| Acinetobacter baumannii |
Acinetobacter baumannii |
IC50 |
4000.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
IC50 |
4900.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
IC50 |
9200.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
IC50 |
33400.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
32.0 |
ug.mL-1 |
10.1007/s00044-012-0394-2 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.10.048 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00015 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64.0 |
ug.mL-1 |
10.1039/d2md00260d |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.06.003 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111850 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
10000.0 |
nM |
10.6019/CHEMBL4513141 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
25000.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
64000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
200000.0 |
nM |
10.1016/j.ejmech.2022.114213 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
200000.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
nan |
None |
10.1016/j.ejmech.2018.06.023 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
nan |
None |
10.1021/jm201467r |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC100 |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC50 |
nan |
None |
10.1021/jm201467r |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC90 |
nan |
None |
10.1021/jm201467r |
| Actinomyces naeslundii |
Actinomyces naeslundii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Actinomyces naeslundii |
Actinomyces naeslundii |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Actinomyces naeslundii |
Actinomyces naeslundii |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Anaerococcus prevotii |
Anaerococcus prevotii |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Anaerococcus tetradius |
Anaerococcus tetradius |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Anaerococcus tetradius |
Anaerococcus tetradius |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Anaerococcus tetradius |
Anaerococcus tetradius |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bacillus |
Bacillus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Bacillus |
Bacillus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Bacillus |
Bacillus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Bacillus anthracis |
Bacillus anthracis |
Activity |
nan |
None |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
11249.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
22498.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
33746.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
36244.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
45553.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
56245.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
56258.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
56283.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
71300.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
71422.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
71540.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
74371.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
78508.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
90081.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
90106.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
91106.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
91216.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
91284.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fAUC |
115702.0 |
ng.hr.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
1.4 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
2.8 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
3.1 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
4.0 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
4.2 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
4.4 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
5.4 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
5.5 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
5.7 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
7.0 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
7.1 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
8.9 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
9.8 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fCmax |
11.3 |
mg/L |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
0.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
4.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
7.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
8.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
9.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
11.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
12.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
13.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
14.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
15.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
18.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
22.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
23.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
fT>MIC |
24.0 |
hr |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.01439-07 |
| Bacillus anthracis |
Bacillus anthracis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01439-07 |
| Bacillus cereus |
Bacillus cereus |
Inhibition |
1.7 |
% |
10.1128/aac.01496-06 |
| Bacillus cereus |
Bacillus cereus |
Inhibition |
3.3 |
% |
10.1128/aac.01496-06 |
| Bacillus cereus |
Bacillus cereus |
Inhibition |
30.0 |
% |
10.1128/aac.01496-06 |
| Bacillus cereus |
Bacillus cereus |
Inhibition |
98.3 |
% |
10.1128/aac.01496-06 |
| Bacillus cereus |
Bacillus cereus |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Bacillus cereus |
Bacillus cereus |
IZ |
10.0 |
mm |
10.1016/j.ejmech.2011.04.041 |
| Bacillus cereus |
Bacillus cereus |
MIC |
0.5 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00379 |
| Bacillus cereus |
Bacillus cereus |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.bmcl.2009.07.106 |
| Bacillus cereus |
Bacillus cereus |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.ejmech.2009.11.009 |
| Bacillus cereus |
Bacillus cereus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00372 |
| Bacillus cereus |
Bacillus cereus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jnatprod.0c00279 |
| Bacillus cereus |
Bacillus cereus |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm501661f |
| Bacillus cereus |
Bacillus cereus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.024 |
| Bacillus cereus |
Bacillus cereus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.05.003 |
| Bacillus cereus |
Bacillus cereus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.096 |
| Bacillus cereus |
Bacillus cereus |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.04.041 |
| Bacillus cereus |
Bacillus cereus |
MIC |
2314.5 |
nM |
10.1016/j.bmcl.2009.04.133 |
| Bacillus cereus |
Bacillus cereus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Bacillus cereus |
Bacillus cereus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Bacillus licheniformis |
Bacillus licheniformis |
MIC |
0.5 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00379 |
| Bacillus licheniformis |
Bacillus licheniformis |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00372 |
| Bacillus licheniformis |
Bacillus licheniformis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm501661f |
| Bacillus pumilus |
Bacillus pumilus |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2021.113723 |
| Bacillus pumilus |
Bacillus pumilus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2007.05.003 |
| Bacillus pumilus |
Bacillus pumilus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115729 |
| Bacillus pumilus |
Bacillus pumilus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.024 |
| Bacillus pumilus |
Bacillus pumilus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.053 |
| Bacillus pumilus |
Bacillus pumilus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2019.06.010 |
| Bacillus pumilus |
Bacillus pumilus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.12.025 |
| Bacillus pumilus |
Bacillus pumilus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113480 |
| Bacillus pumilus |
Bacillus pumilus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113723 |
| Bacillus pumilus |
Bacillus pumilus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.03.028 |
| Bacillus pumilus |
Bacillus pumilus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.017 |
| Bacillus pumilus |
Bacillus pumilus |
MIC |
nan |
None |
10.1016/j.ejmech.2021.113480 |
| Bacillus pumilus |
Bacillus pumilus |
Ratio |
8.0 |
None |
10.1016/j.ejmech.2021.113723 |
| Bacillus pumilus |
Bacillus pumilus |
Ratio |
nan |
None |
10.1016/j.ejmech.2021.113480 |
| Bacillus sp. |
Bacillus sp. |
Inhibition |
0.7 |
% |
10.1128/aac.01496-06 |
| Bacillus sp. |
Bacillus sp. |
Inhibition |
4.9 |
% |
10.1128/aac.01496-06 |
| Bacillus sp. |
Bacillus sp. |
Inhibition |
31.7 |
% |
10.1128/aac.01496-06 |
| Bacillus sp. |
Bacillus sp. |
Inhibition |
97.2 |
% |
10.1128/aac.01496-06 |
| Bacillus sp. |
Bacillus sp. |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Bacillus sp. |
Bacillus sp. |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Bacillus sp. |
Bacillus sp. |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Bacillus subtilis |
Bacillus subtilis |
IC50 |
0.64 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Bacillus subtilis |
Bacillus subtilis |
Inhibition |
98.87 |
% |
10.1016/j.ejmech.2016.07.001 |
| Bacillus subtilis |
Bacillus subtilis |
Inhibition |
99.37 |
% |
10.1016/j.ejmech.2016.07.001 |
| Bacillus subtilis |
Bacillus subtilis |
Inhibition |
99.82 |
% |
10.1016/j.ejmech.2016.07.001 |
| Bacillus subtilis |
Bacillus subtilis |
IZ |
10.0 |
mm |
10.1016/j.ejmech.2013.01.034 |
| Bacillus subtilis |
Bacillus subtilis |
IZ |
20.0 |
mm |
10.1016/j.ejmech.2013.03.027 |
| Bacillus subtilis |
Bacillus subtilis |
IZ |
31.0 |
mm |
10.1016/j.bmcl.2009.10.018 |
| Bacillus subtilis |
Bacillus subtilis |
IZ |
33.0 |
mm |
10.1039/c0md00015a |
| Bacillus subtilis |
Bacillus subtilis |
IZ |
37.0 |
mm |
10.1039/c0md00015a |
| Bacillus subtilis |
Bacillus subtilis |
MBC |
6.25 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Bacillus subtilis |
Bacillus subtilis |
MBC |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2021.113723 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.391 |
ug.mL-1 |
10.1016/j.ejmech.2010.10.015 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2019.06.010 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2020.115729 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.027 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2021.113480 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2021.113723 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.625 |
ug.mL-1 |
10.1016/j.bmcl.2011.05.093 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
0.625 |
ug.mL-1 |
10.1021/jm0510023 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.075 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.053 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.01.034 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
1.8 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.11.019 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
3.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.12.063 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113480 |
| Bacillus subtilis |
Bacillus subtilis |
MIC100 |
3.13 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Bacillus subtilis |
Bacillus subtilis |
Ratio |
128.0 |
None |
10.1016/j.ejmech.2021.113480 |
| Bacillus subtilis |
Bacillus subtilis |
Ratio |
128.0 |
None |
10.1016/j.ejmech.2021.113723 |
| Bacillus subtilis (strain 168) |
Cell division protein ftsZ |
Activity |
nan |
None |
10.1016/j.bmc.2019.06.010 |
| Bacillus subtilis (strain 168) |
Cell division protein ftsZ |
Inhibition |
nan |
% |
10.1016/j.ejmech.2021.113723 |
| Bacillus subtilis (strain 168) |
DNA polymerase III |
Ki |
nan |
None |
10.1021/jm0510023 |
| Bacteria |
Bacteria |
MIC90 |
0.5 |
ug.mL-1 |
10.1021/jm960294s |
| Bacteria |
Bacterial 70S ribosome |
IC50 |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.10.018 |
| Bacteria |
Bacterial 70S ribosome |
IC50 |
920000.0 |
nM |
10.1128/aac.01193-07 |
| Bacteria |
Bacterial 70S ribosome |
IC50 |
1380000.0 |
nM |
10.1128/aac.01193-07 |
| Bacteria |
Cell membrane |
Activity |
nan |
None |
10.1016/j.ejmech.2018.06.054 |
| Bacteria |
Cell membrane |
Activity |
nan |
None |
10.1021/acs.jmedchem.0c00826 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm9509556 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
4.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00194-2 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC90 |
4.0 |
ug.mL-1 |
10.1021/jm960294s |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Bacteroides fragilis |
Bacteroides fragilis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bacteroides ovatus |
Bacteroides ovatus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Bacteroides thetaiotaomicron |
Bacteroides thetaiotaomicron |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bifidobacterium bifidum |
Bifidobacterium bifidum |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bifidobacterium bifidum |
Bifidobacterium bifidum |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bifidobacterium bifidum |
Bifidobacterium bifidum |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bifidobacterium breve |
Bifidobacterium breve |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bifidobacterium breve |
Bifidobacterium breve |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bifidobacterium breve |
Bifidobacterium breve |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bifidobacterium longum |
Bifidobacterium longum |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bifidobacterium longum |
Bifidobacterium longum |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Bifidobacterium longum |
Bifidobacterium longum |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Caenorhabditis elegans |
Caenorhabditis elegans |
Activity |
nan |
None |
10.1021/acs.jmedchem.6b01780 |
| Candida albicans |
Candida albicans |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2008.08.079 |
| Candida albicans |
Candida albicans |
MIC |
32.0 |
ug.mL-1 |
10.1021/np800783b |
| Candida albicans |
Candida albicans |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Candida albicans |
Candida albicans |
MIC |
64.0 |
ug.mL-1 |
10.1073/pnas.0700746104 |
| Candida albicans |
Candida albicans |
MIC |
10000.0 |
nM |
10.6019/CHEMBL4513141 |
| Canis lupus familiaris |
Canis familiaris |
Activity |
nan |
None |
10.1021/jm800038g |
| Canis lupus familiaris |
Canis familiaris |
F |
97.0 |
% |
10.1021/jm800038g |
| Canis lupus familiaris |
MDCK |
Papp |
90.0 |
nm/s |
10.1016/j.bmcl.2010.11.043 |
| Canis lupus familiaris |
MDCK |
Papp |
106.0 |
nm/s |
10.1016/j.bmcl.2010.11.043 |
| Chlamydia pneumoniae |
Chlamydia pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Chlamydia pneumoniae |
Chlamydia pneumoniae |
MIC |
nan |
None |
10.1128/aac.01383-07 |
| Chlamydia pneumoniae |
Chlamydia pneumoniae |
MIC50 |
nan |
None |
10.1128/aac.01017-06 |
| Chlamydia pneumoniae |
Chlamydia pneumoniae |
MIC90 |
nan |
None |
10.1128/aac.01017-06 |
| Chlamydia trachomatis |
Chlamydia trachomatis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Chlamydia trachomatis |
Chlamydia trachomatis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Chlorocebus sabaeus |
Vero |
IC50 |
64.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00500 |
| Chlorocebus sabaeus |
Vero |
IC50 |
64.0 |
ug.mL-1 |
10.1021/acsmedchemlett.7b00068 |
| Chlorocebus sabaeus |
Vero |
IC50 |
200.0 |
ug.mL-1 |
10.1016/j.bmc.2018.07.034 |
| Clostridioides difficile |
Clostridioides difficile |
Activity |
nan |
None |
10.1128/aac.00696-08 |
| Clostridioides difficile |
Clostridioides difficile |
MBC |
3.13 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112046 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC |
nan |
None |
10.1021/acs.jmedchem.9b00720 |
| Clostridioides difficile |
Clostridioides difficile |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridioides difficile |
Clostridioides difficile |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium beijerinckii |
Clostridium beijerinckii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium beijerinckii |
Clostridium beijerinckii |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium beijerinckii |
Clostridium beijerinckii |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium butyricum |
Clostridium butyricum |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium butyricum |
Clostridium butyricum |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium butyricum |
Clostridium butyricum |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
Activity |
11.0 |
% |
10.1128/aac.00696-08 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| [Clostridium] innocuum |
[Clostridium] innocuum |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
Activity |
11.0 |
% |
10.1128/aac.00696-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium paraputrificum |
Clostridium paraputrificum |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium perfringens |
Clostridium perfringens |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Clostridium perfringens |
Clostridium perfringens |
Activity |
2.0 |
mg/L |
10.1128/aac.01208-09 |
| Clostridium perfringens |
Clostridium perfringens |
Activity |
4.0 |
mg/L |
10.1128/aac.01208-09 |
| Clostridium perfringens |
Clostridium perfringens |
Activity |
nan |
None |
10.1128/aac.01208-09 |
| Clostridium perfringens |
Clostridium perfringens |
MIC |
0.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Clostridium perfringens |
Clostridium perfringens |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm9509556 |
| Clostridium perfringens |
Clostridium perfringens |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01208-09 |
| Clostridium perfringens |
Clostridium perfringens |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Clostridium perfringens |
Clostridium perfringens |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium perfringens |
Clostridium perfringens |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Clostridium perfringens |
Clostridium perfringens |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium sporogenes |
Clostridium sporogenes |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium sporogenes |
Clostridium sporogenes |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium sporogenes |
Clostridium sporogenes |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium tertium |
Clostridium tertium |
Activity |
11.0 |
% |
10.1128/aac.00696-08 |
| Clostridium tertium |
Clostridium tertium |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium tertium |
Clostridium tertium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium tertium |
Clostridium tertium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium tertium |
Clostridium tertium |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Clostridium tertium |
Clostridium tertium |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Clostridium tertium |
Clostridium tertium |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Collinsella aerofaciens |
Collinsella aerofaciens |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Collinsella aerofaciens |
Collinsella aerofaciens |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Collinsella aerofaciens |
Collinsella aerofaciens |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Corynebacterium amycolatum |
Corynebacterium amycolatum |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Corynebacterium amycolatum |
Corynebacterium amycolatum |
Inhibition |
27.3 |
% |
10.1128/aac.01496-06 |
| Corynebacterium amycolatum |
Corynebacterium amycolatum |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Corynebacterium amycolatum |
Corynebacterium amycolatum |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Corynebacterium amycolatum |
Corynebacterium amycolatum |
MIC90 |
0.25 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Corynebacterium glutamicum |
Corynebacterium glutamicum |
MIC |
0.781 |
ug.mL-1 |
10.1016/j.ejmech.2010.10.015 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
Inhibition |
1.7 |
% |
10.1128/aac.01496-06 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
Inhibition |
5.1 |
% |
10.1128/aac.01496-06 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
Inhibition |
67.8 |
% |
10.1128/aac.01496-06 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
Inhibition |
98.3 |
% |
10.1128/aac.01496-06 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Corynebacterium jeikeium |
Corynebacterium jeikeium |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Corynebacterium pseudodiphtheriticum |
Corynebacterium pseudodiphtheriticum |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Corynebacterium pseudodiphtheriticum |
Corynebacterium pseudodiphtheriticum |
Inhibition |
36.4 |
% |
10.1128/aac.01496-06 |
| Corynebacterium pseudodiphtheriticum |
Corynebacterium pseudodiphtheriticum |
Inhibition |
90.9 |
% |
10.1128/aac.01496-06 |
| Corynebacterium pseudodiphtheriticum |
Corynebacterium pseudodiphtheriticum |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Corynebacterium pseudodiphtheriticum |
Corynebacterium pseudodiphtheriticum |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Corynebacterium pseudodiphtheriticum |
Corynebacterium pseudodiphtheriticum |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Corynebacterium sp. |
Corynebacterium sp. |
Activity |
nan |
None |
10.1128/aac.00845-09 |
| Corynebacterium sp. |
Corynebacterium sp. |
Inhibition |
2.1 |
% |
10.1128/aac.01496-06 |
| Corynebacterium sp. |
Corynebacterium sp. |
Inhibition |
13.6 |
% |
10.1128/aac.01496-06 |
| Corynebacterium sp. |
Corynebacterium sp. |
Inhibition |
68.2 |
% |
10.1128/aac.01496-06 |
| Corynebacterium sp. |
Corynebacterium sp. |
Inhibition |
92.4 |
% |
10.1128/aac.01496-06 |
| Corynebacterium sp. |
Corynebacterium sp. |
Inhibition |
99.6 |
% |
10.1128/aac.01496-06 |
| Corynebacterium sp. |
Corynebacterium sp. |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Corynebacterium sp. |
Corynebacterium sp. |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Corynebacterium sp. |
Corynebacterium sp. |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Corynebacterium sp. |
Corynebacterium sp. |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Corynebacterium sp. |
Corynebacterium sp. |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Corynebacterium sp. |
Corynebacterium sp. |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Corynebacterium sp. |
Corynebacterium sp. |
MIC90 |
0.12 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Corynebacterium sp. |
Corynebacterium sp. |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Corynebacterium sp. |
Corynebacterium sp. |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Corynebacterium striatum |
Corynebacterium striatum |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Corynebacterium striatum |
Corynebacterium striatum |
Inhibition |
12.0 |
% |
10.1128/aac.01496-06 |
| Corynebacterium striatum |
Corynebacterium striatum |
Inhibition |
88.0 |
% |
10.1128/aac.01496-06 |
| Corynebacterium striatum |
Corynebacterium striatum |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Corynebacterium striatum |
Corynebacterium striatum |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Corynebacterium striatum |
Corynebacterium striatum |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Coxiella burnetii |
Coxiella burnetii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01424-08 |
| Coxiella burnetii |
Coxiella burnetii |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01424-08 |
| Coxiella burnetii |
Coxiella burnetii |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01424-08 |
| Coxiella burnetii |
Coxiella burnetii |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01424-08 |
| Cricetulus griseus |
CHO |
CC50 |
nan |
None |
10.1021/jm2002124 |
| Cronobacter sakazakii |
Cronobacter sakazakii |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Cryptococcus neoformans |
Cryptococcus neoformans |
MIC |
10000.0 |
nM |
10.6019/CHEMBL4513141 |
| Cutibacterium acnes |
Cutibacterium acnes |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Cutibacterium acnes |
Cutibacterium acnes |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Cutibacterium acnes |
Cutibacterium acnes |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Cutibacterium acnes |
Cutibacterium acnes |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Eggerthella lenta |
Eggerthella lenta |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Eggerthella lenta |
Eggerthella lenta |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Eggerthella lenta |
Eggerthella lenta |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.10.048 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00072-07 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
16000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
64000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC |
200000.0 |
nM |
10.1016/j.ejmech.2022.114213 |
| Enterobacter cloacae |
Enterobacter cloacae |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Enterobacteriaceae |
Enterobacteriaceae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Enterocloster clostridioformis |
Enterocloster clostridioformis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Enterocloster clostridioformis |
Enterocloster clostridioformis |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Enterocloster clostridioformis |
Enterocloster clostridioformis |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Enterococcus |
Enterococcus |
Activity |
93.8 |
% |
10.1021/jm500960s |
| Enterococcus |
Enterococcus |
Activity |
nan |
None |
10.1021/jm070708p |
| Enterococcus |
Enterococcus |
Efficacy |
88.0 |
% |
10.1021/jm800038g |
| Enterococcus |
Enterococcus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.005 |
| Enterococcus |
Enterococcus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2007.07.006 |
| Enterococcus |
Enterococcus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2009.03.024 |
| Enterococcus |
Enterococcus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.05.041 |
| Enterococcus |
Enterococcus |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Enterococcus |
Enterococcus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00247-07 |
| Enterococcus |
Enterococcus |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.034 |
| Enterococcus |
Enterococcus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115776 |
| Enterococcus |
Enterococcus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.07.005 |
| Enterococcus |
Enterococcus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.01.014 |
| Enterococcus |
Enterococcus |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm500960s |
| Enterococcus |
Enterococcus |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.034 |
| Enterococcus |
Enterococcus |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2009.03.025 |
| Enterococcus |
Enterococcus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.005 |
| Enterococcus |
Enterococcus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.07.006 |
| Enterococcus |
Enterococcus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c00480 |
| Enterococcus |
Enterococcus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm500960s |
| Enterococcus |
Enterococcus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus |
Enterococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Enterococcus |
Enterococcus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus |
Enterococcus |
MIC50 |
4.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115776 |
| Enterococcus |
Enterococcus |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Enterococcus |
Enterococcus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus |
Enterococcus |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115776 |
| Enterococcus avium |
Enterococcus avium |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Enterococcus avium |
Enterococcus avium |
Inhibition |
4.3 |
% |
10.1128/aac.01496-06 |
| Enterococcus avium |
Enterococcus avium |
Inhibition |
52.6 |
% |
10.1128/aac.01496-06 |
| Enterococcus avium |
Enterococcus avium |
Inhibition |
99.1 |
% |
10.1128/aac.01496-06 |
| Enterococcus avium |
Enterococcus avium |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Enterococcus avium |
Enterococcus avium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus avium |
Enterococcus avium |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00908-07 |
| Enterococcus avium |
Enterococcus avium |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Enterococcus avium |
Enterococcus avium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus avium |
Enterococcus avium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus avium |
Enterococcus avium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Enterococcus casseliflavus |
Enterococcus casseliflavus |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Enterococcus casseliflavus |
Enterococcus casseliflavus |
Inhibition |
23.1 |
% |
10.1128/aac.01496-06 |
| Enterococcus casseliflavus |
Enterococcus casseliflavus |
Inhibition |
96.9 |
% |
10.1128/aac.01496-06 |
| Enterococcus casseliflavus |
Enterococcus casseliflavus |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Enterococcus casseliflavus |
Enterococcus casseliflavus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus casseliflavus |
Enterococcus casseliflavus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus casseliflavus |
Enterococcus casseliflavus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Enterococcus casseliflavus |
Enterococcus casseliflavus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus casseliflavus |
Enterococcus casseliflavus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Enterococcus durans |
Enterococcus durans |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Enterococcus durans |
Enterococcus durans |
Inhibition |
2.0 |
% |
10.1128/aac.01496-06 |
| Enterococcus durans |
Enterococcus durans |
Inhibition |
8.2 |
% |
10.1128/aac.01496-06 |
| Enterococcus durans |
Enterococcus durans |
Inhibition |
32.7 |
% |
10.1128/aac.01496-06 |
| Enterococcus durans |
Enterococcus durans |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Enterococcus durans |
Enterococcus durans |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus durans |
Enterococcus durans |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.096 |
| Enterococcus durans |
Enterococcus durans |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus durans |
Enterococcus durans |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Enterococcus durans |
Enterococcus durans |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus durans |
Enterococcus durans |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
ABBC |
-2.66 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
ABBC |
-1.49 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
ABBC |
1.32 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
ABBC |
2.32 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
ABBC |
3.6 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
ABBC |
5.11 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
0.0 |
% |
10.1128/aac.00129-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
0.0 |
% |
10.1128/aac.00149-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
0.0 |
% |
10.1128/aac.00400-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
0.0 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
0.1 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
0.1 |
% |
10.1128/aac.01453-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
0.2 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
1.1 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
1.3 |
% |
10.1128/aac.00400-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
1.4 |
% |
10.1128/aac.01453-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
1.5 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
98.5 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
98.6 |
% |
10.1128/aac.01453-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
98.7 |
% |
10.1128/aac.00400-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
98.9 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
99.8 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
99.8 |
% |
10.1128/aac.01453-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
99.9 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
100.0 |
% |
10.1128/aac.00129-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
100.0 |
% |
10.1128/aac.00149-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
100.0 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
nan |
None |
10.1016/j.ejmech.2008.07.005 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
nan |
None |
10.1021/acs.jmedchem.6b01780 |
| Enterococcus faecalis |
Enterococcus faecalis |
Activity |
nan |
None |
10.1128/aac.00744-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
AUBC |
210.5 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
AUBC |
212.2 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
AUBC |
214.0 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
AUBC |
215.6 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
AUBC |
217.1 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
AUBC |
217.8 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
DIZ |
nan |
None |
10.1016/j.bmcl.2009.10.018 |
| Enterococcus faecalis |
Enterococcus faecalis |
ED50 |
5.6 |
mg.kg-1 |
10.1021/jm401931e |
| Enterococcus faecalis |
Enterococcus faecalis |
ED50 |
6.0 |
mg.kg-1 |
10.1021/jm401931e |
| Enterococcus faecalis |
Enterococcus faecalis |
ED50 |
13.4 |
mg.kg-1 |
10.1021/jm401931e |
| Enterococcus faecalis |
Enterococcus faecalis |
fT>MIC |
0.0 |
% |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
fT>MIC |
8.08 |
% |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
fT>MIC |
69.0 |
% |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
fT>MIC |
69.1 |
% |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
fT>MIC |
80.9 |
% |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
IZ |
25.0 |
mm |
10.1016/j.bmcl.2009.10.018 |
| Enterococcus faecalis |
Enterococcus faecalis |
IZ |
34.0 |
mm |
10.1039/c0md00015a |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/g |
3.0 |
None |
10.1128/aac.00984-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/g |
6.88 |
None |
10.1128/aac.00984-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-1.16 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.5 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.35 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.16 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.14 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.13 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.12 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.08 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.05 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.04 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.03 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.02 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.01 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
-0.009 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.02 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.04 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.06 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.08 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.08 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.09 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.1 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.11 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.13 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.13 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.14 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.15 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.16 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.18 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.19 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.22 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.23 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.25 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.26 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.28 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.29 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.32 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.35 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.39 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.41 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.44 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.45 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.52 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.53 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.55 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.78 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.79 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
