Molecule

Gefitinib

AlkaPlorer ID: AK049825

Synonym: None

IUPAC Name: N-(3-chloro-4-fluorophenyl)-7-methoxy-6-(3-morpholin-4-ylpropoxy)quinazolin-4-amine

Structure

SMILES: COC1=CC2=NC=NC(NC3=CC=C(F)C(Cl)=C3)=C2C=C1OCCCN1CCOCC1

InChI: InChI=1S/C22H24ClFN4O3/c1-29-20-13-19-16(12-21(20)31-8-2-5-28-6-9-30-10-7-28)22(26-14-25-19)27-15-3-4-18(24)17(23)11-15/h3-4,11-14H,2,5-10H2,1H3,(H,25,26,27)

InChIKey: XGALLCVXEZPNRQ-UHFFFAOYSA-N

Reference

PubChem CID: 123631

CAS: 184475-35-2

NPASS: NPC56271

COCONUT: CNP0077274

Source

Species	Genus	Family	Order	Class	Phylum	Kingdom	Domain
Streptomyces sp.	Streptomyces	Streptomycetaceae	Kitasatosporales	Actinomycetes	Actinomycetota	None	Bacteria
Asarum heterotropoides	Asarum	Asaraceae	Piperales	Magnoliopsida	Streptophyta	Viridiplantae	Eukaryota
Asarum sieboldii	Asarum	Asaraceae	Piperales	Magnoliopsida	Streptophyta	Viridiplantae	Eukaryota

