bmcl.2012.08.003
Enterococcus faecalis Enterococcus faecalis MIC nan None 10.1021/np050424c
Enterococcus faecalis Enterococcus faecalis MIC100 0.78 ug ml-1 10.1016/j.bmc.2018.07.034
Enterococcus faecalis Enterococcus faecalis MIC100 25.0 ug ml-1 10.1016/j.bmc.2018.07.034
Enterococcus faecalis Enterococcus faecalis MIC>90 0.2 ug ml-1 10.1021/np400145u
Enterococcus faecium Enterococcus faecium EC50 130.0 nM 10.1021/acs.jmedchem.8b01293
Enterococcus faecium Enterococcus faecium EC50 1200.0 nM 10.1016/j.bmcl.2016.04.089
Enterococcus faecium Enterococcus faecium IC50 8.75 ug.mL-1 10.1021/np2006555
Enterococcus faecium Enterococcus faecium IZ 9.0 mm 10.1016/j.bmc.2019.115097
Enterococcus faecium Enterococcus faecium IZ nan None 10.1021/np900382x
Enterococcus faecium Enterococcus faecium MBC nan None 10.1021/acs.jnatprod.2c00065
Enterococcus faecium Enterococcus faecium MIC 0.04 ug.mL-1 10.1021/np050176k
Enterococcus faecium Enterococcus faecium MIC 0.125 ug.mL-1 10.1016/j.ejmech.2022.114360
Enterococcus faecium Enterococcus faecium MIC 0.25 ug.mL-1 10.1016/j.ejmech.2019.04.034
Enterococcus faecium Enterococcus faecium MIC 2.0 ug.mL-1 10.1016/j.ejmech.2019.05.090
Enterococcus faecium Enterococcus faecium MIC 3.1 ug.mL-1 10.1021/acs.jnatprod.0c01212
Enterococcus faecium Enterococcus faecium MIC 4.0 ug.mL-1 10.1128/aac.00576-06
Enterococcus faecium Enterococcus faecium MIC 8.0 ug.mL-1 10.1016/j.ejmech.2022.114360
Enterococcus faecium Enterococcus faecium MIC 8.0 ug.mL-1 10.1021/acs.jnatprod.2c00065
Enterococcus faecium Enterococcus faecium MIC 32.0 ug.mL-1 10.1128/aac.01710-09
Enterococcus faecium Enterococcus faecium MIC 21000.0 nM 10.1021/acs.jmedchem.1c02122
Equus caballus Cholinesterase Inhibition 1.88 % 10.1016/j.bmc.2012.09.040
Escherichia coli DNA repair protein RecN Activity nan None 10.1021/acs.jmedchem.0c00328
Escherichia coli Escherichia coli AC50 32271.0 nM None
Escherichia coli Escherichia coli Activity 0.0 % 10.1128/aac.00375-07
Escherichia coli Escherichia coli Activity 1.17 % 10.1021/np010076o
Escherichia coli Escherichia coli Activity 27.82 % 10.1021/np010076o
Escherichia coli Escherichia coli Activity 32.6 % 10.1128/aac.00375-07
Escherichia coli Escherichia coli Activity 32.8 % 10.1128/aac.00375-07
Escherichia coli Escherichia coli Activity 35.8 % 10.1128/aac.00375-07
Escherichia coli Escherichia coli Activity 64.0 mg/L 10.1021/jm501082n
Escherichia coli Escherichia coli Activity 80.2 % 10.1128/aac.00375-07
Escherichia coli Escherichia coli Activity 85.1 % 10.1128/aac.00375-07
Escherichia coli Escherichia coli Activity 89.56 % 10.1021/np010076o
Escherichia coli Escherichia coli Activity nan None 10.1016/j.bmcl.2013.02.005
Escherichia coli Escherichia coli Activity nan None 10.1016/j.ejmech.2019.111636
Escherichia coli Escherichia coli Activity nan None 10.1021/acs.jmedchem.2c01076
Escherichia coli Escherichia coli Activity nan None 10.1021/jm400485e
Escherichia coli Escherichia coli Activity nan None 10.1128/aac.00043-09
Escherichia coli Escherichia coli Activity nan None 10.1128/aac.00375-07
Escherichia coli Escherichia coli Antibiotic resistance nan None 10.1016/s0960-894x(98)00536-8
Escherichia coli Escherichia coli FC 16.0 None 10.1021/acs.jmedchem.2c01076
Escherichia coli Escherichia coli FICI 0.071 None 10.1128/aac.00405-08
Escherichia coli Escherichia coli FICI 0.111 None 10.1128/aac.01439-09
Escherichia coli Escherichia coli FICI 0.126 None 10.1128/aac.01439-09
Escherichia coli Escherichia coli FICI 0.128 None 10.1128/aac.00405-08
Escherichia coli Escherichia coli GI 98.0 % 10.1016/j.bmc.2016.01.040
Escherichia coli Escherichia coli IC90 0.5 ug.mL-1 10.1021/np400002p
Escherichia coli Escherichia coli Inhibition 10.0 % 10.1128/aac.00471-08
Escherichia coli Escherichia coli Inhibition 100.0 % 10.1021/jm0703901
Escherichia coli Escherichia coli Inhibition nan % 10.1016/j.bmc.2018.07.034
Escherichia coli Escherichia coli Inhibition nan % 10.1128/aac.00471-08
Escherichia coli Escherichia coli Inhibition nan % 10.1128/aac.00691-09
Escherichia coli Escherichia coli IZ 6.0 mm 10.1021/np900382x
Escherichia coli Escherichia coli IZ 11.0 mm 10.1016/j.bmc.2018.02.049
Escherichia coli Escherichia coli IZ 14.0 mm 10.1016/j.bmc.2007.09.025
Escherichia coli Escherichia coli IZ 20.0 mm 10.1021/np900382x
Escherichia coli Escherichia coli IZ 27.0 mm 10.1016/j.bmcl.2016.04.038
Escherichia coli Escherichia coli IZ 48.0 mm 10.1016/j.ejmech.2008.09.035
Escherichia coli Escherichia coli log10cfu 8.58 None 10.1128/aac.00471-08
Escherichia coli Escherichia coli MBC 3.0 ug ml-1 10.1128/aac.00375-07
Escherichia coli Escherichia coli MBC 8.0 ug ml-1 10.1016/j.bmcl.2023.129320
Escherichia coli Escherichia coli MBC 8.0 ug ml-1 10.1021/acs.jnatprod.5b00770
Escherichia coli Escherichia coli MBC 25.0 ug ml-1 10.1016/j.bmc.2018.07.034
Escherichia coli Escherichia coli MIC 0.006 ug.mL-1 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC 0.008 ug.mL-1 10.1128/aac.00471-08
Escherichia coli Escherichia coli MIC 0.01333 ug.mL-1 10.1016/j.ejmech.2022.114108
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC 0.016 ug.mL-1 10.1128/aac.01439-09
Escherichia coli Escherichia coli MIC 0.02 ug.mL-1 10.1021/np050176k
Escherichia coli Escherichia coli MIC 0.023 ug.mL-1 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC 0.031 ug.mL-1 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC 0.031 ug.mL-1 10.1128/aac.01439-09
Escherichia coli Escherichia coli MIC 0.047 ug.mL-1 10.1128/aac.01439-09
Escherichia coli Escherichia coli MIC 0.055 ug.mL-1 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1021/acs.jnatprod.1c00578
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1021/acs.jnatprod.2c00621
Escherichia coli Escherichia coli MIC 0.06 ug.mL-1 10.1021/jm501082n
Escherichia coli Escherichia coli MIC 0.063 ug.mL-1 10.1128/aac.01439-09
Escherichia coli Escherichia coli MIC 0.064 ug.mL-1 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1016/j.ejmech.2018.08.070
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1021/jm301499r
Escherichia coli Escherichia coli MIC 0.125 ug.mL-1 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC 0.19 ug.mL-1 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC 0.19 ug.mL-1 10.1128/aac.01439-09
Escherichia coli Escherichia coli MIC 0.24 ug.mL-1 10.1016/j.bmcl.2006.10.016
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1016/j.ejmech.2008.09.035
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC 0.25 ug.mL-1 10.1128/aac.01439-09
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1016/j.bmc.2018.02.049
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1021/jm501082n
Escherichia coli Escherichia coli MIC 0.5 ug.mL-1 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC 0.64 ug.mL-1 10.1128/aac.01439-09
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1016/j.ejmech.2014.07.066
Escherichia coli Escherichia coli MIC 1.0 ug.mL-1 10.1128/aac.01439-09
Escherichia coli Escherichia coli MIC 1.024 ug.mL-1 10.1016/j.ejmech.2022.114108
Escherichia coli Escherichia coli MIC 1.9 ug.mL-1 10.1016/j.ejmech.2007.12.019
Escherichia coli Escherichia coli MIC 1.9 ug.mL-1 10.1128/aac.00580-10
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1016/j.bmcl.2016.05.077
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1016/j.ejmech.2016.03.061
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1016/j.ejmech.2022.114360
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1021/jm020183v
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00375-07
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.00748-09
Escherichia coli Escherichia coli MIC 2.0 ug.mL-1 10.1128/aac.01783-09
Escherichia coli Escherichia coli MIC 2.1 ug.mL-1 10.1128/aac.00580-10
Escherichia coli Escherichia coli MIC 2.5 ug.mL-1 10.1021/acs.jmedchem.7b00204
Escherichia coli Escherichia coli MIC 3.0 ug.mL-1 10.1128/aac.00375-07
Escherichia coli Escherichia coli MIC 3.9 ug.mL-1 10.1016/j.ejmech.2007.12.019
Escherichia coli Escherichia coli MIC 3.9 ug.mL-1 10.1128/aac.00580-10
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1016/j.bmcl.2023.129320
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1016/j.ejmech.2018.08.070
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1021/acs.jnatprod.0c01309
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00310-09
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.00375-07
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01439-09
Escherichia coli Escherichia coli MIC 4.0 ug.mL-1 10.1128/aac.01783-09
Escherichia coli Escherichia coli MIC 5.0 ug.mL-1 10.1016/j.ejmech.2013.04.060
Escherichia coli Escherichia coli MIC 6.0 ug.mL-1 10.1021/jm00143a010
Escherichia coli Escherichia coli MIC 6.0 ug.mL-1 10.1021/jm00145a020
Escherichia coli Escherichia coli MIC 6.0 ug.mL-1 10.1021/jm00220a012
Escherichia coli Escherichia coli MIC 6.0 ug.mL-1 10.1128/aac.00375-07
Escherichia coli Escherichia coli MIC 6.25 ug.mL-1 10.1128/aac.00475-08
Escherichia coli Escherichia coli MIC 6.3 ug.mL-1 10.1021/acs.jnatprod.0c01212
Escherichia coli Escherichia coli MIC 7.0 ug.mL-1 10.1016/j.ejmech.2013.04.060
Escherichia coli Escherichia coli MIC 7.0 ug.mL-1 10.1021/jm400485e
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1016/j.bmcl.2006.10.016
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1016/j.bmcl.2020.127146
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1016/j.ejmech.2008.04.001
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1016/j.ejmech.2019.02.009
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1016/j.ejmech.2022.114360
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1021/acs.jnatprod.1c00578
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1021/acs.jnatprod.2c00621
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1021/acs.jnatprod.5b00770
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1021/jm00167a029
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1021/jm301499r
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1021/jm501082n
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1021/ml300350p
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1039/d2md00041e
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00017-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.00638-08
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.01052-07
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.01439-09
Escherichia coli Escherichia coli MIC 8.0 ug.mL-1 10.1128/aac.01783-09
Escherichia coli Escherichia coli MIC 10.0 ug.mL-1 10.1021/jm400485e
Escherichia coli Escherichia coli MIC 12.0 ug.mL-1 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1016/j.ejmech.2020.113049
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00043-09
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.00638-08
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.01052-07
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.01053-06
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.01128-06
Escherichia coli Escherichia coli MIC 16.0 ug.mL-1 10.1128/aac.01783-09
Escherichia coli Escherichia coli MIC 20.0 ug.mL-1 10.1021/jm970791o
Escherichia coli Escherichia coli MIC 22.0 ug.mL-1 10.1016/j.bmcl.2017.05.032
Escherichia coli Escherichia coli MIC 24.0 ug.mL-1 10.1128/aac.01128-06
Escherichia coli Escherichia coli MIC 31.0 ug.mL-1 10.1021/jm501082n
Escherichia coli Escherichia coli MIC 50.0 ug.mL-1 10.1016/j.bmcl.2009.09.095
Escherichia coli Escherichia coli MIC 50.0 ug.mL-1 10.1016/j.bmcl.2010.12.084
Escherichia coli Escherichia coli MIC 62.5 ug.mL-1 10.1016/j.bmc.2006.12.035
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/j.bmcl.2015.01.026
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/j.ejmech.2008.04.001
Escherichia coli Escherichia coli MIC 64.0 ug.mL-1 10.1016/j.ejmech.2022.114360
Escherichia coli Escherichia coli MIC 100.0 ug.mL-1 10.1021/jm0703901
Escherichia coli Escherichia coli MIC 250.0 ug.mL-1 10.1016/j.bmcl.2006.10.016
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1016/j.bmc.2006.12.035
Escherichia coli Escherichia coli MIC 512.0 ug.mL-1 10.1128/aac.00310-09
Escherichia coli Escherichia coli MIC 2000.0 nM 10.1016/j.ejmech.2019.111636
Escherichia coli Escherichia coli MIC 4000.0 nM 10.1016/j.ejmech.2019.111636
Escherichia coli Escherichia coli MIC 4000.0 nM 10.1021/acs.jmedchem.1c00614
Escherichia coli Escherichia coli MIC 4000.0 nM 10.1021/acs.jmedchem.1c02122
Escherichia coli Escherichia coli MIC 4000.0 nM 10.1021/acs.jmedchem.1c02140
Escherichia coli Escherichia coli MIC 4000.0 nM 10.1021/acs.jmedchem.2c01076
Escherichia coli Escherichia coli MIC 4000.0 nM 10.1021/acs.jmedchem.9b00288
Escherichia coli Escherichia coli MIC 8000.0 nM 10.1021/acs.jmedchem.9b00288
Escherichia coli Escherichia coli MIC 10000.0 nM 10.1021/acs.jnatprod.5b01129
Escherichia coli Escherichia coli MIC 16000.0 nM 10.1016/j.bmc.2016.04.058
Escherichia coli Escherichia coli MIC 55000.0 nM 10.1016/j.bmc.2016.04.058
Escherichia coli Escherichia coli MIC 25922000.0 nM 10.1021/acs.jmedchem.1c02140
Escherichia coli Escherichia coli MIC nan None 10.1016/j.bmc.2010.05.016
Escherichia coli Escherichia coli MIC nan None 10.1016/j.bmc.2013.10.011
Escherichia coli Escherichia coli MIC nan None 10.1016/j.bmc.2019.04.032
Escherichia coli Escherichia coli MIC nan None 10.1016/j.bmcl.2012.08.003
Escherichia coli Escherichia coli MIC nan None 10.1016/j.bmcl.2013.11.024
Escherichia coli Escherichia coli MIC nan None 10.1016/j.ejmech.2019.04.067
Escherichia coli Escherichia coli MIC nan None 10.1021/np050424c
Escherichia coli Escherichia coli MIC nan None 10.1021/np200320u
Escherichia coli Escherichia coli MIC nan None 10.1128/aac.00405-08
Escherichia coli Escherichia coli MIC100 3.13 ug ml-1 10.1016/j.bmc.2018.07.034
Escherichia coli Escherichia coli MIC90 100.0 nM 10.1016/j.bmcl.2011.08.054
Escherichia coli Escherichia coli MIC90 128.0 ug.mL-1 10.1016/j.bmcl.2009.11.042
Escherichia coli Escherichia coli MIC90 12500.0 nM 10.1016/j.bmcl.2011.08.054
Escherichia coli Escherichia coli MIC99 nan None 10.1016/j.ejmech.2013.10.055
Escherichia coli Escherichia coli Ratio 1.0 None 10.1128/aac.00748-09
Escherichia coli Escherichia coli Ratio 8.0 None 10.1021/jm501082n
Escherichia coli Escherichia coli Ratio 32.0 None 10.1016/j.bmcl.2006.10.016
Escherichia coli Escherichia coli Ratio 32.0 None 10.1016/j.ejmech.2019.111636
Escherichia coli Escherichia coli Ratio 85.0 None 10.1128/aac.00405-08
Escherichia coli Escherichia coli Ratio 85.0 None 10.1128/aac.01439-09
Escherichia coli Escherichia coli Ratio 125.0 None 10.1128/aac.00405-08
Escherichia coli Escherichia coli Ratio 170.0 None 10.1128/aac.00405-08
Escherichia coli Escherichia coli Ratio 250.0 None 10.1128/aac.00405-08
Escherichia coli Escherichia coli Ratio 250.0 None 10.1128/aac.01439-09
Escherichia coli GroEL/GroES IC50 100000.0 nM 10.1021/acs.jmedchem.8b01293
Escherichia coli LexA repressor Activity nan None 10.1021/acs.jmedchem.0c00328
Escherichia coli K-12 Beta-lactamase AmpC Potency 707.9 nM None
Escherichia coli K-12 Cell division inhibitor sulA Activity nan None 10.1021/acs.jmedchem.0c00328
Escherichia coli K-12 DNA-directed RNA polymerase beta chain Inhibition 57.0 % 10.1021/jm00125a022
Escherichia coli K-12 Phospho-N-acetylmuramoyl-pentapeptide-transferase IC50 nan ug.mL-1 10.1016/s0960-894x(03)00597-3
Escherichia coli K-12 Recombinase A Activity nan None 10.1021/acs.jmedchem.0c00328
Escherichia coli O127:H6 (strain E2348/69 / EPEC) DNA-directed RNA polymerase subunit beta IC50 171000.0 nM 10.1021/jm4004889
Escherichia coli O127:H6 (strain E2348/69 / EPEC) DNA-directed RNA polymerase subunit beta IC50 233000.0 nM 10.1021/jm4004889
Escherichia coli O127:H6 (strain E2348/69 / EPEC) DNA-directed RNA polymerase subunit beta IC50 1130000.0 nM 10.1021/jm4004889
Fannyhessea vaginae Fannyhessea vaginae MIC 0.25 ug.mL-1 10.1021/acs.jmedchem.1c02045
Fusobacterium nucleatum Fusobacterium nucleatum MIC 0.5 ug.mL-1 10.1021/acs.jmedchem.1c02045
Fusobacterium nucleatum Fusobacterium nucleatum MIC 1.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Gardnerella vaginalis Gardnerella vaginalis MIC 0.5 ug.mL-1 10.1021/acs.jmedchem.1c02045
Haemophilus influenzae Haemophilus influenzae Inhibition 10.0 % 10.1128/aac.00471-08
Haemophilus influenzae Haemophilus influenzae Inhibition nan % 10.1128/aac.00471-08
Haemophilus influenzae Haemophilus influenzae log10cfu 8.14 None 10.1128/aac.00471-08
Haemophilus influenzae Haemophilus influenzae MIC 0.0008 ug.mL-1 10.1128/aac.00471-08
Haemophilus influenzae Haemophilus influenzae MIC 0.125 ug.mL-1 10.1021/jm00167a029
Haemophilus influenzae Haemophilus influenzae MIC 0.25 ug.mL-1 10.1128/aac.01545-06
Haemophilus influenzae Haemophilus influenzae MIC 0.5 ug.mL-1 10.1128/aac.01545-06
Haemophilus influenzae Haemophilus influenzae MIC 25.0 nM 10.1021/acs.jmedchem.5b00050
Haemophilus influenzae Haemophilus influenzae MIC 128.0 ug.mL-1 10.1128/aac.01545-06
Helicobacter pylori Helicobacter pylori MIC 0.007 ug.mL-1 10.1021/acs.jmedchem.1c02045
Helicobacter pylori Helicobacter pylori MIC 0.06 ug.mL-1 10.1021/acs.jmedchem.1c02045
Helicobacter pylori Helicobacter pylori MIC 0.25 ug.mL-1 10.1021/acs.jmedchem.1c02045
Helicobacter pylori Helicobacter pylori MIC 0.5 ug.mL-1 10.1021/acs.jmedchem.1c02045
Helicobacter pylori Helicobacter pylori MIC 2.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Helicobacter pylori Helicobacter pylori MIC 8.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Helicobacter pylori Helicobacter pylori MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Helicobacter pylori Helicobacter pylori MIC 32.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Helicobacter pylori Helicobacter pylori MIC90 0.5 ug.mL-1 10.1021/acs.jmedchem.1c02045
Helicobacter pylori Helicobacter pylori MIC90 2.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Homo sapiens A549 Activity 34.0 % 10.1128/aac.00985-07
Homo sapiens A549 Activity 45.0 % 10.1128/aac.00985-07
Homo sapiens A549 Activity 47.0 % 10.1128/aac.00985-07
Homo sapiens A549 Activity 53.0 % 10.1128/aac.00985-07
Homo sapiens A549 Activity 59.0 % 10.1128/aac.00985-07
Homo sapiens A549 Activity 79.0 % 10.1128/aac.00985-07
Homo sapiens A549 Activity 95.0 % 10.1128/aac.00985-07
Homo sapiens A549 Activity 178.0 ug ml-1 10.1016/j.bmcl.2009.09.095
Homo sapiens A549 Activity nan None 10.1128/aac.00961-08
Homo sapiens A549 Activity nan None 10.1128/aac.00985-07
Homo sapiens A549 CD50 nan None 10.1016/j.bmc.2013.07.003
Homo sapiens A549 FC 1.9 None 10.1128/aac.00961-08
Homo sapiens A549 FC 2.1 None 10.1128/aac.00961-08
Homo sapiens A549 FC 4.0 None 10.1128/aac.00961-08
Homo sapiens A549 GI50 100.0 ug.mL-1 10.1016/j.bmcl.2016.03.045
Homo sapiens A549 GI50 100.0 ug.mL-1 10.1016/j.bmcl.2017.01.004
Homo sapiens A549 GI50 100.0 ug.mL-1 10.1016/j.bmcl.2019.03.020
Homo sapiens A549 GI50 100.0 ug.mL-1 10.1016/j.ejmech.2017.03.065
Homo sapiens A549 GI50 100.0 ug.mL-1 10.1039/C5MD00404G
Homo sapiens A549 GI50 121510000.0 nM 10.1039/C6MD00278A
Homo sapiens A549 GI90 100.0 ug ml-1 10.1016/j.bmcl.2017.01.004
Homo sapiens A549 GI90 100.0 ug ml-1 10.1016/j.bmcl.2019.03.020
Homo sapiens A549 GI90 100.0 ug ml-1 10.1016/j.ejmech.2017.03.065
Homo sapiens A549 Inhibition 5.5 % 10.1128/aac.00985-07
Homo sapiens A549 Inhibition 8.3 % 10.1128/aac.00985-07
Homo sapiens A549 Inhibition nan % 10.1128/aac.00985-07
Homo sapiens Acetylcholinesterase IC50 nan None None
Homo sapiens Acetylcholinesterase Inhibition 12.2 % 10.1016/j.ejmech.2018.04.058
Homo sapiens Acetylcholinesterase Ki nan None None
Homo sapiens Adenosine A1 receptor AC50 18808.1 nM 10.1038/s41467-023-40064-9
Homo sapiens Adenosine A1 receptor IC50 nan None None
Homo sapiens Adenosine A1 receptor Ki nan None None
Homo sapiens Adenosine A2a receptor AC50 12966.1 nM 10.1038/s41467-023-40064-9
Homo sapiens Adenosine A2a receptor IC50 nan None None
Homo sapiens Adenosine A2a receptor Ki nan None None
Homo sapiens Adenosine A3 receptor AC50 26999.8 nM 10.1038/s41467-023-40064-9
Homo sapiens Adenosine A3 receptor IC50 nan None None
Homo sapiens Adenosine A3 receptor Ki nan None None
Homo sapiens Alpha-1a adrenergic receptor AC50 2331.5 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-1a adrenergic receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-1a adrenergic receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-1d adrenergic receptor IC50 nan None None
Homo sapiens Alpha-1d adrenergic receptor Ki nan None None
Homo sapiens Alpha-2a adrenergic receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-2a adrenergic receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-2a adrenergic receptor IC50 nan None None
Homo sapiens Alpha-2a adrenergic receptor Ki nan None None
Homo sapiens Alpha-2b adrenergic receptor AC50 12000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-2b adrenergic receptor IC50 nan None None
Homo sapiens Alpha-2b adrenergic receptor Ki nan None None
Homo sapiens Alpha-2c adrenergic receptor AC50 10999.9 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-2c adrenergic receptor IC50 nan None None
Homo sapiens Alpha-2c adrenergic receptor Ki nan None None
Homo sapiens Alpha-synuclein IC50 7100.0 nM 10.1016/j.ejmech.2019.01.045
Homo sapiens Alpha-synuclein IC50 46200.0 nM 10.1016/j.ejmech.2019.01.045
Homo sapiens Amyloid-beta A4 protein Activity 48.4 % 10.1039/C9MD00030E
Homo sapiens Amyloid-beta A4 protein Inhibition 27.5 % 10.1016/j.ejmech.2018.04.058
Homo sapiens Angiotensin II type 2 (AT-2) receptor IC50 nan None None
Homo sapiens Angiotensin II type 2 (AT-2) receptor Ki nan None None
Homo sapiens Arylacetamide deacetylase Drug metabolism 41.77 pmol/min/mg 10.1124/dmd.112.044537
Homo sapiens Arylacetamide deacetylase Ki 200000.0 nM 10.1124/dmd.111.043067
Homo sapiens Arylacetamide deacetylase Ki 300000.0 nM 10.1124/dmd.111.043067
Homo sapiens Arylacetamide deacetylase Ki 700000.0 nM 10.1124/dmd.111.043067
Homo sapiens Arylacetamide deacetylase Km 200000.0 nM 10.1124/dmd.111.043067
Homo sapiens Arylacetamide deacetylase Km 300000.0 nM 10.1124/dmd.111.043067
Homo sapiens Arylacetamide deacetylase Km 400000.0 nM 10.1124/dmd.111.043067
Homo sapiens Arylacetamide deacetylase Vmax 149.0 pmol/min/U 10.1124/dmd.111.043067
Homo sapiens Arylacetamide deacetylase Vmax 211.8 pmol/min/mg 10.1124/dmd.111.043067
Homo sapiens Arylacetamide deacetylase Vmax 272.6 pmol/min/mg 10.1124/dmd.111.043067
Homo sapiens Arylacetamide deacetylase Vmax/Km 0.9 uL/min/U 10.1124/dmd.111.043067
Homo sapiens ATP-binding cassette sub-family G member 2 IC50 56000.0 nM 10.1016/j.ejmech.2022.114346
Homo sapiens Beta-1 adrenergic receptor AC50 28000.1 nM 10.1038/s41467-023-40064-9
Homo sapiens Beta-1 adrenergic receptor IC50 nan None None
Homo sapiens Beta-1 adrenergic receptor Ki nan None None
Homo sapiens Beta-2 adrenergic receptor AC50 29000.1 nM 10.1038/s41467-023-40064-9
Homo sapiens Beta-2 adrenergic receptor IC50 nan None None
Homo sapiens Beta-2 adrenergic receptor Ki nan None None
Homo sapiens Beta-3 adrenergic receptor AC50 32600.2 nM 10.1038/s41467-023-40064-9
Homo sapiens Beta-3 adrenergic receptor IC50 nan None None
Homo sapiens Beta-3 adrenergic receptor Ki nan None None
Homo sapiens Bile acid receptor FXR AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Bile acid receptor FXR AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Bile salt export pump AC50 9600.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Bile salt export pump Activity nan None 10.1038/nrd3028
Homo sapiens Bile salt export pump IC50 11300.0 nM 10.1124/dmd.111.040758
Homo sapiens Bile salt export pump IC50 18700.0 nM 10.1002/hep.27206
Homo sapiens Bile salt export pump IC50 25300.0 nM 10.1093/toxsci/kfq269
Homo sapiens Bile salt export pump IC50 25300.0 nM 10.1093/toxsci/kft176
Homo sapiens Bradykinin B1 receptor AC50 14249.8 nM 10.1038/s41467-023-40064-9
Homo sapiens Bradykinin B2 receptor AC50 18577.4 nM 10.1038/s41467-023-40064-9
Homo sapiens Bradykinin B2 receptor IC50 nan None None
Homo sapiens Bradykinin B2 receptor Ki nan None None
Homo sapiens Brain Drug uptake 0.29 ug ml-1 10.1021/jm901858n
Homo sapiens Bromodomain adjacent to zinc finger domain protein 2B Potency 50118.7 nM None
Homo sapiens Calcitonin receptor IC50 nan None None
Homo sapiens Calcitonin receptor Ki nan None None
Homo sapiens Canalicular multispecific organic anion transporter 1 Activity 18.0 % 10.1021/jm7015683
Homo sapiens Canalicular multispecific organic anion transporter 1 Activity nan None 10.1016/s0002-9440(10)64794-3
Homo sapiens Canalicular multispecific organic anion transporter 1 Activity nan None 10.1016/s0300-483x(01)00570-4
Homo sapiens Canalicular multispecific organic anion transporter 1 IC50 53000.0 nM 10.1093/toxsci/kft176
Homo sapiens Canalicular multispecific organic anion transporter 2 IC50 69000.0 nM 10.1093/toxsci/kft176
Homo sapiens Cannabinoid CB1 receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Cannabinoid CB1 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Cannabinoid CB1 receptor IC50 nan None None
Homo sapiens Cannabinoid CB1 receptor Ki nan None None
Homo sapiens Carbonic anhydrase II IC50 nan None None
Homo sapiens Carbonic anhydrase II Ki nan None None
Homo sapiens Carboxylesterase 2 Drug metabolism 2.99 pmol/min/mg 10.1124/dmd.112.044537
Homo sapiens Caspase-1 IC50 8319.0 nM None
Homo sapiens Caspase-1 Ki nan None None
Homo sapiens Cathepsin G IC50 nan None None
Homo sapiens Cathepsin G Ki nan None None
Homo sapiens C-C chemokine receptor type 2 IC50 nan None None
Homo sapiens C-C chemokine receptor type 2 Ki nan None None
Homo sapiens C-C chemokine receptor type 4 IC50 nan None None
Homo sapiens C-C chemokine receptor type 4 Ki nan None None
Homo sapiens C-C chemokine receptor type 5 IC50 nan None None
Homo sapiens C-C chemokine receptor type 5 Ki nan None None
Homo sapiens Cholecystokinin A receptor AC50 17080.1 nM 10.1038/s41467-023-40064-9
Homo sapiens Cholecystokinin A receptor IC50 nan None None
Homo sapiens Cholecystokinin A receptor Ki nan None None
Homo sapiens Cholecystokinin B receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Chromobox protein homolog 1 Potency 39810.7 nM None
Homo sapiens Corticotropin releasing factor receptor 1 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Corticotropin releasing factor receptor 2 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Cyclooxygenase-1 IC50 nan None None
Homo sapiens Cyclooxygenase-1 Ki nan None None
Homo sapiens Cyclooxygenase-2 AC50 6400.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Cyclooxygenase-2 IC50 nan None None
Homo sapiens Cyclooxygenase-2 Ki nan None None
Homo sapiens Cysteinyl leukotriene receptor 1 IC50 nan None None
Homo sapiens Cysteinyl leukotriene receptor 1 Ki nan None None
Homo sapiens Cytochrome P450 Activity 65.0 % 10.1021/acs.jmedchem.0c02245
Homo sapiens Cytochrome P450 1A2 FC 1.37 None 10.1128/aac.00660-09
Homo sapiens Cytochrome P450 1A2 IC50 nan None None
Homo sapiens Cytochrome P450 1A2 Inhibition nan % 10.1021/tx300075j
Homo sapiens Cytochrome P450 1A2 Ki nan None None
Homo sapiens Cytochrome P450 2A6 IC50 nan None None
Homo sapiens Cytochrome P450 2A6 Ki nan None None
Homo sapiens Cytochrome P450 2B6 Activity nan None None
Homo sapiens Cytochrome P450 2B6 EC50 1300.0 nM 10.1124/dmd.112.047118
Homo sapiens Cytochrome P450 2B6 Emax 16.9 None 10.1124/dmd.112.047118
Homo sapiens Cytochrome P450 2B6 FC 3.6 None 10.1128/aac.00660-09
Homo sapiens Cytochrome P450 2B6 FC 13.9 None 10.1124/dmd.112.045765
Homo sapiens Cytochrome P450 2C19 Activity nan None None
Homo sapiens Cytochrome P450 2C19 IC50 nan None None
Homo sapiens Cytochrome P450 2C19 Inhibition nan % 10.1021/tx300075j
Homo sapiens Cytochrome P450 2C19 Ki nan None None
Homo sapiens Cytochrome P450 2C8 Activity nan None None
Homo sapiens Cytochrome P450 2C9 Activity nan None None
Homo sapiens Cytochrome P450 2C9 FC 1.0 None 10.1016/j.bmcl.2016.06.088
Homo sapiens Cytochrome P450 2C9 FC 2.96 None 10.1124/dmd.112.047928
Homo sapiens Cytochrome P450 2C9 FC 3.6 None 10.1124/dmd.112.045765
Homo sapiens Cytochrome P450 2C9 IC50 nan None None
Homo sapiens Cytochrome P450 2C9 Inhibition nan % 10.1021/tx300075j
Homo sapiens Cytochrome P450 2C9 Ki nan None None
Homo sapiens Cytochrome P450 2D6 FC 1.0 None 10.1016/j.bmcl.2016.06.088
Homo sapiens Cytochrome P450 2D6 IC50 nan None None
Homo sapiens Cytochrome P450 2D6 Inhibition nan % 10.1021/tx300075j
Homo sapiens Cytochrome P450 2D6 Ki nan None None
Homo sapiens Cytochrome P450 2E1 IC50 nan None None
Homo sapiens Cytochrome P450 2E1 Ki nan None None
Homo sapiens Cytochrome P450 3A Activity 98.0 % 10.1021/acs.jmedchem.0c02245
Homo sapiens Cytochrome P450 3A Activity 99.7 % 10.1021/acs.jmedchem.0c02245
Homo sapiens Cytochrome P450 3A4 Activity 6.0 % 10.1021/jm300601d
Homo sapiens Cytochrome P450 3A4 Activity 20.0 % 10.1016/j.bmcl.2022.128843
Homo sapiens Cytochrome P450 3A4 Activity 46.0 % 10.1021/acs.jmedchem.0c02245
Homo sapiens Cytochrome P450 3A4 Activity 86.0 % 10.1021/acs.jmedchem.0c02245
Homo sapiens Cytochrome P450 3A4 Activity 92.0 % 10.1021/acs.jmedchem.0c02245
Homo sapiens Cytochrome P450 3A4 Activity 100.0 % 10.1021/jm801073z
Homo sapiens Cytochrome P450 3A4 Activity nan None 10.1021/acs.jmedchem.5b01078
Homo sapiens Cytochrome P450 3A4 Activity nan None None
Homo sapiens Cytochrome P450 3A4 Emax 5.0 % 10.1021/acs.jmedchem.1c01887
Homo sapiens Cytochrome P450 3A4 FC 1.0 None 10.1016/j.bmcl.2016.06.088
Homo sapiens Cytochrome P450 3A4 FC 6.63 None 10.1128/aac.00660-09
Homo sapiens Cytochrome P450 3A4 FC 12.5 None 10.1124/dmd.112.047928
Homo sapiens Cytochrome P450 3A4 FC 24.4 None 10.1124/dmd.112.045765
Homo sapiens Cytochrome P450 3A4 FC 30.0 None 10.1124/dmd.110.035840
Homo sapiens Cytochrome P450 3A4 IC50 nan None None
Homo sapiens Cytochrome P450 3A4 Inhibition nan % 10.1021/tx300075j
Homo sapiens Cytochrome P450 3A4 Ki nan None None
Homo sapiens Cytochrome P450 3A4 Ratio 4.3 None 10.1016/j.bmcl.2014.10.032
Homo sapiens Cytochrome P450 3A5 Activity nan None 10.1021/acs.jmedchem.5b01078
Homo sapiens Cytochrome P450 51 IC50 30000.0 nM 10.1124/dmd.106.013888
Homo sapiens Delta opioid receptor AC50 17000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Delta opioid receptor IC50 nan None None
Homo sapiens Delta opioid receptor Ki nan None None
Homo sapiens DLD-1 Activity nan None 10.1128/aac.00961-08
Homo sapiens DNA polymerase iota Potency 89125.1 nM None
Homo sapiens Dopamine D1 receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine D1 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine D1 receptor IC50 nan None None
Homo sapiens Dopamine D1 receptor Ki nan None None
Homo sapiens Dopamine D2 receptor AC50 9200.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine D2 receptor IC50 nan None None
Homo sapiens Dopamine D2 receptor Ki nan None None
Homo sapiens Dopamine D3 receptor AC50 10999.9 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine D3 receptor IC50 nan None None
Homo sapiens Dopamine D3 receptor Ki nan None None
Homo sapiens Dopamine D4 receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine D4 receptor IC50 nan None None
Homo sapiens Dopamine D4 receptor Ki nan None None
Homo sapiens Dopamine transporter AC50 20000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine transporter IC50 nan None None
Homo sapiens Dopamine transporter Ki nan None None
Homo sapiens Endothelin receptor ET-A AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Endothelin receptor ET-A IC50 nan None None
Homo sapiens Endothelin receptor ET-A Ki nan None None
Homo sapiens Endothelin receptor ET-B AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Epidermal growth factor receptor erbB1 IC50 nan None None
Homo sapiens Epidermal growth factor receptor erbB1 Ki nan None None
Homo sapiens Equilibrative nucleoside transporter 1 AC50 12445.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Estrogen receptor alpha AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Estrogen receptor alpha IC50 nan None None
Homo sapiens Estrogen receptor alpha Ki nan None None
Homo sapiens Estrogen receptor beta AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Estrogen receptor beta IC50 nan None None
Homo sapiens Estrogen receptor beta Ki nan None None
Homo sapiens Galactocerebrosidase Potency 631.0 nM None
Homo sapiens Gastric inhibitory polypeptide receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Geminin Potency 29092.9 nM None
Homo sapiens Ghrelin receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Glucagon receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Glucocorticoid receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Glucocorticoid receptor IC50 nan None None
Homo sapiens Glucocorticoid receptor Ki nan None None
Homo sapiens Glutathione transferase omega 1 IC50 75000.0 nM 10.1021/acs.jmedchem.8b00318
Homo sapiens Guanine nucleotide-binding protein G(s), subunit alpha Potency 39810.7 nM None
Homo sapiens HaCaT Survival 55.0 % 10.1021/acs.jnatprod.5b01033
Homo sapiens HCT-116 GI50 100.0 ug.mL-1 10.1016/j.bmcl.2017.01.004
Homo sapiens HCT-116 GI50 121510000.0 nM 10.1039/C6MD00278A
Homo sapiens HCT-116 GI90 100.0 ug ml-1 10.1016/j.bmcl.2017.01.004
Homo sapiens HEK293 CC50 100000.0 nM 10.1021/acs.jmedchem.8b01293
Homo sapiens HEK293 IC50 nan None 10.1016/j.bmcl.2012.12.096
Homo sapiens HEK293 Inhibition nan % 10.1016/j.ejmech.2018.07.047
Homo sapiens HEK293 LC50 200.0 ug.mL-1 10.1016/j.bmc.2008.10.042
Homo sapiens HEK293 LC50 100000.0 nM 10.1021/jm400240r
Homo sapiens HEK-293T Activity nan None 10.1016/j.bmcl.2012.10.060
Homo sapiens HeLa Activity 100.4 % 10.1021/acs.jmedchem.5b00608
Homo sapiens HeLa Activity 101.7 % 10.1021/acs.jmedchem.5b00608
Homo sapiens HeLa CC50 100.0 ug.mL-1 10.1016/j.bmcl.2016.05.093
Homo sapiens HeLa CD50 190.0 uM 10.1016/j.bmcl.2008.03.025
Homo sapiens HeLa GI50 100.0 ug.mL-1 10.1016/j.bmcl.2016.03.045
Homo sapiens HeLa GI50 100.0 ug.mL-1 10.1016/j.bmcl.2019.03.020
Homo sapiens HeLa GI50 100.0 ug.mL-1 10.1016/j.ejmech.2017.03.065
Homo sapiens HeLa GI90 100.0 ug ml-1 10.1016/j.bmcl.2019.03.020
Homo sapiens HeLa GI90 100.0 ug ml-1 10.1016/j.ejmech.2017.03.065
Homo sapiens HeLa IC20 180.0 ug ml-1 10.1128/aac.00729-05
Homo sapiens HeLa IC20 nan None 10.1128/aac.00729-05
Homo sapiens HeLa IC50 270.0 ug.mL-1 10.1128/aac.00729-05
Homo sapiens HeLa IC50 20000.0 nM 10.1021/acs.jmedchem.5b00608
Homo sapiens HeLa IC50 nan None 10.1128/aac.00729-05
Homo sapiens Hepatocyte Activity 50.0 uM 10.1124/dmd.112.045765
Homo sapiens Hepatocyte Activity 100.0 % 10.1021/jm801073z
Homo sapiens Hepatocyte Activity 123.2 % 10.1021/acs.jmedchem.5b00608
Homo sapiens Hepatocyte Activity nan None 10.1016/j.bmcl.2014.10.032
Homo sapiens Hepatocyte Activity nan None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte EC50 980.0 nM 10.1124/dmd.112.047118
Homo sapiens Hepatocyte Emax 16.9 None 10.1124/dmd.112.047118
Homo sapiens Hepatocyte FC 0.7 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 0.8 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 1.0 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 1.1 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 1.2 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 1.3 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 1.4 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 2.3 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 2.5 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 2.6 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 4.3 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 8.4 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 20.2 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte FC 60.0 None 10.1124/dmd.110.035840
Homo sapiens Hepatocyte FC 74.8 None 10.1124/dmd.112.045765
Homo sapiens Hepatocyte IC50 20000.0 nM 10.1021/acs.jmedchem.5b00608
Homo sapiens HepG2 Activity 114.66 % 10.1007/s00044-010-9405-3
Homo sapiens HepG2 Activity 116.03 % 10.1007/s00044-010-9405-3
Homo sapiens HepG2 Activity 192.41 % 10.1007/s00044-010-9405-3
Homo sapiens HepG2 Activity nan None 10.1016/j.bmc.2014.11.043
Homo sapiens HepG2 CC50 175.9 ug.mL-1 10.1016/j.ejmech.2021.113472
Homo sapiens HepG2 IC50 145330.0 nM 10.1016/j.bmcl.2020.127146
Homo sapiens HERG AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens HERG IC50 nan None None
Homo sapiens HERG Inhibition nan % 10.1016/j.bmc.2019.01.022
Homo sapiens HERG Ki nan None None
Homo sapiens Histamine H1 receptor AC50 8700.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Histamine H1 receptor IC50 nan None None
Homo sapiens Histamine H1 receptor Ki nan None None
Homo sapiens Histamine H2 receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Histamine H2 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Histamine H2 receptor IC50 nan None None
Homo sapiens Histamine H2 receptor Ki nan None None
Homo sapiens Histamine H3 receptor AC50 25000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens HMG-CoA reductase IC50 nan None None
Homo sapiens HMG-CoA reductase Ki nan None None
Homo sapiens Homo sapiens Activity 5.8 % 10.1128/aac.00247-07
Homo sapiens Homo sapiens Activity 99.0 % 10.1128/aac.00579-07
Homo sapiens Homo sapiens Activity nan None 10.1002/hep.27206
Homo sapiens Homo sapiens Activity nan None 10.1128/aac.00247-07
Homo sapiens Homo sapiens AUC 13.1 ug ml-1 10.1128/aac.01474-06
Homo sapiens Homo sapiens AUC 24.5 ug ml-1 10.1128/aac.01474-06
Homo sapiens Homo sapiens AUC 100.0 ug ml-1 10.1128/aac.01474-06
Homo sapiens Homo sapiens AUC 171.0 ug ml-1 10.1128/aac.01474-06
Homo sapiens Homo sapiens AUC 6400.0 ng.hr.mL-1 10.1128/aac.01550-06
Homo sapiens Homo sapiens AUC 13200.0 ng.hr.mL-1 10.1128/aac.01550-06
Homo sapiens Homo sapiens AUC 19600.0 ng.hr.mL-1 10.1128/aac.00461-07
Homo sapiens Homo sapiens AUC 21500.0 ng.hr.mL-1 10.1128/aac.00749-08
Homo sapiens Homo sapiens AUC 23100.0 ng.hr.mL-1 10.1128/aac.00461-07
Homo sapiens Homo sapiens AUC 28200.0 ng.hr.mL-1 10.1128/aac.00461-07
Homo sapiens Homo sapiens AUC 29700.0 ng.hr.mL-1 10.1371/journal.pmed.0030466
Homo sapiens Homo sapiens AUC 30100.0 ng.hr.mL-1 10.1128/aac.00461-07
Homo sapiens Homo sapiens AUC 30700.0 ng.hr.mL-1 10.1128/aac.00461-07
Homo sapiens Homo sapiens AUC 41700.0 ng.hr.mL-1 10.1128/aac.00341-07
Homo sapiens Homo sapiens AUC 44000.0 ng.hr.mL-1 10.1128/aac.01621-06
Homo sapiens Homo sapiens AUC 44600.0 ng.hr.mL-1 10.1128/aac.00461-07
Homo sapiens Homo sapiens AUC 45700.0 ng.hr.mL-1 10.1128/aac.00341-07
Homo sapiens Homo sapiens AUC 48500.0 ng.hr.mL-1 10.1128/aac.00461-07
Homo sapiens Homo sapiens AUC 48500.0 ng.hr.mL-1 10.1128/aac.01550-06
Homo sapiens Homo sapiens AUC 49000.0 ng.hr.mL-1 10.1128/aac.00447-09
Homo sapiens Homo sapiens AUC 50600.0 ng.hr.mL-1 10.1128/aac.00447-09
Homo sapiens Homo sapiens AUC 60300.0 ng.hr.mL-1 10.1128/aac.00461-07
Homo sapiens Homo sapiens AUC 73604.65 ng.hr.mL-1 10.1093/toxsci/kft176
Homo sapiens Homo sapiens AUC 79700.0 ng.hr.mL-1 10.1128/aac.00461-07
Homo sapiens Homo sapiens AUC 79700.0 ng.hr.mL-1 10.1128/aac.01550-06
Homo sapiens Homo sapiens AUC 112000.0 ng.hr.mL-1 10.1128/aac.01533-06
Homo sapiens Homo sapiens CL 1.3 mL.min-1.kg-1 10.1021/jm901371v
Homo sapiens Homo sapiens CL 1.5 mL.min-1.kg-1 10.1021/jm900403j
Homo sapiens Homo sapiens CL 1.5 mL.min-1.kg-1 10.1021/jm901371v
Homo sapiens Homo sapiens CL 8.9 L/hr 10.1128/aac.00447-09
Homo sapiens Homo sapiens CL/F 7.5 L/hr 10.1128/aac.01550-06
Homo sapiens Homo sapiens CL/F 9.2 L/hr 10.1128/aac.00447-09
Homo sapiens Homo sapiens CL/F 9.2 L/hr 10.1128/aac.01550-06
Homo sapiens Homo sapiens CL/F 15.1 L/hr 10.1128/aac.00341-07
Homo sapiens Homo sapiens CL/F 16.5 L/hr 10.1128/aac.00341-07
Homo sapiens Homo sapiens CL/F 19.2 L/hr 10.1128/aac.00461-07
Homo sapiens Homo sapiens CL/F 19.4 L/hr 10.1128/aac.00461-07
Homo sapiens Homo sapiens CL/F 20.2 L/hr 10.1128/aac.00461-07
Homo sapiens Homo sapiens CL_renal 0.2 mL.min-1.kg-1 10.1021/jm900403j
Homo sapiens Homo sapiens CL_renal 0.2 mL.min-1.kg-1 10.1021/jm901371v
Homo sapiens Homo sapiens Cmax 1458.17 nM 10.1128/aac.01550-06
Homo sapiens Homo sapiens Cmax 2673.31 nM 10.1128/aac.01550-06
Homo sapiens Homo sapiens Cmax 3074.31 nM 10.1128/aac.01474-06
Homo sapiens Homo sapiens Cmax 3876.3 nM 10.1128/aac.01474-06
Homo sapiens Homo sapiens Cmax 4252.99 nM None
Homo sapiens Homo sapiens Cmax 6683.27 nM 10.1371/journal.pmed.0030466
Homo sapiens Homo sapiens Cmax 8000.0 nM 10.1128/aac.00527-07
Homo sapiens Homo sapiens Cmax 8500.0 nM 10.1002/hep.27206
Homo sapiens Homo sapiens Cmax 8505.98 nM None
Homo sapiens Homo sapiens Cmax 9721.13 nM 10.1128/aac.00749-08
Homo sapiens Homo sapiens Cmax 11531.68 nM 10.1128/aac.00341-07
Homo sapiens Homo sapiens Cmax 11665.35 nM 10.1128/aac.00447-09
Homo sapiens Homo sapiens Cmax 12151.41 nM 10.1128/aac.01605-07
Homo sapiens Homo sapiens Cmax 12285.07 nM 10.1128/aac.00341-07
Homo sapiens Homo sapiens Cmax 12758.98 nM 10.1128/aac.00375-07
Homo sapiens Homo sapiens Cmax 12758.98 nM 10.1128/aac.00447-09
Homo sapiens Homo sapiens Cmax 12758.98 nM 10.1128/aac.01550-06
Homo sapiens Homo sapiens Cmax 13002.0 nM None
Homo sapiens Homo sapiens Cmax 13974.12 nM None
Homo sapiens Homo sapiens Cmax 15796.83 nM 10.1128/aac.01474-06
Homo sapiens Homo sapiens Cmax 17011.97 nM 10.1128/aac.01474-06
Homo sapiens Homo sapiens Cmax 18956.19 nM 10.1128/aac.01550-06
Homo sapiens Homo sapiens Cmin 329.0 ng/ml 10.1128/aac.00341-07
Homo sapiens Homo sapiens Cmin 360.0 ng/ml 10.1128/aac.00341-07
Homo sapiens Homo sapiens Cp 9.9 ug ml-1 10.1128/aac.01621-06
Homo sapiens Homo sapiens Css 3.726 uM 10.1093/toxsci/kft176
Homo sapiens Homo sapiens DILI_Concern nan None 10.1016/j.drudis.2016.02.015
Homo sapiens Homo sapiens DILI_severity_class 8.0 None 10.1016/j.drudis.2016.02.015
Homo sapiens Homo sapiens F 50.0 % 10.1021/jm400887j
Homo sapiens Homo sapiens F 68.0 % 10.1128/aac.00749-08
Homo sapiens Homo sapiens F 69.0 % 10.1128/aac.00447-09
Homo sapiens Homo sapiens F 74.0 % 10.1128/aac.00447-09
Homo sapiens Homo sapiens F 88.8 % 10.1016/j.bmc.2007.08.060
Homo sapiens Homo sapiens Fa 1.0 None 10.1021/jm901371v
Homo sapiens Homo sapiens fAUC 16000.0 ng.hr.mL-1 10.1128/aac.01533-06
Homo sapiens Homo sapiens fAUC 112000.0 ng.hr.mL-1 10.1128/aac.01533-06
Homo sapiens Homo sapiens FC 45.0 None 10.1128/aac.00579-07
Homo sapiens Homo sapiens FC 178.0 None 10.1128/aac.00579-07
Homo sapiens Homo sapiens FC 422.0 None 10.1128/aac.00579-07
Homo sapiens Homo sapiens fCmax 2.0 mg/L 10.1128/aac.01533-06
Homo sapiens Homo sapiens fCmax 2.0 ug ml-1 10.1128/aac.00766-08
Homo sapiens Homo sapiens fCmax 7.0 mg/L 10.1128/aac.01533-06
Homo sapiens Homo sapiens fCmax 14.0 mg/L 10.1128/aac.01533-06
Homo sapiens Homo sapiens F_fraction 0.93 None 10.1021/jm901371v
Homo sapiens Homo sapiens Fg 0.99 None 10.1021/jm901371v
Homo sapiens Homo sapiens Fh 0.94 None 10.1021/jm901371v
Homo sapiens Homo sapiens Ka 1.15 L/hr 10.1128/aac.00461-07
Homo sapiens Homo sapiens Ka 1.23 L/hr 10.1128/aac.00461-07
Homo sapiens Homo sapiens Ka 1.61 L/hr 10.1128/aac.00461-07
Homo sapiens Homo sapiens Ka 1.64 L/hr 10.1128/aac.00461-07
Homo sapiens Homo sapiens MTT 0.424 hr 10.1128/aac.00461-07
Homo sapiens Homo sapiens Ratio 0.82 None 10.1128/aac.01550-06
Homo sapiens Homo sapiens Ratio 0.92 None 10.1128/aac.01550-06
Homo sapiens Homo sapiens Ratio 0.94 None 10.1128/aac.00447-09
Homo sapiens Homo sapiens Ratio 0.97 None 10.1128/aac.00447-09
Homo sapiens Homo sapiens Ratio 0.98 None 10.1128/aac.00447-09
Homo sapiens Homo sapiens Ratio 1.04 None 10.1128/aac.00447-09
Homo sapiens Homo sapiens Ratio 1.09 None 10.1128/aac.00447-09
Homo sapiens Homo sapiens Ratio 1.13 None 10.1128/aac.01550-06
Homo sapiens Homo sapiens Ratio 70.8 None 10.1128/aac.00749-08
Homo sapiens Homo sapiens Ratio AUC 1.49 None 10.1128/aac.01550-06
Homo sapiens Homo sapiens Ratio AUC 1.65 None 10.1128/aac.01550-06
Homo sapiens Homo sapiens T1/2 1.4 hr 10.1128/aac.00341-07
Homo sapiens Homo sapiens T1/2 1.6 hr 10.1128/aac.00341-07
Homo sapiens Homo sapiens T1/2 1.9 hr 10.1128/aac.01550-06
Homo sapiens Homo sapiens T1/2 1.9 hr 10.1128/aac.01621-06
Homo sapiens Homo sapiens T1/2 2.0 hr 10.1128/aac.00749-08
Homo sapiens Homo sapiens T1/2 2.0 hr None
Homo sapiens Homo sapiens T1/2 2.1 hr 10.1128/aac.00447-09
Homo sapiens Homo sapiens T1/2 2.2 hr 10.1128/aac.00447-09
Homo sapiens Homo sapiens T1/2 2.2 hr 10.1128/aac.01550-06
Homo sapiens Homo sapiens T1/2 2.5 hr 10.1128/aac.01550-06
Homo sapiens Homo sapiens T1/2 2.9 hr None
Homo sapiens Homo sapiens T1/2 3.0 hr 10.1128/aac.01533-06
Homo sapiens Homo sapiens T1/2 3.0 hr 10.1128/aac.01605-07
Homo sapiens Homo sapiens T1/2 3.2 hr 10.1128/aac.01550-06
Homo sapiens Homo sapiens T1/2 3.35 hr None
Homo sapiens Homo sapiens T1/2 3.5 hr 10.1128/aac.00527-07
Homo sapiens Homo sapiens T1/2 3.6 hr None
Homo sapiens Homo sapiens T1/2 5.0 hr None
Homo sapiens Homo sapiens T1/2 5.08 hr None
Homo sapiens Homo sapiens T1/2 7.3 hr None
Homo sapiens Homo sapiens T1/2 11.0 hr None
Homo sapiens Homo sapiens TIME 3.611e-06 hr 10.1128/aac.01204-07
Homo sapiens Homo sapiens Tmax 1.0 hr 10.1128/aac.00527-07
Homo sapiens Homo sapiens Tmax 1.0 hr 10.1128/aac.01550-06
Homo sapiens Homo sapiens Tmax 1.0 hr None
Homo sapiens Homo sapiens Tmax 1.5 hr 10.1128/aac.00749-08
Homo sapiens Homo sapiens Tmax 2.0 hr 10.1128/aac.00447-09
Homo sapiens Homo sapiens Tmax 2.0 hr 10.1128/aac.01550-06
Homo sapiens Homo sapiens Tmax 2.5 hr 10.1128/aac.00447-09
Homo sapiens Homo sapiens Tmax 2.5 hr 10.1128/aac.01474-06
Homo sapiens Homo sapiens Tmax 2.7 hr 10.1128/aac.00341-07
Homo sapiens Homo sapiens Tmax 3.12 hr 10.1128/aac.01474-06
Homo sapiens Homo sapiens Tmax 3.27 hr 10.1128/aac.01474-06
Homo sapiens Homo sapiens Tmax 3.67 hr 10.1128/aac.01474-06
Homo sapiens Homo sapiens Tmax 4.0 hr 10.1128/aac.01550-06
Homo sapiens Homo sapiens Vbeta 32.0 l 10.1128/aac.00341-07
Homo sapiens Homo sapiens Vbeta 33.0 l 10.1128/aac.00341-07
Homo sapiens Homo sapiens Vc/F 23.3 l 10.1128/aac.01550-06
Homo sapiens Homo sapiens Vc/F 25.3 l 10.1128/aac.01550-06
Homo sapiens Homo sapiens Vc/F 27.4 l 10.1128/aac.00447-09
Homo sapiens Homo sapiens Vc/F 27.6 l 10.1128/aac.00447-09
Homo sapiens Homo sapiens Vd 8.05 l 10.1128/aac.01520-08
Homo sapiens Homo sapiens Vd 10.16 l 10.1128/aac.01520-08
Homo sapiens Homo sapiens Vd 11.56 l 10.1128/aac.01520-08
Homo sapiens Homo sapiens Vdss 0.97 L.kg-1 10.1021/jm901371v
Homo sapiens Homo sapiens Vz 51.5 l 10.1128/aac.00461-07
Homo sapiens Homo sapiens Vz 52.8 l 10.1128/aac.00461-07
Homo sapiens Homo sapiens Vz 53.2 l 10.1128/aac.00461-07
Homo sapiens Homo sapiens Vz 53.4 l 10.1128/aac.00461-07
Homo sapiens HSP60/HSP10 IC50 100000.0 nM 10.1021/acs.jmedchem.8b01293
Homo sapiens HT-29 Activity nan None 10.1128/aac.00961-08
Homo sapiens Interleukin-8 receptor A IC50 nan None None
Homo sapiens Interleukin-8 receptor A Ki nan None None
Homo sapiens Interleukin-8 receptor B IC50 nan None None
Homo sapiens Interleukin-8 receptor B Ki nan None None
Homo sapiens Jurkat CD50 nan None 10.1016/j.bmc.2013.07.003
Homo sapiens Kappa opioid receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Kappa opioid receptor IC50 nan None None
Homo sapiens Kappa opioid receptor Ki nan None None
Homo sapiens Leukocyte common antigen IC50 nan None None
