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name Structure Reference Source Properties Activities Metabolism

efavirenz

AlkaPlorer ID: AK043601

Synonym: None

IUPAC Name: (4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluoromethyl)-1H-3,1-benzoxazin-2-one

Structure

SMILES: OC1=NC2=CC=C(Cl)C=C2[C@@](C#CC2CC2)(C(F)(F)F)O1

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InChI: InChI=1S/C14H9ClF3NO2/c15-9-3-4-11-10(7-9)13(14(16,17)18,21-12(20)19-11)6-5-8-1-2-8/h3-4,7-8H,1-2H2,(H,19,20)/t13-/m0/s1

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InChIKey: XPOQHMRABVBWPR-ZDUSSCGKSA-N

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Reference

PubChem CID: 64139

CAS: 154598-52-4

SuperNatural Ⅲ: SN0436588-01

NPASS: NPC168951

Properties Information

Molecule Weight: 315.67799999999994

TPSA？: 41.82000000000001

MolLogP？: 4.086700000000001

Number of H-Donors: 1

Number of H-Acceptors: 2

RingCount: 3

Activities Information

Organism Target Name Standard Type Standard Value Standard Units doi
Acinetobacter baumannii Acinetobacter baumannii Inhibition 17.76 % 10.6019/CHEMBL4513141
Bovine viral diarrhea virus 1 Bovine viral diarrhea virus 1 EC50 nan None 10.1016/j.bmc.2015.09.035
Candida albicans Candida albicans Inhibition 3.86 % 10.6019/CHEMBL4513141
Canis lupus familiaris Canis familiaris F nan % 10.1016/j.bmcl.2010.01.085
Canis lupus familiaris Canis familiaris F nan % 10.1016/j.bmcl.2010.01.086
Canis lupus familiaris Canis familiaris t1/2 nan None 10.1016/j.bmcl.2010.01.085
Canis lupus familiaris Canis familiaris t1/2 nan None 10.1016/j.bmcl.2010.01.086
Canis lupus familiaris Canis familiaris Vdss nan None 10.1016/j.bmcl.2010.01.085
Canis lupus familiaris Canis familiaris Vdss nan None 10.1016/j.bmcl.2010.01.086
Chlorocebus sabaeus Vero CC50 100000.0 nM 10.1016/j.bmcl.2016.06.065
Chlorocebus sabaeus Vero CC50 nan None 10.1007/s00044-007-9004-0
Coxsackievirus B5 Coxsackievirus B5 EC50 nan None 10.1016/j.bmc.2015.09.035
Cryptococcus neoformans Cryptococcus neoformans Inhibition -5.8 % 10.6019/CHEMBL4513141
Equus caballus Ferritin light chain Potency 31622.8 nM None
Escherichia coli Escherichia coli Inhibition -2.05 % 10.6019/CHEMBL4513141
Homo sapiens A-375 Activity 51.0 % 10.1021/jm200734j
Homo sapiens A-375 Activity nan None 10.1021/jm200734j
Homo sapiens A-375 Inhibition 51.0 % 10.1021/jm0507330
Homo sapiens Adenosine A1 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Adenosine A2a receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Adenosine A3 receptor AC50 5999.2 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-1a adrenergic receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-1a adrenergic receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-2a adrenergic receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-2b adrenergic receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Alpha-2c adrenergic receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens ATP-binding cassette sub-family G member 2 Activity nan None 10.1128/aac.01527-10
Homo sapiens ATP-binding cassette sub-family G member 2 IC50 20600.0 nM 10.1016/j.ejmech.2022.114346
Homo sapiens ATP-binding cassette sub-family G member 2 Inhibition nan % 10.1128/aac.01527-10
Homo sapiens Beta-1 adrenergic receptor AC50 18999.8 nM 10.1038/s41467-023-40064-9
Homo sapiens Beta-2 adrenergic receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Bile salt export pump AC50 109999.3 nM 10.1038/s41467-023-40064-9
Homo sapiens Bile salt export pump IC50 133000.0 nM 10.1093/toxsci/kft176
Homo sapiens Bradykinin B2 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens C8166 EC90 0.008 uM 10.1021/jm031147e
Homo sapiens C8166 EC90 0.008 uM 10.1021/jm040854k
Homo sapiens C8166 EC90 1.8 uM 10.1021/jm040854k
Homo sapiens C8166 TC50 1.0 uM 10.1021/jm801395v
Homo sapiens Canalicular multispecific organic anion transporter 1 Activity nan None 10.1038/nrd3028
Homo sapiens Canalicular multispecific organic anion transporter 1 Activity nan None 10.1124/dmd.106.012765
Homo sapiens Canalicular multispecific organic anion transporter 1 Activity nan None 10.1128/aac.01527-10
Homo sapiens Canalicular multispecific organic anion transporter 1 IC50 133000.0 nM 10.1093/toxsci/kft176
Homo sapiens Canalicular multispecific organic anion transporter 2 Activity nan None 10.1038/nrd3028
Homo sapiens Canalicular multispecific organic anion transporter 2 Activity nan None 10.1124/dmd.106.012765
Homo sapiens Canalicular multispecific organic anion transporter 2 Activity nan None 10.1128/aac.01527-10
Homo sapiens Canalicular multispecific organic anion transporter 2 IC50 133000.0 nM 10.1093/toxsci/kft176
Homo sapiens Cannabinoid CB1 receptor AC50 20668.1 nM 10.1038/s41467-023-40064-9
Homo sapiens Cannabinoid CB1 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens CCRF-CEM CC50 100000.0 nM 10.1016/j.bmcl.2016.06.065
Homo sapiens CCRF-CEM CC50 200000.0 nM 10.1016/j.bmcl.2005.07.046
Homo sapiens CCRF-CEM CC50 10000000.0 nM 10.1021/jm101614j
Homo sapiens CEM-SS CC50 550.0 nM 10.1039/C4MD00282B
Homo sapiens CEM-SS CC50 nan None 10.1016/j.bmc.2016.05.010
Homo sapiens CEM-SS TC50 1.0 uM 10.1016/j.bmcl.2010.09.034
Homo sapiens Cholecystokinin A receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Cholecystokinin B receptor AC50 44999.7 nM 10.1038/s41467-023-40064-9
Homo sapiens Cholesterol 24-hydroxylase Activity nan None 10.1021/acs.jmedchem.9b01383
Homo sapiens Cholesterol 24-hydroxylase FC 4.1 None 10.1021/acs.jmedchem.9b01383
Homo sapiens Cholesterol 24-hydroxylase FC 4.9 None 10.1021/acs.jmedchem.9b01383
Homo sapiens Cholesterol 24-hydroxylase Inhibition nan % 10.1021/acs.jmedchem.9b01383
Homo sapiens Cholesterol 24-hydroxylase K 2.2 10'6/M/s 10.1021/acs.jmedchem.9b01383
Homo sapiens Cholesterol 24-hydroxylase K 11.2 /s 10.1021/acs.jmedchem.9b01383
Homo sapiens Cholesterol 24-hydroxylase Kd 800.0 nM 10.1021/acs.jmedchem.9b01383
Homo sapiens Cholesterol 24-hydroxylase Kd 5000.0 nM 10.1021/acs.jmedchem.9b01383
Homo sapiens Cholesterol 24-hydroxylase Kd 10200.0 nM 10.1021/acs.jmedchem.9b01383
Homo sapiens Cyclooxygenase-2 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Cytochrome P450 2B6 Activity nan None None
Homo sapiens Cytochrome P450 2B6 Drug metabolism nan None 10.1124/dmd.112.049601
Homo sapiens Cytochrome P450 2B6 Inhibition 95.0 % 10.1021/ml500297n
Homo sapiens Cytochrome P450 2B6 K 0.023 /min 10.1021/ml500297n
Homo sapiens Cytochrome P450 2B6 Km 450.0 nM 10.1021/ml500297n
Homo sapiens Cytochrome P450 2B6 Vmax 1.0 pmol/min 10.1021/ml500297n
Homo sapiens Cytochrome P450 2C8 Drug metabolism nan None 10.1124/dmd.112.049601
Homo sapiens Cytochrome P450 3A Activity 76.0 % 10.1021/acs.jmedchem.0c02245
Homo sapiens Cytochrome P450 3A4 Activity nan None None
Homo sapiens Delta opioid receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine D1 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine D2 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine D3 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Dopamine transporter AC50 17999.9 nM 10.1038/s41467-023-40064-9
Homo sapiens Endothelin receptor ET-A AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Equilibrative nucleoside transporter 1 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Estrogen receptor alpha AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Ghrelin receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Glucocorticoid receptor AC50 2710.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Glucocorticoid receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens HEK293 CC50 10000.0 nM 10.1016/j.bmcl.2006.01.066
Homo sapiens HEK293 CC50 10000.0 nM 10.1016/j.bmcl.2006.01.073
Homo sapiens HEK293 CC50 10000.0 nM 10.1016/j.bmcl.2006.05.073
Homo sapiens HEK293 IC50 40600.0 nM 10.1016/j.ejmech.2020.112790
Homo sapiens HEK-293T Activity nan None 10.1016/j.ejmech.2014.07.072
Homo sapiens HEK-293T CC50 30000.0 nM 10.1016/j.ejmech.2020.112071
Homo sapiens HeLa EC50 0.4 nM 10.1016/j.bmcl.2006.06.048
Homo sapiens HeLa EC50 11.0 nM 10.1016/j.bmcl.2006.06.048
Homo sapiens HeLa EC50 73.0 nM 10.1016/j.bmcl.2006.06.048
Homo sapiens HeLa IC50 0.5 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 0.8 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 0.9 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 1.0 nM 10.1021/jm040072r
Homo sapiens HeLa IC50 1.2 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 1.4 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 1.4 nM 10.1021/jm040072r
Homo sapiens HeLa IC50 1.5 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 1.8 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 2.0 nM 10.1021/jm040072r
Homo sapiens HeLa IC50 3.0 nM 10.1021/jm040072r
Homo sapiens HeLa IC50 3.3 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 6.4 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 7.0 nM 10.1021/jm040072r
Homo sapiens HeLa IC50 23.0 nM 10.1021/jm040072r
Homo sapiens HeLa IC50 24.0 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 42.0 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 43.0 nM 10.1021/jm040072r
Homo sapiens HeLa IC50 74.0 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 74.0 nM 10.1021/jm040072r
Homo sapiens HeLa IC50 130.0 nM 10.1021/jm0004906
Homo sapiens HeLa IC50 552.0 nM 10.1021/jm040072r
Homo sapiens HeLa IC50 1600.0 nM 10.1021/jm0004906
Homo sapiens Hepatocyte t1/2 nan None 10.1021/jm801322h
Homo sapiens HERG AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Histamine H1 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Histamine H2 receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Histamine H3 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Histone deacetylase 6 Inhibition -3.53 % 10.6019/CHEMBL4808148
Homo sapiens Histone deacetylase 6 Inhibition 7.2 % 10.6019/CHEMBL4808148
Homo sapiens Homo sapiens Activity nan None 10.1128/aac.00283-10
Homo sapiens Homo sapiens AUC 47.72 None 10.1128/aac.00283-10
Homo sapiens Homo sapiens AUC 97.46 None 10.1128/aac.00283-10
Homo sapiens Homo sapiens AUC 60000.0 ng.hr.mL-1 10.1128/aac.01594-08
Homo sapiens Homo sapiens AUC 63600.0 ng.hr.mL-1 10.1128/aac.01594-08
Homo sapiens Homo sapiens AUC 65200.0 ng.hr.mL-1 10.1128/aac.01594-08
Homo sapiens Homo sapiens CL/F 3.167 mL.min-1.kg-1 10.1128/aac.01594-08
Homo sapiens Homo sapiens CL/F 3.5 mL.min-1.kg-1 10.1128/aac.01594-08
Homo sapiens Homo sapiens CL/F 5.0 mL.min-1.kg-1 10.1128/aac.01594-08
Homo sapiens Homo sapiens CL/F 9.22 L/hr 10.1128/aac.01537-08
Homo sapiens Homo sapiens CL/F 70.67 ml/min 10.1128/aac.00283-10
Homo sapiens Homo sapiens CL/F 147.5 ml/min 10.1128/aac.00283-10
Homo sapiens Homo sapiens Cmax 8663.84 nM 10.1128/aac.00283-10
Homo sapiens Homo sapiens Cmax 11752.41 nM 10.1128/aac.01594-08
Homo sapiens Homo sapiens Cmax 11904.46 nM 10.1128/aac.00283-10
Homo sapiens Homo sapiens Cmax 12956.16 nM 10.1128/aac.01594-08
Homo sapiens Homo sapiens Cmax 17486.06 nM 10.1128/aac.01594-08
Homo sapiens Homo sapiens Cmin 1.18 mg/L 10.1128/aac.01594-08
Homo sapiens Homo sapiens Cmin 1.29 mg/L 10.1128/aac.01594-08
Homo sapiens Homo sapiens Cmin 1.45 mg/L 10.1128/aac.01594-08
Homo sapiens Homo sapiens Cmin 1.64 mg/L 10.1128/aac.01594-08
Homo sapiens Homo sapiens DILI_Concern nan None 10.1016/j.drudis.2016.02.015
Homo sapiens Homo sapiens DILI_severity_class 7.0 None 10.1016/j.drudis.2016.02.015
Homo sapiens Homo sapiens Free 0.5 % 10.1021/jm990580e
Homo sapiens Homo sapiens T1/2 33.0 hr 10.1128/aac.00283-10
Homo sapiens Homo sapiens T1/2 40.0 hr 10.1016/j.ejmech.2015.11.025
Homo sapiens Homo sapiens T1/2 52.0 hr 10.1016/j.ejmech.2015.11.025
Homo sapiens Homo sapiens T1/2 78.7 hr 10.1128/aac.00283-10
Homo sapiens Homo sapiens Tmax 2.2 hr 10.1128/aac.00283-10
Homo sapiens Homo sapiens Tmax 2.3 hr 10.1128/aac.00283-10
Homo sapiens Homo sapiens Tmax 5.0 hr 10.1016/j.ejmech.2015.11.025
Homo sapiens Homo sapiens Vc/F 295.0 l 10.1128/aac.01537-08
Homo sapiens Homo sapiens Vd 401.6 l 10.1128/aac.00283-10
Homo sapiens Homo sapiens Vd 462.8 l 10.1128/aac.00283-10
Homo sapiens Kappa opioid receptor AC50 4854.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Liver microsome Drug metabolism nan None 10.1124/dmd.112.049601
Homo sapiens Liver microsomes t1/2 nan None 10.1021/jm801322h
Homo sapiens MAP kinase ERK2 Potency 15848.9 nM None
Homo sapiens Melanocortin receptor 3 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Melanocortin receptor 4 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Microtubule-associated protein tau Potency 28183.8 nM None
Homo sapiens Monoamine oxidase A AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Motilin receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens MT2 CC50 100.0 nM 10.1016/j.bmcl.2006.08.037
Homo sapiens MT2 CC50 100.0 nM 10.1016/j.bmcl.2010.03.006
Homo sapiens MT2 CC50 3000.0 nM 10.1021/jm070683u
Homo sapiens MT2 CC50 15000.0 nM 10.1016/j.bmc.2016.07.039
Homo sapiens MT2 CC50 15000.0 nM 10.1016/j.bmcl.2012.11.115
Homo sapiens MT2 CC50 15000.0 nM 10.1016/j.bmcl.2013.06.091
Homo sapiens MT2 CC50 15000.0 nM 10.1016/j.bmcl.2013.06.093
Homo sapiens MT2 CC50 15000.0 nM 10.1021/jm201134m
Homo sapiens MT2 CC50 15000.0 nM 10.1021/ml5003713
Homo sapiens MT2 EC50 15000.0 nM 10.1021/acs.jmedchem.1c01758
Homo sapiens MT2 IC90 1.7 nM 10.1021/jm990580e
Homo sapiens MT2 IC90 2.4 nM 10.1021/jm990580e
Homo sapiens MT2 IC90 2.8 nM 10.1021/jm990580e
Homo sapiens MT2 IC90 17.0 nM 10.1021/jm990580e
Homo sapiens MT2 IC90 3000.0 nM 10.1021/jm990580e
Homo sapiens MT4 Activity 40.02 uM 10.1128/aac.00986-09
Homo sapiens MT4 CC50 1.0 ug.mL-1 10.1016/j.ejmech.2012.04.038
Homo sapiens MT4 CC50 6.33 nM 10.1021/acs.jmedchem.7b00332
Homo sapiens MT4 CC50 300.0 nM 10.1021/jm070811e
Homo sapiens MT4 CC50 320.0 nM 10.1016/j.bmcl.2006.03.080
Homo sapiens MT4 CC50 320.0 nM 10.1021/jm050744t
Homo sapiens MT4 CC50 320.0 nM 10.1021/jm801330n
Homo sapiens MT4 CC50 320.0 nM 10.1039/C4MD00282B
Homo sapiens MT4 CC50 2000.0 nM 10.1016/j.bmc.2012.12.049
Homo sapiens MT4 CC50 2000.0 nM 10.1016/j.ejmech.2018.01.016
Homo sapiens MT4 CC50 2000.0 nM 10.1016/j.ejmech.2019.05.011
Homo sapiens MT4 CC50 3000.0 nM 10.1021/acs.jmedchem.8b01238
Homo sapiens MT4 CC50 3000.0 nM 10.1021/jm500284x
Homo sapiens MT4 CC50 3000.0 nM 10.1021/jm800340w
Homo sapiens MT4 CC50 3160.0 nM 10.1016/j.bmc.2018.12.039
Homo sapiens MT4 CC50 3167.8 nM 10.1021/jm101626c
Homo sapiens MT4 CC50 3200.0 nM 10.1021/jm201308v
Homo sapiens MT4 CC50 6000.0 nM 10.1016/j.bmc.2008.06.012
Homo sapiens MT4 CC50 6000.0 nM 10.1016/j.bmc.2009.06.068
Homo sapiens MT4 CC50 6000.0 nM 10.1016/j.bmc.2009.12.059
Homo sapiens MT4 CC50 6000.0 nM 10.1016/j.bmc.2015.01.002
Homo sapiens MT4 CC50 6000.0 nM 10.1016/j.bmcl.2007.01.025
Homo sapiens MT4 CC50 6000.0 nM 10.1021/jm070382k
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmc.2010.05.081
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmc.2012.07.026
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmc.2012.09.058
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmc.2013.09.051
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmc.2013.10.033
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmc.2014.02.030
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmc.2014.03.020
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmc.2014.08.001
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmc.2016.04.010
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmc.2017.03.009
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmc.2020.115927
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmcl.2012.09.062
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.bmcl.2013.10.059
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.ejmech.2012.02.019
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.ejmech.2012.04.004
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.ejmech.2015.01.042
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.ejmech.2015.02.022
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.ejmech.2016.10.009
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.ejmech.2019.111864
Homo sapiens MT4 CC50 6300.0 nM 10.1016/j.ejmech.2020.113063
Homo sapiens MT4 CC50 6300.0 nM 10.1021/acs.jmedchem.1c00987
Homo sapiens MT4 CC50 6330.0 nM 10.1016/j.bmc.2011.07.023
Homo sapiens MT4 CC50 6330.0 nM 10.1016/j.bmc.2017.05.040
Homo sapiens MT4 CC50 6330.0 nM 10.1016/j.bmc.2017.12.033
Homo sapiens MT4 CC50 6330.0 nM 10.1016/j.ejmech.2022.114471
Homo sapiens MT4 CC50 6330.0 nM 10.1021/acs.jmedchem.1c00128
Homo sapiens MT4 CC50 6330.0 nM 10.1021/acs.jmedchem.1c00708
Homo sapiens MT4 CC50 6330.0 nM 10.1021/acs.jmedchem.1c01676
Homo sapiens MT4 CC50 6335.0 nM 10.1016/j.ejmech.2021.113204
Homo sapiens MT4 CC50 6335.6 nM 10.1016/j.ejmech.2014.05.059
Homo sapiens MT4 CC50 6336.0 nM 10.1007/s00044-009-9220-x
Homo sapiens MT4 CC50 6336.0 nM 10.1016/j.bmc.2009.07.028
Homo sapiens MT4 CC50 6336.0 nM 10.1016/j.bmcl.2008.09.055
Homo sapiens MT4 CC50 6336.0 nM 10.1016/j.ejmech.2009.06.037
Homo sapiens MT4 CC50 6336.0 nM 10.1016/j.ejmech.2015.04.050
Homo sapiens MT4 CC50 6336.0 nM 10.1016/j.ejmech.2015.08.007
Homo sapiens MT4 CC50 6336.0 nM 10.1021/acsmedchemlett.8b00054
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2008.01.039
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2010.03.007
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2011.05.024
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2011.10.002
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2012.04.030
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2013.08.040
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2013.12.045
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2014.11.032
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2015.09.020
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2016.05.010
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2016.07.041
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2018.03.003
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmc.2021.116195
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.bmcl.2018.03.012
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2013.04.052
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2014.02.047
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2014.09.054
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2016.02.068
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2017.02.047
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2017.07.012
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2018.03.059
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2019.111603
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2019.111874
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2020.112549
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2020.112811
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2020.113051
Homo sapiens MT4 CC50 6340.0 nM 10.1016/j.ejmech.2022.114512
Homo sapiens MT4 CC50 6340.0 nM 10.1021/acs.jmedchem.1c01015
Homo sapiens MT4 CC50 6340.0 nM 10.1021/acs.jmedchem.2c00468
Homo sapiens MT4 CC50 6340.0 nM 10.1021/acs.jmedchem.8b01729
Homo sapiens MT4 CC50 6340.0 nM 10.1021/acs.jmedchem.9b01446
Homo sapiens MT4 CC50 6340.0 nM 10.1021/acs.jmedchem.9b01769
Homo sapiens MT4 CC50 6340.0 nM 10.1039/C3MD00028A
Homo sapiens MT4 CC50 6340.0 nM 10.1039/C3MD00247K
Homo sapiens MT4 CC50 6350.0 nM 10.1016/j.bmc.2021.116239
Homo sapiens MT4 CC50 6350.0 nM 10.1016/j.ejmech.2019.111619
Homo sapiens MT4 CC50 6380.0 nM 10.1016/j.ejmech.2020.112237
Homo sapiens MT4 CC50 6500.0 nM 10.1016/j.bmc.2015.03.037
Homo sapiens MT4 CC50 9000.0 nM 10.1016/j.bmcl.2017.03.009
Homo sapiens MT4 CC50 15839.0 nM 10.1016/j.ejmech.2014.04.027
Homo sapiens MT4 CC50 15839.0 nM 10.1016/j.ejmech.2020.112696
Homo sapiens MT4 CC50 15839.0 nM 10.1021/acs.jmedchem.6b01906
Homo sapiens MT4 CC50 15839.0 nM 10.1021/jm300477h
Homo sapiens MT4 CC50 15839.0 nM 10.1021/jm5011622
Homo sapiens MT4 CC50 32314.0 nM 10.1016/j.ejmech.2006.11.014
Homo sapiens MT4 CC50 35000.0 nM 10.1007/s00044-008-9149-5
Homo sapiens MT4 CC50 35000.0 nM 10.1016/j.ejmech.2009.08.013
Homo sapiens MT4 CC50 35000.0 nM 10.1021/jm031147e
Homo sapiens MT4 CC50 37000.0 nM 10.1016/j.bmcl.2015.04.006
Homo sapiens MT4 CC50 37000.0 nM 10.1016/j.ejmech.2012.07.020
Homo sapiens MT4 CC50 38000.0 nM 10.1016/j.bmc.2014.06.043
Homo sapiens MT4 CC50 38000.0 nM 10.1016/j.bmc.2015.09.035
Homo sapiens MT4 CC50 40000.0 nM 10.1016/j.bmc.2011.10.009
Homo sapiens MT4 CC50 40000.0 nM 10.1016/j.bmc.2015.08.028
Homo sapiens MT4 CC50 40000.0 nM 10.1016/j.ejmech.2012.03.038
Homo sapiens MT4 CC50 40000.0 nM 10.1016/j.ejmech.2014.07.011
Homo sapiens MT4 CC50 40000.0 nM 10.1016/j.ejmech.2015.06.027
Homo sapiens MT4 CC50 40000.0 nM 10.1016/j.ejmech.2015.10.002
Homo sapiens MT4 CC50 40000.0 nM 10.1016/j.ejmech.2017.09.060
Homo sapiens MT4 CC50 40000.0 nM 10.1016/j.ejmech.2017.12.083
Homo sapiens MT4 CC50 40000.0 nM 10.1021/jm500139a
Homo sapiens MT4 CC50 40196.0 nM 10.1021/acs.jmedchem.1c01758
Homo sapiens MT4 CC50 45000.0 nM 10.1007/s00044-013-0740-z
Homo sapiens MT4 CC50 45000.0 nM 10.1016/j.ejmech.2009.08.012
Homo sapiens MT4 CC50 63000.0 nM 10.1016/j.bmc.2011.08.025
Homo sapiens MT4 CC50 63360.0 nM 10.1016/j.bmc.2010.05.036
Homo sapiens MT4 CC50 80000.0 nM 10.1016/j.bmcl.2004.04.008
Homo sapiens MT4 CD50 100.0 uM 10.1021/jm020949r
Homo sapiens MT4 EC50 1.0 nM 10.1021/jm040127p
Homo sapiens MT4 EC50 2.0 nM 10.1021/jm040127p
Homo sapiens MT4 EC50 4.0 nM 10.1021/jm010853h
Homo sapiens MT4 EC50 4.0 nM 10.1021/jm0309856
Homo sapiens MT4 EC50 4.0 nM 10.1021/jm040854k
Homo sapiens MT4 EC50 25.0 nM 10.1021/jm010853h
Homo sapiens MT4 EC50 25.0 nM 10.1021/jm0309856
Homo sapiens MT4 EC50 25.0 nM 10.1021/jm040854k
Homo sapiens MT4 EC50 40.0 nM 10.1021/jm040127p
Homo sapiens MT4 EC50 150.0 nM 10.1021/jm040854k
Homo sapiens MT4 EC50 160.0 nM 10.1021/jm040127p
Homo sapiens MT4 EC50 10000.0 nM 10.1021/jm040127p
Homo sapiens MT4 ED50 0.05 uM 10.1021/jm990095j
Homo sapiens MT4 IC50 1.0 nM 10.1016/j.bmcl.2003.09.045
Homo sapiens MT4 IC50 2.0 nM 10.1016/j.bmcl.2003.09.045
Homo sapiens MT4 IC50 2.7 nM 10.1021/jm030255y
Homo sapiens MT4 IC50 3.5 nM 10.1021/jm030255y
Homo sapiens MT4 IC50 40.0 nM 10.1016/j.bmcl.2003.09.045
Homo sapiens MT4 IC50 40.0 nM 10.1016/s0960-894x(04)00205-7
Homo sapiens MT4 IC50 200.0 nM 10.1016/j.bmcl.2003.09.045
Homo sapiens MT4 IC50 10000.0 nM 10.1016/j.bmcl.2003.09.045
Homo sapiens MT4 IC50 nan nM 10.1016/j.bmcl.2004.04.008
Homo sapiens Multidrug resistance-associated protein 1 Activity nan None 10.1124/dmd.106.012765
Homo sapiens Multidrug resistance-associated protein 1 Activity nan None 10.1128/aac.01527-10
Homo sapiens Multidrug resistance-associated protein 4 IC50 133000.0 nM 10.1093/toxsci/kft176
Homo sapiens Mu opioid receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Muscarinic acetylcholine receptor M1 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Muscarinic acetylcholine receptor M2 AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Muscarinic acetylcholine receptor M3 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Neuronal acetylcholine receptor protein alpha-4 subunit AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Neuropeptide S receptor Potency 10000.0 nM None
Homo sapiens Neuropeptide Y receptor type 1 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Norepinephrine transporter AC50 15000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens PBMC CC50 100000.0 nM 10.1016/j.bmcl.2016.06.065
Homo sapiens PBMC Drug uptake 974.0 ng/ml 10.1128/aac.00283-10
Homo sapiens PBMC Drug uptake 1469.0 ng/ml 10.1128/aac.00283-10