0.83 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
1.0 |
None |
10.1128/aac.00984-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
log10CFU/ml |
1.23 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111593 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111830 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2020.112497 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2019.04.063 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2021.113723 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2022.114550 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
64.0 |
ug ml-1 |
10.1039/D1MD00211B |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2022.114550 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC |
128.0 |
ug ml-1 |
10.1039/D1MD00211B |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC50 |
2.0 |
mg/L |
10.1128/aac.00344-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC50 |
2.0 |
mg/L |
10.1128/aac.00666-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC50 |
4.0 |
mg/L |
10.1128/aac.00344-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC50 |
4.0 |
mg/L |
10.1128/aac.00666-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC50 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC50 |
64.0 |
ug ml-1 |
10.1021/acs.jmedchem.6b01780 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC90 |
4.0 |
mg/L |
10.1128/aac.00344-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC90 |
4.0 |
mg/L |
10.1128/aac.00666-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.093 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2007.01.012 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.076 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1016/s0960-894x(02)00043-4 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00734 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1021/acsmedchemlett.0c00653 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
0.8 |
ug.mL-1 |
10.1016/j.bmcl.2016.04.086 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2008.08.079 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.018 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.029 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.033 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.05.066 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.12.025 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.075 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.12.027 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.05.003 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.09.010 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.10.048 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.063 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111593 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111830 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112497 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114550 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1016/s0960-894x(02)00043-4 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00734 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00372 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00379 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm200614t |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm500960s |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm501661f |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1021/np0702032 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1039/c9md00391f |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1039/D1MD00211B |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1073/pnas.0700746104 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00744-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00984-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.25 |
ug.mL-1 |
10.1016/j.bmcl.2011.05.093 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.25 |
ug.mL-1 |
10.1021/jm0510023 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.034 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2009.03.025 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1007/s00044-012-0394-2 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2011.10.041 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116397 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.028 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.021 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.031 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.068 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.02.047 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.024 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.096 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.10.073 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.04.045 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.06.063 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.12.025 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.01.109 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.05.071 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.06.023 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.07.064 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.056 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.075 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.09.024 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.10.061 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.03.043 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.011 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.054 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.03.075 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.07.034 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.023 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.03.013 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.03.053 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.04.046 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.12.027 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.06.022 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128531 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.013 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.007 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113723 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114550 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(01)00305-5 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00249-x |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00194-2 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(99)00473-4 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00295 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00372 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/acsmedchemlett.7b00263 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm020092y |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm070638m |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm4000598 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm401931e |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm500960s |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm501661f |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm980274l |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/np800783b |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00744-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00908-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00984-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01633-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
3.12 |
ug.mL-1 |
10.1016/j.bmcl.2009.07.106 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
3.12 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.033 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
3.12 |
ug.mL-1 |
10.1016/j.ejmech.2009.11.009 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
3.13 |
ug.mL-1 |
10.1016/j.bmcl.2004.07.064 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.017 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.024 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.037 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.03.099 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.11.093 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.056 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.085 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.02.052 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.003 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.08.002 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113480 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00295 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm020248u |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm058204j |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm070638m |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm9509556 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm980546k |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm990373e |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/ml400280z |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/np0702032 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1039/d2md00260d |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00744-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00908-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01193-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.10.010 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113480 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm200614t |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1021/np800783b |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01347-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01633-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.011 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.12.012 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.126746 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.126747 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2020.127660 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.004 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111781 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm4000598 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01633-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.03.043 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.011 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.014 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01193-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01347-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01633-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01347-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01633-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
3000.0 |
nM |
10.1021/acs.jmedchem.0c01198 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
6000.0 |
nM |
10.1016/j.bmcl.2004.08.059 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
6250.0 |
nM |
10.1016/j.ejmech.2020.113002 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
9258.1 |
nM |
10.1016/j.bmcl.2009.04.133 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1016/j.ejmech.2018.09.067 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC100 |
12.5 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC100 |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01780 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00344-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00666-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2009.08.026 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1021/jm1014023 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.004 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
32.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
nan |
None |
10.1128/aac.01017-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC50 |
nan |
None |
10.1128/aac.01398-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.022 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2009.08.026 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm070708p |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm1014023 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00344-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00666-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.07.022 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.004 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
nan |
None |
10.1128/aac.01017-06 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC90 |
nan |
None |
10.1128/aac.01398-07 |
| Enterococcus faecalis |
Enterococcus faecalis |
PD50 |
3.0 |
mg kg-1 |
10.1016/j.bmcl.2010.11.022 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
0.3 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
0.34 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
0.88 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
0.9 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
1.0 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
2.0 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
2.01 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
2.1 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
4.0 |
None |
10.1021/acs.jmedchem.6b01780 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
5.83 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
6.99 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
7.17 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
7.7 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
9.51 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
9.76 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
Ratio |
32.0 |
None |
10.1016/j.ejmech.2021.113723 |
| Enterococcus faecalis |
Enterococcus faecalis |
RatioAUC/MIC |
1.24 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
RatioAUC/MIC |
3.9 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
RatioAUC/MIC |
10.2 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
RatioAUC/MIC |
35.4 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
RatioAUC/MIC |
37.1 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecalis |
Enterococcus faecalis |
RatioAUC/MIC |
42.9 |
None |
10.1128/aac.01022-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
0.0 |
% |
10.1128/aac.00149-08 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
0.0 |
% |
10.1128/aac.00400-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
0.0 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
0.3 |
% |
10.1128/aac.01453-08 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
0.4 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
0.5 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
0.6 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
0.7 |
% |
10.1128/aac.00129-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
0.87 |
log10CFU |
10.1021/acsmedchemlett.3c00032 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
1.07 |
log10CFU |
10.1021/acsmedchemlett.3c00032 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
1.8 |
% |
10.1128/aac.01453-08 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
3.4 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
8.6 |
% |
10.1128/aac.00400-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
86.5 |
% |
10.1021/acsmedchemlett.3c00032 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
91.4 |
% |
10.1128/aac.00400-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
91.5 |
% |
10.1021/acsmedchemlett.3c00032 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
93.1 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
96.0 |
% |
10.1128/aac.01398-07 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
97.6 |
% |
10.1128/aac.01453-08 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
99.0 |
% |
10.1128/aac.01398-07 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
99.1 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
99.3 |
% |
10.1128/aac.00129-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
99.3 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
99.4 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
99.5 |
% |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
99.6 |
% |
10.1128/aac.01453-08 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
100.0 |
% |
10.1128/aac.00149-08 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
nan |
None |
10.1021/acs.jmedchem.0c00734 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
nan |
None |
10.1021/acs.jmedchem.6b01780 |
| Enterococcus faecium |
Enterococcus faecium |
Activity |
nan |
None |
10.1021/acsmedchemlett.3c00032 |
| Enterococcus faecium |
Enterococcus faecium |
AUPAP |
40.0 |
% |
10.1128/aac.01194-06 |
| Enterococcus faecium |
Enterococcus faecium |
ED50 |
3.91 |
mg.kg-1 |
10.1016/j.bmcl.2007.09.024 |
| Enterococcus faecium |
Enterococcus faecium |
ED50 |
11.4 |
mg.kg-1 |
10.1016/j.bmcl.2016.04.086 |
| Enterococcus faecium |
Enterococcus faecium |
log10CFU/ml |
-2.0 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecium |
Enterococcus faecium |
log10CFU/ml |
-0.72 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecium |
Enterococcus faecium |
log10CFU/ml |
-0.63 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecium |
Enterococcus faecium |
log10CFU/ml |
-0.42 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecium |
Enterococcus faecium |
log10CFU/ml |
-0.35 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecium |
Enterococcus faecium |
log10CFU/ml |
0.2 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecium |
Enterococcus faecium |
log10CFU/ml |
3.0 |
None |
10.1128/aac.01194-06 |
| Enterococcus faecium |
Enterococcus faecium |
log10CFU/ml |
3.8 |
None |
10.1128/aac.01194-06 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
4.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
4.69 |
uM |
10.1021/acs.jmedchem.1c00168 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
4.69 |
uM |
10.1021/acs.jmedchem.5b02004 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
4.69 |
uM |
10.1021/acs.jmedchem.7b01903 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
4.69 |
uM |
10.1039/C6MD00381H |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
8.0 |
ug ml-1 |
10.1016/j.ejmech.2019.04.063 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111593 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111830 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2020.112497 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
32.0 |
ug ml-1 |
10.1021/acs.jmedchem.6b00233 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.023 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2021.113723 |
| Enterococcus faecium |
Enterococcus faecium |
MBC |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2022.114550 |
| Enterococcus faecium |
Enterococcus faecium |
MBC50 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Enterococcus faecium |
Enterococcus faecium |
MBC50 |
16.0 |
ug ml-1 |
10.1021/acs.jmedchem.6b01780 |
| Enterococcus faecium |
Enterococcus faecium |
MBC50 |
128.0 |
ug ml-1 |
10.1021/acs.jmedchem.6b01780 |
| Enterococcus faecium |
Enterococcus faecium |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Enterococcus faecium |
Enterococcus faecium |
MBEC |
1.56 |
uM |
10.1021/acs.jmedchem.1c00168 |
| Enterococcus faecium |
Enterococcus faecium |
MBEC |
1.56 |
uM |
10.1021/acs.jmedchem.5b02004 |
| Enterococcus faecium |
Enterococcus faecium |
MBEC |
1.56 |
uM |
10.1021/acs.jmedchem.7b01903 |
| Enterococcus faecium |
Enterococcus faecium |
MBEC |
1.56 |
uM |
10.1039/C6MD00381H |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.25 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00734 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2011.10.041 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.022 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.063 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00734 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01780 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.034 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.12.012 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.126746 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2020.127660 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.05.003 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.10.048 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.023 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.004 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111593 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111781 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111830 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112497 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114550 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1016/s0960-894x(99)00473-4 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00734 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00233 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1021/acsmedchemlett.3c00032 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00379 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm500960s |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm501661f |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00197-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.25 |
ug.mL-1 |
10.1016/j.bmcl.2011.05.093 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.25 |
ug.mL-1 |
10.1021/jm0510023 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.01710-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.034 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2009.03.025 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.033 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
1.6 |
ug.mL-1 |
10.1016/j.bmcl.2016.04.086 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116397 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.028 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.021 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.031 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.068 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.096 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.10.073 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.03.099 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.04.045 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.06.063 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.05.071 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.06.023 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.12.081 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.056 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.09.024 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.10.061 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.03.043 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.054 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.08.037 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.03.013 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.12.012 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.126746 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.126747 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2020.127660 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.013 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.003 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.08.002 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.004 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111781 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(01)00305-5 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(02)00352-9 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(99)00473-4 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00295 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00372 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1021/acsmedchemlett.7b00263 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm020092y |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm500960s |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm501661f |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm800800c |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm9509556 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1021/ml400280z |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1073/pnas.0700746104 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00197-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01194-06 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.5 |
ug.mL-1 |
10.1016/j.bmcl.2011.05.093 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2.5 |
ug.mL-1 |
10.1021/jm0510023 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.037 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.03.104 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128531 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113723 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
4.0 |
ug.mL-1 |
10.1039/d2md00260d |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm200614t |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01347-06 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm4000598 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01193-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01347-06 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
30.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00153 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
32.0 |
ug.mL-1 |
10.1021/np800783b |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01347-06 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01347-06 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
64.0 |
ug/sq.cm |
10.1128/aac.01347-06 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
500.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
3000.0 |
nM |
10.1021/acs.jmedchem.0c01198 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
3130.0 |
nM |
10.1016/j.ejmech.2018.06.045 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
3130.0 |
nM |
10.1021/acs.jmedchem.5b02004 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
3130.0 |
nM |
10.1039/C6MD00381H |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
6000.0 |
nM |
10.1016/j.ejmech.2022.114213 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
6250.0 |
nM |
10.1016/j.ejmech.2020.113002 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
11860.0 |
nM |
10.1016/j.ejmech.2019.02.004 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
12500.0 |
nM |
10.1016/j.ejmech.2020.113002 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
89000.0 |
nM |
10.1021/acs.jnatprod.2c00153 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
100000.0 |
nM |
10.1016/j.bmcl.2004.08.059 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
2000000.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.021 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
4000000.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.021 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
8000000.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.021 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
16000000.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.021 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
nan |
None |
10.1016/j.bmcl.2007.06.075 |
| Enterococcus faecium |
Enterococcus faecium |
MIC |
nan |
None |
10.1021/np800503z |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01780 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm1014023 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2009.08.026 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.004 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01780 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
32.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC50 |
nan |
None |
10.1128/aac.01017-06 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2009.08.026 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.022 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm1014023 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.004 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
4.0 |
ug.mL-1 |
10.1021/jm070708p |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
4.0 |
ug.mL-1 |
10.1021/jm960294s |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
nan |
None |
10.1128/aac.01017-06 |
| Enterococcus faecium |
Enterococcus faecium |
PD50 |
4.0 |
mg kg-1 |
10.1016/j.bmcl.2010.11.022 |
| Enterococcus faecium |
Enterococcus faecium |
Ratio |
1.0 |
None |
10.1021/acs.jmedchem.6b01780 |
| Enterococcus faecium |
Enterococcus faecium |
Ratio |
2.0 |
None |
10.1128/aac.00197-09 |
| Enterococcus faecium |
Enterococcus faecium |
Ratio |
4.0 |
None |
10.1021/acs.jmedchem.6b01780 |
| Enterococcus faecium |
Enterococcus faecium |
Ratio |
16.0 |
None |
10.1016/j.ejmech.2021.113723 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
Inhibition |
1.7 |
% |
10.1128/aac.01496-06 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
Inhibition |
30.3 |
% |
10.1128/aac.01496-06 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
Inhibition |
99.2 |
% |
10.1128/aac.01496-06 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
MIC50 |
nan |
None |
10.1128/aac.01017-06 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Enterococcus gallinarum |
Enterococcus gallinarum |
MIC90 |
nan |
None |
10.1128/aac.01017-06 |
| Enterococcus hirae |
Enterococcus hirae |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Enterococcus hirae |
Enterococcus hirae |
Inhibition |
37.5 |
% |
10.1128/aac.01496-06 |
| Enterococcus hirae |
Enterococcus hirae |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Enterococcus hirae |
Enterococcus hirae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus hirae |
Enterococcus hirae |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus hirae |
Enterococcus hirae |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Enterococcus hirae |
Enterococcus hirae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Enterococcus hirae |
Enterococcus hirae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Enterococcus sp. |
Enterococcus sp. |
Activity |
0.0 |
% |
10.1128/aac.01538-07 |
| Enterococcus sp. |
Enterococcus sp. |
Activity |
1.5 |
% |
10.1128/aac.01538-07 |
| Enterococcus sp. |
Enterococcus sp. |
Activity |
1.6 |
% |
10.1128/aac.01538-07 |
| Enterococcus sp. |
Enterococcus sp. |
Activity |
1.8 |
% |
10.1128/aac.01538-07 |
| Enterococcus sp. |
Enterococcus sp. |
Activity |
2.9 |
% |
10.1128/aac.01538-07 |
| Enterococcus sp. |
Enterococcus sp. |
MBC |
4.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Enterococcus sp. |
Enterococcus sp. |
MBC50 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Enterococcus sp. |
Enterococcus sp. |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Enterococcus sp. |
Enterococcus sp. |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Enterococcus sp. |
Enterococcus sp. |
MIC50 |
2.0 |
ug.mL-1 |
10.1021/jm020328y |
| Enterococcus sp. |
Enterococcus sp. |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Enterococcus sp. |
Enterococcus sp. |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm020328y |
| Enterococcus sp. |
Enterococcus sp. |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Enterococcus sp. |
Enterococcus sp. |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.023 |
| Escherichia coli |
DNA gyrase |
IC50 |
32000.0 |
nM |
10.1021/jm501174m |
| Escherichia coli |
DNA gyrase |
IC50 |
nan |
nM |
10.1016/j.bmcl.2003.07.028 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1016/j.bmcl.2008.10.045 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1016/j.ejmech.2008.07.005 |
| Escherichia coli |
Escherichia coli |
IC50 |
0.05 |
ug.mL-1 |
10.1016/j.bmc.2018.07.034 |
| Escherichia coli |
Escherichia coli |
IC50 |
0.49 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Escherichia coli |
Escherichia coli |
IC50 |
950.0 |
nM |
10.1016/j.bmcl.2007.05.056 |
| Escherichia coli |
Escherichia coli |
IC50 |
950.0 |
nM |
10.1016/j.bmcl.2007.05.085 |
| Escherichia coli |
Escherichia coli |
IC50 |
3300.0 |
nM |
10.1016/j.bmcl.2006.07.064 |
| Escherichia coli |
Escherichia coli |
IC50 |
3600.0 |
nM |
10.1016/j.bmcl.2008.02.052 |
| Escherichia coli |
Escherichia coli |
IC50 |
3600.0 |
nM |
10.1021/jm070708p |
| Escherichia coli |
Escherichia coli |
IC50 |
4100.0 |
nM |
10.1016/j.bmcl.2003.07.028 |
| Escherichia coli |
Escherichia coli |
IC50 |
4600.0 |
nM |
10.1016/j.bmcl.2008.10.011 |
| Escherichia coli |
Escherichia coli |
IC50 |
4600.0 |
nM |
10.1016/j.bmcl.2008.10.014 |
| Escherichia coli |
Escherichia coli |
IC50 |
8700.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Escherichia coli |
Escherichia coli |
IC50 |
9300.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Escherichia coli |
Escherichia coli |
IC50 |
11000.0 |
nM |
10.1016/j.bmcl.2007.07.022 |
| Escherichia coli |
Escherichia coli |
IC50 |
18000.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Escherichia coli |
Escherichia coli |
IC50 |
100000.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Escherichia coli |
Escherichia coli |
Inhibition |
99.34 |
% |
10.1016/j.ejmech.2016.07.001 |
| Escherichia coli |
Escherichia coli |
Inhibition |
99.77 |
% |
10.1016/j.ejmech.2016.07.001 |
| Escherichia coli |
Escherichia coli |
Inhibition |
100.15 |
% |
10.1016/j.ejmech.2016.07.001 |
| Escherichia coli |
Escherichia coli |
Inhibition |
nan |
% |
10.1016/j.bmc.2018.07.034 |
| Escherichia coli |
Escherichia coli |
IZ |
0.0 |
mm |
10.1016/j.bmcl.2009.10.018 |
| Escherichia coli |
Escherichia coli |
IZ |
12.0 |
mm |
10.1016/j.ejmech.2011.04.041 |
| Escherichia coli |
Escherichia coli |
IZ |
23.0 |
mm |
10.1039/c0md00015a |
| Escherichia coli |
Escherichia coli |
IZ |
28.0 |
mm |
10.1039/c0md00015a |
| Escherichia coli |
Escherichia coli |
IZ |
nan |
None |
10.1016/j.ejmech.2013.01.034 |
| Escherichia coli |
Escherichia coli |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Escherichia coli |
Escherichia coli |
MBEC |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.054 |
| Escherichia coli |
Escherichia coli |
MBEC80 |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.054 |
| Escherichia coli |
Escherichia coli |
MBEC90 |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.054 |
| Escherichia coli |
Escherichia coli |
MBIC80 |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.054 |
| Escherichia coli |
Escherichia coli |
MBIC90 |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.054 |
| Escherichia coli |
Escherichia coli |
MIC |
1.15 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Escherichia coli |
Escherichia coli |
MIC |
1.95 |
ug.mL-1 |
10.1128/aac.00580-10 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.12.063 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Escherichia coli |
Escherichia coli |
MIC |
2.0 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00015 |
| Escherichia coli |
Escherichia coli |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.02.002 |
| Escherichia coli |
Escherichia coli |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.bmcl.2004.07.064 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.028 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.005 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.11.019 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.07.006 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.023 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111850 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112046 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1016/s0960-894x(01)00305-5 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01780 |
| Escherichia coli |
Escherichia coli |
MIC |
8.0 |
ug.mL-1 |
10.1039/d2md00260d |
| Escherichia coli |
Escherichia coli |
MIC |
11.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.10.018 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.037 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.096 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.04.045 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.03.075 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128531 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00580-10 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00921-08 |
| Escherichia coli |
Escherichia coli |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01015-07 |
| Escherichia coli |
Escherichia coli |
MIC |
31.25 |
ug.mL-1 |
10.1128/aac.00580-10 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2008.08.079 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2011.10.041 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.037 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1016/s0960-894x(01)00305-5 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00015 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm020248u |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1021/np0702032 |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1039/C5MD00101C |
| Escherichia coli |
Escherichia coli |
MIC |
32.0 |
ug.mL-1 |
10.1073/pnas.0700746104 |
| Escherichia coli |
Escherichia coli |
MIC |
36.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.10.018 |
| Escherichia coli |
