| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
512.0 |
ug.mL-1 |
10.1016/j.bmc.2022.117095 |
| Aspergillus niger |
Aspergillus niger |
IZ |
0.0 |
mm |
10.1016/j.ejmech.2011.10.022 |
| Bacillus |
Bacillus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Bacillus |
Bacillus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Bacillus |
Bacillus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Bacillus anthracis |
Bacillus anthracis |
Inhibition |
nan |
% |
10.1128/aac.01594-07 |
| Bacillus cereus |
Bacillus cereus |
IZ |
9.0 |
mm |
10.1007/s00044-007-9024-9 |
| Bacillus cereus |
Bacillus cereus |
IZ |
9.0 |
mm |
10.1016/j.bmc.2007.05.037 |
| Bacillus cereus |
Bacillus cereus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Bacillus licheniformis |
Bacillus licheniformis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Bacillus subtilis |
Bacillus subtilis |
Inhibition |
nan |
% |
10.1016/j.ejmech.2017.08.039 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.078 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00174 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jnatprod.8b00979 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
319200.0 |
nM |
10.1016/j.ejmech.2019.01.038 |
| Bos taurus |
Monoamine oxidase A |
Activity |
nan |
None |
10.1021/jm800656v |
| Brachyspira pilosicoli |
Class D beta-lactamase |
Kcat |
113.0 |
/s |
10.1128/aac.00684-07 |
| Brachyspira pilosicoli |
Class D beta-lactamase |
Kcat/Km |
9.8 |
10'5/M/s |
10.1128/aac.00684-07 |
| Brachyspira pilosicoli |
Class D beta-lactamase |
Km |
115000.0 |
nM |
10.1128/aac.00684-07 |
| Candida albicans |
Candida albicans |
IZ |
0.0 |
mm |
10.1021/np900382x |
| Candida albicans |
Candida albicans |
MIC |
nan |
None |
10.1016/j.ejmech.2013.04.023 |
| Carnobacterium divergens |
Carnobacterium divergens |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01145-07 |
| Carnobacterium divergens |
Carnobacterium divergens |
MIC |
24.0 |
ug.mL-1 |
10.1128/aac.01145-07 |
| Carnobacterium divergens |
Carnobacterium divergens |
MIC |
nan |
None |
10.1128/aac.01145-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
48.0 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
96.0 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterococcus |
Enterococcus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus |
Enterococcus |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus |
Enterococcus |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus avium |
Enterococcus avium |
MIC |
nan |
None |
10.1021/acs.jnatprod.9b01024 |
| Enterococcus avium |
Enterococcus avium |
MIC |
nan |
None |
10.1128/aac.00908-07 |
| Enterococcus casseliflavus |
Enterococcus casseliflavus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Enterococcus casseliflavus |
Enterococcus casseliflavus |
MIC |
nan |
None |
10.1021/acs.jnatprod.9b01024 |
| Enterococcus durans |
Enterococcus durans |
MIC |
nan |
None |
10.1021/acs.jnatprod.9b01024 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
nan |
None |
10.1021/jm9803572 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
50.0 |
ug ml-1 |
10.1021/np010599w |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
nan |
None |
10.1021/np010599w |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/np4006794 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116142 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.08.123 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.09.097 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.048 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.12.027 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1016/s0960-894x(01)00024-5 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00326-6 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm9803572 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
25.0 |
ug.mL-1 |
10.1021/np010599w |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.08.123 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.09.097 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.048 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.12.027 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
64.0 |
ug.mL-1 |
10.1016/s0960-894x(01)00024-5 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
64.0 |
ug.mL-1 |
10.1039/D1MD00230A |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
100.0 |
ug.mL-1 |
10.1021/np010599w |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
256.0 |
ug.mL-1 |
10.1021/np4006794 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
319200.0 |
nM |
10.1016/j.ejmech.2019.01.038 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1016/j.bmcl.2010.02.037 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1016/j.ejmech.2013.04.023 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1021/acs.jnatprod.9b01024 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1021/np4006794 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1128/aac.00908-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC=>90 |
8.0 |
ug ml-1 |
10.1016/j.bmcl.2013.02.016 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC=>90 |
64.0 |
ug ml-1 |
10.1016/j.bmcl.2013.02.016 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
8.0 |
ug.mL-1 |
10.1016/j.bmc.2012.10.009 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2012.10.009 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus faecium |
Enterococcus faecium |
IZ |
0.0 |
mm |
10.1021/np900382x |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
nan |
None |
10.1021/np010599w |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113402 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jnatprod.6b00229 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jnatprod.8b00979 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
64.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00326-6 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm9803572 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
64.0 |
ug.mL-1 |
10.1039/D1MD00230A |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
100.0 |
ug.mL-1 |
10.1021/np010599w |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
256.0 |
ug.mL-1 |
10.1021/np4006794 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
nan |
None |
10.1016/j.bmcl.2010.02.037 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
nan |
None |
10.1021/acs.jnatprod.9b01024 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
MIC |
nan |
None |
10.1021/acs.jnatprod.9b01024 |
| Escherichia coli |
Beta-lactamase OXA-7 |
Km |
52000.0 |
nM |
10.1128/aac.01714-09 |
| Escherichia coli |
Beta-lactamase OXA-7 |
Vmax |
9.3 |
nmol/sec |
10.1128/aac.01714-09 |
| Escherichia coli |
Beta-lactamase SCO-1 |
Activity |
4.0 |
None |
10.1128/aac.01439-06 |
| Escherichia coli |
Beta-lactamase TEM |
Activity |
nan |
None |
10.1128/aac.01439-06 |
| Escherichia coli |
Escherichia coli |
Activity |
12.0 |
uM |
10.1128/aac.01714-09 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1128/aac.01677-09 |
| Escherichia coli |
Escherichia coli |
IZ |
0.0 |
mm |
10.1016/j.ejmech.2011.10.022 |
| Escherichia coli |
Escherichia coli |
IZ |
0.0 |
mm |
10.1021/np900382x |
| Escherichia coli |
Escherichia coli |
IZ |
8.0 |
mm |
10.1021/np900382x |
| Escherichia coli |
Escherichia coli |
MBC |
nan |
None |
10.1016/j.ejmech.2013.04.023 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00921-08 |
| Escherichia coli |
Escherichia coli |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01677-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01677-09 |
| Escherichia coli |
Escherichia coli |
MIC |
1.024 |
ug.mL-1 |
10.1128/aac.01472-06 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00011-07 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01677-09 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00242-07 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01677-09 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01677-09 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1007/s00044-012-0417-z |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.09.107 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.082 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2010.09.031 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.05.012 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.12.011 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.05.023 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.08.026 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.10.012 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00011-07 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Escherichia coli |