Homo sapiens PBMC Drug uptake 2029.0 ng/ml 10.1128/aac.00283-10
Homo sapiens PBMC Drug uptake 3597.0 ng/ml 10.1128/aac.00283-10
Homo sapiens PBMC Ratio 1.36 None 10.1128/aac.00283-10
Homo sapiens PBMC Ratio 1.53 None 10.1128/aac.00283-10
Homo sapiens PBMC Ratio 1.63 None 10.1128/aac.00283-10
Homo sapiens PBMC Ratio 1.76 None 10.1128/aac.00283-10
Homo sapiens Peroxisome proliferator-activated receptor gamma AC50 17999.9 nM 10.1038/s41467-023-40064-9
Homo sapiens Peroxisome proliferator-activated receptor gamma AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens P-glycoprotein 1 Activity nan None 10.1128/aac.01527-10
Homo sapiens P-glycoprotein 1 Inhibition nan % 10.1128/aac.01527-10
Homo sapiens Phosphodiesterase 3A AC50 23999.9 nM 10.1038/s41467-023-40064-9
Homo sapiens Phosphodiesterase 4D AC50 14966.7 nM 10.1038/s41467-023-40064-9
Homo sapiens Plasma Activity 99.5 % 10.1128/aac.01559-08
Homo sapiens Plasma Cp 95.0 ng/ml 10.1124/dmd.112.049601
Homo sapiens Plasma Cp 2170.0 ng/ml 10.1124/dmd.112.049601
Homo sapiens Plasma Drug metabolism nan None 10.1124/dmd.112.049601
Homo sapiens Plasma Fu 0.0047 None 10.1128/aac.00283-10
Homo sapiens Plasma Fu 0.0052 None 10.1128/aac.00283-10
Homo sapiens Pregnane X receptor AC50 19099.9 nM 10.1038/s41467-023-40064-9
Homo sapiens Pregnane X receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Progesterone receptor AC50 14000.1 nM 10.1038/s41467-023-40064-9
Homo sapiens Progesterone receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 1a (5-HT1a) receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2a (5-HT2a) receptor AC50 3786.2 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2a (5-HT2a) receptor AC50 26999.8 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2a (5-HT2a) receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2b (5-HT2b) receptor AC50 10000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 2c (5-HT2c) receptor AC50 5612.5 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin 3a (5-HT3a) receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serotonin transporter AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Serum albumin PPB 99.9 % 10.1016/j.bmcl.2010.01.085
Homo sapiens Serum albumin PPB 99.9 % 10.1016/j.bmcl.2010.01.086
Homo sapiens Solute carrier family 22 member 1 Inhibition 37.0 % 10.1021/jm8003152
Homo sapiens Solute carrier organic anion transporter family member 1B1 Activity nan None 10.1128/aac.01527-10
Homo sapiens Solute carrier organic anion transporter family member 1B1 Inhibition 40.9 % 10.1021/jm300212s
Homo sapiens Solute carrier organic anion transporter family member 1B3 Inhibition 18.2 % 10.1021/jm300212s
Homo sapiens Solute carrier organic anion transporter family member 2B1 Inhibition 43.2 % 10.1021/jm300212s
Homo sapiens SUP-T1 CC50 nan None 10.1021/acs.jnatprod.6b00878
Homo sapiens Thromboxane A2 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Type-1 angiotensin II receptor AC50 12999.9 nM 10.1038/s41467-023-40064-9
Homo sapiens Tyrosyl-DNA phosphodiesterase 1 Potency 16788.9 nM None
Homo sapiens Tyrosyl-DNA phosphodiesterase 1 Potency 29855.4 nM None
Homo sapiens TZM CC50 6300.0 nM 10.1016/j.ejmech.2020.113063
Homo sapiens TZM CC50 nan None 10.1016/j.bmc.2019.06.044
Homo sapiens Vasopressin V1a receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Homo sapiens Vasopressin V2 receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Human alphaherpesvirus 1 Human alphaherpesvirus 1 EC50 nan None 10.1016/j.bmc.2015.09.035
Human immunodeficiency virus Human immunodeficiency virus EC50 0.5 nM 10.1016/j.bmcl.2006.09.047
Human immunodeficiency virus Human immunodeficiency virus EC50 0.55 nM 10.1016/j.bmcl.2012.12.049
Human immunodeficiency virus Human immunodeficiency virus EC50 1.0 nM 10.1021/jm800527x
Human immunodeficiency virus Human immunodeficiency virus EC50 1.6 nM 10.1016/j.bmcl.2012.12.049
Human immunodeficiency virus Human immunodeficiency virus EC50 2.0 nM 10.1021/jm800527x
Human immunodeficiency virus Human immunodeficiency virus EC50 3.0 nM 10.1021/jm800527x
Human immunodeficiency virus Human immunodeficiency virus EC50 4.0 nM 10.1021/jm800527x
Human immunodeficiency virus Human immunodeficiency virus EC50 6.0 nM 10.1021/jm800527x
Human immunodeficiency virus Human immunodeficiency virus EC50 7.0 nM 10.1021/jm800527x
Human immunodeficiency virus Human immunodeficiency virus EC50 8.0 nM 10.1021/jm800527x
Human immunodeficiency virus Human immunodeficiency virus EC50 12.0 nM 10.1021/jm800527x
Human immunodeficiency virus Human immunodeficiency virus EC50 18.0 nM 10.1021/jm800527x
Human immunodeficiency virus Human immunodeficiency virus EC50 66.0 nM 10.1021/jm800527x
Human immunodeficiency virus Human immunodeficiency virus EC50 100.0 nM 10.1021/jm800527x
Human immunodeficiency virus Human immunodeficiency virus EC50 780.0 nM 10.1016/j.bmcl.2005.07.046
Human immunodeficiency virus Human immunodeficiency virus EC50 20000.0 nM 10.1021/jm0512490
Human immunodeficiency virus Human immunodeficiency virus FC 1.0 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 2.2 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 7.2 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 15.4 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 16.0 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 33.6 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 34.8 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 42.0 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 55.6 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 213.0 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 229.0 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 248.6 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 281.4 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 306.2 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus FC 454.0 None 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 0.5 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 0.6 nM 10.1016/j.bmcl.2009.08.080
Human immunodeficiency virus Human immunodeficiency virus IC50 1.1 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 3.6 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 7.7 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 8.0 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 16.8 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 17.4 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 21.0 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 27.8 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 106.5 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 114.5 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 124.3 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 140.7 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 153.1 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC50 500.0 nM 10.1021/jm901230r
Human immunodeficiency virus Human immunodeficiency virus IC90 1.2 nM 10.1016/j.bmcl.2009.08.080
Human immunodeficiency virus Human immunodeficiency virus IC95 39.0 nM 10.1016/j.bmcl.2013.12.070
Human immunodeficiency virus Human immunodeficiency virus IC95 90.0 nM 10.1016/j.bmcl.2013.12.070
Human immunodeficiency virus Human immunodeficiency virus IC95 1400.0 nM 10.1016/j.bmcl.2013.12.070
Human immunodeficiency virus Human immunodeficiency virus IC95 3200.0 nM 10.1016/j.bmcl.2013.12.070
Human immunodeficiency virus Human immunodeficiency virus Ratio EC50 0.8 None 10.1128/aac.00210-08
Human immunodeficiency virus Human immunodeficiency virus Ratio EC50 0.9 None 10.1128/aac.00210-08
Human immunodeficiency virus Human immunodeficiency virus Ratio EC50 1.2 None 10.1128/aac.00210-08
Human immunodeficiency virus Human immunodeficiency virus Ratio EC50 1.9 None 10.1128/aac.00210-08
Human immunodeficiency virus Human immunodeficiency virus Ratio EC50 3.0 None 10.1016/j.bmcl.2012.12.049
Human immunodeficiency virus Human immunodeficiency virus Ratio EC50 15.3 None 10.1128/aac.00210-08
Human immunodeficiency virus Human immunodeficiency virus Ratio EC50 70.0 None 10.1021/acsmedchemlett.5b00036
Human immunodeficiency virus Human immunodeficiency virus Ratio EC50 2128.0 None 10.1128/aac.00210-08
Human immunodeficiency virus Human immunodeficiency virus Selectivity index 256.0 None 10.1016/j.bmcl.2005.07.046
Human immunodeficiency virus 1 Envelope glycoprotein gp160 IC50 3.5 nM 10.1016/j.bmcl.2019.01.011
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Activity 0.02 uM 10.1128/aac.00972-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Activity nan None 10.1016/j.ejmech.2008.10.032
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Activity nan None 10.1021/acs.jnatprod.7b00659
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Activity nan None 10.1128/aac.00972-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Activity nan None 10.1128/aac.01064-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Activity nan None 10.1128/aac.01218-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 CC50 30000.0 nM 10.1016/j.bmc.2007.09.015
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.00019 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.00025 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.0003 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.00044 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.00085 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.00103 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.005 nM 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.049 ug.mL-1 10.1016/j.bmc.2015.09.020
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.05 nM 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.1 nM 10.1128/aac.00972-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.1 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.12 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.15 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.16 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.17 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.19 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.2 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.27 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.3 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.3 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.31 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.33 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.34 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.34 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.39 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.4 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.42 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.43 nM 10.1016/j.ejmech.2018.01.016
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.48 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.48 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.49 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.5 nM 10.1016/j.bmcl.2006.01.066
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.5 nM 10.1016/j.bmcl.2006.01.073
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.5 nM 10.1016/j.bmcl.2006.04.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.5 nM 10.1021/jm301294g
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.5 nM 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.5 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.5 nM 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.52 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.53 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.6 nM 10.1128/aac.00759-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.62 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.64 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.66 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.7 nM 10.1016/j.bmcl.2007.11.127
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.7 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.7 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.72 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.74 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.74 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.76 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.78 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.8 nM 10.1021/np200087d
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.8 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.8 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.9 nM 10.1016/j.bmc.2008.06.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.9 nM 10.1016/j.bmc.2009.06.068
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.9 nM 10.1016/j.bmc.2009.12.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.9 nM 10.1016/j.bmcl.2007.01.025
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.9 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.92 nM 10.1039/C4MD00282B
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.95 nM 10.1128/aac.00210-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 0.98 nM 10.1039/C4MD00282B
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1016/j.bmc.2014.08.005
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1016/j.bmcl.2006.01.066
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1016/j.bmcl.2006.04.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1016/j.bmcl.2006.05.073
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1016/j.bmcl.2006.05.096
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1016/j.bmcl.2016.06.065
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1016/j.ejmech.2018.01.016
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1016/j.ejmech.2020.112071
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1021/jm030558s
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1021/jm040838n
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1021/jm050744t
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1021/jm070382k
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1021/jm301294g
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1021/jm801330n
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1128/aac.00759-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.0 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.1 nM 10.1016/j.bmcl.2006.01.066
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.1 nM 10.1016/j.bmcl.2010.01.085
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.1 nM 10.1016/j.bmcl.2010.01.086
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.1 nM 10.1128/aac.00643-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.1 nM 10.1128/aac.01064-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.1 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.11 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.17 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.19 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.2 nM 10.1016/j.ejmech.2011.06.020
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.2 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.288 nM 10.1021/acs.jmedchem.8b01729
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.3 nM 10.1021/acs.jmedchem.8b01729
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.3 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.4 nM 10.1021/jm040840e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.4 nM 10.1021/jm201134m
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.47 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.5 nM 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.5 nM 10.1016/j.ejmech.2018.01.016
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.5 nM 10.1021/jm101614j
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.5 nM 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.58 nM 10.1016/j.bmc.2018.03.003
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.6 nM 10.1016/j.ejmech.2006.11.014
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.6 nM 10.1016/j.ejmech.2018.01.016
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.6 nM 10.1016/j.ejmech.2019.05.011
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.6 nM 10.1021/acs.jmedchem.0c00117
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.6 nM 10.1128/aac.00210-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.7 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.73 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.8 nM 10.1021/acs.jmedchem.5b01430
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1.9 nM 10.1128/aac.00210-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1007/s00044-013-0740-z
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmc.2007.09.015
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmc.2011.08.060
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmc.2011.10.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmc.2015.08.028
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmc.2016.07.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmcl.2006.01.066
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmcl.2006.05.073
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmcl.2006.08.037
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmcl.2010.03.006
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmcl.2012.11.115
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmcl.2013.06.091
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmcl.2013.06.093
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.bmcl.2015.04.006
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.ejmech.2009.08.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.ejmech.2012.03.038
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.ejmech.2012.07.020
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.ejmech.2014.07.011
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.ejmech.2015.06.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.ejmech.2015.10.002
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.ejmech.2017.09.060
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.ejmech.2017.12.083
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.ejmech.2019.05.011
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.ejmech.2020.112071
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1016/j.ejmech.2020.112811
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1021/jm030558s
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1021/jm040838n
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1021/jm040840e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1021/jm201134m
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1021/jm500139a
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1021/ml5003713
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1021/np200087d
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1128/aac.00643-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.0 nM 10.1128/aac.01480-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.08 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.1 nM 10.1016/j.bmc.2010.05.081
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.1 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.2 nM 10.1016/j.bmc.2010.05.081
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.2 nM 10.1021/acs.jmedchem.2c00468
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.26 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.31 nM 10.1021/acs.jmedchem.9b01769
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.5 nM 10.1016/j.bmc.2021.116195
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.5 nM 10.1016/j.ejmech.2020.113063
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.6 nM 10.1016/j.bmcl.2010.01.085
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.6 nM 10.1016/j.bmcl.2010.01.086
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.6 nM 10.1016/j.ejmech.2019.111864
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.7 nM 10.1016/j.bmc.2016.05.010
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.7 nM 10.1016/j.bmcl.2007.01.025
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.7 nM 10.1021/jm801395v
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.73 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.8 nM 10.1016/j.ejmech.2020.113051
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.818 nM 10.1016/j.ejmech.2020.113051
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2.9 nM 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1007/s00044-008-9149-5
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1016/j.bmc.2008.01.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1016/j.bmc.2010.03.007
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1016/j.bmc.2010.05.036
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1016/j.bmc.2011.08.025
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1016/j.bmc.2021.116239
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1016/j.ejmech.2009.08.013
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1016/j.ejmech.2012.04.038
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1016/j.ejmech.2016.10.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1016/j.ejmech.2022.114512
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1021/jm801330n
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.0 nM 10.1128/aac.01480-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.17 nM 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.2 nM 10.1016/j.ejmech.2022.114471
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.2 nM 10.1021/acs.jmedchem.1c01758
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.5 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.57 nM 10.1128/aac.01795-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.7 nM 10.1016/j.bmcl.2017.03.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.8 nM 10.1016/j.ejmech.2019.111874
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3.9 nM 10.1016/j.ejmech.2006.11.014
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1016/j.bmc.2016.05.010
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1016/j.bmc.2017.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1016/j.bmc.2017.12.033
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1016/j.bmcl.2006.01.066
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1016/j.bmcl.2006.05.073
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1016/j.bmcl.2010.09.034
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1016/j.ejmech.2022.114471
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1021/acs.jmedchem.1c00128
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1021/acs.jmedchem.1c00708
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1021/acs.jmedchem.1c01676
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1021/jm031147e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1021/jm0512490
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1021/jm070811e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1021/jm500139a
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.0 nM 10.1128/aac.01480-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.1 nM 10.1016/j.ejmech.2006.11.014
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.24 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.3 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.4 nM 10.1007/s00044-009-9220-x
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.4 nM 10.1016/j.bmc.2009.07.028
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.4 nM 10.1016/j.bmc.2011.05.024
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.4 nM 10.1016/j.bmcl.2008.09.055
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.4 nM 10.1016/j.ejmech.2009.06.037