Homo sapiens Leukocyte common antigen Ki nan None None
Homo sapiens Leukocyte elastase IC50 nan None None
Homo sapiens Leukocyte elastase Ki nan None None
Homo sapiens Liver microsome CL 0.7 mL.min-1.g-1 10.1124/dmd.111.043067
Homo sapiens Liver microsome Stability nan % 10.1021/acs.jmedchem.5b01542
Homo sapiens Liver microsomes Activity nan None 10.1021/tx300075j
Homo sapiens Liver microsomes Stability nan % 10.1021/tx300075j
Homo sapiens LS180 Activity nan None 10.1039/C6MD00300A
Homo sapiens LXR-alpha AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens LXR-beta AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens MAP kinase ERK1 IC50 nan None None
Homo sapiens MAP kinase ERK1 Ki nan None None
Homo sapiens MAP kinase ERK2 IC50 nan None None
Homo sapiens MAP kinase ERK2 Ki nan None None
Homo sapiens MAP kinase p38 alpha IC50 nan None None
Homo sapiens MAP kinase p38 alpha Ki nan None None
Homo sapiens Matrix metalloproteinase-1 IC50 nan None None
Homo sapiens Matrix metalloproteinase-1 Ki nan None None
Homo sapiens Matrix metalloproteinase 9 IC50 nan None None
Homo sapiens Matrix metalloproteinase 9 Ki nan None None
Homo sapiens MCF7 GI50 100.0 ug.mL-1 10.1016/j.bmcl.2017.01.004
Homo sapiens MCF7 GI50 100.0 ug.mL-1 10.1039/C5MD00404G
Homo sapiens MCF7 GI50 121510000.0 nM 10.1039/C6MD00278A
Homo sapiens MCF7 GI90 100.0 ug ml-1 10.1016/j.bmcl.2017.01.004
Homo sapiens Melanocortin receptor 3 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Melanocortin receptor 3 IC50 nan None None
Homo sapiens Melanocortin receptor 3 Ki nan None None
Homo sapiens Melanocortin receptor 4 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Melanocortin receptor 4 IC50 nan None None
Homo sapiens Melanocortin receptor 4 Ki nan None None
Homo sapiens Melanocortin receptor 5 IC50 nan None None
Homo sapiens Melanocortin receptor 5 Ki nan None None
Homo sapiens MG-63 IC20 120.0 ug ml-1 10.1128/aac.00729-05
Homo sapiens MG-63 IC20 nan None 10.1128/aac.00729-05
Homo sapiens MG-63 IC50 240.0 ug.mL-1 10.1128/aac.00729-05
Homo sapiens MG-63 IC50 nan None 10.1128/aac.00729-05
Homo sapiens Monoamine oxidase A AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Monoamine oxidase A Activity nan None 10.1021/jm800656v
Homo sapiens Monoamine oxidase A IC50 nan None None
Homo sapiens Monoamine oxidase A Ki nan None None
Homo sapiens Motilin receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens MRC5 Activity 65.0 ug ml-1 10.1016/j.bmcl.2009.09.095
Homo sapiens MRC5 CC50 nan None 10.1016/j.ejmech.2017.06.061
Homo sapiens MRC5 IC50 100000.0 nM 10.1021/acs.jnatprod.5b00266
Homo sapiens MRC5 IC50 nan None 10.1016/j.bmcl.2019.02.019
Homo sapiens MRC5 IC50 nan None 10.1016/j.ejmech.2022.114831
Homo sapiens MRC5 IC50 nan None 10.1021/acs.jmedchem.7b01332
Homo sapiens MRC5 IC90 100000.0 nM 10.1021/acs.jnatprod.5b00266
Homo sapiens MRC5 Survival 53.0 % 10.1021/acs.jnatprod.5b01033
Homo sapiens Multidrug resistance-associated protein 1 Activity 110.0 % 10.1016/s0304-3835(99)00024-5
Homo sapiens Multidrug resistance-associated protein 4 IC50 41900.0 nM 10.1093/toxsci/kft176
Homo sapiens Multidrug resistance-associated protein 5 Activity nan None 10.1016/s0378-4274(01)00306-x
Homo sapiens Mu opioid receptor AC50 8000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Mu opioid receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Mu opioid receptor IC50 nan None None
Homo sapiens Mu opioid receptor Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M1 AC50 7100.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Muscarinic acetylcholine receptor M1 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M1 Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M2 AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Muscarinic acetylcholine receptor M2 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Muscarinic acetylcholine receptor M2 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M2 Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M3 AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Muscarinic acetylcholine receptor M3 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M3 Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M4 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M4 Ki nan None None
Homo sapiens Muscarinic acetylcholine receptor M5 IC50 nan None None
Homo sapiens Muscarinic acetylcholine receptor M5 Ki nan None None
Homo sapiens Neurokinin 1 receptor IC50 nan None None
Homo sapiens Neurokinin 1 receptor Ki nan None None
Homo sapiens Neurokinin 2 receptor IC50 nan None None
Homo sapiens Neurokinin 2 receptor Ki nan None None
Homo sapiens Neuronal acetylcholine receptor protein alpha-4 subunit AC50 21999.9 nM 10.1038/s41467-023-40064-9
Homo sapiens Neuropeptide Y receptor type 1 AC50 22539.8 nM 10.1038/s41467-023-40064-9
Homo sapiens Neuropeptide Y receptor type 1 IC50 nan None None
Homo sapiens Neuropeptide Y receptor type 1 Ki nan None None
Homo sapiens Neuropeptide Y receptor type 2 AC50 21579.9 nM 10.1038/s41467-023-40064-9
Homo sapiens Neuropeptide Y receptor type 2 IC50 nan None None
Homo sapiens Neuropeptide Y receptor type 2 Ki nan None None
Homo sapiens Neurotensin receptor 1 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Nitric oxide synthase, inducible Activity nan None 10.1128/aac.00961-08
Homo sapiens Norepinephrine transporter AC50 20000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Norepinephrine transporter IC50 nan None None
Homo sapiens Norepinephrine transporter Ki nan None None
Homo sapiens Nuclear factor erythroid 2-related factor 2 Potency 4109.5 nM None
Homo sapiens Nuclear factor erythroid 2-related factor 2 Potency 4610.9 nM None
Homo sapiens Nuclear receptor subfamily 1 group I member 3 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Nuclear receptor subfamily 1 group I member 3 Activity nan None 10.1016/j.ejmech.2019.06.031
Homo sapiens PANC-1 GI50 100.0 ug.mL-1 10.1016/j.bmcl.2019.03.020
Homo sapiens PANC-1 GI50 100.0 ug.mL-1 10.1016/j.ejmech.2017.03.065
Homo sapiens PANC-1 GI90 100.0 ug ml-1 10.1016/j.bmcl.2019.03.020
Homo sapiens PANC-1 GI90 100.0 ug ml-1 10.1016/j.ejmech.2017.03.065
Homo sapiens Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 Potency 50118.7 nM None
Homo sapiens Peroxisome proliferator-activated receptor alpha AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens P-glycoprotein 1 Activity nan None 10.1016/0006-2952(95)00045-2
Homo sapiens P-glycoprotein 1 Activity nan None 10.1023/b:pham.0000026434.82855.69
Homo sapiens P-glycoprotein 1 Activity nan None 10.1074/jbc.m010173200
Homo sapiens P-glycoprotein 1 Activity nan None 10.1172/jci6663
Homo sapiens P-glycoprotein 1 Activity nan None None
Homo sapiens Phosphodiesterase 3A AC50 18330.3 nM 10.1038/s41467-023-40064-9
Homo sapiens Phosphodiesterase 4D AC50 12999.9 nM 10.1038/s41467-023-40064-9
Homo sapiens Phosphodiesterase 5A IC50 nan None None
Homo sapiens Phosphodiesterase 5A Ki nan None None
Homo sapiens Plasma Cmax 21872.53 nM 10.1128/aac.01145-08
Homo sapiens Plasma Drug uptake 0.001 ug ml-1 10.1126/science.1106753
Homo sapiens Plasma fCmax 2.43 uM 10.1124/dmd.111.040758
Homo sapiens Plasma Fu 0.15 None 10.1128/aac.01145-08
Homo sapiens Plasma Fu 0.165 None 10.1021/acs.jmedchem.5b00050
Homo sapiens Plasma K(p,uu,CSF) 2.2 None 10.1021/jm901036q
Homo sapiens Plasma PPB 85.0 % 10.1128/aac.00749-08
Homo sapiens Platelet activating factor receptor IC50 nan None None
Homo sapiens Platelet activating factor receptor Ki nan None None
Homo sapiens Pregnane X receptor AC50 19899.6 nM 10.1038/s41467-023-40064-9
Homo sapiens Pregnane X receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Pregnane X receptor Activity 70.0 % 10.1021/acs.jmedchem.9b01032
Homo sapiens Pregnane X receptor Activity 77.3 % 10.1039/C6MD00300A
Homo sapiens Pregnane X receptor Activity 100.0 % 10.1021/acs.jmedchem.0c02201
Homo sapiens Pregnane X receptor Activity 100.0 % 10.1021/acs.jmedchem.2c01640
Homo sapiens Pregnane X receptor Activity 107.0 % 10.1016/j.bmcl.2008.06.018
Homo sapiens Pregnane X receptor Activity 114.0 % 10.1021/acs.jmedchem.0c02245
Homo sapiens Pregnane X receptor Activity nan None 10.1016/j.bmc.2014.11.043
Homo sapiens Pregnane X receptor Activity nan None 10.1021/acs.jmedchem.6b00415
Homo sapiens Pregnane X receptor Activity nan None 10.1021/acsmedchemlett.1c00277
Homo sapiens Pregnane X receptor Activity nan None 10.1021/acsmedchemlett.9b00079
Homo sapiens Pregnane X receptor Activity nan None 10.1021/jm200025f
Homo sapiens Pregnane X receptor Activity nan None None
Homo sapiens Pregnane X receptor EC50 190.0 nM 10.1021/acs.jmedchem.5b01891
Homo sapiens Pregnane X receptor EC50 200.0 nM 10.1124/dmd.110.035105
Homo sapiens Pregnane X receptor EC50 226.0 nM 10.1039/C6MD00300A
Homo sapiens Pregnane X receptor EC50 1100.0 nM 10.1016/j.bmcl.2016.02.031
Homo sapiens Pregnane X receptor EC50 1170.0 nM 10.1021/acs.jmedchem.2c01640
Homo sapiens Pregnane X receptor EC50 1190.0 nM 10.1021/acs.jmedchem.0c02245
Homo sapiens Pregnane X receptor EC50 1400.0 nM 10.1021/acs.jmedchem.0c02201
Homo sapiens Pregnane X receptor EC50 2000.0 nM 10.1016/j.bmc.2018.07.038
Homo sapiens Pregnane X receptor EC50 2300.0 nM 10.1021/jm201716n
Homo sapiens Pregnane X receptor EC50 3200.0 nM 10.1124/dmd.110.035105
Homo sapiens Pregnane X receptor EC50 3500.0 nM 10.1124/dmd.110.035105
Homo sapiens Pregnane X receptor EC50 5600.0 nM 10.1016/j.bmcl.2011.08.054
Homo sapiens Pregnane X receptor Efficacy 43.9 % 10.1124/dmd.110.035105
Homo sapiens Pregnane X receptor Efficacy 75.0 % 10.1016/j.bmcl.2016.02.031
Homo sapiens Pregnane X receptor FC 2.9 None 10.1021/acsmedchemlett.1c00277
Homo sapiens Pregnane X receptor FC 9.5 None 10.1016/j.bmcl.2011.08.054
Homo sapiens Pregnane X receptor FC 11.0 None 10.1124/dmd.111.042879
Homo sapiens Pregnane X receptor FC 12.0 None 10.1124/dmd.111.042879
Homo sapiens Pregnane X receptor FC 12.6 None 10.1021/jm201716n
Homo sapiens Pregnane X receptor FC 38.0 None 10.1124/dmd.111.042879
Homo sapiens Pregnane X receptor FC 43.0 None 10.1124/dmd.111.042879
Homo sapiens Pregnane X receptor FC 50.0 None 10.1124/dmd.111.042879
Homo sapiens Pregnane X receptor FC 53.0 None 10.1124/dmd.111.042879
Homo sapiens Pregnane X receptor IC50 nan None 10.1021/acs.jmedchem.0c02201
Homo sapiens Pregnane X receptor Imax 117.0 % 10.1021/acs.jmedchem.5b01891
Homo sapiens Pregnane X receptor Inhibition 18.0 % 10.1016/j.bmcl.2008.06.018
Homo sapiens Pregnane X receptor Inhibition nan % 10.1021/acs.jmedchem.2c01640
Homo sapiens Progesterone receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Protein kinase C alpha IC50 nan None None
Homo sapiens Protein kinase C alpha Ki nan None None
Homo sapiens Receptor protein-tyrosine kinase erbB-2 IC50 nan None None
Homo sapiens Receptor protein-tyrosine kinase erbB-2 Ki nan None None
Homo sapiens Retinoic acid receptor alpha AC50 3000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Retinoic acid receptor alpha AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Retinoic acid receptor beta AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Retinoic acid receptor beta AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Retinoic acid receptor gamma AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform IC50 nan None None
Homo sapiens Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform Ki nan None None
Homo sapiens Serotonin 1a (5-HT1a) receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 1a (5-HT1a) receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2a (5-HT2a) receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2a (5-HT2a) receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2a (5-HT2a) receptor IC50 nan None None
Homo sapiens Serotonin 2a (5-HT2a) receptor Ki nan None None
Homo sapiens Serotonin 2b (5-HT2b) receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2b (5-HT2b) receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2b (5-HT2b) receptor IC50 nan None None
Homo sapiens Serotonin 2b (5-HT2b) receptor Ki nan None None
Homo sapiens Serotonin 2c (5-HT2c) receptor AC50 12000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2c (5-HT2c) receptor IC50 nan None None
Homo sapiens Serotonin 2c (5-HT2c) receptor Ki nan None None
Homo sapiens Serotonin 3a (5-HT3a) receptor AC50 5200.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 6 (5-HT6) receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 6 (5-HT6) receptor IC50 nan None None
Homo sapiens Serotonin 6 (5-HT6) receptor Ki nan None None
Homo sapiens Serotonin 7 (5-HT7) receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin transporter AC50 15000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin transporter IC50 nan None None
Homo sapiens Serotonin transporter Ki nan None None
Homo sapiens Serum Activity 80.0 % 10.1128/aac.01605-07
Homo sapiens Serum Cmax 2430.28 nM 10.1128/aac.00922-07
Homo sapiens Serum Cmax 18227.11 nM 10.1128/aac.00961-08
Homo sapiens Serum Drug uptake 5.3 mg/L 10.1128/aac.01081-09
Homo sapiens Serum Drug uptake 8.9 mg/L 10.1128/aac.01081-09
Homo sapiens Serum T1/2 2.0 hr 10.1128/aac.00922-07
Homo sapiens Serum Tmax 1.2 hr 10.1128/aac.00922-07
Homo sapiens Serum albumin Binding 73.3 % 10.1021/jm991174y
Homo sapiens Serum albumin Kd 12000.0 nM 10.1128/aac.00971-08
Homo sapiens Serum albumin Ratio 0.5 None 10.1128/aac.00971-08
Homo sapiens Serum albumin Ratio 1.0 None 10.1128/aac.00971-08
Homo sapiens Serum albumin Ratio 1.5 None 10.1128/aac.00971-08
Homo sapiens Sigma opioid receptor IC50 nan None None
Homo sapiens Sigma opioid receptor Ki nan None None
Homo sapiens Solute carrier family 22 member 1 Inhibition 26.2 % 10.1021/jm8003152
Homo sapiens Solute carrier organic anion transporter family member 1A2 Activity nan None 10.1038/nrd3028
Homo sapiens Solute carrier organic anion transporter family member 1A2 Activity nan None 10.1053/jhep.2002.34133
Homo sapiens Solute carrier organic anion transporter family member 1A2 Ki 51000.0 nM 10.1053/jhep.2002.34133
Homo sapiens Solute carrier organic anion transporter family member 1B1 Activity nan None 10.1038/nrd3028
Homo sapiens Solute carrier organic anion transporter family member 1B1 Activity nan None 10.1074/jbc.m004968200
Homo sapiens Solute carrier organic anion transporter family member 1B1 Activity nan None 10.1124/jpet.102.043026
Homo sapiens Solute carrier organic anion transporter family member 1B1 IC50 300.0 nM 10.1124/dmd.111.042382
Homo sapiens Solute carrier organic anion transporter family member 1B1 IC50 1200.0 nM 10.1021/jm300212s
Homo sapiens Solute carrier organic anion transporter family member 1B1 IC50 2200.0 nM 10.1124/dmd.111.042382
Homo sapiens Solute carrier organic anion transporter family member 1B1 IC50 2300.0 nM 10.1124/dmd.111.042382
Homo sapiens Solute carrier organic anion transporter family member 1B1 Inhibition 33.63 % 10.1124/mol.112.084152
Homo sapiens Solute carrier organic anion transporter family member 1B1 Inhibition 88.3 % 10.1021/jm300212s
Homo sapiens Solute carrier organic anion transporter family member 1B1 Inhibition 98.4 % 10.1124/dmd.112.048470
Homo sapiens Solute carrier organic anion transporter family member 1B1 Ki 1100.0 nM 10.1021/jm300212s
Homo sapiens Solute carrier organic anion transporter family member 1B1 Ki 17000.0 nM 10.1053/jhep.2002.34133
Homo sapiens Solute carrier organic anion transporter family member 1B1 Km 1500.0 nM 10.1124/jpet.102.043026
Homo sapiens Solute carrier organic anion transporter family member 1B1 Km 13000.0 nM 10.1053/jhep.2002.34133
Homo sapiens Solute carrier organic anion transporter family member 1B3 Activity nan None 10.1038/nrd3028
Homo sapiens Solute carrier organic anion transporter family member 1B3 Activity nan None 10.1074/jbc.m004968200
Homo sapiens Solute carrier organic anion transporter family member 1B3 IC50 1500.0 nM 10.1021/jm300212s
Homo sapiens Solute carrier organic anion transporter family member 1B3 Inhibition 22.01 % 10.1124/mol.112.084152
Homo sapiens Solute carrier organic anion transporter family member 1B3 Inhibition 97.4 % 10.1124/dmd.112.048470
Homo sapiens Solute carrier organic anion transporter family member 1B3 Inhibition 101.7 % 10.1021/jm300212s
Homo sapiens Solute carrier organic anion transporter family member 1B3 Ki 1400.0 nM 10.1021/jm300212s
Homo sapiens Solute carrier organic anion transporter family member 1B3 Ki 5000.0 nM 10.1053/jhep.2002.34133
Homo sapiens Solute carrier organic anion transporter family member 1B3 Km 2300.0 nM 10.1053/jhep.2002.34133
Homo sapiens Solute carrier organic anion transporter family member 2B1 Activity nan None 10.1038/nrd3028
Homo sapiens Solute carrier organic anion transporter family member 2B1 Activity nan None 10.1053/jhep.2002.34133
Homo sapiens Solute carrier organic anion transporter family member 2B1 IC50 65000.0 nM 10.1021/jm300212s
Homo sapiens Solute carrier organic anion transporter family member 2B1 Inhibition 21.2 % 10.1021/jm300212s
Homo sapiens Solute carrier organic anion transporter family member 2B1 Ki 63000.0 nM 10.1021/jm300212s
Homo sapiens TAR DNA-binding protein 43 Potency 501.2 nM None
Homo sapiens Thiosulfate sulfurtransferase IC50 100000.0 nM 10.1021/acs.jmedchem.8b01293
Homo sapiens THP-1 Activity 65.0 ug ml-1 10.1016/j.bmcl.2009.09.095
Homo sapiens THP-1 GI50 0.14 ug.mL-1 10.1016/j.ejmech.2017.01.009
Homo sapiens THP-1 IC50 100000.0 nM 10.1021/acs.jnatprod.5b00266
Homo sapiens THP-1 IC90 100000.0 nM 10.1021/acs.jnatprod.5b00266
Homo sapiens Thromboxane A2 receptor AC50 17364.6 nM 10.1038/s41467-023-40064-9
Homo sapiens Thromboxane-A synthase IC50 nan None None
Homo sapiens Thromboxane-A synthase Ki nan None None
Homo sapiens Type-1 angiotensin II receptor AC50 19395.9 nM 10.1038/s41467-023-40064-9
Homo sapiens Tyrosine-protein kinase FYN IC50 nan None None
Homo sapiens Tyrosine-protein kinase FYN Ki nan None None
Homo sapiens Tyrosine-protein kinase LCK IC50 nan None None
Homo sapiens Tyrosine-protein kinase LCK Ki nan None None
Homo sapiens Tyrosyl-DNA phosphodiesterase 1 Potency 5173.5 nM None
Homo sapiens Tyrosyl-DNA phosphodiesterase 1 Potency 18837.5 nM None
Homo sapiens Tyrosyl-DNA phosphodiesterase 1 Potency 23715.0 nM None
Homo sapiens UDP-glucuronosyltransferase 1-1 Activity 0.0 pm/min/mg 10.1146/annurev.pharmtox.40.1.581
Homo sapiens UDP-glucuronosyltransferase 1-6 Activity 0.0 pm/min/mg 10.1146/annurev.pharmtox.40.1.581
Homo sapiens UDP-glucuronosyltransferase 1-9 Activity 0.0 pm/min/mg 10.1146/annurev.pharmtox.40.1.581
Homo sapiens Vascular endothelial growth factor receptor 1 IC50 nan None None
Homo sapiens Vascular endothelial growth factor receptor 1 Ki nan None None
Homo sapiens Vasoactive intestinal polypeptide receptor 1 IC50 nan None None
Homo sapiens Vasoactive intestinal polypeptide receptor 1 Ki nan None None
Homo sapiens Vasopressin V1a receptor AC50 26699.9 nM 10.1038/s41467-023-40064-9
Homo sapiens Vasopressin V1a receptor IC50 nan None None
Homo sapiens Vasopressin V1a receptor Ki nan None None
Homo sapiens Vasopressin V2 receptor AC50 29999.9 nM 10.1038/s41467-023-40064-9
Klebsiella aerogenes Klebsiella aerogenes Inhibition 100.0 % 10.1021/jm0703901
Klebsiella aerogenes Klebsiella aerogenes MIC 100.0 ug.mL-1 10.1021/jm0703901
Klebsiella aerogenes Klebsiella aerogenes MIC 8000.0 nM 10.1021/acs.jmedchem.1c02122
Klebsiella oxytoca Klebsiella oxytoca MBC nan None 10.1021/acs.jnatprod.2c00065
Klebsiella oxytoca Klebsiella oxytoca MIC 0.012 ug.mL-1 10.1128/aac.00405-08
Klebsiella oxytoca Klebsiella oxytoca MIC 0.032 ug.mL-1 10.1128/aac.00405-08
Klebsiella oxytoca Klebsiella oxytoca MIC 4.0 ug.mL-1 10.1021/acs.jnatprod.2c00065
Klebsiella oxytoca Klebsiella oxytoca Ratio 680.0 None 10.1128/aac.00405-08
Klebsiella oxytoca Klebsiella oxytoca Ratio 700.0 None 10.1128/aac.00405-08
Klebsiella pneumoniae Klebsiella pneumoniae EC50 11000.0 nM 10.1021/acs.jmedchem.8b01293
Klebsiella pneumoniae Klebsiella pneumoniae FICI 0.125 None 10.1128/aac.01439-09
Klebsiella pneumoniae Klebsiella pneumoniae Inhibition 10.0 % 10.1128/aac.00471-08
Klebsiella pneumoniae Klebsiella pneumoniae Inhibition nan % 10.1128/aac.00471-08
Klebsiella pneumoniae Klebsiella pneumoniae IZ 7.0 mm 10.1016/j.bmc.2018.02.049
Klebsiella pneumoniae Klebsiella pneumoniae IZ 27.0 mm 10.1016/j.bmcl.2016.04.038
Klebsiella pneumoniae Klebsiella pneumoniae IZ 45.0 mm 10.1016/j.ejmech.2008.09.035
Klebsiella pneumoniae Klebsiella pneumoniae IZ nan None 10.1016/j.bmc.2007.09.025
Klebsiella pneumoniae Klebsiella pneumoniae log10cfu 8.5 None 10.1128/aac.00471-08
Klebsiella pneumoniae Klebsiella pneumoniae MBC 3.13 ug ml-1 10.1016/j.bmc.2018.07.034
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.016 ug.mL-1 10.1128/aac.00471-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.064 ug.mL-1 10.1128/aac.00405-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.073 ug.mL-1 10.1128/aac.00405-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.19 ug.mL-1 10.1128/aac.00405-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.25 ug.mL-1 10.1016/j.bmc.2018.02.049
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.25 ug.mL-1 10.1016/j.ejmech.2008.09.035
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.25 ug.mL-1 10.1128/aac.00405-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 0.5 ug.mL-1 10.1128/aac.01439-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.0 ug.mL-1 10.1128/aac.01439-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.5 ug.mL-1 10.1128/aac.00405-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1.9 ug.mL-1 10.1016/j.ejmech.2007.12.019
Klebsiella pneumoniae Klebsiella pneumoniae MIC 2.0 ug.mL-1 10.1128/aac.00405-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 6.0 ug.mL-1 10.1128/aac.00017-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 7.8 ug.mL-1 10.1016/j.ejmech.2007.12.019
Klebsiella pneumoniae Klebsiella pneumoniae MIC 8.0 ug.mL-1 10.1128/aac.00017-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 12.0 ug.mL-1 10.1128/aac.01439-09
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1016/j.ejmech.2008.04.001
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1021/jm00167a029
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.00405-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16.0 ug.mL-1 10.1128/aac.01053-06
Klebsiella pneumoniae Klebsiella pneumoniae MIC 22.0 ug.mL-1 10.1016/j.bmcl.2017.05.032
Klebsiella pneumoniae Klebsiella pneumoniae MIC 25.0 ug.mL-1 10.1021/acs.jnatprod.0c01212
Klebsiella pneumoniae Klebsiella pneumoniae MIC 25.0 ug.mL-1 10.1021/jm00143a010
Klebsiella pneumoniae Klebsiella pneumoniae MIC 25.0 ug.mL-1 10.1021/jm00145a020
Klebsiella pneumoniae Klebsiella pneumoniae MIC 25.0 ug.mL-1 10.1021/jm00220a012
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1021/acs.jmedchem.8b01287
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.00017-08
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32.0 ug.mL-1 10.1128/aac.01247-10
Klebsiella pneumoniae Klebsiella pneumoniae MIC 64.0 ug.mL-1 10.1016/j.ejmech.2022.114360
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1016/j.bmc.2006.12.035
Klebsiella pneumoniae Klebsiella pneumoniae MIC 256.0 ug.mL-1 10.1016/j.ejmech.2008.04.001
Klebsiella pneumoniae Klebsiella pneumoniae MIC 1024.0 ug.mL-1 10.1021/acs.jmedchem.6b01742
Klebsiella pneumoniae Klebsiella pneumoniae MIC 4096.0 ug.mL-1 10.1016/j.bmc.2006.12.035
Klebsiella pneumoniae Klebsiella pneumoniae MIC 16000.0 nM 10.1021/acs.jmedchem.1c02122
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32000.0 nM 10.1016/j.ejmech.2019.111636
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32000.0 nM 10.1021/acs.jmedchem.1c00614
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32000.0 nM 10.1021/acs.jmedchem.1c02140
Klebsiella pneumoniae Klebsiella pneumoniae MIC 32000.0 nM 10.1021/acs.jmedchem.2c01076
Klebsiella pneumoniae Klebsiella pneumoniae MIC nan None 10.1016/j.bmc.2019.04.032
Klebsiella pneumoniae Klebsiella pneumoniae MIC nan None 10.1016/j.ejmech.2019.04.067
Klebsiella pneumoniae Klebsiella pneumoniae MIC100 1.56 ug ml-1 10.1016/j.bmc.2018.07.034
Klebsiella pneumoniae Klebsiella pneumoniae Ratio 10.0 None 10.1128/aac.00405-08
Klebsiella pneumoniae Klebsiella pneumoniae Ratio 24.0 None 10.1128/aac.01439-09
Klebsiella pneumoniae Klebsiella pneumoniae Ratio 43.0 None 10.1128/aac.00405-08
Klebsiella pneumoniae Klebsiella pneumoniae Ratio 250.0 None 10.1128/aac.00405-08
Klebsiella pneumoniae subsp. pneumoniae Klebsiella pneumoniae subsp. pneumoniae EC50 5400.0 nM 10.1016/j.bmcl.2016.04.089
Leishmania donovani Leishmania donovani IC50 nan None 10.1021/np020592u
Leishmania donovani Leishmania donovani IC50 nan None 10.1021/np0400095
Leishmania donovani Leishmania donovani IC50 nan None 10.1021/np0601399
Leishmania donovani Leishmania donovani IC90 nan None 10.1021/np020592u
Leishmania donovani Leishmania donovani IC90 nan None 10.1021/np0400095
Leishmania donovani Leishmania donovani IC90 nan None 10.1021/np0601399
Listeria monocytogenes Listeria monocytogenes Inhibition 100.0 % 10.1021/jm0703901
Listeria monocytogenes Listeria monocytogenes MIC nan None 10.1016/j.bmc.2019.04.032
Macaca fascicularis Brain Fu 0.162 None 10.1124/dmd.111.038778
Mammaliicoccus sciuri Mammaliicoccus sciuri Activity 0.0 % 10.1128/aac.00426-10
Mammaliicoccus sciuri Mammaliicoccus sciuri Activity 11.1 % 10.1128/aac.00426-10
Mammaliicoccus sciuri Mammaliicoccus sciuri Activity 15.4 % 10.1128/aac.00426-10
Micrococcus luteus Micrococcus luteus IZ 49.0 mm 10.1016/j.bmc.2007.09.025
Micrococcus luteus Micrococcus luteus MIC 0.125 ug.mL-1 10.1021/ml300350p
Mobiluncus curtisii subsp. curtisii Mobiluncus curtisii subsp. curtisii MIC 0.004 ug.mL-1 10.1021/acs.jmedchem.1c02045
Morganella morganii Morganella morganii MIC 10.0 ug.mL-1 10.1021/acs.jnatprod.2c00174
Morganella morganii Morganella morganii MIC nan None 10.1016/j.bmcl.2012.08.003
Mus musculus Brain Drug uptake 10.25 ug ml-1 10.1021/jm901858n
Mus musculus Brain Fu 0.121 None 10.1124/dmd.111.038778
Mus musculus Canalicular multispecific organic anion transporter 2 Activity nan None 10.1124/dmd.31.11.1296
Mus musculus Integrin alpha M MIC 2.0 ug.mL-1 10.1021/jm00167a029
Mus musculus Integrin alpha M MIC 64.0 ug.mL-1 10.1021/jm00167a029
Mus musculus J774 Activity 73.0 % 10.1016/j.bmc.2016.01.028
Mus musculus J774 Activity 78.0 % 10.1016/j.ejmech.2013.12.013
Mus musculus J774 Activity 80.0 % 10.1016/j.bmcl.2016.03.066
Mus musculus J774 Activity 82.0 % 10.1016/j.ejmech.2013.12.013
Mus musculus J774 Activity 85.0 % 10.1016/j.bmc.2016.01.028
Mus musculus J774 Activity 86.0 % 10.1016/j.ejmech.2013.12.013
Mus musculus J774 Activity 87.0 % 10.1016/j.bmcl.2016.03.066
Mus musculus J774 Activity 93.0 % 10.1016/j.bmcl.2016.03.066
Mus musculus J774 Activity 95.0 % 10.1016/j.bmc.2016.01.028
Mus musculus J774.A1 Activity 1.03 deltalog10CFU 10.1016/j.ejmech.2022.114145
Mus musculus J774.A1 Activity 90.0 % 10.1128/aac.00375-07
Mus musculus J774.A1 Activity 94.4 None 10.1128/aac.00375-07
Mus musculus J774.A1 CC50 207.03 ug.mL-1 10.1016/j.bmc.2010.09.006
Mus musculus J774.A1 IC50 64.0 ug.mL-1 10.1016/j.bmc.2022.117006
Mus musculus J774.A1 IC50 nan None 10.1016/j.bmc.2019.07.045
Mus musculus J774.A1 IC50 nan None 10.1016/j.bmcl.2019.02.019
Mus musculus Mus musculus Activity 85.0 % 10.1021/np50025a010
Mus musculus Mus musculus Activity 174.0 % 10.1021/np50025a010
Mus musculus Mus musculus AUC 24760.0 ng.hr.mL-1 10.1128/aac.00367-09
Mus musculus Mus musculus AUC 48200.0 ng.hr.mL-1 10.1371/journal.pmed.0030466
Mus musculus Mus musculus Cmax 6197.22 nM 10.1371/journal.pmed.0030466
Mus musculus Mus musculus Cmax 19138.47 nM 10.1128/aac.00367-09
Mus musculus Mus musculus Cp 0.66 ug ml-1 10.1371/journal.pmed.0030466
Mus musculus Mus musculus Cp 3.18 ug ml-1 10.1371/journal.pmed.0030466
Mus musculus Mus musculus Cp 3.33 ug ml-1 10.1371/journal.pmed.0030466
Mus musculus Mus musculus Cp 3.82 ug ml-1 10.1371/journal.pmed.0030466
Mus musculus Mus musculus Cp 4.49 ug ml-1 10.1371/journal.pmed.0030466
Mus musculus Mus musculus Cp 4.52 ug ml-1 10.1371/journal.pmed.0030466
Mus musculus Mus musculus Cp 5.1 ug ml-1 10.1371/journal.pmed.0030466
Mus musculus Mus musculus EC90 0.007 None 10.1016/s0960-894x(01)00283-9
Mus musculus Mus musculus EC99 0.451 None 10.1016/s0960-894x(01)00283-9
Mus musculus Mus musculus FC 1.3 None 10.1124/dmd.112.048009
Mus musculus Mus musculus FC 1.5 None 10.1124/dmd.112.048009
Mus musculus Mus musculus FC 1.8 None 10.1124/dmd.112.048009
Mus musculus Mus musculus FC 1.9 None 10.1124/dmd.112.048009
Mus musculus Mus musculus FC 2.0 None 10.1124/dmd.112.048009
Mus musculus Mus musculus FC 2.1 None 10.1124/dmd.112.048009
Mus musculus Mus musculus FC 2.5 None 10.1124/dmd.112.048009
Mus musculus Mus musculus FC 2.7 None 10.1124/dmd.112.048009
Mus musculus Mus musculus FC 3.7 None 10.1124/dmd.112.048009
Mus musculus Mus musculus FC 4.5 None 10.1124/dmd.112.048009
Mus musculus Mus musculus FC 8.4 None 10.1124/dmd.112.048009
Mus musculus Mus musculus FC 16.5 None 10.1124/dmd.112.048009
Mus musculus Mus musculus FC 171.9 None 10.1124/dmd.112.048009
Mus musculus Mus musculus IC50 nan None 10.1016/j.ejmech.2016.07.039
Mus musculus Mus musculus Inhibition 9.56 % 10.1016/j.bmc.2016.09.012
Mus musculus Mus musculus Inhibition nan % 10.1016/j.ejmech.2016.08.034
Mus musculus Mus musculus T1/2 2.86 hr 10.1128/aac.00367-09
Mus musculus Mus musculus T1/2 3.4 hr 10.1371/journal.pmed.0030466
Mus musculus Mus musculus Tmax 6.0 hr 10.1371/journal.pmed.0030466
Mus musculus NIH3T3 Survival 62.0 % 10.1021/acs.jnatprod.5b01033
Mus musculus Nitric oxide synthase, inducible IC50 nan None None
Mus musculus Nitric oxide synthase, inducible Ki nan None None
Mus musculus Nuclear receptor subfamily 1 group I member 2 FC 1.6 None 10.1124/dmd.112.048009
Mus musculus Nuclear receptor subfamily 1 group I member 2 FC 1.7 None 10.1124/dmd.112.048009
Mus musculus RAW264.7 Activity nan None 10.1016/j.ejmech.2017.12.088
Mus musculus RAW264.7 CC50 80.39 ug.mL-1 10.1016/j.ejmech.2021.113472
Mus musculus RAW264.7 CC50 24000.0 nM 10.1016/j.ejmech.2020.112908
Mus musculus RAW264.7 GI 23.48 % 10.1016/j.bmc.2017.03.053
Mus musculus RAW264.7 GI nan None 10.1016/j.bmc.2015.03.004
Mus musculus RAW264.7 GI nan None 10.1016/j.bmc.2017.11.031
Mus musculus RAW264.7 GI nan None 10.1016/j.ejmech.2018.07.046
Mus musculus RAW264.7 GI50 700.0 ug.mL-1 10.1016/j.bmc.2015.04.001
Mus musculus RAW264.7 GI50 850000.0 nM 10.1039/C3MD00251A
Mus musculus RAW264.7 GI50 nan None 10.1016/j.ejmech.2018.07.046
Mus musculus RAW264.7 IC50 nan None 10.1016/j.ejmech.2022.114831
Mus musculus RAW264.7 Inhibition nan % 10.1016/j.bmc.2014.10.016
Mus musculus RAW264.7 Inhibition nan % 10.1016/j.bmc.2015.02.032
Mus musculus RAW264.7 Inhibition nan % 10.1016/j.bmc.2016.01.011
Mus musculus RAW264.7 Inhibition nan % 10.1016/j.ejmech.2014.09.028
Mus musculus RAW264.7 Inhibition nan % 10.1016/j.ejmech.2014.12.046
Mus musculus RAW264.7 Inhibition nan % 10.1016/j.ejmech.2015.06.032
Mycobacterium avium Mycobacterium avium Activity 0.0 % 10.1016/j.bmcl.2006.08.090
Mycobacterium avium Mycobacterium avium GI 90.0 % 10.1016/j.bmc.2012.05.004
Mycobacterium avium Mycobacterium avium GI 90.0 % 10.1016/j.bmc.2016.09.008
Mycobacterium avium Mycobacterium avium GI 90.0 % 10.1016/j.bmcl.2011.11.114
Mycobacterium avium Mycobacterium avium Inhibition 90.0 % 10.1016/j.bmc.2006.12.032
Mycobacterium avium Mycobacterium avium Inhibition 90.0 % 10.1021/jm058167w
Mycobacterium avium Mycobacterium avium Inhibition 90.0 % 10.1021/jm0703901
Mycobacterium avium Mycobacterium avium Inhibition 90.0 % 10.1021/jm070391t
Mycobacterium avium Mycobacterium avium Inhibition 100.0 % 10.1016/j.bmc.2006.12.032
Mycobacterium avium Mycobacterium avium MIC 0.004 ug.mL-1 10.1016/j.bmcl.2007.02.024
Mycobacterium avium Mycobacterium avium MIC 0.004 ug.mL-1 10.1016/j.bmcl.2009.09.095
Mycobacterium avium Mycobacterium avium MIC 0.05 ug.mL-1 10.1016/j.bmcl.2009.09.095
Mycobacterium avium Mycobacterium avium MIC 0.05 ug.mL-1 10.1016/j.bmcl.2010.12.084
Mycobacterium avium Mycobacterium avium MIC 0.125 ug.mL-1 10.1016/s0960-894x(03)00596-1
Mycobacterium avium Mycobacterium avium MIC 0.125 ug.mL-1 10.1016/s0960-894x(03)00597-3
Mycobacterium avium Mycobacterium avium MIC 0.15 ug.mL-1 10.1128/aac.00749-08
Mycobacterium avium Mycobacterium avium MIC 0.25 ug.mL-1 10.1016/j.ejmech.2009.06.005
Mycobacterium avium Mycobacterium avium MIC 0.25 ug.mL-1 10.1021/jm701560p
Mycobacterium avium Mycobacterium avium MIC 0.25 ug.mL-1 10.1128/aac.01545-09
Mycobacterium avium Mycobacterium avium MIC 0.3 ug.mL-1 10.1016/s0960-894x(99)00510-7
Mycobacterium avium Mycobacterium avium MIC 0.3 ug.mL-1 10.1021/jm0602662
Mycobacterium avium Mycobacterium avium MIC 0.78 ug.mL-1 10.1039/C8MD00056E
Mycobacterium avium Mycobacterium avium MIC 2.0 ug.mL-1 10.1016/j.bmc.2013.10.011
Mycobacterium avium Mycobacterium avium MIC 3.1 ug.mL-1 10.1021/jm070638m
Mycobacterium avium Mycobacterium avium MIC 4.0 ug.mL-1 10.1021/acs.jmedchem.2c00972
Mycobacterium avium Mycobacterium avium MIC 90.0 ug.mL-1 10.1016/j.ejmech.2017.11.083
Mycobacterium avium Mycobacterium avium MIC 100.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium avium Mycobacterium avium MIC 780.0 nM 10.1016/j.bmcl.2014.05.062
Mycobacterium avium Mycobacterium avium MIC 16000.0 nM 10.1016/j.ejmech.2010.02.037
Mycobacterium avium Mycobacterium avium MIC 65000.0 nM 10.1016/j.ejmech.2010.02.037
Mycobacterium avium Mycobacterium avium MIC nan ug.mL-1 10.1016/s0960-894x(00)00159-1
Mycobacterium avium Mycobacterium avium MIC nan None 10.1016/j.bmc.2010.05.016
Mycobacterium avium Mycobacterium avium MIC50 16.0 ug.mL-1 10.1021/jm00167a029
Mycobacterium avium Mycobacterium avium MIC50 32.0 ug.mL-1 10.1128/aac.01545-09
Mycobacterium avium Mycobacterium avium MIC90 2.0 ug.mL-1 10.1016/j.bmc.2016.03.003
Mycobacterium avium Mycobacterium avium MIC90 2.0 ug.mL-1 10.1021/jm058167w
Mycobacterium avium Mycobacterium avium MIC90 2.0 ug.mL-1 10.1021/jm0703901
Mycobacterium avium Mycobacterium avium MIC90 2.0 ug.mL-1 10.1021/jm070391t
Mycobacterium avium Mycobacterium avium MIC90 128.0 ug.mL-1 10.1128/aac.01545-09
Mycobacterium avium Mycobacterium avium MIC90 780.0 nM 10.1021/ml200036r
Mycobacterium avium Mycobacterium avium MIC>99 32.0 uM 10.1016/j.bmc.2017.08.010
Mycobacterium avium Mycobacterium avium MIC>99 32.0 uM 10.1016/j.ejmech.2017.02.058
Mycobacterium avium Mycobacterium avium MIC>99 32.0 uM 10.1021/acs.jmedchem.9b00912
Mycobacterium avium Mycobacterium avium MIC>99 62.0 uM 10.1021/acs.jmedchem.9b00912
Mycobacterium avium complex sp. Mycobacterium avium complex sp. MIC 30.0 ug.mL-1 10.1016/j.ejmech.2017.11.083
Mycobacterium avium complex sp. Mycobacterium avium complex sp. MIC=>90 10.0 uM 10.1016/j.bmc.2015.03.018
Mycobacterium avium complex sp. Mycobacterium avium complex sp. MIC>90 10.0 uM 10.1016/j.bmc.2015.06.047
Mycobacterium avium subsp. paratuberculosis Mycobacterium avium subsp. paratuberculosis Activity 2.0 ug ml-1 10.1128/aac.00678-07
Mycobacterium avium subsp. paratuberculosis Mycobacterium avium subsp. paratuberculosis Activity 64.0 ug ml-1 10.1128/aac.00678-07
Mycobacterium avium subsp. paratuberculosis Mycobacterium avium subsp. paratuberculosis Activity nan None 10.1128/aac.00678-07
Mycobacterium avium subsp. paratuberculosis Mycobacterium avium subsp. paratuberculosis MIC=>90 109.0 uM 10.1016/j.bmc.2015.03.018
Mycobacterium avium subsp. paratuberculosis Mycobacterium avium subsp. paratuberculosis MIC>90 109.0 uM 10.1016/j.bmc.2015.06.047
Mycobacterium gordonae Mycobacterium gordonae MIC 0.5 ug.mL-1 10.1021/jm00167a029
Mycobacterium gordonae Mycobacterium gordonae MIC 0.6 ug.mL-1 10.1016/s0960-894x(99)00510-7
Mycobacterium gordonae Mycobacterium gordonae MIC 4.0 ug.mL-1 10.1021/jm00167a029
Mycobacterium intracellulare Mycobacterium intracellulare Activity nan None 10.1021/acs.jnatprod.7b00903
Mycobacterium intracellulare Mycobacterium intracellulare IC50 nan None 10.1021/jm900672t
Mycobacterium intracellulare Mycobacterium intracellulare IC50 nan None 10.1021/np900281r
Mycobacterium intracellulare Mycobacterium intracellulare MIC 0.125 ug.mL-1 10.1016/s0960-894x(03)00596-1
Mycobacterium intracellulare Mycobacterium intracellulare MIC 0.125 ug.mL-1 10.1016/s0960-894x(03)00597-3
Mycobacterium intracellulare Mycobacterium intracellulare MIC 0.2 ug.mL-1 10.1021/jm00150a006
Mycobacterium intracellulare Mycobacterium intracellulare MIC 0.25 ug.mL-1 10.1128/aac.01545-09
Mycobacterium intracellulare Mycobacterium intracellulare MIC 0.3 ug.mL-1 10.1021/np9901940
Mycobacterium intracellulare Mycobacterium intracellulare MIC 0.5 ug.mL-1 10.1016/j.ejmech.2013.06.010
Mycobacterium intracellulare Mycobacterium intracellulare MIC 0.5 ug.mL-1 10.1016/j.ejmech.2013.12.037
Mycobacterium intracellulare Mycobacterium intracellulare MIC 0.78 ug.mL-1 10.1021/jm00100a012
Mycobacterium intracellulare Mycobacterium intracellulare MIC 1.0 ug.mL-1 10.1016/j.bmc.2013.10.011
Mycobacterium intracellulare Mycobacterium intracellulare MIC 3.1 ug.mL-1 10.1021/jm070638m
Mycobacterium intracellulare Mycobacterium intracellulare MIC nan None 10.1016/j.bmc.2010.05.016
Mycobacterium intracellulare Mycobacterium intracellulare MIC nan None 10.1021/np900281r
Mycobacterium intracellulare Mycobacterium intracellulare MIC50 2.0 ug.mL-1 10.1128/aac.01545-09
Mycobacterium intracellulare Mycobacterium intracellulare MIC90 32.0 ug.mL-1 10.1128/aac.01545-09
Mycobacterium kansasii Mycobacterium kansasii Activity 100.0 % 10.1016/j.bmcl.2006.08.090
Mycobacterium kansasii Mycobacterium kansasii MIC 0.05 ug.mL-1 10.1021/jm00150a006
Mycobacterium kansasii Mycobacterium kansasii MIC 0.06 ug.mL-1 10.1128/aac.01545-09
Mycobacterium kansasii Mycobacterium kansasii MIC 0.125 ug.mL-1 10.1021/jm00167a029
Mycobacterium kansasii Mycobacterium kansasii MIC 0.25 ug.mL-1 10.1016/s0960-894x(03)00596-1
Mycobacterium kansasii Mycobacterium kansasii MIC 0.25 ug.mL-1 10.1016/s0960-894x(03)00597-3
Mycobacterium kansasii Mycobacterium kansasii MIC 0.5 ug.mL-1 10.1016/j.bmc.2013.10.011
Mycobacterium kansasii Mycobacterium kansasii MIC 0.78 ug.mL-1 10.1039/C8MD00056E
Mycobacterium kansasii Mycobacterium kansasii MIC 8.0 ug.mL-1 10.1021/jm00167a029
Mycobacterium kansasii Mycobacterium kansasii MIC 16.0 ug.mL-1 10.1021/jm00167a029
Mycobacterium kansasii Mycobacterium kansasii MIC 30.0 nM 10.1016/j.bmcl.2014.05.062
Mycobacterium kansasii Mycobacterium kansasii MIC 100.0 nM 10.1021/ml5003458
Mycobacterium kansasii Mycobacterium kansasii MIC 125.0 nM 10.1016/j.ejmech.2010.02.037
Mycobacterium kansasii Mycobacterium kansasii MIC 250.0 nM 10.1016/j.ejmech.2010.02.037
Mycobacterium kansasii Mycobacterium kansasii MIC 7590.0 nM 10.1016/j.bmcl.2008.12.088
Mycobacterium kansasii Mycobacterium kansasii MIC nan None 10.1016/j.bmc.2010.05.016
Mycobacterium kansasii Mycobacterium kansasii MIC50 0.25 ug.mL-1 10.1128/aac.01545-09
Mycobacterium kansasii Mycobacterium kansasii MIC90 0.25 ug.mL-1 10.1128/aac.01545-09
Mycobacterium kansasii Mycobacterium kansasii MIC90 780.0 nM 10.1021/ml200036r
Mycobacterium kansasii Mycobacterium kansasii MIC>99 0.125 uM 10.1016/j.bmc.2017.08.010
Mycobacterium kansasii Mycobacterium kansasii MIC>99 0.125 uM 10.1016/j.ejmech.2017.02.058
Mycobacterium kansasii Mycobacterium kansasii MIC>99 0.125 uM 10.1021/acs.jmedchem.9b00912
Mycobacterium kansasii Mycobacterium kansasii MIC>99 0.25 uM 10.1016/j.bmc.2017.08.010
Mycobacterium kansasii Mycobacterium kansasii MIC>99 0.25 uM 10.1016/j.ejmech.2017.02.058
Mycobacterium kansasii Mycobacterium kansasii MIC>99 0.25 uM 10.1021/acs.jmedchem.9b00912
Mycobacterium leprae Mycobacterium leprae Activity 0.0 pg 10.1016/j.bmc.2019.04.032
Mycobacterium leprae Mycobacterium leprae Activity 0.0 pmol 10.1016/j.bmc.2019.04.032
Mycobacterium leprae Mycobacterium leprae Activity 0.7 pmol 10.1016/j.bmc.2019.04.032
Mycobacterium leprae Mycobacterium leprae Activity 0.73 pmol 10.1016/j.bmc.2019.04.032
Mycobacterium leprae Mycobacterium leprae Activity 211.0 pg 10.1016/j.bmc.2019.04.032
Mycobacterium leprae Mycobacterium leprae Activity 215.0 pg 10.1016/j.bmc.2019.04.032
Mycobacterium leprae Mycobacterium leprae Inhibition 86.0 % 10.1016/j.bmc.2019.04.032
Mycobacterium marinum Mycobacterium marinum Activity 1.9 deltalog10CFU/ml 10.1016/j.bmc.2016.01.059
Mycobacterium marinum Mycobacterium marinum Activity 27.0 % 10.1021/acs.jmedchem.1c02122
Mycobacterium marinum Mycobacterium marinum Activity nan None 10.1016/j.ejmech.2015.01.020
Mycobacterium marinum Mycobacterium marinum Activity nan None 10.1021/acs.jmedchem.1c01407
Mycobacterium marinum Mycobacterium marinum MIC 0.5 ug.mL-1 10.1021/jm00167a029
Mycobacterium marinum Mycobacterium marinum MIC 0.5 ug.mL-1 10.1021/jm701560p
Mycobacterium marinum Mycobacterium marinum MIC 0.6 ug.mL-1 10.1016/s0960-894x(99)00510-7
Mycobacterium marinum Mycobacterium marinum MIC 0.6 ug.mL-1 10.1021/jm0602662
Mycobacterium marinum Mycobacterium marinum MIC 1.0 ug.mL-1 10.1021/jm00167a029
Mycobacterium marinum Mycobacterium marinum MIC 2.0 ug.mL-1 10.1021/jm00167a029
Mycobacterium marinum Mycobacterium marinum MIC 230.0 nM 10.1021/ml5003458
Mycobacterium marinum Mycobacterium marinum MIC 1200.0 nM 10.1016/j.bmcl.2014.05.062
Mycobacterium marinum Mycobacterium marinum MIC90 780.0 nM 10.1021/ml200036r
Mycobacterium scrofulaceum Mycobacterium scrofulaceum MIC 0.063 ug.mL-1 10.1021/jm00167a029
Mycobacterium scrofulaceum Mycobacterium scrofulaceum MIC 0.125 ug.mL-1 10.1021/jm00167a029
Mycobacterium scrofulaceum Mycobacterium scrofulaceum MIC 0.5 ug.mL-1 10.1016/j.ejmech.2013.12.037
Mycobacterium scrofulaceum Mycobacterium scrofulaceum MIC 8.0 ug.mL-1 10.1021/jm00167a029
Mycobacterium smegmatis DNA gyrase subunit B IC50 nan None 10.1016/j.bmc.2014.10.016
Mycobacterium smegmatis DNA gyrase subunit B IC50 nan None 10.1016/j.bmc.2015.02.032
Mycobacterium smegmatis DNA gyrase subunit B IC50 nan None 10.1016/j.bmc.2015.03.004
Mycobacterium smegmatis DNA gyrase subunit B IC50 nan None 10.1016/j.ejmech.2015.06.032
Mycobacterium smegmatis DNA gyrase subunit B IC50 nan None 10.1016/j.ejmech.2016.08.034
Mycobacterium smegmatis (strain ATCC 700084 / mc(2)155) DNA gyrase subunit B IC50 nan None 10.1016/j.ejmech.2016.06.042
Mycobacterium szulgai Mycobacterium szulgai MIC 0.5 ug.mL-1 10.1016/j.ejmech.2013.12.037
Mycobacterium tuberculosis ATP-dependent Clp protease ATP-binding subunit ClpC1 Kd nan None 10.1021/acs.jnatprod.9b01095
Mycobacterium tuberculosis DNA-directed RNA polymerase beta chain IC50 10.0 nM 10.1016/j.bmcl.2011.08.054
Mycobacterium tuberculosis DNA-directed RNA polymerase beta chain logIC50 -2.399 None 10.1016/j.bmcl.2011.08.054
Mycobacterium tuberculosis Enoyl-[acyl-carrier-protein] reductase IC50 30.0 nM 10.1021/jm500833f
Mycobacterium tuberculosis Enoyl-[acyl-carrier-protein] reductase MIC 0.2 ug.mL-1 10.1016/j.ejmech.2018.07.047
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 0.5 None 10.1021/jm060957y
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 1.0 log10CFU 10.1021/acs.jmedchem.2c01493
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 1.0 log10CFU/ml 10.1021/acs.jmedchem.1c02122
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 1.03 deltalog10CFU 10.1021/acs.jmedchem.1c00263
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 1.06 deltalog10CFU 10.1016/j.bmc.2016.01.028
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 1.1 log10CFU 10.1016/j.ejmech.2021.113932
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 1.58 log10CFU 10.1021/acsmedchemlett.5b00324
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 1.76 log10CFU 10.1039/C4MD00288A
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 1.93 log10CFU 10.1039/C4MD00288A
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 2.0 log10CFU 10.1021/acs.jmedchem.0c01727
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 2.1 deltalog10CFU/ml 10.1016/j.bmc.2016.01.059
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 2.39 deltalog10CFU 10.1016/j.bmc.2016.01.028
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 2.44 log10CFU 10.1016/j.ejmech.2016.11.048
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 2.8 log10CFU 10.1039/C4MD00288A
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 2.86 deltalog10CFU 10.1016/j.bmc.2016.01.028
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 3.0 log10CFU/ml 10.1016/j.ejmech.2021.113932
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 3.3 10'5CFU 10.1016/j.bmc.2017.03.053
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 3.31 log10CFU 10.1039/C4MD00288A
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 3.9 log10CFU 10.1016/j.bmcl.2016.09.043
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 4.49 log10CFU 10.1021/acs.jmedchem.1c00263
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 5.2 None 10.1016/j.bmcl.2016.09.043
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 5.6 % 10.1128/aac.00897-07
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 9.2 % 10.1128/aac.01124-07
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 29.19 % 10.1016/j.bmcl.2012.10.032
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 61.2 % 10.1128/aac.00964-09
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 79.8 % 10.1128/aac.00964-09
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 82.58 % 10.1016/j.bmcl.2012.10.032
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 87.0 % 10.1016/j.ejmech.2016.08.039
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 87.0 % 10.1016/j.ejmech.2022.114454
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 87.2 % 10.1128/aac.00964-09
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 90.9 % 10.1128/aac.00964-09
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 93.8 % 10.1128/aac.00964-09
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 94.2 % 10.1128/aac.00964-09
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 94.5 % 10.1128/aac.01124-07
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 95.0 % 10.1371/journal.pmed.0030466
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 95.79 % 10.1021/jm701560p
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 95.9 % 10.1128/aac.00964-09
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 96.3 % 10.1128/aac.00964-09
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 96.59 % 10.1016/j.bmc.2010.09.006
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 98.0 % 10.1021/jm100165w
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 98.0 % 10.1039/C5MD00131E
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 98.42 % 10.1021/jm701560p
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 99.4 % 10.1128/aac.01124-07
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 99.79 % 10.1021/jm701560p
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 99.83 % 10.1016/j.bmc.2010.09.006
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 99.93 % 10.1016/j.bmc.2010.09.006
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 99.97 % 10.1016/j.bmc.2010.09.006
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 100.0 % 10.1021/np0703702
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 391.0 mg 10.1126/science.1106753