Escherichia coli |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.04.086 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2019.06.010 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115729 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.028 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.123 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128531 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.03.024 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.05.041 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.106 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.053 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112046 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113480 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113723 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jnatprod.9b00321 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm058204j |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm9509556 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1021/np800503z |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1073/pnas.0700746104 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01015-07 |
| Escherichia coli |
Escherichia coli |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01208-09 |
| Escherichia coli |
Escherichia coli |
MIC |
80.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.05.093 |
| Escherichia coli |
Escherichia coli |
MIC |
80.0 |
ug.mL-1 |
10.1021/jm0510023 |
| Escherichia coli |
Escherichia coli |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.09.019 |
| Escherichia coli |
Escherichia coli |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2010.10.015 |
| Escherichia coli |
Escherichia coli |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.04.041 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.023 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111850 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b01780 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00015 |
| Escherichia coli |
Escherichia coli |
MIC |
128.0 |
ug.mL-1 |
10.1021/jm070638m |
| Escherichia coli |
Escherichia coli |
MIC |
130.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.10.018 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.02.002 |
| Escherichia coli |
Escherichia coli |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01015-07 |
| Escherichia coli |
Escherichia coli |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00921-08 |
| Escherichia coli |
Escherichia coli |
MIC |
1024.0 |
ug.mL-1 |
10.1128/aac.00921-08 |
| Escherichia coli |
Escherichia coli |
MIC |
6250.0 |
nM |
10.1016/j.ejmech.2020.113002 |
| Escherichia coli |
Escherichia coli |
MIC |
10000.0 |
nM |
10.6019/CHEMBL4513141 |
| Escherichia coli |
Escherichia coli |
MIC |
16000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Escherichia coli |
Escherichia coli |
MIC |
20000.0 |
nM |
10.1021/jm501174m |
| Escherichia coli |
Escherichia coli |
MIC |
25000.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Escherichia coli |
Escherichia coli |
MIC |
47400.0 |
nM |
10.1021/acs.jmedchem.0c01198 |
| Escherichia coli |
Escherichia coli |
MIC |
50000.0 |
nM |
10.1016/j.ejmech.2022.114333 |
| Escherichia coli |
Escherichia coli |
MIC |
50000.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Escherichia coli |
Escherichia coli |
MIC |
64000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Escherichia coli |
Escherichia coli |
MIC |
75000.0 |
nM |
10.1016/j.ejmech.2020.113002 |
| Escherichia coli |
Escherichia coli |
MIC |
100000.0 |
nM |
10.1016/j.bmcl.2004.08.059 |
| Escherichia coli |
Escherichia coli |
MIC |
100000.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Escherichia coli |
Escherichia coli |
MIC |
200000.0 |
nM |
10.1016/j.ejmech.2022.114213 |
| Escherichia coli |
Escherichia coli |
MIC |
200000.0 |
nM |
10.1021/jm501174m |
| Escherichia coli |
Escherichia coli |
MIC |
1897000.0 |
nM |
10.1021/acs.jmedchem.0c01198 |
| Escherichia coli |
Escherichia coli |
MIC |
64000000.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.021 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.bmc.2015.02.016 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.bmc.2019.05.012 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1021/acs.jmedchem.0c00295 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1021/np800503z |
| Escherichia coli |
Escherichia coli |
MIC100 |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Escherichia coli |
Escherichia coli |
MIC90 |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Escherichia coli |
Escherichia coli |
MIC90 |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Escherichia coli |
Escherichia coli |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Escherichia coli |
Escherichia coli |
MIC90 |
128.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Escherichia coli |
Escherichia coli |
MIC90 |
256.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.06.022 |
| Escherichia coli |
Escherichia coli |
MIC99 |
32.0 |
ug ml-1 |
10.1016/j.bmcl.2014.02.025 |
| Escherichia coli |
Escherichia coli |
Ratio |
3.6 |
None |
10.1016/j.bmcl.2017.10.018 |
| Escherichia coli |
Escherichia coli |
Ratio |
4.0 |
None |
10.1128/aac.00921-08 |
| Escherichia coli |
Escherichia coli |
Ratio |
12.0 |
None |
10.1016/j.bmcl.2017.10.018 |
| Finegoldia magna |
Finegoldia magna |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Finegoldia magna |
Finegoldia magna |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Finegoldia magna |
Finegoldia magna |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Finegoldia magna |
Finegoldia magna |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Finegoldia magna |
Finegoldia magna |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Finegoldia magna |
Finegoldia magna |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Finegoldia magna |
Finegoldia magna |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Fusobacterium mortiferum |
Fusobacterium mortiferum |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Fusobacterium varium |
Fusobacterium varium |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Fusobacterium varium |
Fusobacterium varium |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Fusobacterium varium |
Fusobacterium varium |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Haemophilus influenzae |
Haemophilus influenzae |
Activity |
nan |
None |
10.1016/j.ejmech.2008.07.005 |
| Haemophilus influenzae |
Haemophilus influenzae |
MBC |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MBC50 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.033 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.034 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2009.03.025 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.056 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.03.013 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128842 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
4.0 |
ug.mL-1 |
10.1021/acsmedchemlett.7b00263 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.022 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.028 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.076 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.01.109 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.10.063 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.056 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.085 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.03.043 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.011 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.014 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.005 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.07.006 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.07.005 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.03.024 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.01.014 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.05.041 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm201467r |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1021/np800503z |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
12.0 |
ug.mL-1 |
10.1021/np0702032 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmc.2011.10.041 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.017 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.018 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.029 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.11.093 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.03.104 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.07.064 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.011 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.014 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.03.013 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.03.024 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.003 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.08.002 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm020248u |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm058204j |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm800800c |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm980546k |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm990373e |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1021/ml400280z |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2008.08.079 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.011 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
12500.0 |
nM |
10.1021/acs.jmedchem.5b00050 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
23000.0 |
nM |
10.1021/jm501174m |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
32000.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.04.003 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
16000000.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.021 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC |
nan |
None |
10.1016/j.bmcl.2010.11.102 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
0.03 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
8.0 |
ug.mL-1 |
10.1021/jm1014023 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
8.0 |
ug.mL-1 |
10.1021/jm201467r |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC50 |
nan |
None |
10.1128/aac.01017-06 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
16.0 |
ug.mL-1 |
10.1021/jm1014023 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
16.0 |
ug.mL-1 |
10.1021/jm201467r |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
16.0 |
ug.mL-1 |
10.1021/jm960294s |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
32.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.023 |
| Haemophilus influenzae |
Haemophilus influenzae |
MIC90 |
nan |
None |
10.1128/aac.01017-06 |
| Haemophilus parainfluenzae |
Haemophilus parainfluenzae |
MIC |
16.0 |
ug.mL-1 |
10.1021/np800503z |
| Homo sapiens |
A549 |
IC50 |
nan |
None |
10.1021/acs.jnatprod.9b00321 |
| Homo sapiens |
Adenosine A1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A2a receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2b adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2c adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Anandamide amidohydrolase |
Inhibition |
5.7 |
% |
10.1016/j.bmcl.2009.09.086 |
| Homo sapiens |
Beta-1 adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-2 adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bile salt export pump |
AC50 |
300000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bile salt export pump |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Bile salt export pump |
IC50 |
1000000.0 |
nM |
10.1124/dmd.112.047068 |
| Homo sapiens |
Bradykinin B2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Caco-2 |
IC50 |
nan |
None |
10.1021/acs.jnatprod.9b00321 |
| Homo sapiens |
Calmodulin-like protein 3 |
IC50 |
9300.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 1 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 2 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Cannabinoid CB1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cholecystokinin A receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cholecystokinin B receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-1 |
IC50 |
8190.0 |
nM |
10.1016/j.bmcl.2019.07.024 |
| Homo sapiens |
Cyclooxygenase-2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cytochrome P450 1A2 |
IC50 |
20000.0 |
nM |
10.1016/j.ejmech.2013.03.003 |
| Homo sapiens |
Cytochrome P450 1A2 |
IC50 |
20000.0 |
nM |
10.1021/ml400280z |
| Homo sapiens |
Cytochrome P450 1A2 |
INH |
100.0 |
uM |
10.1016/j.bmcl.2019.07.024 |
| Homo sapiens |
Cytochrome P450 1A2 |
Inhibition |
nan |
% |
10.1016/j.ejmech.2013.08.002 |
| Homo sapiens |
Cytochrome P450 2C19 |
INH |
100.0 |
uM |
10.1016/j.bmcl.2019.07.024 |
| Homo sapiens |
Cytochrome P450 2C9 |
IC50 |
20000.0 |
nM |
10.1016/j.ejmech.2013.03.003 |
| Homo sapiens |
Cytochrome P450 2C9 |
IC50 |
20000.0 |
nM |
10.1021/ml400280z |
| Homo sapiens |
Cytochrome P450 2C9 |
INH |
100.0 |
uM |
10.1016/j.bmcl.2019.07.024 |
| Homo sapiens |
Cytochrome P450 2C9 |
Inhibition |
nan |
% |
10.1016/j.ejmech.2013.08.002 |
| Homo sapiens |
Cytochrome P450 2D6 |
IC50 |
20000.0 |
nM |
10.1016/j.ejmech.2013.03.003 |
| Homo sapiens |
Cytochrome P450 2D6 |
IC50 |
20000.0 |
nM |
10.1021/ml400280z |
| Homo sapiens |
Cytochrome P450 2D6 |
INH |
100.0 |
uM |
10.1016/j.bmcl.2019.07.024 |
| Homo sapiens |
Cytochrome P450 2D6 |
Inhibition |
nan |
% |
10.1016/j.ejmech.2013.08.002 |
| Homo sapiens |
Cytochrome P450 3A4 |
IC50 |
20000.0 |
nM |
10.1016/j.ejmech.2013.03.003 |
| Homo sapiens |
Cytochrome P450 3A4 |
IC50 |
20000.0 |
nM |
10.1021/ml400280z |
| Homo sapiens |
Cytochrome P450 3A4 |
INH |
100.0 |
uM |
10.1016/j.bmcl.2019.07.024 |
| Homo sapiens |
Cytochrome P450 3A4 |
Inhibition |
nan |
% |
10.1016/j.ejmech.2013.08.002 |
| Homo sapiens |
Delta opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Endothelin receptor ET-A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Equilibrative nucleoside transporter 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Ghrelin receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
HaCaT |
Activity |
nan |
None |
10.1016/j.ejmech.2013.03.069 |
| Homo sapiens |
HEK293 |
CC50 |
4460.0 |
nM |
10.6019/CHEMBL4513141 |
| Homo sapiens |
HeLa |
Activity |
nan |
None |
10.1128/aac.00729-05 |
| Homo sapiens |
HeLa |
CC50 |
nan |
None |
10.1021/jm2002124 |
| Homo sapiens |
HeLa |
IC20 |
300.0 |
ug ml-1 |
10.1128/aac.00729-05 |
| Homo sapiens |
HeLa |
IC50 |
100.0 |
ug.mL-1 |
10.1073/pnas.0700746104 |
| Homo sapiens |
HeLa |
IC50 |
400.0 |
ug.mL-1 |
10.1128/aac.00729-05 |
| Homo sapiens |
HEp-2 |
CC50 |
nan |
None |
10.1021/jm2002124 |
| Homo sapiens |
HepG2 |
Activity |
20.0 |
% |
10.1016/j.bmc.2014.10.037 |
| Homo sapiens |
HepG2 |
Activity |
nan |
None |
10.1016/j.ejmech.2013.03.069 |
| Homo sapiens |
HepG2 |
CC50 |
nan |
None |
10.1021/jm2002124 |
| Homo sapiens |
HepG2 |
EC50 |
30000.0 |
nM |
10.1016/j.bmcl.2019.07.024 |
| Homo sapiens |
HepG2 |
IC50 |
25000.0 |
nM |
10.1016/j.bmcl.2018.12.012 |
| Homo sapiens |
HepG2 |
IC50 |
25000.0 |
nM |
10.1016/j.ejmech.2018.09.004 |
| Homo sapiens |
HepG2 |
IC50 |
25000.0 |
nM |
10.1016/j.ejmech.2019.111781 |
| Homo sapiens |
HepG2 |
IC50 |
64000.0 |
nM |
10.1016/j.bmcl.2019.126746 |
| Homo sapiens |
HERG |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
HERG |
Inhibition |
nan |
% |
10.1021/jm2002124 |
| Homo sapiens |
Histamine H1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histone deacetylase 6 |
Inhibition |
-36.28 |
% |
10.6019/CHEMBL4808148 |
| Homo sapiens |
Histone deacetylase 6 |
Inhibition |
-3.13 |
% |
10.6019/CHEMBL4808148 |
| Homo sapiens |
Homo sapiens |
Activity |
nan |
None |
10.1021/jm020248u |
| Homo sapiens |
Homo sapiens |
AUC |
60100.0 |
ng.hr.mL-1 |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
AUC |
66800.0 |
ng.hr.mL-1 |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
AUC |
80300.0 |
ng.hr.mL-1 |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
AUC |
84600.0 |
ng.hr.mL-1 |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
AUC |
88100.0 |
ng.hr.mL-1 |
10.1128/aac.01022-09 |
| Homo sapiens |
Homo sapiens |
AUC |
96800.0 |
ng.hr.mL-1 |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
AUC |
124500.0 |
ng.hr.mL-1 |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
AUC |
136400.0 |
ng.hr.mL-1 |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
AUC |
160700.0 |
ng.hr.mL-1 |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
AUC |
196080.0 |
ng.hr.mL-1 |
10.1128/aac.00177-10 |
| Homo sapiens |
Homo sapiens |
AUC |
260000.0 |
ng.hr.mL-1 |
10.1128/aac.00247-07 |
| Homo sapiens |
Homo sapiens |
AUC |
412550.0 |
ng.hr.mL-1 |
10.1128/aac.00177-10 |
| Homo sapiens |
Homo sapiens |
CL |
1.2 |
mL.min-1.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
CL |
1.8 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
CL |
1.8 |
mL.min-1.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
CL |
70.0 |
ml/min |
10.1021/jm800038g |
| Homo sapiens |
Homo sapiens |
CL |
100.0 |
ml/min |
10.1021/jm800038g |
| Homo sapiens |
Homo sapiens |
CL/F |
4.8 |
L/hr |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
CL/F |
7.1 |
L/hr |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
CL_renal |
0.6 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
CL_renal |
0.6 |
mL.min-1.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
CL_renal |
30.0 |
ml/min |
10.1021/jm800038g |
| Homo sapiens |
Homo sapiens |
Cmax |
30532.09 |
nM |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
Cmax |
39721.36 |
nM |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
Cmax |
41796.35 |
nM |
10.1128/aac.01022-09 |
| Homo sapiens |
Homo sapiens |
Cmax |
43574.92 |
nM |
10.1128/aac.00177-10 |
| Homo sapiens |
Homo sapiens |
Cmax |
44167.78 |
nM |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
Cmax |
47428.49 |
nM |
10.1128/aac.00197-09 |
| Homo sapiens |
Homo sapiens |
Cmax |
57507.04 |
nM |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
Cmin |
0.68 |
mg/L |
10.1128/aac.00177-10 |
| Homo sapiens |
Homo sapiens |
Cmin |
2.94 |
mg/L |
10.1128/aac.00177-10 |
| Homo sapiens |
Homo sapiens |
Cmin |
3.8 |
mg/L |
10.1128/aac.00177-10 |
| Homo sapiens |
Homo sapiens |
Cmin |
4.0 |
ug ml-1 |
10.1128/aac.00197-09 |
| Homo sapiens |
Homo sapiens |
Cmin |
4.78 |
mg/L |
10.1128/aac.00177-10 |
| Homo sapiens |
Homo sapiens |
Cmin |
7.0 |
ug ml-1 |
10.1021/jm800038g |
| Homo sapiens |
Homo sapiens |
Cmin |
26.99 |
mg/L |
10.1128/aac.00177-10 |
| Homo sapiens |
Homo sapiens |
DILI_Concern |
nan |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
DILI_severity_class |
3.0 |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
Dose non renally cleared |
65.0 |
% |
10.1128/aac.00177-10 |
| Homo sapiens |
Homo sapiens |
F |
100.0 |
% |
10.1016/j.bmc.2007.08.060 |
| Homo sapiens |
Homo sapiens |
F |
100.0 |
% |
10.1021/jm800038g |
| Homo sapiens |
Homo sapiens |
F |
100.0 |
% |
10.1128/aac.00638-07 |
| Homo sapiens |
Homo sapiens |
Fa |
1.0 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
F_fraction |
1.0 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Fg |
1.05 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Fh |
0.95 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
ka |
1.5 |
/hr |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
ka |
2.7 |
/hr |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
Kel |
0.2 |
/hr |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
T1/2 |
0.3 |
hr |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
T1/2 |
0.5 |
hr |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.9 |
hr |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
T1/2 |
4.6 |
hr |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
T1/2 |
5.0 |
hr |
10.1021/jm800038g |
| Homo sapiens |
Homo sapiens |
T1/2 |
5.1 |
hr |
10.1128/aac.01022-09 |
| Homo sapiens |
Homo sapiens |
Tmax |
1.0 |
hr |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
Tmax |
1.5 |
hr |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
Vc/F |
29.6 |
l |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
Vc/F |
32.1 |
l |
10.1128/aac.01378-08 |
| Homo sapiens |
Homo sapiens |
Vdss |
0.58 |
L.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Huh-7 |
CC50 |
nan |
nM |
10.1016/j.bmcl.2004.08.059 |
| Homo sapiens |
Kappa opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Liver microsome |
Stability |
100.0 |
% |
10.1021/acsmedchemlett.5b00213 |
| Homo sapiens |
Melanocortin receptor 3 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
MG-63 |
Activity |
nan |
None |
10.1128/aac.00729-05 |
| Homo sapiens |
MG-63 |
IC20 |
250.0 |
ug ml-1 |
10.1128/aac.00729-05 |
| Homo sapiens |
MG-63 |
IC50 |
400.0 |
ug.mL-1 |
10.1128/aac.00729-05 |
| Homo sapiens |
Monoamine oxidase A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Monoamine oxidase A |
IC50 |
3.8 |
ug.mL-1 |
10.1021/jm401931e |
| Homo sapiens |
Monoamine oxidase A |
IC50 |
8.1 |
ug.mL-1 |
10.1021/jm401931e |
| Homo sapiens |
Monoamine oxidase A |
IC50 |
46000.0 |
nM |
10.1016/j.ejmech.2015.10.025 |
| Homo sapiens |
Monoamine oxidase A |
Inhibition |
6.79 |
% |
10.1016/j.bmcl.2013.01.033 |
| Homo sapiens |
Monoamine oxidase A |
Inhibition |
50.0 |
% |
10.1016/j.ejmech.2015.10.025 |
| Homo sapiens |
Monoamine oxidase A |
Inhibition |
74.0 |
% |
10.1016/j.ejmech.2018.09.004 |
| Homo sapiens |
Monoamine oxidase A |
Inhibition |
75.0 |
% |
10.1016/j.bmcl.2019.126746 |
| Homo sapiens |
Monoamine oxidase A |
Inhibition |
76.0 |
% |
10.1016/j.bmcl.2018.12.012 |
| Homo sapiens |
Monoamine oxidase A |
Inhibition |
76.0 |
% |
10.1016/j.ejmech.2019.111781 |
| Homo sapiens |
Monoamine oxidase A |
Ki |
7900.0 |
nM |
10.1016/j.bmc.2012.11.036 |
| Homo sapiens |
Monoamine oxidase A |
Ki |
20000.0 |
nM |
10.1016/j.bmcl.2006.10.063 |
| Homo sapiens |
Monoamine oxidase A |
Ki |
53000.0 |
nM |
10.1021/jm070708p |
| Homo sapiens |
Monoamine oxidase A |
Ki |
55000.0 |
nM |
10.1021/jm800038g |
| Homo sapiens |
Monoamine oxidase B |
IC50 |
2100.0 |
nM |
10.1016/j.ejmech.2015.10.025 |
| Homo sapiens |
Monoamine oxidase B |
IC50 |
17000.0 |
nM |
10.1016/j.ejmech.2009.02.031 |
| Homo sapiens |
Monoamine oxidase B |
Inhibition |
31.41 |
% |
10.1016/j.bmcl.2013.01.033 |
| Homo sapiens |
Monoamine oxidase B |
Inhibition |
50.0 |
% |
10.1016/j.ejmech.2015.10.025 |
| Homo sapiens |
Motilin receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Multidrug resistance-associated protein 4 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Mu opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuronal acetylcholine receptor protein alpha-4 subunit |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
PBMC |
Activity |
16.0 |
% |
10.1128/aac.01190-06 |
| Homo sapiens |
PBMC |
Activity |
51.0 |
% |
10.1128/aac.01190-06 |
| Homo sapiens |
PBMC |
Activity |
59.0 |
% |
10.1128/aac.01190-06 |
| Homo sapiens |
PBMC |
Activity |
60.0 |
% |
10.1128/aac.01190-06 |
| Homo sapiens |
PBMC |
Activity |
82.0 |
% |
10.1128/aac.01190-06 |
| Homo sapiens |
PBMC |
Activity |
297.0 |
% |
10.1128/aac.01190-06 |
| Homo sapiens |
Phosphodiesterase 3A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 4D |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Plasma |
Cmax |
47428.49 |
nM |
10.1128/aac.01145-08 |
| Homo sapiens |
Plasma |
Fu |
0.31 |
None |
10.1128/aac.01145-08 |
| Homo sapiens |
Plasma |
Fu |
0.7 |
None |
10.1021/acs.jmedchem.5b00050 |
| Homo sapiens |
Plasma |
Fu |
0.71 |
None |
10.1021/jm501174m |
| Homo sapiens |
Plasma |
Stability |
100.0 |
% |
10.1021/acsmedchemlett.5b00213 |
| Homo sapiens |
Pregnane X receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Prelamin-A/C |
Potency |
35481.3 |
nM |
None |
| Homo sapiens |
Progesterone receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 1a (5-HT1a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 3a (5-HT3a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serum |
Drug uptake |
6.0 |
ug ml-1 |
10.1128/aac.00247-07 |
| Homo sapiens |
Serum |
PPB |
31.0 |
% |
10.1128/aac.00766-09 |
| Homo sapiens |
Sodium channel protein type V alpha subunit |
AC50 |
50000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Succinate dehydrogenase [ubiquinone] flavoprotein subunit, mitochondrial |
IC50 |
8190.0 |
nM |
10.1016/j.bmcl.2019.07.024 |
| Homo sapiens |
THP-1 |
Drug uptake |
10.0 |
% |
10.1128/aac.01723-09 |
| Homo sapiens |
THP-1 |
Drug uptake |
20.0 |
% |
10.1128/aac.01723-09 |
| Homo sapiens |
THP-1 |
Drug uptake |
25.0 |
% |
10.1128/aac.01723-09 |
| Homo sapiens |
Thromboxane A2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Type-1 angiotensin II receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Tyrosyl-DNA phosphodiesterase 1 |
Potency |
21136.0 |
nM |
None |
| Homo sapiens |
Tyrosyl-DNA phosphodiesterase 1 |
Potency |
33498.3 |
nM |
None |
| Homo sapiens |
Vasopressin V1a receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vasopressin V2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Voltage-gated L-type calcium channel |
IC50 |
105400.0 |
nM |
10.1038/srep02100 |
| Homo sapiens |
Voltage-gated L-type calcium channel alpha-1C subunit |
AC50 |
50000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Hoylesella loescheii |
Hoylesella loescheii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Hoylesella loescheii |
Hoylesella loescheii |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Hoylesella loescheii |
Hoylesella loescheii |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Hoylesella oralis |
Hoylesella oralis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Hoylesella oralis |
Hoylesella oralis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Hoylesella oralis |
Hoylesella oralis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
200000.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Activity |
nan |
None |
10.1016/j.bmcl.2008.10.045 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.ejmech.2009.11.009 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.bmcl.2004.07.064 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2010.10.015 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.024 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.096 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1007/s00044-012-0394-2 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.10.048 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1021/acs.jnatprod.9b00321 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm9509556 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1021/np800503z |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64.0 |
ug.mL-1 |
10.1039/d2md00260d |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111850 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
128.0 |
ug.mL-1 |
10.1021/jm070638m |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
4629.0 |
nM |
10.1016/j.bmcl.2009.04.133 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
10000.0 |
nM |
10.6019/CHEMBL4513141 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
64000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
100000.0 |
nM |
10.1016/j.bmcl.2004.08.059 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
200000.0 |
nM |
10.1016/j.ejmech.2022.114213 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
200000.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
nan |
None |
10.1016/j.ejmech.2018.06.023 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
nan |
None |
10.1021/acs.jmedchem.0c00295 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC100 |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC90 |
128.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Lactococcus lactis |
Lactococcus lactis |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Lactococcus lactis |
Lactococcus lactis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Lactococcus lactis |
Lactococcus lactis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Legionella pneumophila |
Legionella pneumophila |
Activity |
5.14 |
mg/L |
10.1128/aac.01724-09 |
| Legionella pneumophila |
Legionella pneumophila |
EC50 |
8.45 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Legionella pneumophila |
Legionella pneumophila |
log10cfu |
-1.2 |
None |
10.1128/aac.01724-09 |
| Legionella pneumophila |
Legionella pneumophila |
log10cfu |
0.78 |
None |
10.1128/aac.01724-09 |
| Legionella pneumophila |
Legionella pneumophila |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Legionella pneumophila |
Legionella pneumophila |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Legionella pneumophila |
Legionella pneumophila |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Legionella pneumophila |
Legionella pneumophila |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Legionella pneumophila |
Legionella pneumophila |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Leuconostoc |
Leuconostoc |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| Leuconostoc |
Leuconostoc |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| Listeria monocytogenes |
Listeria monocytogenes |
Activity |
5.47 |
mg/L |
10.1128/aac.01724-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
Activity |
nan |
None |
10.1128/aac.00845-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
EC50 |
0.62 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Listeria monocytogenes |
Listeria monocytogenes |
Inhibition |
0.7 |
% |
10.1128/aac.01496-06 |
| Listeria monocytogenes |
Listeria monocytogenes |
Inhibition |
29.2 |
% |
10.1128/aac.01496-06 |
| Listeria monocytogenes |
Listeria monocytogenes |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Listeria monocytogenes |
Listeria monocytogenes |
log10cfu |
-0.37 |
None |
10.1128/aac.01724-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
log10cfu |
3.19 |
None |
10.1128/aac.01724-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111830 |
| Listeria monocytogenes |
Listeria monocytogenes |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2020.112497 |
| Listeria monocytogenes |
Listeria monocytogenes |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2019.04.063 |
| Listeria monocytogenes |
Listeria monocytogenes |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111593 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.063 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.111593 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.111830 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2020.112497 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
0.5 |
ug.mL-1 |
10.1039/c9md00391f |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114550 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
2.0 |
ug.mL-1 |
10.1039/D1MD00211B |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC50 |
2000.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC90 |
2000.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| Mammaliicoccus lentus |
Mammaliicoccus lentus |
MIC |
1.563 |
ug.mL-1 |
10.1016/j.ejmech.2010.10.015 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
Activity |
96.0 |
% |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MBC |
0.5 |
ug ml-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MBC50 |
2.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MBC90 |
4.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC50 |
nan |
None |
10.1128/aac.00859-08 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Mammaliicoccus sciuri |
Mammaliicoccus sciuri |
MIC90 |
nan |
None |
10.1128/aac.00859-08 |
| Metamycoplasma hominis |
Metamycoplasma hominis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| Metamycoplasma hominis |
Metamycoplasma hominis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Metamycoplasma hominis |
Metamycoplasma hominis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Metamycoplasma hominis |
Metamycoplasma hominis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Metamycoplasma hominis |
Metamycoplasma hominis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| Metamycoplasma hominis |
Metamycoplasma hominis |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| Micrococcus |
Micrococcus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Micrococcus |
Micrococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Micrococcus |
Micrococcus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Micrococcus luteus |
Micrococcus luteus |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Micrococcus luteus |
Micrococcus luteus |
Inhibition |
3.4 |
% |
10.1128/aac.01496-06 |
| Micrococcus luteus |
Micrococcus luteus |
Inhibition |
75.9 |
% |
10.1128/aac.01496-06 |
| Micrococcus luteus |
Micrococcus luteus |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Micrococcus luteus |
Micrococcus luteus |
IZ |
20.0 |
mm |
10.1016/j.ejmech.2013.01.034 |
| Micrococcus luteus |
Micrococcus luteus |
IZ |
20.0 |
mm |
10.1016/j.ejmech.2013.03.027 |
| Micrococcus luteus |
Micrococcus luteus |
IZ |
38.0 |
mm |
10.1016/j.bmcl.2009.10.018 |
| Micrococcus luteus |
Micrococcus luteus |
IZ |
38.0 |
mm |
10.1039/c0md00015a |
| Micrococcus luteus |
Micrococcus luteus |
IZ |
45.0 |
mm |
10.1039/c0md00015a |
| Micrococcus luteus |
Micrococcus luteus |
MIC |
0.781 |
ug.mL-1 |
10.1016/j.ejmech.2010.10.015 |
| Micrococcus luteus |
Micrococcus luteus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.01.034 |
| Micrococcus luteus |
Micrococcus luteus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.027 |
| Micrococcus luteus |
Micrococcus luteus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Micrococcus luteus |
Micrococcus luteus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm201467r |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
4.0 |
ug.mL-1 |
10.1007/s00044-012-0394-2 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.022 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.056 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.03.043 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
4.0 |
ug.mL-1 |
10.1016/s0960-894x(02)00352-9 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm058204j |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
4.0 |
ug.mL-1 |
10.1021/np800503z |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
4.0 |
ug.mL-1 |
10.1039/d2md00260d |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.017 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.018 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.029 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.11.093 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.01.109 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.03.104 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.07.064 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.056 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.085 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.005 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.07.006 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.03.024 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.003 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.05.041 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.08.002 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm020248u |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm980546k |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm990373e |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1021/ml400280z |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC |
8000000.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.021 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
8.0 |
ug.mL-1 |
10.1021/jm1014023 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
8.0 |
ug.mL-1 |
10.1021/jm201467r |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
4.0 |
ug.mL-1 |
10.1021/jm960294s |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.023 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
8.0 |
ug.mL-1 |
10.1021/jm201467r |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
16.0 |
ug.mL-1 |
10.1021/jm1014023 |
| Moraxella catarrhalis |
Moraxella catarrhalis |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Mus musculus |
Brain |
AUC |
0.9 |
ug.hr/g |
10.1021/acsmedchemlett.5b00213 |
| Mus musculus |
Brain |
AUCt |
0.83 |
ug.hr/g |
10.1021/acsmedchemlett.5b00213 |
| Mus musculus |
Brain |
Cmax |
0.45 |
ug/g |
10.1021/acsmedchemlett.5b00213 |
| Mus musculus |
Mus musculus |
Activity |
0.05 |
None |
10.1016/j.bmcl.2003.07.033 |
| Mus musculus |
Mus musculus |
Activity |
1.4 |
None |
10.1016/j.bmcl.2003.07.033 |
| Mus musculus |
Mus musculus |
Activity |
nan |
None |
10.1016/j.ejmech.2018.09.053 |
| Mus musculus |
Mus musculus |
AUC |
780.0 |
ng.hr.mL-1 |
10.1128/aac.01567-06 |
| Mus musculus |
Mus musculus |
AUC |
2100.0 |
ng.hr.mL-1 |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
AUC |
10980.0 |
ng.hr.mL-1 |
10.1016/j.bmcl.2008.03.043 |
| Mus musculus |
Mus musculus |
AUC |
16000.0 |
ng.hr.mL-1 |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
AUC |
19000.0 |
ng.hr.mL-1 |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
AUC |
29090.0 |
ng.hr.mL-1 |
10.1128/aac.01315-06 |
| Mus musculus |
Mus musculus |
AUC |
112020.0 |
ng.hr.mL-1 |
10.1128/aac.01315-06 |
| Mus musculus |
Mus musculus |
AUC |
161850.0 |
ng.hr.mL-1 |
10.1021/ml400280z |
| Mus musculus |
Mus musculus |
AUC |
45700000000.0 |
ng.hr.mL-1 |
10.1021/jm070428+ |
| Mus musculus |
Mus musculus |
AUC |
105000000000.0 |
ng.hr.mL-1 |
10.1021/jm070428+ |
| Mus musculus |
Mus musculus |
CFU |
75.0 |
% |
10.1016/j.bmcl.2006.10.063 |
| Mus musculus |
Mus musculus |
CL |
15.67 |
mL.min-1.kg-1 |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
CL/F |
8.667 |
mL.min-1.kg-1 |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