Properties Information

Molecule Weight: 446.9100000000004

TPSA？: 68.74000000000001

MolLogP？: 4.275600000000003

Number of H-Donors: 1

Number of H-Acceptors: 7

RingCount: 4

Activities Information

Organism	Target Name	Standard Type	Standard Value	Standard Units	doi
Canis lupus familiaris	MDCK	GI50	1450.0	nM	10.1016/j.bmc.2013.10.007
Canis lupus familiaris	MDCK-II	Activity	nan	None	10.1016/j.bmc.2013.10.007
Canis lupus familiaris	MDCK-II	GI50	1360.0	nM	10.1016/j.ejmech.2018.10.026
Canis lupus familiaris	MDCK-II	GI50	2100.0	nM	10.1016/j.ejmech.2018.10.026
Chlorocebus sabaeus	Vero	Activity	34.0	%	10.1021/acsmedchemlett.8b00270
Chlorocebus sabaeus	Vero	IC50	10000.0	nM	10.1021/acsmedchemlett.8b00270
Chlorocebus sabaeus	Vero	IC50	100000.0	nM	10.1016/j.bmcl.2017.08.063
Cricetulus griseus	CHO-K1	GI50	43700.0	nM	10.1021/acs.jmedchem.6b01774
Gallus gallus	Myosin light chain kinase, smooth muscle	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	16HBE14o-	Activity	nan	None	10.1016/j.ejmech.2013.05.026
Homo sapiens	23132-87	IC50	864.28	nM	10.6019/CHEMBL1201861
Homo sapiens	26S protease regulatory subunit 6B	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	3-phosphoinositide dependent protein kinase-1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	3-phosphoinositide dependent protein kinase-1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	3-phosphoinositide dependent protein kinase-1	Ki	3981.07	nM	None
Homo sapiens	3-phosphoinositide dependent protein kinase-1	Thermal melting change	-0.5	degrees C	10.1073/pnas.0708800104
Homo sapiens	5637	IC50	8310.55	nM	10.6019/CHEMBL1201861
Homo sapiens	639-V	IC50	3577.92	nM	10.6019/CHEMBL1201861
Homo sapiens	647-V	IC50	3162.2	nM	10.6019/CHEMBL1201861
Homo sapiens	697	IC50	1441.04	nM	10.6019/CHEMBL1201861
Homo sapiens	769-P	IC50	1279.18	nM	10.6019/CHEMBL1201861
Homo sapiens	786-0	IC50	2184.06	nM	10.6019/CHEMBL1201861
Homo sapiens	8305C	IC50	33993.69	nM	10.6019/CHEMBL1201861
Homo sapiens	8505C	IC50	26912.61	nM	10.6019/CHEMBL1201861
Homo sapiens	8-MG-BA	IC50	6193.79	nM	10.6019/CHEMBL1201861
Homo sapiens	A101D	IC50	9517.19	nM	10.6019/CHEMBL1201861
Homo sapiens	A 172	IC50	4555.21	nM	10.6019/CHEMBL1201861
Homo sapiens	A204	IC50	10046.62	nM	10.6019/CHEMBL1201861
Homo sapiens	A2058	IC50	10549.06	nM	10.6019/CHEMBL1201861
Homo sapiens	A2780	IC50	3640.89	nM	10.6019/CHEMBL1201861
Homo sapiens	A-375	IC50	20550.0	nM	10.1016/j.ejmech.2010.03.001
Homo sapiens	A-375	IC50	21056.66	nM	10.6019/CHEMBL1201861
Homo sapiens	A388	IC50	6895.2	nM	10.6019/CHEMBL1201861
Homo sapiens	A3-KAW	IC50	31447.08	nM	10.6019/CHEMBL1201861
Homo sapiens	A-427	IC50	59574.46	nM	10.6019/CHEMBL1201861
Homo sapiens	A-431	EC50	1710.0	nM	10.1021/acs.jmedchem.7b00515
Homo sapiens	A-431	EC50	2200.0	nM	10.1021/acs.jmedchem.7b00316
Homo sapiens	A-431	FC	0.229	None	10.1016/j.bmc.2020.115889
Homo sapiens	A-431	GI50	514.0	nM	10.1016/j.bmc.2009.11.035
Homo sapiens	A-431	IC50	0.276	ug.mL-1	10.1016/s0960-894x(02)00598-x
Homo sapiens	A-431	IC50	550.0	nM	10.1016/j.bmcl.2013.12.079
Homo sapiens	A-431	IC50	550.0	nM	10.1016/j.bmcl.2016.08.007
Homo sapiens	A-431	IC50	550.0	nM	10.1016/j.bmcl.2020.127045
Homo sapiens	A-431	IC50	768.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	A-431	IC50	780.04	nM	10.6019/CHEMBL1201861
Homo sapiens	A-431	IC50	1282.0	nM	10.1016/j.bmc.2018.11.009
Homo sapiens	A-431	IC50	1330.0	nM	10.1016/j.ejmech.2016.01.045
Homo sapiens	A-431	IC50	1410.0	nM	10.1016/j.bmc.2012.05.034
Homo sapiens	A-431	IC50	1890.0	nM	10.1007/s00044-013-0734-x
Homo sapiens	A-431	IC50	1980.0	nM	10.1016/j.bmc.2013.09.027
Homo sapiens	A-431	IC50	2150.0	nM	10.1021/jm201591k
Homo sapiens	A-431	IC50	2470.0	nM	10.1021/acs.jmedchem.8b01612
Homo sapiens	A-431	IC50	2600.0	nM	10.1016/j.ejmech.2019.111966