Escherichia coli |
MIC |
190.0 |
ug.mL-1 |
10.1021/acs.jmedchem.7b00204 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1021/np4006794 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00921-08 |
| Escherichia coli |
Escherichia coli |
MIC |
282.0 |
ug.mL-1 |
10.1128/aac.01714-09 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00921-08 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01472-06 |
| Escherichia coli |
Escherichia coli |
MIC |
650.0 |
ug.mL-1 |
10.1021/np500775e |
| Escherichia coli |
Escherichia coli |
MIC |
1024.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.03.008 |
| Escherichia coli |
Escherichia coli |
MIC |
1300.0 |
ug.mL-1 |
10.1021/np500775e |
| Escherichia coli |
Escherichia coli |
MIC |
8000.0 |
ug.mL-1 |
10.1128/aac.00011-07 |
| Escherichia coli |
Escherichia coli |
MIC |
319200.0 |
nM |
10.1016/j.ejmech.2019.01.038 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.ejmech.2013.04.023 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.ejmech.2019.01.038 |
| Escherichia coli |
Escherichia coli |
MIC=>80 |
0.25 |
ug ml-1 |
10.1021/acs.jmedchem.1c01551 |
| Escherichia coli |
Escherichia coli |
permeability |
0.6 |
um/s |
10.1128/aac.01714-09 |
| Escherichia coli |
Escherichia coli |
Ratio |
4.0 |
None |
10.1128/aac.00921-08 |
| Escherichia coli |
Escherichia coli |
Ratio |
256.0 |
None |
10.1016/j.ejmech.2012.03.008 |
| Escherichia coli |
Escherichia coli |
Ratio |
512.0 |
None |
10.1016/j.ejmech.2012.03.008 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.008 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.015 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Homo sapiens |
Acetylcholinesterase |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Androgen Receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bile salt export pump |
AC50 |
219998.6 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Gamma-aminobutyric acid receptor subunit alpha-1/alpha-2/beta-2/gamma-2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
HERG |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Homo sapiens |
CL |
6.3 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
CL_renal |
2.6 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
DILI_Concern |
nan |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
DILI_severity_class |
3.0 |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Monoamine oxidase A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Mu opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Norepinephrine transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Oligopeptide transporter small intestine isoform |
Ki |
12000000.0 |
nM |
10.1016/j.ejpb.2004.07.008 |
| Homo sapiens |
Oligopeptide transporter small intestine isoform |
Ki |
12000000.0 |
nM |
10.1021/jm048982w |
| Homo sapiens |
Phosphodiesterase 3A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 4A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Plasma |
Cmax |
159426.07 |
nM |
10.1128/aac.01145-08 |
| Homo sapiens |
Plasma |
Fu |
0.07 |
None |
10.1128/aac.01145-08 |
| Homo sapiens |
Progesterone receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 1a (5-HT1a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Solute carrier family 15 member 2 |
Ki |
3300000.0 |
nM |
10.1016/j.bmc.2011.06.027 |
| Homo sapiens |
Solute carrier family 15 member 2 |
Ki |
3311311.21 |
nM |
10.1016/j.bmc.2011.06.027 |
| Homo sapiens |
Solute carrier family 22 member 8 |
Inhibition |
nan |
% |
10.1124/dmd.112.049569 |
| Homo sapiens |
THP-1 |
Ratio |
0.2 |
None |
10.1128/aac.00123-08 |
| Homo sapiens |
Thrombin |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Thromboxane A2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vascular endothelial growth factor receptor 2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
256.0 |
ug.mL-1 |
10.1021/np4006794 |
| Kocuria rhizophila |
Kocuria rhizophila |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Lactococcus lactis |
Lactococcus lactis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Lactococcus lactis |
Lactococcus lactis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Lactococcus lactis |
Lactococcus lactis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Listeria monocytogenes |
Listeria monocytogenes |
IZ |
9.6 |
mm |
10.1128/aac.00503-10 |
| Listeria monocytogenes |
Listeria monocytogenes |
IZ |
10.7 |
mm |
10.1128/aac.00290-10 |
| Listeria monocytogenes |
Listeria monocytogenes |
IZ |
11.9 |
mm |
10.1128/aac.00503-10 |
| Listeria monocytogenes |
Listeria monocytogenes |
IZ |
12.3 |
mm |
10.1128/aac.00290-10 |
| Mammaliicoccus lentus |
Mammaliicoccus lentus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00356-10 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
Activity |
4.0 |
% |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
Activity |
74.0 |
% |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
Activity |
96.0 |
% |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MBC |
1.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MBC50 |
2.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MBC50 |
128.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MBC90 |
256.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Micrococcus |
Micrococcus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Micrococcus |
Micrococcus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Micrococcus |
Micrococcus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Micrococcus luteus |
Micrococcus luteus |
MIC |
nan |
None |
10.1021/np4006794 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
Activity |
nan |
None |
10.1128/aac.00418-09 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Morganella morganii |
Morganella morganii |
MIC |
40.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00174 |
| Morganella morganii |
Morganella morganii |
MIC |
160.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00174 |
| Morganella morganii |
Morganella morganii |
MIC |
256.0 |
ug.mL-1 |
10.1021/np4006794 |
| Mus musculus |
Solute carrier family 22 member 6 |
Inhibition |
nan |
% |
10.1124/dmd.112.049569 |
| Mus musculus |
Solute carrier family 22 member 8 |
Drug uptake |
nan |
None |
10.1124/dmd.112.049569 |
| Mus musculus |
Solute carrier family 22 member 8 |
IC50 |
35000.0 |
nM |
10.1124/dmd.112.049569 |
| Mus musculus |
Solute carrier family 22 member 8 |
Inhibition |
nan |
% |
10.1124/dmd.112.049569 |
| Mycobacterium |
Mycobacterium |
IZ |
0.0 |
mm |
10.1016/j.ejmech.2011.10.022 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
nan |
None |
10.1021/np800572r |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
nan |
None |
10.1021/np800572r |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.060 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
nan |
None |
10.1021/np800572r |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
nan |
None |
10.1016/j.ejmech.2013.04.023 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
nan |
None |
10.1016/j.ejmech.2013.04.023 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
256.0 |
ug.mL-1 |
10.1021/np4006794 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
319200.0 |
nM |
10.1016/j.ejmech.2019.01.038 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
512000.0 |
nM |
10.1016/j.ejmech.2019.111623 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1016/j.ejmech.2013.04.023 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1016/j.ejmech.2019.01.038 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1021/acs.jnatprod.7b00496 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC=>80 |
1.98 |