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity 466.0 mg 10.1126/science.1106753
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1016/j.bmc.2009.04.055
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1016/j.bmc.2016.03.003
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1016/j.bmc.2018.07.034
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1016/j.bmc.2022.116777
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1016/j.bmcl.2012.10.060
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1016/j.bmcl.2022.128824
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1016/j.bmcl.2022.128871
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1016/j.ejmech.2012.04.014
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1016/j.ejmech.2020.112772
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1021/acs.jmedchem.0c01374
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1021/acs.jmedchem.2c01493
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1021/acs.jmedchem.5b01699
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1021/acs.jmedchem.5b01833
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1021/acs.jnatprod.7b00903
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1021/acsmedchemlett.7b00287
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1021/jm0703901
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1021/ml200157f
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1039/C4MD00288A
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1039/d1md00387a
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1128/aac.00661-10
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1128/aac.00898-06
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1128/aac.01468-06
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1128/aac.01486-07
Mycobacterium tuberculosis Mycobacterium tuberculosis Activity nan None 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis C50g 2.019 mg/L 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis C50g 1932.0 mg/L 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis C50k 7.652 mg/L 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis C50k 22.41 mg/L 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis CFU 0.0 /ml 10.1128/aac.00086-07
Mycobacterium tuberculosis Mycobacterium tuberculosis CFU 1.95 /ml 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis CFU 39.0 None 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis CFU 2000.0 None 10.1016/j.ejmech.2015.03.036
Mycobacterium tuberculosis Mycobacterium tuberculosis DIZ nan None 10.1007/s00044-013-0487-6
Mycobacterium tuberculosis Mycobacterium tuberculosis Drug uptake nan None 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis EC50 20.0 nM 10.1016/j.bmcl.2012.12.069
Mycobacterium tuberculosis Mycobacterium tuberculosis EC90 0.02 uM 10.1016/j.bmcl.2012.12.069
Mycobacterium tuberculosis Mycobacterium tuberculosis EC90 0.03 uM 10.1016/j.bmcl.2012.12.069
Mycobacterium tuberculosis Mycobacterium tuberculosis EC90 0.1 ug ml-1 10.1016/j.bmcl.2004.09.052
Mycobacterium tuberculosis Mycobacterium tuberculosis EC90/MIC 1.67 None 10.1016/j.bmcl.2004.09.052
Mycobacterium tuberculosis Mycobacterium tuberculosis EC99 1.5 ug ml-1 10.1016/j.bmcl.2004.09.052
Mycobacterium tuberculosis Mycobacterium tuberculosis ED99 9.8 mg kg-1 10.1128/aac.01423-09
Mycobacterium tuberculosis Mycobacterium tuberculosis Emax 4.2 log10CFU/ml 10.1016/j.bmcl.2018.11.002
Mycobacterium tuberculosis Mycobacterium tuberculosis Emax 6.2 log10CFU/ml 10.1016/j.bmcl.2018.11.002
Mycobacterium tuberculosis Mycobacterium tuberculosis Emax 6.3 log10CFU/ml 10.1016/j.bmcl.2018.11.002
Mycobacterium tuberculosis Mycobacterium tuberculosis Emax 30.0 mg kg-1 10.1128/aac.01423-09
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 0.46 None 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 0.48 None 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 0.81 None 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 0.98 None 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 1.34 log10RLU 10.1021/acsmedchemlett.8b00410
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 1.42 log10RLU 10.1021/acsmedchemlett.8b00410
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 1.49 None 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 1.5 None 10.1016/j.ejmech.2019.112010
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 1.6 None 10.1016/j.ejmech.2020.112035
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 1.6 None 10.1016/j.ejmech.2020.112402
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 1.73 None 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 1.8 None 10.1021/acs.jnatprod.9b00475
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 1.83 None 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 1.85 None 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 2.0 None 10.1016/j.bmc.2016.09.012
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 2.0 None 10.1016/j.ejmech.2009.12.074
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 2.0 None 10.1016/j.ejmech.2014.12.046
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 2.2 None 10.1016/j.bmc.2016.07.051
Mycobacterium tuberculosis Mycobacterium tuberculosis FC 2.68 None 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 0.0 % 10.1016/j.bmc.2012.09.019
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 46.21 % 10.1016/j.bmc.2016.09.008
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 53.0 % 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 55.0 % 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 62.27 % 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 63.0 % 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 65.0 % 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 66.33 % 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 68.0 % 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 71.0 % 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 72.0 % 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 73.67 % 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 74.0 % 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 76.33 % 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 84.0 % 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 86.0 % 10.1016/j.ejmech.2017.04.002
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 91.0 % 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 94.6 % 10.1016/j.ejmech.2017.03.065
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 95.0 % 10.1007/s00044-012-0451-x
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 95.0 % 10.1016/j.bmcl.2013.06.072
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 95.0 % 10.1016/j.ejmech.2011.07.033
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 95.0 % 10.1016/j.ejmech.2011.07.049
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 95.0 % 10.1016/j.ejmech.2012.01.008
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 96.0 % 10.1016/j.ejmech.2008.12.001
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 96.4 % 10.1016/j.ejmech.2017.03.065
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 96.8 % 10.1016/j.ejmech.2017.03.065
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 97.0 % 10.1016/j.bmc.2007.05.063
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 97.0 % 10.1016/j.bmcl.2013.06.076
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 97.0 % 10.1016/j.ejmech.2006.12.001
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 97.6 % 10.1021/np9000569
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 98.0 % 10.1007/s00044-011-9808-9
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 98.0 % 10.1007/s00044-011-9857-0
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 98.0 % 10.1007/s00044-012-0322-5
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 98.0 % 10.1007/s00044-013-0803-1
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 98.0 % 10.1016/j.bmc.2013.06.027
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 98.0 % 10.1016/j.ejmech.2011.09.023
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 98.0 % 10.1016/j.ejmech.2013.03.017
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 98.0 % 10.1016/j.ejmech.2013.05.003
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 98.0 % 10.1016/j.ejmech.2017.03.065
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 99.0 % 10.1007/s00044-012-0026-x
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 99.0 % 10.1007/s00044-012-0041-y
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 99.0 % 10.1007/s00044-012-0073-3
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 99.0 % 10.1007/s00044-012-0129-4
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 99.0 % 10.1016/j.ejmech.2012.12.055
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 99.0 % 10.1016/j.ejmech.2013.06.010
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 99.0 % 10.1016/j.ejmech.2014.02.005
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 99.0 % 10.1016/j.ejmech.2017.03.065
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 99.5 % 10.1016/j.ejmech.2017.03.065
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 100.0 % 10.1016/j.bmc.2012.05.004
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 100.0 % 10.1016/j.bmc.2012.09.019
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 100.0 % 10.1016/j.bmc.2013.07.003
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 100.0 % 10.1016/j.bmc.2016.09.008
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 100.0 % 10.1016/j.bmcl.2011.11.114
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 100.0 % 10.1016/j.bmcl.2020.127351
Mycobacterium tuberculosis Mycobacterium tuberculosis GI 100.0 % 10.1016/j.ejmech.2013.06.010
Mycobacterium tuberculosis Mycobacterium tuberculosis GI nan None 10.1007/s00044-012-0255-z
Mycobacterium tuberculosis Mycobacterium tuberculosis GI nan None 10.1016/j.bmc.2012.05.004
Mycobacterium tuberculosis Mycobacterium tuberculosis GI nan None 10.1016/j.bmc.2013.07.003
Mycobacterium tuberculosis Mycobacterium tuberculosis GI nan None 10.1016/j.bmc.2016.02.035
Mycobacterium tuberculosis Mycobacterium tuberculosis GI nan None 10.1021/acs.jmedchem.5b00608
Mycobacterium tuberculosis Mycobacterium tuberculosis GI nan None 10.1039/C7MD00146K
Mycobacterium tuberculosis Mycobacterium tuberculosis GI50 30.0 nM 10.1016/j.ejmech.2013.06.010
Mycobacterium tuberculosis Mycobacterium tuberculosis Hg 0.361 None 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis Hg 4.542 None 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis Hk 1.388 None 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis Hk 45.33 None 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0014 ug.mL-1 10.1016/j.bmcl.2015.08.006
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0014 ug.mL-1 10.1016/j.bmcl.2016.03.055
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0016 ug.mL-1 10.1016/j.bmcl.2016.02.043
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0017 ug.mL-1 10.1016/j.bmcl.2016.02.043
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0017 ug.mL-1 10.1016/j.bmcl.2016.05.093
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0018 ug.mL-1 10.1016/j.bmcl.2015.08.006
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0018 ug.mL-1 10.1016/j.bmcl.2015.11.071
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0018 ug.mL-1 10.1016/j.bmcl.2016.02.056
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0019 ug.mL-1 10.1016/j.ejmech.2016.09.059
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0019 ug.mL-1 10.1039/C8MD00055G
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.002 ug.mL-1 10.1039/C5MD00057B
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0021 ug.mL-1 10.1016/j.bmcl.2015.08.006
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0021 ug.mL-1 10.1016/j.ejmech.2016.09.059
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0024 ug.mL-1 10.1016/j.bmcl.2016.05.093
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.004 ug.mL-1 10.1016/j.bmcl.2016.03.055
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.004 ug.mL-1 10.1016/j.ejmech.2016.09.059
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0043 ug.mL-1 10.1016/j.ejmech.2016.09.059
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.0047 ug.mL-1 10.1021/np9000703
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.02 ug.mL-1 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.02 ug.mL-1 10.1039/C8MD00055G
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.08 ug.mL-1 10.1021/acs.jnatprod.0c01104
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.72 nM 10.1016/j.bmc.2017.09.037
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 0.72 nM 10.1016/j.ejmech.2017.07.060
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 2.0 ug.mL-1 10.1021/ml5001933
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 2.4 nM 10.1016/j.bmcl.2019.03.020
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 2.4 nM 10.1016/j.ejmech.2017.03.065
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 2.9 ug.mL-1 10.1021/ml5001933
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 4.1 nM 10.1021/acsmedchemlett.5b00176
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 4.6 nM 10.1016/j.bmc.2017.09.037
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 4.6 nM 10.1016/j.ejmech.2017.07.060
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 4.7 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 8.4 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 10.0 nM 10.1016/j.bmc.2020.115797
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 13.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 20.0 nM 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 20.0 nM 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 20.0 nM 10.1016/j.ejmech.2017.11.035
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 30.0 nM 10.1016/j.bmcl.2017.07.067
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 40.0 nM 10.1016/j.ejmech.2017.03.065
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 60.0 nM 10.1016/j.bmc.2020.115797
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 91.0 nM 10.1021/acs.jmedchem.2c01493
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 147.0 ug.mL-1 10.1016/s0960-894x(01)00283-9
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 152.0 nM 10.1021/np500617u
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 550.0 nM 10.1016/j.ejmech.2019.01.026
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 1200.0 nM 10.1016/j.bmc.2021.116506
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 1200.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 1220.0 nM 10.1016/j.ejmech.2019.01.026
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 50000.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 nan None 10.1021/ml5001933
Mycobacterium tuberculosis Mycobacterium tuberculosis IC50 nan None 10.1021/np900281r
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.015 ug.mL-1 10.1016/j.ejmech.2010.06.036
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.0151 ug.mL-1 10.1016/j.ejmech.2016.09.059
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.0173 ug.mL-1 10.1016/j.ejmech.2016.09.059
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.02 ug.mL-1 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.02 ug.mL-1 10.1016/j.ejmech.2016.09.059
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.028 ug.mL-1 10.1016/j.ejmech.2016.09.059
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.043 ug.mL-1 10.1016/j.bmcl.2015.08.006
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.043 ug.mL-1 10.1016/j.bmcl.2016.02.056
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.048 ug.mL-1 10.1016/j.bmcl.2015.08.006
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.05 ug.mL-1 10.1016/j.bmcl.2016.03.045
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.051 ug.mL-1 10.1016/j.bmcl.2015.08.006
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.53 ug.mL-1 10.1039/C8MD00055G
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.72 ug.mL-1 10.1016/j.bmcl.2016.03.045
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 0.8 ug.mL-1 10.1039/C8MD00055G
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 3.7 nM 10.1016/j.bmc.2017.09.037
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 3.7 nM 10.1016/j.ejmech.2017.07.060
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 4.9 nM 10.1016/j.bmc.2017.09.037
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 4.9 nM 10.1016/j.ejmech.2017.07.060
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 6.9 nM 10.1021/acsmedchemlett.5b00176
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 12.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 20.0 nM 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 22.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 30.0 nM 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 30.0 nM 10.1016/j.ejmech.2017.11.035
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 39.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 2300.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis IC90 50000.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis Imax 54.0 % 10.1016/j.bmcl.2019.04.010
Mycobacterium tuberculosis Mycobacterium tuberculosis INH 0.13 ug ml-1 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 0.0 % 10.1021/jm100165w
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 13.0 % 10.1016/j.bmcl.2019.04.010
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 49.0 % 10.1016/j.bmcl.2008.09.029
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 54.8 % 10.1021/jm030479g
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 56.0 % 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 61.0 % 10.1021/acs.jmedchem.5b00608
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 61.2 % 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 63.0 % 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 68.0 % 10.1021/acs.jmedchem.5b00608
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 73.0 % 10.1016/j.bmcl.2008.09.029
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 80.0 % 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 90.0 % 10.1016/j.bmc.2008.10.086
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 90.0 % 10.1021/np050424c
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 91.7 % 10.1021/jm030479g
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 91.9 % 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 93.0 % 10.1021/jm061288r
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 94.0 % 10.1016/j.bmcl.2008.09.029
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 94.3 % 10.1021/jm030479g
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 95.0 % 10.1016/j.bmc.2017.07.034
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 95.0 % 10.1016/j.bmcl.2004.05.060
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 95.0 % 10.1016/j.ejmech.2011.03.039
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 95.0 % 10.1016/j.ejmech.2011.08.014
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 95.0 % 10.1016/j.ejmech.2013.11.002
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 97.0 % 10.1016/j.ejmech.2009.09.024
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 97.6 % 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1007/s00044-011-9952-2
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1016/j.bmc.2017.09.035
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1016/j.bmcl.2015.07.071
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1016/j.bmcl.2016.06.038
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1016/j.ejmech.2007.07.001
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1016/j.ejmech.2010.06.031
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1016/j.ejmech.2012.05.004
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1016/j.ejmech.2012.08.047
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1016/j.ejmech.2014.02.015
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1016/j.ejmech.2014.06.071
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1016/j.ejmech.2014.07.008
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1016/j.ejmech.2016.02.016
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1016/j.ejmech.2020.112886
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 98.0 % 10.1039/d2md00076h
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 99.0 % 10.1007/s00044-011-9950-4
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 99.0 % 10.1007/s00044-013-0472-0
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 99.0 % 10.1007/s00044-013-0839-2
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 99.0 % 10.1016/j.bmc.2015.11.018
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 99.0 % 10.1016/j.bmcl.2008.09.029
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 99.0 % 10.1016/j.ejmech.2009.11.036
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 99.0 % 10.1016/j.ejmech.2010.04.022
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 99.0 % 10.1016/j.ejmech.2012.03.033
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 99.0 % 10.1016/j.ejmech.2014.07.100
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 99.0 % 10.1016/j.ejmech.2020.112358
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 99.5 % 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 100.0 % 10.1007/s00044-012-9971-7
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 100.0 % 10.1016/j.bmc.2006.12.032
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 100.0 % 10.1016/j.bmc.2014.10.007
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 100.0 % 10.1016/j.bmcl.2007.04.007
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 100.0 % 10.1016/j.bmcl.2008.09.029
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 100.0 % 10.1016/j.bmcl.2021.128261
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 100.0 % 10.1016/j.ejmech.2012.08.047
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 100.0 % 10.1016/j.ejmech.2022.114831
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 100.0 % 10.1021/jm0703901
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 100.0 % 10.1021/jm070391t
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 100.0 % 10.1021/jm100165w
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition 100.0 % 10.1021/jm100568q
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition nan % 10.1007/s00044-013-0472-0
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition nan % 10.1016/j.ejmech.2015.03.036
Mycobacterium tuberculosis Mycobacterium tuberculosis Inhibition nan % 10.1016/j.ejmech.2019.05.082
Mycobacterium tuberculosis Mycobacterium tuberculosis IZ 28.0 mm 10.1016/j.bmc.2007.09.025
Mycobacterium tuberculosis Mycobacterium tuberculosis Kgmax 6.195 10'-3 log10CFU/ml/hr 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis Kgmax 9.756 10'-3 log10CFU/ml/hr 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis Kkmax 15.83 10'-3 log10CFU/ml/hr 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis Kkmax 29.38 10'-3 log10CFU/ml/hr 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 1.0 None 10.1021/jm4019228
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 1.76 None 10.1016/j.ejmech.2014.05.005
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 1.89 None 10.1126/science.1106753
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 1.93 None 10.1016/j.ejmech.2014.05.005
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 2.75 None 10.1126/science.1106753
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 2.8 None 10.1016/j.ejmech.2014.05.005
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 3.21 None 10.1016/j.ejmech.2010.05.035
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 3.279 None 10.1371/journal.pmed.0030466
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 3.31 None 10.1016/j.ejmech.2014.05.005
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 3.71 None 10.1016/j.ejmech.2014.05.005
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 3.8 None 10.1016/j.ejmech.2010.07.015
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 3.972 None 10.1371/journal.pmed.0030466
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 3.98 None 10.1016/j.ejmech.2010.05.035
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 4.05 None 10.1126/science.1106753
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 4.53 None 10.1021/np3007167
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 4.72 None 10.1126/science.1106753
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 5.231 None 10.1371/journal.pmed.0030466
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 5.634 None 10.1371/journal.pmed.0030466
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 5.75 None 10.1021/np3007167
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 6.14 None 10.1016/j.ejmech.2014.05.005
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu 7.409 None 10.1371/journal.pmed.0030466
Mycobacterium tuberculosis Mycobacterium tuberculosis log10cfu nan None 10.1016/j.ejmech.2010.07.015
Mycobacterium tuberculosis Mycobacterium tuberculosis Log10 cfu 4.1 None 10.1128/aac.00898-06
Mycobacterium tuberculosis Mycobacterium tuberculosis Log10 cfu 6.0 None 10.1128/aac.00898-06
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml -1.82 None 10.1128/aac.01204-07
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml -1.7 None 10.1128/aac.01204-07
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml -1.55 None 10.1128/aac.01204-07
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml -1.25 None 10.1128/aac.01204-07
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml -1.17 None 10.1128/aac.01204-07
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml -0.89 None 10.1128/aac.01204-07
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml -0.88 None 10.1128/aac.01204-07
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml -0.28 None 10.1128/aac.01204-07
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml 0.221 None 10.1128/aac.01474-06
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml 0.3 None 10.1128/aac.01474-06
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml 0.44 None 10.1128/aac.01474-06
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml 1.32 None 10.1128/aac.00753-07
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml 1.7 None 10.1016/j.ejmech.2012.02.033
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml 4.63 None 10.1128/aac.00753-07
Mycobacterium tuberculosis Mycobacterium tuberculosis log10CFU/ml 6.36 None 10.1128/aac.00753-07
Mycobacterium tuberculosis Mycobacterium tuberculosis log(1/C) 5.91 None 10.1021/jm00210a025
Mycobacterium tuberculosis Mycobacterium tuberculosis log(activity) 0.5 None 10.1016/j.bmc.2017.11.031
Mycobacterium tuberculosis Mycobacterium tuberculosis log(activity) 0.8 None 10.1016/j.ejmech.2017.12.088
Mycobacterium tuberculosis Mycobacterium tuberculosis log(activity) 0.9 None 10.1016/j.ejmech.2020.112178
Mycobacterium tuberculosis Mycobacterium tuberculosis log(activity) 1.2 None 10.1016/j.bmc.2017.11.031
Mycobacterium tuberculosis Mycobacterium tuberculosis log(activity) 1.3 None 10.1016/j.bmc.2017.03.053
Mycobacterium tuberculosis Mycobacterium tuberculosis log(activity) 1.5 None 10.1016/j.ejmech.2017.12.088
Mycobacterium tuberculosis Mycobacterium tuberculosis log(activity) 1.8 None 10.1016/j.ejmech.2020.112178
Mycobacterium tuberculosis Mycobacterium tuberculosis log(activity) 2.0 None 10.1016/j.bmc.2017.03.053
Mycobacterium tuberculosis Mycobacterium tuberculosis log(activity) 2.0 None 10.1016/j.bmc.2017.12.044
Mycobacterium tuberculosis Mycobacterium tuberculosis log(activity) 2.7 None 10.1021/acs.jmedchem.2c00972
Mycobacterium tuberculosis Mycobacterium tuberculosis -logMIC 6.924 None 10.1007/s00044-012-0385-3
Mycobacterium tuberculosis Mycobacterium tuberculosis MBC 0.01 ug ml-1 10.1016/j.bmc.2018.07.034
Mycobacterium tuberculosis Mycobacterium tuberculosis MBC 0.12 uM 10.1021/acs.jnatprod.9b01095
Mycobacterium tuberculosis Mycobacterium tuberculosis MBC 0.24 uM 10.1021/acs.jnatprod.9b01095
Mycobacterium tuberculosis Mycobacterium tuberculosis MBC 0.39 uM 10.1016/j.bmc.2008.12.006
Mycobacterium tuberculosis Mycobacterium tuberculosis MBC 100.0 ug ml-1 10.1016/j.bmc.2007.09.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MBC 161.0 ng/ml 10.1021/acs.jnatprod.5b00770
Mycobacterium tuberculosis Mycobacterium tuberculosis MBC nan None 10.1016/j.ejmech.2018.02.067
Mycobacterium tuberculosis Mycobacterium tuberculosis MBC90 0.1 ug ml-1 10.1021/np400145u
Mycobacterium tuberculosis Mycobacterium tuberculosis MBC90 0.5 ug ml-1 10.1021/np400145u
Mycobacterium tuberculosis Mycobacterium tuberculosis MBC99.9 0.78 ug ml-1 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis MBC99.9 1.56 ug ml-1 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis MBC99.9 1.56 ug ml-1 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis MCC 3.0 ug.mL-1 10.1021/jm0602662
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.0008 ug.mL-1 10.1128/aac.00550-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.001 ug.mL-1 10.1128/aac.00287-10
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.0016 ug.mL-1 10.1128/aac.00550-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.002 ug.mL-1 10.1128/aac.00287-10
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.0021 ug.mL-1 10.1016/j.bmcl.2016.03.055
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.0025 ug.mL-1 10.1021/np800082e
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.0025 ug.mL-1 10.1039/d2md00401a
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.003 ug.mL-1 10.1007/s00044-012-0222-8
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.003 ug.mL-1 10.1016/j.bmcl.2016.11.003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.003 ug.mL-1 10.1039/C8MD00212F
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.0032 ug.mL-1 10.1128/aac.00550-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.004 ug.mL-1 10.1016/j.bmcl.2009.09.095
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.004 ug.mL-1 10.1016/j.bmcl.2010.12.084
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.004 ug.mL-1 10.1016/j.ejmech.2010.07.003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.004 ug.mL-1 10.1016/j.ejmech.2020.112045
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.004 ug.mL-1 10.1016/j.ejmech.2020.112440
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.004 ug.mL-1 10.1128/aac.00287-10
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.005 ug.mL-1 10.1016/j.ejmech.2014.07.066
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.005 ug.mL-1 10.1021/acs.jmedchem.2c00972
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.006 ug.mL-1 10.1016/j.ejmech.2018.12.001
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.0063 ug.mL-1 10.1021/acs.jnatprod.5b00961
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.007 ug.mL-1 10.1016/j.ejmech.2016.09.030
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.007 ug.mL-1 10.1021/jm4012033
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.008 ug.mL-1 10.1016/j.bmcl.2007.02.024
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.008 ug.mL-1 10.1021/jm500432n
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.008 ug.mL-1 10.1128/aac.00287-10
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.01 ug.mL-1 10.1016/j.bmcl.2014.09.080
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.01 ug.mL-1 10.1016/j.ejmech.2020.112175
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.01 ug.mL-1 10.1016/j.ejmech.2020.112835
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.01 ug.mL-1 10.1021/jm4012033
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.0125 ug.mL-1 10.1016/j.bmcl.2018.12.053
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.013 ug.mL-1 10.1016/j.bmcl.2018.05.049
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.015 ug.mL-1 10.1016/j.bmc.2007.04.003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.015 ug.mL-1 10.1016/j.bmc.2010.02.024
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.015 ug.mL-1 10.1016/j.bmcl.2008.09.096
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.015 ug.mL-1 10.1016/j.bmcl.2013.06.076
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.015 ug.mL-1 10.1016/j.ejmech.2008.12.001
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.015 ug.mL-1 10.1016/j.ejmech.2017.11.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.015 ug.mL-1 10.1016/j.ejmech.2022.114145
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.015 ug.mL-1 10.1021/jm500432n
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.015 ug.mL-1 10.1128/aac.00287-10
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.015 ug.mL-1 10.1128/aac.01545-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.016 ug.mL-1 10.1016/j.bmcl.2006.12.066
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.016 ug.mL-1 10.1016/j.ejmech.2016.09.030
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.016 ug.mL-1 10.1021/acs.jmedchem.2c00972
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.017 ug.mL-1 10.1016/j.ejmech.2016.09.030
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.019 ug.mL-1 10.1016/j.bmcl.2018.05.049
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.02 ug.mL-1 10.1016/j.bmcl.2006.08.090
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.02 ug.mL-1 10.1016/j.bmcl.2016.05.093
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.02 ug.mL-1 10.1016/j.bmcl.2018.11.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.02 ug.mL-1 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.02 ug.mL-1 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.02 ug.mL-1 10.1016/j.ejmech.2014.10.079
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.02 ug.mL-1 10.1016/j.ejmech.2017.03.015
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.02 ug.mL-1 10.1016/j.ejmech.2020.112835
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.025 ug.mL-1 10.1016/j.ejmech.2021.113603
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.025 ug.mL-1 10.1021/jm00150a006
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.025 ug.mL-1 10.1021/np5005328
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1016/j.bmc.2010.05.016
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1016/j.bmc.2013.09.034
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1016/j.bmc.2013.10.011
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1016/j.bmc.2019.07.045
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1016/j.bmc.2022.116777
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1016/j.bmcl.2016.05.093
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1016/j.bmcl.2018.11.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1016/j.ejmech.2016.09.030
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1016/j.ejmech.2019.04.067
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1016/j.ejmech.2020.112835
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1016/j.ejmech.2021.113580
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1021/acs.jmedchem.0c00500
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1021/jm201608g
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1021/np049831z
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1039/d1md00387a
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1128/aac.00287-10
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.03 ug.mL-1 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.037 ug.mL-1 10.1016/j.bmc.2022.117006
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.037 ug.mL-1 10.1016/j.ejmech.2020.112409
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.038 ug.mL-1 10.1016/j.ejmech.2016.11.048
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.0382 ug.mL-1 10.1016/j.ejmech.2021.113398
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.04 ug.mL-1 10.1016/j.bmcl.2016.03.055
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.04 ug.mL-1 10.1016/j.ejmech.2020.112835
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.04 ug.mL-1 10.1021/acs.jmedchem.0c00500
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.04 ug.mL-1 10.1039/C5MD00057B
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.041 ug.mL-1 10.1016/j.bmcl.2016.02.043
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.042 ug.mL-1 10.1016/j.ejmech.2022.114502
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.043 ug.mL-1 10.1016/j.bmcl.2015.11.071
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.043 ug.mL-1 10.1016/j.ejmech.2017.06.051
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.043 ug.mL-1 10.1016/j.ejmech.2022.114454
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.045 ug.mL-1 10.1016/j.bmcl.2016.02.043
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.049 ug.mL-1 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.049 ug.mL-1 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.049 ug.mL-1 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1016/j.bmc.2015.04.001
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1016/j.bmcl.2016.03.050
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1016/j.bmcl.2016.06.075
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1016/j.bmcl.2018.11.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1016/j.ejmech.2014.09.029
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1016/j.ejmech.2017.06.005
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1016/j.ejmech.2017.11.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1016/j.ejmech.2019.06.038
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1021/jm00150a006
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1021/jm500853v
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1128/aac.01288-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.05 ug.mL-1 10.1128/aac.01486-07
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.057 ug.mL-1 10.1016/j.ejmech.2020.112075
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1016/j.bmc.2008.10.042
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1016/j.bmcl.2008.09.029
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1016/j.ejmech.2008.04.013
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1016/j.ejmech.2010.11.020
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1016/j.ejmech.2011.10.041
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1016/j.ejmech.2014.02.017
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1016/j.ejmech.2019.07.057
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1016/j.ejmech.2020.112996
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1016/j.ejmech.2021.113580
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1016/s0960-894x(00)00058-5
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1016/s0960-894x(00)00648-x
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1021/acsmedchemlett.9b00515
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1021/np0303411
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1021/np2000667
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.06 ug.mL-1 10.1039/d1md00387a
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.062 ug.mL-1 10.1016/j.ejmech.2021.113472
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.062 ug.mL-1 10.1021/jm000413a
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.0625 ug.mL-1 10.1016/j.bmcl.2012.08.003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.0625 ug.mL-1 10.1016/j.ejmech.2012.03.012
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.0625 ug.mL-1 10.1016/j.ejmech.2021.113657
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.063 ug.mL-1 10.1016/j.bmc.2011.01.050
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.063 ug.mL-1 10.1016/j.bmc.2011.02.034
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.063 ug.mL-1 10.1021/np050554l
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.07 ug.mL-1 10.1016/j.bmc.2008.02.009
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.07 ug.mL-1 10.1021/jm201608g
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.07 ug.mL-1 10.1021/np400391p
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.074 ug.mL-1 10.1016/j.ejmech.2022.114454
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.075 ug.mL-1 10.1016/j.ejmech.2022.114454
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.078 ug.mL-1 10.1016/j.ejmech.2019.01.042
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.078 ug.mL-1 10.1039/C7MD00350A
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.078 ug.mL-1 10.1039/C7MD00366H
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.08 ug.mL-1 10.1021/acs.jmedchem.2c00972
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.08 ug.mL-1 10.1021/jm061288r
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.09 ug.mL-1 10.1021/jm900672t
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.095 ug.mL-1 10.1016/j.bmcl.2018.07.005
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1007/s00044-013-0787-x
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1016/j.bmc.2016.01.059
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1016/j.bmcl.2005.08.045
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1016/j.bmcl.2007.10.083
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1016/j.bmcl.2009.04.029
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1016/j.bmcl.2011.05.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1016/j.bmcl.2015.07.069
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1016/j.bmcl.2019.06.055
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1016/j.ejmech.2010.09.019
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1016/j.ejmech.2014.07.067
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1016/j.ejmech.2017.04.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1016/j.ejmech.2019.112010
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1021/acs.jnatprod.1c00812
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1021/acs.jnatprod.7b00300
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1021/acsmedchemlett.1c00431
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1021/jm060339h
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1021/jm060957y
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.1 ug.mL-1 10.1021/np400391p
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.12 ug.mL-1 10.1016/j.bmcl.2007.07.027
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.12 ug.mL-1 10.1016/j.bmcl.2011.09.031
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.12 ug.mL-1 10.1016/j.ejmech.2010.12.028
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.12 ug.mL-1 10.1016/j.ejmech.2011.10.041
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.12 ug.mL-1 10.1021/jm020891g
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.12 ug.mL-1 10.1021/np5001494
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1007/s00044-013-0781-3
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/j.bmc.2007.05.063
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/j.bmc.2008.10.086
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/j.bmc.2013.09.034
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/j.bmcl.2005.01.073
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/j.bmcl.2007.04.007
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/j.bmcl.2011.02.022
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/j.bmcl.2012.05.063
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/j.ejmech.2009.10.050
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/j.ejmech.2013.12.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/j.ejmech.2018.03.016
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/j.ejmech.2018.11.032
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/j.ejmech.2021.113472
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/s0960-894x(00)00188-8
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1016/s0960-894x(01)00266-9
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1021/jm049952w
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1021/np049640w
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1021/np980066w
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.125 ug.mL-1 10.1128/aac.00643-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.127 ug.mL-1 10.1016/j.bmc.2018.03.004
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.15 ug.mL-1 10.1016/j.ejmech.2011.04.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.15 ug.mL-1 10.1016/j.ejmech.2014.06.071
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.15 ug.mL-1 10.1021/np500538c
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.15 ug.mL-1 10.1128/aac.00749-08
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.16 ug.mL-1 10.1021/np0002233
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.161 ug.mL-1 10.1021/acs.jnatprod.5b00770
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.195 ug.mL-1 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.195 ug.mL-1 10.1016/j.ejmech.2017.11.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.197 ug.mL-1 10.1016/j.ejmech.2018.05.049
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1007/s00044-011-9948-y
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.bmcl.2005.08.045
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.bmcl.2007.07.089
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.bmcl.2011.06.076
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.bmcl.2012.12.073
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.bmcl.2016.07.039
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.bmcl.2017.10.071
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.bmcl.2018.11.036
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.bmcl.2019.01.004
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.bmcl.2019.07.040
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.bmcl.2020.127434
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.ejmech.2011.06.014
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.ejmech.2013.03.027
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.ejmech.2013.10.082
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.ejmech.2017.07.059
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.ejmech.2018.07.046
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.ejmech.2018.12.043
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.ejmech.2019.05.082
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.ejmech.2020.112886
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1016/j.ejmech.2022.114454
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1021/jm070638m
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1039/C7MD00350A
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1039/C7MD00366H
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1128/aac.00643-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.2 ug.mL-1 10.1371/journal.pmed.0030466
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.23 ug.mL-1 10.1016/j.bmcl.2018.11.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.24 nM 10.1007/s00044-011-9662-9