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.4 nM 10.1016/j.ejmech.2019.111864
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.5 nM 10.1021/acs.jmedchem.1c00987
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.7 nM 10.1016/j.bmcl.2017.03.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.7 nM 10.1016/j.ejmech.2020.112237
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 4.8 nM 10.1016/j.bmcl.2018.03.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.bmc.2011.07.023
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.bmc.2012.09.058
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.bmc.2014.06.043
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.bmc.2015.09.035
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.bmcl.2010.09.034
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.bmcl.2012.09.062
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.ejmech.2012.04.004
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.ejmech.2015.11.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.ejmech.2016.10.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.ejmech.2017.07.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.ejmech.2019.111864
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.ejmech.2020.112811
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.ejmech.2020.113051
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1016/j.ejmech.2022.114471
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1021/acs.jmedchem.2c00468
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1021/jm070382k
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.0 nM 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.03 nM 10.1021/acs.jmedchem.7b00332
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.1 nM 10.1016/j.bmc.2016.07.041
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.1 nM 10.1016/j.ejmech.2017.02.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.12 nM 10.1021/acs.jmedchem.1c01015
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.2 nM 10.1016/j.bmc.2021.116195
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.2 nM 10.1016/j.ejmech.2017.02.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.2 nM 10.1016/j.ejmech.2020.113063
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.23 nM 10.1016/j.bmc.2016.07.041
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.26 nM 10.1021/acs.jmedchem.1c01015
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.3 nM 10.1016/j.bmc.2014.08.001
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.3 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.4 nM 10.1016/j.bmc.2010.05.081
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.4 nM 10.1016/j.bmc.2011.10.002
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.4 nM 10.1016/j.bmc.2015.03.037
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.4 nM 10.1016/j.bmcl.2017.03.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.4 nM 10.1016/j.ejmech.2012.02.019
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.4 nM 10.1016/j.ejmech.2015.08.007
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.4 nM 10.1016/j.ejmech.2015.11.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.4 nM 10.1016/j.ejmech.2016.02.068
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.4 nM 10.1021/acs.jmedchem.1c00708
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.4 nM 10.1021/acs.jmedchem.1c01676
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.4 nM 10.1021/acs.jmedchem.1c01758
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.4 nM 10.1039/C3MD00028A
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.5 nM 10.1016/j.ejmech.2011.08.011
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.5 nM 10.1016/j.ejmech.2020.113051
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.6 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.7 nM 10.1016/j.bmc.2010.05.081
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.7 nM 10.1016/j.bmc.2021.116195
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.7 nM 10.1016/j.ejmech.2014.02.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 5.7 nM 10.1016/j.ejmech.2020.113063
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1016/j.bmc.2013.12.045
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1016/j.bmc.2014.03.020
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1016/j.bmc.2015.01.002
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1016/j.bmc.2016.04.010
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1016/j.bmc.2018.03.003
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1016/j.bmc.2021.116239
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1016/j.bmcl.2006.01.066
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1016/j.bmcl.2006.05.073
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1016/j.bmcl.2008.06.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1016/j.ejmech.2015.02.022
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1016/j.ejmech.2019.111603
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1016/j.ejmech.2020.112811
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1021/acs.jmedchem.1c00987
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1021/acs.jmedchem.8b01729
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.0 nM 10.1021/jm070811e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.1 nM 10.1016/j.bmcl.2007.01.025
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.2 nM 10.1016/j.bmc.2014.11.032
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.2 nM 10.1016/j.ejmech.2022.114512
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.3 nM 10.1016/j.bmc.2015.09.020
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.3 nM 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.3 nM 10.1016/j.ejmech.2014.09.054
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.3 nM 10.1016/j.ejmech.2015.01.042
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.3 nM 10.1016/j.ejmech.2015.04.050
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.3 nM 10.1016/j.ejmech.2015.08.007
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.3 nM 10.1016/j.ejmech.2019.111619
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.3 nM 10.1021/acs.jmedchem.9b01446
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.3 nM 10.1021/jm300477h
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.57 nM 10.1016/j.bmc.2012.04.030
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.6 nM 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.7 nM 10.1016/j.bmc.2013.08.040
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.8 nM 10.1016/j.bmc.2016.07.041
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.8 nM 10.1016/j.ejmech.2015.11.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.8 nM 10.1016/j.ejmech.2017.02.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6.8 nM 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.0 nM 10.1016/j.bmc.2012.12.049
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.0 nM 10.1016/j.bmc.2018.12.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.0 nM 10.1016/j.bmc.2021.116239
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.0 nM 10.1016/j.bmcl.2013.10.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.0 nM 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.0 nM 10.1016/j.ejmech.2019.111603
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.0 nM 10.1021/acs.jmedchem.2c00468
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.0 nM 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.0 nM 10.1021/jm0512490
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.0 nM 10.1021/jm500284x
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.0 nM 10.1021/jm800340w
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.1 nM 10.1016/j.ejmech.2022.114512
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.3 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.3 nM 10.1021/acs.jmedchem.9b01446
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.3 nM 10.1021/jm201308v
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.4 nM 10.1016/j.bmc.2013.10.033
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.4 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.4 nM 10.1021/acs.jmedchem.9b01446
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.5 nM 10.1021/acs.jmedchem.1c00708
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7.5 nM 10.1021/acs.jmedchem.1c01676
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 8.0 nM 10.1016/j.bmc.2007.09.015
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 8.0 nM 10.1016/j.bmcl.2006.01.066
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 8.0 nM 10.1021/jm801330n
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 8.2 nM 10.1016/j.ejmech.2015.08.007
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 8.3 nM 10.1016/j.ejmech.2019.111619
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 8.5 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 8.6 nM 10.1016/j.ejmech.2019.111619
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 8.63 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 8.9 nM 10.1039/C3MD00247K
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 9.0 nM 10.1016/j.bmc.2013.09.051
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 9.6 nM 10.1016/j.bmcl.2007.01.025
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1007/s00044-009-9192-x
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.bmc.2007.12.046
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.bmc.2007.12.050
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.bmc.2008.05.010
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.bmc.2016.07.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.bmcl.2006.01.066
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.bmcl.2006.04.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.bmcl.2006.05.073
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.bmcl.2010.03.006
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.bmcl.2012.11.115
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.bmcl.2013.06.091
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.ejmech.2008.10.032
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.ejmech.2009.08.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1016/j.ejmech.2013.04.052
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1021/jm040838n
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1021/jm201134m
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1021/jm201308v
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1021/jm500139a
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.0 nM 10.1021/ml5003713
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.1 nM 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.3 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10.7 nM 10.1021/acs.jmedchem.1c01676
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 11.0 nM 10.1021/jm030558s
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 12.66 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 12.8 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 13.0 nM 10.1016/j.bmcl.2006.05.096
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 13.0 nM 10.1021/jm500284x
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 13.0 nM 10.1128/aac.01480-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 14.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 14.27 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 15.0 nM 10.1021/acsmedchemlett.5b00254
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 15.0 nM 10.1128/aac.00210-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 15.9 nM 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 15.9 nM 10.1016/j.ejmech.2020.112696
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 15.9 nM 10.1021/acs.jmedchem.6b01906
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 15.9 nM 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 17.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 19.0 nM 10.1016/j.bmcl.2006.05.096
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 19.0 nM 10.1016/j.bmcl.2008.06.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 19.0 nM 10.1016/j.ejmech.2018.01.016
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 20.0 nM 10.1016/j.ejmech.2008.09.024
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 20.0 nM 10.1021/jm301294g
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 22.0 nM 10.1016/j.bmc.2014.02.030
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 22.0 nM 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 22.0 nM 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 24.0 nM 10.1021/np200087d
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 24.43 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 25.0 nM 10.1021/jm031147e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 25.1 nM 10.1021/jm040838n
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 25.14 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 28.0 nM 10.1016/j.ejmech.2021.113204
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 28.0 nM 10.1021/jm040840e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 29.0 nM 10.1128/aac.01480-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 30.0 nM 10.1016/j.bmc.2016.07.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 30.0 nM 10.1016/j.bmcl.2010.03.006
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 30.0 nM 10.1016/j.bmcl.2012.11.115
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 30.0 nM 10.1016/j.bmcl.2013.06.091
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 30.0 nM 10.1016/j.ejmech.2020.112071
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 30.0 nM 10.1021/acs.jmedchem.2c00468
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 30.0 nM 10.1021/jm201134m
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 30.0 nM 10.1021/ml5003713
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 30.8 nM 10.1016/j.bmc.2021.116195
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 30.8 nM 10.1016/j.ejmech.2020.113063
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 31.0 nM 10.1016/j.ejmech.2006.11.014
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 31.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 32.0 nM 10.1016/j.bmc.2010.05.081
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 32.0 nM 10.1016/j.bmcl.2006.01.066
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 32.0 nM 10.1016/j.bmcl.2006.04.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 32.0 nM 10.1016/j.bmcl.2006.05.073
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 32.0 nM 10.1016/j.ejmech.2020.113051
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 34.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 34.88 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 35.0 nM 10.1016/j.bmcl.2010.01.085
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 35.0 nM 10.1016/j.bmcl.2010.01.086
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 35.0 nM 10.1021/jm040840e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 37.0 nM 10.1016/j.bmc.2021.116239
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 37.0 nM 10.1021/acs.jmedchem.5b01430
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 37.0 nM 10.1021/jm040840e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 37.0 nM 10.1021/jm201134m
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 37.1 nM 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 37.1 nM 10.1016/j.ejmech.2022.114512
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 38.0 nM 10.1016/j.bmcl.2017.03.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 38.0 nM 10.1021/jm030558s
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 39.0 nM 10.1021/jm030558s
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 40.0 nM 10.1016/j.bmc.2007.12.046
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 40.0 nM 10.1016/j.bmc.2007.12.050
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 40.0 nM 10.1016/j.bmc.2008.05.010
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 40.0 nM 10.1016/j.ejmech.2018.01.016
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 40.0 nM 10.1016/j.ejmech.2020.112811
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 40.0 nM 10.1021/jm040838n
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 41.0 nM 10.1021/acsmedchemlett.5b00254
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 44.0 nM 10.1016/j.ejmech.2019.111603
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 44.0 nM 10.1016/j.ejmech.2019.111619
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 44.0 nM 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 44.0 nM 10.1021/acs.jmedchem.9b01446
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 44.0 nM 10.1021/jm800340w
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 44.7 nM 10.1021/acs.jmedchem.1c00708
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 46.4 nM 10.1016/j.ejmech.2006.11.014
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 46.9 nM 10.1016/j.ejmech.2006.11.014
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 47.0 nM 10.1016/j.bmc.2018.03.003
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 49.0 nM 10.1016/j.bmc.2018.03.003
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 49.0 nM 10.1016/j.bmcl.2007.01.025
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 50.0 nM 10.1016/j.ejmech.2018.01.016
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 50.0 nM 10.1016/j.ejmech.2020.112071
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 51.6 nM 10.1021/acs.jmedchem.1c00987
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 52.0 nM 10.1021/acs.jmedchem.8b01729
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 54.0 nM 10.1016/j.ejmech.2011.08.011
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 55.0 nM 10.1016/j.ejmech.2006.11.014
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 55.0 nM 10.1016/j.ejmech.2019.05.011
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 57.0 nM 10.1016/j.ejmech.2016.10.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 57.0 nM 10.1016/j.ejmech.2022.114471
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 57.0 nM 10.1021/jm050744t
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 57.0 nM 10.1021/jm801330n
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 57.2 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 57.3 nM 10.1016/j.bmcl.2007.01.025
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 58.0 nM 10.1021/acs.jmedchem.5b01430
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 59.0 nM 10.1016/j.ejmech.2018.01.016
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 60.0 nM 10.1016/j.ejmech.2009.08.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 60.0 nM 10.1016/j.ejmech.2020.112071
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 60.0 nM 10.1021/jm500139a
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 63.7 nM 10.1016/j.ejmech.2020.113063
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 63.8 nM 10.1016/j.bmc.2021.116195
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 64.0 nM 10.1021/acs.jmedchem.2c00468
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 64.3 nM 10.1128/aac.01795-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 66.0 nM 10.1016/j.bmc.2010.05.081
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 67.93 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 69.3 nM 10.1021/jm300477h
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 71.0 nM 10.1016/j.ejmech.2020.113051
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 72.0 nM 10.1016/j.ejmech.2022.114471
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 72.8 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 76.0 nM 10.1016/j.ejmech.2016.10.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 76.0 nM 10.1016/j.ejmech.2019.111864
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 77.06 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 78.0 nM 10.1021/jm040840e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 78.39 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 80.0 nM 10.1021/jm070811e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 80.0 nM 10.1021/jm500139a
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 81.0 nM 10.1021/acsmedchemlett.7b00524
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 83.0 nM 10.1016/j.bmcl.2008.06.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 85.5 nM 10.1016/j.ejmech.2015.08.007
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 85.9 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 86.0 nM 10.1128/aac.00210-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 89.0 nM 10.1016/j.ejmech.2022.114471
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 89.0 nM 10.1021/acs.jmedchem.8b01729
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 89.2 nM 10.1021/acs.jmedchem.1c00987
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 90.0 nM 10.1021/jm070811e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 90.0 nM 10.1021/jm500139a
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 91.5 nM 10.1021/acs.jmedchem.1c00708
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 91.5 nM 10.1021/acs.jmedchem.1c01676
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 92.0 nM 10.1016/j.ejmech.2016.10.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 94.0 nM 10.1016/j.ejmech.2020.112811
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 94.2 nM 10.1016/j.ejmech.2022.114512
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 95.0 nM 10.1016/j.ejmech.2015.08.007
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 95.0 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 97.0 nM 10.1016/j.ejmech.2022.114471
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 98.0 nM 10.1016/j.ejmech.2016.10.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 98.0 nM 10.1016/j.ejmech.2019.111619
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 100.0 nM 10.1016/j.bmc.2016.07.041
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 100.0 nM 10.1016/j.ejmech.2015.11.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 100.0 nM 10.1016/j.ejmech.2017.02.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 100.0 nM 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 100.0 nM 10.1021/jm500139a
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 102.0 nM 10.1016/j.ejmech.2019.111603
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 102.0 nM 10.1021/acs.jmedchem.9b01446
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 102.5 nM 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 103.0 nM 10.1016/j.bmc.2021.116239
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 104.0 nM 10.1016/j.bmc.2010.05.081
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 105.0 nM 10.1016/j.ejmech.2022.114471
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 108.0 nM 10.1016/j.ejmech.2011.08.011
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 110.0 nM 10.1016/j.bmc.2010.05.081
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 110.0 nM 10.1016/j.bmc.2018.03.003
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 110.0 nM 10.1016/j.ejmech.2016.10.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 111.0 nM 10.1021/acs.jmedchem.1c01015
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 120.0 nM 10.1016/j.bmc.2016.07.041
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 120.0 nM 10.1016/j.bmc.2018.03.003