ug ml-1 |
10.1021/acs.jmedchem.1c01551 |
| Pseudomonas fluorescens |
Beta-lactamase |
Kcat/Km |
100.0 |
/mM/s |
10.1128/aac.00961-09 |
| Rattus norvegicus |
Oligopeptide transporter, kidney isoform |
Ki |
3300000.0 |
nM |
10.1016/j.ejpb.2004.07.008 |
| Rattus norvegicus |
Serum |
Drug uptake |
125.0 |
ug ml-1 |
10.1128/aac.00506-06 |
| Salmonella enterica |
Salmonella enterica |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00371-09 |
| Salmonella enterica |
Salmonella enterica |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00371-09 |
| Salmonella enterica |
Salmonella enterica |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00371-09 |
| Salmonella enterica |
Salmonella enterica |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00371-09 |
| Salmonella enterica |
Salmonella enterica |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00371-09 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01472-06 |
| Staphylococcus |
Staphylococcus |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus |
Staphylococcus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus |
Staphylococcus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus |
Staphylococcus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus |
Staphylococcus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus |
Staphylococcus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus |
Staphylococcus |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus |
Staphylococcus |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus |
Staphylococcus |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus |
Staphylococcus |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus |
Staphylococcus |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus |
Staphylococcus |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus |
Staphylococcus |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus |
Staphylococcus |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus |
Staphylococcus |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus |
Staphylococcus |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus |
Staphylococcus |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus |
Staphylococcus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus |
Staphylococcus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus |
Staphylococcus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus |
Staphylococcus |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus |
Staphylococcus |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus aureus |
Accessory gene regulator protein A |
Activity |
nan |
None |
10.1128/aac.00064-10 |
| Staphylococcus aureus |
Cell division protein ftsZ |
Activity |
nan |
None |
10.1016/j.bmcl.2012.08.123 |
| Staphylococcus aureus |
MecA |
Activity |
300.0 |
ug ml-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
MecA |
Activity |
nan |
None |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
MecA |
IC50 |
710000.0 |
nM |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
MecA |
Inhibition |
5.0 |
% |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.00952-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.01562-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
ug ml-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.5 |
ug ml-1 |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1.0 |
ug ml-1 |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
2.0 |
ug ml-1 |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
4.3 |
% |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
6.05 |
log10CFU/ml |
10.1016/j.ejmech.2016.03.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
6.2 |
% |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
7.62 |
log10CFU/ml |
10.1016/j.ejmech.2016.03.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
8.35 |
log10CFU/ml |
10.1016/j.ejmech.2016.03.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
8.8 |
% |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
9.1 |
% |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
9.7 |
% |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
10.4 |
% |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
11.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
11.2 |
log10CFU/ml |
10.1016/j.ejmech.2016.03.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
11.95 |
log10CFU/ml |
10.1016/j.ejmech.2016.03.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
12.34 |
log10CFU/ml |
10.1016/j.ejmech.2016.03.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
12.4 |
% |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
32.0 |
ug ml-1 |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
36.4 |
% |
10.1128/aac.00418-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
46.2 |
% |
10.1128/aac.00952-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
53.8 |
% |
10.1128/aac.00952-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
64.0 |
ug ml-1 |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
78.9 |
% |
10.1128/aac.00418-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
89.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00351-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00952-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.01562-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
ug ml-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
128.0 |
ug ml-1 |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
200.0 |
ug ml-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
400.0 |
ug ml-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
800.0 |
ug ml-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.bmc.2022.116648 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.bmcl.2006.08.062 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/acsmedchemlett.1c00648 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/acsmedchemlett.5b00142 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/jm0703183 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00064-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00722-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01201-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01472-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
CFU/ml |
3.0 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
CFU/ml |
4.0 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
2.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
2.49 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
2.71 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
2.89 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
2.99 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.14 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.2 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.34 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.34 |
None |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.36 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.4 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.48 |
None |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.5 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.64 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.67 |
None |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.68 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.83 |
None |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.93 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
3.99 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
4.0 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
4.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
4.26 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
4.32 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
4.36 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
4.48 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
4.79 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
4.99 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
5.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
6.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
6.12 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