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.24 nM 10.1007/s00044-011-9705-2
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.24 ug.mL-1 10.1039/C6MD00085A
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.24 ug.mL-1 10.1039/C6MD00593D
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1007/s00044-011-9950-4
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1007/s00044-012-0026-x
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1007/s00044-012-0041-y
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1007/s00044-012-0073-3
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1007/s00044-013-0472-0
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1007/s00044-013-0839-2
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.bmc.2007.03.086
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.bmc.2010.08.016
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.bmc.2010.09.006
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.bmc.2016.10.027
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.bmcl.2005.06.010
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.bmcl.2019.07.041
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.ejmech.2007.07.001
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.ejmech.2009.06.005
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.ejmech.2010.07.015
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.ejmech.2012.03.033
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.ejmech.2016.12.042
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.ejmech.2017.04.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.ejmech.2018.11.032
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1016/j.ejmech.2018.12.001
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1021/acs.jnatprod.2c00360
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1021/jm00167a029
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1021/jm0110284
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1021/jm701560p
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1021/np010101q
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1021/np010216u
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1021/np050424c
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1128/aac.00643-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.25 ug.mL-1 10.1128/aac.00661-10
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.29 ug.mL-1 10.1016/j.ejmech.2017.11.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.3 ug.mL-1 10.1016/j.ejmech.2018.08.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.3 ug.mL-1 10.1016/s0960-894x(99)00510-7
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.3 ug.mL-1 10.1021/jm0602662
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.37 ug.mL-1 10.1016/j.ejmech.2017.11.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.39 ug.mL-1 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.39 ug.mL-1 10.1016/j.bmcl.2017.07.023
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.39 ug.mL-1 10.1016/j.ejmech.2017.06.051
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.39 ug.mL-1 10.1016/j.ejmech.2017.11.090
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.39 ug.mL-1 10.1016/j.ejmech.2018.01.080
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.39 ug.mL-1 10.1371/journal.pmed.0030466
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.4 ug.mL-1 10.1016/j.ejmech.2015.03.014
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.4 ug.mL-1 10.1016/j.ejmech.2015.10.047
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.4 ug.mL-1 10.1016/j.ejmech.2016.05.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.4 ug.mL-1 10.1016/j.ejmech.2016.11.032
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.4 ug.mL-1 10.1016/j.ejmech.2018.08.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.41 ug.mL-1 10.1016/j.ejmech.2017.01.009
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.42 ug.mL-1 10.1016/j.ejmech.2016.09.030
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.48 ug.mL-1 10.1016/j.ejmech.2017.01.009
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 nM 10.1016/j.ejmech.2019.111578
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1007/s00044-012-0451-x
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.bmc.2015.11.018
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.bmc.2019.04.017
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.bmcl.2005.01.073
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.bmcl.2005.11.087
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.bmcl.2009.12.045
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.bmcl.2013.06.072
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.bmcl.2023.129189
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.ejmech.2009.11.036
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.ejmech.2010.11.020
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.ejmech.2011.03.039
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.ejmech.2011.07.033
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.ejmech.2011.07.049
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.ejmech.2011.08.014
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.ejmech.2012.01.008
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.ejmech.2013.11.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.ejmech.2013.12.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1016/j.ejmech.2018.09.049
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1021/np020592u
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1021/np0400095
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1021/np0601399
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.5 ug.mL-1 10.1021/np9700681
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.51 ug.mL-1 10.1016/j.ejmech.2017.01.009
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.51 ug.mL-1 10.1016/j.ejmech.2020.113102
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.6 ug.mL-1 10.1016/j.ejmech.2010.05.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.62 ug.mL-1 10.1016/j.ejmech.2017.11.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.64 ug.mL-1 10.1021/acs.jnatprod.5b00975
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.65 ug.mL-1 10.1021/acsmedchemlett.1c00431
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.72 ug.mL-1 10.1016/j.bmcl.2016.03.045
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.72 ug.mL-1 10.1016/j.bmcl.2019.06.055
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.75 ug.mL-1 10.1016/j.bmcl.2006.07.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.75 ug.mL-1 10.1016/j.ejmech.2017.01.009
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.75 ug.mL-1 10.1016/j.ejmech.2020.113102
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.75 ug.mL-1 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.78 ug.mL-1 10.1016/j.bmcl.2012.01.052
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.78 ug.mL-1 10.1039/C8MD00056E
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.78 ug.mL-1 10.1371/journal.pmed.0030466
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.8 ug.mL-1 10.1016/j.bmc.2010.09.006
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.8 ug.mL-1 10.1016/j.bmcl.2020.127655
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.84 ug.mL-1 10.1016/j.ejmech.2011.04.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 0.91 ug.mL-1 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 mg 10.1016/j.bmc.2007.07.023
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 nM 10.1016/j.bmcl.2019.04.010
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 nM 10.1021/acs.jmedchem.1c00837
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1007/s00044-012-0074-2
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.bmc.2007.08.045
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.bmc.2009.04.055
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.bmcl.2007.07.073
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.bmcl.2007.09.096
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2007.01.009
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2007.08.003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2008.06.014
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2009.03.027
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2009.07.015
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2014.09.043
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2015.10.054
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2017.04.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2018.01.080
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2019.111882
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2021.113266
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.0 ug.mL-1 10.1021/jm00210a025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.2 ug.mL-1 10.1016/j.bmc.2011.11.020
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.2 ug.mL-1 10.1016/j.ejmech.2014.10.031
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.47 ug.mL-1 10.1016/j.bmc.2018.07.034
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.47 ug.mL-1 10.1021/jm201608g
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.56 ug.mL-1 10.1016/j.ejmech.2013.12.013
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1.6 ug.mL-1 10.1016/j.bmcl.2016.11.047
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 nM 10.1021/acs.jmedchem.1c00837
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1007/s00044-012-0268-7
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.bmc.2011.01.050
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.bmc.2013.09.034
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.bmc.2019.04.032
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.bmcl.2009.11.107
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.bmcl.2011.05.016
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.bmcl.2012.02.053
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.bmcl.2012.12.096
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.ejmech.2010.06.006
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.ejmech.2011.03.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.ejmech.2011.10.041
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.ejmech.2013.03.027
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.ejmech.2014.10.026
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1016/j.ejmech.2020.112835
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1021/acsmedchemlett.5b00202
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1021/jm000149l
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1021/np050554l
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.0 ug.mL-1 10.1039/C9MD00057G
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.5 ug.mL-1 10.1016/j.bmc.2011.11.020
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.5 ug.mL-1 10.1016/j.ejmech.2014.10.031
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2.5 ug.mL-1 10.1016/j.ejmech.2021.113266
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3.0 nM 10.1021/acs.jmedchem.1c00837
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3.0 nM 10.1021/ml5001933
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3.0 ug.mL-1 10.1016/j.bmcl.2018.05.049
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3.1 ug.mL-1 10.1016/j.ejmech.2019.111882
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3.12 ug.mL-1 10.1021/jm060339h
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3.13 ug.mL-1 10.1016/j.bmcl.2009.04.029
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3.13 ug.mL-1 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3.64 nM 10.1021/acsmedchemlett.5b00176
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 4.0 nM 10.1021/acs.jmedchem.1c00837
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 4.0 nM 10.1021/jm5005978
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 4.0 ug.mL-1 10.1016/j.bmcl.2018.11.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 4.0 ug.mL-1 10.1016/j.ejmech.2019.01.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 4.0 ug.mL-1 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 4.0 ug.mL-1 10.1021/jm201608g
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 4.0 ug.mL-1 10.1039/d2md00260d
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 4.2 ug.mL-1 10.1016/j.ejmech.2010.05.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 5.0 nM 10.1021/acs.jmedchem.1c00837
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 5.0 nM 10.1021/acsmedchemlett.9b00343
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 5.0 ug.mL-1 10.1016/j.bmcl.2006.08.090
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 6.0 nM 10.1016/j.bmcl.2011.06.018
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 6.0 nM 10.1016/j.bmcl.2011.07.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 6.0 nM 10.1021/acs.jnatprod.1c00232
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 6.25 nM 10.1021/acs.jnatprod.0c00804
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 6.25 ug.mL-1 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 6.5 nM 10.1021/acsmedchemlett.5b00176
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 6.5 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 7.5 ug.mL-1 10.1007/s00044-013-0485-8
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 8.0 nM 10.1021/ml5001728
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 8.0 nM 10.1021/ml500531p
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 8.0 ug.mL-1 10.1016/j.bmc.2019.07.045
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 8.0 ug.mL-1 10.1016/j.ejmech.2015.03.014
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 8.0 ug.mL-1 10.1016/j.ejmech.2017.11.083
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 8.0 ug.mL-1 10.1016/s0960-894x(01)00266-9
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 8.0 ug.mL-1 10.1021/acs.jnatprod.2c00360
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 8.0 ug.mL-1 10.1128/aac.00287-10
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 9.0 nM 10.1021/acs.jmedchem.1c00707
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 9.24 ug.mL-1 10.1016/j.ejmech.2022.114145
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 10.0 nM 10.1016/j.bmc.2010.07.010
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 10.0 nM 10.1016/j.ejmech.2009.12.074
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 10.0 nM 10.1021/acsmedchemlett.9b00343
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 10.0 nM 10.1021/jm5005978
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 10.0 ug.mL-1 10.1016/j.ejmech.2020.112075
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 10.0 ug.mL-1 10.1016/j.ejmech.2020.112409
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 10.0 ug.mL-1 10.1016/j.ejmech.2021.113398
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 10.0 ug.mL-1 10.1016/j.ejmech.2021.113603
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 10.0 ug.mL-1 10.1016/j.ejmech.2022.114145
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 10.0 ug.mL-1 10.1021/acs.jmedchem.0c00500
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 10.0 ug.mL-1 10.1021/acs.jmedchem.0c02153
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 11.0 nM 10.1016/j.bmc.2017.09.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 11.0 nM 10.1016/j.ejmech.2017.07.060
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 12.0 nM 10.1016/j.bmc.2017.09.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 12.0 nM 10.1016/j.ejmech.2017.07.060
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 15.0 nM 10.1016/j.bmc.2017.09.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 15.0 nM 10.1016/j.ejmech.2017.07.060
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 15.0 nM 10.1021/jm401268f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 15.0 nM 10.1021/ml5001728
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 15.0 nM 10.1021/ml500531p
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 15.0 ug.mL-1 10.1016/j.ejmech.2006.12.001
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 16.0 nM 10.1016/j.bmcl.2015.04.099
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 16.0 ug.mL-1 10.1016/j.bmc.2011.02.034
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 16.0 ug.mL-1 10.1016/j.bmc.2016.10.027
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 16.0 ug.mL-1 10.1016/j.bmc.2021.116529
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 16.0 ug.mL-1 10.1016/j.bmcl.2005.01.073
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 16.0 ug.mL-1 10.1016/j.bmcl.2012.08.003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 16.0 ug.mL-1 10.1021/acs.jnatprod.2c00360
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 16.0 ug.mL-1 10.1128/aac.00287-10
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 16.0 ug.mL-1 10.1128/aac.00643-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 16.0 ug.mL-1 10.1128/aac.00661-10
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 16.0 ug.mL-1 10.1128/aac.01545-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 18.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 20.0 nM 10.1016/j.bmc.2010.08.016
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 20.0 nM 10.1016/j.ejmech.2018.02.067
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 20.0 nM 10.1021/jm5002937
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 20.0 nM 10.1021/jm5005978
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 20.0 ug.mL-1 10.1016/j.bmcl.2011.09.031
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 22.0 nM 10.1016/j.bmc.2017.09.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 22.0 nM 10.1016/j.ejmech.2017.07.060
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 25.0 ug.mL-1 10.1007/s00044-012-0451-x
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 25.0 ug.mL-1 10.1016/j.bmc.2019.04.032
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 25.0 ug.mL-1 10.1016/j.bmcl.2013.06.072
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 25.0 ug.mL-1 10.1016/j.ejmech.2011.07.033
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 25.0 ug.mL-1 10.1016/j.ejmech.2011.08.014
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 25.0 ug.mL-1 10.1016/j.ejmech.2012.01.008
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 25.0 ug.mL-1 10.1016/j.ejmech.2013.11.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 25.0 ug.mL-1 10.1016/j.ejmech.2018.08.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 25.0 ug.mL-1 10.1021/acsmedchemlett.1c00431
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 25.0 ug.mL-1 10.1021/jm070638m
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 27.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 30.0 nM 10.1016/j.bmcl.2015.04.099
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 30.0 nM 10.1021/acs.jnatprod.9b01095
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 30.0 nM 10.1021/jm401268f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 30.0 nM 10.1021/jm5005978
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 30.0 ug.mL-1 10.1007/s00044-013-0485-8
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32.0 ug.mL-1 10.1007/s00044-011-9573-9
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32.0 ug.mL-1 10.1016/j.bmc.2021.116529
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32.0 ug.mL-1 10.1016/j.bmcl.2008.10.045
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32.0 ug.mL-1 10.1016/j.bmcl.2012.08.003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32.0 ug.mL-1 10.1016/j.bmcl.2017.07.023
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32.0 ug.mL-1 10.1016/j.ejmech.2009.05.015
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32.0 ug.mL-1 10.1016/j.ejmech.2012.03.012
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32.0 ug.mL-1 10.1016/j.ejmech.2017.11.090
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.01.080
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32.0 ug.mL-1 10.1016/j.ejmech.2018.11.032
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32.0 ug.mL-1 10.1016/j.ejmech.2019.01.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32.0 ug.mL-1 10.1016/j.ejmech.2019.111882
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 36.4 nM 10.1021/acsmedchemlett.5b00176
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 36.89 ug.mL-1 10.1016/j.ejmech.2019.06.038
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 36.89 ug.mL-1 10.1021/acsmedchemlett.6b00330
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 37.0 nM 10.1016/j.bmc.2009.06.051
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 38.0 nM 10.1016/j.bmcl.2013.11.024
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 38.65 ug.mL-1 10.1016/j.ejmech.2019.06.038
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 38.65 ug.mL-1 10.1021/acsmedchemlett.6b00330
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 nM 10.1016/j.bmc.2010.08.016
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 nM 10.1016/j.bmc.2017.09.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 nM 10.1016/j.bmcl.2012.12.069
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 nM 10.1016/j.bmcl.2016.02.076
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 nM 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 nM 10.1016/j.ejmech.2017.07.060
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 nM 10.1016/j.ejmech.2017.11.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 nM 10.1021/acs.jnatprod.2c01003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 nM 10.1021/acsmedchemlett.5b00424
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 nM 10.1021/ml5003458
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 nM 10.1039/c5md00340g
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 nM 10.1039/C6MD00231E
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1007/s00044-010-9399-x
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1007/s00044-011-9952-2
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1007/s00044-012-0060-8
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1007/s00044-012-0129-4
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1007/s00044-012-0322-5
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1007/s00044-013-0803-1
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1016/j.bmcl.2018.07.005
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1016/j.ejmech.2010.06.031
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1016/j.ejmech.2010.08.014
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1016/j.ejmech.2011.09.023
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1016/j.ejmech.2012.12.055
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1016/j.ejmech.2013.03.017
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1016/j.ejmech.2013.05.003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1016/j.ejmech.2014.09.029
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1016/j.ejmech.2019.01.042
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40.0 ug.mL-1 10.1016/j.ejmech.2021.113266
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 41.0 ug.mL-1 10.1016/j.ejmech.2016.09.030
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 45.7 ug.mL-1 10.1007/s00044-013-0485-8
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 49.0 nM 10.1021/acsmedchemlett.7b00356
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50.0 nM 10.1016/j.bmcl.2009.12.062
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50.0 nM 10.1016/j.bmcl.2011.02.008
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50.0 nM 10.1016/j.bmcl.2016.02.076
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50.0 nM 10.1016/j.ejmech.2013.11.007
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50.0 nM 10.1021/acsmedchemlett.2c00254
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50.0 nM 10.1021/acsmedchemlett.5b00424
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50.0 nM 10.1021/jm900003c
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50.0 nM 10.1021/ml5003458
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50.0 nM 10.1039/c5md00340g
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50.0 ug.mL-1 10.1016/j.ejmech.2019.111882
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 60.0 nM 10.1016/j.bmcl.2013.11.050
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 60.0 nM 10.1016/j.bmcl.2020.127074
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 60.0 nM 10.1016/j.ejmech.2009.12.074
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 60.0 nM 10.1016/j.ejmech.2013.11.007
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 60.0 nM 10.1021/acs.jnatprod.0c00194
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 60.0 nM 10.1021/jm401268f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 60.0 nM 10.1021/jm900003c
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 60.0 nM 10.1021/jm901235p
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 60.7 nM 10.1039/C3MD00251A
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1016/j.bmc.2010.09.006
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1016/j.bmc.2019.04.017
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1016/j.bmc.2022.116777
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1016/j.bmcl.2019.07.041
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1016/j.ejmech.2012.03.012
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1016/j.ejmech.2018.09.049
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1016/j.ejmech.2019.01.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1016/j.ejmech.2019.111678
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1016/j.ejmech.2021.113580
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1016/j.ejmech.2022.114454
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1021/acs.jnatprod.2c00360
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1021/jm701560p
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1039/d1md00387a
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1039/d2md00260d
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64.0 ug.mL-1 10.1128/aac.00287-10
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 70.0 nM 10.1016/j.bmc.2007.05.053
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 70.0 nM 10.1039/C3MD00366C
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 70.0 nM 10.1039/C7MD00146K
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 80.0 nM 10.1016/j.bmc.2013.11.011
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 80.0 nM 10.1016/j.bmc.2014.10.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 80.0 nM 10.1039/C7MD00146K
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 89.0 nM 10.1016/j.bmcl.2013.11.024
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 90.0 nM 10.1016/j.bmc.2011.04.023
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 90.0 nM 10.1016/j.bmcl.2015.12.080
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 90.0 nM 10.1016/j.bmcl.2015.12.083
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 90.0 nM 10.1021/acs.jnatprod.2c01003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 90.0 nM 10.1021/acs.jnatprod.6b00839
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1007/s00044-011-9770-6
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1007/s00044-013-0850-7
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1016/j.bmc.2009.08.061
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1016/j.bmc.2010.03.018
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1016/j.bmc.2012.08.041
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1016/j.bmcl.2009.10.107
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1016/j.bmcl.2009.11.105
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1016/j.bmcl.2010.10.080
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1016/j.bmcl.2011.03.045
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1016/j.bmcl.2011.12.119
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1016/j.ejmech.2011.07.029
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1016/j.ejmech.2011.07.046
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1016/j.ejmech.2011.09.007
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1016/j.ejmech.2013.11.007
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1021/jm900003c
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1021/jm900340a
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1021/jm901112f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1021/jm901273n
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 nM 10.1021/np800751j
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 ug.mL-1 10.1016/j.ejmech.2009.06.005
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 ug.mL-1 10.1016/j.ejmech.2017.11.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 ug.mL-1 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 ug.mL-1 10.1021/np2000667
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100.0 ug.mL-1 10.1371/journal.pmed.0030466
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 110.0 nM 10.1016/j.ejmech.2021.113932
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 110.0 ug.mL-1 10.1016/j.bmc.2007.09.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 119.0 nM 10.1007/s00044-012-0385-3
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.bmc.2011.04.033
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.bmc.2019.01.022
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.bmcl.2014.02.052
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.ejmech.2009.09.001
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.ejmech.2009.09.033
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.ejmech.2009.09.034
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.ejmech.2010.10.020
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.ejmech.2011.07.026
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.ejmech.2012.04.021
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.ejmech.2017.06.051
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.ejmech.2020.112035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.ejmech.2020.112402
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 120.0 nM 10.1016/j.ejmech.2022.114454
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 128.0 ug.mL-1 10.1016/j.ejmech.2013.03.027
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 128.0 ug.mL-1 10.1016/j.ejmech.2019.01.002
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 128.0 ug.mL-1 10.1016/j.ejmech.2019.07.057
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 128.0 ug.mL-1 10.1016/j.ejmech.2019.111678
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 128.0 ug.mL-1 10.1021/acsmedchemlett.5b00202
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 140.0 nM 10.1016/j.ejmech.2013.11.007
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 140.0 nM 10.1021/np200022b
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 150.0 nM 10.1016/j.bmc.2014.08.031
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 150.0 nM 10.1016/j.bmc.2014.10.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 150.0 nM 10.1016/j.bmc.2016.07.051
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 150.0 nM 10.1016/j.bmc.2017.11.031
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 150.0 nM 10.1016/j.ejmech.2014.09.028
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 150.0 nM 10.1016/j.ejmech.2014.12.046
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 150.0 nM 10.1021/jm020891g
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 152.0 nM 10.1016/j.bmcl.2009.07.147
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 160.0 nM 10.1016/j.bmcl.2012.12.069
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 164.0 nM 10.1016/j.ejmech.2019.06.053
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 190.0 nM 10.1016/j.ejmech.2010.11.023
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 200.0 nM 10.1016/j.bmcl.2009.11.105
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 200.0 nM 10.1016/j.bmcl.2019.02.019
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 200.0 ug.mL-1 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 210.0 nM 10.1016/j.bmcl.2013.11.024
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 210.0 nM 10.1016/j.ejmech.2017.12.088
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 210.0 nM 10.1021/np900281r
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 230.0 nM 10.1007/s00044-011-9638-9
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 230.0 nM 10.1016/j.bmc.2014.10.016
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 230.0 nM 10.1016/j.bmc.2015.02.032
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 230.0 nM 10.1016/j.bmc.2015.03.004
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 230.0 nM 10.1016/j.bmc.2016.01.011
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 230.0 nM 10.1016/j.bmc.2016.09.012
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 230.0 nM 10.1016/j.bmcl.2008.12.088
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 230.0 nM 10.1016/j.bmcl.2020.127074
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 230.0 nM 10.1016/j.ejmech.2015.06.032
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 230.0 nM 10.1016/j.ejmech.2016.06.042
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 240.0 nM 10.1016/j.bmc.2012.01.041
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 240.0 nM 10.1016/j.bmc.2012.06.030
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 240.0 nM 10.1016/j.bmc.2013.11.011
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 240.0 nM 10.1016/j.bmcl.2007.01.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 240.0 nM 10.1016/j.bmcl.2020.127037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 240.0 nM 10.1016/j.ejmech.2016.03.060
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 240.0 nM 10.1016/j.ejmech.2021.113266
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 240.0 nM 10.1021/np0580210
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 240.0 ug.mL-1 10.1128/aac.01486-07
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 243.0 nM 10.1016/j.ejmech.2013.01.017
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 250.0 nM 10.1016/j.bmc.2019.02.053
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 250.0 nM 10.1016/j.ejmech.2010.02.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 256.0 ug.mL-1 10.1016/j.bmcl.2021.128088
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 256.0 ug.mL-1 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 256.0 ug.mL-1 10.1021/acsmedchemlett.5b00202
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 280.0 ug.mL-1 10.1007/s00044-013-0487-6
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 290.0 nM 10.1016/j.ejmech.2014.06.075
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 300.0 nM 10.1016/j.bmc.2014.10.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 300.0 nM 10.1016/j.ejmech.2017.10.010
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 300.0 nM 10.1016/j.ejmech.2020.112699
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 300.0 nM 10.1021/acs.jnatprod.0c00151
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 300.0 nM 10.1021/np000267b
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 350.0 nM 10.1016/j.ejmech.2021.113932
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 377.0 nM 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 480.0 nM 10.1016/j.bmcl.2010.06.096
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 480.0 nM 10.1016/j.bmcl.2012.10.060
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 490.0 nM 10.1016/j.bmcl.2013.11.024
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 500.0 nM 10.1016/j.bmc.2017.03.053
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 500.0 nM 10.1016/j.ejmech.2010.02.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 500.0 nM 10.1016/j.ejmech.2010.04.022
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 500.0 nM 10.1016/j.ejmech.2020.112178
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 500.0 nM 10.1021/acs.jmedchem.6b00674
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 500.0 nM 10.1128/aac.00055-06
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 600.0 nM 10.1021/acs.jnatprod.9b00475
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 610.0 nM 10.1016/j.bmc.2014.10.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 610.0 nM 10.1016/j.ejmech.2020.112898
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 610.0 nM 10.1021/np0202226
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 640.0 nM 10.1021/acsmedchemlett.7b00356
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 910.0 nM 10.1016/j.ejmech.2018.04.039
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 940.0 nM 10.1016/j.bmc.2007.05.053
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 950.0 nM 10.1016/j.ejmech.2021.113932
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 970.0 nM 10.1016/j.bmc.2011.04.023
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 970.0 nM 10.1016/j.ejmech.2018.04.039
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1000.0 nM 10.1016/j.bmc.2008.12.070
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1000.0 nM 10.1016/j.ejmech.2014.05.069
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1000.0 nM 10.1016/j.ejmech.2015.11.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1130.0 nM 10.1016/j.ejmech.2021.113932
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1210.0 nM 10.1021/jm2003624
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1220.0 nM 10.1016/j.ejmech.2018.01.071
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1400.0 nM 10.1016/j.bmc.2015.03.008
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1410.0 nM 10.1016/j.bmc.2008.12.006
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1500.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1800.0 nM 10.1128/aac.00055-06
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1900.0 nM 10.1016/j.bmc.2010.03.018
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1900.0 nM 10.1016/j.ejmech.2021.113932
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1900.0 nM 10.1021/jm900003c
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 1900.0 nM 10.1021/jm901273n
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2000.0 nM 10.1016/j.bmcl.2009.11.105
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2000.0 nM 10.1016/j.bmcl.2013.08.101
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2000.0 nM 10.1016/j.bmcl.2015.12.083
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2000.0 nM 10.1016/j.ejmech.2014.05.069
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2000.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2000.0 nM 10.1021/jm900340a
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2400.0 nM 10.1016/j.bmcl.2009.12.062
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2400.0 nM 10.1016/j.bmcl.2011.02.008
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2400.0 nM 10.1016/j.ejmech.2020.112358
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2430.0 nM 10.1016/j.bmcl.2009.07.147
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2430.0 nM 10.1016/j.ejmech.2011.07.026
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 2800.0 nM 10.1016/j.bmc.2015.03.008
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3000.0 nM 10.1016/j.bmc.2018.07.049
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3120.0 nM 10.1016/j.bmcl.2011.06.018
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3120.0 nM 10.1016/j.bmcl.2011.07.035
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3790.0 nM 10.1007/s00044-011-9638-9
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3790.0 nM 10.1016/j.bmc.2007.05.053
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3790.0 nM 10.1016/j.ejmech.2009.09.033
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3800.0 nM 10.1007/s00044-013-0850-7
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3800.0 nM 10.1016/j.bmcl.2009.10.107
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3800.0 nM 10.1016/j.ejmech.2009.09.001
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3800.0 nM 10.1016/j.ejmech.2012.04.021
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 3820.0 nM 10.1016/j.ejmech.2021.113932
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 4000.0 nM 10.1016/j.bmc.2010.08.016
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 4000.0 nM 10.1016/j.ejmech.2013.11.007
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 4800.0 nM 10.1016/j.bmc.2012.08.041
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 4800.0 nM 10.1016/j.bmcl.2017.01.024
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 5000.0 nM 10.1021/jm5002937
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 6700.0 nM 10.1016/j.ejmech.2015.03.021
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 7200.0 nM 10.1016/j.bmc.2017.09.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 7200.0 nM 10.1016/j.ejmech.2017.07.060
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 8000.0 nM 10.1016/j.ejmech.2014.05.069
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 8000.0 nM 10.1016/j.ejmech.2016.11.041
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 12100.0 nM 10.1016/j.ejmech.2018.04.039
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 12200.0 nM 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 12500.0 nM 10.1021/ml5001933
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 15180.0 nM 10.1016/j.bmcl.2010.06.096
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 15190.0 nM 10.1016/j.ejmech.2010.10.020
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 15200.0 nM 10.1016/j.bmcl.2008.12.088
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 16000.0 nM 10.1016/j.ejmech.2014.05.069
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 19000.0 nM 10.1039/C7MD00146K
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 19400.0 nM 10.1016/j.bmcl.2017.01.024
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 21000.0 nM 10.1039/C6MD00278A
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 24000.0 nM 10.1039/C6MD00278A
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 25000.0 nM 10.1016/j.ejmech.2010.04.022
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 30370.0 nM 10.1016/j.bmc.2014.08.031
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 30370.0 nM 10.1016/j.ejmech.2014.09.028
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 30400.0 nM 10.1016/j.bmcl.2019.02.019
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32000.0 nM 10.1021/jm900003c
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 32000.0 nM 10.1021/jm901273n
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40000.0 nM 10.1016/j.bmc.2019.01.022
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 40000.0 nM 10.1016/j.ejmech.2019.06.053
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 48000.0 nM 10.1016/j.ejmech.2016.02.016
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 48600.0 nM 10.1021/acsmedchemlett.2c00254
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 48610.0 nM 10.1016/j.ejmech.2020.112967
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50000.0 nM 10.1016/j.bmc.2017.09.037
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50000.0 nM 10.1016/j.ejmech.2017.07.060
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 50000.0 nM 10.1021/acsmedchemlett.6b00088
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 64000.0 nM 10.1039/C3MD00366C
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 100000.0 nM 10.1016/j.ejmech.2016.11.048
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 121510.0 nM 10.1016/j.bmc.2007.05.053
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 151900.0 nM 10.1016/j.ejmech.2018.02.067
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 250000.0 ug.mL-1 10.1016/j.ejmech.2008.01.016
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 256000.0 nM 10.1039/C3MD00366C
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 311000.0 nM 10.1016/j.ejmech.2010.11.023
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC 311080.0 nM 10.1016/j.ejmech.2020.112898
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC nan ug.mL-1 10.1016/s0960-894x(00)00159-1
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC nan None 10.1007/s00044-013-0472-0
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC nan None 10.1016/j.bmc.2007.05.053
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC nan None 10.1016/j.bmcl.2018.05.049
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC nan None 10.1016/j.ejmech.2014.09.028
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC nan None 10.1039/C3MD00366C
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC nan None 10.1128/aac.01486-07
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC100 0.2 ug ml-1 10.1016/j.bmc.2018.07.034
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC100 0.25 microg/ml 10.1016/j.ejmech.2009.09.024
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC100 0.5 uM 10.1021/acs.jnatprod.5b00266
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.0019 ug.mL-1 10.1016/j.bmcl.2017.01.004
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.0043 ug.mL-1 10.1016/j.bmcl.2017.01.004
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.035 ug.mL-1 10.1016/j.bmcl.2022.128824
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.035 ug.mL-1 10.1016/j.bmcl.2022.128871
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.06 ug.mL-1 10.1128/aac.01545-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.1 ug.mL-1 10.1021/jm030479g
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.5 ug.mL-1 10.1007/s00044-010-9322-5
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.5 ug.mL-1 10.1016/j.bmc.2021.116560
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.5 ug.mL-1 10.1021/jm100165w
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.7 ug.mL-1 10.1016/j.bmcl.2020.127351
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.7 ug.mL-1 10.1016/j.bmcl.2021.128261
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.8 ug.mL-1 10.1016/j.bmcl.2020.127351
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 0.8 ug.mL-1 10.1016/j.bmcl.2021.128261
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 1.0 ug.mL-1 10.1021/jm100568q
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 4.21 ug.mL-1 10.1007/s00044-010-9322-5
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 21.0 nM 10.1021/acs.jmedchem.2c00266
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 40.0 ug.mL-1 10.1016/j.bmcl.2022.128824
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 40.0 ug.mL-1 10.1016/j.bmcl.2022.128871
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 128.0 ug.mL-1 10.1128/aac.01545-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 200.0 nM 10.1016/j.bmc.2021.116506
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC50 240.0 nM 10.1021/acs.jmedchem.2c00266