CL/F |
10.67 |
mL.min-1.kg-1 |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
Cmax |
9782.13 |
nM |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
Cmax |
18704.61 |
nM |
10.1016/j.bmcl.2008.03.043 |
| Mus musculus |
Mus musculus |
Cmax |
26382.1 |
nM |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
Cmax |
32607.08 |
nM |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
Cmax |
36134.58 |
nM |
10.1128/aac.01315-06 |
| Mus musculus |
Mus musculus |
Cmax |
75648.44 |
nM |
10.1128/aac.01315-06 |
| Mus musculus |
Mus musculus |
Cmax |
109678.38 |
nM |
10.1021/ml400280z |
| Mus musculus |
Mus musculus |
Cmax |
148214.02 |
nM |
10.1128/aac.00148-08 |
| Mus musculus |
Mus musculus |
ED50 |
1.14 |
mg.kg-1 |
10.1021/jm050035f |
| Mus musculus |
Mus musculus |
ED50 |
2.0 |
mg.kg-1 |
10.1016/s0960-894x(98)00194-2 |
| Mus musculus |
Mus musculus |
ED50 |
2.0 |
mg.kg-1 |
10.1021/jm9509556 |
| Mus musculus |
Mus musculus |
ED50 |
2.4 |
mg.kg-1 |
10.1021/jm050035f |
| Mus musculus |
Mus musculus |
ED50 |
3.1 |
mg.kg-1 |
10.1021/jm050035f |
| Mus musculus |
Mus musculus |
ED50 |
3.9 |
mg.kg-1 |
10.1021/jm980274l |
| Mus musculus |
Mus musculus |
ED50 |
3.9 |
mg kg-1 day-1 |
10.1021/jm990373e |
| Mus musculus |
Mus musculus |
ED50 |
3.91 |
mg.kg-1 |
10.1021/jm020092y |
| Mus musculus |
Mus musculus |
ED50 |
5.0 |
mg.kg-1 |
10.1016/j.bmcl.2003.07.022 |
| Mus musculus |
Mus musculus |
ED50 |
5.6 |
mg.kg-1 |
10.1016/j.bmcl.2003.07.029 |
| Mus musculus |
Mus musculus |
ED50 |
5.6 |
mg.kg-1 |
10.1021/jm9509556 |
| Mus musculus |
Mus musculus |
ED50 |
5.6 |
mg.kg-1 |
10.1021/jm980274l |
| Mus musculus |
Mus musculus |
ED50 |
5.6 |
mg kg-1 day-1 |
10.1016/j.bmcl.2003.07.017 |
| Mus musculus |
Mus musculus |
ED50 |
5.6 |
mg kg-1 day-1 |
10.1021/jm990373e |
| Mus musculus |
Mus musculus |
ED50 |
6.8 |
mg kg-1 day-1 |
10.1016/j.bmcl.2004.04.037 |
| Mus musculus |
Mus musculus |
ED50 |
8.0 |
mg kg-1 day-1 |
10.1016/j.bmcl.2003.08.031 |
| Mus musculus |
Mus musculus |
ED50 |
10.0 |
mg.kg-1 |
10.1021/jm9509556 |
| Mus musculus |
Mus musculus |
ED50 |
24.0 |
mg.kg-1 |
10.1021/jm9509556 |
| Mus musculus |
Mus musculus |
F |
100.0 |
% |
10.1128/aac.01567-06 |
| Mus musculus |
Mus musculus |
fAUC |
1400.0 |
ng.hr.mL-1 |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
fAUC |
11000.0 |
ng.hr.mL-1 |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
fAUC |
13000.0 |
ng.hr.mL-1 |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
fCmax |
2.3 |
ug ml-1 |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
fCmax |
6.0 |
ug ml-1 |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
fCmax |
7.1 |
ug ml-1 |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
Kel |
0.51 |
/hr |
10.1016/j.bmcl.2008.03.043 |
| Mus musculus |
Mus musculus |
MIC |
1.2 |
ug.mL-1 |
10.1016/s0960-894x(00)00304-8 |
| Mus musculus |
Mus musculus |
MIC |
2.5 |
ug.mL-1 |
10.1016/s0960-894x(00)00304-8 |
| Mus musculus |
Mus musculus |
PD50 |
1.8 |
mg kg-1 |
10.1016/s0960-894x(00)00304-8 |
| Mus musculus |
Mus musculus |
PD50 |
2.1 |
mg kg-1 |
10.1016/s0960-894x(00)00304-8 |
| Mus musculus |
Mus musculus |
PD50 |
2.4 |
mg kg-1 |
10.1016/s0960-894x(00)00304-8 |
| Mus musculus |
Mus musculus |
PD50 |
3.0 |
mg kg-1 |
10.1016/s0960-894x(00)00304-8 |
| Mus musculus |
Mus musculus |
PD50 |
4.2 |
mg kg-1 |
10.1016/s0960-894x(00)00304-8 |
| Mus musculus |
Mus musculus |
PD50 |
5.8 |
mg kg-1 |
10.1016/s0960-894x(00)00304-8 |
| Mus musculus |
Mus musculus |
PD50 |
6.0 |
mg/kg/day |
10.1016/j.bmcl.2005.04.003 |
| Mus musculus |
Mus musculus |
PD50 |
8.6 |
mg kg-1 |
10.1016/s0960-894x(00)00304-8 |
| Mus musculus |
Mus musculus |
PD50 |
8.7 |
mg kg-1 |
10.1016/s0960-894x(00)00304-8 |
| Mus musculus |
Mus musculus |
T1/2 |
0.5 |
hr |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
T1/2 |
0.8 |
hr |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
T1/2 |
1.0 |
hr |
10.1021/acsmedchemlett.7b00068 |
| Mus musculus |
Mus musculus |
T1/2 |
1.17 |
hr |
10.1128/aac.01315-06 |
| Mus musculus |
Mus musculus |
T1/2 |
1.37 |
hr |
10.1016/j.bmcl.2008.03.043 |
| Mus musculus |
Mus musculus |
T1/2 |
1.4 |
hr |
10.1128/aac.00833-08 |
| Mus musculus |
Mus musculus |
T1/2 |
2.18 |
hr |
10.1128/aac.01315-06 |
| Mus musculus |
Mus musculus |
Tmax |
0.25 |
hr |
10.1016/j.bmcl.2008.03.043 |
| Mus musculus |
Mus musculus |
Tmax |
0.5 |
hr |
10.1021/ml400280z |
| Mus musculus |
Mus musculus |
Tmax |
0.5 |
hr |
10.1128/aac.01315-06 |
| Mus musculus |
Mus musculus |
Tmax |
1.0 |
hr |
10.1128/aac.01315-06 |
| Mus musculus |
Plasma |
AUC |
7580.0 |
ng.hr.mL-1 |
10.1021/acsmedchemlett.5b00213 |
| Mus musculus |
Plasma |
AUC |
7700.0 |
ng.hr.mL-1 |
10.1021/acsmedchemlett.5b00213 |
| Mus musculus |
Plasma |
Cmax |
10819.62 |
nM |
10.1021/acsmedchemlett.5b00213 |
| Mus musculus |
Plasma |
Cp |
nan |
None |
10.1021/acs.jmedchem.6b00372 |
| Mus musculus |
Plasma |
fAUC |
29916.67 |
ng.hr.mL-1 |
10.1128/aac.00642-09 |
| Mus musculus |
Plasma |
fCmax |
14.0 |
ug ml-1 |
10.1128/aac.00642-09 |
| Mus musculus |
Plasma |
PPB |
32.0 |
% |
10.1128/aac.00642-09 |
| Mus musculus |
Plasma |
PPB |
68.0 |
% |
10.1128/aac.01567-06 |
| Mus musculus |
Plasma |
T1/2 |
1.7 |
hr |
10.1128/aac.00642-09 |
| Mus musculus |
Plasma |
Tmax |
0.5 |
hr |
10.1128/aac.00642-09 |
| Mus musculus |
Serum |
Tmax |
0.13 |
hr |
10.1128/aac.00833-08 |
| Mycobacterium avium |
Mycobacterium avium |
MIC90 |
nan |
None |
10.1016/j.bmcl.2016.06.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
0.5 |
log10CFU/ml |
10.1016/j.bmc.2016.08.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.7 |
log10CFU/ml |
10.1016/j.bmc.2016.08.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.4 |
log10CFU |
10.1021/acs.jmedchem.2c00227 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
3.0 |
log10CFU |
10.1021/acs.jmedchem.2c00227 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
3.0 |
log10CFU/ml |
10.1016/j.bmc.2016.08.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
3.9 |
log10CFU |
10.1021/acs.jmedchem.7b00631 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
4.136 |
log10CFU |
10.1021/acs.jmedchem.0c00500 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acs.jmedchem.0c00500 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
ED99 |
28.0 |
mg kg-1 |
10.1128/aac.01423-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Emax |
300.0 |
mg kg-1 |
10.1128/aac.01423-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.71 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.8 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
84.02 |
% |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.52 |
% |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
96.58 |
% |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
1.61 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2012.02.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1021/jm9509556 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1039/C9MD00057G |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00414-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.23 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00500 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2014.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.3 |
ug.mL-1 |
10.1016/j.bmcl.2015.12.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.32 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00500 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2017.06.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00414-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01378-08 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.63 |
ug.mL-1 |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.88 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.10.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.08.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.06.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1039/C9MD00057G |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01189-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01378-08 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.25 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.31 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.68 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.91 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2010.12.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.33 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.65 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.92 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00500 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00414-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01189-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.34 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
14.08 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
14.54 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01189-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01189-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01189-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.bmc.2012.04.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1021/acs.jnatprod.2c01003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1500.0 |
nM |
10.1021/acs.jmedchem.2c00227 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1560.0 |
nM |
10.1039/C6MD00236F |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1700.0 |
nM |
10.1021/acs.jnatprod.2c01003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1860.0 |
nM |
10.1016/j.bmcl.2017.01.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1900.0 |
nM |
10.1128/aac.00055-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2300.0 |
nM |
10.1039/C6MD00236F |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2780.0 |
nM |
10.1016/j.bmcl.2017.01.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2800.0 |
nM |
10.1021/acsmedchemlett.7b00356 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2900.0 |
nM |
10.1021/acsmedchemlett.7b00356 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3700.0 |
nM |
10.1016/j.bmcl.2017.01.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6300.0 |
nM |
10.1128/aac.00055-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
65200.0 |
nM |
10.1128/aac.00055-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128000.0 |
nM |
10.1128/aac.00055-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1016/j.bmc.2012.04.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1016/j.bmcl.2014.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC100 |
0.6 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00414-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b02075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.304 |
ug ml-1 |
10.1021/acsmedchemlett.7b00068 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.953 |
ug ml-1 |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
1.254 |
ug ml-1 |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
1.87 |
ug ml-1 |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.9b02075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00414-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
5.98 |
ug.mL-1 |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
700.0 |
nM |
10.1016/j.ejmech.2022.114201 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
800.0 |
nM |
10.1016/j.ejmech.2022.114201 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
900.0 |
nM |
10.1016/j.ejmech.2022.114201 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1900.0 |
nM |
10.1016/j.ejmech.2022.114201 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
1.0 |
None |
10.1021/jm500833f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Selectivity ratio |
1.05 |
None |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
IC50 |
0.029 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
IC50 |
0.31 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
Inhibition |
100.59 |
% |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
Inhibition |
101.14 |
% |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
Inhibition |
101.46 |
% |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.42 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.43 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00400-10 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00400-10 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00400-10 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC90 |
nan |
None |
10.1016/j.bmcl.2016.06.019 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00590-09 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
5.0 |
ug.mL-1 |
10.1128/aac.00590-09 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
25.0 |
ug.mL-1 |
10.1128/aac.00590-09 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
100.0 |
ug.mL-1 |
10.1128/aac.00590-09 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MBC |
0.8 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00644-10 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.10.073 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00644-10 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128531 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00644-10 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01189-07 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00644-10 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00644-10 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00644-10 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00644-10 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC100 |
0.2 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Mycolicibacterium vaccae |
Mycolicibacterium vaccae |
IZ |
42.0 |
mm |
10.1016/j.bmcl.2009.10.018 |
| Mycolicibacterium vaccae |
Mycolicibacterium vaccae |
IZ |
52.0 |
mm |
10.1039/c0md00015a |
| Mycoplasmoides pneumoniae |
Mycoplasmoides pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| Mycoplasmoides pneumoniae |
Mycoplasmoides pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Mycoplasmoides pneumoniae |
Mycoplasmoides pneumoniae |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Mycoplasmoides pneumoniae |
Mycoplasmoides pneumoniae |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| Mycoplasmoides pneumoniae |
Mycoplasmoides pneumoniae |
MIC50 |
64.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Mycoplasmoides pneumoniae |
Mycoplasmoides pneumoniae |
MIC90 |
64.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Mycoplasmoides pneumoniae |
Mycoplasmoides pneumoniae |
MIC90 |
128.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| Neisseria meningitidis |
Neisseria meningitidis |
MIC |
8.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00213 |
| Nocardia asteroides |
Nocardia asteroides |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| Nocardia asteroides |
Nocardia asteroides |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| Nocardia brasiliensis |
Nocardia brasiliensis |
Activity |
nan |
None |
10.1128/aac.00148-08 |
| Nocardia brasiliensis |
Nocardia brasiliensis |
MIC |
0.001 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia brasiliensis |
Nocardia brasiliensis |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00148-08 |
| Nocardia brasiliensis |
Nocardia brasiliensis |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| Nocardia brasiliensis |
Nocardia brasiliensis |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| Nocardia carnea |
Nocardia carnea |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia cyriacigeorgica |
Nocardia cyriacigeorgica |
MIC |
0.00012 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia farcinica |
Nocardia farcinica |
MIC |
0.00012 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia nova |
Nocardia nova |
MIC |
0.00012 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia otitidiscaviarum |
Nocardia otitidiscaviarum |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia sp. |
Nocardia sp. |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Nocardia sp. |
Nocardia sp. |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| Nocardia sp. |
Nocardia sp. |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| Nocardia transvalensis |
Nocardia transvalensis |
MIC |
0.001 |
ug.mL-1 |
10.1128/aac.01102-06 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Activity |
2.35 |
Kg |
10.1128/aac.00638-07 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Activity |
2.36 |
Kg |
10.1128/aac.00638-07 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Activity |
2.42 |
Kg |
10.1128/aac.00638-07 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Activity |
2.44 |
Kg |
10.1128/aac.00638-07 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Activity |
nan |
None |
10.1128/aac.00638-07 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
AUC |
76300.0 |
ng.hr.mL-1 |
10.1128/aac.01242-06 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
AUC |
136900.0 |
ng.hr.mL-1 |
10.1128/aac.01242-06 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
AUC |
173000.0 |
ng.hr.mL-1 |
10.1128/aac.00638-07 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
AUC |
334000.0 |
ng.hr.mL-1 |
10.1128/aac.00638-07 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
CFU |
0.18 |
10'7/g |
10.1128/aac.00638-07 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
CFU |
2.02 |
10'9/g |
10.1128/aac.00638-07 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Cmax |
35274.94 |
nM |
10.1128/aac.01242-06 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Cmax |
58099.9 |
nM |
10.1128/aac.01242-06 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Cmax |
80628.43 |
nM |
10.1128/aac.00638-07 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Cmin |
17.0 |
ug ml-1 |
10.1128/aac.00638-07 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
Cp |
28.2 |
ug ml-1 |
10.1128/aac.00886-09 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
T1/2 |
2.7 |
hr |
10.1128/aac.01242-06 |
| Oryctolagus cuniculus |
Oryctolagus cuniculus |
T1/2 |
3.3 |
hr |
10.1128/aac.01242-06 |
| Paeniclostridium sordellii |
Paeniclostridium sordellii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Paeniclostridium sordellii |
Paeniclostridium sordellii |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Paeniclostridium sordellii |
Paeniclostridium sordellii |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Parabacteroides distasonis |
Parabacteroides distasonis |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Parabacteroides merdae |
Parabacteroides merdae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Parabacteroides merdae |
Parabacteroides merdae |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Parabacteroides merdae |
Parabacteroides merdae |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Paraclostridium bifermentans |
Paraclostridium bifermentans |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Paraclostridium bifermentans |
Paraclostridium bifermentans |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Paraclostridium bifermentans |
Paraclostridium bifermentans |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Parvimonas micra |
Parvimonas micra |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Parvimonas micra |
Parvimonas micra |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Parvimonas micra |
Parvimonas micra |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Parvimonas micra |
Parvimonas micra |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Parvimonas micra |
Parvimonas micra |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Parvimonas micra |
Parvimonas micra |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Parvimonas micra |
Parvimonas micra |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Parvimonas micra |
Parvimonas micra |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Parvimonas micra |
Parvimonas micra |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Parvimonas micra |
Parvimonas micra |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Pasteurella multocida |
Pasteurella multocida |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Pasteurella multocida |
Pasteurella multocida |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Pasteurella multocida |
Pasteurella multocida |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Peptoniphilus asaccharolyticus |
Peptoniphilus asaccharolyticus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Peptostreptococcus anaerobius |
Peptostreptococcus anaerobius |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Peptostreptococcus sp. |
Peptostreptococcus sp. |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Peptostreptococcus sp. |
Peptostreptococcus sp. |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Peptostreptococcus sp. |
Peptostreptococcus sp. |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Peptostreptococcus sp. |
Peptostreptococcus sp. |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Phocaeicola vulgatus |
Phocaeicola vulgatus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Plasmodium falciparum |
Plasmodium falciparum |
Activity |
nan |
None |
10.1128/aac.00892-07 |
| Porphyromonas asaccharolytica |
Porphyromonas asaccharolytica |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Porphyromonas asaccharolytica |
Porphyromonas asaccharolytica |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Porphyromonas asaccharolytica |
Porphyromonas asaccharolytica |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Prescottella equi |
Prescottella equi |
MBC50 |
8.0 |
mg/L |
10.1128/aac.00344-06 |
| Prescottella equi |
Prescottella equi |
MBC90 |
16.0 |
mg/L |
10.1128/aac.00344-06 |
| Prescottella equi |
Prescottella equi |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00344-06 |
| Prescottella equi |
Prescottella equi |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00344-06 |
| Prevotella bivia |
Prevotella bivia |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella bivia |
Prevotella bivia |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella bivia |
Prevotella bivia |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella buccae |
Prevotella buccae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella buccae |
Prevotella buccae |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella buccae |
Prevotella buccae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella corporis |
Prevotella corporis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella corporis |
Prevotella corporis |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella corporis |
Prevotella corporis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella denticola |
Prevotella denticola |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella denticola |
Prevotella denticola |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella denticola |
Prevotella denticola |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella disiens |
Prevotella disiens |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella disiens |
Prevotella disiens |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella disiens |
Prevotella disiens |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella intermedia |
Prevotella intermedia |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella intermedia |
Prevotella intermedia |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella intermedia |
Prevotella intermedia |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella melaninogenica |
Prevotella melaninogenica |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella nigrescens |
Prevotella nigrescens |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella nigrescens |
Prevotella nigrescens |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Prevotella nigrescens |
Prevotella nigrescens |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Priestia megaterium |
Priestia megaterium |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.017 |
| Propionibacterium |
Propionibacterium |
Activity |
0.0 |
% |
10.1128/aac.00696-08 |
| Propionibacterium |
Propionibacterium |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Propionibacterium |
Propionibacterium |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Propionibacterium |
Propionibacterium |
MIC90 |
0.5 |
ug.mL-1 |
10.1128/aac.00696-08 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
128.0 |
ug.mL-1 |
10.1021/jm070638m |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
25000.0 |
nM |
10.1016/j.bmcl.2004.08.059 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Activity |
nan |
None |
10.1016/j.bmcl.2008.10.045 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IC50 |
0.49 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IC50 |
1700.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IC50 |
15930.0 |
nM |
10.1016/j.bmcl.2014.12.063 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IC50 |
19800.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IC50 |
24700.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IC50 |
100000.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Inhibition |
99.01 |
% |
10.1016/j.ejmech.2016.07.001 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Inhibition |
99.22 |
% |
10.1016/j.ejmech.2016.07.001 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Inhibition |
99.9 |
% |
10.1016/j.ejmech.2016.07.001 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
0.0 |
mm |
10.1016/j.bmcl.2009.10.018 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
0.0 |
mm |
10.1039/c0md00015a |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
8.5 |
mm |
10.1016/j.ejmech.2011.04.041 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
10.0 |
mm |
10.1016/j.bmcl.2009.10.018 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
10.0 |
mm |
10.1039/c0md00015a |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IZ |
12.0 |
mm |
10.1016/j.ejmech.2013.01.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1.31 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2.5 |
ug.mL-1 |
10.1016/j.bmcl.2014.12.063 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.017 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.096 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.04.045 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.03.028 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2011.10.041 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
32.0 |
ug.mL-1 |
10.1039/C5MD00101C |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.04.086 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2019.06.010 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115729 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.10.048 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.053 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113480 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113723 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm9509556 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1021/np800503z |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64.0 |
ug.mL-1 |
10.1039/d2md00260d |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.09.019 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2010.10.015 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.04.041 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111850 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
128.0 |
ug.mL-1 |
10.1021/jm070638m |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
10000.0 |
nM |
10.6019/CHEMBL4513141 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
12500.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
50000.0 |
nM |
10.1016/j.ejmech.2022.114333 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
64000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
100000.0 |
nM |
10.1016/j.bmcl.2004.08.059 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
200000.0 |
nM |
10.1016/j.ejmech.2022.114213 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
200000.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
1024000.0 |
nM |
10.1016/j.bmcl.2023.129282 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1016/j.ejmech.2018.06.023 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1128/aac.00642-09 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
128.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC99 |
32.0 |
ug ml-1 |
10.1016/j.bmcl.2014.02.025 |
| Raoultella planticola |
Raoultella planticola |
IZ |
nan |
None |
10.1016/j.ejmech.2013.01.034 |
| Rattus norvegicus |
Androgen Receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Cyclooxygenase-1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
GABA receptor alpha-1 subunit |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Glutamate (NMDA) receptor subunit zeta 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
H9c2 |
IC50 |
8710.0 |
nM |
10.1021/acsmedchemlett.7b00068 |
| Rattus norvegicus |
Liver microsome |
Stability |
88.3 |
% |
10.1021/acsmedchemlett.5b00213 |
| Rattus norvegicus |
Monoamine oxidase A |
Inhibition |
61.3 |
% |
10.1016/j.ejmech.2013.03.003 |
| Rattus norvegicus |
Monoamine oxidase A |
Inhibition |
61.3 |
% |
10.1021/ml400280z |
| Rattus norvegicus |
Monoamine oxidase B |
IC50 |
17000.0 |
nM |
10.1016/s0960-894x(02)00352-9 |
| Rattus norvegicus |
Monoamine oxidase B |
Inhibition |
70.4 |
% |
10.1016/j.ejmech.2013.03.003 |
| Rattus norvegicus |
Monoamine oxidase B |
Inhibition |
70.4 |
% |
10.1021/ml400280z |
| Rattus norvegicus |
Plasma |
Cp |
7.3 |
ug ml-1 |
10.1021/jm800038g |
| Rattus norvegicus |
Plasma |
Cp |
17.0 |
ug ml-1 |
10.1021/jm800038g |
| Rattus norvegicus |
Plasma |
Fu |
0.69 |
None |
10.1021/jm901371v |
| Rattus norvegicus |
Plasma |
PPB |
31.0 |
% |
10.1021/jm800038g |
| Rattus norvegicus |
Plasma |
Stability |
100.0 |
% |
10.1021/acsmedchemlett.5b00213 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
1.64 |
% |
10.1021/jm401931e |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
1.9 |
10'9/L |
10.1021/jm401931e |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
5.52 |
10'12/L |
10.1021/jm401931e |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
9.0 |
% |
10.1021/jm070708p |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
13.0 |
% |
10.1021/jm401931e |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
20.52 |
pg |
10.1021/jm401931e |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
30.18 |
% |
10.1021/jm401931e |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
54.74 |
fL |
10.1021/jm401931e |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
86.2 |
% |
10.1021/jm401931e |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
97.0 |
% |
10.1021/jm070708p |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
112.8 |
g/L |
10.1021/jm401931e |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
487.4 |
10'9/L |
10.1021/jm401931e |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
nan |
None |
10.1021/jm070708p |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
nan |
None |
10.1021/jm800038g |
| Rattus norvegicus |
Rattus norvegicus |
AUC |
4240.0 |
ng.hr.mL-1 |
10.1016/s0960-894x(03)00249-x |
| Rattus norvegicus |
Rattus norvegicus |
AUC |
15500.0 |
ng.hr.mL-1 |
10.1016/j.bmc.2012.08.023 |
| Rattus norvegicus |
Rattus norvegicus |
AUC |
105000.0 |
ng.hr.mL-1 |
10.1021/jm070708p |
| Rattus norvegicus |
Rattus norvegicus |
AUC |
666000.0 |
ng.hr.mL-1 |
10.1021/jm070708p |
| Rattus norvegicus |
Rattus norvegicus |
AUC/dose |
1.1 |
microg.hr/mL |
10.1016/j.bmcl.2014.03.022 |
| Rattus norvegicus |
Rattus norvegicus |
CL |
10.5 |
mL.min-1.kg-1 |
10.1016/j.bmc.2012.08.023 |
| Rattus norvegicus |
Rattus norvegicus |
CL |
10.5 |
mL.min-1.kg-1 |
10.1016/j.bmcl.2003.07.029 |
| Rattus norvegicus |
Rattus norvegicus |
CL |
10.5 |
mL.min-1.kg-1 |
10.1021/jm020248u |
| Rattus norvegicus |
Rattus norvegicus |
CL |
14.5 |
mL.min-1.kg-1 |
10.1016/j.bmcl.2014.03.022 |
| Rattus norvegicus |
Rattus norvegicus |
CL |
nan |
None |
10.1021/jm020248u |
| Rattus norvegicus |
Rattus norvegicus |
CL/F |
10.5 |
mL.min-1.kg-1 |
10.1021/jm980546k |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
4117.39 |
nM |
10.1016/s0960-894x(03)00249-x |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
15800.0 |
nM |
10.1021/jm980546k |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
44464.21 |
nM |
10.1016/j.bmc.2012.08.023 |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
46835.63 |
nM |
10.1016/j.bmcl.2003.07.029 |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
46835.63 |
nM |
10.1016/j.ejmech.2007.05.003 |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
46835.63 |
nM |
10.1021/jm020248u |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
51874.91 |
nM |
10.1128/aac.00744-06 |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
55135.62 |
nM |
10.1128/aac.00744-06 |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
57210.61 |
nM |
10.1128/aac.00744-06 |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
nan |
None |
10.1021/jm020248u |
| Rattus norvegicus |
Rattus norvegicus |
Cmin |
3.81 |
mg/L |
10.1128/aac.00744-06 |
| Rattus norvegicus |
Rattus norvegicus |
Cmin |
4.57 |
mg/L |
10.1128/aac.00744-06 |
| Rattus norvegicus |
Rattus norvegicus |
Cmin |
5.93 |
mg/L |
10.1128/aac.00744-06 |
| Rattus norvegicus |
Rattus norvegicus |
F |
100.0 |
% |
10.1016/j.ejmech.2007.05.003 |
| Rattus norvegicus |
Rattus norvegicus |
F |
109.0 |
% |
10.1016/j.bmc.2012.08.023 |
| Rattus norvegicus |
Rattus norvegicus |
F |
109.0 |
% |
10.1016/j.bmcl.2003.07.029 |
| Rattus norvegicus |
Rattus norvegicus |
F |
109.0 |
% |
10.1021/jm800038g |
| Rattus norvegicus |
Rattus norvegicus |
IC50 |
12000.0 |
nM |
10.1016/s0960-894x(02)00352-9 |
| Rattus norvegicus |
Rattus norvegicus |
PD50 |
4.07 |
mg kg-1 |
10.1016/s0960-894x(03)00249-x |
| Rattus norvegicus |
Rattus norvegicus |
Ratio |
8.4 |
None |
10.1021/jm070708p |
| Rattus norvegicus |
Rattus norvegicus |
Remaining at 40 min |
97.0 |
% |
10.1021/jm020248u |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
0.7 |
hr |
10.1016/j.bmcl.2014.03.022 |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
0.95 |
hr |
10.1016/j.bmcl.2003.07.029 |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
0.95 |
hr |
10.1016/j.ejmech.2007.05.003 |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
0.95 |
hr |
10.1021/jm020248u |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
0.95 |
hr |
10.1021/jm980546k |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
1.0 |
hr |
10.1016/j.bmc.2012.08.023 |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
1.05 |
hr |
10.1016/j.bmcl.2003.07.029 |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
1.05 |
hr |
10.1016/j.ejmech.2007.05.003 |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
1.05 |
hr |
10.1021/jm020248u |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
1.05 |
hr |
10.1021/jm980546k |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
3.093 |
hr |
10.1016/s0960-894x(03)00249-x |
| Rattus norvegicus |
Rattus norvegicus |
T max |
nan |
None |
10.1021/jm020248u |
| Rattus norvegicus |
Rattus norvegicus |
Tmax |
0.0 |
hr |
10.1016/j.ejmech.2007.05.003 |
| Rattus norvegicus |
Rattus norvegicus |
Tmax |
0.3 |
hr |
10.1016/j.bmcl.2003.07.029 |
| Rattus norvegicus |
Rattus norvegicus |
Tmax |
0.3 |
hr |
10.1021/jm980546k |
| Rattus norvegicus |
Rattus norvegicus |
Tmax |
0.31 |
hr |
10.1016/j.ejmech.2007.05.003 |
| Rattus norvegicus |
Rattus norvegicus |
Tmax |
0.31 |
hr |
10.1021/jm020248u |
| Rattus norvegicus |
Rattus norvegicus |
Tmax |
0.333 |
hr |
10.1016/s0960-894x(03)00249-x |
| Rattus norvegicus |
Rattus norvegicus |
Tmax |
1.0 |
hr |
10.1128/aac.00744-06 |
| Rattus norvegicus |
Rattus norvegicus |
T>MIC |
12.0 |
hr |
10.1128/aac.00744-06 |
| Rattus norvegicus |
Rattus norvegicus |
T>MIC |
24.0 |
hr |
10.1128/aac.00744-06 |
| Rattus norvegicus |
Rattus norvegicus |
T>MIC |
48.0 |
hr |
10.1128/aac.00744-06 |
| Rattus norvegicus |
Rattus norvegicus |
Vd |
0.72 |
L.kg-1 |
10.1016/j.bmc.2012.08.023 |
| Rattus norvegicus |
Rattus norvegicus |
Vd |
nan |
None |
10.1021/jm020248u |
| Rattus norvegicus |
Rattus norvegicus |
Vdss |
0.72 |
L.kg-1 |
10.1016/j.bmcl.2003.07.029 |
| Rattus norvegicus |
Rattus norvegicus |
Vdss |
0.72 |
L.kg-1 |
10.1021/jm020248u |
| Rattus norvegicus |
Rattus norvegicus |
Vdss |
0.72 |
L.kg-1 |
10.1021/jm980546k |
| Rattus norvegicus |
Rattus norvegicus |
Vdss |
1.0 |
L.kg-1 |
10.1016/j.bmcl.2014.03.022 |
| Rhodococcus sp. |
Rhodococcus sp. |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| Rhodococcus sp. |
Rhodococcus sp. |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| Ruminococcus sp. |
Ruminococcus sp. |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Ruminococcus sp. |
Ruminococcus sp. |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Ruminococcus sp. |
Ruminococcus sp. |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Salmonella enterica |
Salmonella enterica |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Salmonella enterica subsp. enterica serovar Abony |
Salmonella enterica subsp. enterica serovar Abony |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.096 |
| Salmonella enterica subsp. enterica serovar Abony |
Salmonella enterica subsp. enterica serovar Abony |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.04.045 |
| Salmonella enterica subsp. enterica serovar Typhi |
Salmonella typhi |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.11.019 |
| Salmonella enterica subsp. enterica serovar Typhi |
Salmonella typhi |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.096 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.09.019 |