6.82 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
6.83 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
7.4 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
8.0 |
None |
10.1016/j.ejmech.2019.111686 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
8.88 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
9.03 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
9.6 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
9.61 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
10.0 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
12.4 |
None |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
13.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
15.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
16.0 |
None |
10.1128/aac.00049-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
18.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
20.43 |
None |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
25.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
27.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
31.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
41.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
50.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
64.0 |
None |
10.1016/j.bmc.2023.117232 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
64.0 |
None |
10.1128/aac.00049-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
66.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
69.0 |
None |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
128.0 |
None |
10.1128/aac.00049-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
GI |
nan |
None |
10.1016/j.bmc.2015.04.069 |
| Staphylococcus aureus |
Staphylococcus aureus |
GI |
nan |
None |
10.1021/acsmedchemlett.5b00142 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
nan |
% |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
0.0 |
mm |
10.1021/np900382x |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
6.0 |
mm |
10.1016/j.bmcl.2016.05.030 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
15.0 |
mm |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
18.0 |
mm |
10.1021/np900382x |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
21.0 |
mm |
10.1016/j.ejmech.2011.10.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
22.0 |
mm |
10.1021/np900382x |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
28.86 |
mm |
10.1016/j.bmcl.2016.05.030 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
-0.39 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
0.83 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
3.0 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-3.91 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-3.0 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-2.7 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-2.52 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-2.05 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-1.75 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-1.72 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-1.54 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-1.51 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-1.47 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-1.35 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-1.32 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-1.28 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-1.27 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-1.02 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.94 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.91 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.85 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.48 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.05 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
0.21 |
None |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
5.5 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
1000.0 |
None |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.2 |
ug ml-1 |
10.1016/j.ejmech.2013.04.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.00506-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.39 |
ug ml-1 |
10.1021/np010599w |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.4 |
ug ml-1 |
10.1016/j.ejmech.2013.04.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.5 |
mg/L |
10.1128/aac.01376-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.8 |
ug ml-1 |
10.1016/j.ejmech.2013.04.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
1.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
1.25 |
uM |
10.1016/j.bmcl.2016.05.030 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
1.5 |
ug ml-1 |
10.1016/j.ejmech.2013.04.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
19.9 |
uM |
10.1016/j.bmcl.2016.05.030 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
150.0 |
ug ml-1 |
10.1016/j.ejmech.2013.04.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
256.0 |
ug ml-1 |
10.1128/aac.00049-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
256.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
nan |
None |
10.1021/np010599w |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
16.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
256.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
64.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
512.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.01173-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.01192-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.048 |
ug.mL-1 |
10.1128/aac.00437-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2012.08.123 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2012.09.097 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.048 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2012.12.027 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2021.113659 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01091-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01201-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01376-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.078 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00174 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmc.2021.116580 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.bmc.2021.116142 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01113-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01124-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01201-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01472-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmc.2010.02.005 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2009.06.092 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00684 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1021/np8002673 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00506-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.13 |
ug.mL-1 |
10.1021/acs.jnatprod.6b00229 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.13 |
ug.mL-1 |
10.1021/acs.jnatprod.8b00979 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.19 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2013.04.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.037 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2021.128192 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/s0960-894x(01)00024-5 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/s0960-894x(98)00326-6 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00684 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jnatprod.0c00444 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jnatprod.7b00452 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1021/acsmedchemlett.1c00680 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm9803572 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1021/np8002673 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1021/np800572r |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1039/D1MD00230A |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00534-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01164-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01376-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01480-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.256 |