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC70 0.08 uM 10.1016/j.bmcl.2017.07.067
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>80 0.003 ug ml-1 10.1021/jm500833f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>80 0.004 uM 10.1021/acs.jmedchem.6b01358
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>80 0.007 ug ml-1 10.1021/jm500833f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>80 0.008 uM 10.1021/acs.jmedchem.6b01358
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>80 0.016 uM 10.1021/acs.jmedchem.6b01358
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>80 0.04 uM 10.1039/C5MD00589B
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>80 1.2 uM 10.1039/C5MD00589B
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>80 16.0 ug ml-1 10.1021/jm500833f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC80 26.6 nM 10.1021/jm5003606
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC80 180.0 nM 10.1021/jm5003606
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=<90 0.0625 ug ml-1 10.1016/j.ejmech.2021.113202
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=<90 0.125 ug ml-1 10.1021/acs.jmedchem.7b00582
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=<90 4.0 ug ml-1 10.1016/j.ejmech.2021.113202
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=<90 128.0 ug ml-1 10.1016/j.ejmech.2021.113202
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.003 ug ml-1 10.1016/j.ejmech.2016.09.030
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.008 ug ml-1 10.1021/acsmedchemlett.8b00410
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.05 ug ml-1 10.1016/j.bmcl.2015.10.027
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.05 ug ml-1 10.1016/j.ejmech.2015.09.030
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.05 uM 10.1016/j.ejmech.2015.05.048
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.057 ug ml-1 10.1021/acsmedchemlett.7b00068
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.06 ug ml-1 10.1016/j.ejmech.2020.112420
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.06 uM 10.1016/j.bmcl.2014.05.062
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.071 uM 10.1016/j.ejmech.2017.05.044
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.078 ug ml-1 10.1016/j.ejmech.2019.111595
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.084 ug ml-1 10.1016/j.ejmech.2018.03.060
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.096 ug ml-1 10.1016/j.ejmech.2018.09.042
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.11 uM 10.1016/j.bmcl.2014.05.062
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.13 uM 10.1016/j.ejmech.2015.10.024
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.152 uM 10.1016/j.ejmech.2019.01.073
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 0.5 mg/L 10.1016/j.bmcl.2015.09.072
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 2.0 ug ml-1 10.1021/acsmedchemlett.8b00410
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 10.0 uM 10.1016/j.bmc.2015.03.018
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 20.0 ug ml-1 10.1021/acsmedchemlett.7b00068
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 40.0 ug ml-1 10.1016/j.bmcl.2015.10.027
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 40.0 ug ml-1 10.1016/j.ejmech.2015.09.030
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 40.0 ug ml-1 10.1016/j.ejmech.2018.03.060
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 40.0 ug ml-1 10.1016/j.ejmech.2018.09.042
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 40.0 ug ml-1 10.1016/j.ejmech.2019.111595
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 40.0 ug ml-1 10.1021/acsmedchemlett.7b00068
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 57.0 uM 10.1016/j.ejmech.2017.05.044
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 128.0 ug ml-1 10.1016/j.ejmech.2020.112420
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 128.0 uM 10.1016/j.ejmech.2019.01.073
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC=>90 256.0 mg/L 10.1016/j.bmcl.2015.09.072
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 0.01 ug ml-1 10.1021/np400145u
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 0.02 ug ml-1 10.1021/np400145u
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 0.03 ug ml-1 10.1021/np400145u
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 0.038 uM 10.1016/j.ejmech.2018.12.071
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 0.04 ug ml-1 10.1021/np400145u
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 0.05 ug ml-1 10.1021/acs.jnatprod.8b00567
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 0.05 ug ml-1 10.1021/acsmedchemlett.6b00330
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 0.059 ug ml-1 10.1016/j.bmcl.2018.07.046
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 0.0781 ug ml-1 10.1021/acsmedchemlett.8b00177
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 0.092 uM 10.1021/acsmedchemlett.7b00106
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 0.1 ug ml-1 10.1021/np400145u
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 0.2 ug ml-1 10.1021/np400145u
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 3.3 ug ml-1 10.1021/np400145u
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 10.0 uM 10.1016/j.bmc.2015.06.047
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 27.24 uM 10.1021/acsmedchemlett.7b00106
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 40.0 ug ml-1 10.1016/j.bmcl.2018.07.046
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 40.0 ug ml-1 10.1021/acsmedchemlett.8b00177
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 40.0 uM 10.1016/j.ejmech.2018.12.071
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>90 48.6 uM 10.1021/acsmedchemlett.7b00106
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.003 ug.mL-1 10.1021/jm300123s
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.004 ug.mL-1 10.1021/acsmedchemlett.0c00381
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.005 ug.mL-1 10.1021/acs.jmedchem.1c01349
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.0173 ug.mL-1 10.1016/j.bmcl.2017.01.004
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.02 ug.mL-1 10.1016/j.bmcl.2017.01.004
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.02 ug.mL-1 10.1021/np400497f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.02 ug.mL-1 10.1038/nchembio884
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.03 ug.mL-1 10.1021/acs.jmedchem.1c01349
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.04 ug.mL-1 10.1021/np400497f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.041 ug.mL-1 10.1021/jm300123s
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.043 ug.mL-1 10.1021/acsmedchemlett.6b00077
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.048 ug.mL-1 10.1021/acsmedchemlett.6b00077
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.05 ug.mL-1 10.1016/j.bmcl.2012.05.096
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.05 ug.mL-1 10.1016/j.ejmech.2022.114404
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.05 ug.mL-1 10.1021/np400497f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.057 ug.mL-1 10.1016/j.bmcl.2022.128824
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.06 ug.mL-1 10.1021/acsmedchemlett.5b00202
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.0625 ug.mL-1 10.1016/j.bmcl.2012.09.041
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.064 ug.mL-1 10.1016/j.bmcl.2022.128871
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.08 ug.mL-1 10.1021/np400497f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.09 ug.mL-1 10.1021/np400497f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.125 ug.mL-1 10.1021/acs.jmedchem.2c01064
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.125 ug.mL-1 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.125 ug.mL-1 10.1128/aac.01545-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.13 ug.mL-1 10.1038/nchembio884
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.2 ug.mL-1 10.1016/j.ejmech.2022.114404
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.25 ug.mL-1 10.1039/C8MD00389K
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.3 ug.mL-1 10.1016/j.ejmech.2016.12.042
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.39 ug.mL-1 10.1016/j.ejmech.2017.05.057
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.39 ug.mL-1 10.1016/j.ejmech.2018.07.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.5 ug.mL-1 10.1016/j.bmc.2016.03.003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.5 ug.mL-1 10.1016/j.bmcl.2007.06.064
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.5 ug.mL-1 10.1021/acsmedchemlett.6b00077
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.5 ug.mL-1 10.1021/jm0703901
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.5 ug.mL-1 10.1021/jm070391t
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.51 ug.mL-1 10.1039/C5MD00404G
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.7 ug.mL-1 10.1016/j.bmcl.2007.06.064
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.75 ug.mL-1 10.1039/C5MD00404G
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.8 ug.mL-1 10.1016/j.bmcl.2007.06.064
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 0.8 ug.mL-1 10.1021/acsmedchemlett.6b00077
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 1.0 ug.mL-1 10.1016/j.bmc.2016.03.003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 1.47 ug.mL-1 10.1016/j.bmcl.2012.05.096
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 1.5 nM 10.1016/j.bmcl.2019.05.001
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 1.6 nM 10.1021/acs.jmedchem.5b01542
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 2.0 ug.mL-1 10.1007/s00044-010-9322-5
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 2.0 ug.mL-1 10.1021/jm300123s
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 2.91 nM 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 2.95 ug.mL-1 10.1021/acsmedchemlett.8b00410
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 3.2 nM 10.1021/acs.jmedchem.5b01542
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 3.29 ug.mL-1 10.1021/np400497f
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 4.0 ug.mL-1 10.1016/j.bmcl.2007.06.064
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 4.0 ug.mL-1 10.1016/j.bmcl.2016.06.019
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 4.5 nM 10.1016/j.ejmech.2021.113734
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 6.0 nM 10.1039/d1md00063b
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 7.0 nM 10.1016/j.bmcl.2019.126911
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 7.37 ug.mL-1 10.1007/s00044-010-9322-5
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 8.0 nM 10.1016/j.bmcl.2008.03.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 8.0 ug.mL-1 10.1016/j.ejmech.2016.12.042
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 9.0 nM 10.1021/acs.jmedchem.5b01542
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 9.0 nM 10.1039/C9MD00161A
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 10.0 nM 10.1016/j.bmcl.2021.127784
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 10.0 nM 10.1016/j.ejmech.2021.113207
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 10.0 nM 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 10.0 nM 10.1021/ml200036r
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 10.0 ug.mL-1 10.1021/acsmedchemlett.6b00077
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 13.0 nM 10.1016/j.ejmech.2022.114105
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 15.0 nM 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 15.6 nM 10.1016/j.ejmech.2019.06.069
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 18.0 nM 10.1016/j.ejmech.2019.06.069
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 19.0 nM 10.1016/j.bmcl.2019.126911
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 20.0 nM 10.1016/j.bmc.2016.12.038
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 20.0 nM 10.1016/j.ejmech.2021.113734
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 20.0 nM 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 20.0 nM 10.1021/ml200036r
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 20.0 nM 10.1039/C9MD00161A
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 21.7 nM 10.1016/j.ejmech.2019.06.069
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 23.0 nM 10.1016/j.ejmech.2022.114105
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 25.0 ug.mL-1 10.1016/j.ejmech.2016.12.042
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 25.0 ug.mL-1 10.1016/j.ejmech.2022.114404
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 28.0 nM 10.1021/acs.jnatprod.1c00198
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 30.0 nM 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 32.0 ug.mL-1 10.1016/j.ejmech.2017.05.057
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 32.0 ug.mL-1 10.1016/j.ejmech.2018.07.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 40.0 nM 10.1016/j.bmc.2012.02.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 40.0 nM 10.1016/j.ejmech.2013.09.061
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 40.0 nM 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 40.0 ug.mL-1 10.1007/s00044-011-9718-x
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 40.0 ug.mL-1 10.1016/j.bmcl.2022.128824
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 40.0 ug.mL-1 10.1016/j.bmcl.2022.128871
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 50.0 nM 10.1016/j.ejmech.2012.08.047
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 50.0 nM 10.1016/j.ejmech.2017.05.026
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 50.0 nM 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 50.0 nM 10.1021/ml200036r
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 60.0 nM 10.1007/s00044-012-9971-7
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 60.0 nM 10.1016/j.bmcl.2019.02.019
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 60.0 nM 10.1039/C8MD00480C
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 70.0 nM 10.1016/j.bmcl.2013.09.013
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 70.0 nM 10.1016/j.ejmech.2015.05.020
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 70.0 nM 10.1021/acsmedchemlett.5b00141
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 70.0 nM 10.1021/ml200036r
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 90.0 nM 10.1007/s00044-007-9073-0
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 90.0 nM 10.1016/j.bmc.2012.02.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 90.0 nM 10.1016/j.bmcl.2012.06.095
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 100.0 nM 10.1016/j.ejmech.2017.06.061
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 100.0 nM 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 100.0 nM 10.1021/acs.jnatprod.5b00266
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 100.0 nM 10.1021/jm900513a
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 120.0 nM 10.1016/j.ejmech.2013.06.010
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 128.0 ug.mL-1 10.1016/j.bmcl.2016.06.019
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 128.0 ug.mL-1 10.1128/aac.01545-09
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 130.0 nM 10.1016/j.bmcl.2011.08.054
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 130.0 nM 10.1021/jm201716n
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 150.0 nM 10.1021/np900806j
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 190.0 nM 10.1016/j.ejmech.2017.05.026
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 200.0 nM 10.1016/j.bmc.2012.02.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 200.0 nM 10.1021/ml200036r
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 210.0 nM 10.1016/j.ejmech.2015.05.048
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 210.0 nM 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 300.0 nM 10.1039/d2md00155a
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 460.0 nM 10.1021/jm201716n
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 500.0 nM 10.1016/j.ejmech.2016.07.039
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 610.0 nM 10.1016/j.bmcl.2012.06.095
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 610.0 nM 10.1021/acs.jnatprod.5b01033
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 760.0 nM 10.1016/j.ejmech.2020.112821
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 780.0 nM 10.1021/ml200036r
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 800.0 nM 10.1021/ml200036r
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 910.0 nM 10.1016/j.bmcl.2019.03.020
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 910.0 nM 10.1016/j.ejmech.2017.03.065
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 980.0 nM 10.1016/j.ejmech.2017.03.065
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 1000.0 nM 10.1016/j.ejmech.2017.05.026
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 1000.0 nM 10.1021/acs.jmedchem.7b01332
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 1000.0 nM 10.1021/ml200036r
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 1900.0 nM 10.1016/j.bmcl.2011.08.054
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 1900.0 nM 10.1021/jm900513a
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 1930.0 nM 10.1016/j.ejmech.2012.08.047
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 2400.0 nM 10.1021/acsmedchemlett.5b00141
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 2600.0 nM 10.1016/j.bmc.2012.02.025
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 2600.0 nM 10.1016/j.bmcl.2014.05.062
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 2600.0 nM 10.1021/ml200036r
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 8000.0 nM 10.1016/j.ejmech.2021.113734
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 38900.0 nM 10.1016/j.ejmech.2015.05.020
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 155500.0 nM 10.1021/acsmedchemlett.5b00141
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 311070.0 nM 10.1021/acsmedchemlett.5b00141
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 311100.0 nM 10.1016/j.ejmech.2015.05.020
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 nan None 10.1016/j.ejmech.2016.07.039
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 nan None 10.1021/acs.jmedchem.5b01542
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC90 nan None 10.1021/acs.jnatprod.5b01033
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC95 0.03 ug ml-1 10.1016/j.bmc.2017.07.034
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC95 0.25 ug ml-1 10.1016/j.bmcl.2011.06.074
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC97 0.015 ug ml-1 10.1016/j.bmcl.2011.06.074
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC98 40.0 ug ml-1 10.1016/j.ejmech.2017.06.051
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC98 40.0 ug ml-1 10.1016/j.ejmech.2018.03.016
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>99 0.012 uM 10.1016/j.bmc.2015.10.021
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>99 0.25 uM 10.1016/j.bmc.2017.08.010
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>99 0.25 uM 10.1016/j.ejmech.2017.02.058
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>99 0.25 uM 10.1021/acs.jmedchem.9b00912
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>99 8.0 uM 10.1016/j.bmc.2017.08.010
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>99 8.0 uM 10.1021/acs.jmedchem.5b00608
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC>99 8.0 uM 10.1021/acs.jmedchem.9b00912
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.00167 uM 10.1016/j.bmcl.2019.05.001
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.003 uM 10.1021/ml400088y
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.004 uM 10.1016/j.bmc.2014.10.007
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.00482 uM 10.1021/acs.jmedchem.0c01833
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.005 uM 10.1016/j.bmc.2020.115530
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.007 uM 10.1016/j.ejmech.2020.112772
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.0083 uM 10.1016/j.bmcl.2014.05.022
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.012 uM 10.1021/acs.jmedchem.7b01347
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.013 uM 10.1016/j.bmc.2014.10.007
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.02 ug ml-1 10.1016/j.bmcl.2013.10.016
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.02 ug ml-1 10.1016/j.ejmech.2014.01.005
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.037 uM 10.1021/acs.jmedchem.2c00266
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.041 uM 10.1021/acs.jmedchem.2c00266
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.125 ug ml-1 10.1016/j.bmc.2013.06.027
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.14 uM 10.1016/j.ejmech.2013.10.055
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.19 uM 10.1021/jm401735w
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.197 ug ml-1 10.1016/j.bmcl.2016.04.012
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.197 ug ml-1 10.1016/j.bmcl.2016.10.082
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.197 ug ml-1 10.1039/C4MD00224E
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.2 ug ml-1 10.1016/j.ejmech.2014.07.100
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.2 ug ml-1 10.1016/j.ejmech.2015.01.013
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.2 ug ml-1 10.1016/j.ejmech.2015.02.034
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.25 ug ml-1 10.1016/j.ejmech.2014.03.085
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.25 ug ml-1 10.1016/j.ejmech.2019.07.019
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 0.5 uM 10.1016/j.bmcl.2017.02.021
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 1.0 ug ml-1 10.1016/j.bmc.2012.09.019
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 1.0 ug ml-1 10.1016/j.bmc.2013.07.003
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 40.0 ug ml-1 10.1007/s00044-011-9942-4
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 40.0 ug ml-1 10.1007/s00044-012-0273-x
Mycobacterium tuberculosis Mycobacterium tuberculosis MIC99 nan None 10.1016/j.bmc.2013.07.003
Mycobacterium tuberculosis Mycobacterium tuberculosis PAE 5.2 day 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis PAE 12.0 day 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis PAE 12.9 day 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis PAE 19.3 day 10.1128/aac.01533-06
Mycobacterium tuberculosis Mycobacterium tuberculosis Ratio 0.5 None 10.1021/jm500833f
Mycobacterium tuberculosis Mycobacterium tuberculosis Ratio 1.0 None 10.1016/j.bmcl.2008.03.025
Mycobacterium tuberculosis Mycobacterium tuberculosis Ratio 4.0 None 10.1128/aac.00550-09
Mycobacterium tuberculosis Mycobacterium tuberculosis Ratio 15.6 None 10.1016/j.bmcl.2016.03.066
Mycobacterium tuberculosis Mycobacterium tuberculosis Ratio 65.0 None 10.1016/j.bmcl.2009.07.147
Mycobacterium tuberculosis Mycobacterium tuberculosis Ratio 650.0 None 10.1016/j.bmcl.2009.07.147
Mycobacterium tuberculosis Mycobacterium tuberculosis Ratio nan None 10.1016/j.ejmech.2018.02.067
Mycobacterium tuberculosis Mycobacterium tuberculosis Selectivity Index 0.2 None 10.1021/acs.jmedchem.1c01349
Mycobacterium tuberculosis Mycobacterium tuberculosis Selectivity ratio 4.0 None 10.1021/acs.jmedchem.6b01358
Mycobacterium tuberculosis Mycobacterium tuberculosis Selectivity ratio 7.35 None 10.1016/j.bmc.2018.07.034
Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC50 1.53 nM 10.1021/acs.jmedchem.1c01407
Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC50 10.0 nM 10.1016/j.ejmech.2020.112908
Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC50 2900.0 nM 10.1016/j.ejmech.2020.112908
Mycobacterium tuberculosis H37Rv Mycobacterium tuberculosis H37Rv MIC90 8000.0 nM 10.1016/j.ejmech.2021.113734
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) Cytochrome bc1 complex cytochrome b subunit Inhibition nan % 10.1021/acs.jmedchem.8b00172
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) DNA gyrase subunit A/DNA gyrase subunit B IC50 50000.0 nM 10.1016/j.bmc.2016.01.011
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) DNA gyrase subunit A/DNA gyrase subunit B IC50 nan None 10.1016/j.bmc.2014.10.016
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) DNA gyrase subunit A/DNA gyrase subunit B IC50 nan None 10.1016/j.bmc.2015.03.004
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) DNA gyrase subunit A/DNA gyrase subunit B IC50 nan None 10.1016/j.ejmech.2015.06.032
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) DNA gyrase subunit A/DNA gyrase subunit B IC50 nan None 10.1016/j.ejmech.2016.08.034
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) DNA gyrase subunit A/DNA gyrase subunit B IC50 nan None 10.1021/ml500531p
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) FAD-dependent decaprenylphosphoryl-beta-D-ribofuranose 2-oxidase MIC 0.015 ug.mL-1 10.1021/acs.jmedchem.1c00263
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) Polyketide synthase Pks13 MIC=<90 0.0625 ug ml-1 10.1021/acs.jmedchem.9b00010
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) Polyketide synthase Pks13 MIC=<90 0.125 ug ml-1 10.1021/acs.jmedchem.9b00010
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) Polyketide synthase Pks13 MIC=<90 4.0 ug ml-1 10.1021/acs.jmedchem.9b00010
Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) Polyketide synthase Pks13 MIC=<90 128.0 ug ml-1 10.1021/acs.jmedchem.9b00010
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis Activity 3.0 log10CFU/ml 10.1016/j.ejmech.2021.113932
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis Activity nan None 10.1016/j.ejmech.2016.07.068
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis IC50 10.0 nM None
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis IC50 910.0 nM 10.1016/j.bmcl.2019.03.020
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis Inhibition 100.0 % 10.1016/j.ejmech.2022.114831
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis Inhibition 100.0 % 10.1021/jm058167w
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis MIC 0.016 ug.mL-1 10.1128/aac.01302-08
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis MIC 0.031 ug.mL-1 10.1128/aac.01302-08
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis MIC 0.063 ug.mL-1 10.1128/aac.01302-08
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis MIC 0.45 ug.mL-1 10.1016/j.ejmech.2020.113102
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis MIC 0.81 ug.mL-1 10.1016/j.ejmech.2020.113102
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis MIC 350.0 nM 10.1016/j.ejmech.2021.113932
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis MIC nan None 10.1016/j.bmcl.2019.06.055
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis MIC90 1.0 ug.mL-1 10.1021/jm058167w
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis MIC90 20.0 nM 10.1016/j.ejmech.2016.07.068
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis MIC90 980.0 nM 10.1016/j.bmcl.2019.03.020
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis MIC90 2200.0 nM 10.1016/j.bmcl.2019.126671
Mycobacterium tuberculosis variant bovis Mycobacterium tuberculosis variant bovis MIC>99 0.25 ug ml-1 10.1016/j.ejmech.2014.07.066
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG Activity 25.0 % 10.1021/acs.jmedchem.8b00832
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG IC50 0.0012 ug.mL-1 10.1016/j.bmcl.2016.02.043
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG IC50 0.0015 ug.mL-1 10.1016/j.bmcl.2016.02.043
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG IC50 0.0016 ug.mL-1 10.1016/j.bmcl.2015.11.071
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG IC50 0.0027 ug.mL-1 10.1016/j.bmcl.2016.05.093
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG IC50 0.003 ug.mL-1 10.1016/j.bmcl.2016.05.093
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 0.0002 ug.mL-1 10.1128/aac.00550-09
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 0.0004 ug.mL-1 10.1128/aac.00550-09
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 0.0008 ug.mL-1 10.1128/aac.00550-09
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 0.0016 ug.mL-1 10.1128/aac.00550-09
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 0.0032 ug.mL-1 10.1128/aac.00550-09
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 0.015 ug.mL-1 10.1016/j.bmcl.2016.02.043
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 0.017 ug.mL-1 10.1016/j.bmcl.2016.02.043
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 0.041 ug.mL-1 10.1016/j.bmcl.2015.11.071
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 0.05 ug.mL-1 10.1016/j.bmcl.2016.05.093
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 0.08 ug.mL-1 10.1016/j.bmcl.2016.05.093
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 0.1 ug.mL-1 10.1021/jm070638m
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 4.0 nM 10.1016/j.bmcl.2014.05.062
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 20.0 nM 10.1021/ml5003458
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC 60.7 nM 10.1039/C3MD00251A
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC90 0.004 ug.mL-1 10.1021/acsmedchemlett.6b00077
Mycobacterium tuberculosis variant bovis BCG Mycobacterium tuberculosis variant bovis BCG MIC90 0.0042 ug.mL-1 10.1021/acsmedchemlett.6b00077
Mycobacterium tuberculosis variant microti Mycobacterium tuberculosis variant microti MIC 30380.0 nM 10.1016/j.bmcl.2008.12.088
Mycobacterium ulcerans Mycobacterium ulcerans Activity nan None 10.1128/aac.00730-07
Mycobacterium ulcerans Mycobacterium ulcerans log10cfu 0.46 None 10.1128/aac.00730-07
Mycobacterium ulcerans Mycobacterium ulcerans log10cfu 1.52 None 10.1128/aac.00730-07
Mycobacterium ulcerans Mycobacterium ulcerans Log10 cfu 4.13 None 10.1128/aac.00821-06
Mycobacterium ulcerans Mycobacterium ulcerans MIC 0.016 ug.mL-1 10.1128/aac.00400-10
Mycobacterium ulcerans Mycobacterium ulcerans MIC 0.03 ug.mL-1 10.1128/aac.00400-10
Mycobacterium ulcerans Mycobacterium ulcerans MIC 0.06 ug.mL-1 10.1128/aac.00400-10
Mycobacterium ulcerans Mycobacterium ulcerans MIC 0.13 ug.mL-1 10.1128/aac.00400-10
Mycobacterium ulcerans Mycobacterium ulcerans MIC 0.5 ug.mL-1 10.1128/aac.00400-10
Mycobacterium ulcerans Mycobacterium ulcerans MIC 2.0 ug.mL-1 10.1128/aac.00730-07
Mycobacterium xenopi Mycobacterium xenopi MIC 1.0 ug.mL-1 10.1021/jm00167a029
Mycobacteroides abscessus Mycobacteroides abscessus DIZ nan None 10.1016/j.bmcl.2019.07.001
Mycobacteroides abscessus Mycobacteroides abscessus IZ 0.0 mm 10.1016/j.bmcl.2019.07.001
Mycobacteroides abscessus Mycobacteroides abscessus MIC 128.0 ug.mL-1 10.1128/aac.01545-09
Mycobacteroides abscessus Mycobacteroides abscessus MIC 4000.0 nM 10.1021/acs.jnatprod.9b01095
Mycobacteroides abscessus Mycobacteroides abscessus MIC 162000.0 nM 10.1016/j.bmcl.2014.05.062
Mycobacteroides abscessus Mycobacteroides abscessus MIC nan None 10.1016/j.bmc.2022.116777
Mycobacteroides abscessus Mycobacteroides abscessus MIC nan None 10.1016/j.ejmech.2020.112996
Mycobacteroides abscessus Mycobacteroides abscessus MIC50 128.0 ug.mL-1 10.1128/aac.01545-09
Mycobacteroides abscessus Mycobacteroides abscessus MIC90 128.0 ug.mL-1 10.1128/aac.01545-09
Mycobacteroides abscessus Mycobacteroides abscessus MIC90 162300.0 nM 10.1021/ml200036r
Mycobacteroides chelonae Mycobacteroides chelonae MIC 0.125 ug.mL-1 10.1016/j.ejmech.2013.12.037
Mycobacteroides chelonae Mycobacteroides chelonae MIC 5.0 ug.mL-1 10.1128/aac.00590-09
Mycobacteroides chelonae Mycobacteroides chelonae MIC 25.0 ug.mL-1 10.1128/aac.00590-09
Mycobacteroides chelonae Mycobacteroides chelonae MIC 32.0 ug.mL-1 10.1016/j.bmc.2013.10.011
Mycobacteroides chelonae Mycobacteroides chelonae MIC 64.0 ug.mL-1 10.1016/j.bmcl.2019.07.001
Mycobacteroides chelonae Mycobacteroides chelonae MIC 100.0 ug.mL-1 10.1128/aac.00590-09
Mycobacteroides chelonae Mycobacteroides chelonae MIC 128.0 ug.mL-1 10.1128/aac.01545-09
Mycobacteroides chelonae Mycobacteroides chelonae MIC 500.0 ug.mL-1 10.1128/aac.00590-09
Mycobacteroides chelonae Mycobacteroides chelonae MIC 100000.0 nM 10.1016/j.bmcl.2014.05.062
Mycobacteroides chelonae Mycobacteroides chelonae MIC nan None 10.1016/j.bmc.2010.05.016
Mycobacteroides chelonae Mycobacteroides chelonae MIC nan None 10.1016/j.bmc.2022.116777
Mycobacteroides chelonae Mycobacteroides chelonae MIC nan None 10.1016/j.ejmech.2020.112996
Mycobacteroides chelonae Mycobacteroides chelonae MIC50 128.0 ug.mL-1 10.1128/aac.01545-09
Mycobacteroides chelonae Mycobacteroides chelonae MIC90 128.0 ug.mL-1 10.1128/aac.01545-09
Mycobacteroides chelonae Mycobacteroides chelonae MIC90 150000.0 nM 10.1021/ml200036r
Mycolicibacterium aurum Mycolicibacterium aurum MIC 0.78 ug.mL-1 10.1021/jm070638m
Mycolicibacterium aurum Mycolicibacterium aurum MIC 2.0 ug.mL-1 10.1021/acs.jnatprod.9b01015
Mycolicibacterium aurum Mycolicibacterium aurum MIC 470.0 nM 10.1016/j.ejmech.2019.111578
Mycolicibacterium diernhoferi Mycolicibacterium diernhoferi MIC 4.0 ug.mL-1 10.1021/np2006555
Mycolicibacterium flavescens Mycolicibacterium flavescens MIC 0.25 ug.mL-1 10.1021/jm00167a029
Mycolicibacterium flavescens Mycolicibacterium flavescens MIC 128.0 ug.mL-1 10.1021/jm00167a029
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 0.25 ug.mL-1 10.1016/s0960-894x(01)00283-9
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 0.5 ug.mL-1 10.1016/j.ejmech.2013.12.037
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 1.0 ug.mL-1 10.1021/jm00167a029
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 1.0 ug.mL-1 10.1128/aac.01545-09
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 1.5 ug.mL-1 10.1007/s00044-012-0451-x
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 1.5 ug.mL-1 10.1016/j.bmcl.2009.12.045
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 1.5 ug.mL-1 10.1016/j.bmcl.2013.06.072
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 1.5 ug.mL-1 10.1016/j.ejmech.2011.03.039
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 1.5 ug.mL-1 10.1016/j.ejmech.2011.07.033
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 1.5 ug.mL-1 10.1016/j.ejmech.2011.07.049
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 1.5 ug.mL-1 10.1016/j.ejmech.2011.08.014
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 1.5 ug.mL-1 10.1016/j.ejmech.2012.01.008
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 1.5 ug.mL-1 10.1016/j.ejmech.2013.11.002
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 2.0 ug.mL-1 10.1021/jm00167a029
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 4.0 ug.mL-1 10.1021/jm00167a029
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 25.0 ug.mL-1 10.1021/jm070638m
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 32.0 ug.mL-1 10.1016/j.bmc.2013.10.011
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 32.0 ug.mL-1 10.1021/jm00167a029
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 64.0 ug.mL-1 10.1016/j.bmcl.2019.07.001
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 64.0 ug.mL-1 10.1021/jm00167a029
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 128.0 ug.mL-1 10.1021/jm00167a029
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC 1890.0 nM 10.1016/j.bmcl.2008.12.088
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC nan None 10.1016/j.bmc.2010.05.016
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC nan None 10.1016/j.bmc.2022.116777
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC nan None 10.1016/j.ejmech.2020.112996
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC50 32.0 ug.mL-1 10.1128/aac.01545-09
Mycolicibacterium fortuitum Mycolicibacterium fortuitum MIC90 64.0 ug.mL-1 10.1128/aac.01545-09
Mycolicibacterium phlei Mycolicibacterium phlei DIZ nan None 10.1007/s00044-013-0487-6
Mycolicibacterium phlei Mycolicibacterium phlei IZ 25.0 mm 10.1016/j.bmc.2007.09.025
Mycolicibacterium phlei Mycolicibacterium phlei log(1/C) 6.48 None 10.1021/jm00210a025
Mycolicibacterium phlei Mycolicibacterium phlei MBC 0.06 ug ml-1 10.1021/acs.jnatprod.2c00065
Mycolicibacterium phlei Mycolicibacterium phlei MIC 0.03 ug.mL-1 10.1021/acs.jnatprod.2c00065
Mycolicibacterium phlei Mycolicibacterium phlei MIC 0.032 ug.mL-1 10.1021/jm00167a029
Mycolicibacterium phlei Mycolicibacterium phlei MIC 0.25 ug.mL-1 10.1021/jm00167a029
Mycolicibacterium phlei Mycolicibacterium phlei MIC 0.27 ug.mL-1 10.1021/jm00210a025
Mycolicibacterium phlei Mycolicibacterium phlei MIC 8.0 ug.mL-1 10.1021/jm00167a029
Mycolicibacterium phlei Mycolicibacterium phlei MIC 40.0 ug.mL-1 10.1007/s00044-013-0487-6
Mycolicibacterium phlei Mycolicibacterium phlei MIC 30380.0 nM 10.1016/j.bmcl.2008.12.088
Mycolicibacterium smegmatis Mycolicibacterium smegmatis Activity 32.4 % 10.1016/j.ejmech.2016.07.068
Mycolicibacterium smegmatis Mycolicibacterium smegmatis Activity 66.5 % 10.1016/j.ejmech.2016.07.068
Mycolicibacterium smegmatis Mycolicibacterium smegmatis Activity 95.6 % 10.1016/j.ejmech.2016.07.068
Mycolicibacterium smegmatis Mycolicibacterium smegmatis Activity 123.4 % 10.1016/j.ejmech.2016.07.068
Mycolicibacterium smegmatis Mycolicibacterium smegmatis Activity nan None 10.1016/j.ejmech.2016.07.068
Mycolicibacterium smegmatis Mycolicibacterium smegmatis Activity nan None 10.1016/j.ejmech.2019.05.081
Mycolicibacterium smegmatis Mycolicibacterium smegmatis DIZ nan None 10.1007/s00044-013-0487-6
Mycolicibacterium smegmatis Mycolicibacterium smegmatis FICI 0.5 None 10.1016/j.bmc.2014.06.012
Mycolicibacterium smegmatis Mycolicibacterium smegmatis FICI 0.63 None 10.1016/j.bmc.2014.06.012
Mycolicibacterium smegmatis Mycolicibacterium smegmatis FICI 1.0 None 10.1016/j.bmc.2014.06.012
Mycolicibacterium smegmatis Mycolicibacterium smegmatis GI50 1.04 ug.mL-1 10.1016/j.ejmech.2014.02.042
Mycolicibacterium smegmatis Mycolicibacterium smegmatis GI50 1220.0 nM 10.1016/j.ejmech.2014.06.075
Mycolicibacterium smegmatis Mycolicibacterium smegmatis IC50 1870.0 nM 10.1016/j.bmcl.2015.02.052
Mycolicibacterium smegmatis Mycolicibacterium smegmatis IC50 3110.0 nM 10.1128/aac.00803-09
Mycolicibacterium smegmatis Mycolicibacterium smegmatis IC50 4360.0 nM 10.1128/aac.00803-09
Mycolicibacterium smegmatis Mycolicibacterium smegmatis IC90 0.2 ug.mL-1 10.1021/np400002p
Mycolicibacterium smegmatis Mycolicibacterium smegmatis IZ 30.0 mm 10.1016/j.bmc.2007.09.025
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MBC 8.0 ug ml-1 10.1021/acs.jnatprod.2c00065
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MBC 25.0 ug ml-1 10.1016/j.bmc.2018.07.034
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MBC 130.0 ug ml-1 10.1016/j.bmc.2007.09.025
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 0.1 ug.mL-1 10.1021/acs.jnatprod.1c00812
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 0.5 ug.mL-1 10.1016/j.bmcl.2006.10.016
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 0.5 ug.mL-1 10.1039/d2md00260d
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 0.5 ug.mL-1 10.1126/science.1106753
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 0.78 ug.mL-1 10.1039/C8MD00056E
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2014.08.066
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.5 ug.mL-1 10.1007/s00044-012-0451-x
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.5 ug.mL-1 10.1016/j.bmcl.2009.12.045
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.5 ug.mL-1 10.1016/j.bmcl.2013.06.072
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.5 ug.mL-1 10.1016/j.ejmech.2011.03.039
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.5 ug.mL-1 10.1016/j.ejmech.2011.07.033
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.5 ug.mL-1 10.1016/j.ejmech.2011.07.049
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.5 ug.mL-1 10.1016/j.ejmech.2011.08.014
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.5 ug.mL-1 10.1016/j.ejmech.2012.01.008
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.5 ug.mL-1 10.1016/j.ejmech.2013.11.002
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.5 ug.mL-1 10.1016/j.ejmech.2020.112835
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.56 ug.mL-1 10.1016/j.bmcl.2009.09.095
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1.75 ug.mL-1 10.1016/j.ejmech.2016.07.058
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 2.15 ug.mL-1 10.1016/j.bmcl.2015.05.044
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 4.0 ug.mL-1 10.1021/acs.jmedchem.2c00972
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 4.0 ug.mL-1 10.1021/np2006555
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 4.0 ug.mL-1 10.1128/aac.00012-09
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 8.0 ug.mL-1 10.1016/j.ejmech.2010.11.020
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 8.0 ug.mL-1 10.1021/acs.jnatprod.2c00065
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 12.5 ug.mL-1 10.1016/j.ejmech.2019.111578
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 16.0 ug.mL-1 10.1016/j.bmcl.2018.05.049
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 25.0 ug.mL-1 10.1021/jm070638m
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 32.0 ug.mL-1 10.1016/j.bmc.2012.02.039
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 32.0 ug.mL-1 10.1016/j.bmcl.2006.10.016
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 32.0 ug.mL-1 10.1016/j.bmcl.2019.07.001
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 32.0 ug.mL-1 10.1016/s0960-894x(99)00510-7
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 32.0 ug.mL-1 10.1021/jm0602662
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 32.0 ug.mL-1 10.1021/jm701560p
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 32.0 ug.mL-1 10.1128/aac.00012-09
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 55.0 ug.mL-1 10.1016/j.ejmech.2010.05.017
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 64.0 ug.mL-1 10.1016/j.bmc.2010.05.016
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 64.0 ug.mL-1 10.1016/j.bmc.2013.10.011
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 64.0 ug.mL-1 10.1021/jm00167a029
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 100.0 ug.mL-1 10.1039/C7MD00350A
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 140.0 ug.mL-1 10.1016/j.bmc.2007.09.025
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 350.0 nM 10.1016/j.ejmech.2021.113932
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 480.0 ug.mL-1 10.1007/s00044-013-0487-6
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 1890.0 nM 10.1016/j.bmcl.2008.12.088
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 3790.0 nM 10.1016/j.ejmech.2010.11.023
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 5000.0 nM 10.1016/j.ejmech.2021.113212
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 6250.0 nM 10.1128/aac.00803-09
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 10000.0 nM 10.1016/j.ejmech.2021.113212
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 16700.0 nM 10.1016/j.bmcl.2013.11.024
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 22600.0 nM 10.1016/j.bmcl.2008.12.088
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC 100000.0 ug.mL-1 10.1039/C7MD00366H
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC nan ug.mL-1 10.1016/s0960-894x(03)00597-3
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC nan None 10.1016/j.bmcl.2012.08.003
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC nan None 10.1016/j.ejmech.2009.09.001
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC nan None 10.1128/aac.00012-09
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC100 25.0 ug ml-1 10.1016/j.bmc.2018.07.034
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC50 0.57 ug.mL-1 10.1016/j.bmcl.2022.128692
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC50 0.63 ug.mL-1 10.1016/j.bmcl.2022.128692
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC50 0.76 ug.mL-1 10.1016/j.bmcl.2022.128692
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC50 2.08 ug.mL-1 10.1016/j.ejmech.2013.10.034
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC>90 0.3 ug ml-1 10.1021/np400145u
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC90 0.76 ug.mL-1 10.1016/j.bmcl.2022.128692
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC90 2.15 ug.mL-1 10.1016/j.ejmech.2013.10.034
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC90 2.4 ug.mL-1 10.1016/j.bmcl.2022.128692
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC90 2.83 ug.mL-1 10.1016/j.bmcl.2022.128692
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC90 8.0 ug.mL-1 10.1021/acs.jmedchem.1c01349
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC90 8.2 ug.mL-1 10.1038/nchembio884
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC90 2500.0 nM 10.1016/j.ejmech.2016.07.068
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC90 10000.0 nM 10.1016/j.ejmech.2017.05.026
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC90 162300.0 nM 10.1021/ml200036r
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC99 0.2 uM 10.1016/j.bmc.2014.06.012
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC99 0.32 uM 10.1016/j.bmc.2014.06.012
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC99 0.63 uM 10.1016/j.bmc.2014.06.012
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC99 1.26 uM 10.1039/C3MD00387F
Mycolicibacterium smegmatis Mycolicibacterium smegmatis MIC99 2.53 uM 10.1016/j.bmc.2014.06.012
Mycolicibacterium smegmatis Mycolicibacterium smegmatis Ratio 0.126 None 10.1016/j.bmc.2014.06.012
Mycolicibacterium smegmatis Mycolicibacterium smegmatis Ratio 0.254 None 10.1016/j.bmc.2014.06.012
Mycolicibacterium smegmatis Mycolicibacterium smegmatis Ratio 0.5 None 10.1016/j.bmc.2014.06.012
Mycolicibacterium smegmatis Mycolicibacterium smegmatis Ratio 64.0 None 10.1016/j.bmcl.2006.10.016
Mycolicibacterium smegmatis Mycolicibacterium smegmatis Selectivity Index 1.0 None 10.1021/acs.jmedchem.1c01349
Mycolicibacterium vaccae Mycolicibacterium vaccae MIC 3800.0 nM 10.1016/j.bmcl.2008.12.088
Neisseria gonorrhoeae Neisseria gonorrhoeae MIC 0.125 ug.mL-1 10.1021/jm00167a029
Neisseria meningitidis Neisseria meningitidis Activity 0.0 % 10.1128/aac.00994-08
Neisseria meningitidis Neisseria meningitidis Activity 0.0 % 10.1128/aac.01812-09
Neisseria meningitidis Neisseria meningitidis Activity 1.0 % 10.1128/aac.00994-08
Neisseria meningitidis Neisseria meningitidis Activity 99.0 % 10.1128/aac.00994-08
Neisseria meningitidis Neisseria meningitidis Activity 100.0 % 10.1128/aac.01812-09