| Salmonella enterica subsp. enterica serovar Typhi str. CT18 |
Salmonella enterica subsp. enterica serovar Typhi str. CT18 |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.03.028 |
| Serratia marcescens |
Serratia marcescens |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.096 |
| Serratia marcescens |
Serratia marcescens |
MIC |
64.0 |
ug.mL-1 |
10.1021/np800503z |
| Serratia marcescens |
Serratia marcescens |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.02.002 |
| Severe acute respiratory syndrome coronavirus 2 |
Replicase polyprotein 1ab |
Inhibition |
6.413 |
% |
10.6019/CHEMBL4495564 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Hit score |
0.0228 |
None |
10.1101/2020.04.21.054387 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
19952.62 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
20000.0 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
0.38 |
% |
10.6019/CHEMBL4495565 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
18.98 |
% |
10.21203/rs.3.rs-23951/v1 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition index |
0.04947 |
None |
10.1101/2020.04.03.023846 |
| Staphylococcus |
Staphylococcus |
Activity |
0.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus |
Staphylococcus |
Activity |
99.5 |
% |
10.1128/aac.01453-08 |
| Staphylococcus |
Staphylococcus |
Activity |
99.9 |
% |
10.1128/aac.01453-08 |
| Staphylococcus |
Staphylococcus |
Activity |
100.0 |
% |
10.1128/aac.00845-09 |
| Staphylococcus |
Staphylococcus |
Activity |
100.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus |
Staphylococcus |
Activity |
nan |
None |
10.1021/jm070708p |
| Staphylococcus |
Staphylococcus |
Inhibition |
3.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus |
Staphylococcus |
Inhibition |
8.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus |
Staphylococcus |
Inhibition |
60.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus |
Staphylococcus |
Inhibition |
80.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus |
Staphylococcus |
Inhibition |
80.4 |
% |
10.1128/aac.01653-09 |
| Staphylococcus |
Staphylococcus |
Inhibition |
99.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus |
Staphylococcus |
Inhibition |
100.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus |
Staphylococcus |
IZ |
18.0 |
mm |
10.1016/j.ejmech.2013.01.034 |
| Staphylococcus |
Staphylococcus |
IZ |
18.0 |
mm |
10.1016/j.ejmech.2013.03.027 |
| Staphylococcus |
Staphylococcus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.005 |
| Staphylococcus |
Staphylococcus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2007.07.006 |
| Staphylococcus |
Staphylococcus |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus |
Staphylococcus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus |
Staphylococcus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Staphylococcus |
Staphylococcus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus |
Staphylococcus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Staphylococcus |
Staphylococcus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2008.07.005 |
| Staphylococcus |
Staphylococcus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2009.03.024 |
| Staphylococcus |
Staphylococcus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.027 |
| Staphylococcus |
Staphylococcus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.05.041 |
| Staphylococcus |
Staphylococcus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00247-07 |
| Staphylococcus |
Staphylococcus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus |
Staphylococcus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.005 |
| Staphylococcus |
Staphylococcus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.07.006 |
| Staphylococcus |
Staphylococcus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus |
Staphylococcus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus |
Staphylococcus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus |
Staphylococcus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Staphylococcus |
Staphylococcus |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.01.034 |
| Staphylococcus |
Staphylococcus |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.034 |
| Staphylococcus |
Staphylococcus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Staphylococcus |
Staphylococcus |
MIC |
3.12 |
ug.mL-1 |
10.1016/j.bmcl.2009.03.025 |
| Staphylococcus |
Staphylococcus |
MIC |
3.12 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.033 |
| Staphylococcus |
Staphylococcus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Staphylococcus |
Staphylococcus |
MIC50 |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus |
Staphylococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus |
Staphylococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus |
Staphylococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus |
Staphylococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Staphylococcus |
Staphylococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus |
Staphylococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus |
Staphylococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Staphylococcus |
Staphylococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus |
Staphylococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01653-09 |
| Staphylococcus |
Staphylococcus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus |
Staphylococcus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus |
Staphylococcus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus |
Staphylococcus |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.01653-09 |
| Staphylococcus |
Staphylococcus |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus |
Staphylococcus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus |
Staphylococcus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus |
Staphylococcus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Staphylococcus |
Staphylococcus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus |
Staphylococcus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus |
Staphylococcus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus |
Staphylococcus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Staphylococcus |
Staphylococcus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus |
Staphylococcus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus |
Staphylococcus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus |
Staphylococcus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Enoyl-[acyl-carrier-protein] reductase (FabI) |
IC50 |
nan |
None |
10.1016/j.bmcl.2015.08.077 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
-0.53 |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
-0.27 |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
-0.12 |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.00301-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.00400-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.00846-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.01538-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.04 |
% |
10.1128/aac.01453-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.1 |
% |
10.1128/aac.00301-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
0.58 |
% |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1.0 |
log10CFU/ml |
10.1016/j.bmc.2019.06.010 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1.09 |
mg/L |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1.16 |
% |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1.19 |
log10CFU |
10.1021/acs.jmedchem.7b00949 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1.41 |
deltalog10CFU |
10.1016/j.ejmech.2017.12.090 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1.44 |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1.59 |
mg/L |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1.6 |
log10CFU/ml |
10.1021/acs.jnatprod.2c00621 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1.7 |
log10CFU/ml |
10.1039/c9md00391f |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
2.26 |
mg/L |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
2.3 |
mg/L |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
2.71 |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
2.77 |
mg/L |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
2.95 |
mg/L |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
4.27 |
mg/L |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
4.27 |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
4.55 |
mg/L |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
6.07 |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
8.0 |
% |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
10.15 |
mg/L |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
17.0 |
% |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
25.0 |
% |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
31.2 |
% |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
33.3 |
% |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
59.0 |
% |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
68.0 |
% |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
82.7 |
% |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
85.0 |
% |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
85.2 |
% |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
89.0 |
% |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
90.0 |
% |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
91.0 |
% |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
91.5 |
% |
10.1021/acs.jmedchem.7b00949 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
91.7 |
% |
10.1021/acs.jmedchem.7b00949 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
95.0 |
% |
10.1021/acs.jmedchem.7b00949 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
96.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
96.6 |
% |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
98.0 |
% |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
98.2 |
% |
10.1021/acs.jmedchem.7b00949 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
99.0 |
% |
10.1128/aac.01398-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
99.2 |
% |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
99.3 |
% |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
99.9 |
% |
10.1021/acs.jmedchem.7b00949 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
99.9 |
% |
10.1128/aac.00301-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
99.9 |
% |
10.1128/aac.01453-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00129-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00301-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00400-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00845-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.00952-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.01351-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.01453-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.01562-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
100.0 |
mg/L |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
567.0 |
mm3 |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
858.0 |
mm3 |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
932.0 |
mm3 |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1018.0 |
mm3 |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1234.0 |
mm3 |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1277.0 |
mm3 |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1407.0 |
mm3 |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
1644.0 |
mm3 |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.bmc.2020.115729 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.bmcl.2014.03.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.bmcl.2014.07.037 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.bmcl.2017.06.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.ejmech.2008.07.005 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.ejmech.2017.12.090 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.ejmech.2018.09.053 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.ejmech.2019.112022 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1016/j.ejmech.2021.113723 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/acs.jmedchem.6b00372 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/acs.jmedchem.6b01834 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/acs.jmedchem.7b00113 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/acs.jmedchem.7b00949 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/acs.jmedchem.7b01300 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/acsmedchemlett.7b00501 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/jm200938f |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/jm900519b |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1021/np050438i |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1039/C5MD00101C |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1039/D1MD00211B |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1039/d2md00351a |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1073/pnas.0700746104 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00064-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00129-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00208-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00301-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00350-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00638-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00766-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00833-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.00887-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01052-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01201-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01302-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
Activity |
nan |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
AUPAP |
70.2 |
% |
10.1128/aac.01194-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
AUPAP |
90.2 |
% |
10.1128/aac.01194-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
AUPAP |
178.0 |
% |
10.1128/aac.01194-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
-0.4 |
None |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
0.0 |
None |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
0.1 |
None |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
0.2 |
None |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
0.4 |
None |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
0.6 |
None |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
1.05 |
None |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
1.4 |
None |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
2.69 |
None |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
2.82 |
None |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
3.51 |
None |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
3.64 |
None |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
3.7 |
None |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
4.07 |
None |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
4.4 |
None |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
deltalog10CFU |
4.49 |
None |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
DIZ |
nan |
None |
10.1016/j.bmcl.2009.10.018 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.18 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2017.02.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.29 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.35 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.4 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.47 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.63 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.7 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
0.84 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
EC50 |
2.78 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
1.73 |
mg.kg-1 |
10.1016/j.ejmech.2013.03.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
1.73 |
mg.kg-1 |
10.1021/ml400280z |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
1.98 |
mg.kg-1 |
10.1021/ml400280z |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
2.0 |
mg.kg-1 |
10.1128/aac.00026-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
2.02 |
mg.kg-1 |
10.1016/j.ejmech.2013.03.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
2.3 |
mg.kg-1 |
10.1016/j.ejmech.2014.07.036 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
2.5 |
mg.kg-1 |
10.1016/j.bmcl.2022.128842 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
2.8 |
mg.kg-1 |
10.1021/jm501661f |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
3.7 |
mg/kg/day |
10.1128/aac.00833-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
4.0 |
mg.kg-1 |
10.1016/j.bmcl.2004.05.066 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
4.53 |
mg.kg-1 |
10.1021/acs.jmedchem.8b01750 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
4.83 |
mg.kg-1 |
10.1021/acs.jmedchem.8b01750 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
5.0 |
mg.kg-1 |
10.1016/j.bmc.2022.116614 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
5.0 |
mg.kg-1 |
10.1016/j.bmcl.2016.04.086 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
5.1 |
mg/kg/day |
10.1128/aac.00833-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
5.3 |
mg.kg-1 |
10.1016/j.bmcl.2008.03.043 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
5.3 |
mg/kg/day |
10.1016/j.bmcl.2006.01.109 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
5.4 |
mg kg-1 day-1 |
10.1016/j.bmcl.2004.04.037 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
5.6 |
mg.kg-1 |
10.1016/j.bmcl.2005.06.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
5.6 |
mg.kg-1 |
10.1016/j.bmcl.2007.10.061 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
5.9 |
mg.kg-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
6.3 |
mg.kg-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
6.3 |
mg/kg/day |
10.1128/aac.00833-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
6.4 |
mg/kg/day |
10.1128/aac.00833-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
7.0 |
mg.kg-1 |
10.1128/aac.00026-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
7.0 |
mg/kg/day |
10.1128/aac.00833-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
7.07 |
mg.kg-1 |
10.1021/jm4000598 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
7.4 |
mg.kg-1 |
10.1128/aac.00026-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
7.4 |
mg.kg-1 |
10.1128/aac.00084-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
7.89 |
mg.kg-1 |
10.1021/jm500312x |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
8.28 |
mg.kg-1 |
10.1021/jm4000598 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
8.45 |
mg.kg-1 |
10.1016/j.ejmech.2007.09.010 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
8.5 |
mg/kg/day |
10.1128/aac.00833-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
8.7 |
mg.kg-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
9.0 |
mg.kg-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
9.39 |
mg.kg-1 |
10.1021/jm500312x |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
9.4 |
mg.kg-1 |
10.1016/j.ejmech.2011.01.014 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
9.5 |
mg.kg-1 |
10.1021/jm200614t |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
9.87 |
mg.kg-1 |
10.1021/jm4000598 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
10.2 |
mg.kg-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
10.3 |
mg.kg-1 |
10.1128/aac.00026-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
11.9 |
mg.kg-1 |
10.1016/j.ejmech.2014.07.106 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
12.9 |
mg.kg-1 |
10.1016/j.ejmech.2011.01.014 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
14.1 |
mg.kg-1 |
10.1021/jm200614t |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
15.6 |
mg.kg-1 |
10.1016/j.ejmech.2011.01.014 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
15.6 |
mg.kg-1 |
10.1021/jm500312x |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
17.88 |
mg.kg-1 |
10.1016/j.ejmech.2007.01.012 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
21.4 |
mg.kg-1 |
10.1016/j.ejmech.2011.01.014 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
23.96 |
mg.kg-1 |
10.1016/j.ejmech.2007.01.012 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED50 |
29.1 |
mg.kg-1 |
10.1016/j.ejmech.2011.01.014 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED99 |
5.2 |
mg kg-1 |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED99 |
6.9 |
mg kg-1 |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED99 |
7.0 |
mg kg-1 |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED99 |
12.0 |
mg kg-1 |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED99 |
12.0 |
mg Kg-1 |
10.1016/j.bmcl.2009.04.144 |
| Staphylococcus aureus |
Staphylococcus aureus |
ED99 |
85.0 |
mg kg-1 |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Efficacy |
77.0 |
% |
10.1021/jm800038g |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
0.5 |
None |
10.1128/aac.00833-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
FC |
1.4 |
None |
10.1016/j.bmcl.2014.03.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
FIC |
0.25 |
None |
10.1021/acs.jnatprod.2c00621 |
| Staphylococcus aureus |
Staphylococcus aureus |
GI |
0.0 |
% |
10.1128/aac.01242-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
0.42 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
nan |
None |
10.1073/pnas.0700746104 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
0.5 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
1.3 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
2.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
2.4 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
2.5 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
4.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
4.6 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
4.9 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
9.8 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
40.5 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
45.2 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
51.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
75.6 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
81.6 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
84.6 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
91.1 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
98.7 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
99.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
99.13 |
% |
10.1016/j.ejmech.2016.07.001 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
99.46 |
% |
10.1016/j.ejmech.2016.07.001 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
99.51 |
% |
10.1016/j.ejmech.2016.07.001 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
100.0 |
% |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
nan |
% |
10.1128/aac.00633-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
nan |
% |
10.1128/aac.00887-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
18.0 |
mm |
10.1016/j.ejmech.2011.04.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
19.0 |
mm |
10.1128/aac.00231-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
26.0 |
mm |
10.1039/C2MD00252C |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
27.0 |
mm |
10.1016/j.bmcl.2009.10.018 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
28.0 |
mm |
10.1016/j.ejmech.2013.01.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
28.0 |
mm |
10.1016/j.ejmech.2013.03.027 |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
34.0 |
mm |
10.1039/c0md00015a |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
35.0 |
mm |
10.1039/c0md00015a |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
39.0 |
mm |
10.1039/c0md00015a |
| Staphylococcus aureus |
Staphylococcus aureus |
IZ |
42.0 |
mm |
10.1039/c0md00015a |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
-0.91 |
None |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
-0.69 |
None |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
-0.54 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
-0.42 |
None |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
-0.41 |
None |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
-0.39 |
None |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
-0.37 |
None |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
0.27 |
None |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
0.61 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
0.62 |
None |
10.1128/aac.00237-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
0.93 |
None |
10.1128/aac.00208-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
1.0 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
1.06 |
None |
10.1128/aac.00208-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
1.5 |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
1.51 |
None |
10.1128/aac.00237-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
2.0 |
None |
10.1128/aac.00633-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
2.0 |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
2.4 |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
2.5 |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
2.52 |
None |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
3.7 |
None |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
6.9 |
None |
10.1128/aac.01242-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10cfu |
7.1 |
None |
10.1128/aac.01242-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Log10 cfu |
0.2 |
None |
10.1021/jm060844e |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/g |
1.29 |
None |
10.1021/jm201467r |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/g |
2.46 |
None |
10.1021/jm201467r |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/g |
2.5 |
None |
10.1128/aac.00886-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/g |
2.9 |
None |
10.1128/aac.00886-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/g |
5.9 |
None |
10.1128/aac.00886-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-3.24 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.81 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.58 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.26 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.24 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.22 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.21 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.17 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.15 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.07 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.06 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
-0.04 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
0.02 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
0.21 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
0.32 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
0.52 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
0.74 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
1.31 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
1.55 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
1.7 |
None |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
2.13 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
2.72 |
None |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.0 |
None |
10.1128/aac.01194-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.1 |
None |
10.1128/aac.01194-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.19 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.24 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.26 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.3 |
None |
10.1128/aac.01194-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.64 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.66 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.9 |
None |
10.1128/aac.01194-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
3.98 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
4.2 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
4.24 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
4.25 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
4.5 |
None |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
4.52 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
4.6 |
None |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
4.8 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
4.89 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
4.95 |
None |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
5.1 |
None |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
7.1 |
None |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
log10CFU/ml |
7.3 |
None |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
Log 1/MIC |
-0.19 |
None |
10.1016/s0960-894x(99)00474-6 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
0.5 |
ug ml-1 |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
1.0 |
mg/ml |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
1.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
1.0 |
ug ml-1 |
10.1128/aac.00257-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
1.0 |
ug ml-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
1.56 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
2.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
2.0 |
ug ml-1 |
10.1021/acs.jmedchem.6b00233 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
2.0 |
ug ml-1 |
10.1128/aac.00257-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
2.0 |
ug ml-1 |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
2.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
2.0 |
ug ml-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
2.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
4.0 |
ug ml-1 |
10.1021/acs.jmedchem.6b00233 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
4.0 |
ug ml-1 |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
4.0 |
ug ml-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
4.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
8.0 |
ug ml-1 |
10.1016/j.ejmech.2016.11.042 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
8.0 |
ug ml-1 |
10.1016/j.ejmech.2017.02.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
8.0 |
ug ml-1 |
10.1016/j.ejmech.2017.08.039 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
8.0 |
ug ml-1 |
10.1016/j.ejmech.2021.113723 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
8.0 |
ug ml-1 |
10.1021/acs.jmedchem.6b00233 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
8.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
8.0 |
ug ml-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
10.7 |
ug ml-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
12.5 |
ug ml-1 |
10.1128/aac.00638-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
15.6 |
uM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
15.6 |
uM |
10.1021/acs.jmedchem.7b01903 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
15.6 |
uM |
10.1039/C6MD00381H |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
16.0 |
mg/L |
10.1128/aac.01242-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2016.11.042 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2017.02.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2017.08.039 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2018.03.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.04.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111593 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111830 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2020.112497 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2021.113723 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
16.0 |
ug ml-1 |
10.1021/acs.jmedchem.6b00233 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
16.0 |
ug ml-1 |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
20.0 |
ug ml-1 |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
31.3 |
uM |
10.1021/acs.jmedchem.1c00168 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
31.3 |
uM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
31.3 |
uM |
10.1021/acs.jmedchem.7b01903 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2016.11.042 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2017.02.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2017.08.039 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2018.03.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2018.09.053 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2019.04.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111593 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111830 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2020.112497 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1021/acs.jmedchem.6b00233 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1128/aac.00208-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
32.0 |
ug ml-1 |
10.1128/aac.00766-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
46.2 |
uM |
10.1016/j.ejmech.2020.113134 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
64.0 |
mg/L |
10.1128/aac.01242-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
64.0 |
ug ml-1 |
10.1016/j.bmc.2019.06.010 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
64.0 |
ug ml-1 |
10.1016/j.bmc.2020.115729 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2018.03.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2019.04.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111593 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111830 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2020.112497 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
64.0 |
ug ml-1 |
10.1016/j.ejmech.2022.114550 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
64.0 |
ug ml-1 |
10.1021/acs.jmedchem.6b00233 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
64.0 |
ug ml-1 |
10.1039/D1MD00211B |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2021.113723 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2022.114550 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC |
128.0 |
ug ml-1 |
10.1039/c9md00391f |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
0.5 |
mg/L |
10.1128/aac.00344-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
0.5 |
mg/L |
10.1128/aac.00666-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
1.0 |
mg/L |
10.1128/aac.00344-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
2.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
4.0 |
ug ml-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
6.0 |
ug ml-1 |
10.1128/aac.00257-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
8.0 |
mg/ml |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
8.0 |
ug ml-1 |
10.1128/aac.00257-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
8.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
8.0 |
ug ml-1 |
10.1128/aac.01325-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
8.0 |
ug ml-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC50 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
2.0 |
mg/L |
10.1128/aac.00344-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
2.0 |
mg/L |
10.1128/aac.00666-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
4.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
16.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
32.0 |
mg/ml |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
32.0 |
ug ml-1 |
10.1128/aac.00257-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
32.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
64.0 |
ug ml-1 |
10.1128/aac.00257-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC90 |
64.0 |
ug ml-1 |
10.1128/aac.01325-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC99.9 |
8.0 |
ug ml-1 |
10.1021/acs.jmedchem.6b00372 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBC99.9 |
16.0 |
ug ml-1 |
10.1021/acs.jmedchem.6b00372 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC |
128.0 |
ug ml-1 |
10.1128/aac.00766-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC |
2000.0 |
uM |
10.1021/acs.jmedchem.1c00168 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC |
2000.0 |
uM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC |
2000.0 |
uM |
10.1021/acs.jmedchem.7b01903 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC |
2000.0 |
uM |
10.1039/C6MD00381H |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC80 |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBEC90 |
128.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBIC80 |
26.8 |
ug ml-1 |
10.1016/j.ejmech.2018.06.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MBIC90 |
36.1 |
ug ml-1 |
10.1016/j.ejmech.2018.06.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.0005 |
ug.mL-1 |
10.1128/aac.01173-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmc.2014.10.037 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmc.2021.116580 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2007.01.012 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2004.05.066 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1016/s0960-894x(02)00043-4 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00350-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00550-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00307-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.38 |