ug.mL-1 |
10.1128/aac.00437-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.256 |
ug.mL-1 |
10.1128/aac.01173-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.39 |
ug.mL-1 |
10.1021/np010599w |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2013.04.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.4 |
ug.mL-1 |
10.1128/aac.01099-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.42 |
ug.mL-1 |
10.1016/j.bmc.2021.116580 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2009.06.092 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.137 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.111686 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2020.112276 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2021.113402 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/np4001703 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/np4006794 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/np500080m |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1039/D1MD00230A |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00464-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00534-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01164-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01480-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.78 |
ug.mL-1 |
10.1016/S0960-894X(01)80927-6 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.8 |
ug.mL-1 |
10.1016/j.ejmech.2013.04.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.8 |
ug.mL-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.8 |
ug.mL-1 |
10.1128/aac.01099-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1007/s00044-012-0417-z |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2015.08.031 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.09.107 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.082 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.10.028 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.001 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.02.033 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2010.09.031 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.05.012 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.12.011 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.05.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.08.026 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.10.012 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.12.007 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.03.059 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111686 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113402 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jnatprod.5b01038 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00049-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00273-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00533-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00534-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01192-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.04.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.00533-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.00834-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.56 |
ug.mL-1 |
10.1016/S0960-894X(01)80927-6 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jnatprod.7b00226 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00049-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00231-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00534-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.00533-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.12 |
ug.mL-1 |
10.1016/S0960-894X(01)80927-6 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/acsmedchemlett.1c00680 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm101604v |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00049-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00534-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01001-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
5.0 |
ug.mL-1 |
10.1128/aac.00834-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6.0 |
ug.mL-1 |
10.1128/aac.00834-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6.25 |
ug.mL-1 |
10.1016/S0960-894X(01)80927-6 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115776 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00684 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jnatprod.8b00979 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00142 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1021/np050438i |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00001-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00534-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01091-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01128-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01164-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01201-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
12.0 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
12.5 |
ug.mL-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116142 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.06.092 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.137 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.03.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.060 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00684 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00142 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00001-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00064-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00361-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00533-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00534-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00576-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00908-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01124-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01201-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01472-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
24.0 |
ug.mL-1 |
10.1128/aac.00417-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
25.0 |
ug.mL-1 |
10.1021/np0780147 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.03.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.037 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.03.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.113134 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jnatprod.6b00229 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jnatprod.7b00226 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/acsmedchemlett.1c00680 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/np8002673 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/np800572r |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00361-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00533-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01001-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01113-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01201-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01376-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
50.0 |
ug.mL-1 |
10.1016/S0960-894X(01)80927-6 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
50.0 |
ug.mL-1 |