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 120.0 nM 10.1016/j.bmcl.2017.03.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 120.0 nM 10.1016/j.ejmech.2015.11.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 120.0 nM 10.1016/j.ejmech.2017.02.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 120.0 nM 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 120.0 nM 10.1016/j.ejmech.2020.112071
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 124.0 nM 10.1016/j.ejmech.2019.111874
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 130.0 nM 10.1016/j.bmc.2018.03.003
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 130.0 nM 10.1016/j.bmcl.2017.03.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 130.0 nM 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 130.0 nM 10.1016/j.ejmech.2020.112696
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 130.0 nM 10.1021/acs.jmedchem.6b01906
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 130.0 nM 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 135.57 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 138.0 nM 10.1021/jm030558s
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 140.0 nM 10.1016/j.bmc.2015.03.037
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 140.0 nM 10.1016/j.bmcl.2018.03.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 140.0 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 144.0 nM 10.1021/acs.jmedchem.1c00987
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 147.4 nM 10.1021/acs.jmedchem.1c01758
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 148.0 nM 10.1016/j.ejmech.2020.113063
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 148.3 nM 10.1016/j.bmc.2021.116195
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 150.0 nM 10.1021/jm031147e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 155.0 nM 10.1016/j.ejmech.2015.04.050
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 155.0 nM 10.1016/j.ejmech.2015.08.007
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 157.0 nM 10.1021/jm301294g
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 157.5 nM 10.1021/jm300477h
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 160.0 nM 10.1016/j.bmc.2014.11.032
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 160.0 nM 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 160.0 nM 10.1016/j.ejmech.2014.09.054
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 160.0 nM 10.1016/j.ejmech.2015.01.042
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 160.0 nM 10.1016/j.ejmech.2015.02.022
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 160.0 nM 10.1016/j.ejmech.2020.112696
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 160.0 nM 10.1021/acs.jmedchem.6b01906
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 160.0 nM 10.1021/jm040838n
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 160.0 nM 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 167.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 168.5 nM 10.1016/j.bmc.2021.116195
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 169.0 nM 10.1016/j.ejmech.2020.113063
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 170.0 nM 10.1016/j.bmcl.2017.03.009
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 180.0 nM 10.1016/j.bmc.2010.03.007
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 180.0 nM 10.1016/j.ejmech.2020.112071
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 186.0 nM 10.1021/acs.jmedchem.9b01769
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 190.0 nM 10.1016/j.bmc.2016.05.010
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 194.0 nM 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 196.0 nM 10.1021/acs.jmedchem.2c00468
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 200.0 nM 10.1021/jm050744t
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 204.8 nM 10.1016/j.ejmech.2022.114512
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 210.0 nM 10.1016/j.bmc.2016.07.041
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 210.0 nM 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 210.0 nM 10.1016/j.ejmech.2015.11.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 210.0 nM 10.1016/j.ejmech.2017.02.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 210.0 nM 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 212.0 nM 10.1016/j.bmc.2021.116239
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 218.0 nM 10.1016/j.bmcl.2007.01.025
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 220.0 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 222.0 nM 10.1016/j.bmc.2010.05.081
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 225.0 nM 10.1016/j.ejmech.2016.02.068
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 228.0 nM 10.1016/j.ejmech.2015.08.007
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 230.0 nM 10.1016/j.bmc.2014.08.001
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 235.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 240.0 nM 10.1016/j.ejmech.2019.111864
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 240.0 nM 10.1021/acs.jmedchem.8b01729
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 244.0 nM 10.1016/j.bmc.2018.12.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 244.0 nM 10.1021/acs.jmedchem.1c00987
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 250.0 nM 10.1016/j.ejmech.2019.111619
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 258.37 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 260.0 nM 10.1016/j.ejmech.2019.111619
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 260.0 nM 10.1016/j.ejmech.2020.113051
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 262.0 nM 10.1016/j.ejmech.2020.112811
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 264.0 nM 10.1016/j.ejmech.2020.112237
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 265.0 nM 10.1021/acs.jmedchem.1c01015
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 267.0 nM 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 268.0 nM 10.1016/j.bmc.2021.116239
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 269.0 nM 10.1021/acs.jmedchem.1c00708
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 269.0 nM 10.1021/acs.jmedchem.1c01015
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 269.0 nM 10.1021/acs.jmedchem.1c01676
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 270.0 nM 10.1016/j.bmc.2014.03.020
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 270.0 nM 10.1016/j.ejmech.2019.111619
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 270.0 nM 10.1021/acs.jmedchem.8b01729
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 273.0 nM 10.1016/j.ejmech.2020.113063
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 273.3 nM 10.1016/j.bmc.2021.116195
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 274.0 nM 10.1021/acs.jmedchem.1c00987
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 275.0 nM 10.1021/jm040840e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 280.0 nM 10.1016/j.bmcl.2006.01.066
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 280.0 nM 10.1016/j.bmcl.2006.05.073
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 290.0 nM 10.1021/acs.jmedchem.9b01446
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 298.5 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 300.0 nM 10.1016/j.bmc.2007.09.015
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 300.0 nM 10.1021/jm050744t
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 307.0 nM 10.1021/acs.jmedchem.1c01015
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 310.0 nM 10.1016/j.ejmech.2017.07.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 310.0 nM 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 313.0 nM 10.1016/j.bmcl.2006.05.096
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 314.0 nM 10.1016/j.ejmech.2020.112811
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 315.0 nM 10.1021/jm300477h
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 317.0 nM 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 317.0 nM 10.1016/j.ejmech.2020.112696
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 317.0 nM 10.1021/acs.jmedchem.6b01906
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 317.0 nM 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 320.0 nM 10.1016/j.ejmech.2014.02.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 320.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 330.0 nM 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 330.0 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 332.0 nM 10.1016/j.bmc.2021.116239
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 340.0 nM 10.1016/j.bmc.2016.07.041
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 340.0 nM 10.1016/j.ejmech.2015.11.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 340.0 nM 10.1016/j.ejmech.2017.02.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 340.0 nM 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 340.0 nM 10.1016/j.ejmech.2020.113051
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 340.0 nM 10.1021/jm201308v
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 340.0 nM 10.1021/jm500284x
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 343.4 nM 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 348.0 nM 10.1016/j.ejmech.2015.08.007
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 360.0 nM 10.1021/jm030558s
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 365.0 nM 10.1016/j.ejmech.2020.112811
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 380.0 nM 10.1016/j.bmc.2008.01.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 380.0 nM 10.1016/j.ejmech.2020.113051
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 390.0 nM 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 390.0 nM 10.1021/jm800340w
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 400.0 nM 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 410.0 nM 10.1021/acs.jmedchem.1c01676
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 416.6 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 440.0 nM 10.1016/j.ejmech.2012.04.004
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 443.0 nM 10.1016/j.bmc.2011.07.023
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 460.0 nM 10.1016/j.bmc.2013.08.040
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 465.0 nM 10.1021/acs.jmedchem.1c01015
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 500.0 nM 10.1016/j.bmcl.2008.06.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 507.0 nM 10.1016/j.bmc.2014.02.030
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 510.0 nM 10.1016/j.bmc.2011.10.002
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 510.0 nM 10.1016/j.ejmech.2013.04.052
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 510.0 nM 10.1039/C3MD00247K
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 520.0 nM 10.1016/j.bmc.2013.09.051
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 520.0 nM 10.1016/j.bmc.2013.10.033
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 520.0 nM 10.1016/j.bmcl.2013.10.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 525.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 530.0 nM 10.1021/acs.jmedchem.1c00535
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 550.0 nM 10.1016/j.bmc.2012.04.030
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 550.0 nM 10.1016/j.bmc.2012.07.026
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 560.0 nM 10.1016/j.bmc.2010.05.036
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 560.0 nM 10.1016/j.bmc.2011.08.025
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 560.0 nM 10.1021/acs.jmedchem.1c01676
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 570.0 nM 10.1016/j.bmcl.2012.09.062
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 570.0 nM 10.1016/j.ejmech.2012.02.019
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 590.0 nM 10.1016/j.bmc.2012.12.049
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 630.0 nM 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 633.5 nM 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 760.0 nM 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 760.0 nM 10.1016/j.ejmech.2020.112696
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 760.0 nM 10.1021/acs.jmedchem.6b01906
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 760.0 nM 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 814.9 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 836.0 nM 10.1021/acsmedchemlett.5b00254
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 870.0 nM 10.1021/acsmedchemlett.5b00254
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 889.0 nM 10.1021/np200855d
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 980.0 nM 10.1021/jm300477h
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1000.0 nM 10.1016/j.bmcl.2010.09.034
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1000.0 nM 10.1128/aac.01064-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1016.1 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1080.0 nM 10.1016/j.ejmech.2020.112071
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1382.1 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1460.0 nM 10.1016/j.ejmech.2006.11.014
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1560.0 nM 10.1021/acs.jmedchem.0c00117
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1570.0 nM 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1570.0 nM 10.1021/jm800340w
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1600.0 nM 10.1021/jm201308v
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1608.4 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1615.0 nM 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 1970.0 nM 10.1021/jm500284x
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2000.0 nM 10.1021/acs.jmedchem.1c01758
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2030.0 nM 10.1021/acs.jmedchem.0c00117
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2500.0 nM 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2526.0 nM 10.1016/j.bmcl.2006.04.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 2526.0 nM 10.1016/j.bmcl.2006.05.096
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3000.0 nM 10.1016/j.bmc.2007.09.015
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3170.0 nM 10.1021/acs.jmedchem.0c00117
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 3700.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6000.0 nM 10.1021/jm500139a
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 6600.0 nM 10.1016/j.bmc.2012.07.026
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7000.0 nM 10.1016/j.ejmech.2009.08.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 7000.0 nM 10.1021/jm500139a
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 8500.0 nM 10.1016/j.bmc.2020.115927
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10000.0 nM 10.1021/acs.jmedchem.1c01758
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10000.0 nM 10.1021/jm070811e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 10000.0 nM 10.1021/jm801438e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 30000.0 nM 10.1021/acs.jmedchem.1c01758
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 183630.0 nM 10.1016/j.bmc.2016.03.043
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 nan None 10.1016/j.bmc.2016.05.010
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 nan None 10.1016/j.bmc.2016.07.041
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 nan None 10.1016/j.ejmech.2019.111864
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC50 nan None 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC90 1.8 uM 10.1021/jm031147e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC95 0.008 uM 10.1128/aac.01064-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC95 3.8 nM 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC95 8.4 nM 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC95 38.0 nM 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC95 89.0 nM 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC95 245.0 nM 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC95 322.0 nM 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC95 1734.0 nM 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC95 3394.0 nM 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC99 0.0001 uM 10.1021/jm500139a
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC99 0.01 uM 10.1021/jm500139a
Human immunodeficiency virus 1 Human immunodeficiency virus 1 EC99 nan None 10.1021/jm500139a
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 0.001 uM 10.1016/j.bmcl.2008.09.070
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 0.008 uM 10.1016/j.bmcl.2008.09.070
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 0.01 uM 10.1021/jm020949r
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 0.04 uM 10.1021/jm020949r
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 0.133 uM 10.1016/j.bmcl.2008.09.070
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 0.3 uM 10.1021/jm020949r
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 0.35 uM 10.1021/jm020949r
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 2.7 uM 10.1021/jm020949r
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 3.0 nM 10.1021/jm070488f
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 7.0 nM 10.1021/jm070488f
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 10.0 nM 10.1021/jm070488f
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 200.0 nM 10.1021/jm070488f
Human immunodeficiency virus 1 Human immunodeficiency virus 1 ED50 20000.0 nM 10.1021/jm070488f
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.17 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.2 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.3 None 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.38 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.51 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.71 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.73 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.77 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.81 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.83 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.86 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.88 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.9 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 0.9 None 10.1128/aac.01593-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 1.0 None 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 1.0 None 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 1.0 None 10.1128/aac.01593-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 1.16 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 1.2 None 10.1128/aac.01593-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 1.3 None 10.1128/aac.01593-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 1.7 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 1.9 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 2.4 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 2.4 None 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 2.5 None 10.1128/aac.01594-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 2.9 None 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 3.1 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 3.2 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 3.2 None 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 3.6 None 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 4.0 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 5.2 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 5.4 None 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 8.1 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 9.0 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 13.6 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 16.0 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 16.3 None 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 17.0 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 21.3 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 23.0 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 26.0 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 33.7 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 56.0 None 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 63.0 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 79.8 None 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 115.0 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 137.7 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 154.0 None 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 164.1 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 300.0 None 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 461.5 None 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 538.0 None 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 700.0 None 10.1128/aac.00870-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FC 2394.0 None 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 0.2 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 0.5 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 0.7 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 0.8 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 0.9 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 1.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 1.2 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 1.3 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 1.4 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 1.5 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 1.6 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 1.7 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 2.1 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 2.5 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 2.9 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 3.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 3.3 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 4.1 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 4.4 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 4.5 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 5.3 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 5.7 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 6.7 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 8.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 8.2 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 8.6 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 8.7 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 10.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 14.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 16.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 17.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 18.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 26.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 28.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 31.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 37.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 43.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 47.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 52.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 64.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 71.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 72.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 77.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 86.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 97.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 100.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 300.0 None 10.1021/jm0708230