ug.mL-1 |
10.1128/aac.00676-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.069 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ucm/s |
10.1016/j.bmcl.2009.07.115 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.033 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.021 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2004.05.066 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.093 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.102 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2011.12.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2015.06.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.047 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.005 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2007.07.006 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2007.09.010 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2008.07.005 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2009.03.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.05.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/s0960-894x(02)00043-4 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1016/s0960-894x(03)00249-x |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jnatprod.0c00279 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/acsmedchemlett.0c00653 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00015 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm500462x |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1021/np800503z |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1039/c9md00391f |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00247-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00350-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00550-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01091-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01201-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01376-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.62 |
ug.mL-1 |
10.1016/j.bmc.2017.02.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.75 |
ug.mL-1 |
10.1128/aac.00307-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.bmcl.2004.07.064 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.781 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.077 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.781 |
ug.mL-1 |
10.1016/j.ejmech.2010.10.015 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.8 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.069 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
0.85 |
ug.mL-1 |
10.1016/j.bmc.2021.116580 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2011.10.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2019.06.010 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115729 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.028 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.033 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.031 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.068 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.076 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.03.099 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.12.025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.01.109 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.05.071 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.06.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.12.081 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.093 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.075 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.03.043 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.07.115 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.137 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.102 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.10.052 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.10.069 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.03.053 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.04.046 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.06.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.12.027 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.08.032 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.047 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.12.012 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.126746 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.126747 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2020.127660 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.128203 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128531 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.005 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.013 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.01.012 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.05.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.07.006 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.09.010 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.02.002 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.09.035 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.007 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.053 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111593 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111781 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111830 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112046 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112497 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113659 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114204 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114550 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/s0960-894x(02)00043-4 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1016/s0960-894x(99)00473-4 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00153 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00233 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b01580 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jnatprod.0c00279 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00621 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jnatprod.7b00745 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jnatprod.9b00321 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jnatprod.9b01285 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acsmedchemlett.7b00263 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00015 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00379 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm020092y |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm058204j |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm101604v |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm200614t |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm300690s |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm4000598 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm500312x |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm500462x |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm800800c |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1021/np800503z |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1039/C8MD00081F |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1039/c9md00391f |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00026-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00064-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00169-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00247-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00350-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00361-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00533-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00550-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00633-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00676-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00915-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01098-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01113-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01201-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01242-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01350-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01351-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01432-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.13 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.001 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.25 |
ug.mL-1 |
10.1016/j.bmcl.2011.05.093 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.25 |
ug.mL-1 |
10.1021/jm0510023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.25 |
ug.mL-1 |
10.1128/aac.00676-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.48 |
ug.mL-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.01.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.027 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.5 |
ug.mL-1 |
10.1021/np0702032 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.00533-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.5 |
ug.mL-1 |
10.1128/aac.00676-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2004.07.064 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2009.03.025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2009.07.106 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2014.03.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.ejmech.2009.11.009 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.56 |
ug.mL-1 |
10.1016/s0960-894x(99)00474-6 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.56 |
ug.mL-1 |
10.1128/aac.00638-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.6 |
ug.mL-1 |
10.1016/j.bmc.2014.10.037 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.6 |
ug.mL-1 |
10.1016/j.bmcl.2016.04.086 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.6 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.069 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.75 |
ug.mL-1 |
10.1016/j.bmc.2021.116580 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1.75 |
ug.mL-1 |
10.1128/aac.00676-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1007/s00044-012-0394-2 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2008.08.079 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2011.10.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2015.02.016 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2019.06.010 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115729 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115776 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116397 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.017 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.018 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.028 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.029 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.021 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.031 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.068 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.02.047 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.037 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.096 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.10.073 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.03.099 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.04.045 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.06.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.10.053 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.12.025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.01.109 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.05.071 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.06.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.07.064 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.10.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.056 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.085 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.056 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.075 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.09.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.10.061 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.02.052 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.03.043 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.011 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.11.021 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.123 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.137 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.08.037 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.102 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.03.075 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.11.002 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.03.013 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.03.053 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.04.046 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.12.027 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.08.032 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.12.016 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.06.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128531 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128842 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.005 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.013 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.05.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.07.006 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.07.005 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.03.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.09.019 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.01.014 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.04.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.02.002 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.05.041 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.08.002 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.106 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2015.10.025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.11.042 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.060 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.02.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.08.039 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.053 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111644 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111830 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112497 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112686 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113442 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113480 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113723 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113741 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114204 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114550 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(01)00305-5 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00249-x |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00430-x |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00194-2 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(99)00473-4 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00295 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c00480 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00372 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jnatprod.7b00133 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acsmedchemlett.7b00263 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00379 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm020092y |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm070638m |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm2002124 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm201467r |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm300690s |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm500462x |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm501661f |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm980274l |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm980546k |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm990373e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/ml400280z |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/np0702032 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/np300544a |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1021/np800783b |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1039/C5MD00101C |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1039/c9md00391f |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1039/D1MD00211B |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1039/d2md00260d |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1073/pnas.0700746104 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00044-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00062-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00064-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00183-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00208-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00209-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00237-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00350-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00361-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00417-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00533-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00550-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00676-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00714-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00766-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00833-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00887-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00908-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00915-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00985-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01022-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01032-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01194-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01201-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01242-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01347-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01350-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01422-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01583-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.5 |
ug.mL-1 |
10.1016/j.bmcl.2011.05.093 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.5 |
ug.mL-1 |
10.1016/j.ejmech.2009.09.019 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.5 |
ug.mL-1 |
10.1021/jm0510023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.5 |
ug.mL-1 |
10.1128/aac.00676-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.5 |
ug.mL-1 |
10.1128/aac.00775-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2.55 |
ug.mL-1 |
10.1128/aac.00766-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.0 |
ug.mL-1 |
10.1128/aac.00676-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.1 |
ug.mL-1 |
10.1016/j.bmcl.2017.10.018 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.12 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.12 |
ug.mL-1 |
10.1016/j.bmcl.2009.03.025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.12 |
ug.mL-1 |
10.1016/j.bmcl.2009.07.106 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.12 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.033 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.12 |
ug.mL-1 |
10.1016/j.ejmech.2009.11.009 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.125 |
ug.mL-1 |
10.1016/j.bmc.2014.10.037 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.13 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.069 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3.73 |
ug.mL-1 |
10.1128/aac.00766-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1007/s00044-012-0394-2 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.017 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.11.093 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.03.104 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.123 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.102 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.04.046 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.12.016 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.11.019 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.03.028 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.02.002 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.106 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.007 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.054 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.017 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113480 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113723 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/s0960-894x(02)00352-9 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00249-x |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00194-2 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jnatprod.1c00578 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00621 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jnatprod.7b00133 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm020248u |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm058204j |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm070708p |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm2002124 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm501661f |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm800318d |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm9509556 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm980274l |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm980546k |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm990373e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/np300544a |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/np800503z |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1021/np800783b |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1039/d2md00260d |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1073/pnas.0700746104 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00062-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00169-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00183-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00209-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00350-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00550-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00642-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00676-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00714-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00766-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00833-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00846-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00908-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00915-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01015-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01098-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01113-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01145-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01193-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01302-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01350-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01376-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01422-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01583-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
7.8 |
ug.mL-1 |
10.1016/j.bmc.2019.05.012 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.10.010 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128842 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm4000598 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00183-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00231-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00350-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00550-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00714-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00766-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00985-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01032-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01098-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01113-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01194-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01347-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01376-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01422-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.01583-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.12.025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.075 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.05.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113480 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1021/acsmedchemlett.7b00263 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm060844e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm200614t |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm300690s |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00183-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00550-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00714-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01302-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01347-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.03.043 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.08.002 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.044 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.06.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.063 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114204 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00233 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00372 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00379 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm070638m |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm501661f |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/ml400280z |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1021/np800783b |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1073/pnas.0700746104 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00183-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00550-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00714-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01098-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01302-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01347-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.028 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111593 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111830 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112497 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1039/c9md00391f |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00714-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01015-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01098-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01193-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01567-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.10.048 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01098-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
500.0 |
ug.mL-1 |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
512.0 |
ug.mL-1 |
10.1128/aac.00846-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2015.06.031 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1000.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.04.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1500.0 |
nM |
10.1021/acsmedchemlett.0c00425 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1560.0 |
nM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2000.0 |
nM |
10.1016/j.ejmech.2015.06.031 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2500.0 |
nM |
10.6019/CHEMBL4513141 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
2600.0 |
nM |
10.1016/j.ejmech.2020.113134 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3000.0 |
nM |
10.1016/j.ejmech.2018.09.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3000.0 |
nM |
10.1016/j.ejmech.2020.112444 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3125.0 |
nM |
10.1016/j.ejmech.2022.114333 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3130.0 |
nM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3130.0 |
nM |
10.1021/acs.jmedchem.7b01903 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
3130.0 |
nM |
10.1039/C6MD00381H |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4000.0 |
nM |
10.1021/acsmedchemlett.0c00425 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4629.0 |
nM |
10.1016/j.bmcl.2009.04.133 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
5200.0 |
nM |
10.1016/j.ejmech.2020.113134 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6000.0 |
nM |
10.1016/j.bmcl.2004.08.059 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6000.0 |
nM |
10.1016/j.ejmech.2022.114213 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6200.0 |
nM |
10.1021/jm501174m |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6250.0 |
nM |
10.1016/j.ejmech.2020.113002 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6250.0 |
nM |
10.1016/j.ejmech.2022.114333 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6250.0 |
nM |
10.1021/acs.jmedchem.2c01349 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
6250.0 |
nM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
9258.1 |
nM |
10.1016/j.bmcl.2009.04.133 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
12000.0 |
nM |
10.1021/jm501174m |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
12500.0 |
nM |
10.1016/j.ejmech.2018.06.045 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
12500.0 |
nM |
10.1021/acs.jmedchem.1c00168 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
12500.0 |
nM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
12500.0 |
nM |
10.1021/acs.jmedchem.7b01903 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
32000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64000.0 |
nM |
10.1016/j.ejmech.2015.06.031 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
190000.0 |
nM |
10.1016/j.ejmech.2018.09.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
190000.0 |
nM |
10.1016/j.ejmech.2020.112444 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
250000.0 |
ug.mL-1 |
10.1016/j.bmc.2014.10.037 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4000000.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.021 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
64000000.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.021 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmc.2008.08.079 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmc.2015.02.016 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmc.2019.05.012 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmcl.2007.06.075 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmcl.2013.10.069 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmcl.2013.11.002 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmcl.2015.08.077 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.ejmech.2017.10.048 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.ejmech.2018.09.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.ejmech.2021.113480 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1021/acs.jmedchem.8b01750 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1021/jm2002124 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1128/aac.00550-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1128/aac.00676-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC100 |
0.78 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC100 |
12.5 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC100 |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00344-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00666-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
0.75 |
ug.mL-1 |
10.1128/aac.00307-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2009.08.026 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm1014023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm101604v |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00301-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00307-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00550-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01325-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.007 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1021/jm020328y |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1021/jm060844e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1021/jm201467r |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00257-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00301-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01351-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
4.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115776 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
16.0 |
ug.mL-1 |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2000.0 |
ug.mL-1 |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
2000000.0 |
ug.mL-1 |
10.1016/j.bmc.2014.10.037 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC50 |
nan |
None |
10.1128/aac.01017-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2009.08.026 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.019 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00307-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00344-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00846-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
1.5 |
ug.mL-1 |
10.1128/aac.00307-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.06.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.007 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm020328y |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm060844e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm1014023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm101604v |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm301113w |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00206-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00301-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00344-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00550-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00666-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00846-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01325-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01351-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01516-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmc.2020.115776 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.07.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.004 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1021/jm070708p |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1021/jm201467r |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1021/jm960294s |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00257-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.023 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
8.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
16.0 |
ug.mL-1 |
10.1021/jm301113w |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
2000.0 |
ug.mL-1 |
10.1128/aac.00452-10 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
4000000.0 |
ug.mL-1 |
10.1016/j.bmc.2014.10.037 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
nan |
None |
10.1128/aac.01017-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC99 |
1.0 |
ug ml-1 |
10.1016/j.bmcl.2014.02.025 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC99 |
2.0 |
ug ml-1 |
10.1016/j.bmcl.2014.02.025 |
| Staphylococcus aureus |
Staphylococcus aureus |
mortality |
16.0 |
% |
10.1016/j.ejmech.2014.07.106 |
| Staphylococcus aureus |
Staphylococcus aureus |
mortality |
66.0 |
% |
10.1016/j.ejmech.2014.07.106 |
| Staphylococcus aureus |
Staphylococcus aureus |
mortality |
83.0 |
% |
10.1016/j.ejmech.2014.07.106 |
| Staphylococcus aureus |
Staphylococcus aureus |
PD50 |
3.1 |
mg Kg-1 |
10.1021/jm070708p |
| Staphylococcus aureus |
Staphylococcus aureus |
PD50 |
4.0 |
mg kg-1 |
10.1016/j.bmcl.2010.11.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
PD50 |
5.0 |
mg Kg-1 |
10.1021/jm070708p |
| Staphylococcus aureus |
Staphylococcus aureus |
PD50 |
6.25 |
mg Kg-1 |
10.1021/jm070708p |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
0.5 |
None |
10.1021/jm500462x |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
1.0 |
None |
10.1021/jm500462x |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
2.0 |
None |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