10.1021/np0780147 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1007/s00044-012-0417-z |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.08.123 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.09.097 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.09.107 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.082 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.048 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.10.028 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.001 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.02.033 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2010.09.031 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.05.012 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.12.011 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.05.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.08.026 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.10.012 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.12.007 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.12.027 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.03.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.03.059 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112276 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/s0960-894x(01)00024-5 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00326-6 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00142 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm9803572 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1039/D1MD00230A |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00001-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00049-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00973-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01001-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
75.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.04.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
80.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00174 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
100.0 |
ug.mL-1 |
10.1016/S0960-894X(01)80927-6 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
100.0 |
ug.mL-1 |
10.1021/np010599w |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
100.0 |
ug.mL-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.06.092 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.03.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112276 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b01518 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jnatprod.5b01038 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jnatprod.7b00226 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00142 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1021/np8002673 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1021/np800572r |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00049-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01001-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01255-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01466-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
160.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00174 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
192.0 |
ug.mL-1 |
10.1128/aac.00417-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.03.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112233 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1021/acsmedchemlett.1c00680 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00142 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1021/np0304823 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1021/np4006794 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1039/D1MD00211B |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00001-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00040-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00049-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00209-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00417-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00504-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00533-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00653-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00834-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01024-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01255-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01466-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
310.0 |
nM |
10.1016/j.ejmech.2019.01.038 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
400.0 |
ug.mL-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
400.0 |
ug.mL-1 |
10.1128/aac.01099-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
470.0 |
nM |
10.1016/j.ejmech.2015.06.013 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.03.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.09.116 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112233 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1021/acsmedchemlett.1c00680 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00142 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1021/np0304823 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1039/D1MD00211B |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00001-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00209-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00534-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01466-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.01472-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
600.0 |
nM |
10.1021/acs.jnatprod.7b00496 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
620.0 |
nM |
10.1016/j.bmcl.2016.05.030 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
800.0 |
ug.mL-1 |
10.1128/aac.00266-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
800.0 |
ug.mL-1 |
10.1128/aac.01099-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2017.01.038 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1024.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00142 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1024.0 |
ug.mL-1 |
10.1128/aac.00209-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1025.0 |
ug.mL-1 |
10.1128/aac.00534-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1200.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111686 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2500.0 |
nM |
10.1016/j.ejmech.2021.113212 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
19900.0 |
nM |
10.1016/j.bmcl.2016.05.030 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
19950.0 |
nM |
10.1016/j.ejmech.2019.01.038 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
50000.0 |
nM |
10.1016/j.ejmech.2017.01.038 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64000.0 |
nM |
10.1016/j.ejmech.2020.113134 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
79000.0 |
nM |
10.1021/np2003319 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
80000.0 |
nM |
10.1016/j.ejmech.2017.01.038 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
80000.0 |
nM |
10.1016/j.ejmech.2021.113212 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
159600.0 |
nM |
10.1016/j.ejmech.2019.01.038 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
160000.0 |
nM |
10.1016/j.ejmech.2017.01.038 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
319000.0 |
nM |
10.1021/acs.jnatprod.7b00496 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
320000.0 |
nM |
10.1016/j.ejmech.2017.01.038 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512000.0 |
nM |
10.1016/j.ejmech.2019.111623 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
638000.0 |
nM |
10.1021/acs.jnatprod.7b00496 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
638000.0 |
nM |
10.1021/acs.jnatprod.9b01024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
640000.0 |
nM |
10.1016/j.ejmech.2017.01.038 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
710000.0 |
nM |
10.1016/j.ejmech.2015.06.013 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1275000.0 |
nM |
10.1021/acs.jnatprod.9b01024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1276000.0 |
nM |
10.1021/np2003319 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1021/np4006794 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1128/aac.01255-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC100 |
64.0 |
ug ml-1 |
10.1021/acs.jmedchem.2c01151 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
16.0 |
ug.mL-1 |
10.1021/jm101604v |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