Neisseria meningitidis Neisseria meningitidis MIC 1.5e-05 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 2.4e-05 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 2.5e-05 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 2.9e-05 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 3.4e-05 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 5.7e-05 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 6.1e-05 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 6.5e-05 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 8.9e-05 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 0.000125 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 0.00015 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 0.000225 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 0.002 ug.mL-1 10.1128/aac.00994-08
Neisseria meningitidis Neisseria meningitidis MIC 0.008 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 0.015 ug.mL-1 10.1128/aac.01812-09
Neisseria meningitidis Neisseria meningitidis MIC 0.032 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC 0.256 ug.mL-1 10.1128/aac.00315-10
Neisseria meningitidis Neisseria meningitidis MIC50 0.015 ug.mL-1 10.1128/aac.01812-09
Neisseria meningitidis Neisseria meningitidis MIC50 0.064 ug.mL-1 10.1128/aac.00994-08
Neisseria meningitidis Neisseria meningitidis MIC90 0.03 ug.mL-1 10.1128/aac.01812-09
Neisseria meningitidis Neisseria meningitidis MIC90 0.125 ug.mL-1 10.1128/aac.00994-08
Oryctolagus cuniculus Angiotensin-converting enzyme IC50 nan None None
Oryctolagus cuniculus Angiotensin-converting enzyme Ki nan None None
Oryctolagus cuniculus Arachidonate 15-lipoxygenase IC50 2949.0 nM None
Oryctolagus cuniculus Arachidonate 15-lipoxygenase Ki nan None None
Oryctolagus cuniculus Oryctolagus cuniculus Activity 8.2 % 10.1128/aac.00367-09
Oryctolagus cuniculus Oryctolagus cuniculus Activity 411.7 /uL 10.1128/aac.00367-09
Oryctolagus cuniculus Oryctolagus cuniculus Activity nan None 10.1128/aac.00367-09
Oryctolagus cuniculus Oryctolagus cuniculus AUC 40280.0 ng.hr.mL-1 10.1128/aac.00367-09
Oryctolagus cuniculus Oryctolagus cuniculus Cmax 20195.64 nM 10.1128/aac.00367-09
Oryctolagus cuniculus Oryctolagus cuniculus T1/2 3.38 hr 10.1128/aac.00367-09
Papio hamadryas Plasma PPB 27.32 % 10.1021/jm901858n
Pasteurella multocida Pasteurella multocida MIC 0.1 ug.mL-1 10.1128/aac.00245-08
Pasteurella multocida Pasteurella multocida MIC 0.2 ug.mL-1 10.1128/aac.00245-08
Pasteurella multocida Pasteurella multocida MIC 0.78 ug.mL-1 10.1128/aac.00245-08
Pasteurella multocida Pasteurella multocida MIC 50.0 ug.mL-1 10.1128/aac.00245-08
Pasteurella multocida Pasteurella multocida Ratio 64.0 None 10.1128/aac.00245-08
Pasteurella multocida Pasteurella multocida Ratio 512.0 None 10.1128/aac.00245-08
Peptococcus niger Peptococcus niger MIC 0.004 ug.mL-1 10.1021/acs.jmedchem.1c02045
Peptoniphilus asaccharolyticus Peptoniphilus asaccharolyticus MIC 0.004 ug.mL-1 10.1021/acs.jmedchem.1c02045
Peptostreptococcus anaerobius Peptostreptococcus anaerobius MIC 0.004 ug.mL-1 10.1021/acs.jmedchem.1c02045
Peptostreptococcus sp. Peptostreptococcus sp. MIC 1.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Phocaeicola vulgatus Phocaeicola vulgatus MIC 0.25 ug.mL-1 10.1021/acs.jmedchem.1c02045
Plasmodium falciparum Plasmodium falciparum Activity 10.0 % 10.1128/aac.00808-06
Plasmodium falciparum Plasmodium falciparum Activity 13.0 % 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum Activity 14.0 % 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum Activity 15.0 % 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum Activity 16.0 % 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum Activity 25.0 % 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum Activity 36.0 % 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum Activity 49.0 % 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum Activity 65.0 % 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum Activity 93.0 % 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum Activity nan None 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum Activity nan None 10.1128/aac.00808-06
Plasmodium falciparum Plasmodium falciparum IC50 190.0 nM 10.1128/aac.00808-06
Plasmodium falciparum Plasmodium falciparum IC50 274.0 nM 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum IC50 528.0 nM 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum IC50 1000.0 nM 10.1016/j.bmc.2010.01.068
Plasmodium falciparum Plasmodium falciparum IC50 2830.0 nM 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum IC50 2990.0 nM 10.1128/aac.00527-07
Plasmodium falciparum Plasmodium falciparum IC50 4200.0 nM 10.1128/aac.00808-06
Plasmodium falciparum Plasmodium falciparum IC50 nan None 10.1021/np020592u
Plasmodium falciparum Plasmodium falciparum IC50 nan None 10.1021/np0400095
Plasmodium falciparum Plasmodium falciparum IC50 nan None 10.1021/np0601399
Plasmodium falciparum Plasmodium falciparum MIC 0.0023 ug.mL-1 10.1021/np0602012
Plasmodium falciparum Plasmodium falciparum MIC90 2000.0 nM 10.1128/aac.00808-06
Plasmodium falciparum Plasmodium falciparum MIC90 109600.0 nM 10.1128/aac.00808-06
Plasmodium falciparum Plasmodium falciparum Potency 1168.9 nM None
Plasmodium falciparum Plasmodium falciparum Potency 1852.6 nM None
Plasmodium yoelii Plasmodium yoelii IC50 22200.0 nM 10.1021/jm201095h
Porphyromonas asaccharolytica Porphyromonas asaccharolytica MIC 0.004 ug.mL-1 10.1021/acs.jmedchem.1c02045
Prevotella bivia Prevotella bivia MIC 0.004 ug.mL-1 10.1021/acs.jmedchem.1c02045
Prevotella bivia Prevotella bivia MIC 0.06 ug.mL-1 10.1021/acs.jmedchem.1c02045
Prevotella bivia Prevotella bivia MIC 0.5 ug.mL-1 10.1021/acs.jmedchem.1c02045
Prevotella disiens Prevotella disiens MIC 0.12 ug.mL-1 10.1021/acs.jmedchem.1c02045
Prevotella disiens Prevotella disiens MIC 0.5 ug.mL-1 10.1021/acs.jmedchem.1c02045
Prevotella intermedia Prevotella intermedia MIC 0.12 ug.mL-1 10.1021/acs.jmedchem.1c02045
Priestia megaterium Priestia megaterium MIC 64.0 ug.mL-1 10.1016/j.bmcl.2015.01.026
Proteus mirabilis Proteus mirabilis MIC 1.0 ug.mL-1 10.1128/aac.00405-08
Proteus mirabilis Proteus mirabilis Ratio 2.0 None 10.1128/aac.00405-08
Proteus vulgaris Proteus vulgaris IZ 10.0 mm 10.1016/j.bmc.2018.02.049
Proteus vulgaris Proteus vulgaris MIC 0.125 ug.mL-1 10.1016/j.bmc.2018.02.049
Proteus vulgaris Proteus vulgaris MIC 1.0 ug.mL-1 10.1128/aac.00405-08
Proteus vulgaris Proteus vulgaris MIC 8.0 ug.mL-1 10.1021/jm00167a029
Proteus vulgaris Proteus vulgaris MIC 100.0 ug.mL-1 10.1021/jm0703901
Proteus vulgaris Proteus vulgaris Ratio 2.0 None 10.1128/aac.00405-08
Providencia alcalifaciens Providencia alcalifaciens MIC 8000.0 nM 10.1021/acs.jmedchem.1c02122
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity nan None 10.1021/acs.jmedchem.6b01742
Pseudomonas aeruginosa Pseudomonas aeruginosa Activity nan None 10.1021/acs.jnatprod.5b01129
Pseudomonas aeruginosa Pseudomonas aeruginosa EC50 5200.0 nM 10.1016/j.bmcl.2016.04.089
Pseudomonas aeruginosa Pseudomonas aeruginosa EC50 7800.0 nM 10.1021/acs.jmedchem.8b01293
Pseudomonas aeruginosa Pseudomonas aeruginosa FC 3.0 None 10.1021/acs.jnatprod.5b01129
Pseudomonas aeruginosa Pseudomonas aeruginosa FC 128.0 None 10.1021/acs.jmedchem.1c00614
Pseudomonas aeruginosa Pseudomonas aeruginosa FC 100000.0 None 10.1128/aac.01071-07
Pseudomonas aeruginosa Pseudomonas aeruginosa FIC 0.25 None 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa FIC 0.5 None 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa FICI 0.05 None 10.1128/aac.01071-07
Pseudomonas aeruginosa Pseudomonas aeruginosa FICI 1.25 None 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa FICI 1.5 None 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa Inhibition 10.0 % 10.1128/aac.00471-08
Pseudomonas aeruginosa Pseudomonas aeruginosa Inhibition 100.0 % 10.1021/jm0703901
Pseudomonas aeruginosa Pseudomonas aeruginosa Inhibition nan % 10.1128/aac.00471-08
Pseudomonas aeruginosa Pseudomonas aeruginosa IZ 6.0 mm 10.1016/j.bmc.2018.02.049
Pseudomonas aeruginosa Pseudomonas aeruginosa IZ 29.0 mm 10.1016/j.bmcl.2016.04.038
Pseudomonas aeruginosa Pseudomonas aeruginosa log10cfu 8.56 None 10.1128/aac.00471-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MBC 32.0 ug ml-1 10.1021/acs.jnatprod.2c00065
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 0.016 ug.mL-1 10.1128/aac.00471-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2.0 ug.mL-1 10.1016/j.ejmech.2016.03.061
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4.0 ug.mL-1 10.1128/aac.00405-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1021/acs.jmedchem.6b01742
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 8.0 ug.mL-1 10.1021/jm00167a029
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 10.0 ug.mL-1 10.1128/aac.01071-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 12.0 ug.mL-1 10.1021/jm00145a020
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 12.0 ug.mL-1 10.1128/aac.00405-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 13.0 ug.mL-1 10.1016/j.ejmech.2013.04.060
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 13.0 ug.mL-1 10.1021/jm400485e
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.6b01742
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1039/d2md00041e
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16.0 ug.mL-1 10.1128/aac.00405-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 20.0 ug.mL-1 10.1128/aac.01071-07
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 31.0 ug.mL-1 10.1021/jm501082n
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1016/j.bmc.2006.12.035
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1016/j.bmcl.2015.01.026
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1016/j.ejmech.2008.04.001
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1021/acs.jnatprod.2c00065
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1021/ml300350p
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00017-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32.0 ug.mL-1 10.1128/aac.00405-08
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 62.5 ug.mL-1 10.1021/acs.jnatprod.0c01309
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1016/j.bmcl.2020.127146
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 64.0 ug.mL-1 10.1016/j.ejmech.2022.114360
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 100.0 ug.mL-1 10.1021/jm0703901
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 128.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1016/j.bmc.2006.12.035
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 256.0 ug.mL-1 10.1016/j.ejmech.2019.05.090
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 500.0 ug.mL-1 10.1016/j.ejmech.2007.12.019
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 512.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1024.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 1024.0 ug.mL-1 10.1021/acs.jmedchem.6b01742
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2000.0 nM 10.1021/acs.jmedchem.1c00614
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2048.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4000.0 nM 10.1021/acs.jmedchem.1c00614
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 4096.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 16000.0 nM 10.1021/acs.jmedchem.9b00288
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 19000.0 nM 10.1021/acs.jnatprod.5b01129
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 25000.0 nM 10.1016/j.bmc.2016.04.058
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 27000.0 nM 10.1021/acs.jnatprod.5b01129
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32000.0 nM 10.1016/j.ejmech.2019.111636
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32000.0 nM 10.1021/acs.jmedchem.1c00614
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32000.0 nM 10.1021/acs.jmedchem.1c02140
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 32000.0 nM 10.1021/acs.jmedchem.2c01076
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 53000.0 nM 10.1021/acs.jmedchem.1c02122
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC 2048000.0 nM 10.1021/acs.jmedchem.1c00614
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC nan None 10.1016/j.bmc.2018.02.049
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC nan None 10.1016/j.bmc.2019.04.032
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC nan None 10.1016/j.bmcl.2012.08.003
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC nan None 10.1016/j.ejmech.2019.04.067
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC nan None 10.1021/np050424c
Pseudomonas aeruginosa Pseudomonas aeruginosa MIC>90 17.8 ug ml-1 10.1021/np400145u
Pseudomonas aeruginosa Pseudomonas aeruginosa mortality 100.0 % 10.1021/acs.jmedchem.6b01742
Pseudomonas aeruginosa Pseudomonas aeruginosa Ratio 2.0 None 10.1128/aac.00405-08
Rattus norvegicus Aldose reductase IC50 nan None None
Rattus norvegicus Aldose reductase Ki nan None None
Rattus norvegicus Alpha-1a adrenergic receptor IC50 nan None None
Rattus norvegicus Alpha-1a adrenergic receptor Ki nan None None
Rattus norvegicus Alpha-1b adrenergic receptor IC50 nan None None
Rattus norvegicus Alpha-1b adrenergic receptor Ki nan None None
Rattus norvegicus Androgen Receptor AC50 3000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Androgen Receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Androgen Receptor IC50 nan None None
Rattus norvegicus Androgen Receptor Ki nan None None
Rattus norvegicus Bile salt export pump IC50 34700.0 nM 10.1124/dmd.111.040758
Rattus norvegicus Bile salt export pump Ki 11900.0 nM 10.1016/s0016-5085(00)70224-1
Rattus norvegicus Brain Fu 0.068 None 10.1124/dmd.111.038778
Rattus norvegicus Brain Fu 0.121 None 10.1124/dmd.111.038778
Rattus norvegicus Brain Fu 0.13 None 10.1124/dmd.110.035998
Rattus norvegicus Brain Kp 0.92 None 10.1124/dmd.110.035998
Rattus norvegicus Brain Vd 6.9 L.kg-1 10.1124/dmd.110.035998
Rattus norvegicus Brain Vdu 6.9 ml 10.1021/jm901036q
Rattus norvegicus Cyclooxygenase-1 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus GABA receptor alpha-1 subunit AC50 30000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Glutamate (NMDA) receptor subunit zeta 1 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Glycine receptor IC50 nan None None
Rattus norvegicus Glycine receptor Ki nan None None
Rattus norvegicus Insulin receptor IC50 nan None None
Rattus norvegicus Insulin receptor Ki nan None None
Rattus norvegicus Jejunum CL 0.0 mL.min-1.g-1 10.1124/dmd.111.043067
Rattus norvegicus Kidney CL 0.0 mL.min-1.g-1 10.1124/dmd.111.043067
Rattus norvegicus Liver IC50 nan None 10.1002/hep.27206
Rattus norvegicus Liver microsome CL 0.0 mL.min-1.g-1 10.1124/dmd.111.043067
Rattus norvegicus Liver microsome Stability nan % 10.1021/acs.jmedchem.5b01542
Rattus norvegicus Multidrug resistance protein 1a Activity nan None 10.1016/0006-2952(95)00045-2
Rattus norvegicus Nitric-oxide synthase, brain IC50 nan None None
Rattus norvegicus Nitric-oxide synthase, brain Ki nan None None
Rattus norvegicus Nuclear receptor subfamily 1 group I member 2 Activity nan None 10.1124/dmd.110.035105
Rattus norvegicus Nuclear receptor subfamily 1 group I member 2 Activity nan None 10.1124/dmd.111.042879
Rattus norvegicus Plasma Cp(f) 0.83 uM 10.1021/jm901036q
Rattus norvegicus Plasma Fu 0.12 None 10.1021/jm901036q
Rattus norvegicus Plasma Fu 0.2 None 10.1021/jm901371v
Rattus norvegicus Plasma K(p,uu,CSF) 0.34 None 10.1021/jm901036q
Rattus norvegicus Rattus norvegicus Activity -31.0 % 10.1021/jm00164a013
Rattus norvegicus Rattus norvegicus Activity -30.0 % 10.1021/jm00164a013
Rattus norvegicus Rattus norvegicus Activity -27.0 % 10.1021/jm00164a013
Rattus norvegicus Rattus norvegicus ALB 34000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALB 35000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALB 36000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALB 36000.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALB 37000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALB 37000.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALB 38000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALB 38000.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALB 39000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALB 40000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALB 41000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALBGLOB 1.6 None 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALBGLOB 1.7 None 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALBGLOB 1.8 None 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALBGLOB 1.9 None 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALBGLOB 2.0 None 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 274.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALP 325.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALP 360.33 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALP 384.33 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALP 548.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 557.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 610.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 668.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 712.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 755.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 771.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 779.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 780.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 781.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 787.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 799.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 806.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 813.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 827.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 830.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 835.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 841.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 851.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 864.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 871.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 897.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 906.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 907.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 922.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 943.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 955.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 966.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 974.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 976.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 1040.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALP 1084.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 26.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 27.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 28.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 30.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 31.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 31.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 31.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 31.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 32.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 33.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 33.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 34.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 34.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 34.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 35.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 35.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 35.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 35.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 36.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALT 36.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 36.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 37.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 41.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALT 41.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus ALT 42.33 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus ALT 46.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus APTT 14.7 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 14.8 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 14.9 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 15.1 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 15.2 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 15.3 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 15.4 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 15.6 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 15.7 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 15.9 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 16.1 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 16.2 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 16.3 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 16.4 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 16.5 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 16.6 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 16.7 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 16.8 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 16.9 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 17.0 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 17.1 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 17.2 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus APTT 17.6 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 54.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 55.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 55.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 56.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 56.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 56.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 58.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 58.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 59.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 60.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus AST 60.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 60.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 60.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 61.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 61.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 62.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 62.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 62.67 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus AST 63.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 63.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 64.33 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus AST 64.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 65.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 65.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 66.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 66.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 68.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 68.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 68.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 69.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 69.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 70.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus AST 74.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BASOLE 0.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BASOLE 0.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BILDIR 0.02 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.04 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.14 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.16 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.18 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.2 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.28 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.32 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.34 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.38 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.4 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.42 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.44 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.5 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.66 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 0.78 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 1.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 2.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 3.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 4.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILDIR 5.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILI 3.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILI 3.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BILI 3.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BILI 3.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BILI 4.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILI 5.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILI 6.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILI 9.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BILI 10.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 90.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BUN 96.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 100.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 105.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 106.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 106.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BUN 110.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 112.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 113.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BUN 122.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 128.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 132.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 136.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus BUN 146.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 158.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 160.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 164.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 168.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 172.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 174.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 178.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 182.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 184.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 186.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 190.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 192.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus BUN 202.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CALCIUM 98.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CALCIUM 100.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CALCIUM 101.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CALCIUM 102.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CALCIUM 103.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CALCIUM 104.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CALCIUM 105.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CALCIUM 106.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CALCIUM 107.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CALCIUM 108.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CALCIUM 109.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHLORIDE 106.67 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHLORIDE 107.33 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHLORIDE 108.0 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHLORIDE 108.33 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHOL 540.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 600.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 632.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 633.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHOL 670.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 680.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 686.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 716.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 730.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 734.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 736.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 746.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 748.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 750.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHOL 760.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 766.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 768.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 774.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 776.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 782.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 783.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CHOL 784.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 796.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 804.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 806.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 810.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 816.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 822.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 830.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 836.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 838.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 848.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 866.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CHOL 936.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CK 115.33 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CK 139.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CK 142.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CK 143.0 U.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus Cl 103.2 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 104.0 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 104.6 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 104.8 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 105.0 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 105.4 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 105.6 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 105.8 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 106.0 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 106.2 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 106.4 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 106.6 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 106.8 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 107.0 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 107.2 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 107.6 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 107.8 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 108.0 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 108.2 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 108.4 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Cl 109.6 meq/L 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CREAT 3.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CREAT 4.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CREAT 4.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CREAT 5.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus CREAT 5.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CREAT 5.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus CREAT 6.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus EOSLE 0.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus EOSLE 0.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOSLE 0.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus EOSLE 0.33 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus EOSLE 0.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus EOSLE 0.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus EOSLE 0.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus EOSLE 1.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2032.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2034.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2036.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2052.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2074.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2078.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2102.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2114.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2126.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2136.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2144.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2146.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2180.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2208.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2210.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2212.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2224.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2250.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2264.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2266.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2268.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2272.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2290.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2318.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2326.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2336.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2356.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2366.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2390.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2394.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus FIBRINO 2396.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GGT 0.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GGT 1.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GGT 1.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GGT 1.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GGT 1.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GGT 1.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GGT 2.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GGT 2.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1663.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus GLUC 1703.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus GLUC 1776.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus GLUC 1798.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1803.3 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus GLUC 1812.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1822.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1824.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1836.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1842.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1850.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1854.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1858.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1866.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1878.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1880.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1884.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1888.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1890.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1902.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1916.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1932.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1934.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1936.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1942.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1948.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1986.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 1992.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 2028.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 2030.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 2104.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus GLUC 2120.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 34.87 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HCT 35.03 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HCT 36.5 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HCT 36.73 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HCT 38.9 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 40.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 40.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 40.5 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 40.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 40.7 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 40.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 40.9 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 41.1 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 41.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 41.3 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 41.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 41.7 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 42.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 42.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 42.3 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 42.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 42.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 43.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 43.3 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 44.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 44.9 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 45.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 46.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HCT 47.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 130000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 134000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 135000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 136000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 137000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 137300.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HGB 138000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 139000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 139300.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HGB 140000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 141000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 143000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 143300.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HGB 145700.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus HGB 147000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 150000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 152000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 156000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus HGB 157000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 70.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 75.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 76.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 77.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 78.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 84.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 89.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 91.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 96.0 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 96.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 98.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 99.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 100.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 101.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 102.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 104.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 106.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 108.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 110.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 113.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 114.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 114.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 128.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 147.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 157.2 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 158.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 160.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 163.8 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 165.4 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LDH 204.6 IU.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 76.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 76.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 77.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 78.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 78.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 79.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 80.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 81.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 81.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 81.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 82.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 82.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 82.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 82.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 84.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 84.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 84.5 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 84.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 84.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 85.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYMLE 85.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 85.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 86.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 86.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 86.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 86.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 87.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 87.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 88.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYMLE 89.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYMLE 89.33 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus LYMLE 90.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 91.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus LYMLE 92.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 17.8 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 18.9 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 19.0 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 19.7 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 19.8 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 20.3 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 20.4 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 20.7 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 20.9 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 21.0 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 21.1 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 21.2 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 21.3 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 21.5 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 21.6 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 21.7 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 21.8 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 21.9 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 22.0 pg 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCH 23.47 pg 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCH 23.73 pg 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCH 23.83 pg 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCH 24.47 pg 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCHC 33.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCHC 33.1 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCHC 33.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCHC 33.3 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCHC 33.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCHC 33.5 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCHC 33.7 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCHC 33.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCHC 390300.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCHC 394000.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCHC 397700.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCHC 399300.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCV 53.7 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 55.8 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 56.7 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 58.7 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 58.8 fL 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCV 58.9 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 59.6 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 60.23 fL 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCV 60.6 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 60.7 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 61.1 fL 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCV 61.5 fL 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MCV 62.5 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 62.8 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 62.9 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 63.2 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 63.4 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 63.8 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 63.9 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 64.0 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 64.2 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 64.6 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 64.9 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 65.0 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 65.1 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 65.2 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 65.5 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 65.6 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 65.9 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 66.0 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MCV 66.3 fL 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 2.