2.0 |
None |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
4.0 |
None |
10.1016/j.ejmech.2021.113480 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
4.0 |
None |
10.1016/j.ejmech.2021.113723 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
4.0 |
None |
10.1128/aac.01653-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
16.0 |
None |
10.1016/j.ejmech.2018.09.053 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
16.0 |
None |
10.1128/aac.00766-09 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
32.0 |
None |
10.1016/j.bmc.2019.06.010 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
32.0 |
None |
10.1016/j.bmc.2020.115729 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
32.0 |
None |
10.1016/j.ejmech.2018.09.053 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
32.0 |
None |
10.1016/j.ejmech.2021.113480 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
64.0 |
None |
10.1016/j.bmc.2020.115729 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
64.0 |
None |
10.1016/j.ejmech.2021.113723 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
nan |
None |
10.1016/j.ejmech.2021.113480 |
| Staphylococcus aureus |
Staphylococcus aureus |
Ratio |
nan |
None |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus aureus |
Staphylococcus aureus |
Survival |
30.0 |
% |
10.1016/j.bmcl.2014.03.022 |
| Staphylococcus aureus |
Staphylococcus aureus |
Survival |
30.0 |
% |
10.1039/C5MD00101C |
| Staphylococcus aureus |
Staphylococcus aureus |
Survival |
60.0 |
% |
10.1128/aac.00738-06 |
| Staphylococcus aureus |
Staphylococcus aureus |
Survival |
100.0 |
% |
10.1128/aac.00738-06 |
| Staphylococcus aureus subsp. aureus RN4220 |
Staphylococcus aureus subsp. aureus RN4220 |
ABBC |
-2.27 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Staphylococcus aureus subsp. aureus RN4220 |
Staphylococcus aureus subsp. aureus RN4220 |
ABBC |
-1.21 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Staphylococcus aureus subsp. aureus RN4220 |
Staphylococcus aureus subsp. aureus RN4220 |
AUBC |
228.8 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Staphylococcus aureus subsp. aureus RN4220 |
Staphylococcus aureus subsp. aureus RN4220 |
AUBC |
229.4 |
log10CFU/ml.hr |
10.1128/aac.01022-09 |
| Staphylococcus aureus subsp. aureus RN4220 |
Staphylococcus aureus subsp. aureus RN4220 |
fT>MIC |
50.0 |
% |
10.1128/aac.01022-09 |
| Staphylococcus aureus subsp. aureus RN4220 |
Staphylococcus aureus subsp. aureus RN4220 |
fT>MIC |
66.6 |
% |
10.1128/aac.01022-09 |
| Staphylococcus aureus subsp. aureus RN4220 |
Staphylococcus aureus subsp. aureus RN4220 |
Ratio |
6.64 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus subsp. aureus RN4220 |
Staphylococcus aureus subsp. aureus RN4220 |
Ratio |
7.77 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus subsp. aureus RN4220 |
Staphylococcus aureus subsp. aureus RN4220 |
Ratio |
7.95 |
None |
10.1128/aac.01022-09 |
| Staphylococcus aureus subsp. aureus RN4220 |
Staphylococcus aureus subsp. aureus RN4220 |
RatioAUC/MIC |
32.9 |
None |
10.1128/aac.01022-09 |
| Staphylococcus capitis |
Staphylococcus capitis |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC |
16.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus capitis |
Staphylococcus capitis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus chromogenes |
Staphylococcus chromogenes |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Staphylococcus cohnii |
Staphylococcus cohnii |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus cohnii |
Staphylococcus cohnii |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus cohnii |
Staphylococcus cohnii |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus cohnii |
Staphylococcus cohnii |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus cohnii |
Staphylococcus cohnii |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus cohnii |
Staphylococcus cohnii |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
0.0 |
% |
10.1128/aac.00400-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
0.0 |
% |
10.1128/aac.01538-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
0.49 |
mg/L |
10.1128/aac.01724-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
96.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
99.1 |
% |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
99.4 |
% |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
99.7 |
% |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
100.0 |
% |
10.1128/aac.00400-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
100.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
nan |
None |
10.1016/j.ejmech.2008.07.005 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
nan |
None |
10.1128/aac.00887-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
nan |
None |
10.1128/aac.01052-06 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Activity |
nan |
None |
10.1128/aac.01538-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
EC50 |
2.99 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
ED50 |
84.77 |
mg.kg-1 |
10.1016/j.ejmech.2007.01.012 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Inhibition |
nan |
% |
10.1128/aac.00887-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
IZ |
6.0 |
mm |
10.1128/aac.00231-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
log10cfu |
-1.0 |
None |
10.1128/aac.01724-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
log10cfu |
0.18 |
None |
10.1128/aac.01724-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
log10cfu |
0.22 |
None |
10.1128/aac.00237-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
log10cfu |
0.61 |
None |
10.1128/aac.00237-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
0.5 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
8.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111593 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.04.063 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111830 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2020.112497 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC50 |
2.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MBC90 |
4.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2009.09.019 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.047 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.25 |
ug.mL-1 |
10.1016/s0960-894x(02)00043-4 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.021 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2009.07.115 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.123 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.102 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2011.12.063 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2007.01.012 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.106 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.063 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.111593 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1016/s0960-894x(02)00043-4 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1016/s0960-894x(03)00249-x |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1016/s0960-894x(03)00430-x |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00379 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
0.781 |
ug.mL-1 |
10.1016/j.ejmech.2010.10.015 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.017 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.018 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.022 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.029 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.08.021 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.12.025 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.075 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.07.115 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.102 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.03.075 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.07.034 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.023 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2016.08.032 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.01.012 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.05.003 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111830 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112497 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114204 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/s0960-894x(02)00352-9 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00194-2 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1016/s0960-894x(99)00473-4 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00372 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm020248u |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm200614t |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm4000598 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm501661f |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm9509556 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm980274l |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm980546k |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm990373e |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1021/np0702032 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1021/np800783b |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1039/c9md00391f |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00237-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01032-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01724-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2004.07.064 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.024 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.06.096 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.04.045 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.075 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.03.053 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.06.022 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2015.10.025 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00249-x |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm4000598 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00887-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.017 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113480 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113723 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.067 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2006.11.019 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm4000598 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
8.0 |
ug.mL-1 |
10.1039/d2md00260d |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2008.03.028 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm200614t |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.02.055 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
32.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.01619-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00231-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01032-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
1560.0 |
nM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
2000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
3130.0 |
nM |
10.1016/j.ejmech.2018.06.045 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
3130.0 |
nM |
10.1021/acs.jmedchem.5b02004 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
3130.0 |
nM |
10.1039/C6MD00381H |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
32000000.0 |
ug.mL-1 |
10.1016/j.bmc.2014.10.037 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
nan |
None |
10.1016/j.ejmech.2021.113480 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
nan |
None |
10.1021/acsmedchemlett.7b00263 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
32.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC50 |
32000000.0 |
ug.mL-1 |
10.1016/j.bmc.2014.10.037 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.022 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm301113w |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm960294s |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.015 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
128.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC90 |
64000000.0 |
ug.mL-1 |
10.1016/j.bmc.2014.10.037 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
Ratio |
nan |
None |
10.1016/j.ejmech.2021.113480 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
96.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
99.0 |
% |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
99.3 |
% |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
100.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
100.0 |
% |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC |
0.5 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC |
1.0 |
mg/ml |
10.1128/aac.00452-10 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC50 |
2.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC50 |
8.0 |
mg/ml |
10.1128/aac.00452-10 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC90 |
4.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MBC90 |
32.0 |
mg/ml |
10.1128/aac.00452-10 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
1.0 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00379 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00372 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm501661f |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
2.0 |
ug.mL-1 |
10.1021/np800783b |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC |
500.0 |
ug.mL-1 |
10.1128/aac.00452-10 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC50 |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC50 |
2000.0 |
ug.mL-1 |
10.1128/aac.00452-10 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm301113w |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00952-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus haemolyticus |
Staphylococcus haemolyticus |
MIC90 |
2000.0 |
ug.mL-1 |
10.1128/aac.00452-10 |
| Staphylococcus hominis |
Staphylococcus hominis |
Activity |
96.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
Activity |
100.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MBC |
0.5 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MBC50 |
2.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MBC90 |
4.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC |
1.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00430-x |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00859-08 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC50 |
nan |
None |
10.1128/aac.00859-08 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus hominis |
Staphylococcus hominis |
MIC90 |
nan |
None |
10.1128/aac.00859-08 |
| Staphylococcus intermedius |
Staphylococcus intermedius |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus intermedius |
Staphylococcus intermedius |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus intermedius |
Staphylococcus intermedius |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
Activity |
0.0 |
% |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
Activity |
20.0 |
% |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
Activity |
80.0 |
% |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
BBC |
4.0 |
ug ml-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
BBC |
128.0 |
ug ml-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MBC50 |
128.0 |
ug ml-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MBC90 |
128.0 |
ug ml-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01052-06 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus lugdunensis |
Staphylococcus lugdunensis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01052-06 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
0.781 |
ug.mL-1 |
10.1016/j.ejmech.2010.10.015 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.04.045 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus saprophyticus |
Staphylococcus saprophyticus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Staphylococcus simulans |
Staphylococcus simulans |
Activity |
96.0 |
% |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MBC |
0.25 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MBC |
0.5 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MBC50 |
2.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MBC90 |
4.0 |
ug ml-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC50 |
0.25 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus simulans |
Staphylococcus simulans |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00624-09 |
| Staphylococcus sp. |
Staphylococcus sp. |
Activity |
100.0 |
% |
10.1128/aac.01562-06 |
| Staphylococcus sp. |
Staphylococcus sp. |
MBC |
2.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Staphylococcus sp. |
Staphylococcus sp. |
MBC |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Staphylococcus sp. |
Staphylococcus sp. |
MBC50 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Staphylococcus sp. |
Staphylococcus sp. |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Staphylococcus sp. |
Staphylococcus sp. |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus sp. |
Staphylococcus sp. |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus sp. |
Staphylococcus sp. |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus sp. |
Staphylococcus sp. |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus sp. |
Staphylococcus sp. |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus sp. |
Staphylococcus sp. |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01562-06 |
| Staphylococcus sp. |
Staphylococcus sp. |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus sp. |
Staphylococcus sp. |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC |
0.781 |
ug.mL-1 |
10.1016/j.ejmech.2010.10.015 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Staphylococcus warneri |
Staphylococcus warneri |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus xylosus |
Staphylococcus xylosus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus xylosus |
Staphylococcus xylosus |
MIC |
0.781 |
ug.mL-1 |
10.1016/j.ejmech.2010.10.015 |
| Staphylococcus xylosus |
Staphylococcus xylosus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Staphylococcus xylosus |
Staphylococcus xylosus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus |
Streptococcus |
Activity |
1.3 |
% |
10.1128/aac.01453-08 |
| Streptococcus |
Streptococcus |
Activity |
99.9 |
% |
10.1128/aac.01453-08 |
| Streptococcus |
Streptococcus |
Activity |
100.0 |
% |
10.1128/aac.01453-08 |
| Streptococcus |
Streptococcus |
EC50 |
645.0 |
nM |
None |
| Streptococcus |
Streptococcus |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
0.5 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
0.8 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
1.5 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
1.9 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
3.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
3.5 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
3.8 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
8.2 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
16.6 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
39.6 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
95.5 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
96.1 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
96.2 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Streptococcus |
Streptococcus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00247-07 |
| Streptococcus |
Streptococcus |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00430-x |
| Streptococcus |
Streptococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Streptococcus |
Streptococcus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus |
Streptococcus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01453-08 |
| Streptococcus |
Streptococcus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
Activity |
100.0 |
% |
10.1128/aac.00149-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
Activity |
100.0 |
% |
10.1128/aac.00400-09 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.034 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2009.03.025 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.033 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.023 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Streptococcus agalactiae |
Streptococcus agalactiae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Streptococcus constellatus |
Streptococcus constellatus |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| Streptococcus constellatus |
Streptococcus constellatus |
Inhibition |
1.1 |
% |
10.1128/aac.01496-06 |
| Streptococcus constellatus |
Streptococcus constellatus |
Inhibition |
3.4 |
% |
10.1128/aac.01496-06 |
| Streptococcus constellatus |
Streptococcus constellatus |
Inhibition |
12.4 |
% |
10.1128/aac.01496-06 |
| Streptococcus constellatus |
Streptococcus constellatus |
Inhibition |
42.7 |
% |
10.1128/aac.01496-06 |
| Streptococcus constellatus |
Streptococcus constellatus |
Inhibition |
98.9 |
% |
10.1128/aac.01496-06 |
| Streptococcus constellatus |
Streptococcus constellatus |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC50 |
nan |
None |
10.1128/aac.01398-07 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Streptococcus constellatus |
Streptococcus constellatus |
MIC90 |
nan |
None |
10.1128/aac.01398-07 |
| Streptococcus dysgalactiae |
Streptococcus dysgalactiae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114495 |
| Streptococcus dysgalactiae subsp. equisimilis |
Streptococcus dysgalactiae subsp. equisimilis |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus dysgalactiae subsp. equisimilis |
Streptococcus dysgalactiae subsp. equisimilis |
MIC50 |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus dysgalactiae subsp. equisimilis |
Streptococcus dysgalactiae subsp. equisimilis |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus equinus |
Streptococcus equinus |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus equinus |
Streptococcus equinus |
Inhibition |
2.7 |
% |
10.1128/aac.01496-06 |
| Streptococcus equinus |
Streptococcus equinus |
Inhibition |
23.8 |
% |
10.1128/aac.01496-06 |
| Streptococcus equinus |
Streptococcus equinus |
Inhibition |
87.2 |
% |
10.1128/aac.01496-06 |
| Streptococcus equinus |
Streptococcus equinus |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus equinus |
Streptococcus equinus |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus equinus |
Streptococcus equinus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus equinus |
Streptococcus equinus |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus equinus |
Streptococcus equinus |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus equinus |
Streptococcus equinus |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus gordonii |
Streptococcus gordonii |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus gordonii |
Streptococcus gordonii |
Inhibition |
33.3 |
% |
10.1128/aac.01496-06 |
| Streptococcus gordonii |
Streptococcus gordonii |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus gordonii |
Streptococcus gordonii |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus gordonii |
Streptococcus gordonii |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus intermedius |
Streptococcus intermedius |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| Streptococcus intermedius |
Streptococcus intermedius |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus intermedius |
Streptococcus intermedius |
Inhibition |
24.2 |
% |
10.1128/aac.01496-06 |
| Streptococcus intermedius |
Streptococcus intermedius |
Inhibition |
87.9 |
% |
10.1128/aac.01496-06 |
| Streptococcus intermedius |
Streptococcus intermedius |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus intermedius |
Streptococcus intermedius |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus intermedius |
Streptococcus intermedius |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus intermedius |
Streptococcus intermedius |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Streptococcus intermedius |
Streptococcus intermedius |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus intermedius |
Streptococcus intermedius |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus intermedius |
Streptococcus intermedius |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Streptococcus intermedius |
Streptococcus intermedius |
MIC50 |
nan |
None |
10.1128/aac.01398-07 |
| Streptococcus intermedius |
Streptococcus intermedius |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus intermedius |
Streptococcus intermedius |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus intermedius |
Streptococcus intermedius |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Streptococcus intermedius |
Streptococcus intermedius |
MIC90 |
nan |
None |
10.1128/aac.01398-07 |
| Streptococcus mitis |
Streptococcus mitis |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| Streptococcus mitis |
Streptococcus mitis |
Inhibition |
0.3 |
% |
10.1128/aac.01496-06 |
| Streptococcus mitis |
Streptococcus mitis |
Inhibition |
1.2 |
% |
10.1128/aac.01496-06 |
| Streptococcus mitis |
Streptococcus mitis |
Inhibition |
4.4 |
% |
10.1128/aac.01496-06 |
| Streptococcus mitis |
Streptococcus mitis |
Inhibition |
33.4 |
% |
10.1128/aac.01496-06 |
| Streptococcus mitis |
Streptococcus mitis |
Inhibition |
99.1 |
% |
10.1128/aac.01496-06 |
| Streptococcus mitis |
Streptococcus mitis |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus mitis |
Streptococcus mitis |
MIC |
0.008 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Streptococcus mitis |
Streptococcus mitis |
MIC |
0.015 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus mitis |
Streptococcus mitis |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus mitis |
Streptococcus mitis |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus mitis |
Streptococcus mitis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus mitis |
Streptococcus mitis |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2004.07.064 |
| Streptococcus mitis |
Streptococcus mitis |
MIC50 |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus mitis |
Streptococcus mitis |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus mitis |
Streptococcus mitis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Streptococcus mitis |
Streptococcus mitis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus mitis |
Streptococcus mitis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus mitis |
Streptococcus mitis |
MIC50 |
nan |
None |
10.1128/aac.01398-07 |
| Streptococcus mitis |
Streptococcus mitis |
MIC90 |
0.06 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus mitis |
Streptococcus mitis |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus mitis |
Streptococcus mitis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus mitis |
Streptococcus mitis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus mitis |
Streptococcus mitis |
MIC90 |
nan |
None |
10.1128/aac.01398-07 |
| Streptococcus mutans |
Streptococcus mutans |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus mutans |
Streptococcus mutans |
Inhibition |
36.8 |
% |
10.1128/aac.01496-06 |
| Streptococcus mutans |
Streptococcus mutans |
Inhibition |
89.5 |
% |
10.1128/aac.01496-06 |
| Streptococcus mutans |
Streptococcus mutans |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus mutans |
Streptococcus mutans |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus mutans |
Streptococcus mutans |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus oralis |
Streptococcus oralis |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| Streptococcus oralis |
Streptococcus oralis |
Inhibition |
0.7 |
% |
10.1128/aac.01496-06 |
| Streptococcus oralis |
Streptococcus oralis |
Inhibition |
3.6 |
% |
10.1128/aac.01496-06 |
| Streptococcus oralis |
Streptococcus oralis |
Inhibition |
34.5 |
% |
10.1128/aac.01496-06 |
| Streptococcus oralis |
Streptococcus oralis |
Inhibition |
96.4 |
% |
10.1128/aac.01496-06 |
| Streptococcus oralis |
Streptococcus oralis |
Inhibition |
99.3 |
% |
10.1128/aac.01496-06 |
| Streptococcus oralis |
Streptococcus oralis |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus oralis |
Streptococcus oralis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus oralis |
Streptococcus oralis |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00372 |
| Streptococcus oralis |
Streptococcus oralis |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm501661f |
| Streptococcus oralis |
Streptococcus oralis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus oralis |
Streptococcus oralis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus oralis |
Streptococcus oralis |
MIC50 |
nan |
None |
10.1128/aac.01398-07 |
| Streptococcus oralis |
Streptococcus oralis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus oralis |
Streptococcus oralis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus oralis |
Streptococcus oralis |
MIC90 |
nan |
None |
10.1128/aac.01398-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
0.0 |
% |
10.1128/aac.00107-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
0.0 |
% |
10.1128/aac.01268-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
0.0 |
% |
10.1128/aac.01538-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
100.0 |
% |
10.1128/aac.00107-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
100.0 |
% |
10.1128/aac.00149-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
100.0 |
% |
10.1128/aac.00400-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
100.0 |
% |
10.1128/aac.00845-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
100.0 |
% |
10.1128/aac.01268-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
100.0 |
% |
10.1128/aac.01384-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
100.0 |
% |
10.1128/aac.01797-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Activity |
nan |
None |
10.1021/jm070708p |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
ED50 |
1.5 |
mg.kg-1 |
10.1016/j.bmcl.2016.04.086 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
ED50 |
5.6 |
mg.kg-1 |
10.1128/aac.00026-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
ED50 |
8.17 |
mg.kg-1 |
10.1021/jm401931e |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
ED50 |
9.3 |
mg.kg-1 |
10.1021/jm401931e |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
ED50 |
14.0 |
mg/kg/day |
10.1128/aac.00833-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
ED50 |
16.8 |
mg.kg-1 |
10.1021/jm401931e |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
ED50 |
20.0 |
mg/kg/day |
10.1128/aac.00833-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
ED50 |
40.0 |
mg/kg/day |
10.1128/aac.00833-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
FC |
0.8 |
None |
10.1016/j.bmcl.2014.03.022 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
FC |
1.0 |
None |
10.1016/j.bmcl.2014.03.022 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
FC |
4.5 |
None |
10.1016/j.bmcl.2014.03.022 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
IC50 |
nan |
None |
10.1073/pnas.0700746104 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
log10cfu |
2.5 |
None |
10.1021/jm800318d |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
log10cfu |
5.9 |
None |
10.1021/jm800318d |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Log10 cfu |
3.89 |
None |
10.1021/jm070428+ |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
Log10 cfu |
nan |
None |
10.1021/jm070428+ |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
log10CFU/g |
3.56 |
None |
10.1021/jm201467r |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC |
2.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC |
4.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.04.063 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111593 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111830 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2020.112497 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2019.04.063 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111593 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111830 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC |
32.0 |
ug ml-1 |
10.1016/j.ejmech.2020.112497 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC50 |
4.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MBC90 |
8.0 |
ug ml-1 |
10.1128/aac.01569-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.06 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01797-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.067 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.125 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2011.10.041 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2005.12.025 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2007.01.012 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2007.05.003 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1021/np800503z |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00026-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.01797-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.39 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.034 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.bmcl.2014.03.022 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.4 |
ug.mL-1 |
10.1021/jm800318d |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2011.10.041 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.018 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.029 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.093 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.075 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.102 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2014.03.013 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2022.128531 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2006.10.005 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2007.07.006 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2008.07.005 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2009.03.024 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.05.041 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/s0960-894x(02)00043-4 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1016/s0960-894x(98)00194-2 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00295 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00213 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1021/acsmedchemlett.7b00263 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm201467r |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1021/ml400280z |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1021/np800783b |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01268-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01797-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.bmcl.2004.07.064 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.bmcl.2009.03.025 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.033 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
0.8 |
ug.mL-1 |
10.1016/j.bmcl.2016.04.086 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2008.08.079 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2011.10.041 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2016.07.029 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.017 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.03.099 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.03.104 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.10.063 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.056 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.085 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.02.052 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.07.115 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.102 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.03.013 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.03.053 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128842 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.09.010 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.02.002 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.003 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.08.002 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.063 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111593 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111644 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111830 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112497 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1016/s0960-894x(02)00352-9 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00295 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00720 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00213 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm020248u |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm058204j |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm200614t |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm800800c |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm9509556 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm980274l |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm980546k |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm990373e |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/ml400280z |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/np0702032 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1021/np800503z |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1039/c9md00391f |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1073/pnas.0700746104 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00026-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.06.063 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.11.093 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.07.064 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.056 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.10.061 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.011 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.014 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.054 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.12.063 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.05.023 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128531 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.063 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00430-x |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm4000598 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00026-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00833-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.022 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01208-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