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Fold change 400.0 None 10.1128/aac.01032-06
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FT50 9.4 hr 10.1016/j.ejmech.2020.112071
Human immunodeficiency virus 1 Human immunodeficiency virus 1 FT50 10.1 hr 10.1021/acs.jnatprod.7b00659
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.00036 ug.mL-1 10.1124/dmd.112.049601
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.00051 ug.mL-1 10.1124/dmd.112.049601
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.09 nM 10.1016/j.bmc.2008.11.075
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.4 nM 10.1021/acs.jnatprod.6b00878
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.4 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.4 nM 10.1021/jm801322h
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.6 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.7 nM 10.1016/j.bmc.2019.06.044
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.7 nM 10.1021/acs.jnatprod.7b00659
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.8 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.8 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.84 nM 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.9 nM 10.1016/j.bmc.2019.06.044
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.9 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 0.9 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.0 nM 10.1016/j.bmcl.2006.10.082
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.0 nM 10.1016/s0960-894x(01)00412-7
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.0 nM 10.1021/acs.jnatprod.7b00659
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.0 nM 10.1021/jm040072r
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.0 nM 10.1021/jm0407658
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.0 nM 10.1021/jm040829e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.0 nM 10.1021/jm0408621
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.0 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.0 nM 10.1021/jm900802y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.2 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.3 nM 10.1016/j.bmc.2009.02.039
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.3 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.3 None 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.4 nM 10.1021/acs.jnatprod.6b00829
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.4 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.5 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.5 nM 10.1021/np500253m
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.6 nM 10.1021/jm050670l
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.7 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.8 nM 10.1016/j.bmcl.2010.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.8 nM 10.1016/j.bmcl.2010.08.068
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.8 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.8 nM 10.1021/jm050670l
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.8 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.99 nM 10.1016/j.bmcl.2006.10.082
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1.99 nM 10.1021/jm900802y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.0 nM 10.1016/s0960-894x(01)00331-6
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.0 nM 10.1016/s0960-894x(01)00412-7
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.0 nM 10.1021/acs.jmedchem.6b00730
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.0 nM 10.1021/jm0407658
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.0 nM 10.1021/jm040829e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.0 nM 10.1021/jm0408621
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.0 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.0 nM 10.1039/C0MD00009D
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.1 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.3 nM 10.1016/j.bmc.2019.06.044
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.3 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.4 None 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.5 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.7 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2.93 nM 10.1021/jm049606e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 3.0 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 3.0 nM 10.1039/C0MD00009D
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 3.1 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 3.6 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 3.98 nM 10.1016/j.bmcl.2006.10.082
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 3.98 nM 10.1021/jm900802y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 4.0 nM 10.1021/acs.jnatprod.7b00014
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 4.0 nM 10.1021/acs.jnatprod.7b00659
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 5.0 nM 10.1021/jm0407658
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 5.0 nM 10.1021/jm0408621
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 5.01 nM 10.1021/jm900802y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 5.1 None 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 5.4 nM 10.1016/j.bmc.2019.06.044
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 5.65 nM 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 5.7 nM 10.1016/j.bmcl.2010.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 5.7 nM 10.1016/j.bmcl.2010.08.068
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 5.8 None 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 5.9 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 6.0 nM 10.1016/j.bmcl.2010.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 6.0 nM 10.1021/jm0407658
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 6.0 nM 10.1021/jm0408621
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 6.3 nM 10.1021/jm900802y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 7.0 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 7.2 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 10.0 nM 10.1021/jm0407658
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 10.0 nM 10.1021/jm0408621
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 10.0 nM 10.1021/jm900802y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 11.0 nM 10.1016/j.bmc.2022.117083
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 12.0 nM 10.1021/jm801470b
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 17.0 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 18.0 nM 10.1039/C0MD00009D
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 18.1 nM 10.1016/j.bmcl.2010.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 18.1 nM 10.1016/j.bmcl.2010.08.068
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 20.0 nM 10.1021/jm0407658
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 20.0 None 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 21.0 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 21.0 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 22.0 nM 10.1021/jm801470b
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 22.6 nM 10.1016/j.ejmech.2014.05.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 24.0 None 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 25.0 nM 10.1021/jm0408621
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 25.0 nM 10.1021/jm050670l
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 25.1 nM 10.1021/jm900802y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 27.0 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 39.8 nM 10.1016/j.bmcl.2006.10.082
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 39.8 nM 10.1021/jm900802y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 40.0 nM 10.1016/s0960-894x(01)00412-7
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 40.0 nM 10.1021/jm0407658
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 40.0 nM 10.1021/jm040829e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 40.0 nM 10.1021/jm0408621
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 44.0 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 46.0 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 56.0 nM 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 58.8 nM 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 60.0 nM 10.1021/np400029d
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 65.0 nM 10.1039/C0MD00009D
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 82.8 nM 10.1016/j.bmcl.2010.08.068
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 83.0 nM 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 89.0 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 93.0 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 94.0 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 100.0 nM 10.1016/j.bmcl.2010.08.068
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 130.0 nM 10.1021/jm801470b
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 140.0 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 150.0 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 150.0 nM 10.1021/jm0407658
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 154.0 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 158.0 nM 10.1016/j.bmcl.2006.10.082
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 158.0 nM 10.1016/s0960-894x(01)00412-7
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 158.0 nM 10.1021/jm040829e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 158.0 nM 10.1021/jm0408621
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 158.0 nM 10.1021/jm900802y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 160.0 nM 10.1016/j.ejmech.2014.05.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 160.0 nM 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 160.0 nM 10.1021/jm801470b
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 162.75 nM 10.1016/j.ejmech.2018.07.067
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 250.0 nM 10.1021/jm0407658
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 251.0 nM 10.1021/jm0408621
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 251.0 nM 10.1021/jm900802y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 480.0 nM 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 485.0 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 490.0 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 500.0 nM 10.1016/j.bmcl.2010.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 760.0 nM 10.1021/jm801470b
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1000.0 nM 10.1016/j.bmcl.2006.10.082
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1000.0 nM 10.1016/j.bmcl.2010.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1000.0 nM 10.1021/jm900802y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1198.0 nM 10.1021/jm8004493
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 1500.0 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 2490.0 nM 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 10000.0 nM 10.1016/j.bmcl.2006.05.096
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 10000.0 nM 10.1016/s0960-894x(01)00412-7
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 10000.0 nM 10.1021/jm0407658
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 10000.0 nM 10.1021/jm040829e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 10000.0 nM 10.1021/jm0408621
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 26000.0 nM 10.1021/acs.jmedchem.6b00730
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 106000.0 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC50 910000.0 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 1.7 nM 10.1016/s0960-894x(00)00662-4
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 1.7 nM 10.1016/s0960-894x(01)00192-5
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 1.7 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 2.8 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 8.5 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 17.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 33.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 64.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 77.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 120.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 650.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 1056.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 2400.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 8100.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 15700.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC90 309500.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC95 4.3 nM 10.1016/j.bmcl.2010.06.083
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC95 4.6 nM 10.1021/jm800856c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC95 8.0 nM 10.1016/j.bmcl.2010.06.083
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC95 38.0 nM 10.1016/j.bmcl.2010.06.083
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC95 42.0 nM 10.1021/jm800856c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC95 87.0 nM 10.1021/jm800856c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC95 232.0 nM 10.1016/j.bmcl.2010.06.083
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC95 245.0 nM 10.1021/jm800856c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 IC95 272.0 nM 10.1016/j.bmcl.2010.06.083
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Inhibition 15.0 % 10.1016/j.ejmech.2021.113498
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Inhibition 24.0 % 10.1128/aac.00759-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Inhibition 42.5 % 10.1021/np2001896
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Inhibition 85.0 % 10.1016/j.ejmech.2021.113498
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Inhibition 99.97 % 10.1016/j.ejmech.2019.111900
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Inhibition 100.0 % 10.1021/acs.jnatprod.7b00659
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Inhibition nan % 10.1016/j.ejmech.2011.08.011
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Inhibition nan % 10.1021/acs.jnatprod.6b00878
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Inhibition nan % 10.1021/np200855d
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.4 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.4 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.5 None 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.6 None 10.1128/aac.00210-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.73 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.8 None 10.1128/aac.00210-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.8 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.83 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.88 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.9 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.92 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.93 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.94 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.95 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 0.98 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.0 None 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.0 None 10.1128/aac.00759-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.0 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.0 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.0 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.0 None 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.1 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.1 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.1 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.1 None 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.2 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.2 None 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.3 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.3 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.3 None 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.4 None 10.1016/j.ejmech.2011.08.011
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.4 None 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.4 None 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.4 None 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.4 None 10.1021/jm201308v
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.4 None 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.4 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.4 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.4 None 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.5 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.5 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.5 None 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.5 None 10.1128/aac.01480-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.6 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.7 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.7 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.9 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1.9 None 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.0 None 10.1021/jm500284x
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.0 None 10.1128/aac.00759-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.0 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.0 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.0 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.0 None 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.0 None 10.1128/aac.01480-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.1 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.1 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.17 None 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.2 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.2 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.27 None 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.3 None 10.1128/aac.01313-07
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.4 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.5 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.6 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.7 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.8 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 2.9 None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 3.0 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 3.0 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 3.4 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 3.7 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 3.8 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 4.0 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 4.3 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 4.6 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 4.8 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 5.0 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 5.0 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 5.7 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 5.9 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 6.0 None 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 6.0 None 10.1021/jm800340w
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 6.0 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 6.4 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 6.5 None 10.1128/aac.01480-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 7.2 None 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 8.1 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 8.2 None 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 8.2 None 10.1016/j.ejmech.2020.112696
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 8.2 None 10.1021/acs.jmedchem.6b01906
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 8.2 None 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 8.9 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 9.3 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 9.5 None 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 10.0 None 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 10.0 None 10.1016/j.ejmech.2020.112696
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 10.0 None 10.1021/acs.jmedchem.6b01906
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 10.0 None 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 11.0 None 10.1021/jm300477h
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 12.1 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 12.3 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 12.79 None 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 13.0 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 13.0 None 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 13.1 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 14.2 None 10.1016/j.ejmech.2011.08.011
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 15.0 None 10.1128/aac.01480-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 16.3 None 10.1021/acsmedchemlett.7b00524
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 16.7 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 16.9 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 17.3 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 18.7 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 20.0 None 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 20.0 None 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 20.0 None 10.1016/j.ejmech.2020.112696
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 20.0 None 10.1021/acs.jmedchem.6b01906
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 20.0 None 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 20.3 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 23.0 None 10.1021/jm301294g
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 24.0 None 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 25.0 None 10.1016/j.ejmech.2015.01.042
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 25.0 None 10.1021/jm300477h
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 25.7 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 28.3 None 10.1016/j.ejmech.2011.08.011
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 30.0 None 10.1016/j.bmcl.2018.03.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 32.5 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 35.0 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 35.34 None 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 35.5 None 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 36.5 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 42.0 None 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 42.6 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 47.0 None 10.1021/jm201308v
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 48.0 None 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 48.0 None 10.1016/j.ejmech.2020.112696
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 48.0 None 10.1021/acs.jmedchem.6b01906
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 48.0 None 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 49.0 None 10.1021/jm500284x