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MONOLE 2.33 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MONOLE 2.67 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus MONOLE 2.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 3.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 3.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 3.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 3.5 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 4.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 4.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 5.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 5.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 5.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 5.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 5.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 6.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 6.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 6.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 6.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 7.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 7.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 7.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 7.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus MONOLE 8.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 2.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 3.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 4.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 6.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 6.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 6.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 7.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 7.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 7.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 7.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 8.0 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTLE 8.67 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTLE 8.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 9.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 9.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 9.67 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTLE 10.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 11.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 11.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 11.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 12.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 12.67 % 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus NEUTLE 13.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 13.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 13.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 14.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 15.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus NEUTLE 16.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 70.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 71.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 72.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 77.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 79.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 80.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 81.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 83.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 88.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 90.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 93.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 95.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 96.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 103.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 104.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 105.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 106.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 107.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 109.7 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PHOS 110.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 111.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 111.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PHOS 112.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOS 113.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PHOS 116.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PHOSLPD 1080.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1155.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1178.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1202.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1248.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1274.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1278.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1286.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1340.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1346.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1354.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1376.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1386.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1396.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1406.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1420.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1422.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1444.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1448.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1454.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1468.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1470.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1500.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1514.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1542.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1562.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1570.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1574.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1596.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1598.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PHOSLPD 1608.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1010670.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PLAT 1035000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1047330.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PLAT 1053000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1065000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1070000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1072000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1077000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1082670.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PLAT 1103000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1105000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1110000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1111330.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PLAT 1112000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1114000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1115000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1116000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1118000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1125000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1134000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1142000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1143000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1152000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1156000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1179000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1181000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1182000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1183000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1219000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1225000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1259000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PLAT 1260000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus POTASSIUM 4.3 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus POTASSIUM 4.4 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus POTASSIUM 4.5 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus POTASSIUM 4.6 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus POTASSIUM 4.7 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus POTASSIUM 4.8 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus POTASSIUM 4.9 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus POTASSIUM 5.0 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus POTASSIUM 5.1 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus POTASSIUM 5.2 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus POTASSIUM 5.5 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus POTASSIUM 6.3 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus POTASSIUM 6.4 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus POTASSIUM 6.6 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus POTASSIUM 6.63 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PROT 55000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PROT 56000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PROT 56700.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PROT 57000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PROT 57300.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PROT 58000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PROT 59000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PROT 60000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PROT 60300.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PROT 61000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PROT 61000.0 ug.mL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus PROT 62000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PROT 63000.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 11.5 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 11.7 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 11.8 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 11.9 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 12.0 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 12.1 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 12.2 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 12.3 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 12.4 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 12.5 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 12.6 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 12.7 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus PT 12.8 s 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 5700000.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus RBC 5790000.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus RBC 5958000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6010000.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus RBC 6092000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6104000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6168000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6208000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6212000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6220000.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus RBC 6236000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6242000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6246000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6282000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6332000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6358000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6402000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6412000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6536000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6576000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6580000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6582000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6730000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6738000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6772000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6832000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 6840000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 7028000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 7262000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 7426000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 7548000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 7866000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 7996000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 8036000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RBC 8190000.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 2.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 2.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 2.3 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 2.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 3.5 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 3.9 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 4.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 4.7 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 5.5 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 5.7 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 5.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 5.9 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 6.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 7.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 8.5 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 8.6 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 8.7 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 9.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 9.4 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 9.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 10.0 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 10.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 10.5 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 10.8 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 10.9 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 11.1 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus RETIRBC 11.2 % 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 136.8 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 137.0 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 137.2 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 137.4 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 137.8 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 138.0 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 138.2 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 138.6 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 138.8 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 139.0 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 139.2 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 139.4 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 139.6 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 139.8 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 140.0 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 140.6 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 140.8 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 141.2 mEq.L-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus SODIUM 149.33 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus SODIUM 150.33 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus SODIUM 152.67 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus SODIUM 153.0 mEq.L-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus TERMBW 189.7 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 190.4 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 190.9 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 191.2 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 191.9 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 192.3 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 192.4 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 193.3 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 194.2 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 194.8 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 196.1 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 196.2 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 201.3 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 203.6 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 206.5 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 223.8 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 234.9 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 238.2 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 242.1 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 249.0 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 259.9 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 264.5 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 275.2 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 298.5 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 298.6 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 308.0 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 316.4 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 356.4 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 375.5 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 379.8 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TERMBW 390.1 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Tissue Severity Score nan None 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus Tissue Severity Score nan None 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus TRIG 228.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 230.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 332.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 358.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 394.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 396.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 452.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 460.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 482.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 506.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 528.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 546.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 556.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 624.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 660.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 664.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 682.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 710.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 730.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 754.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 758.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 906.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 968.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 1128.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 1166.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 1204.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 1214.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 1320.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 1326.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 1650.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 1682.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus TRIG 2058.0 ug.mL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 9070.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus WBC 9940.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 10170.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 10200.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 10490.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 10500.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 10700.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 11630.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 11650.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 11690.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 11900.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 11920.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 11960.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 12040.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 12220.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 12330.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 12390.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 12470.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 12700.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 12700.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus WBC 12800.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 12910.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 12940.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 13090.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 13120.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 13160.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 13840.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 14230.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus WBC 14620.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 15360.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 16120.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 16520.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WBC 17130.0 cells.uL-1 10.6019/CHEMBL3885881
Rattus norvegicus Rattus norvegicus WBC 18560.0 cells.uL-1 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 0.8 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 0.9 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 1.0 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 1.1 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 1.2 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 1.3 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 1.4 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 1.7 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 1.8 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 1.9 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 2.0 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 2.1 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 2.2 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 2.3 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 2.4 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 2.5 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 2.6 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 2.7 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 7.5 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 7.6 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 7.7 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 7.9 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 8.1 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 8.5 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 8.8 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 8.9 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 9.0 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 9.4 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 9.8 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 10.2 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 10.7 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 11.3 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 11.6 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 12.2 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 12.4 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 12.9 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 13.1 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 13.9 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 14.5 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 14.8 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 16.0 g 10.6019/CHEMBL3885861
Rattus norvegicus Rattus norvegicus WEIGHT 16.8 g 10.6019/CHEMBL3885861
Rattus norvegicus Serotonin 1a (5-HT1a) receptor IC50 nan None None
Rattus norvegicus Serotonin 1a (5-HT1a) receptor Ki nan None None
Rattus norvegicus Serotonin 1b (5-HT1b) receptor IC50 nan None None
Rattus norvegicus Serotonin 1b (5-HT1b) receptor Ki nan None None
Rattus norvegicus Serum AUC 277000.0 ng.hr.mL-1 10.1128/aac.00458-08
Rattus norvegicus Solute carrier family 22 member 7 Activity nan None 10.1016/s0014-5793(98)00585-7
Rattus norvegicus Solute carrier organic anion transporter family member 1A1 Activity nan None None
Rattus norvegicus Solute carrier organic anion transporter family member 1A1 Ki 18200.0 nM 10.1023/a:1014264614637
Rattus norvegicus Solute carrier organic anion transporter family member 1A4 Ki 1400.0 nM 10.1053/jhep.2000.8539
Rattus norvegicus Solute carrier organic anion transporter family member 1A4 Ki 1460.0 nM 10.1023/a:1014264614637
Rattus norvegicus Voltage-gated L-type calcium channel alpha-1C subunit AC50 30000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Voltage-gated N-type calcium channel alpha-1B subunit AC50 10000.0 nM 10.1038/s41467-023-40064-9
Saccharomyces cerevisiae Saccharomyces cerevisiae IZ 0.0 mm 10.1016/j.ejmech.2010.07.050
Salmonella enterica Salmonella enterica MIC 4.0 ug.mL-1 10.1128/aac.00310-09
Salmonella enterica Salmonella enterica MIC 2000.0 nM 10.1021/acs.jmedchem.1c02122
Salmonella enterica subsp. enterica serovar Abony Salmonella enterica subsp. enterica serovar Abony MIC 1.0 ug.mL-1 10.1016/j.ejmech.2014.07.066
Salmonella enterica subsp. enterica serovar Paratyphi A Salmonella paratyphi IZ 6.0 mm 10.1016/j.bmc.2018.02.049
Salmonella enterica subsp. enterica serovar Paratyphi A Salmonella paratyphi MIC 12.0 ug.mL-1 10.1021/jm00143a010
Salmonella enterica subsp. enterica serovar Paratyphi A Salmonella paratyphi MIC 12.0 ug.mL-1 10.1021/jm00145a020
Salmonella enterica subsp. enterica serovar Paratyphi A Salmonella paratyphi MIC nan None 10.1016/j.bmc.2018.02.049
Salmonella enterica subsp. enterica serovar Paratyphi B Salmonella enterica subsp. enterica serovar Paratyphi B MIC 12.0 ug.mL-1 10.1021/jm00220a012
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium Activity nan None 10.1016/j.ejmech.2017.06.061
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium Inhibition 100.0 % 10.1021/jm0703901
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 16.0 ug.mL-1 10.1128/aac.00079-09
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 100.0 ug.mL-1 10.1021/jm0703901
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 256.0 ug.mL-1 10.1128/aac.00615-06
Salmonella enterica subsp. enterica serovar Typhimurium Salmonella typhimurium MIC 4000.0 nM 10.1021/acs.jmedchem.9b00288
Serratia marcescens Serratia marcescens MIC 16.0 ug.mL-1 10.1128/aac.00405-08
Serratia marcescens Serratia marcescens MIC 32.0 ug.mL-1 10.1021/ml300350p
Serratia marcescens Serratia marcescens Ratio 2.0 None 10.1128/aac.00405-08
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Hit score 0.08736 None 10.1101/2020.04.21.054387
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 IC50 19952.62 nM 10.6019/CHEMBL4651402
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 IC50 20000.0 nM 10.6019/CHEMBL4651402
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Inhibition index 0.2558 None 10.1101/2020.04.03.023846
Shigella dysenteriae Shigella dysenteriae IZ 8.0 mm 10.1016/j.bmc.2018.02.049
Shigella dysenteriae Shigella dysenteriae MIC 0.25 ug.mL-1 10.1016/j.bmc.2018.02.049
Shigella sonnei Shigella sonnei MIC 1700.0 nM 10.1021/acs.jmedchem.1c02122
Staphylococcus aureus Staphylococcus aureus Activity 0.0 % 10.1128/aac.01244-06
Staphylococcus aureus Staphylococcus aureus Activity 2.0 % 10.1128/aac.00846-07
Staphylococcus aureus Staphylococcus aureus Activity 2.3 % 10.1128/aac.00090-10
Staphylococcus aureus Staphylococcus aureus Activity 4.0 % 10.1128/aac.00846-07
Staphylococcus aureus Staphylococcus aureus Activity 18.8 % 10.1128/aac.00090-10
Staphylococcus aureus Staphylococcus aureus Activity 20.0 % 10.1016/j.bmc.2006.12.027
Staphylococcus aureus Staphylococcus aureus Activity 46.0 % 10.1128/aac.00120-07
Staphylococcus aureus Staphylococcus aureus Activity 50.0 % 10.1128/aac.00775-08
Staphylococcus aureus Staphylococcus aureus Activity 92.0 % 10.1128/aac.00775-08
Staphylococcus aureus Staphylococcus aureus Activity 94.0 % 10.1128/aac.00470-10
Staphylococcus aureus Staphylococcus aureus Activity 94.0 % 10.1128/aac.00775-08
Staphylococcus aureus Staphylococcus aureus Activity 96.0 % 10.1128/aac.00470-10
Staphylococcus aureus Staphylococcus aureus Activity 99.9 % 10.1016/j.bmcl.2023.129320
Staphylococcus aureus Staphylococcus aureus Activity 100.0 % 10.1128/aac.00470-10
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1016/j.bmc.2016.11.056
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1016/j.bmcl.2023.129320
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1016/j.ejmech.2018.04.049
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1016/j.ejmech.2019.112026
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1016/j.ejmech.2021.113691
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1021/acs.jmedchem.2c01076
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1021/jm0703183
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1021/jm3012728
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1021/jm900519b
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.00064-10
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.00350-06
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.00458-08
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.00596-06
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.00766-08
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.00775-08
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.00804-08
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.01145-08
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.01302-07
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.01395-07
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.01480-07
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.01605-07
Staphylococcus aureus Staphylococcus aureus Activity nan None 10.1128/aac.01649-07
Staphylococcus aureus Staphylococcus aureus Antibiotic resistance nan None 10.1016/s0960-894x(98)00536-8
Staphylococcus aureus Staphylococcus aureus AUC 19650.0 ng.hr.mL-1 10.1128/aac.00455-10
Staphylococcus aureus Staphylococcus aureus EC50 50.0 nM 10.1016/j.bmcl.2016.04.089
Staphylococcus aureus Staphylococcus aureus EC50 50.0 nM 10.1021/acs.jmedchem.8b01293
Staphylococcus aureus Staphylococcus aureus EC50 150.0 nM 10.1016/j.bmcl.2016.04.089
Staphylococcus aureus Staphylococcus aureus EC50 230.0 nM 10.1021/acs.jmedchem.8b01293
Staphylococcus aureus Staphylococcus aureus ED50 0.09 mg.kg-1 10.1021/jm00167a029
Staphylococcus aureus Staphylococcus aureus ED50 0.14 mg.kg-1 10.1021/jm00145a020
Staphylococcus aureus Staphylococcus aureus ED50 0.28 mg.kg-1 10.1021/jm00167a029
Staphylococcus aureus Staphylococcus aureus FC 0.98 None 10.1128/aac.00273-08
Staphylococcus aureus Staphylococcus aureus FC 0.99 None 10.1128/aac.00273-08
Staphylococcus aureus Staphylococcus aureus FC 1.19 None 10.1128/aac.00273-08
Staphylococcus aureus Staphylococcus aureus FC 1.2 None 10.1128/aac.00273-08
Staphylococcus aureus Staphylococcus aureus FC 1.9 None 10.1128/aac.00273-08
Staphylococcus aureus Staphylococcus aureus FC 2.0 None 10.1128/aac.01605-07
Staphylococcus aureus Staphylococcus aureus FC 2.5 None 10.1128/aac.01605-07
Staphylococcus aureus Staphylococcus aureus FC 4.0 None 10.1039/d2md00351a
Staphylococcus aureus Staphylococcus aureus FC 8.0 None 10.1016/j.ejmech.2021.113723
Staphylococcus aureus Staphylococcus aureus FC 15.0 None 10.1039/d2md00351a
Staphylococcus aureus Staphylococcus aureus FC 128.0 None 10.1016/j.bmcl.2023.129320
Staphylococcus aureus Staphylococcus aureus FC 500.0 None 10.1021/jm3012728
Staphylococcus aureus Staphylococcus aureus FC 1024.0 None 10.1016/j.bmcl.2023.129320
Staphylococcus aureus Staphylococcus aureus FC 4096.0 None 10.1021/acs.jmedchem.2c01076
Staphylococcus aureus Staphylococcus aureus FC 16000.0 None 10.1016/j.ejmech.2021.113723
Staphylococcus aureus Staphylococcus aureus fCmax 3.82 ug ml-1 10.1128/aac.00455-10
Staphylococcus aureus Staphylococcus aureus FIC 1.0 None 10.1021/acs.jnatprod.2c00621
Staphylococcus aureus Staphylococcus aureus GI nan None 10.1016/j.bmc.2015.04.069
Staphylococcus aureus Staphylococcus aureus IC50 0.0025 ug.mL-1 10.1021/np000436s
Staphylococcus aureus Staphylococcus aureus IC50 0.01 ug.mL-1 10.1021/np000436s
Staphylococcus aureus Staphylococcus aureus IC50 250.0 ug.mL-1 10.1021/np050176k
Staphylococcus aureus Staphylococcus aureus IC50 10000.0 nM 10.1021/acs.jnatprod.2c00444
Staphylococcus aureus Staphylococcus aureus IC50 nan None 10.1021/np2006555
Staphylococcus aureus Staphylococcus aureus IC50 nan None 10.1021/np900281r
Staphylococcus aureus Staphylococcus aureus Inhibition 10.0 % 10.1128/aac.00471-08
Staphylococcus aureus Staphylococcus aureus Inhibition 76.3 % 10.1016/j.ejmech.2021.113402
Staphylococcus aureus Staphylococcus aureus Inhibition 76.3 % 10.1039/D1MD00230A
Staphylococcus aureus Staphylococcus aureus Inhibition 100.0 % 10.1021/jm0703901
Staphylococcus aureus Staphylococcus aureus Inhibition nan % 10.1128/aac.00471-08
Staphylococcus aureus Staphylococcus aureus Inhibition nan % 10.1128/aac.01302-07
Staphylococcus aureus Staphylococcus aureus IZ 10.0 mm 10.1016/j.bmc.2018.02.049
Staphylococcus aureus Staphylococcus aureus IZ 23.0 mm 10.1016/j.bmcl.2017.05.032
Staphylococcus aureus Staphylococcus aureus IZ 25.0 mm 10.1016/j.bmcl.2016.04.038
Staphylococcus aureus Staphylococcus aureus IZ 27.0 mm 10.1016/j.bmcl.2017.05.032
Staphylococcus aureus Staphylococcus aureus IZ 30.0 mm 10.1016/j.bmcl.2017.05.032
Staphylococcus aureus Staphylococcus aureus IZ 31.0 mm 10.1016/j.bmc.2007.09.025
Staphylococcus aureus Staphylococcus aureus IZ 33.0 mm 10.1016/j.bmcl.2017.05.032
Staphylococcus aureus Staphylococcus aureus IZ 49.0 mm 10.1016/j.ejmech.2008.09.035
Staphylococcus aureus Staphylococcus aureus IZ nan None 10.1021/np900382x
Staphylococcus aureus Staphylococcus aureus log10cfu -1.72 None 10.1128/aac.01145-08
Staphylococcus aureus Staphylococcus aureus log10cfu 0.86 None 10.1128/aac.00237-08
Staphylococcus aureus Staphylococcus aureus log10cfu 1.0 None 10.1128/aac.01145-08
Staphylococcus aureus Staphylococcus aureus log10cfu 1.1 None 10.1128/aac.00208-09
Staphylococcus aureus Staphylococcus aureus log10cfu 1.36 None 10.1128/aac.00208-09
Staphylococcus aureus Staphylococcus aureus log10cfu 1.78 None 10.1128/aac.00237-08
Staphylococcus aureus Staphylococcus aureus log10cfu 2.0 None 10.1128/aac.01145-08
Staphylococcus aureus Staphylococcus aureus log10cfu 3.0 None 10.1128/aac.01145-08
Staphylococcus aureus Staphylococcus aureus log10cfu 7.5 None 10.1128/aac.00471-08
Staphylococcus aureus Staphylococcus aureus log10cfu 42.6 None 10.1128/aac.01145-08
Staphylococcus aureus Staphylococcus aureus log10CFU/ml -3.02 None 10.1128/aac.01145-08
Staphylococcus aureus Staphylococcus aureus log10CFU/ml 0.5 None 10.1128/aac.00775-08
Staphylococcus aureus Staphylococcus aureus log10CFU/ml 1.43 None 10.1128/aac.00120-07
Staphylococcus aureus Staphylococcus aureus log10CFU/ml 3.0 None 10.1128/aac.00775-08
Staphylococcus aureus Staphylococcus aureus log10CFU/ml 3.1 None 10.1128/aac.00775-08
Staphylococcus aureus Staphylococcus aureus log10CFU/ml 3.68 None 10.1128/aac.00120-07
Staphylococcus aureus Staphylococcus aureus log10CFU/ml 6.9 None 10.1128/aac.00458-08
Staphylococcus aureus Staphylococcus aureus log10CFU/ml 43.35 None 10.1128/aac.01145-08
Staphylococcus aureus Staphylococcus aureus log(1/C) 8.07 None 10.1021/jm00210a025
Staphylococcus aureus Staphylococcus aureus MBC 0.08 ug ml-1 10.1128/aac.00775-08
Staphylococcus aureus Staphylococcus aureus MBC 0.12 ug ml-1 10.1128/aac.00458-08
Staphylococcus aureus Staphylococcus aureus MBC 0.2 ug ml-1 10.1016/j.bmc.2018.07.034
Staphylococcus aureus Staphylococcus aureus MBC 0.4 ug ml-1 10.1016/j.bmc.2018.07.034
Staphylococcus aureus Staphylococcus aureus MBC 0.5 ug ml-1 10.1128/aac.00208-09
Staphylococcus aureus Staphylococcus aureus MBC 0.8 ug ml-1 10.1128/aac.00120-07
Staphylococcus aureus Staphylococcus aureus MBC 1.0 ug ml-1 10.1016/j.bmcl.2023.129320
Staphylococcus aureus Staphylococcus aureus MBC 2.0 mg/ml 10.1021/acs.jmedchem.6b00485
Staphylococcus aureus Staphylococcus aureus MBC 2.0 ug ml-1 10.1016/j.bmcl.2023.129320
Staphylococcus aureus Staphylococcus aureus MBC 2.0 uM 10.1021/acs.jmedchem.5b02004
Staphylococcus aureus Staphylococcus aureus MBC 2.0 uM 10.1021/acs.jmedchem.7b01903
Staphylococcus aureus Staphylococcus aureus MBC 2.5 ug ml-1 10.1128/aac.00775-08
Staphylococcus aureus Staphylococcus aureus MBC 3.6 ug ml-1 10.1128/aac.00120-07
Staphylococcus aureus Staphylococcus aureus MBC 4.0 ug ml-1 10.1128/aac.00458-08
Staphylococcus aureus Staphylococcus aureus MBC 8.0 ng/ml 10.1021/acs.jnatprod.5b00770
Staphylococcus aureus Staphylococcus aureus MBC 8.0 ug ml-1 10.1128/aac.00208-09
Staphylococcus aureus Staphylococcus aureus MBC 25.0 ug ml-1 10.1016/j.bmc.2018.07.034
Staphylococcus aureus Staphylococcus aureus MBC nan None 10.1021/acs.jnatprod.2c00065
Staphylococcus aureus Staphylococcus aureus MBEC 0.25 ug ml-1 10.1128/aac.00766-08
Staphylococcus aureus Staphylococcus aureus MBEC 4.0 ug ml-1 10.1128/aac.00766-08
Staphylococcus aureus Staphylococcus aureus MBEC 6.25 ug ml-1 10.1128/aac.00457-09
Staphylococcus aureus Staphylococcus aureus MBEC 25.0 ug ml-1 10.1128/aac.00457-09
Staphylococcus aureus Staphylococcus aureus MBEC 46.9 uM 10.1021/acs.jmedchem.5b02004
Staphylococcus aureus Staphylococcus aureus MBEC 46.9 uM 10.1021/acs.jmedchem.7b01903
Staphylococcus aureus Staphylococcus aureus MBIC 0.0625 ug ml-1 10.1128/aac.00455-10
Staphylococcus aureus Staphylococcus aureus MBIC 0.2 ug ml-1 10.1128/aac.00457-09
Staphylococcus aureus Staphylococcus aureus MBIC nan None 10.1128/aac.00455-10
Staphylococcus aureus Staphylococcus aureus MIC 6e-06 ug.mL-1 10.1128/aac.00437-10
Staphylococcus aureus Staphylococcus aureus MIC 0.0002 ug.mL-1 10.1128/aac.01145-08
Staphylococcus aureus Staphylococcus aureus MIC 0.00025 ug.mL-1 10.1128/aac.00471-08
Staphylococcus aureus Staphylococcus aureus MIC 0.0005 ug.mL-1 10.1128/aac.01145-08
Staphylococcus aureus Staphylococcus aureus MIC 0.002 ug.mL-1 10.1016/j.bmcl.2009.09.095
Staphylococcus aureus Staphylococcus aureus MIC 0.002 ug.mL-1 10.1016/j.bmcl.2010.12.084
Staphylococcus aureus Staphylococcus aureus MIC 0.002 ug.mL-1 10.1021/np050176k
Staphylococcus aureus Staphylococcus aureus MIC 0.002 ug.mL-1 10.1021/np200320u
Staphylococcus aureus Staphylococcus aureus MIC 0.002 ug.mL-1 10.1128/aac.00206-09
Staphylococcus aureus Staphylococcus aureus MIC 0.002 ug.mL-1 10.1128/aac.01145-08
Staphylococcus aureus Staphylococcus aureus MIC 0.003 ug.mL-1 10.1021/jm00164a013
Staphylococcus aureus Staphylococcus aureus MIC 0.004 ug.mL-1 10.1016/j.bmcl.2007.02.024
Staphylococcus aureus Staphylococcus aureus MIC 0.004 ug.mL-1 10.1016/j.bmcl.2010.12.084
Staphylococcus aureus Staphylococcus aureus MIC 0.004 ug.mL-1 10.1021/acs.jnatprod.2c00065
Staphylococcus aureus Staphylococcus aureus MIC 0.004 ug.mL-1 10.1021/acs.jnatprod.5b00770
Staphylococcus aureus Staphylococcus aureus MIC 0.004 ug.mL-1 10.1021/np200320u
Staphylococcus aureus Staphylococcus aureus MIC 0.004 ug.mL-1 10.1128/aac.00064-10
Staphylococcus aureus Staphylococcus aureus MIC 0.004 ug.mL-1 10.1128/aac.00206-09
Staphylococcus aureus Staphylococcus aureus MIC 0.004 ug.mL-1 10.1128/aac.00834-08
Staphylococcus aureus Staphylococcus aureus MIC 0.004 ug.mL-1 10.1128/aac.01455-06
Staphylococcus aureus Staphylococcus aureus MIC 0.004 ug.mL-1 10.1128/aac.01544-08
Staphylococcus aureus Staphylococcus aureus MIC 0.004 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC 0.005 ug.mL-1 10.1021/jm00145a020
Staphylococcus aureus Staphylococcus aureus MIC 0.005 ug.mL-1 10.1021/np010173h
Staphylococcus aureus Staphylococcus aureus MIC 0.006 ug.mL-1 10.1016/j.ejmech.2017.10.048
Staphylococcus aureus Staphylococcus aureus MIC 0.006 ug.mL-1 10.1128/aac.00457-09
Staphylococcus aureus Staphylococcus aureus MIC 0.006 ug.mL-1 10.1128/aac.00834-08
Staphylococcus aureus Staphylococcus aureus MIC 0.007 ug.mL-1 10.1021/jm00210a025
Staphylococcus aureus Staphylococcus aureus MIC 0.0078 ug.mL-1 10.1021/acs.jnatprod.1c00578
Staphylococcus aureus Staphylococcus aureus MIC 0.0078 ug.mL-1 10.1021/acs.jnatprod.2c00621
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1016/j.bmcl.2006.10.016
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1016/j.bmcl.2007.08.048
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1016/j.bmcl.2016.05.077
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1016/j.ejmech.2012.09.041
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1016/j.ejmech.2014.07.066
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1016/j.ejmech.2016.03.061
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1021/acs.jmedchem.1c02045
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1021/acs.jmedchem.6b00485
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1021/acsmedchemlett.0c00381
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1128/aac.00206-09
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1128/aac.01455-06
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC 0.008 ug.mL-1 10.1128/aac.01649-07
Staphylococcus aureus Staphylococcus aureus MIC 0.01 ug.mL-1 10.1021/acs.jmedchem.0c00520
Staphylococcus aureus Staphylococcus aureus MIC 0.01 ug.mL-1 10.1128/aac.00775-08
Staphylococcus aureus Staphylococcus aureus MIC 0.012 ug.mL-1 10.1128/aac.00457-09
Staphylococcus aureus Staphylococcus aureus MIC 0.01221 ug.mL-1 10.1016/j.bmc.2010.02.005
Staphylococcus aureus Staphylococcus aureus MIC 0.0125 ug.mL-1 10.1016/j.ejmech.2019.05.090
Staphylococcus aureus Staphylococcus aureus MIC 0.015 ug.mL-1 10.1016/j.ejmech.2012.09.041
Staphylococcus aureus Staphylococcus aureus MIC 0.015 ug.mL-1 10.1016/j.ejmech.2019.04.067
Staphylococcus aureus Staphylococcus aureus MIC 0.015 ug.mL-1 10.1128/aac.00973-06
Staphylococcus aureus Staphylococcus aureus MIC 0.0156 ug.mL-1 10.1016/j.ejmech.2019.02.009
Staphylococcus aureus Staphylococcus aureus MIC 0.016 ug.mL-1 10.1016/j.bmcl.2015.07.043
Staphylococcus aureus Staphylococcus aureus MIC 0.016 ug.mL-1 10.1016/j.ejmech.2014.07.066
Staphylococcus aureus Staphylococcus aureus MIC 0.016 ug.mL-1 10.1016/j.ejmech.2016.03.061
Staphylococcus aureus Staphylococcus aureus MIC 0.016 ug.mL-1 10.1021/jm00167a029
Staphylococcus aureus Staphylococcus aureus MIC 0.016 ug.mL-1 10.1128/aac.00120-07
Staphylococcus aureus Staphylococcus aureus MIC 0.016 ug.mL-1 10.1128/aac.00206-09
Staphylococcus aureus Staphylococcus aureus MIC 0.016 ug.mL-1 10.1128/aac.01455-06
Staphylococcus aureus Staphylococcus aureus MIC 0.016 ug.mL-1 10.1128/aac.01605-07
Staphylococcus aureus Staphylococcus aureus MIC 0.016 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC 0.02 ug.mL-1 10.1016/j.ejmech.2013.04.060
Staphylococcus aureus Staphylococcus aureus MIC 0.02 ug.mL-1 10.1021/jm400485e
Staphylococcus aureus Staphylococcus aureus MIC 0.02 ug.mL-1 10.1021/np000436s
Staphylococcus aureus Staphylococcus aureus MIC 0.02 ug.mL-1 10.1128/aac.00766-08
Staphylococcus aureus Staphylococcus aureus MIC 0.0225 ug.mL-1 10.1007/s00044-011-9918-4
Staphylococcus aureus Staphylococcus aureus MIC 0.025 ug.mL-1 10.1021/jm00143a010
Staphylococcus aureus Staphylococcus aureus MIC 0.025 ug.mL-1 10.1021/jm00220a012
Staphylococcus aureus Staphylococcus aureus MIC 0.03 ug.mL-1 10.1021/acs.jmedchem.0c00520
Staphylococcus aureus Staphylococcus aureus MIC 0.03 ug.mL-1 10.1021/acs.jnatprod.9b00062
Staphylococcus aureus Staphylococcus aureus MIC 0.03 ug.mL-1 10.1021/jm501082n
Staphylococcus aureus Staphylococcus aureus MIC 0.03 ug.mL-1 10.1128/aac.00208-09
Staphylococcus aureus Staphylococcus aureus MIC 0.03 ug.mL-1 10.1128/aac.00766-08
Staphylococcus aureus Staphylococcus aureus MIC 0.03 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC 0.03125 ug.mL-1 10.1016/j.ejmech.2019.02.009
Staphylococcus aureus Staphylococcus aureus MIC 0.049 ug.mL-1 10.1128/aac.00971-08
Staphylococcus aureus Staphylococcus aureus MIC 0.05 ug.mL-1 10.1128/aac.00273-08
Staphylococcus aureus Staphylococcus aureus MIC 0.06 ug.mL-1 10.1016/j.ejmech.2007.12.019
Staphylococcus aureus Staphylococcus aureus MIC 0.06 ug.mL-1 10.1128/aac.00350-06
Staphylococcus aureus Staphylococcus aureus MIC 0.06 ug.mL-1 10.1128/aac.00915-08
Staphylococcus aureus Staphylococcus aureus MIC 0.06 ug.mL-1 10.1128/aac.01480-07
Staphylococcus aureus Staphylococcus aureus MIC 0.0625 ug.mL-1 10.1016/j.bmcl.2020.127146
Staphylococcus aureus Staphylococcus aureus MIC 0.0625 ug.mL-1 10.1128/aac.00455-10
Staphylococcus aureus Staphylococcus aureus MIC 0.07 ug.mL-1 10.1016/j.ejmech.2012.09.041
Staphylococcus aureus Staphylococcus aureus MIC 0.078 ug.mL-1 10.1021/acs.jnatprod.2c00174
Staphylococcus aureus Staphylococcus aureus MIC 0.1 ug.mL-1 10.1016/j.bmc.2021.116580
Staphylococcus aureus Staphylococcus aureus MIC 0.125 ug.mL-1 10.1016/j.bmcl.2020.127146
Staphylococcus aureus Staphylococcus aureus MIC 0.125 ug.mL-1 10.1016/j.ejmech.2016.12.060
Staphylococcus aureus Staphylococcus aureus MIC 0.125 ug.mL-1 10.1016/j.ejmech.2022.114360
Staphylococcus aureus Staphylococcus aureus MIC 0.125 ug.mL-1 10.1128/aac.01480-07
Staphylococcus aureus Staphylococcus aureus MIC 0.21 ug.mL-1 10.1016/j.bmc.2021.116580
Staphylococcus aureus Staphylococcus aureus MIC 0.25 ug.mL-1 10.1016/j.bmc.2018.02.049
Staphylococcus aureus Staphylococcus aureus MIC 0.25 ug.mL-1 10.1016/j.bmcl.2023.129320
Staphylococcus aureus Staphylococcus aureus MIC 0.25 ug.mL-1 10.1016/j.ejmech.2008.09.035
Staphylococcus aureus Staphylococcus aureus MIC 0.25 ug.mL-1 10.1016/j.ejmech.2019.04.034
Staphylococcus aureus Staphylococcus aureus MIC 0.25 ug.mL-1 10.1021/acs.jnatprod.0c01309
Staphylococcus aureus Staphylococcus aureus MIC 0.25 ug.mL-1 10.1021/np050438i
Staphylococcus aureus Staphylococcus aureus MIC 0.25 ug.mL-1 10.1128/aac.01649-07
Staphylococcus aureus Staphylococcus aureus MIC 0.3 ug.mL-1 10.1016/j.ejmech.2012.09.041
Staphylococcus aureus Staphylococcus aureus MIC 0.3125 ug.mL-1 10.1021/np000436s
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1016/j.bmcl.2020.127146
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1016/j.ejmech.2008.04.001
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1016/j.ejmech.2022.114360
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1021/ml300350p
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1128/aac.00206-09
Staphylococcus aureus Staphylococcus aureus MIC 0.5 ug.mL-1 10.1128/aac.00908-07