32.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
32.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
128.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115776 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
128.0 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
nan |
None |
10.1128/aac.01017-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC=>80 |
0.06 |
ug ml-1 |
10.1021/acs.jmedchem.1c01551 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC=>90 |
0.063 |
ug ml-1 |
10.1016/j.bmcl.2013.02.016 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC=>90 |
64.0 |
ug ml-1 |
10.1016/j.bmcl.2013.02.016 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.06 |
ug.mL-1 |
10.1016/j.bmc.2012.10.009 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
16.0 |
ug.mL-1 |
10.1021/jm101604v |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2012.10.009 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
128.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115776 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
128.0 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
nan |
None |
10.1128/aac.01017-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
8.0 |
None |
10.1016/j.ejmech.2019.111686 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
1500.0 |
None |
10.1016/j.ejmech.2015.06.013 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC |
638000.0 |
nM |
10.1021/acs.jnatprod.9b01024 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus cohnii |
Staphylococcus cohnii |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus cohnii |
Staphylococcus cohnii |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus cohnii |
Staphylococcus cohnii |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
0.0 |
% |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
4.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
16.7 |
% |
10.1128/aac.00418-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
26.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
27.3 |
% |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
55.6 |
% |
10.1128/aac.00418-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
72.7 |
% |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
74.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
96.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
100.0 |
% |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
0.2 |
ug ml-1 |
10.1016/j.ejmech.2013.04.023 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
1.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC50 |
2.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC50 |
128.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC90 |
256.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.16 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00174 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2013.04.023 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2021.128192 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jnatprod.8b00979 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00231-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.098 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
256.0 |
ug.mL-1 |
10.1021/np4006794 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
638000.0 |
nM |
10.1021/acs.jnatprod.9b01024 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
nan |
None |
10.1021/np4006794 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
nan |
None |
10.1128/aac.00418-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
0.0 |
% |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
4.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
26.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
26.8 |
% |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
31.7 |
% |
10.1128/aac.00418-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
73.2 |
% |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
74.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
96.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
100.0 |
% |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC |
1.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC50 |
2.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC50 |
128.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC90 |
256.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
39900.0 |
nM |
10.1021/acs.jnatprod.9b01024 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
Activity |
4.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
Activity |
16.0 |
% |
10.1128/aac.00418-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
Activity |
26.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
Activity |
74.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
Activity |
96.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MBC |
1.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MBC50 |
2.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MBC50 |
128.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MBC90 |
256.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC |
39900.0 |
nM |
10.1021/acs.jnatprod.9b01024 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus intermedius |
Staphylococcus intermedius |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus intermedius |
Staphylococcus intermedius |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus intermedius |
Staphylococcus intermedius |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
Activity |
60.0 |
% |
10.1128/aac.00418-09 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC |
1250.0 |
nM |
10.1021/acs.jnatprod.9b01024 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
Activity |
9.9 |
% |
10.1128/aac.00418-09 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01150-07 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01150-07 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01150-07 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
2490.0 |
nM |
10.1021/acs.jnatprod.9b01024 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01150-07 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01150-07 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus simulans |
Staphylococcus simulans |
Activity |
74.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
Activity |
96.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MBC |
1.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MBC50 |
2.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MBC50 |
128.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MBC90 |
256.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC |
620.0 |
nM |
10.1021/acs.jnatprod.9b01024 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC50 |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus sp. |
Staphylococcus sp. |
Activity |
0.0 |
% |
10.1128/aac.01562-06 |
| Staphylococcus sp. |
Staphylococcus sp. |
Activity |
100.0 |
% |
10.1128/aac.01562-06 |
| Staphylococcus sp. |
Staphylococcus sp. |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus sp. |
Staphylococcus sp. |
MIC50 |
32.0 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus sp. |
Staphylococcus sp. |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus sp. |
Staphylococcus sp. |
MIC90 |
128.0 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus warneri |
Staphylococcus warneri |
Activity |
46.0 |
% |
10.1128/aac.00418-09 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC |
319000.0 |
nM |
10.1021/acs.jnatprod.9b01024 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00418-09 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00185-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00185-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00185-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00185-08 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC50 |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus mitis |
Streptococcus mitis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus mitis |
Streptococcus mitis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus mitis |
Streptococcus mitis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus mutans |