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 49.1 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 50.0 None 10.1021/jm300477h
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 54.8 None 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 56.0 None 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 56.0 None 10.1021/jm800340w
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 56.4 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 57.0 None 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 57.2 None 10.1128/aac.00210-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 58.0 None 10.1021/acsmedchemlett.5b00254
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 61.0 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 68.0 None 10.1016/j.ejmech.2018.03.059
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 70.0 None 10.1016/j.bmc.2013.10.033
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 72.3 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 73.1 None 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 83.6 None 10.1016/j.bmc.2012.04.030
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 90.0 None 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 92.17 None 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 94.8 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 96.0 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 114.13 None 10.1016/j.bmc.2021.116531
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 186.0 None 10.1016/j.bmc.2011.08.025
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 200.0 None 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 220.0 None 10.1021/jm201308v
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 221.0 None 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 222.0 None 10.1021/np200855d
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 224.0 None 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 224.0 None 10.1021/jm800340w
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 237.5 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 281.0 None 10.1021/jm500284x
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 281.0 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 327.0 None 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 486.0 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 530.0 None 10.1128/aac.00984-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 575.8 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 925.0 None 10.1021/acs.jmedchem.0c00117
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1206.0 None 10.1021/acs.jmedchem.0c00117
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1695.0 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1812.0 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 1881.0 None 10.1021/acs.jmedchem.0c00117
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 5660.0 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 10866.0 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 12931.1 None 10.1128/aac.00986-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 nan None 10.1016/j.ejmech.2008.10.032
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio EC50 nan None 10.1128/aac.01209-10
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 0.3 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 0.4 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 0.5 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 0.6 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 0.7 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 0.8 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 0.8 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 0.9 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 1.0 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 1.0 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 1.2 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 1.2 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 1.3 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 1.4 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 1.5 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 1.5 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 1.6 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 1.7 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 1.9 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 2.0 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 2.0 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 2.1 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 2.1 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 2.6 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 2.8 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 2.9 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 2.9 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 3.0 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 3.6 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 3.8 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 5.4 None 10.1016/j.ejmech.2016.07.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 7.6 None 10.1016/j.bmc.2019.06.044
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 9.9 None 10.1128/aac.01335-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 10.1 None 10.1016/j.bmcl.2010.08.068
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 11.0 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 38.0 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 39.0 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 42.0 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 43.0 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 56.0 None 10.1016/j.ejmech.2016.07.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 56.4 None 10.1016/j.ejmech.2016.07.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 79.8 None 10.1016/j.ejmech.2016.07.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 138.0 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 154.0 None 10.1016/j.ejmech.2016.07.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 183.0 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 461.5 None 10.1016/j.ejmech.2016.07.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 538.0 None 10.1016/j.ejmech.2016.07.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 2394.0 None 10.1016/j.ejmech.2016.07.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 10000.0 None 10.1128/aac.01156-08
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Ratio IC50 13269.2 None 10.1016/j.ejmech.2016.07.047
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Selectivity index 10000.0 uM 10.1021/jm0407658
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Selectivity index 10000.0 None 10.1021/jm040838n
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Selectivity ratio 2.0 None 10.1016/j.bmcl.2006.04.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Selectivity ratio 18.0 None 10.1128/aac.01795-09
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Selectivity ratio 20.0 None 10.1016/j.bmcl.2006.04.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Selectivity ratio 50.0 None 10.1021/acsmedchemlett.5b00254
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Selectivity ratio 64.0 None 10.1016/j.bmcl.2006.04.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 Selectivity ratio 5000.0 None 10.1016/j.bmcl.2006.04.012
Human immunodeficiency virus 1 Human immunodeficiency virus 1 SI 10000.0 uM 10.1021/jm0408621
Human immunodeficiency virus 1 Human immunodeficiency virus 1 TIME 8.8 hr 10.1016/j.ejmech.2014.07.072
Human immunodeficiency virus 1 Human immunodeficiency virus 1 TIME 13.06 hr 10.1021/np400683h
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 protease IC90 64.0 nM 10.1016/s0960-894x(00)00662-4
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 protease IC90 240.0 nM 10.1016/s0960-894x(00)00662-4
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 protease IC90 7300.0 nM 10.1016/s0960-894x(00)00624-7
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 protease IC90 7300.0 nM 10.1016/s0960-894x(00)00662-4
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Activity 0.0009 uM 10.1021/jm010580q
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Activity 0.478 uM 10.1021/jm010580q
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Activity 3.1 % 10.1039/C4MD00399C
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Activity nan None 10.1128/aac.01308-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase C90 7300.0 nM 10.1016/s0960-894x(01)00331-6
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 1.0 nM 10.1016/j.bmcl.2006.03.080
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 1.0 nM 10.1016/j.bmcl.2008.06.072
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 2.0 nM 10.1016/j.bmcl.2008.06.072
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 2.85 nM 10.1021/acsmedchemlett.8b00054
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 3.0 nM 10.1016/j.ejmech.2018.09.013
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 4.0 nM 10.1016/j.bmc.2017.12.033
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 4.0 nM 10.1021/jm050273a
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 5.0 nM 10.1016/j.bmc.2017.12.033
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 5.0 nM 10.1016/j.ejmech.2016.06.026
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 5.19 nM 10.1021/acs.jmedchem.7b00332
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 5.2 nM 10.1016/j.bmc.2017.03.009
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 5.4 nM 10.1021/acs.jmedchem.1c00128
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 8.2 nM 10.1021/acs.jmedchem.7b00332
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 16.0 nM 10.1016/j.bmc.2017.12.033
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 29.0 nM 10.1016/j.bmc.2017.12.033
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 34.0 nM 10.1016/j.bmcl.2008.06.072
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 38.0 nM 10.1016/j.bmc.2017.12.033
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 44.0 nM 10.1016/j.bmc.2017.12.033
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 44.7 nM 10.1021/acs.jmedchem.1c00128
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 57.0 nM 10.1016/j.bmc.2017.12.033
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 57.0 nM 10.1016/j.bmcl.2006.03.080
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 80.1 nM 10.1021/acs.jmedchem.7b00332
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 91.5 nM 10.1021/acs.jmedchem.1c00128
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 101.0 nM 10.1016/j.ejmech.2016.06.026
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 115.0 nM 10.1021/acs.jmedchem.7b00332
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 156.17 nM 10.1016/j.ejmech.2018.07.067
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 160.0 nM 10.1016/j.bmc.2017.03.009
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 200.0 nM 10.1016/j.bmcl.2006.03.080
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 224.0 nM 10.1021/acsmedchemlett.8b00054
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 300.0 nM 10.1016/j.bmcl.2006.03.080
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 308.0 nM 10.1021/acs.jmedchem.7b00332
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 348.0 nM 10.1021/acs.jmedchem.7b00332
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase EC50 514.0 nM 10.1021/acs.jmedchem.7b00332
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ED50 0.005 uM 10.1021/jm990095j
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ED50 0.016 uM 10.1021/jm990095j
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ED50 0.06 uM 10.1021/jm990095j
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ED50 0.14 uM 10.1021/jm990095j
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 0.003 ug.mL-1 10.1021/jm001095i
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 0.007 ug.mL-1 10.1021/jm001095i
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 0.091 nM 10.1016/j.ejmech.2019.111900
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 0.091 nM 10.1016/j.ejmech.2021.113498
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 0.166 nM 10.1039/C4MD00282B
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 0.31 nM 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 0.42 nM 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 0.75 nM 10.1021/jm030255y
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 0.8 nM 10.1016/j.bmcl.2006.02.049
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 1.0 nM 10.1021/jm800856c
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 1.3 nM 10.1007/s00044-009-9192-x
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 1.3 nM 10.1016/j.ejmech.2008.10.032
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 2.0 nM 10.1016/j.ejmech.2018.01.016
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 3.0 nM 10.1016/j.ejmech.2012.01.056
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 4.0 nM 10.1016/j.bmc.2008.06.012
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 4.0 nM 10.1016/j.bmc.2009.06.068
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 4.0 nM 10.1016/j.bmc.2009.12.059
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 4.0 nM 10.1016/j.bmcl.2004.04.008
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 4.0 nM 10.1016/j.bmcl.2007.01.025
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 4.0 nM 10.1016/j.bmcl.2018.10.010
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 4.0 nM 10.1021/jm990095j
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 6.0 nM 10.1016/j.bmcl.2006.02.049
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 6.0 nM 10.1016/j.ejmech.2019.05.011
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 6.0 nM 10.1021/acsmedchemlett.8b00054
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 6.0 nM 10.1021/jm990095j
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 7.0 nM 10.1016/j.bmc.2018.12.039
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 7.0 nM 10.1021/acs.jmedchem.8b01729
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 7.079 nM 10.1021/acs.jmedchem.8b01729
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 7.2 nM 10.1021/jm800856c
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 7.2 nM 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 8.0 nM 10.1016/j.ejmech.2021.113204
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 8.1 nM 10.1016/j.ejmech.2020.113051
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 8.128 nM 10.1016/j.ejmech.2020.113051
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 9.5 nM 10.1016/j.bmcl.2006.02.049
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 10.0 nM 10.1016/j.bmc.2016.04.010
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 10.0 nM 10.1016/j.bmcl.2016.06.065
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 10.0 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 10.0 nM 10.1021/acs.jmedchem.1c00128
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 10.0 nM 10.1021/acs.jmedchem.1c00708
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 10.0 nM 10.1021/acs.jmedchem.1c01676
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 10.0 nM 10.1039/C3MD00036B
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 10.0 nM 10.1039/C3MD00225J
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 10.0 nM 10.1128/aac.00749-06
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 10.2 nM 10.1128/aac.01559-08
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 11.0 nM 10.1016/j.ejmech.2022.114512
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 11.0 nM 10.1021/acs.jmedchem.2c00468
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 12.0 nM 10.1016/j.ejmech.2015.02.032
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 14.0 nM 10.1016/j.bmc.2007.12.046
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 14.0 nM 10.1016/j.ejmech.2019.111619
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 14.0 nM 10.1021/jm049252r
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 14.0 nM 10.1021/jm801322h
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 17.0 nM 10.1074/jbc.m608274200
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 18.0 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 18.9 nM 10.1021/jm800856c
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 19.0 nM 10.1016/j.bmc.2017.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 19.0 nM 10.1016/j.bmc.2017.12.033
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 20.0 nM 10.1016/j.bmc.2008.05.010
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 20.0 nM 10.1016/j.bmc.2018.03.003
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 20.0 nM 10.1016/j.ejmech.2014.09.054
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 20.0 nM 10.1021/jm049252r
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 22.0 nM 10.1016/j.bmc.2015.01.002
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 22.0 nM 10.1016/j.bmc.2015.03.037
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 22.0 nM 10.1016/j.bmc.2015.06.048
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 22.0 nM 10.1016/j.bmc.2015.09.020
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 24.0 nM 10.1016/j.bmc.2014.11.032
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 30.0 nM 10.1016/j.bmc.2017.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 30.0 nM 10.1016/j.ejmech.2019.111603
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 30.0 nM 10.1021/acs.jmedchem.9b01446
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 30.0 nM 10.1021/acsmedchemlett.7b00524
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 30.0 nM 10.1039/C3MD00036B
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 30.0 nM 10.1039/C3MD00225J
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 30.0 nM 10.1128/aac.01795-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 32.0 nM 10.1016/j.bmc.2013.12.045
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 35.0 nM 10.1016/j.ejmech.2015.08.007
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 35.0 nM 10.1021/acs.jmedchem.1c00535
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 36.0 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 37.0 nM 10.1016/j.bmc.2013.08.040
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 37.0 nM 10.1039/C3MD00247K
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 38.0 nM 10.1016/j.bmc.2014.02.030
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 38.0 nM 10.1016/j.ejmech.2015.11.025
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 38.0 nM 10.1016/j.ejmech.2016.05.054
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 38.0 nM 10.1016/s0960-894x(01)00239-6
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 38.0 nM 10.1021/acs.jmedchem.8b00843
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 40.0 nM 10.1007/s00044-007-9004-0
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 40.0 nM 10.1016/j.ejmech.2017.07.012
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 40.0 nM 10.1021/jm050257d
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 40.0 nM 10.1021/jm801322h
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 42.0 nM 10.1128/aac.00749-06
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 44.0 nM 10.1016/j.ejmech.2015.04.050
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 47.0 nM 10.1016/s0960-894x(00)00624-7
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 47.0 nM 10.1016/s0960-894x(00)00662-4
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 47.0 nM 10.1016/s0960-894x(01)00012-9
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 47.0 nM 10.1016/s0960-894x(99)00672-1
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 47.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 48.0 nM 10.1016/j.ejmech.2013.04.052
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 48.0 nM 10.1016/s0960-894x(00)00321-8
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 48.0 nM 10.1016/s0960-894x(01)00331-6
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 48.0 nM 10.1016/s0960-894x(99)00486-2
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 48.0 nM 10.1016/s0960-894x(99)00565-x
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 50.0 nM 10.1016/j.bmc.2009.12.059
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 50.0 nM 10.1016/j.bmc.2016.04.010
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 50.0 nM 10.1021/jm990095j
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 50.0 nM 10.1039/C3MD00036B
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 50.0 nM 10.1039/C3MD00225J
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 54.0 nM 10.1016/j.bmcl.2006.02.049
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 57.0 nM 10.1016/j.bmc.2017.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 57.0 nM 10.1128/aac.01795-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 60.0 nM 10.1039/C3MD00036B
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 60.0 nM 10.1128/aac.00749-06
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 61.0 nM 10.1021/jm990095j
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 70.0 nM 10.1016/j.bmc.2016.04.010
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 80.0 nM 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 80.0 nM 10.1016/j.ejmech.2020.112696
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 80.0 nM 10.1021/acs.jmedchem.6b01906
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 80.0 nM 10.1021/jm300477h
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 80.0 nM 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 80.0 nM 10.1039/C3MD00036B
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 80.0 nM 10.1039/C3MD00225J
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 93.0 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 100.0 nM 10.1016/j.bmc.2017.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 112.0 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 120.0 nM 10.1016/j.bmcl.2013.10.059
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 120.0 nM 10.1021/jm050257d
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 120.0 nM 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 126.0 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 140.0 nM 10.1039/C3MD00036B
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 140.0 nM 10.1039/C3MD00225J
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 150.0 nM 10.1021/jm050257d
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 160.0 nM 10.1021/jm050257d
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 180.0 nM 10.1016/j.bmc.2020.115927
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 200.0 nM 10.1016/j.bmc.2009.12.059
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 216.0 nM 10.1128/aac.00800-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 250.0 nM 10.1016/j.bmc.2016.04.010
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 260.0 nM 10.1016/j.ejmech.2019.111874
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 270.0 nM 10.1016/j.bmc.2017.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 280.0 nM 10.1016/j.ejmech.2015.02.032
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 360.0 nM 10.1016/j.bmc.2018.03.003
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 364.0 nM 10.1021/jm801322h
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 380.0 nM 10.1021/jm050257d
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 400.0 nM 10.1021/acs.jmedchem.6b01906
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 400.0 nM 10.1021/jm300477h