Staphylococcus aureus Staphylococcus aureus MIC 0.6 ug.mL-1 10.1016/j.ejmech.2012.09.041
Staphylococcus aureus Staphylococcus aureus MIC 0.625 ug.mL-1 10.1128/aac.00247-08
Staphylococcus aureus Staphylococcus aureus MIC 0.9 ug.mL-1 10.1016/j.ejmech.2007.12.019
Staphylococcus aureus Staphylococcus aureus MIC 1.0 ug.mL-1 10.1128/aac.00458-08
Staphylococcus aureus Staphylococcus aureus MIC 1.0 ug.mL-1 10.1128/aac.00971-08
Staphylococcus aureus Staphylococcus aureus MIC 1.0 ug.mL-1 10.1128/aac.01649-07
Staphylococcus aureus Staphylococcus aureus MIC 1.25 ug.mL-1 10.1016/j.ejmech.2012.09.041
Staphylococcus aureus Staphylococcus aureus MIC 1.562 ug.mL-1 10.1007/s00044-011-9918-4
Staphylococcus aureus Staphylococcus aureus MIC 1.6 ug.mL-1 10.1016/j.ejmech.2017.10.048
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1128/aac.00237-08
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1128/aac.00971-08
Staphylococcus aureus Staphylococcus aureus MIC 2.0 ug.mL-1 10.1128/aac.01649-07
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1016/j.bmcl.2007.02.024
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1021/np200320u
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1128/aac.00846-07
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1128/aac.00971-08
Staphylococcus aureus Staphylococcus aureus MIC 4.0 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC 7.8 nM 10.1021/acs.jmedchem.9b00288
Staphylococcus aureus Staphylococcus aureus MIC 8.0 ug.mL-1 10.1016/j.ejmech.2008.04.001
Staphylococcus aureus Staphylococcus aureus MIC 8.0 ug.mL-1 10.1021/acs.jmedchem.6b00485
Staphylococcus aureus Staphylococcus aureus MIC 8.0 ug.mL-1 10.1128/aac.01649-07
Staphylococcus aureus Staphylococcus aureus MIC 10.0 nM 10.1021/acs.jmedchem.1c02122
Staphylococcus aureus Staphylococcus aureus MIC 10.0 ug.mL-1 10.1021/acs.jnatprod.2c00174
Staphylococcus aureus Staphylococcus aureus MIC 16.0 ug.mL-1 10.1016/j.bmcl.2007.08.048
Staphylococcus aureus Staphylococcus aureus MIC 16.0 ug.mL-1 10.1128/aac.00206-09
Staphylococcus aureus Staphylococcus aureus MIC 16.0 ug.mL-1 10.1128/aac.01649-07
Staphylococcus aureus Staphylococcus aureus MIC 18.0 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC 20.0 nM 10.1021/acs.jmedchem.1c02122
Staphylococcus aureus Staphylococcus aureus MIC 21.0 ug.mL-1 10.1016/j.bmcl.2017.05.032
Staphylococcus aureus Staphylococcus aureus MIC 22.0 ug.mL-1 10.1016/j.bmcl.2017.05.032
Staphylococcus aureus Staphylococcus aureus MIC 31.0 ug.mL-1 10.1016/j.ejmech.2019.04.043
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1016/j.bmc.2006.12.035
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1128/aac.00350-06
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1128/aac.00834-08
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC 32.0 ug.mL-1 10.1128/aac.01649-07
Staphylococcus aureus Staphylococcus aureus MIC 63.0 ug.mL-1 10.1016/j.bmcl.2006.10.016
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1016/j.bmcl.2007.08.048
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1016/j.bmcl.2020.127146
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1016/j.ejmech.2022.114360
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1128/aac.00915-08
Staphylococcus aureus Staphylococcus aureus MIC 64.0 ug.mL-1 10.1128/aac.01649-07
Staphylococcus aureus Staphylococcus aureus MIC 100.0 nM 10.1021/acs.jmedchem.5b02004
Staphylococcus aureus Staphylococcus aureus MIC 100.0 nM 10.1021/acs.jmedchem.7b01903
Staphylococcus aureus Staphylococcus aureus MIC 100.0 nM 10.1021/acs.jnatprod.5b01129
Staphylococcus aureus Staphylococcus aureus MIC 125.0 ug.mL-1 10.1128/aac.01649-07
Staphylococcus aureus Staphylococcus aureus MIC 128.0 ug.mL-1 10.1016/j.bmcl.2016.05.077
Staphylococcus aureus Staphylococcus aureus MIC 128.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Staphylococcus aureus Staphylococcus aureus MIC 128.0 ug.mL-1 10.1128/aac.00350-06
Staphylococcus aureus Staphylococcus aureus MIC 128.0 ug.mL-1 10.1128/aac.01081-09
Staphylococcus aureus Staphylococcus aureus MIC 128.0 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC 250.0 nM 10.1021/acs.jmedchem.9b00288
Staphylococcus aureus Staphylococcus aureus MIC 250.0 ug.mL-1 10.1021/acs.jmedchem.6b00485
Staphylococcus aureus Staphylococcus aureus MIC 250.0 ug.mL-1 10.1128/aac.01649-07
Staphylococcus aureus Staphylococcus aureus MIC 256.0 ug.mL-1 10.1128/aac.00206-09
Staphylococcus aureus Staphylococcus aureus MIC 512.0 ug.mL-1 10.1128/aac.00846-07
Staphylococcus aureus Staphylococcus aureus MIC 1000.0 nM 10.1016/j.ejmech.2019.111636
Staphylococcus aureus Staphylococcus aureus MIC 1000.0 nM 10.1021/acs.jmedchem.1c00614
Staphylococcus aureus Staphylococcus aureus MIC 1000.0 nM 10.1021/acs.jmedchem.1c02140
Staphylococcus aureus Staphylococcus aureus MIC 1000.0 nM 10.1021/acs.jmedchem.2c01076
Staphylococcus aureus Staphylococcus aureus MIC 1000.0 nM 10.1021/acs.jnatprod.2c00481
Staphylococcus aureus Staphylococcus aureus MIC 1000.0 ug.mL-1 10.1016/j.bmc.2015.09.027
Staphylococcus aureus Staphylococcus aureus MIC 1024.0 ug.mL-1 10.1128/aac.00209-07
Staphylococcus aureus Staphylococcus aureus MIC 1250.0 nM 10.1021/acs.jmedchem.1c01809
Staphylococcus aureus Staphylococcus aureus MIC 1900.0 nM 10.1021/acs.jnatprod.1c00232
Staphylococcus aureus Staphylococcus aureus MIC 2048.0 ug.mL-1 10.1128/aac.01544-08
Staphylococcus aureus Staphylococcus aureus MIC 4096.0 ug.mL-1 10.1016/j.bmc.2006.12.035
Staphylococcus aureus Staphylococcus aureus MIC 15400.0 nM 10.1021/acs.jnatprod.2c00481
Staphylococcus aureus Staphylococcus aureus MIC 25923000.0 nM 10.1021/acs.jmedchem.1c02140
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1016/j.bmc.2010.05.016
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1016/j.bmc.2013.10.011
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1016/j.bmc.2019.04.032
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1016/j.bmcl.2012.08.003
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1016/j.bmcl.2013.11.024
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1021/np050424c
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1021/np200320u
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1021/np900281r
Staphylococcus aureus Staphylococcus aureus MIC nan None 10.1128/aac.00455-10
Staphylococcus aureus Staphylococcus aureus MIC100 0.15 ug ml-1 10.1016/j.bmc.2018.07.034
Staphylococcus aureus Staphylococcus aureus MIC100 0.2 ug ml-1 10.1016/j.bmc.2018.07.034
Staphylococcus aureus Staphylococcus aureus MIC100 6.25 ug ml-1 10.1016/j.bmc.2018.07.034
Staphylococcus aureus Staphylococcus aureus MIC100 25.0 ug ml-1 10.1016/j.bmc.2018.07.034
Staphylococcus aureus Staphylococcus aureus MIC50 0.004 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC50 0.008 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC50 0.015 ug.mL-1 10.1021/acs.jmedchem.6b00485
Staphylococcus aureus Staphylococcus aureus MIC50 0.016 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC90 0.015 ug.mL-1 10.1021/acs.jmedchem.6b00485
Staphylococcus aureus Staphylococcus aureus MIC90 0.016 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC90 0.5 ug.mL-1 10.1128/aac.00846-07
Staphylococcus aureus Staphylococcus aureus MIC90 2.0 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC90 16.0 ug.mL-1 10.1128/aac.01619-08
Staphylococcus aureus Staphylococcus aureus MIC99 nan None 10.1016/j.ejmech.2013.10.055
Staphylococcus aureus Staphylococcus aureus PAE 1.8 hr 10.1016/j.bmcl.2023.129320
Staphylococcus aureus Staphylococcus aureus PAE 3.45 hr 10.1016/j.bmcl.2023.129320
Staphylococcus aureus Staphylococcus aureus Ratio 4.5 None 10.1128/aac.00120-07
Staphylococcus aureus Staphylococcus aureus Ratio 7.0 None 10.1021/acs.jmedchem.9b00720
Staphylococcus aureus Staphylococcus aureus Ratio 23.0 None 10.1021/acs.jmedchem.5b02004
Staphylococcus aureus Staphylococcus aureus Ratio 29.0 None 10.1016/j.ejmech.2018.03.044
Staphylococcus aureus Staphylococcus aureus Ratio 29.0 None 10.1016/j.ejmech.2019.04.063
Staphylococcus aureus Staphylococcus aureus Ratio 533.0 None 10.1128/aac.00458-08
Staphylococcus aureus Staphylococcus aureus Ratio 2000.0 None 10.1016/j.bmc.2019.02.024
Staphylococcus aureus Staphylococcus aureus Ratio 40000.0 None 10.1016/j.ejmech.2017.10.048
Staphylococcus aureus Staphylococcus aureus Ratio 500000.0 None 10.1016/j.ejmech.2018.03.044
Staphylococcus aureus Staphylococcus aureus Ratio 500000.0 None 10.1016/j.ejmech.2019.04.063
Staphylococcus aureus Staphylococcus aureus Ratio 500000.0 None 10.1021/acs.jmedchem.9b00720
Staphylococcus aureus Staphylococcus aureus T1/2 3.56 hr 10.1128/aac.00455-10
Staphylococcus epidermidis Staphylococcus epidermidis Activity nan None 10.1128/aac.00343-07
Staphylococcus epidermidis Staphylococcus epidermidis Inhibition 100.0 % 10.1021/jm0703901
Staphylococcus epidermidis Staphylococcus epidermidis IZ 40.0 mm 10.1016/j.bmc.2018.02.049
Staphylococcus epidermidis Staphylococcus epidermidis log10cfu 0.17 None 10.1128/aac.00237-08
Staphylococcus epidermidis Staphylococcus epidermidis log10cfu 2.5 None 10.1128/aac.00237-08
Staphylococcus epidermidis Staphylococcus epidermidis MBC 0.006 ug ml-1 10.1128/aac.00343-07
Staphylococcus epidermidis Staphylococcus epidermidis MBC 0.25 ug ml-1 10.1128/aac.01011-09
Staphylococcus epidermidis Staphylococcus epidermidis MBC 3.0 uM 10.1021/acs.jmedchem.5b02004
Staphylococcus epidermidis Staphylococcus epidermidis MBC 3.0 uM 10.1021/acs.jmedchem.7b01903
Staphylococcus epidermidis Staphylococcus epidermidis MBEC 15.6 uM 10.1021/acs.jmedchem.5b02004
Staphylococcus epidermidis Staphylococcus epidermidis MBEC 15.6 uM 10.1021/acs.jmedchem.7b01903
Staphylococcus epidermidis Staphylococcus epidermidis MBEC 50.0 ug ml-1 10.1128/aac.00457-09
Staphylococcus epidermidis Staphylococcus epidermidis MBIC 0.2 ug ml-1 10.1128/aac.00457-09
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.004 ug.mL-1 10.1016/j.ejmech.2014.07.066
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.004 ug.mL-1 10.1016/j.ejmech.2016.03.061
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.004 ug.mL-1 10.1021/acs.jmedchem.6b00485
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.006 ug.mL-1 10.1128/aac.00343-07
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.008 ug.mL-1 10.1016/j.bmcl.2015.07.043
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.008 ug.mL-1 10.1016/j.bmcl.2016.05.077
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.008 ug.mL-1 10.1016/j.ejmech.2016.03.061
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.008 ug.mL-1 10.1021/jm00167a029
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.008 ug.mL-1 10.1128/aac.01011-09
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.008 ug.mL-1 10.1128/aac.01619-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.012 ug.mL-1 10.1128/aac.00457-09
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.0156 ug.mL-1 10.1016/j.ejmech.2019.02.009
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.016 ug.mL-1 10.1128/aac.01619-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.03 ug.mL-1 10.1021/acs.jmedchem.0c00520
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.03 ug.mL-1 10.1021/jm501082n
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.03 ug.mL-1 10.1128/aac.01619-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.078 ug.mL-1 10.1021/acs.jnatprod.2c00174
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.125 ug.mL-1 10.1128/aac.00237-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.25 ug.mL-1 10.1016/j.bmc.2018.02.049
Staphylococcus epidermidis Staphylococcus epidermidis MIC 0.25 ug.mL-1 10.1016/j.ejmech.2019.04.034
Staphylococcus epidermidis Staphylococcus epidermidis MIC 1.0 ug.mL-1 10.1016/j.ejmech.2022.114360
Staphylococcus epidermidis Staphylococcus epidermidis MIC 20.0 nM 10.1021/acs.jmedchem.1c02122
Staphylococcus epidermidis Staphylococcus epidermidis MIC 100.0 nM 10.1021/acs.jmedchem.5b02004
Staphylococcus epidermidis Staphylococcus epidermidis MIC 100.0 nM 10.1021/acs.jmedchem.7b01903
Staphylococcus epidermidis Staphylococcus epidermidis MIC 100.0 nM 10.1021/acs.jnatprod.5b01129
Staphylococcus epidermidis Staphylococcus epidermidis MIC 128.0 ug.mL-1 10.1128/aac.01619-08
Staphylococcus epidermidis Staphylococcus epidermidis MIC 250.0 nM 10.1021/acs.jmedchem.9b00288
Staphylococcus epidermidis Staphylococcus epidermidis MIC 1000.0 nM 10.1021/acs.jmedchem.1c00614
Staphylococcus epidermidis Staphylococcus epidermidis MIC 1000.0 nM 10.1021/acs.jmedchem.1c02140
Staphylococcus epidermidis Staphylococcus epidermidis MIC50 0.015 ug.mL-1 10.1021/acs.jmedchem.6b00485
Staphylococcus epidermidis Staphylococcus epidermidis MIC90 0.015 ug.mL-1 10.1021/acs.jmedchem.6b00485
Staphylococcus epidermidis Staphylococcus epidermidis MIC90 4.0 ug.mL-1 10.1021/acs.jmedchem.6b00485
Staphylococcus epidermidis Staphylococcus epidermidis Ratio 1.0 None 10.1128/aac.00343-07
Staphylococcus lugdunensis Staphylococcus lugdunensis Activity 0.0 % 10.1128/aac.01052-06
Staphylococcus lugdunensis Staphylococcus lugdunensis Activity 7.0 % 10.1128/aac.01052-06
Staphylococcus lugdunensis Staphylococcus lugdunensis Activity 93.0 % 10.1128/aac.01052-06
Staphylococcus lugdunensis Staphylococcus lugdunensis BBC 0.125 ug ml-1 10.1128/aac.01052-06
Staphylococcus lugdunensis Staphylococcus lugdunensis BBC 0.25 ug ml-1 10.1128/aac.01052-06
Staphylococcus lugdunensis Staphylococcus lugdunensis BBC 8.0 ug ml-1 10.1128/aac.01052-06
Staphylococcus lugdunensis Staphylococcus lugdunensis BBC 32.0 ug ml-1 10.1128/aac.01052-06
Staphylococcus lugdunensis Staphylococcus lugdunensis BBC 64.0 ug ml-1 10.1128/aac.01052-06
Staphylococcus lugdunensis Staphylococcus lugdunensis MBC50 8.0 ug ml-1 10.1128/aac.01052-06
Staphylococcus lugdunensis Staphylococcus lugdunensis MBC90 32.0 ug ml-1 10.1128/aac.01052-06
Staphylococcus lugdunensis Staphylococcus lugdunensis MIC50 0.03 ug.mL-1 10.1128/aac.01052-06
Staphylococcus lugdunensis Staphylococcus lugdunensis MIC90 0.03 ug.mL-1 10.1128/aac.01052-06
Staphylococcus saprophyticus Staphylococcus saprophyticus MIC 0.03 ug.mL-1 10.1021/acs.jmedchem.0c00520
Stenotrophomonas maltophilia Stenotrophomonas maltophilia MIC 32.0 ug.mL-1 10.1016/j.ejmech.2019.04.034
Streptococcus agalactiae Streptococcus agalactiae MIC 0.03 ug.mL-1 10.1021/acs.jmedchem.0c00520
Streptococcus agalactiae Streptococcus agalactiae MIC 0.03 ug.mL-1 10.1021/acs.jmedchem.6b00485
Streptococcus agalactiae Streptococcus agalactiae MIC50 0.12 ug.mL-1 10.1021/acs.jmedchem.6b00485
Streptococcus agalactiae Streptococcus agalactiae MIC90 0.12 ug.mL-1 10.1021/acs.jmedchem.6b00485
Streptococcus pneumoniae Streptococcus pneumoniae Activity 0.8 % 10.1128/aac.01384-06
Streptococcus pneumoniae Streptococcus pneumoniae Activity 98.8 % 10.1128/aac.01384-06
Streptococcus pneumoniae Streptococcus pneumoniae Activity nan None 10.1021/acs.jmedchem.0c00520
Streptococcus pneumoniae Streptococcus pneumoniae IZ 25.0 mm 10.1016/j.bmcl.2016.04.038
Streptococcus pneumoniae Streptococcus pneumoniae MBC 25.0 ug ml-1 10.1016/j.bmc.2018.07.034
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.004 ug.mL-1 10.1021/np050176k
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.0625 ug.mL-1 10.1016/j.ejmech.2019.05.090
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.0625 ug.mL-1 10.1021/acs.jmedchem.0c00520
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.063 ug.mL-1 10.1021/jm00167a029
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.12 ug.mL-1 10.1021/acs.jmedchem.6b00485
Streptococcus pneumoniae Streptococcus pneumoniae MIC 0.25 ug.mL-1 10.1016/j.ejmech.2019.04.034
Streptococcus pneumoniae Streptococcus pneumoniae MIC 10.0 nM 10.1021/acs.jnatprod.2c00481
Streptococcus pneumoniae Streptococcus pneumoniae MIC 20.0 nM 10.1021/acs.jnatprod.2c00481
Streptococcus pneumoniae Streptococcus pneumoniae MIC 110.0 nM 10.1021/acs.jmedchem.1c02122
Streptococcus pneumoniae Streptococcus pneumoniae MIC100 25.0 ug ml-1 10.1016/j.bmc.2018.07.034
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.03 ug.mL-1 10.1128/aac.01384-06
Streptococcus pneumoniae Streptococcus pneumoniae MIC50 0.25 ug.mL-1 10.1021/acs.jmedchem.6b00485
Streptococcus pneumoniae Streptococcus pneumoniae MIC>90 0.01 ug ml-1 10.1021/np400145u
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.03 ug.mL-1 10.1128/aac.01384-06
Streptococcus pneumoniae Streptococcus pneumoniae MIC90 0.25 ug.mL-1 10.1021/acs.jmedchem.6b00485
Streptococcus pyogenes Streptococcus pyogenes ED50 0.35 mg.kg-1 10.1021/jm00167a029
Streptococcus pyogenes Streptococcus pyogenes ED50 0.47 mg.kg-1 10.1021/jm00167a029
Streptococcus pyogenes Streptococcus pyogenes Inhibition 10.0 % 10.1128/aac.00471-08
Streptococcus pyogenes Streptococcus pyogenes Inhibition 100.0 % 10.1021/jm0703901
Streptococcus pyogenes Streptococcus pyogenes Inhibition nan % 10.1128/aac.00471-08
Streptococcus pyogenes Streptococcus pyogenes log10cfu 6.44 None 10.1128/aac.00471-08
Streptococcus pyogenes Streptococcus pyogenes MIC 0.00025 ug.mL-1 10.1128/aac.00471-08
Streptococcus pyogenes Streptococcus pyogenes MIC 0.008 ug.mL-1 10.1021/acs.jmedchem.6b00485
Streptococcus pyogenes Streptococcus pyogenes MIC 0.03 ug.mL-1 10.1021/acs.jmedchem.0c00520
Streptococcus pyogenes Streptococcus pyogenes MIC 0.063 ug.mL-1 10.1021/jm00167a029
Streptococcus pyogenes Streptococcus pyogenes MIC nan None 10.1021/np050424c
Streptococcus pyogenes Streptococcus pyogenes MIC50 0.06 ug.mL-1 10.1021/acs.jmedchem.6b00485
Streptococcus pyogenes Streptococcus pyogenes MIC90 0.12 ug.mL-1 10.1021/acs.jmedchem.6b00485
Streptococcus salivarius Streptococcus salivarius MBC 25.0 ug ml-1 10.1016/j.bmc.2018.07.034
Streptococcus salivarius Streptococcus salivarius MIC100 0.2 ug ml-1 10.1016/j.bmc.2018.07.034
Streptomyces albus Streptomyces albus MIC 5.0 ug.mL-1 10.1128/aac.01406-09
Streptomyces albus Streptomyces albus MIC 20.0 ug.mL-1 10.1128/aac.01406-09
Streptomyces albus Streptomyces albus MIC 40.0 ug.mL-1 10.1128/aac.01406-09
Treponema denticola Treponema denticola MIC 0.004 ug.mL-1 10.1021/acs.jmedchem.1c02045
Trichophyton rubrum Trichophyton rubrum MIC 1.0 ug.mL-1 10.1016/j.ejmech.2014.07.066
Veillonella parvula Veillonella parvula MIC 4.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
Vibrio cholerae Vibrio cholerae MIC 128000.0 nM 10.1021/acs.jmedchem.1c02122
Xanthomonas campestris Xanthomonas campestris MIC 32.0 ug.mL-1 10.1016/j.bmcl.2015.01.026
Yersinia pseudotuberculosis Yersinia pseudotuberculosis MIC 11000.0 nM 10.1021/acs.jmedchem.1c02122
None ADMET Activity 0.0 % 10.1021/np50025a010
None ADMET Activity 1.0 % 10.1021/np50025a010
None ADMET Activity 4.0 % 10.1021/np50025a010
None ADMET Activity 48.0 % 10.1021/np50025a010
None ADMET Activity 52.7 % 10.1021/acs.jmedchem.5b00608
None ADMET Activity 58.0 % 10.1021/np50025a010
None ADMET Activity 66.0 % 10.1021/np50025a010
None ADMET Activity 82.0 % 10.1021/np50025a010
None ADMET Activity 85.0 % 10.1016/j.ejmech.2013.09.061
None ADMET Activity 93.0 % 10.1016/j.ejmech.2013.09.061
None ADMET Activity 94.0 % 10.1016/j.ejmech.2013.09.061
None ADMET Activity 98.3 % 10.1021/acs.jmedchem.5b00608
None ADMET Activity 103.1 % 10.1021/acs.jmedchem.5b00608
None ADMET Activity 105.6 % 10.1021/acs.jmedchem.5b00608
None ADMET Activity nan None 10.1016/j.ejmech.2015.10.049
None ADMET AUC 0.0 ng.hr.mL-1 10.1128/aac.01533-06
None ADMET AUC 4600.0 ng.hr.mL-1 10.1128/aac.00775-08
None ADMET AUC 7000.0 ng.hr.mL-1 10.1128/aac.01533-06
None ADMET AUC 14000.0 ng.hr.mL-1 10.1128/aac.01533-06
None ADMET AUC 64400.0 ng.hr.mL-1 10.1128/aac.01544-08
None ADMET AUC 122000.0 ng.hr.mL-1 10.1128/aac.01533-06
None ADMET AUC 304000.0 ng.hr.mL-1 10.1128/aac.00458-08
None ADMET BPR 0.03 None 10.1021/jm901036q
None ADMET CC50 100.0 ug.mL-1 10.1016/j.bmcl.2016.05.093
None ADMET CL 0.0 mL.min-1.g-1 10.1124/dmd.111.043067
None ADMET CL 0.2 mL.min-1.g-1 10.1124/dmd.111.043067
None ADMET CL 0.7 mL.min-1.g-1 10.1124/dmd.111.043067
None ADMET CL 3.5 mL.min-1.kg-1 10.1124/dmd.108.020479
None ADMET CL 32.0 mL.min-1.kg-1 10.1021/jm000407e
None ADMET CL 99.0 L/hr 10.1128/aac.01533-06
None ADMET Cmax 1215.14 nM 10.1128/aac.00775-08
None ADMET Cmax 5954.19 nM 10.1128/aac.01544-08
None ADMET Cmax 8019.93 nM 10.1128/aac.00458-08
None ADMET Cmax 13000.0 nM 10.1021/acs.jmedchem.9b01071
None ADMET Cmin 0.1 ug ml-1 10.1128/aac.00775-08
None ADMET Cmin 1.3 ug ml-1 10.1128/aac.01544-08
None ADMET Cmin 3.8 mg/L 10.1128/aac.00458-08
None ADMET Drug metabolism 90.0 % 10.1016/j.bmcl.2019.07.001
None ADMET Drug metabolism nan None 10.1016/j.bmcl.2019.07.001
None ADMET Drug uptake 10.0 ug ml-1 10.1128/aac.00985-07
None ADMET Fu 0.118 None 10.1124/dmd.111.038778
None ADMET GI50 100.0 ug.mL-1 10.1016/j.bmcl.2016.03.045
None ADMET GI50 100.0 ug.mL-1 10.1039/C5MD00404G
None ADMET IC50 20000.0 nM 10.1021/acs.jmedchem.5b00608
None ADMET IC50 100000.0 nM 10.1016/j.ejmech.2013.01.017
None ADMET IC50 100000.0 nM 10.1021/jm401735w
None ADMET IC50 nan None 10.1016/j.ejmech.2013.06.010
None ADMET Inhibition nan % 10.1016/j.bmcl.2016.04.012
None ADMET Ki 50000.0 nM 10.1021/np50025a010
None ADMET Ki 100000.0 nM 10.1021/np50025a010
None ADMET Ki 140000.0 nM 10.1021/np50025a010
None ADMET K(p,uu,brain) 0.035 None 10.1021/jm901036q
None ADMET MRT 4.6 hr 10.1124/dmd.108.020479
None ADMET PPB 64.0 % 10.1128/aac.00971-08
None ADMET Ratio 1.0 None 10.1128/aac.00971-08
None ADMET Selectivity Index 643.12 None 10.1016/j.ejmech.2021.113472
None ADMET Selectivity Index 1407.2 None 10.1016/j.ejmech.2021.113472
None ADMET Selectivity Index nan None 10.1016/j.bmc.2022.116777
None ADMET Stability nan % 10.1021/acs.jmedchem.2c01076
None ADMET Stability nan % 10.1021/acs.jmedchem.5b01542
None ADMET Survival nan None 10.1016/j.ejmech.2019.06.038
None ADMET T1/2 2.5 hr 10.1128/aac.00775-08
None ADMET T1/2 3.5 hr 10.1021/jm000407e
None ADMET T1/2 3.8 hr 10.1124/dmd.108.020479
None ADMET T1/2 4.1 hr 10.1128/aac.01544-08
None ADMET T1/2 4.7 hr 10.1016/j.bmc.2016.11.008
None ADMET T1/2 9.3 hr 10.1016/j.bmc.2016.11.008
None ADMET TI nan None 10.1016/j.ejmech.2013.06.010
None ADMET TI nan None 10.1016/j.ejmech.2017.06.061
None ADMET Tmax 1.5 hr 10.1021/acs.jmedchem.9b01071
None ADMET Tmax 2.1 hr 10.1128/aac.00775-08
None ADMET Vc 430.89 l 10.1128/aac.01533-06
None ADMET Vd 8.8 L.kg-1 10.1021/jm000407e
None ADMET Vd 33.65 l 10.1128/aac.01520-08
None ADMET Vd 43.66 l 10.1128/aac.01520-08
None ADMET Vd 49.94 l 10.1128/aac.01520-08
None ADMET Vd 52.1 l 10.1128/aac.01520-08
None ADMET Vd 102.6 l 10.1128/aac.01520-08
None ADMET Vd 102.8 l 10.1128/aac.01520-08
None ADMET Vdss 0.97 L.kg-1 10.1124/dmd.108.020479
None Erythrocyte LC50 nan None 10.1021/acs.jnatprod.5b01129
None Erythrocyte MHC10 nan None 10.1021/acs.jmedchem.2c01076
None Hepatotoxicity Alkaline Phosphatase Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity Alkaline Phosphatase Increase - Index Value nan None 10.2174/1570163043334794
None Hepatotoxicity Alkaline Phosphatase Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None Hepatotoxicity Composite Activity - Active 1.0 None 10.2174/1570163043334794
None Hepatotoxicity Composite Activity - Marginal 3.0 None 10.2174/1570163043334794
None Hepatotoxicity Composite Activity - Score nan None 10.2174/1570163043334794
None Hepatotoxicity GGT Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity GGT Increase - Index Value nan None 10.2174/1570163043334794
None Hepatotoxicity GGT Increase - Number of Reports nan None 10.2174/1570163043334794
None Hepatotoxicity Hepatotoxicity nan None 10.1021/tx1000865
None Hepatotoxicity Hepatotoxicity nan None 10.1021/tx900326k
None Hepatotoxicity Hepatotoxicity nan None 10.1124/dmd.110.035113
None Hepatotoxicity HepSE_bilirubinemia 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_cholecystitis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_cholelithiasis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_cirrhosis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_Combined Scores 3.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_elevated liver function tests 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatic failure 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatic necrosis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatitis 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatomegaly 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_jaundice 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_liver disease 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_liver fatty 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_liver function tests abnormal 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity LDH Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity LDH Increase - Index Value nan None 10.2174/1570163043334794
None Hepatotoxicity LDH Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None Hepatotoxicity LTKB_BD DILI severity score 8.0 None 10.1016/j.drudis.2011.05.007
None Hepatotoxicity SGOT Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity SGOT Increase - Index Value nan None 10.2174/1570163043334794
None Hepatotoxicity SGOT Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None Hepatotoxicity SGPT Increase - Activity Score nan None 10.2174/1570163043334794
None Hepatotoxicity SGPT Increase - Index Value nan None 10.2174/1570163043334794
None Hepatotoxicity SGPT Increase - Number of Reports 4.0 None 10.2174/1570163043334794
None Lipid bilayer Activity nan None 10.1016/j.ejmech.2016.07.068
None Molecular identity unknown PPB 91.0 % 10.1021/jm501661f
None NON-PROTEIN TARGET Activity nan None 10.1016/j.ejmech.2016.07.005
None NON-PROTEIN TARGET Activity nan None 10.1021/acs.jmedchem.6b00624
None NON-PROTEIN TARGET fAUC/MIC 300.0 None 10.1016/j.bmcl.2013.07.006
None NON-PROTEIN TARGET fCmax/MIC 20.0 None 10.1016/j.bmcl.2013.07.006
None NON-PROTEIN TARGET fT>MIC 100.0 % 10.1016/j.bmcl.2013.07.006
None NON-PROTEIN TARGET Fu 0.119 None 10.1124/dmd.111.038778
None NON-PROTEIN TARGET Fu 0.2 None 10.1124/dmd.108.020479
None NON-PROTEIN TARGET Fu 0.62 None 10.1021/jm401963n
None NON-PROTEIN TARGET GI nan None 10.1016/j.ejmech.2016.06.042
None NON-PROTEIN TARGET GI50 100.0 ug.mL-1 10.1016/j.bmcl.2016.11.056
None NON-PROTEIN TARGET GI90 100.0 ug ml-1 10.1016/j.bmcl.2016.11.056
None NON-PROTEIN TARGET Hepatotoxicity (acute) 7.3 % 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (animal toxicity known) nan None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (benign tumour) 0.0 None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (granulomatous hepatitis) 0.0 None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (mechanism) nan None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (moderate) 22.0 None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (moderate) 23.0 % 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (time to onset) nan None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET IC20 30.0 ug ml-1 10.1128/aac.00729-05
None NON-PROTEIN TARGET IC50 0.0016 ug.mL-1 10.1016/j.bmcl.2016.02.056
None NON-PROTEIN TARGET IC50 0.45 ug.mL-1 10.1016/j.bmcl.2016.11.056
None NON-PROTEIN TARGET IC50 0.51 ug.mL-1 10.1016/j.bmcl.2016.11.056
None NON-PROTEIN TARGET IC50 0.75 ug.mL-1 10.1016/j.bmcl.2016.11.056
None NON-PROTEIN TARGET IC50 0.81 ug.mL-1 10.1016/j.bmcl.2016.11.056
None NON-PROTEIN TARGET IC50 130.0 ug.mL-1 10.1128/aac.00729-05
None NON-PROTEIN TARGET IC50 96000.0 nM 10.1128/aac.00126-08
None NON-PROTEIN TARGET IC50 nan None 10.1016/j.bmcl.2016.11.003
None NON-PROTEIN TARGET IC50 nan None 10.1016/j.ejmech.2016.07.039
None NON-PROTEIN TARGET IC90 0.041 ug.mL-1 10.1016/j.bmcl.2016.02.056
None NON-PROTEIN TARGET IC90 0.061 ug.mL-1 10.1016/j.bmcl.2016.03.045
None NON-PROTEIN TARGET IC90 0.89 ug.mL-1 10.1016/j.bmcl.2016.03.045
None NON-PROTEIN TARGET Inhibition 75.0 % 10.1128/aac.00126-08
None NON-PROTEIN TARGET MIC 0.004 ug.mL-1 10.1016/j.bmcl.2009.09.095
None NON-PROTEIN TARGET MIC 0.004 ug.mL-1 10.1016/j.bmcl.2010.12.084
None NON-PROTEIN TARGET MIC 0.004 ug.mL-1 10.1128/aac.00477-09
None NON-PROTEIN TARGET MIC 0.008 ug.mL-1 10.1128/aac.00477-09
None NON-PROTEIN TARGET MIC 0.03 ug.mL-1 10.1128/aac.01052-07
None NON-PROTEIN TARGET MIC 0.06 ug.mL-1 10.1128/aac.01052-07
None NON-PROTEIN TARGET MIC 0.12 ug.mL-1 10.1128/aac.01052-07
None NON-PROTEIN TARGET MIC 0.25 ug.mL-1 10.1016/j.bmcl.2010.12.084
None NON-PROTEIN TARGET MIC 0.25 ug.mL-1 10.1128/aac.00477-09
None NON-PROTEIN TARGET MIC 0.89 ug.mL-1 10.1016/j.bmcl.2016.03.045
None NON-PROTEIN TARGET MIC 1.0 ug.mL-1 10.1128/aac.01052-07
None NON-PROTEIN TARGET MIC 2.0 ug.mL-1 10.1128/aac.01052-07
None NON-PROTEIN TARGET MIC 4.0 ug.mL-1 10.1128/aac.01052-07
None NON-PROTEIN TARGET MIC 4.8 ug.mL-1 10.1016/j.ejmech.2013.04.060
None NON-PROTEIN TARGET MIC 16.0 ug.mL-1 10.1128/aac.00477-09
None NON-PROTEIN TARGET MIC 40.0 ug.mL-1 10.1128/aac.01406-09
None NON-PROTEIN TARGET MIC 128.0 ug.mL-1 10.1128/aac.00477-09
None NON-PROTEIN TARGET MIC 1890.0 nM 10.1016/j.bmcl.2010.06.096
None NON-PROTEIN TARGET MIC 15180.0 nM 10.1016/j.bmcl.2010.06.096
None NON-PROTEIN TARGET MIC90 0.45 ug.mL-1 10.1016/j.bmcl.2016.11.056
None NON-PROTEIN TARGET MIC90 0.45 ug.mL-1 10.1039/C5MD00404G
None NON-PROTEIN TARGET MIC90 0.5 ug.mL-1 10.1016/j.bmcl.2016.11.056
None NON-PROTEIN TARGET MIC90 0.51 ug.mL-1 10.1016/j.bmcl.2016.11.056
None NON-PROTEIN TARGET MIC90 0.7 ug.mL-1 10.1016/j.bmcl.2016.11.056
None NON-PROTEIN TARGET MIC90 0.75 ug.mL-1 10.1016/j.bmcl.2016.11.056
None NON-PROTEIN TARGET MIC90 0.81 ug.mL-1 10.1016/j.bmcl.2016.11.056
None NON-PROTEIN TARGET MIC90 0.81 ug.mL-1 10.1039/C5MD00404G
None NON-PROTEIN TARGET MIC95 0.24 uM 10.1016/j.bmc.2011.05.028
None NON-PROTEIN TARGET RatioAUC/MIC 271.0 None 10.1128/aac.01520-08
None NON-PROTEIN TARGET RatioAUC/MIC 665.0 None 10.1128/aac.01520-08
None NON-PROTEIN TARGET RatioAUC/MIC 1500.0 None 10.1016/j.bmcl.2013.07.006
None NON-PROTEIN TARGET %T>MIC 100.0 % 10.1016/j.bmcl.2013.07.006
None NON-PROTEIN TARGET T>MIC 6.54 hr 10.1128/aac.00367-09
None NON-PROTEIN TARGET T>MIC 7.5 hr 10.1128/aac.00367-09
None No relevant target Activity 0.0 mol/mol 10.1016/j.ejmech.2016.07.039
None No relevant target IC50 nan None 10.1016/j.bmcl.2015.11.071
None No relevant target Kinetic_solubility nan None 10.1016/j.ejmech.2012.08.047
None No relevant target Kinetic_solubility nan None 10.1021/acs.jmedchem.1c00707
None No relevant target Kinetic_solubility nan None 10.1021/acs.jmedchem.5b01542
None No relevant target LogD 1.3 None 10.1021/acs.jmedchem.5b00050
None No relevant target LogD 1.31 None 10.1016/j.ejmech.2022.114434
None No relevant target LogD 1.67 None 10.1021/jm901858n
None No relevant target LogP 1.66 None 10.1016/j.bmcl.2015.07.043
None No relevant target LogP 1.66 None 10.1016/j.ejmech.2014.07.066
None No relevant target LogP 1.66 None 10.1016/j.ejmech.2016.03.061
None No relevant target LogP 1.66 None 10.1016/j.ejmech.2019.02.009
None No relevant target LogP 3.72 None 10.1016/j.bmc.2018.07.049
None No relevant target LogP nan None 10.1016/j.ejmech.2016.07.039
None No relevant target LogP nan None 10.1021/acs.jmedchem.7b01332
None No relevant target -log(solubility) 4.01 None 10.1016/j.bmcl.2015.02.013
None No relevant target -log(solubility) 4.02 None 10.1016/j.bmcl.2015.02.013
None No relevant target -log(solubility) 4.14 None 10.1016/j.bmcl.2015.02.013
None No relevant target -log(solubility) 4.21 None 10.1016/j.bmcl.2015.02.013
None No relevant target -log(solubility) 4.31 None 10.1016/j.bmcl.2015.02.013
None No relevant target pKa 2.2 None 10.1124/dmd.110.035998
None No relevant target pKa 7.6 None 10.1124/dmd.110.035998
None No relevant target solubility nan None 10.1016/j.bmc.2017.09.037
None No relevant target Solubility 1400.0 ug.mL-1 10.1016/j.bmcl.2015.07.043
None No relevant target Solubility 1400.0 ug.mL-1 10.1016/j.ejmech.2014.07.066
None No relevant target Solubility 1400.0 ug.mL-1 10.1016/j.ejmech.2016.03.061
None No relevant target Solubility 1400.0 ug.mL-1 10.1016/j.ejmech.2019.02.009
None No relevant target Solubility 174900.0 nM 10.1016/j.ejmech.2022.114434
None No relevant target Solubility 183300.0 nM 10.1016/j.ejmech.2020.112497
None No relevant target Solubility 751000.0 nM 10.1021/acs.jmedchem.5b00050
None Osteoblast Activity 40.0 % 10.1128/aac.00729-05
None Osteoblast IC20 nan None 10.1128/aac.00729-05
None Osteoblast IC50 nan None 10.1128/aac.00729-05
None Phospholipidosis Phospholipidosis nan None 10.1021/ci6004542
None Phospholipidosis Phospholipidosis nan None 10.1021/mp100103e
None Unchecked AbsAC90 6.43 uM None
None Unchecked Ac50 0.5623 uM None
None Unchecked Ac50 14.13 uM None
None Unchecked Ac50 19.95 uM None
None Unchecked Ac50 22.39 uM None
None Unchecked Ac50 28.18 uM None
None Unchecked Ac50 44.67 uM None
None Unchecked AC50 562.3 nM None
None Unchecked AC50 14130.0 nM None
None Unchecked AC50 19952.6 nM None
None Unchecked AC50 22387.2 nM None
None Unchecked AC50 28183.8 nM None
None Unchecked AC50 44668.4 nM None
None Unchecked Activity 0.0 % 10.1128/aac.00126-08
None Unchecked Activity 2.43 % 10.1128/aac.00126-08
None Unchecked Activity 66.9 % 10.1016/j.ejmech.2016.07.005
None Unchecked Activity 67.1 % 10.1016/j.ejmech.2015.10.049
None Unchecked Activity 97.57 % 10.1128/aac.00126-08
None Unchecked Activity nan None 10.1016/j.ejmech.2010.07.050
None Unchecked Activity nan None 10.1021/acs.jmedchem.1c02140
None Unchecked Activity nan None 10.1021/jm200201k
None Unchecked Activity nan None 10.1124/mol.60.5.934
None Unchecked CC50 72000.0 nM 10.1021/acs.jmedchem.8b01293
None Unchecked CC50 nan None 10.1021/acs.jmedchem.2c01076
None Unchecked FC 8.0 None 10.1016/j.ejmech.2022.114204
None Unchecked FC 64.0 None 10.1021/acs.jmedchem.1c02140
None Unchecked FC 4096.0 None 10.1016/j.ejmech.2022.114360
None Unchecked FC 500000.0 None 10.1016/j.ejmech.2022.114204
None Unchecked Hepatotoxicity (acute) 38.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (association with vascular disease) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (choleostasis) 19.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (chronic liver disease) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (cirrhosis) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (comment) nan None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (cytolytic) 14.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (malignant tumour) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (severe hepatitis) 6.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (steatosis) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (successful reintroduction) nan None 10.1016/s0399-8320(04)95062-2
None Unchecked IC50 0.04 ug.mL-1 10.1128/aac.00343-07
None Unchecked IC50 11.5 nM 10.1128/aac.00753-10
None Unchecked IC50 12.0 nM 10.1021/jm4004889
None Unchecked IC50 14.0 nM 10.1021/acs.jmedchem.5b00050
None Unchecked IC50 15.0 nM 10.1021/acs.jmedchem.6b00485
None Unchecked IC50 15.0 nM 10.1128/aac.01649-07
None Unchecked IC50 16.0 nM 10.1021/jm400485e
None Unchecked IC50 17.0 nM 10.1021/jm4004889
None Unchecked IC50 27.0 nM 10.1021/jm400485e
None Unchecked IC50 30.0 nM 10.1016/j.ejmech.2013.04.060
None Unchecked IC50 30.0 nM 10.1021/jm400485e
None Unchecked IC50 30.0 nM 10.1021/ml5001933
None Unchecked IC50 62.92 ug.mL-1 10.1016/j.ejmech.2020.112835
None Unchecked IC50 80.0 nM 10.1021/ml300350p
None Unchecked IC50 140.0 nM 10.1016/j.bmcl.2020.127146
None Unchecked IC50 6410.0 nM None
None Unchecked IC50 7420.0 nM None
None Unchecked IC50 8940.0 nM None
None Unchecked IC50 9700.0 nM None
None Unchecked IC50 10350.0 nM None
None Unchecked IC50 25000.0 nM 10.1016/j.bmc.2016.09.012
None Unchecked IC50 25000.0 nM 10.1016/j.bmc.2017.11.031
None Unchecked IC50 25000.0 nM 10.1016/j.ejmech.2017.12.088
None Unchecked IC50 25000.0 nM 10.1021/acs.jmedchem.6b00485
None Unchecked IC50 25000.0 nM 10.1128/aac.01649-07
None Unchecked IC50 32559.0 nM None
None Unchecked IC50 52100.0 nM 10.1016/j.bmcl.2011.08.054
None Unchecked IC50 63000.0 nM 10.1021/acs.jmedchem.8b01293
None Unchecked IC50 109000.0 nM 10.1021/jm4004889
None Unchecked IC50 126000.0 nM 10.1021/jm201716n
None Unchecked IC50 313000.0 nM 10.1021/jm201716n
None Unchecked IC50 465000.0 nM 10.1021/jm4004889
None Unchecked IC50 500000.0 nM 10.1016/j.ejmech.2021.113568
None Unchecked IC50 610000.0 nM 10.1021/jm4004889
None Unchecked IC50 830000.0 nM 10.1021/jm201716n
None Unchecked IC50 nan None 10.1016/j.bmc.2015.02.032
None Unchecked IC50 nan None 10.1016/j.ejmech.2014.12.046
None Unchecked IC50 nan None 10.1016/j.ejmech.2016.06.042
None Unchecked IC50 nan None 10.1021/ml5001728
None Unchecked IC50 nan None None
None Unchecked Inhibition 5.0 % 10.1021/jm400485e
None Unchecked Inhibition 7.8 % 10.1128/aac.00753-10
None Unchecked Inhibition 8.3 % 10.1128/aac.00753-10
None Unchecked Inhibition 69.6 % 10.1016/j.bmc.2014.12.060
None Unchecked Inhibition 95.0 % 10.1016/j.bmcl.2009.12.045
None Unchecked Inhibition nan % 10.1016/j.ejmech.2020.112671
None Unchecked Kd 195000.0 nM 10.1021/jm991174y
None Unchecked Ki nan None None
None Unchecked logIC50 1.717 None 10.1016/j.bmcl.2011.08.054
None Unchecked MIC 0.004 ug.mL-1 10.1021/acs.jmedchem.1c02045
None Unchecked MIC 0.1 ug.mL-1 10.1021/acs.jnatprod.1c00812
None Unchecked MIC 9.24 ug.mL-1 10.1021/acs.jmedchem.1c00263
None Unchecked MIC 10.0 ug.mL-1 10.1021/acs.jmedchem.1c00263
None Unchecked MIC 16.0 ug.mL-1 10.1021/acs.jmedchem.1c02045
None Unchecked MIC 50.0 nM 10.1016/j.ejmech.2020.112179
None Unchecked MIC 64.0 ug.mL-1 10.1016/j.bmcl.2019.07.001
None Unchecked MIC 190.0 nM 10.1021/acs.jmedchem.1c02122
None Unchecked MIC 256.0 ug.mL-1 10.1016/j.ejmech.2019.05.090
None Unchecked MIC 4000.0 nM 10.1021/acs.jmedchem.1c02122
None Unchecked MIC 12200.0 nM 10.1016/j.ejmech.2020.112179
None Unchecked MIC 48600.0 nM 10.1016/j.ejmech.2020.112179
None Unchecked MIC100 0.01 ug ml-1 10.1016/j.ejmech.2020.112420
None Unchecked MIC=>90 0.015 ug ml-1 10.1016/j.ejmech.2020.112538
None Unchecked MIC=>90 9.317 ug ml-1 10.1016/j.ejmech.2020.112538
None Unchecked MIC=>90 10.0 ug ml-1 10.1016/j.ejmech.2020.112538
None Unchecked PI 256.0 None 10.1016/j.ejmech.2009.06.005
None Unchecked PI 828.12 None 10.1016/j.bmc.2010.09.006
None Unchecked Potency 1778.3 nM None
None Unchecked Potency 10322.5 nM None
None Unchecked Potency 15848.9 nM None
None Unchecked Potency 18356.4 nM None
None Unchecked Potency 25929.0 nM None
None Unchecked Ratio 0.054 None 10.1093/toxsci/kft176
None Unchecked Ratio 0.07 None 10.1093/toxsci/kft176
None Unchecked Ratio 0.089 None 10.1093/toxsci/kft176
None Unchecked Ratio 0.147 None 10.1093/toxsci/kft176
None Unchecked Ratio 0.27 None 10.1128/aac.00120-07
None Unchecked Ratio 0.75 None 10.1016/j.bmcl.2022.128692
None Unchecked Ratio 0.83 None 10.1016/j.bmcl.2022.128692
None Unchecked Ratio 0.93 None 10.1016/j.bmcl.2022.128692
None Unchecked Ratio 1.09 None 10.1016/j.bmcl.2022.128692
None Unchecked Ratio 2.0 None 10.1021/acs.jmedchem.9b00288
None Unchecked Ratio 3.94 None 10.1128/aac.00367-09
None Unchecked Ratio 4.16 None 10.1128/aac.00367-09
None Unchecked Ratio 6.19 None 10.1128/aac.00367-09
None Unchecked Ratio 10.07 None 10.1128/aac.00367-09
None Unchecked Ratio 61.2 None 10.1128/aac.00120-07
None Unchecked Ratio 64.1 None 10.1128/aac.01533-06
None Unchecked Ratio 100.0 None 10.1016/j.bmcl.2013.07.006
None Unchecked Ratio 100.0 None 10.1128/aac.00775-08
None Unchecked Ratio 224.36 None 10.1128/aac.01533-06
None Unchecked Ratio 256.0 None 10.1021/jm701560p
None Unchecked Ratio 440.0 None 10.1128/aac.00458-08
None Unchecked Ratio 448.72 None 10.1128/aac.01533-06
None Unchecked Ratio 460.0 None 10.1128/aac.00775-08
None Unchecked Ratio 465.0 None 10.1128/aac.01533-06
None Unchecked Ratio 800.0 None 10.1016/j.bmc.2008.10.086
None Unchecked Ratio 16250.0 None 10.1016/j.bmcl.2009.09.095
None Unchecked Ratio 16256.0 None 10.1016/j.bmcl.2009.09.095
None Unchecked Ratio 20260.0 None 10.1128/aac.00458-08
None Unchecked Ratio 44510.0 None 10.1016/j.bmcl.2009.09.095
None Unchecked RatioAUC/MIC 24.14 None 10.1128/aac.01533-06
None Unchecked RatioAUC/MIC 169.0 None 10.1128/aac.01533-06
None Unchecked RatioAUC/MIC 224.36 None 10.1128/aac.01533-06
None Unchecked RatioAUC/MIC 448.72 None 10.1128/aac.01533-06
None Unchecked Ratio IC50 1.0 None 10.1021/jm400485e
None Unchecked Ratio IC50 61.0 None 10.1021/jm900340a
None Unchecked Ratio IC50 1080.0 None 10.1016/j.bmc.2010.03.018
None Unchecked Ratio IC50 1220.0 None 10.1021/jm900340a
None Unchecked Ratio IC50 2033.0 None 10.1021/jm901235p
None Unchecked Selectivity index 8000.0 SI 10.1016/s0960-894x(01)00266-9
None Unchecked Selectivity Index 8.0 None 10.1016/j.ejmech.2019.111678
None Unchecked Selectivity Index 10.0 None 10.1007/s00044-012-0074-2
None Unchecked Selectivity Index 61.0 None 10.1016/j.bmcl.2009.11.105
None Unchecked Selectivity Index 112.35 None 10.1016/j.bmcl.2016.03.045
None Unchecked Selectivity Index 123.0 None 10.1016/j.bmcl.2016.11.056
None Unchecked Selectivity Index 123.0 None 10.1016/j.bmcl.2017.01.004
None Unchecked Selectivity Index 123.0 None 10.1016/j.ejmech.2017.03.065
None Unchecked Selectivity Index 133.0 None 10.1016/j.bmcl.2016.11.056
None Unchecked Selectivity Index 133.0 None 10.1016/j.bmcl.2017.01.004
None Unchecked Selectivity Index 133.0 None 10.1016/j.ejmech.2017.01.009
None Unchecked Selectivity Index 133.0 None 10.1016/j.ejmech.2017.03.065
None Unchecked Selectivity Index 138.88 None 10.1016/j.bmcl.2016.03.045
None Unchecked Selectivity Index 196.0 None 10.1016/j.bmcl.2016.11.056
None Unchecked Selectivity Index 196.0 None 10.1016/j.ejmech.2017.01.009
None Unchecked Selectivity Index 196.0 None 10.1039/C5MD00404G
None Unchecked Selectivity Index 208.0 None 10.1016/j.ejmech.2017.01.009
None Unchecked Selectivity Index 222.0 None 10.1016/j.bmcl.2016.11.056
None Unchecked Selectivity Index 222.0 None 10.1039/C5MD00404G
None Unchecked Selectivity Index 244.0 None 10.1016/j.ejmech.2017.01.009
None Unchecked Selectivity Index 400.0 None 10.1016/j.ejmech.2009.10.050
None Unchecked Selectivity Index 512.0 None 10.1016/j.bmcl.2019.07.041
None Unchecked Selectivity Index 512.0 None 10.1016/j.ejmech.2019.07.057
None Unchecked Selectivity Index 526.31 None 10.1021/jm401735w
None Unchecked Selectivity Index 714.0 None 10.1016/j.bmcl.2016.05.093
None Unchecked Selectivity Index 800.0 None 10.1016/j.bmc.2008.08.050
None Unchecked Selectivity Index 800.0 None 10.1016/j.ejmech.2010.06.036
None Unchecked Selectivity Index 909.0 None 10.1016/j.bmcl.2012.06.095
None Unchecked Selectivity Index 947.0 None 10.1016/j.ejmech.2010.11.023
None Unchecked Selectivity Index 1000.0 None 10.1016/j.bmc.2018.07.034
None Unchecked Selectivity Index 1024.0 None 10.1016/j.bmc.2019.04.017
None Unchecked Selectivity Index 1024.0 None 10.1016/j.ejmech.2018.09.049
None Unchecked Selectivity Index 1100.0 None 10.1016/j.bmcl.2015.12.080
None Unchecked Selectivity Index 1167.0 None 10.1007/s00044-007-9073-0
None Unchecked Selectivity Index 1220.0 None 10.1016/j.bmcl.2009.11.105
None Unchecked Selectivity Index 1250.0 None 10.1016/j.bmcl.2016.05.093
None Unchecked Selectivity Index 1250.0 None 10.1021/np400497f
None Unchecked Selectivity Index 1312.0 None 10.1016/j.ejmech.2017.11.090
None Unchecked Selectivity Index 1363.4 None 10.1016/j.ejmech.2015.10.024
None Unchecked Selectivity Index 1488.0 None 10.1016/j.bmcl.2008.09.029
None Unchecked Selectivity Index 1543.0 None 10.1016/j.bmcl.2013.09.013
None Unchecked Selectivity Index 1754.4 None 10.1039/C6MD00278A
None Unchecked Selectivity Index 2000.0 None 10.1016/j.ejmech.2017.05.026
None Unchecked Selectivity Index 2050.0 None 10.1021/acs.jmedchem.7b00582
None Unchecked Selectivity Index 2325.5 None 10.1016/j.bmcl.2015.11.071
None Unchecked Selectivity Index 2439.0 None 10.1016/j.bmcl.2015.11.071
None Unchecked Selectivity Index 2500.0 None 10.1016/j.bmc.2016.12.038
None Unchecked Selectivity Index 2500.0 None 10.1016/j.ejmech.2016.09.059
None Unchecked Selectivity Index 2702.7 None 10.1016/j.bmcl.2016.02.043
None Unchecked Selectivity Index 2857.1 None 10.1016/j.bmcl.2016.02.043
None Unchecked Selectivity Index 2857.14 None 10.1016/j.bmcl.2016.02.043
None Unchecked Selectivity Index 4066.0 None 10.1021/acs.jnatprod.9b01095
None Unchecked Selectivity Index 5000.0 None 10.1039/C6MD00278A
None Unchecked Selectivity Index 6564.0 None 10.1016/j.ejmech.2019.01.042
None Unchecked Selectivity Index 12500.0 None 10.1021/acsmedchemlett.8b00410
None Unchecked Selectivity Index 14000.0 None 10.1016/j.bmc.2015.04.001
None Unchecked Selectivity Index 14000.0 None 10.1039/C3MD00251A
None Unchecked Selectivity Index 15000.0 None 10.1021/jm300123s
None Unchecked Selectivity Index 34400.0 None 10.1016/j.ejmech.2020.112045
None Unchecked Selectivity Index nan None 10.1016/j.bmc.2019.07.045
None Unchecked Selectivity Index nan None 10.1016/j.bmcl.2019.02.019
None Unchecked Selectivity Index nan None 10.1016/j.ejmech.2016.07.039
None Unchecked Selectivity Index nan None 10.1021/acs.jmedchem.7b01332
None Unchecked Selectivity ratio 1.1 None 10.1021/acs.jmedchem.2c00266
None Unchecked Selectivity ratio 1.3 None 10.1021/acs.jmedchem.2c00266
None Unchecked Selectivity ratio 98.0 None 10.1016/j.bmc.2008.12.006
None Unchecked Selectivity ratio 500.0 None 10.1039/C7MD00350A
None Unchecked Selectivity ratio 500.0 None 10.1039/C7MD00366H
None Unchecked Selectivity ratio 800.0 None 10.1016/j.bmc.2010.02.024
None Unchecked Time nan None 10.1128/aac.00620-10
None Unchecked TIME 0.005556 hr 10.1128/aac.00620-10

Metabolism Information

AKRT ID Reaction Reaction Link ID
AKRT004061 CC(=O)O.CO[C@H]1/C=C/O[C@@]2(C)Oc3c(C)c(O)c4c(c3C2=O)C(=O)/C(=C/NN2CCN(C)CC2)C(=C4O)N=C(O)/C(C)=C/C=C/[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](O)[C@H]1C>>CO[C@H]1/C=C/O[C@@]2(C)Oc3c(C)c(O)c4c(O)c(c(/C=N/N5CCN(C)CC5)c(O)c4c3C2=O)NC(=O)/C(C)=C\C=C\[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C MNXR132055
AKRT011282 CO[C@H]1/C=C/O[C@@]2(C)Oc3c(C)c(O)c4c(O)c(c(/C=N/N5CCN(C)CC5)c(O)c4c3C2=O)NC(=O)/C(C)=C\C=C\[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C>>CO[C@@H](/C=C/O[C@@]1(C)Oc2c(C)c(O)c3c(c2C1=O)C(=O)C(/C=N/N1CCN(C)CC1)=C(O)C3=O)[C@@H](C)[C@@H](OC(C)=O)[C@H](C)[C@H](O)[C@H](C)[C@@H](O)[C@@H](C)/C=C/C=C(/C)C(N)=O 58696
AKRT011283 CO[C@H]1/C=C/O[C@@]2(C)Oc3c(C)c(O)c4c(O)c(c(/C=N/N5CCN(C)CC5)c(O)c4c3C2=O)NC(=O)/C(C)=C\C=C\[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C>>CO[C@H]1/C=C/O[C@@]2(C)Oc3c(C)c(O)c4c(O)c(c(/C=N/N5CCN(C)CC5)c(O)c4c3C2=O)NC(=O)/C(C)=C\C=C\[C@H](C)[C@H](OP(=O)(O)O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C RXN-18733
AKRT011284 CO[C@H]1/C=C/O[C@@]2(C)Oc3c(C)c(O)c4c(O)c(c(/C=N/N5CCN(C)CC5)c(O)c4c3C2=O)NC(=O)/C(C)=C\C=C\[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C>>CO[C@H]1/C=C/O[C@@]2(C)Oc3c(C)c(O)c4c(c3C2=O)C(=O)/C(=C/N(O)N2CCN(C)CC2)C(=C4O)NC(=O)/C(C)=C\C=C\[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C RXN-17329
AKRT011285 CO[C@H]1/C=C/O[C@@]2(C)Oc3c(C)c(O)c4c(O)c(c(/C=N/N5CCN(C)CC5)c(O)c4c3C2=O)NC(=O)/C(C)=C\C=C\[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C>>CO[C@H]1/C=C/O[C@@]2(C)Oc3c(C)c(O)c4c(c3C2=O)C(O)=C(/C=N/N2CCN(C)CC2)C(O)(NC(=O)/C(C)=C\C=C\[C@H](C)[C@H](O)[C@@H](C)[C@@H](O)[C@@H](C)[C@H](OC(C)=O)[C@@H]1C)C4=O 58700