Streptococcus mutans |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2010.09.031 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.08 |
ug.mL-1 |
10.1128/aac.01107-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.16 |
ug.mL-1 |
10.1128/aac.01107-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.18 |
ug.mL-1 |
10.1128/aac.01107-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.2 |
ug.mL-1 |
10.1128/aac.01107-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.21 |
ug.mL-1 |
10.1128/aac.01107-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.23 |
ug.mL-1 |
10.1128/aac.01107-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.24 |
ug.mL-1 |
10.1128/aac.01107-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01107-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.85 |
ug.mL-1 |
10.1128/aac.01107-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.95 |
ug.mL-1 |
10.1128/aac.01107-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00185-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01107-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
319200.0 |
nM |
10.1016/j.ejmech.2019.01.038 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
nan |
None |
10.1128/aac.01107-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
319200.0 |
nM |
10.1016/j.ejmech.2019.01.038 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Yamadazyma tenuis |
Yamadazyma tenuis |
IZ |
0.0 |
mm |
10.1016/j.ejmech.2011.10.022 |
| None |
ADMET |
CL |
6.3 |
mL.min-1.kg-1 |
10.1124/dmd.108.020479 |
| None |
ADMET |
delta logD |
0.9 |
None |
10.1021/jm0000564 |
| None |
ADMET |
F |
49.0 |
% |
10.1021/jm0000564 |
| None |
ADMET |
MRT |
0.5 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
PPB |
90.0 |
% |
10.1016/j.ejmech.2020.112829 |
| None |
ADMET |
T1/2 |
0.7 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
Vdss |
0.19 |
L.kg-1 |
10.1124/dmd.108.020479 |
| None |
Hepatotoxicity |
HepSE_bilirubinemia |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholecystitis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholelithiasis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cirrhosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_Combined Scores |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_elevated liver function tests |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic failure |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic necrosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatitis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatomegaly |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_jaundice |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver disease |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver fatty |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver function tests abnormal |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Molecular identity unknown |
PPB |
91.0 |
% |
10.1021/jm501661f |
| None |
NON-PROTEIN TARGET |
Fu |
0.07 |
None |
10.1124/dmd.108.020479 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (acute) |
22.0 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (animal toxicity known) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (benign tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (granulomatous hepatitis) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (mechanism) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
12.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
81.0 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (time to onset) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00575-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00684-07 |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00242-07 |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00356-10 |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00575-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00356-10 |
| None |
NON-PROTEIN TARGET |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00356-10 |
| None |
NON-PROTEIN TARGET |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00356-10 |
| None |
NON-PROTEIN TARGET |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00356-10 |
| None |
NON-PROTEIN TARGET |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00575-09 |
| None |
NON-PROTEIN TARGET |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00356-10 |
| None |
NON-PROTEIN TARGET |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00575-09 |
| None |
NON-PROTEIN TARGET |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00049-08 |
| None |
NON-PROTEIN TARGET |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00356-10 |
| None |
NON-PROTEIN TARGET |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00575-09 |
| None |
NON-PROTEIN TARGET |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00049-08 |
| None |
NON-PROTEIN TARGET |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00684-07 |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| None |
No relevant target |
Activity |
91.8 |
% |
10.1128/aac.00123-08 |
| None |
No relevant target |
Activity |
94.2 |
% |
10.1128/aac.00123-08 |
| None |
No relevant target |
LogD |
-1.32 |
None |
10.1021/jm0000564 |
| None |
No relevant target |
LogP |
2.1 |
None |
10.1128/aac.01714-09 |
| None |
No relevant target |
pKa |
2.8 |
None |
10.1021/jm0000564 |
| None |
Unchecked |
Activity |
12.0 |
None |
10.1128/aac.01439-06 |
| None |
Unchecked |
Activity |
25.0 |
% |
10.1128/aac.00684-07 |
| None |
Unchecked |
Activity |
210.0 |
mU |
10.1128/aac.00978-07 |
| None |
Unchecked |
Activity |
220.0 |
mU |
10.1128/aac.00978-07 |
| None |
Unchecked |
Activity |
230.0 |
mU |
10.1128/aac.00978-07 |
| None |
Unchecked |
Activity |
nan |
None |
10.1021/acsmedchemlett.1c00680 |
| None |
Unchecked |
Activity |
nan |
None |
10.1128/aac.00978-07 |
| None |
Unchecked |
Hepatotoxicity (acute) |
17.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (association with vascular disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (choleostasis) |
4.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (chronic liver disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cirrhosis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (comment) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cytolytic) |
14.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (malignant tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (severe hepatitis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (steatosis) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (successful reintroduction) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
K0.5 |
0.97 |
uM |
10.1128/aac.01714-09 |
| None |
Unchecked |
Kcat |
0.01 |
/s |
10.1128/aac.01463-07 |
| None |
Unchecked |
Kcat |
1.2 |
/s |
10.1128/aac.00856-09 |
| None |
Unchecked |
Kcat |
15.0 |
/s |
10.1128/aac.00961-09 |
| None |
Unchecked |
Kcat |
62.0 |
/s |
10.1128/aac.01145-07 |
| None |
Unchecked |
Kcat |
577.0 |
/s |
10.1128/aac.00743-09 |
| None |
Unchecked |
Kcat |
780.0 |
/s |
10.1128/aac.00684-07 |
| None |
Unchecked |
Kcat/Km |
0.003 |
/s/microM |
10.1128/aac.00856-09 |
| None |
Unchecked |
Kcat/Km |
2.1 |
10'7/M/s |
10.1128/aac.00684-07 |
| None |
Unchecked |
Kcat/Km |
19.0 |
/uM/s |
10.1128/aac.00743-09 |
| None |
Unchecked |
Kcat/Km |
45.0 |
None |
10.1128/aac.01145-07 |
| None |
Unchecked |
Kcat/Km |
2952.0 |
/mM/s |
10.1128/aac.01145-07 |
| None |
Unchecked |
Km |
21000.0 |
nM |
10.1128/aac.01145-07 |
| None |
Unchecked |
Km |
31000.0 |
nM |
10.1128/aac.00743-09 |
| None |
Unchecked |
Km |
36000.0 |
nM |
10.1128/aac.00684-07 |
| None |
Unchecked |
Km |
110000.0 |
nM |
10.1128/aac.00961-09 |
| None |
Unchecked |
Km |
450000.0 |
nM |
10.1128/aac.00856-09 |
| None |
Unchecked |
Km |
nan |
None |
10.1128/aac.01463-07 |
| None |
Unchecked |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| None |
Unchecked |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.090 |
| None |
Unchecked |
MIC |
512.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112233 |
| None |
Unchecked |
Vmax |
0.94 |
nmol/sec |
10.1128/aac.01714-09 |