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 400.0 nM 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 414.0 nM 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 480.0 nM 10.1016/j.ejmech.2022.114471
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 500.0 nM 10.1016/j.bmc.2009.12.059
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 500.0 nM 10.1021/jm049252r
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 580.0 nM 10.1039/C3MD00036B
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 580.0 nM 10.1039/C3MD00225J
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 630.0 nM 10.1016/j.bmc.2017.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 680.0 nM 10.1016/j.ejmech.2012.01.056
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 680.0 nM 10.1016/j.ejmech.2015.02.032
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 730.0 nM 10.1016/j.bmc.2016.04.010
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 740.0 nM 10.1016/j.bmc.2016.05.010
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 740.0 nM 10.1128/aac.01795-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 800.0 nM 10.1016/j.bmcl.2006.04.012
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 910.0 nM 10.1128/aac.01795-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 1200.0 nM 10.1016/j.bmc.2016.04.010
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 1200.0 nM 10.1016/j.bmc.2017.05.040
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 1420.0 nM 10.1021/acs.jmedchem.6b00738
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 1520.0 nM 10.1016/j.bmc.2011.08.060
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 2100.0 nM 10.1021/jm049252r
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 20000.0 nM 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 20000.0 nM 10.1016/j.ejmech.2020.112696
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 20000.0 nM 10.1021/acs.jmedchem.6b01906
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 20000.0 nM 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 100000.0 nM 10.1016/j.ejmech.2012.01.056
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 nan None 10.1016/j.bmc.2010.05.036
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 nan None 10.1016/j.ejmech.2012.01.056
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 nan None 10.1016/j.ejmech.2015.02.032
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 nan None 10.1021/jm070382k
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 nan None 10.1021/jm300477h
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 nan None 10.1021/jm5011622
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC50 nan None 10.1074/jbc.m608274200
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 1.7 nM 10.1016/j.ejmech.2015.11.025
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 1.7 nM 10.1016/s0960-894x(00)00624-7
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 1.7 nM 10.1021/acs.jmedchem.8b00843
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 1.9 nM 10.1016/s0960-894x(01)00239-6
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 2.0 nM 10.1016/s0960-894x(00)00321-8
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 2.03 nM 10.1016/s0960-894x(99)00486-2
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 2.03 nM 10.1016/s0960-894x(99)00565-x
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 28.0 nM 10.1021/jm990580e
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 49.0 nM 10.1016/s0960-894x(01)00239-6
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 64.0 nM 10.1016/s0960-894x(00)00624-7
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 64.0 nM 10.1016/s0960-894x(01)00192-5
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 64.0 nM 10.1016/s0960-894x(01)00331-6
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 77.0 nM 10.1016/s0960-894x(01)00331-6
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase IC90 310.0 nM 10.1016/s0960-894x(00)00662-4
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.03 uM 10.1021/jm500284x
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.03 uM 10.1021/jm800340w
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.04 uM 10.1016/j.bmcl.2006.03.080
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.04 uM 10.1021/jm050744t
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.04 uM 10.1021/jm801330n
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.08 uM 10.1021/jm050273a
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.08 uM 10.1021/jm500284x
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.08 uM 10.1021/jm800340w
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.09 uM 10.1021/jm050273a
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.1 uM 10.1016/j.bmcl.2006.03.080
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.1 uM 10.1021/jm050273a
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.1 uM 10.1021/jm050744t
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.1 uM 10.1021/jm801330n
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.2 uM 10.1021/jm050273a
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.4 uM 10.1016/j.bmcl.2006.03.080
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.4 uM 10.1021/jm050273a
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.4 uM 10.1021/jm050744t
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 0.4 uM 10.1021/jm801330n
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 3.0 uM 10.1021/jm500284x
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 3.0 uM 10.1021/jm800340w
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 25.0 uM 10.1021/jm050273a
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 30.0 nM 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 30.0 nM 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 30.0 nM 10.1021/jm201308v
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 80.0 nM 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 80.0 nM 10.1021/jm070488f
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 80.0 nM 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 80.0 nM 10.1021/jm201308v
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 400.0 nM 10.1021/jm070488f
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 3000.0 nM 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 3000.0 nM 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 3000.0 nM 10.1021/jm201308v
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 20000.0 nM 10.1021/jm070488f
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 nan None 10.1021/acs.jmedchem.8b01238
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 nan None 10.1021/jm070488f
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 nan None 10.1021/jm101626c
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 nan None 10.1021/jm201308v
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 nan None 10.1021/jm500284x
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase ID50 nan None 10.1021/jm800340w
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Inhibition 17.6 % 10.1128/aac.01308-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Inhibition 50.0 % 10.1128/aac.00749-06
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Inhibition 93.27 % 10.1016/j.ejmech.2018.07.067
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Inhibition 98.0 % 10.1128/aac.00749-06
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Inhibition 100.0 % 10.1016/j.ejmech.2021.113785
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Inhibition nan % 10.1016/j.bmc.2020.115927
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Inhibition nan % 10.1016/j.ejmech.2021.113785
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Inhibition nan % 10.1128/aac.01455-09
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 0.3 nM 10.1016/j.bmcl.2010.06.083
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 0.4 nM 10.1016/j.bmcl.2010.06.083
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 2.93 nM 10.1021/acs.jmedchem.8b00843
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 3.0 nM 10.1016/s0960-894x(01)00510-8
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 4.0 nM 10.1021/jm801330n
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 8.5 nM 10.1016/j.bmcl.2010.06.083
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 10.0 nM 10.1016/j.bmc.2012.12.027
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 17.0 nM 10.1016/s0960-894x(01)00510-8
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 25.0 nM 10.1016/s0960-894x(01)00510-8
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 30.0 nM 10.1016/j.bmc.2012.12.027
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 30.0 nM 10.1021/jm0010365
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 30.0 nM 10.1021/jm070811e
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 30.0 nM 10.1021/jm801330n
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 30.0 nM 10.1021/jm801395v
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 40.0 nM 10.1021/jm0010365
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 50.0 nM 10.1016/j.bmc.2012.12.027
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 80.0 nM 10.1016/j.bmc.2011.08.025
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 80.0 nM 10.1016/j.bmc.2012.12.027
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 120.0 nM 10.1021/jm0010365
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 120.0 nM 10.1021/jm801395v
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 140.0 nM 10.1016/j.bmc.2012.12.027
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 150.0 nM 10.1021/jm0010365
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 150.0 nM 10.1021/jm801395v
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 160.0 nM 10.1021/jm0010365
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 160.0 nM 10.1021/jm801395v
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 200.0 nM 10.1021/jm801330n
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 300.0 nM 10.1021/jm0010365
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 580.0 nM 10.1016/j.bmc.2011.08.025
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 580.0 nM 10.1016/j.bmc.2012.12.027
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 730.0 nM 10.1016/j.bmc.2011.08.025
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 1500.0 nM 10.1021/jm801330n
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 1600.0 nM 10.1021/jm801330n
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki 3000.0 nM 10.1021/jm070811e
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Ki nan None 10.1021/jm070811e
Human immunodeficiency virus 1 Human immunodeficiency virus type 1 reverse transcriptase Selectivity index 20000.0 None 10.1016/j.bmcl.2004.04.008
Human immunodeficiency virus 1 Protease Activity nan None 10.1128/aac.01308-09
Human immunodeficiency virus 1 Reverse transcriptase EC50 4.8 nM 10.1016/j.ejmech.2020.112549
Human immunodeficiency virus 1 Reverse transcriptase EC50 5.0 nM 10.1016/j.ejmech.2021.113204
Human immunodeficiency virus 1 Reverse transcriptase EC50 7.0 nM 10.1016/j.ejmech.2020.112549
Human immunodeficiency virus 1 Reverse transcriptase EC50 31.0 nM 10.1016/j.ejmech.2021.113204
Human immunodeficiency virus 1 Reverse transcriptase EC50 47.5 nM 10.1016/j.ejmech.2020.112549
Human immunodeficiency virus 1 Reverse transcriptase EC50 71.0 nM 10.1016/j.ejmech.2021.113204
Human immunodeficiency virus 1 Reverse transcriptase EC50 76.0 nM 10.1016/j.ejmech.2020.112549
Human immunodeficiency virus 1 Reverse transcriptase EC50 171.1 nM 10.1016/j.ejmech.2020.112549
Human immunodeficiency virus 1 Reverse transcriptase EC50 260.0 nM 10.1016/j.ejmech.2021.113204
Human immunodeficiency virus 1 Reverse transcriptase EC50 380.0 nM 10.1016/j.ejmech.2021.113204
Human immunodeficiency virus 1 Reverse transcriptase IC50 10.0 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Reverse transcriptase IC50 20.0 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Reverse transcriptase IC50 100.0 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Reverse transcriptase IC50 120.0 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 1 Reverse transcriptase IC50 170.0 nM 10.1016/j.ejmech.2021.113868
Human immunodeficiency virus 2 Human immunodeficiency virus 2 Activity nan None 10.1016/j.bmc.2020.115927
Human immunodeficiency virus 2 Human immunodeficiency virus 2 Activity nan None 10.1021/jm070382k
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 20.0 nM 10.1016/j.bmc.2012.12.049
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 6340.0 nM 10.1016/j.ejmech.2013.04.052
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 6340.0 nM 10.1021/acs.jmedchem.1c01015
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 10000.0 nM 10.1016/j.ejmech.2014.04.027
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 10000.0 nM 10.1021/jm101614j
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 10000.0 nM 10.1021/jm5011622
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 24830.0 nM 10.1128/aac.00986-09
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 31680.0 nM 10.1128/aac.00210-08
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 nan None 10.1016/j.bmc.2011.10.002
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 nan None 10.1016/j.bmc.2013.08.040
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 nan None 10.1016/j.bmc.2013.09.051
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 nan None 10.1016/j.bmc.2014.02.030
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 nan None 10.1016/j.bmc.2014.03.020
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 nan None 10.1016/j.bmc.2014.11.032
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 nan None 10.1016/j.bmc.2015.09.020
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 nan None 10.1016/j.ejmech.2012.04.004
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 nan None 10.1016/j.ejmech.2014.09.054
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 nan None 10.1016/j.ejmech.2015.08.007
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 nan None 10.1016/j.ejmech.2017.02.047
Human immunodeficiency virus 2 Human immunodeficiency virus 2 EC50 nan None 10.1039/C3MD00247K
Human orthopneumovirus Human orthopneumovirus EC50 nan None 10.1016/j.bmc.2015.09.035
Klebsiella pneumoniae Klebsiella pneumoniae Inhibition -2.99 % 10.6019/CHEMBL4513141
Leishmania infantum Leishmania infantum IC50 7400.0 nM 10.1016/j.bmc.2014.08.005
Murine leukemia virus Murine leukemia virus IC50 10000.0 nM 10.1021/acs.jnatprod.7b00659
Mus musculus BV-2 Activity nan None 10.1021/acs.jmedchem.6b01906
Mus musculus Indoleamine 2,3-dioxygenase 2 Inhibition 55.0 % 10.1016/j.bmcl.2012.10.010
Mus musculus Nuclear receptor ROR-gamma Potency 12589.3 nM None
Plasmodium falciparum Plasmodium falciparum IC50 43820.0 nM 10.1016/j.bmc.2014.08.005
Poliovirus 1 Poliovirus 1 EC50 nan None 10.1016/j.bmc.2015.09.035
Pseudomonas aeruginosa Pseudomonas aeruginosa Inhibition 7.84 % 10.6019/CHEMBL4513141
Rattus norvegicus Androgen Receptor AC50 26999.8 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Androgen Receptor AC50 30000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Cyclooxygenase-1 AC50 30000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus GABA receptor alpha-1 subunit AC50 10000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Glutamate (NMDA) receptor subunit zeta 1 AC50 10000.0 nM 10.1038/s41467-023-40064-9
Rattus norvegicus Plasma t1/2 nan None 10.1021/jm070382k
Rattus norvegicus Plasma T1/2 1.481 hr 10.1039/C4MD00282B
Rattus norvegicus Voltage-gated L-type calcium channel alpha-1C subunit AC50 18839.5 nM 10.1038/s41467-023-40064-9
Severe acute respiratory syndrome coronavirus 2 Replicase polyprotein 1ab Inhibition 8.045 % 10.6019/CHEMBL4495564
Severe acute respiratory syndrome coronavirus 2 Replicase polyprotein 1ab Inhibition 13.07 % 10.6019/CHEMBL4495564
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Hit score 0.3102 None 10.1101/2020.04.21.054387
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Inhibition -0.1 % 10.6019/CHEMBL4495565
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Inhibition 0.22 % 10.6019/CHEMBL4495565
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Inhibition 32.07 % 10.21203/rs.3.rs-23951/v1
Severe acute respiratory syndrome coronavirus 2 SARS-CoV-2 Inhibition index -0.107 None 10.1101/2020.04.03.023846
Simian immunodeficiency virus Simian immunodeficiency virus EC50 31680.0 nM 10.1128/aac.00210-08
Staphylococcus aureus Staphylococcus aureus Inhibition 10.66 % 10.6019/CHEMBL4513141
Trypanosoma brucei brucei Trypanosoma brucei brucei IC50 30200.0 nM 10.1016/j.bmc.2014.08.005
Trypanosoma brucei rhodesiense Trypanosoma brucei rhodesiense IC50 19600.0 nM 10.1016/j.bmc.2014.08.005
Trypanosoma cruzi Trypanosoma cruzi IC50 8560.0 nM 10.1016/j.bmc.2014.08.005
Vaccinia virus Vaccinia virus EC50 nan None 10.1016/j.bmc.2015.09.035
Vesicular stomatitis virus Vesicular stomatitis virus EC50 0.43 nM 10.1021/jm3016377
Vesicular stomatitis virus Vesicular stomatitis virus EC50 nan None 10.1016/j.bmc.2015.09.035
Yellow fever virus Yellow fever virus EC50 nan None 10.1016/j.bmc.2015.09.035
None ADMET CC30 2.0 uM 10.1016/j.bmcl.2009.08.080
None ADMET CC50 6340.0 nM 10.1016/j.bmc.2021.116531
None ADMET CC50 10000.0 nM 10.1016/j.bmcl.2006.09.047
None ADMET CC50 10000.0 nM 10.1021/jm040838n
None ADMET CC50 15000.0 nM 10.1021/acsmedchemlett.5b00254
None ADMET CC50 15500.0 nM 10.1128/aac.00984-08
None ADMET CC50 35000.0 nM 10.1128/aac.01064-10
None ADMET CC50 50000.0 nM 10.1016/j.bmc.2014.08.005
None ADMET CC50 nan None 10.1016/j.bmc.2015.09.035
None ADMET CL 0.0024 mL.min-1.g-1 10.1124/dmd.111.042416
None ADMET CL 0.0064 mL.min-1.g-1 10.1124/dmd.111.042416
None ADMET CL 0.0145 mL.min-1.g-1 10.1124/dmd.111.042416
None ADMET CL 0.17 uL/min 10.1124/dmd.111.042416
None ADMET CL 0.19 uL/min 10.1124/dmd.111.042416
None ADMET CL 0.3 uL/min 10.1124/dmd.111.042416
None ADMET CL 0.39 uL/min 10.1124/dmd.111.042416
None ADMET CL 8.51 uL.min-1.(10^6cells)-1 10.6019/CHEMBL3301361
None ADMET Drug metabolism nan None 10.1124/dmd.112.049601
None ADMET Drug uptake 19.0 ng/ml 10.1124/dmd.112.049601
None ADMET IC50 25840.0 nM 10.1016/j.bmc.2014.08.005
None ADMET Km 3200.0 nM 10.1124/dmd.111.042416
None ADMET Km 3400.0 nM 10.1124/dmd.111.042416
None ADMET Km 6200.0 nM 10.1124/dmd.111.042416
None ADMET Km 8800.0 nM 10.1124/dmd.111.042416
None ADMET Km 11200.0 nM 10.1124/dmd.111.042416
None ADMET Km 15200.0 nM 10.1124/dmd.111.042416
None ADMET Km 24000.0 nM 10.1124/dmd.111.042416
None ADMET Ratio 370.37 None 10.1021/jm801395v
None ADMET Ratio CC50/EC50 1.0 None 10.1021/acs.jmedchem.1c01015
None ADMET Ratio CC50/EC50 21.0 None 10.1021/acs.jmedchem.1c01015
None ADMET Ratio CC50/EC50 24.0 None 10.1021/acs.jmedchem.1c00128
None ADMET Ratio CC50/EC50 44.0 None 10.1021/acs.jmedchem.1c00987
None ADMET Ratio CC50/EC50 57.0 None 10.1021/acs.jmedchem.1c01015
None ADMET Ratio CC50/EC50 69.0 None 10.1021/acs.jmedchem.1c00128
None ADMET Ratio CC50/EC50 136.0 None 10.1021/acs.jmedchem.1c01015
None ADMET Ratio CC50/EC50 142.0 None 10.1021/acs.jmedchem.1c00128
None ADMET Ratio CC50/EC50 326.53 None 10.1039/C4MD00282B
None ADMET Ratio CC50/EC50 347.82 None 10.1039/C4MD00282B
None ADMET Ratio CC50/EC50 429.0 None 10.1021/acs.jmedchem.8b01238
None ADMET Ratio CC50/EC50 842.0 None 10.1021/acs.jmedchem.1c00128
None ADMET Ratio CC50/EC50 1000.0 None 10.1021/acs.jmedchem.1c01015
None ADMET Ratio CC50/EC50 1176.0 None 10.1021/acs.jmedchem.1c00128
None ADMET Ratio CC50/EC50 1187.0 None 10.1039/C3MD00028A
None ADMET Ratio CC50/EC50 1212.0 None 10.1016/j.ejmech.2020.113063
None ADMET Ratio CC50/EC50 1237.0 None 10.1021/acs.jmedchem.1c01015
None ADMET Ratio CC50/EC50 1394.0 None 10.1021/acs.jmedchem.1c00987
None ADMET Ratio CC50/EC50 1600.0 None 10.1021/acs.jmedchem.1c00128
None ADMET Ratio CC50/EC50 1600.0 None 10.1021/acs.jmedchem.1c01676
None ADMET Ratio CC50/EC50 2143.0 None 10.1016/j.ejmech.2022.114512
None ADMET Ratio CC50/EC50 2222.0 None 10.1016/j.bmc.2021.116531
None ADMET Ratio CC50/EC50 2372.0 None 10.1016/j.ejmech.2022.114471
None ADMET Ratio CC50/EC50 2572.0 None 10.1016/j.ejmech.2020.113063
None ADMET Ratio CC50/EC50 2857.0 None 10.1021/acs.jmedchem.2c00468
None ADMET Ratio CC50/IC50 24.0 None 10.1021/acs.jmedchem.1c01015
None ADMET Ratio CC50/IC50 248.79 None 10.1016/j.ejmech.2018.07.067
None ADMET Ratio CC50/IC50 1205.0 None 10.1021/acs.jmedchem.1c01015
None ADMET Selectivity index 6000.0 None 10.1016/j.bmcl.2007.11.127
None ADMET Selectivity Index 1463.0 None 10.1016/j.ejmech.2021.113868
None ADMET Selectivity Index 1600.0 None 10.1021/acs.jmedchem.1c00708
None ADMET Selectivity Index 2222.0 None 10.1016/j.bmc.2021.116239
None ADMET T1/2 1.633 hr 10.1016/j.bmcl.2010.01.086
None ADMET T1/2 40.0 hr 10.1021/acs.jmedchem.8b00843
None ADMET TC50 20000.0 nM 10.1021/jm070488f
None ADMET Vmax 0.95 pmol/min 10.1124/dmd.111.042416
None ADMET Vmax 1.02 pmol/min 10.1124/dmd.111.042416
None ADMET Vmax 1.21 pmol/min 10.1124/dmd.111.042416
None ADMET Vmax 1.61 pmol/min 10.1124/dmd.111.042416
None ADMET Vmax 25.0 pmol/min 10.1124/dmd.111.042416
None ADMET Vmax 87.1 pmol/min 10.1124/dmd.111.042416
None ADMET Vmax 100.6 pmol/min 10.1124/dmd.111.042416
None Hepatotoxicity Hepatotoxicity nan None 10.1021/tx900326k
None Hepatotoxicity HepSE_bilirubinemia 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_cholecystitis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_cholelithiasis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_cirrhosis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_Combined Scores 4.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_elevated liver function tests 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatic failure 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatic necrosis 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatitis 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_hepatomegaly 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_jaundice 1.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_liver disease 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_liver fatty 0.0 None 10.1371/journal.pcbi.1002310
None Hepatotoxicity HepSE_liver function tests abnormal 0.0 None 10.1371/journal.pcbi.1002310
None Lymphocyte Selectivity index 14285.0 None 10.1021/jm0512490
None Lymphocyte TC50 100.0 uM 10.1021/jm0512490
None Molecular identity unknown PPB 95.1 % 10.1124/dmd.112.049601
None Molecular identity unknown PPB 99.82 % 10.1124/dmd.112.049601
None NON-PROTEIN TARGET CC50 6300.0 nM 10.1016/j.ejmech.2016.05.054
None NON-PROTEIN TARGET CC50 6340.0 nM 10.1021/acs.jmedchem.6b00738
None NON-PROTEIN TARGET CC50 20600.0 nM 10.1016/j.ejmech.2016.06.026
None NON-PROTEIN TARGET EC50 0.7 nM 10.1021/acs.jmedchem.5b01430
None NON-PROTEIN TARGET EC50 5.0 nM 10.1021/acs.jmedchem.6b00738
None NON-PROTEIN TARGET EC50 5.2 nM 10.1021/acs.jmedchem.6b00738
None NON-PROTEIN TARGET EC50 6.8 nM 10.1016/j.ejmech.2016.05.054
None NON-PROTEIN TARGET EC50 8.2 nM 10.1021/acs.jmedchem.6b00738
None NON-PROTEIN TARGET EC50 80.1 nM 10.1021/acs.jmedchem.6b00738
None NON-PROTEIN TARGET EC50 115.5 nM 10.1021/acs.jmedchem.6b00738
None NON-PROTEIN TARGET EC50 156.1 nM 10.1021/acs.jmedchem.6b00738
None NON-PROTEIN TARGET EC50 240.0 nM 10.1016/j.ejmech.2016.05.054
None NON-PROTEIN TARGET EC50 348.5 nM 10.1021/acs.jmedchem.6b00738
None NON-PROTEIN TARGET EC50 514.8 nM 10.1021/acs.jmedchem.6b00738
None NON-PROTEIN TARGET EC50 nan None 10.1016/j.bmc.2015.09.035