5.8 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.011 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
32.0 |
ug.mL-1 |
10.1021/acsmedchemlett.5b00213 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
2000.0 |
nM |
10.1016/j.bmc.2019.03.034 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
3100.0 |
nM |
10.1021/jm501174m |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC100 |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1021/jm020328y |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00107-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01797-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2009.08.026 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm1014023 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm201467r |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01268-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01384-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01797-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
0.5 |
ug.mL-1 |
10.1021/jm020328y |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.07.022 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.11.022 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm070708p |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm201467r |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm960294s |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00107-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01268-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01384-06 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01797-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2009.08.026 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.023 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm1014023 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00484-10 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
PD50 |
10.0 |
mg kg-1 |
10.1016/j.bmcl.2010.11.022 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
PD50 |
38.81 |
mg kg-1 |
10.1016/j.bmc.2016.07.029 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
Activity |
98.0 |
% |
10.1128/aac.01398-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
Activity |
100.0 |
% |
10.1128/aac.00149-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
Activity |
100.0 |
% |
10.1128/aac.00400-09 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
ED50 |
7.8 |
mg.kg-1 |
10.1021/jm401931e |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MBC50 |
1.0 |
mg/L |
10.1128/aac.00344-06 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MBC50 |
1.0 |
mg/L |
10.1128/aac.00666-06 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MBC90 |
2.0 |
mg/L |
10.1128/aac.00344-06 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MBC90 |
2.0 |
mg/L |
10.1128/aac.00666-06 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.012 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.ejmech.2012.02.002 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.067 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2005.12.025 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2012.02.002 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.39 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.034 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2004.04.024 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.075 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2017.06.022 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.025 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1016/s0960-894x(02)00043-4 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1016/s0960-894x(99)00473-4 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1021/acsmedchemlett.7b00263 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1021/np800783b |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.bmcl.2013.01.033 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2003.07.033 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2006.07.064 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.011 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.014 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.05.003 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.02.002 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113480 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113723 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00372 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm201467r |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1021/jm501661f |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2009.03.025 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2009.07.106 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.ejmech.2009.11.009 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.06.063 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.05.056 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.06.056 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.10.061 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.02.052 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.054 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
2.0 |
ug.mL-1 |
10.1021/jm9509556 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
3.13 |
ug.mL-1 |
10.1016/j.bmcl.2004.07.064 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
4.0 |
ug.mL-1 |
10.1021/jm070708p |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
3000.0 |
nM |
10.1016/j.bmcl.2004.08.059 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
3100.0 |
nM |
10.1021/jm501174m |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
4629.0 |
nM |
10.1016/j.bmcl.2009.04.133 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00344-06 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.00666-06 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm201467r |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00344-06 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00400-09 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00666-06 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01047-08 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm201467r |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/jm960294s |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00723-10 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01017-06 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01326-07 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
PD50 |
3.0 |
mg kg-1 |
10.1016/j.bmcl.2010.11.022 |
| Streptococcus pyogenes serotype M1 |
Streptokinase A |
EC50 |
158.0 |
nM |
None |
| Streptococcus pyogenes serotype M1 |
Streptokinase A |
EC50 |
5998.0 |
nM |
None |
| Streptococcus salivarius |
Streptococcus salivarius |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus salivarius |
Streptococcus salivarius |
Inhibition |
1.1 |
% |
10.1128/aac.01496-06 |
| Streptococcus salivarius |
Streptococcus salivarius |
Inhibition |
3.3 |
% |
10.1128/aac.01496-06 |
| Streptococcus salivarius |
Streptococcus salivarius |
Inhibition |
46.2 |
% |
10.1128/aac.01496-06 |
| Streptococcus salivarius |
Streptococcus salivarius |
Inhibition |
98.9 |
% |
10.1128/aac.01496-06 |
| Streptococcus salivarius |
Streptococcus salivarius |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus salivarius |
Streptococcus salivarius |
MBC |
25.0 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Streptococcus salivarius |
Streptococcus salivarius |
MIC100 |
3.13 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Streptococcus salivarius |
Streptococcus salivarius |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus salivarius |
Streptococcus salivarius |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus sanguinis |
Streptococcus sanguinis |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus sanguinis |
Streptococcus sanguinis |
Inhibition |
0.7 |
% |
10.1128/aac.01496-06 |
| Streptococcus sanguinis |
Streptococcus sanguinis |
Inhibition |
4.2 |
% |
10.1128/aac.01496-06 |
| Streptococcus sanguinis |
Streptococcus sanguinis |
Inhibition |
36.6 |
% |
10.1128/aac.01496-06 |
| Streptococcus sanguinis |
Streptococcus sanguinis |
Inhibition |
97.9 |
% |
10.1128/aac.01496-06 |
| Streptococcus sanguinis |
Streptococcus sanguinis |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| Streptococcus sanguinis |
Streptococcus sanguinis |
MIC |
0.06 |
ug.mL-1 |
10.1021/jm401931e |
| Streptococcus sanguinis |
Streptococcus sanguinis |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus sanguinis |
Streptococcus sanguinis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus sanguinis |
Streptococcus sanguinis |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus sanguinis |
Streptococcus sanguinis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| Streptococcus sanguinis |
Streptococcus sanguinis |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus sp. |
Streptococcus sp. |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus sp. |
Streptococcus sp. |
MIC |
0.25 |
ug.mL-1 |
10.1016/s0960-894x(02)00043-4 |
| Streptococcus sp. |
Streptococcus sp. |
MIC |
0.5 |
ug.mL-1 |
10.1016/s0960-894x(02)00043-4 |
| Streptococcus sp. |
Streptococcus sp. |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus sp. |
Streptococcus sp. |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus sp. |
Streptococcus sp. |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
Activity |
100.0 |
% |
10.1128/aac.00129-09 |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
Activity |
100.0 |
% |
10.1128/aac.00845-09 |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
Activity |
nan |
None |
10.1128/aac.00129-09 |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
EC50 |
170.0 |
nM |
None |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Streptococcus sp. 'group A' |
Streptococcus sp. 'group A' |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
Activity |
100.0 |
% |
10.1128/aac.00129-09 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
Activity |
100.0 |
% |
10.1128/aac.00845-09 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
Activity |
nan |
None |
10.1128/aac.00129-09 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00129-09 |
| Streptococcus sp. 'group B' |
Streptococcus sp. 'group B' |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| Streptococcus viridans |
Streptococcus viridans |
Activity |
0.0 |
% |
10.1128/aac.00149-08 |
| Streptococcus viridans |
Streptococcus viridans |
Activity |
100.0 |
% |
10.1128/aac.00149-08 |
| Streptococcus viridans |
Streptococcus viridans |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| Streptococcus viridans |
Streptococcus viridans |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Streptococcus viridans |
Streptococcus viridans |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus viridans |
Streptococcus viridans |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus viridans |
Streptococcus viridans |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Streptococcus viridans |
Streptococcus viridans |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| Streptococcus viridans |
Streptococcus viridans |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Streptococcus viridans |
Streptococcus viridans |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Streptococcus viridans |
Streptococcus viridans |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus viridans |
Streptococcus viridans |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Streptococcus viridans |
Streptococcus viridans |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Streptococcus viridans |
Streptococcus viridans |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Streptococcus viridans |
Streptococcus viridans |
MIC50 |
nan |
None |
10.1128/aac.01398-07 |
| Streptococcus viridans |
Streptococcus viridans |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00100-07 |
| Streptococcus viridans |
Streptococcus viridans |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00149-08 |
| Streptococcus viridans |
Streptococcus viridans |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01315-06 |
| Streptococcus viridans |
Streptococcus viridans |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01197-09 |
| Streptococcus viridans |
Streptococcus viridans |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01569-09 |
| Streptococcus viridans |
Streptococcus viridans |
MIC90 |
nan |
None |
10.1128/aac.01398-07 |
| Thomasclavelia ramosa |
Thomasclavelia ramosa |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Thomasclavelia ramosa |
Thomasclavelia ramosa |
MIC50 |
8.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Thomasclavelia ramosa |
Thomasclavelia ramosa |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| Yersinia pestis |
Yersinia pestis |
MIC |
nan |
None |
10.1016/j.bmc.2015.02.016 |
| None |
ADMET |
Activity |
1.0 |
% |
10.1021/acs.jmedchem.5b02004 |
| None |
ADMET |
Activity |
20.83 |
g |
10.1021/acs.jmedchem.0c00500 |
| None |
ADMET |
Activity |
30.0 |
% |
10.1128/aac.00177-10 |
| None |
ADMET |
Activity |
67.0 |
ug ml-1 |
10.1073/pnas.0700746104 |
| None |
ADMET |
Activity |
nan |
None |
10.1016/j.ejmech.2013.03.069 |
| None |
ADMET |
AUC |
0.53 |
ug.hr/kg |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
AUC |
1.24 |
ug.hr/kg |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
AUC |
19.9 |
ug.hr/kg |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
AUC |
10100.0 |
ng.hr.mL-1 |
10.1128/aac.01022-09 |
| None |
ADMET |
AUC |
35400.0 |
ng.hr.mL-1 |
10.1128/aac.01022-09 |
| None |
ADMET |
AUC |
38200.0 |
ng.hr.mL-1 |
10.1128/aac.01022-09 |
| None |
ADMET |
AUC |
43000.0 |
ng.hr.mL-1 |
10.1128/aac.01022-09 |
| None |
ADMET |
AUC |
47700.0 |
ng.hr.mL-1 |
10.1128/aac.01022-09 |
| None |
ADMET |
AUC |
87800.0 |
ng.hr.mL-1 |
10.1128/aac.00775-08 |
| None |
ADMET |
AUC |
118700.0 |
ng.hr.mL-1 |
10.1128/aac.00775-08 |
| None |
ADMET |
AUC |
125800.0 |
ng.hr.mL-1 |
10.1128/aac.00775-08 |
| None |
ADMET |
CL |
0.0 |
mL.min-1.kg-1 |
10.1016/j.bmcl.2019.126746 |
| None |
ADMET |
CL |
0.0 |
mL.min-1.kg-1 |
10.1016/j.ejmech.2018.09.004 |
| None |
ADMET |
CL |
0.0 |
mL.min-1.kg-1 |
10.1016/j.ejmech.2019.111781 |
| None |
ADMET |
CL |
1.74 |
mL.min-1.kg-1 |
10.1016/j.bmc.2019.03.034 |
| None |
ADMET |
CL |
1.8 |
mL.min-1.kg-1 |
10.1124/dmd.108.020479 |
| None |
ADMET |
CL |
3.167 |
mL.min-1.kg-1 |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
CL |
9.333 |
mL.min-1.kg-1 |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
CL |
12.9 |
L/hr |
10.1128/aac.01022-09 |
| None |
ADMET |
CL |
13.7 |
L/hr |
10.1128/aac.01022-09 |
| None |
ADMET |
CL |
13.9 |
L/hr |
10.1128/aac.01022-09 |
| None |
ADMET |
CL |
14.9 |
L/hr |
10.1128/aac.01022-09 |
| None |
ADMET |
CL |
15.1 |
L/hr |
10.1128/aac.01022-09 |
| None |
ADMET |
CL |
17.2 |
L/hr |
10.1128/aac.01022-09 |
| None |
ADMET |
CL |
34.0 |
mL.min-1.kg-1 |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
Cmax |
4802.13 |
nM |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
Cmax |
12983.55 |
nM |
10.1128/aac.01022-09 |
| None |
ADMET |
Cmax |
14198.9 |
nM |
10.1128/aac.01022-09 |
| None |
ADMET |
Cmax |
20157.11 |
nM |
10.1128/aac.00775-08 |
| None |
ADMET |
Cmax |
25789.24 |
nM |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
Cmax |
37646.36 |
nM |
10.1016/j.bmc.2019.03.034 |
| None |
ADMET |
Cmax |
37646.36 |
nM |
10.1128/aac.00775-08 |
| None |
ADMET |
Cmax |
39721.36 |
nM |
10.1016/j.bmc.2019.03.034 |
| None |
ADMET |
Cmax |
39721.36 |
nM |
10.1128/aac.01022-09 |
| None |
ADMET |
Cmax |
43278.49 |
nM |
10.1128/aac.01022-09 |
| None |
ADMET |
Cmax |
53653.48 |
nM |
10.1128/aac.00775-08 |
| None |
ADMET |
Cmax |
56914.18 |
nM |
10.1128/aac.01022-09 |
| None |
ADMET |
Cmax |
57803.47 |
nM |
10.1128/aac.01022-09 |
| None |
ADMET |
Cmax |
80924.86 |
nM |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
Cmin |
2.5 |
ug ml-1 |
10.1128/aac.00775-08 |
| None |
ADMET |
Cmin |
3.0 |
ug ml-1 |
10.1128/aac.00775-08 |
| None |
ADMET |
Cmin |
3.7 |
ug ml-1 |
10.1128/aac.00775-08 |
| None |
ADMET |
Drugexcretion |
73.0 |
% |
10.1016/j.bmc.2012.08.023 |
| None |
ADMET |
Drug uptake |
0.31 |
ug ml-1 |
10.1128/aac.01022-09 |
| None |
ADMET |
Drug uptake |
0.39 |
ug ml-1 |
10.1128/aac.01022-09 |
| None |
ADMET |
Drug uptake |
1.15 |
ug ml-1 |
10.1128/aac.01022-09 |
| None |
ADMET |
Drug uptake |
1.17 |
ug ml-1 |
10.1128/aac.01022-09 |
| None |
ADMET |
Drug uptake |
1.26 |
ug ml-1 |
10.1128/aac.01022-09 |
| None |
ADMET |
Drug uptake |
1.42 |
ug ml-1 |
10.1128/aac.01022-09 |
| None |
ADMET |
Drug uptake |
20.0 |
% |
10.1021/jm800038g |
| None |
ADMET |
Drug uptake |
64.3 |
ug ml-1 |
10.1021/jm800038g |
| None |
ADMET |
Drug uptake |
nan |
None |
10.1021/acs.jmedchem.6b00372 |
| None |
ADMET |
Drug uptake |
nan |
None |
10.1021/acsmedchemlett.9b00379 |
| None |
ADMET |
F |
100.0 |
% |
10.1021/jm020248u |
| None |
ADMET |
F |
109.0 |
% |
10.1021/jm020248u |
| None |
ADMET |
F |
109.0 |
% |
10.1021/jm980546k |
| None |
ADMET |
Fabs |
1.03 |
None |
10.1016/j.bmc.2019.03.034 |
| None |
ADMET |
IC50 |
3.37 |
ug.mL-1 |
10.1128/aac.00247-07 |
| None |
ADMET |
IC50 |
6.3 |
ug.mL-1 |
10.1021/jm401931e |
| None |
ADMET |
IC50 |
213.0 |
ug.mL-1 |
10.1039/C5MD00101C |
| None |
ADMET |
IC50 |
215.0 |
ug.mL-1 |
10.1039/C5MD00101C |
| None |
ADMET |
IC50 |
465.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.09.019 |
| None |
ADMET |
MRT |
5.4 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
MRT |
6.55 |
hr |
10.1128/aac.01022-09 |
| None |
ADMET |
MRT |
6.81 |
hr |
10.1128/aac.01022-09 |
| None |
ADMET |
MRT |
7.95 |
hr |
10.1128/aac.01022-09 |
| None |
ADMET |
MRT |
8.1 |
hr |
10.1128/aac.01022-09 |
| None |
ADMET |
MRT |
8.65 |
hr |
10.1128/aac.01022-09 |
| None |
ADMET |
Papp |
6.9 |
10^-6 cm/s |
10.1021/acsmedchemlett.3c00032 |
| None |
ADMET |
Papp |
9.0 |
10^-6 cm/s |
10.1021/acsmedchemlett.3c00032 |
| None |
ADMET |
Papp |
295.3 |
nm/s |
10.1016/j.bmcl.2015.12.002 |
| None |
ADMET |
Papp |
516.4 |
nm/s |
10.1016/j.bmcl.2015.12.002 |
| None |
ADMET |
PPB |
22.38 |
% |
10.6019/CHEMBL3301361 |
| None |
ADMET |
PPB |
22.79 |
% |
10.6019/CHEMBL3301361 |
| None |
ADMET |
PPB |
23.19 |
% |
10.6019/CHEMBL3301361 |
| None |
ADMET |
PPB |
52.3 |
% |
10.6019/CHEMBL3301361 |
| None |
ADMET |
Ratio |
0.11 |
None |
10.1021/acsmedchemlett.5b00213 |
| None |
ADMET |
Ratio |
0.12 |
None |
10.1021/acsmedchemlett.5b00213 |
| None |
ADMET |
Ratio |
0.6 |
None |
10.1016/j.bmcl.2015.12.002 |
| None |
ADMET |
Ratio |
1.3 |
None |
10.1021/acsmedchemlett.3c00032 |
| None |
ADMET |
Stability |
18.0 |
% |
10.1016/j.bmcl.2019.126746 |
| None |
ADMET |
Stability |
100.0 |
% |
10.1021/acsmedchemlett.5b00213 |
| None |
ADMET |
Stability |
104.18 |
% |
10.1016/j.ejmech.2018.09.004 |
| None |
ADMET |
Stability |
104.18 |
% |
10.1016/j.ejmech.2019.111781 |
| None |
ADMET |
Stability |
110.9 |
% |
10.1021/acs.jmedchem.0c00500 |
| None |
ADMET |
Stability |
nan |
% |
10.1016/j.ejmech.2019.111781 |
| None |
ADMET |
Stability |
nan |
% |
10.1021/acs.jmedchem.0c00500 |
| None |
ADMET |
T1/2 |
1.3 |
hr |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
T1/2 |
2.23 |
hr |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
T1/2 |
2.6 |
hr |
10.1128/aac.00775-08 |
| None |
ADMET |
T1/2 |
3.5 |
hr |
10.1128/aac.00775-08 |
| None |
ADMET |
T1/2 |
3.613 |
hr |
10.1016/j.bmcl.2019.07.024 |
| None |
ADMET |
T1/2 |
4.4 |
hr |
10.1016/j.bmc.2019.03.034 |
| None |
ADMET |
T1/2 |
4.5 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
T1/2 |
5.01 |
hr |
10.1128/aac.01022-09 |
| None |
ADMET |
T1/2 |
5.2 |
hr |
10.1128/aac.01022-09 |
| None |
ADMET |
T1/2 |
5.32 |
hr |
10.1128/aac.01194-06 |
| None |
ADMET |
T1/2 |
6.18 |
hr |
10.1128/aac.01022-09 |
| None |
ADMET |
T1/2 |
6.27 |
hr |
10.1128/aac.01022-09 |
| None |
ADMET |
T1/2 |
6.54 |
hr |
10.1128/aac.01022-09 |
| None |
ADMET |
T1/2 |
6.72 |
hr |
10.1128/aac.01022-09 |
| None |
ADMET |
T1/2 |
6.8 |
hr |
10.1128/aac.00775-08 |
| None |
ADMET |
T1/2 |
67.6 |
hr |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
T1/2 |
100.0 |
hr |
10.1016/j.bmcl.2015.12.002 |
| None |
ADMET |
Tmax |
0.5 |
hr |
10.1016/j.bmc.2019.03.034 |
| None |
ADMET |
Tmax |
0.5 |
hr |
10.1128/aac.01022-09 |
| None |
ADMET |
Tmax |
1.33 |
hr |
10.1016/j.bmc.2019.03.034 |
| None |
ADMET |
Tmax |
2.8 |
hr |
10.1128/aac.00775-08 |
| None |
ADMET |
Tmax |
3.0 |
hr |
10.1128/aac.00775-08 |
| None |
ADMET |
Tmax |
3.3 |
hr |
10.1128/aac.00775-08 |
| None |
ADMET |
Vd |
0.4 |
L.kg-1 |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
Vd |
0.58 |
L.kg-1 |
10.1016/j.bmc.2019.03.034 |
| None |
ADMET |
Vd |
17.82 |
L.kg-1 |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
Vd |
78.24 |
L.kg-1 |
10.1016/j.bmcl.2022.128842 |
| None |
ADMET |
Vd |
102.2 |
l |
10.1128/aac.01022-09 |
| None |
ADMET |
Vd |
114.9 |
l |
10.1128/aac.01022-09 |
| None |
ADMET |
Vd |
124.5 |
l |
10.1128/aac.01022-09 |
| None |
ADMET |
Vd |
129.7 |
l |
10.1128/aac.01022-09 |
| None |
ADMET |
Vd |
136.7 |
l |
10.1128/aac.01022-09 |
| None |
ADMET |
Vd |
140.7 |
l |
10.1128/aac.01022-09 |
| None |
ADMET |
Vdss |
0.58 |
L.kg-1 |
10.1124/dmd.108.020479 |
| None |
ADMET |
Vdss |
89.3 |
l |
10.1128/aac.01022-09 |
| None |
ADMET |
Vdss |
100.2 |
l |
10.1128/aac.01022-09 |
| None |
ADMET |
Vdss |
103.9 |
l |
10.1128/aac.01022-09 |
| None |
ADMET |
Vdss |
112.1 |
l |
10.1128/aac.01022-09 |
| None |
ADMET |
Vdss |
116.9 |
l |
10.1128/aac.01022-09 |
| None |
ADMET |
Vdss |
119.7 |
l |
10.1128/aac.01022-09 |
| None |
Erythrocyte |
Activity |
1.0 |
% |
10.1021/acs.jmedchem.7b01903 |
| None |
Erythrocyte |
Activity |
1.0 |
% |
10.1039/C6MD00381H |
| None |
Erythrocyte |
HC50 |
550.0 |
ug ml-1 |
10.1016/j.ejmech.2018.06.054 |
| None |
Hepatotoxicity |
HepSE_bilirubinemia |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholecystitis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholelithiasis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cirrhosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_Combined Scores |
2.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_elevated liver function tests |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic failure |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic necrosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatitis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatomegaly |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_jaundice |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver disease |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver fatty |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver function tests abnormal |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Molecular identity unknown |
PPB |
17.8 |
% |
10.1016/j.bmcl.2015.12.002 |
| None |
Molecular identity unknown |
PPB |
26.04 |
% |
10.1021/acsmedchemlett.5b00213 |
| None |
NON-PROTEIN TARGET |
Activity |
11.0 |
% |
10.1128/aac.00696-08 |
| None |
NON-PROTEIN TARGET |
Activity |
100.0 |
% |
10.1128/aac.00845-09 |
| None |
NON-PROTEIN TARGET |
Activity |
100.0 |
% |
10.1128/aac.01398-07 |
| None |
NON-PROTEIN TARGET |
fT>MIC |
62.8 |
% |
10.1128/aac.01378-08 |
| None |
NON-PROTEIN TARGET |
fT>MIC |
100.0 |
% |
10.1128/aac.01378-08 |
| None |
NON-PROTEIN TARGET |
Fu |
0.69 |
None |
10.1124/dmd.108.020479 |
| None |
NON-PROTEIN TARGET |
Fu |
0.69 |
None |
10.1128/aac.00197-09 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (acute) |
0.0 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (animal toxicity known) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (benign tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (granulomatous hepatitis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (mechanism) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
1.0 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (time to onset) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
IC20 |
240.0 |
ug ml-1 |
10.1128/aac.00729-05 |
| None |
NON-PROTEIN TARGET |
IC50 |
12.8 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.024 |
| None |
NON-PROTEIN TARGET |
IC50 |
400.0 |
ug.mL-1 |
10.1128/aac.00729-05 |
| None |
NON-PROTEIN TARGET |
Inhibition |
0.0 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
2.9 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
4.5 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
5.6 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
7.7 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
16.7 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
31.8 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
33.7 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
36.4 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
46.2 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
57.1 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
63.6 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
83.3 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
94.4 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
96.2 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
Inhibition |
100.0 |
% |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
MIC |
6e-05 |
ug.mL-1 |
10.1128/aac.01102-06 |
| None |
NON-PROTEIN TARGET |
MIC |
0.00025 |
ug.mL-1 |
10.1128/aac.01102-06 |
| None |
NON-PROTEIN TARGET |
MIC |
0.12 |
ug.mL-1 |
10.1128/aac.00336-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm401931e |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00228-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00336-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2004.05.066 |
| None |
NON-PROTEIN TARGET |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00090-09 |
| None |
NON-PROTEIN TARGET |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.01398-07 |
| None |
NON-PROTEIN TARGET |
MIC |
0.8 |
ug.mL-1 |
10.1016/j.bmc.2014.10.037 |
| None |
NON-PROTEIN TARGET |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2004.02.047 |
| None |
NON-PROTEIN TARGET |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| None |
NON-PROTEIN TARGET |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| None |
NON-PROTEIN TARGET |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| None |
NON-PROTEIN TARGET |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| None |
NON-PROTEIN TARGET |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00169-10 |
| None |
NON-PROTEIN TARGET |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| None |
NON-PROTEIN TARGET |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| None |
NON-PROTEIN TARGET |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2015.02.016 |
| None |
NON-PROTEIN TARGET |
MIC |
64.0 |
ug.mL-1 |
10.1128/aac.01383-07 |
| None |
NON-PROTEIN TARGET |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| None |
NON-PROTEIN TARGET |
MIC |
128.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.5 |
ug.mL-1 |
10.1021/jm401931e |
| None |
NON-PROTEIN TARGET |
MIC50 |
0.5 |
ug.mL-1 |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| None |
NON-PROTEIN TARGET |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| None |
NON-PROTEIN TARGET |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| None |
NON-PROTEIN TARGET |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
MIC50 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| None |
NON-PROTEIN TARGET |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| None |
NON-PROTEIN TARGET |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| None |
NON-PROTEIN TARGET |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| None |
NON-PROTEIN TARGET |
MIC50 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
128.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC50 |
256.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| None |
NON-PROTEIN TARGET |
MIC90 |
1.0 |
ug.mL-1 |
10.1021/jm401931e |
| None |
NON-PROTEIN TARGET |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
MIC90 |
1.0 |
ug.mL-1 |
10.1128/aac.01641-07 |
| None |
NON-PROTEIN TARGET |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00336-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00845-09 |
| None |
NON-PROTEIN TARGET |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01398-07 |
| None |
NON-PROTEIN TARGET |
MIC90 |
2.0 |
ug.mL-1 |
10.1128/aac.01496-06 |
| None |
NON-PROTEIN TARGET |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| None |
NON-PROTEIN TARGET |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00228-09 |
| None |
NON-PROTEIN TARGET |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
4.0 |
ug.mL-1 |
10.1128/aac.01352-06 |
| None |
NON-PROTEIN TARGET |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00696-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
8.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
16.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
128.0 |
ug.mL-1 |
10.1128/aac.00908-08 |
| None |
NON-PROTEIN TARGET |
MIC90 |
256.0 |
ug.mL-1 |
10.1128/aac.00090-09 |
| None |
No relevant target |
CLogP |
0.01 |
None |
10.1016/s0960-894x(99)00474-6 |
| None |
No relevant target |
CLogP |
0.58 |
None |
10.1016/j.bmcl.2004.08.059 |
| None |
No relevant target |
Drug degradation |
1.0 |
% |
10.1021/acs.jmedchem.1c00790 |
| None |
No relevant target |
Drug degradation |
40.0 |
% |
10.1021/acs.jmedchem.1c00790 |
| None |
No relevant target |
LogD |
-1.38 |
None |
10.1021/acsmedchemlett.3c00032 |
| None |
No relevant target |
LogD |
0.7 |
None |
10.1021/acs.jmedchem.5b00050 |
| None |
No relevant target |
LogD7.4 |
0.67 |
None |
10.6019/CHEMBL3301361 |
| None |
No relevant target |
LogP |
0.48 |
None |
10.1039/C5MD00101C |
| None |
No relevant target |
LogP |
0.5321 |
None |
10.1016/j.ejmech.2008.07.005 |
| None |
No relevant target |
pKa |
6.0 |
None |
10.1021/acs.jmedchem.1c00790 |
| None |
No relevant target |
pKa |
nan |
None |
10.1021/acs.jmedchem.5b02004 |
| None |
No relevant target |
pKa_B1 |
6.81 |
None |
10.6019/CHEMBL3301361 |
| None |
No relevant target |
solubility |
nan |
None |
10.1021/acs.jmedchem.5b02004 |
| None |
No relevant target |
Solubility |
67.47 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.024 |
| None |
No relevant target |
Solubility |
125.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.126747 |
| None |
No relevant target |
Solubility |
49000.0 |
nM |
10.1021/acsmedchemlett.5b00213 |
| None |
No relevant target |
Solubility |
50000.0 |
nM |
10.1021/acsmedchemlett.5b00213 |
| None |
No relevant target |
Solubility |
1000000.0 |
nM |
10.1021/acs.jmedchem.5b00050 |
| None |
No relevant target |
Solubility |
1000000.0 |
nM |
10.1021/jm501174m |
| None |
No relevant target |
Solubility |
7559000.0 |
nM |
10.1039/C5MD00101C |
| None |
No relevant target |
Solubility |
8800000.0 |
nM |
10.1021/acsmedchemlett.3c00032 |
| None |
No relevant target |
Stability |
98.0 |
% |
10.1016/j.bmcl.2019.07.024 |
| None |
No relevant target |
Stability |
nan |
% |
10.1128/aac.00633-09 |
| None |
Osteoblast |
Activity |
13.0 |
% |
10.1128/aac.00729-05 |
| None |
Osteoblast |
Activity |
120.0 |
% |
10.1128/aac.00729-05 |
| None |
Osteoblast |
IC20 |
400.0 |
ug ml-1 |
10.1128/aac.00729-05 |
| None |
Osteoblast |
IC50 |
400.0 |
ug.mL-1 |
10.1128/aac.00729-05 |
| None |
Ribosome |
IC50 |
11900000.0 |
nM |
10.1128/aac.00887-08 |
| None |
Unchecked |
Ac50 |
0.7079 |
uM |
None |
| None |
Unchecked |
Ac50 |
1.259 |
uM |
None |
| None |
Unchecked |
Ac50 |
12.59 |
uM |
None |
| None |
Unchecked |
AC50 |
707.9 |
nM |
None |
| None |
Unchecked |
AC50 |
1260.0 |
nM |
None |
| None |
Unchecked |
AC50 |
12589.3 |
nM |
None |
| None |
Unchecked |
Activity |
nan |
None |
10.1016/j.ejmech.2022.114495 |
| None |
Unchecked |
deltaTm |
nan |
None |
10.1016/j.bmc.2015.02.016 |
| None |
Unchecked |
fAUC/MIC |
1.8 |
None |
10.1128/aac.00833-08 |
| None |
Unchecked |
fAUC/MIC |
2.6 |
None |
10.1128/aac.00833-08 |
| None |
Unchecked |
fAUC/MIC |
3.3 |
None |
10.1128/aac.00833-08 |
| None |
Unchecked |
fAUC/MIC |
3.6 |
None |
10.1128/aac.00833-08 |
| None |
Unchecked |
fAUC/MIC |
5.3 |
None |
10.1128/aac.00833-08 |
| None |
Unchecked |
fAUC/MIC |
6.6 |
None |
10.1128/aac.00833-08 |
| None |
Unchecked |
fAUC/MIC |
449.0 |
None |
10.1128/aac.00642-09 |
| None |
Unchecked |
fAUC/MIC |
898.0 |
None |
10.1128/aac.00642-09 |
| None |
Unchecked |
Hepatotoxicity (acute) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (association with vascular disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (choleostasis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (chronic liver disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cirrhosis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (comment) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cytolytic) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (malignant tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (severe hepatitis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (steatosis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (successful reintroduction) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
IC50 |
900.0 |
nM |
10.1128/aac.01193-07 |
| None |
Unchecked |
IC50 |
2400.0 |
nM |
10.1021/acs.jmedchem.5b00050 |
| None |
Unchecked |
IC50 |
7980.0 |
nM |
10.1021/acs.jmedchem.0c00500 |
| None |
Unchecked |
IC50 |
8400.0 |
nM |
10.1128/aac.01193-07 |
| None |
Unchecked |
IC50 |
100000.0 |
nM |
10.1128/aac.00887-08 |
| None |
Unchecked |
IC50 |
100000.0 |
nM |
10.1128/aac.01193-07 |
| None |
Unchecked |
IC50 |
nan |
nM |
10.1016/j.bmcl.2003.07.028 |
| None |
Unchecked |
IC50 |
nan |
None |
10.1016/j.bmc.2015.07.062 |
| None |
Unchecked |
Inhibition |
15.0 |
% |
10.1016/j.ejmech.2016.09.007 |
| None |
Unchecked |
Inhibition |
70.7 |
% |
10.1016/j.ejmech.2021.113402 |
| None |
Unchecked |
Inhibition |
70.7 |
% |
10.1039/D1MD00230A |
| None |
Unchecked |
Inhibition |
nan |
% |
10.1016/j.bmc.2015.02.016 |
| None |
Unchecked |
Inhibition |
nan |
% |
10.1016/j.bmc.2020.115729 |
| None |
Unchecked |
Inhibition |
nan |
% |
10.1021/acs.jmedchem.9b00616 |
| None |
Unchecked |
Inhibition |
nan |
% |
10.1039/C6MD00236F |
| None |
Unchecked |
Inhibition |
nan |
% |
10.1128/aac.00620-10 |
| None |
Unchecked |
Kd |
nan |
None |
10.1016/j.bmc.2015.07.062 |
| None |
Unchecked |
MIC |
1.0 |
ug.mL-1 |
10.1021/acs.jmedchem.9b00616 |
| None |
Unchecked |
MIC |
nan |
None |
10.1021/acsmedchemlett.0c00653 |
| None |
Unchecked |
MIC100 |
0.87 |
ug ml-1 |
10.1016/j.ejmech.2020.112420 |
| None |
Unchecked |
Potency |
2238.7 |
nM |
None |
| None |
Unchecked |
Potency |
12995.3 |
nM |
None |
| None |
Unchecked |
Ratio |
1.0 |
None |
10.1016/j.ejmech.2020.113002 |
| None |
Unchecked |
Ratio |
2.7 |
None |
10.1128/aac.00775-08 |
| None |
Unchecked |
Ratio |
4.0 |
None |
10.1021/acs.jmedchem.0c00500 |
| None |
Unchecked |
Ratio |
5.1 |
None |
10.1128/aac.00775-08 |
| None |
Unchecked |
Ratio |
7.2 |
None |
10.1128/aac.00775-08 |
| None |
Unchecked |
Ratio |
8.0 |
None |
10.1016/j.ejmech.2018.06.054 |
| None |
Unchecked |
Ratio |
16.2 |
None |
10.1128/aac.01378-08 |
| None |
Unchecked |
Ratio |
20.0 |
None |
10.1128/aac.01378-08 |
| None |
Unchecked |
Ratio |
35.1 |
None |
10.1128/aac.00775-08 |
| None |
Unchecked |
Ratio |
47.5 |
None |
10.1128/aac.00775-08 |
| None |
Unchecked |
Ratio |
50.3 |
None |
10.1128/aac.00775-08 |
| None |
Unchecked |
Ratio |
118.0 |
None |
10.1128/aac.00887-08 |
| None |
Unchecked |
RatioAUC/MIC |
107.8 |
None |
10.1128/aac.01378-08 |
| None |
Unchecked |
RatioAUC/MIC |
116.2 |
None |
10.1128/aac.01378-08 |
| None |
Unchecked |
RatioAUC/MIC |
121.6 |
None |
10.1128/aac.01378-08 |
| None |
Unchecked |
RatioAUC/MIC |
243.2 |
None |
10.1128/aac.01378-08 |
| None |
Unchecked |
Ratio IC50 |
12.0 |
None |
10.1021/acs.jmedchem.2c01349 |
| None |
Unchecked |
Ratio IC50 |
15.0 |
None |
10.1021/acs.jmedchem.2c01349 |
| None |
Unchecked |
Selectivity Index |
197.0 |
None |
10.1021/acsmedchemlett.7b00068 |
| None |
Unchecked |
Selectivity Index |
333.0 |
None |
10.1016/j.bmc.2018.07.034 |
| None |
Unchecked |
Time |
nan |
None |
10.1128/aac.00620-10 |
| None |
Unchecked |
TIME |
0.005556 |
hr |
10.1128/aac.00620-10 |