None NON-PROTEIN TARGET Hepatotoxicity (acute) 10.9 % 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (animal toxicity known) nan None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (benign tumour) 0.0 None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (granulomatous hepatitis) 0.0 None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (mechanism) nan None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (moderate) 2.0 None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (moderate) 18.8 % 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET Hepatotoxicity (time to onset) nan None 10.1016/s0399-8320(04)95062-2
None NON-PROTEIN TARGET IC50 1.04 nM 10.1016/j.ejmech.2016.07.047
None NON-PROTEIN TARGET IC50 1.4 nM 10.1021/acs.jnatprod.6b00299
None NON-PROTEIN TARGET IC50 5.65 nM 10.1016/j.ejmech.2016.07.047
None NON-PROTEIN TARGET IC50 56.0 nM 10.1016/j.ejmech.2016.07.047
None NON-PROTEIN TARGET IC50 58.7 nM 10.1016/j.ejmech.2016.07.047
None NON-PROTEIN TARGET IC50 58.8 nM 10.1016/j.ejmech.2016.07.047
None NON-PROTEIN TARGET IC50 83.0 nM 10.1016/j.ejmech.2016.07.047
None NON-PROTEIN TARGET IC50 160.0 nM 10.1016/j.ejmech.2016.07.047
None NON-PROTEIN TARGET IC50 480.0 nM 10.1016/j.ejmech.2016.07.047
None NON-PROTEIN TARGET IC50 2490.0 nM 10.1016/j.ejmech.2016.07.047
None NON-PROTEIN TARGET IC50 13800.0 nM 10.1016/j.ejmech.2016.07.047
None NON-PROTEIN TARGET IC90 1.7 nM 10.1016/s0960-894x(99)00672-1
None NON-PROTEIN TARGET IC90 220.0 nM 10.1021/jm990580e
None NON-PROTEIN TARGET Ratio CC50/EC50 1585.0 None 10.1016/j.bmc.2016.05.010
None NON-PROTEIN TARGET Ratio CC50/EC50 nan None 10.1016/j.bmc.2016.05.010
None No relevant target pKa 7.18 None 10.1124/dmd.112.050278
None No relevant target solubility nan None 10.1016/j.ejmech.2016.05.054
None No relevant target Solubility 68.0 ug.mL-1 10.1016/j.bmc.2016.07.039
None No relevant target Solubility 68.0 ug.mL-1 10.1016/j.bmcl.2013.06.091
None No relevant target Solubility 68.0 ug.mL-1 10.1016/j.bmcl.2013.06.093
None No relevant target Solubility 68.0 ug.mL-1 10.1021/acsmedchemlett.5b00254
None No relevant target Solubility 68.0 ug.mL-1 10.1021/ml5003713
None No relevant target Solubility 68.3 ug.mL-1 10.1016/j.bmcl.2017.06.049
None No relevant target Solubility 500.0 nM 10.1021/acs.jmedchem.5b01430
None Nucleic Acid IC90 1.7 nM 10.1016/s0960-894x(01)00012-9
None Unchecked Ac50 5.012 uM None
None Unchecked Ac50 17.78 uM None
None Unchecked Ac50 22.39 uM None
None Unchecked Ac50 28.18 uM None
None Unchecked Ac50 31.62 uM None
None Unchecked AC50 5011.9 nM None
None Unchecked AC50 6380.0 nM None
None Unchecked AC50 7550.0 nM None
None Unchecked AC50 17782.8 nM None
None Unchecked AC50 22387.2 nM None
None Unchecked AC50 28183.8 nM None
None Unchecked AC50 28190.0 nM None
None Unchecked AC50 31622.8 nM None
None Unchecked Activity nan None 10.1016/j.bmc.2021.116239
None Unchecked Activity nan None 10.1021/acs.jmedchem.9b01383
None Unchecked CC50 20000.0 nM 10.1016/j.bmcl.2019.01.011
None Unchecked CC50 40490.0 nM 10.1016/j.ejmech.2018.07.067
None Unchecked EC50 1.0 nM 10.1016/j.ejmech.2016.06.026
None Unchecked EC50 2.9 nM 10.1016/j.ejmech.2020.112549
None Unchecked EC50 5.0 nM 10.1016/j.ejmech.2021.113204
None Unchecked EC50 7.3 nM 10.1016/j.bmc.2017.03.009
None Unchecked EC50 7.5 nM 10.1021/acs.jmedchem.1c00128
None Unchecked EC50 161.6 nM 10.1016/j.ejmech.2020.112549
None Unchecked EC50 269.0 nM 10.1021/acs.jmedchem.1c00128
None Unchecked EC50 316.8 nM 10.1016/j.ejmech.2020.112549
None Unchecked EC50 335000.0 nM 10.1016/j.ejmech.2021.113204
None Unchecked Fold resistance 6.0 None 10.1021/jm010853h
None Unchecked FR 5.9 None 10.1016/s0960-894x(01)00510-8
None Unchecked FR 8.6 None 10.1016/s0960-894x(01)00510-8
None Unchecked Free 27.0 % 10.1021/jm990580e
None Unchecked Hepatotoxicity (acute) 8.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (association with vascular disease) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (choleostasis) 2.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (chronic liver disease) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (cirrhosis) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (comment) nan None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (cytolytic) 8.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (malignant tumour) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (severe hepatitis) 4.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (steatosis) 0.0 None 10.1016/s0399-8320(04)95062-2
None Unchecked Hepatotoxicity (successful reintroduction) nan None 10.1016/s0399-8320(04)95062-2
None Unchecked IC50 2.0 nM 10.1016/j.bmcl.2013.12.070
None Unchecked IC50 8.4 nM 10.1016/j.bmcl.2009.08.039
None Unchecked IC50 8.4 nM 10.1016/j.bmcl.2009.08.043
None Unchecked IC50 8.4 nM 10.1016/j.bmcl.2009.08.080
None Unchecked IC50 9.8 nM 10.1016/j.ejmech.2020.112549
None Unchecked IC50 10.0 nM 10.1016/j.ejmech.2020.112071
None Unchecked IC50 12.0 nM 10.1016/j.ejmech.2017.02.054
None Unchecked IC50 24.0 nM 10.1016/j.ejmech.2018.10.029
None Unchecked IC50 25.0 nM 10.1016/j.bmc.2016.05.010
None Unchecked IC50 30.0 nM 10.1016/j.bmcl.2012.12.049
None Unchecked IC50 30.0 nM 10.1021/acs.jmedchem.6b00738
None Unchecked IC50 30.0 nM 10.1021/jm050257d
None Unchecked IC50 37.0 nM 10.1016/j.bmcl.2016.11.030
None Unchecked IC50 60.0 nM 10.1016/j.bmc.2016.04.010
None Unchecked IC50 60.0 nM 10.1039/C3MD00225J
None Unchecked IC50 100.0 nM 10.1128/aac.00800-09
None Unchecked IC50 240.0 nM 10.1016/j.bmc.2020.115927
None Unchecked IC50 380.0 nM 10.1128/aac.00800-09
None Unchecked IC50 400.0 nM 10.1016/j.ejmech.2012.01.056
None Unchecked IC50 400.0 nM 10.1016/j.ejmech.2014.04.027
None Unchecked IC50 400.0 nM 10.1016/j.ejmech.2020.112696
None Unchecked IC50 2476.0 nM None
None Unchecked IC50 3867.4 nM None
None Unchecked IC50 21246.04 nM None
None Unchecked IC50 50000.0 nM 10.1039/C3MD00014A
None Unchecked IC50 nan None 10.1016/j.bmc.2016.05.010
None Unchecked IC50 nan None 10.1016/j.bmc.2020.115927
None Unchecked IC50 nan None 10.1016/j.ejmech.2012.01.056
None Unchecked IC50 nan None 10.1016/j.ejmech.2017.02.054
None Unchecked IC50 nan None 10.1016/j.ejmech.2020.112071
None Unchecked IC50 nan None 10.1021/acs.jmedchem.6b01906
None Unchecked Ki 30.0 nM 10.1016/j.bmc.2011.08.025
None Unchecked Ki 40.0 nM 10.1021/jm801395v
None Unchecked Ki 60.0 nM 10.1016/j.bmc.2012.12.027
None Unchecked Ki 80.0 nM 10.1016/j.bmc.2011.08.025
None Unchecked Ki 80.0 nM 10.1021/jm070811e
None Unchecked Ki 100.0 nM 10.1021/jm801395v
None Unchecked Ki 330.0 nM 10.1016/j.bmc.2011.08.025
None Unchecked Ki 360.0 nM 10.1016/j.bmc.2011.08.025
None Unchecked Ki 380.0 nM 10.1021/jm801395v
None Unchecked Potency 12995.3 nM None
None Unchecked Potency 17061.9 nM None
None Unchecked Potency 24100.5 nM None
None Unchecked Potency 42857.5 nM None
None Unchecked Potency 48086.9 nM None
None Unchecked Ratio 3.0 None 10.1021/acs.jmedchem.8b01238
None Unchecked Ratio 3.0 None 10.1021/jm101626c
None Unchecked Ratio 3.0 None 10.1021/jm201308v
None Unchecked Ratio 3.0 None 10.1021/jm500284x
None Unchecked Ratio 3.0 None 10.1021/jm800340w
None Unchecked Ratio 5.67 None 10.1016/j.ejmech.2021.113498
None Unchecked Ratio 6.0 None 10.1021/jm0309856
None Unchecked Ratio 93.0 None 10.1021/acs.jmedchem.8b01238
None Unchecked Ratio 100.0 None 10.1021/jm101626c
None Unchecked Ratio 100.0 None 10.1021/jm201308v
None Unchecked Ratio 100.0 None 10.1021/jm500284x
None Unchecked Ratio 100.0 None 10.1021/jm800340w
None Unchecked Ratio 8750.0 None 10.1021/jm031147e
None Unchecked Ratio nan None 10.1021/jm500284x
None Unchecked Ratio CC50/EC50 6.34 None 10.1016/j.ejmech.2015.11.039
None Unchecked Ratio CC50/EC50 11.0 None 10.1016/j.bmcl.2012.09.062
None Unchecked Ratio CC50/EC50 12.0 None 10.1016/j.bmc.2012.04.030
None Unchecked Ratio CC50/EC50 12.0 None 10.1016/j.bmc.2013.10.033
None Unchecked Ratio CC50/EC50 12.0 None 10.1016/j.bmcl.2013.10.059
None Unchecked Ratio CC50/EC50 12.0 None 10.1021/acs.jmedchem.6b00738
None Unchecked Ratio CC50/EC50 12.0 None 10.1021/acs.jmedchem.7b00332
None Unchecked Ratio CC50/EC50 17.0 None 10.1016/j.bmc.2008.01.039
None Unchecked Ratio CC50/EC50 18.0 None 10.1021/acs.jmedchem.6b00738
None Unchecked Ratio CC50/EC50 18.0 None 10.1021/acs.jmedchem.7b00332
None Unchecked Ratio CC50/EC50 19.0 None 10.1016/j.bmc.2016.07.041
None Unchecked Ratio CC50/EC50 19.0 None 10.1016/j.ejmech.2018.03.059
None Unchecked Ratio CC50/EC50 19.0 None 10.1016/j.ejmech.2020.113051
None Unchecked Ratio CC50/EC50 20.0 None 10.1016/j.ejmech.2020.112811
None Unchecked Ratio CC50/EC50 21.0 None 10.1016/j.ejmech.2014.02.047
None Unchecked Ratio CC50/EC50 21.0 None 10.1021/acs.jmedchem.6b00738
None Unchecked Ratio CC50/EC50 21.0 None 10.1021/acs.jmedchem.7b00332
None Unchecked Ratio CC50/EC50 24.0 None 10.1016/j.ejmech.2019.111619
None Unchecked Ratio CC50/EC50 24.0 None 10.1016/j.ejmech.2020.112237
None Unchecked Ratio CC50/EC50 24.0 None 10.1021/acs.jmedchem.9b01769
None Unchecked Ratio CC50/EC50 26.0 None 10.1021/acs.jmedchem.8b01729
None Unchecked Ratio CC50/EC50 27.0 None 10.1016/j.bmc.2014.08.001
None Unchecked Ratio CC50/EC50 27.0 None 10.1016/j.ejmech.2016.05.054
None Unchecked Ratio CC50/EC50 28.0 None 10.1016/j.ejmech.2016.02.068
None Unchecked Ratio CC50/EC50 28.2 None 10.1021/acsmedchemlett.8b00054
None Unchecked Ratio CC50/EC50 30.0 None 10.1016/j.bmc.2016.07.041
None Unchecked Ratio CC50/EC50 30.0 None 10.1016/j.ejmech.2018.03.059
None Unchecked Ratio CC50/EC50 41.0 None 10.1016/j.ejmech.2015.01.042
None Unchecked Ratio CC50/EC50 44.0 None 10.1016/j.bmcl.2018.03.012
None Unchecked Ratio CC50/EC50 51.0 None 10.1016/j.ejmech.2019.111874
None Unchecked Ratio CC50/EC50 52.0 None 10.1016/j.bmc.2016.07.041
None Unchecked Ratio CC50/EC50 52.0 None 10.1016/j.ejmech.2018.03.059
None Unchecked Ratio CC50/EC50 55.0 None 10.1016/j.ejmech.2016.10.009
None Unchecked Ratio CC50/EC50 55.0 None 10.1021/acs.jmedchem.6b00738
None Unchecked Ratio CC50/EC50 55.0 None 10.1021/acs.jmedchem.7b00332
None Unchecked Ratio CC50/EC50 62.0 None 10.1016/j.bmc.2016.07.041
None Unchecked Ratio CC50/EC50 62.0 None 10.1016/j.ejmech.2018.03.059
None Unchecked Ratio CC50/EC50 64.0 None 10.1016/j.ejmech.2016.10.009
None Unchecked Ratio CC50/EC50 68.0 None 10.1016/j.ejmech.2016.10.009
None Unchecked Ratio CC50/EC50 75.0 None 10.1021/jm070811e
None Unchecked Ratio CC50/EC50 79.0 None 10.1021/acs.jmedchem.6b00738
None Unchecked Ratio CC50/EC50 79.0 None 10.1021/acs.jmedchem.7b00332
None Unchecked Ratio CC50/EC50 82.0 None 10.1016/j.ejmech.2016.10.009
None Unchecked Ratio CC50/EC50 110.0 None 10.1016/j.ejmech.2016.10.009
None Unchecked Ratio CC50/EC50 113.0 None 10.1016/j.bmc.2011.08.025
None Unchecked Ratio CC50/EC50 286.0 None 10.1016/j.bmc.2012.12.049
None Unchecked Ratio CC50/EC50 429.0 None 10.1021/jm500284x
None Unchecked Ratio CC50/EC50 429.0 None 10.1021/jm800340w
None Unchecked Ratio CC50/EC50 433.9 None 10.1021/jm101626c
None Unchecked Ratio CC50/EC50 440.0 None 10.1021/jm201308v
None Unchecked Ratio CC50/EC50 693.0 None 10.1016/j.bmc.2013.09.051
None Unchecked Ratio CC50/EC50 727.0 None 10.1016/j.ejmech.2013.04.052
None Unchecked Ratio CC50/EC50 727.0 None 10.1039/C3MD00247K
None Unchecked Ratio CC50/EC50 755.0 None 10.1016/j.ejmech.2019.111619
None Unchecked Ratio CC50/EC50 772.0 None 10.1021/acs.jmedchem.6b00738
None Unchecked Ratio CC50/EC50 772.0 None 10.1021/acs.jmedchem.7b00332
None Unchecked Ratio CC50/EC50 855.0 None 10.1016/j.bmc.2013.10.033
None Unchecked Ratio CC50/EC50 855.0 None 10.1016/j.bmcl.2013.10.059
None Unchecked Ratio CC50/EC50 863.0 None 10.1016/j.ejmech.2019.111603
None Unchecked Ratio CC50/EC50 863.0 None 10.1021/acs.jmedchem.9b01446
None Unchecked Ratio CC50/EC50 868.0 None 10.1016/j.bmc.2017.03.009
None Unchecked Ratio CC50/EC50 928.0 None 10.1016/j.bmc.2016.07.041
None Unchecked Ratio CC50/EC50 928.0 None 10.1016/j.ejmech.2018.03.059
None Unchecked Ratio CC50/EC50 938.0 None 10.1016/j.ejmech.2016.05.054
None Unchecked Ratio CC50/EC50 943.0 None 10.1016/j.bmc.2013.08.040
None Unchecked Ratio CC50/EC50 964.0 None 10.1016/j.bmc.2012.04.030
None Unchecked Ratio CC50/EC50 964.0 None 10.1016/j.bmc.2012.07.026
None Unchecked Ratio CC50/EC50 964.0 None 10.1016/j.bmcl.2012.09.062
None Unchecked Ratio CC50/EC50 996.0 None 10.1016/j.ejmech.2014.04.027
None Unchecked Ratio CC50/EC50 996.0 None 10.1016/j.ejmech.2020.112696
None Unchecked Ratio CC50/EC50 996.0 None 10.1021/acs.jmedchem.6b01906
None Unchecked Ratio CC50/EC50 996.0 None 10.1021/jm5011622
None Unchecked Ratio CC50/EC50 1000.0 None 10.1016/j.bmc.2015.01.002
None Unchecked Ratio CC50/EC50 1000.0 None 10.1016/j.ejmech.2012.04.038
None Unchecked Ratio CC50/EC50 1000.0 None 10.1016/j.ejmech.2020.112071
None Unchecked Ratio CC50/EC50 1006.0 None 10.1016/j.ejmech.2015.08.007
None Unchecked Ratio CC50/EC50 1014.0 None 10.1016/j.bmc.2014.11.032
None Unchecked Ratio CC50/EC50 1014.0 None 10.1016/j.bmc.2015.09.020
None Unchecked Ratio CC50/EC50 1014.0 None 10.1016/j.ejmech.2014.09.054
None Unchecked Ratio CC50/EC50 1014.0 None 10.1016/j.ejmech.2015.01.042
None Unchecked Ratio CC50/EC50 1014.0 None 10.1021/acs.jmedchem.6b00738
None Unchecked Ratio CC50/EC50 1056.0 None 10.1016/j.bmc.2013.12.045
None Unchecked Ratio CC50/EC50 1056.0 None 10.1016/j.bmc.2016.04.010
None Unchecked Ratio CC50/EC50 1112.0 None 10.1016/j.ejmech.2014.02.047
None Unchecked Ratio CC50/EC50 1136.0 None 10.1016/j.bmc.2014.03.020
None Unchecked Ratio CC50/EC50 1146.0 None 10.1016/j.bmc.2011.07.023
None Unchecked Ratio CC50/EC50 1146.0 None 10.1016/j.bmc.2011.10.002
None Unchecked Ratio CC50/EC50 1146.0 None 10.1016/j.ejmech.2012.04.004
None Unchecked Ratio CC50/EC50 1183.0 None 10.1016/j.bmc.2014.08.001
None Unchecked Ratio CC50/EC50 1187.0 None 10.1016/j.bmc.2012.09.058
None Unchecked Ratio CC50/EC50 1187.0 None 10.1016/j.ejmech.2012.02.019
None Unchecked Ratio CC50/EC50 1204.0 None 10.1016/j.bmc.2015.03.037
None Unchecked Ratio CC50/EC50 1212.0 None 10.1016/j.bmc.2016.07.041
None Unchecked Ratio CC50/EC50 1212.0 None 10.1016/j.ejmech.2015.11.039
None Unchecked Ratio CC50/EC50 1212.0 None 10.1016/j.ejmech.2016.02.068
None Unchecked Ratio CC50/EC50 1212.0 None 10.1016/j.ejmech.2017.02.047
None Unchecked Ratio CC50/EC50 1212.0 None 10.1016/j.ejmech.2018.03.059
None Unchecked Ratio CC50/EC50 1220.0 None 10.1021/acs.jmedchem.6b00738
None Unchecked Ratio CC50/EC50 1220.0 None 10.1021/acs.jmedchem.7b00332
None Unchecked Ratio CC50/EC50 1235.0 None 10.1016/j.bmc.2016.07.041
None Unchecked Ratio CC50/EC50 1235.0 None 10.1016/j.ejmech.2018.03.059
None Unchecked Ratio CC50/EC50 1258.0 None 10.1016/j.ejmech.2017.07.012
None Unchecked Ratio CC50/EC50 1258.0 None 10.1021/acs.jmedchem.7b00332
None Unchecked Ratio CC50/EC50 1269.0 None 10.1016/j.ejmech.2019.05.011
None Unchecked Ratio CC50/EC50 1282.0 None 10.1016/j.ejmech.2016.10.009
None Unchecked Ratio CC50/EC50 1316.0 None 10.1016/j.bmc.2017.05.040
None Unchecked Ratio CC50/EC50 1316.0 None 10.1016/j.bmc.2017.12.033
None Unchecked Ratio CC50/EC50 1316.0 None 10.1016/j.bmcl.2018.03.012
None Unchecked Ratio CC50/EC50 1333.0 None 10.1016/j.ejmech.2020.112237
None Unchecked Ratio CC50/EC50 1356.0 None 10.1016/j.ejmech.2016.10.009
None Unchecked Ratio CC50/EC50 1434.0 None 10.1007/s00044-009-9220-x
None Unchecked Ratio CC50/EC50 1434.0 None 10.1016/j.bmc.2009.07.028
None Unchecked Ratio CC50/EC50 1434.0 None 10.1016/j.bmc.2011.05.024
None Unchecked Ratio CC50/EC50 1434.0 None 10.1016/j.bmcl.2008.09.055
None Unchecked Ratio CC50/EC50 1434.0 None 10.1016/j.ejmech.2009.06.037
None Unchecked Ratio CC50/EC50 1667.0 None 10.1016/j.ejmech.2019.111874
None Unchecked Ratio CC50/EC50 1717.0 None 10.1016/j.bmcl.2017.03.009
None Unchecked Ratio CC50/EC50 1843.0 None 10.1016/j.bmc.2010.03.007
None Unchecked Ratio CC50/EC50 2112.0 None 10.1016/j.bmc.2010.05.036
None Unchecked Ratio CC50/EC50 2112.0 None 10.1016/j.bmc.2011.08.025
None Unchecked Ratio CC50/EC50 2113.0 None 10.1016/j.bmc.2008.01.039
None Unchecked Ratio CC50/EC50 2223.0 None 10.1021/acsmedchemlett.8b00054
None Unchecked Ratio CC50/EC50 2268.0 None 10.1016/j.ejmech.2020.113051
None Unchecked Ratio CC50/EC50 2268.0 None 10.1016/j.ejmech.2021.113204
None Unchecked Ratio CC50/EC50 2372.0 None 10.1016/j.ejmech.2016.10.009
None Unchecked Ratio CC50/EC50 2514.0 None 10.1021/jm300477h
None Unchecked Ratio CC50/EC50 2540.0 None 10.1021/acs.jmedchem.9b01769
None Unchecked Ratio CC50/EC50 2824.0 None 10.1016/j.ejmech.2020.112811
None Unchecked Ratio CC50/EC50 3082.0 None 10.1016/j.bmc.2010.05.081
None Unchecked Ratio CC50/EC50 4012.0 None 10.1016/j.bmc.2018.03.003
None Unchecked Ratio CC50/EC50 4624.0 None 10.1016/j.ejmech.2018.01.016
None Unchecked Ratio CC50/EC50 4969.0 None 10.1021/acs.jmedchem.8b01729
None Unchecked Ratio CC50/EC50 6666.0 None 10.1016/j.bmc.2008.06.012
None Unchecked Ratio CC50/EC50 6666.0 None 10.1016/j.bmc.2009.06.068
None Unchecked Ratio CC50/EC50 6666.0 None 10.1016/j.bmc.2009.12.059
None Unchecked Ratio CC50/EC50 6666.0 None 10.1016/j.bmcl.2007.01.025
None Unchecked Ratio CC50/EC50 15000.0 None 10.1016/j.bmc.2007.09.015
None Unchecked Ratio CC50/EC50 19850.0 None 10.1016/j.ejmech.2006.11.014
None Unchecked Ratio CC50/EC50 20600.0 None 10.1016/j.ejmech.2016.06.026
None Unchecked Ratio CC50/EC50 31818.0 None 10.1128/aac.01064-10
None Unchecked Ratio CC50/EC50 52183.0 None 10.1016/j.ejmech.2020.112549
None Unchecked Ratio CC50/EC50 58000.0 None 10.1021/jm801438e
None Unchecked Ratio CC50/IC50 280.0 None 10.1016/j.bmc.2014.02.030
None Unchecked Ratio CC50/IC50 280.0 None 10.1016/j.ejmech.2014.05.059
None Unchecked Ratio CC50/IC50 10000.0 None 10.1016/j.bmcl.2006.10.082
None Unchecked Ratio CC50/IC50 10000.0 None 10.1021/jm900802y
None Unchecked Ratio EC50 1.0 None 10.1016/j.ejmech.2021.113868
None Unchecked Ratio EC50 1.0 None 10.1021/acs.jmedchem.1c01015
None Unchecked Ratio EC50 1.2 None 10.1021/acs.jmedchem.1c01015
None Unchecked Ratio EC50 1.5 None 10.1021/jm070811e
None Unchecked Ratio EC50 1.7 None 10.1016/j.ejmech.2020.112071
None Unchecked Ratio EC50 2.0 None 10.1016/j.ejmech.2021.113868
None Unchecked Ratio EC50 2.0 None 10.1016/j.ejmech.2022.114512
None Unchecked Ratio EC50 2.3 None 10.1016/j.ejmech.2020.112811
None Unchecked Ratio EC50 2.5 None 10.1016/j.ejmech.2020.112811
None Unchecked Ratio EC50 8.0 None 10.1016/j.bmcl.2008.09.070
None Unchecked Ratio EC50 8.8 None 10.1021/acs.jmedchem.1c01015
None Unchecked Ratio EC50 12.0 None 10.1016/j.ejmech.2022.114512
None Unchecked Ratio EC50 17.8 None 10.1016/j.ejmech.2020.112811
None Unchecked Ratio EC50 20.0 None 10.1021/jm070811e
None Unchecked Ratio EC50 21.2 None 10.1021/acs.jmedchem.1c01015
None Unchecked Ratio EC50 22.0 None 10.1016/j.ejmech.2021.113868
None Unchecked Ratio EC50 22.0 None 10.1021/jm070811e
None Unchecked Ratio EC50 27.0 None 10.1016/j.ejmech.2020.112071
None Unchecked Ratio EC50 31.0 None 10.1016/j.ejmech.2022.114512
None Unchecked Ratio EC50 33.0 None 10.1016/j.ejmech.2021.113868
None Unchecked Ratio EC50 41.9 None 10.1016/j.ejmech.2020.112811
None Unchecked Ratio EC50 50.2 None 10.1016/j.ejmech.2020.112071
None Unchecked Ratio EC50 51.0 None 10.1016/j.ejmech.2021.113868
None Unchecked Ratio EC50 51.1 None 10.1021/acs.jmedchem.1c01015
None Unchecked Ratio EC50 55.5 None 10.1016/j.ejmech.2020.112071
None Unchecked Ratio EC50 57.0 None 10.1021/jm070811e
None Unchecked Ratio EC50 58.3 None 10.1021/acs.jmedchem.1c01015
None Unchecked Ratio EC50 68.0 None 10.1016/j.ejmech.2022.114512
None Unchecked Ratio EC50 76.0 None 10.1016/j.ejmech.2021.113868
None Unchecked Ratio EC50 116.7 None 10.1016/j.ejmech.2020.112811
None Unchecked Ratio EC50 124.3 None 10.1016/j.ejmech.2020.112071
None Unchecked Ratio EC50 133.0 None 10.1016/j.bmcl.2008.09.070
None Unchecked Ratio EC50 162.5 None 10.1016/j.ejmech.2020.112811
None Unchecked Ratio EC50 183.0 None 10.1016/j.ejmech.2020.112071
None Unchecked Ratio EC50 1080.3 None 10.1016/j.ejmech.2020.112071
None Unchecked Ratio EC50 2128.0 None 10.1128/aac.00210-08
None Unchecked Ratio IC50 0.4 None 10.1016/j.bmcl.2009.08.039
None Unchecked Ratio IC50 0.4 None 10.1016/j.bmcl.2009.08.043
None Unchecked Ratio IC50 0.4 None 10.1016/j.bmcl.2009.08.080
None Unchecked Ratio IC50 0.8 None 10.1016/j.bmcl.2009.08.039
None Unchecked Ratio IC50 0.8 None 10.1016/j.bmcl.2009.08.043
None Unchecked Ratio IC50 0.8 None 10.1016/j.bmcl.2009.08.080
None Unchecked Ratio IC50 1.0 None 10.1016/j.bmcl.2009.08.039
None Unchecked Ratio IC50 1.0 None 10.1016/j.bmcl.2009.08.043
None Unchecked Ratio IC50 1.0 None 10.1016/j.bmcl.2009.08.080
None Unchecked Ratio IC50 1.8 None 10.1016/j.bmcl.2009.08.039
None Unchecked Ratio IC50 1.8 None 10.1016/j.bmcl.2009.08.043
None Unchecked Ratio IC50 1.8 None 10.1016/j.bmcl.2009.08.080
None Unchecked Ratio IC50 2.2 None 10.1016/j.bmcl.2009.08.039
None Unchecked Ratio IC50 2.2 None 10.1016/j.bmcl.2009.08.043
None Unchecked Ratio IC50 2.2 None 10.1016/j.bmcl.2009.08.080
None Unchecked Ratio IC50 2.5 None 10.1016/j.bmcl.2009.08.080
None Unchecked Ratio IC50 2.8 None 10.1016/j.bmcl.2009.08.039
None Unchecked Ratio IC50 2.8 None 10.1016/j.bmcl.2009.08.043
None Unchecked Ratio IC50 2.8 None 10.1016/j.bmcl.2009.08.080
None Unchecked Ratio IC50 3.0 None 10.1039/C3MD00225J
None Unchecked Ratio IC50 3.8 None 10.1016/j.bmcl.2009.08.039
None Unchecked Ratio IC50 3.8 None 10.1016/j.bmcl.2009.08.043
None Unchecked Ratio IC50 3.8 None 10.1016/j.bmcl.2009.08.080
None Unchecked Ratio IC50 5.0 None 10.1039/C3MD00225J
None Unchecked Ratio IC50 5.6 None 10.1016/j.bmcl.2009.08.080
None Unchecked Ratio IC50 6.0 None 10.1039/C3MD00225J
None Unchecked Ratio IC50 8.0 None 10.1039/C3MD00225J
None Unchecked Ratio IC50 10.0 None 10.1128/aac.01455-09
None Unchecked Ratio IC50 13.1 None 10.1128/aac.01455-09
None Unchecked Ratio IC50 14.0 None 10.1039/C3MD00225J
None Unchecked Ratio IC50 20.2 None 10.1128/aac.01455-09
None Unchecked Ratio IC50 37.4 None 10.1128/aac.01455-09
None Unchecked Ratio IC50 44.0 None 10.1016/j.bmcl.2009.08.039
None Unchecked Ratio IC50 44.0 None 10.1016/j.bmcl.2009.08.043
None Unchecked Ratio IC50 44.0 None 10.1016/j.bmcl.2009.08.080
None Unchecked Ratio IC50 47.3 None 10.1021/acs.jmedchem.6b00738
None Unchecked Ratio IC50 58.0 None 10.1039/C3MD00225J
None Unchecked Ratio IC50 60.0 None 10.1128/aac.01455-09
None Unchecked Ratio IC50 90.0 None 10.1021/acs.jmedchem.6b00730
None Unchecked Ratio IC50 200.0 None 10.1021/acs.jmedchem.6b00730
None Unchecked Ratio Ki 2.6 None 10.1016/j.bmc.2011.08.025
None Unchecked Ratio Ki 2.7 None 10.1016/j.bmc.2011.08.025
None Unchecked Ratio Ki 3.0 None 10.1021/jm070811e
None Unchecked Ratio Ki 10.0 None 10.1016/j.bmc.2011.08.025
None Unchecked Ratio Ki 12.0 None 10.1016/j.bmc.2011.08.025
None Unchecked Ratio Ki 19.3 None 10.1016/j.bmc.2011.08.025
None Unchecked Ratio Ki 24.0 None 10.1016/j.bmc.2011.08.025
None Unchecked Ratio Ki 100.0 None 10.1021/jm070811e
None Unchecked Selectivity index 2857.0 None 10.1021/jm070488f
None Unchecked Selectivity Index 13.0 None 10.1016/j.bmc.2018.12.039
None Unchecked Selectivity Index 41.0 None 10.1016/j.ejmech.2015.02.022
None Unchecked Selectivity Index 451.0 None 10.1016/j.bmc.2018.12.039
None Unchecked Selectivity Index 1006.0 None 10.1016/j.ejmech.2015.04.050
None Unchecked Selectivity Index 1014.0 None 10.1016/j.ejmech.2015.02.022
None Unchecked Selectivity Index 2423.0 None 10.1016/j.ejmech.2019.111864
None Unchecked Selectivity Index 6667.0 None 10.1021/jm101614j
None Unchecked Selectivity ratio 16.0 None 10.1128/aac.01795-09
None Unchecked Selectivity ratio 24.7 None 10.1128/aac.01795-09
None Unchecked SI 2500.0 None 10.1021/jm020949r
None Unchecked SI 10000.0 None 10.1021/jm020949r

Metabolism Information