Homo sapiens	A-431	IC50	2980.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	A-431	IC50	3300.0	nM	10.1016/j.ejmech.2017.03.083
Homo sapiens	A-431	IC50	3308.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	A-431	IC50	3740.0	nM	10.1016/j.bmc.2015.12.001
Homo sapiens	A-431	IC50	4000.0	nM	10.1021/jm301365e
Homo sapiens	A-431	IC50	4000.0	nM	10.1021/jm5014659
Homo sapiens	A-431	IC50	4450.0	nM	10.1016/j.ejmech.2017.06.023
Homo sapiens	A-431	IC50	4450.0	nM	10.1016/j.ejmech.2018.01.090
Homo sapiens	A-431	IC50	4450.0	nM	10.1016/j.ejmech.2019.06.015
Homo sapiens	A-431	IC50	4485.0	nM	10.1016/j.ejmech.2014.02.032
Homo sapiens	A-431	IC50	4485.0	nM	10.1021/jm400463q
Homo sapiens	A-431	IC50	4580.0	nM	10.1016/j.bmc.2016.04.046
Homo sapiens	A-431	IC50	6120.0	nM	10.1016/j.bmc.2017.03.032
Homo sapiens	A-431	IC50	8370.0	nM	10.1016/j.ejmech.2021.113300
Homo sapiens	A-431	IC50	8982.0	nM	10.1016/j.ejmech.2013.05.026
Homo sapiens	A-431	IC50	12050.0	nM	10.1016/j.ejmech.2008.07.023
Homo sapiens	A-431	IC50	12580.0	nM	10.1016/j.bmcl.2017.02.023
Homo sapiens	A-431	IC50	16020.0	nM	10.1016/j.ejmech.2021.113589
Homo sapiens	A-431	IC50	24550.0	nM	10.1016/j.ejmech.2021.113589
Homo sapiens	A-431	IC50	31200.0	nM	10.1016/j.bmc.2020.115889
Homo sapiens	A-431	IC50	32170.0	nM	10.1016/j.ejmech.2021.113589
Homo sapiens	A-431	IC50	nan	None	10.1016/j.ejmech.2019.111888
Homo sapiens	A-431	IG50	4.45	uM	10.1016/j.bmcl.2017.02.027
Homo sapiens	A-431	TGI	35.9	%	10.1021/ml4002437
Homo sapiens	A-431	TGI	62.0	%	10.1021/jm500973a
Homo sapiens	A-431	TGI	79.0	%	10.1021/acsmedchemlett.6b00058
Homo sapiens	A-431	TGI	79.0	%	10.1021/jm400822z
Homo sapiens	A-431	TGI	119.0	%	10.1021/jm500973a
Homo sapiens	A498	GI50	400.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	A498	IC50	2294.15	nM	10.6019/CHEMBL1201861
Homo sapiens	A498	IC50	8600.0	nM	10.1016/j.ejmech.2012.06.055
Homo sapiens	A4-Fuk	IC50	350.02	nM	10.6019/CHEMBL1201861
Homo sapiens	A549	Activity	0.94	%	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	Activity	0.95	%	10.1016/j.ejmech.2019.06.015
Homo sapiens	A549	Activity	1.0	%	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	Activity	1.67	%	10.1016/j.ejmech.2017.12.022
Homo sapiens	A549	Activity	3.61	%	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	Activity	4.04	%	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	Activity	4.92	%	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	Activity	5.27	%	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	Activity	5.81	%	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	Activity	5.84	%	10.1016/j.ejmech.2017.12.022
Homo sapiens	A549	Activity	5.95	%	10.1016/j.ejmech.2019.06.015
Homo sapiens	A549	Activity	6.72	%	10.1016/j.ejmech.2017.12.022
Homo sapiens	A549	Activity	7.05	%	10.1021/acs.jmedchem.8b01612
Homo sapiens	A549	Activity	7.86	%	10.1016/j.ejmech.2019.06.015
Homo sapiens	A549	Activity	7.93	%	10.1016/j.ejmech.2019.06.015
Homo sapiens	A549	Activity	11.0	%	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	Activity	16.98	%	10.1016/j.ejmech.2019.06.015
Homo sapiens	A549	Activity	20.72	%	10.1021/acs.jmedchem.8b01612
Homo sapiens	A549	Activity	60.8	%	10.1016/j.bmcl.2014.09.056
Homo sapiens	A549	Activity	61.5	%	10.1016/j.ejmech.2011.07.045
Homo sapiens	A549	Activity	64.6	%	10.1016/j.bmcl.2014.09.056
Homo sapiens	A549	Activity	74.3	%	10.1016/j.bmcl.2014.09.056
Homo sapiens	A549	Activity	76.94	%	10.1016/j.ejmech.2019.06.015
Homo sapiens	A549	Activity	82.1	%	10.1016/j.bmcl.2014.09.056
Homo sapiens	A549	Activity	83.1	%	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	Activity	83.26	%	10.1016/j.ejmech.2019.06.015
Homo sapiens	A549	Activity	84.12	%	10.1016/j.ejmech.2017.12.022
Homo sapiens	A549	Activity	84.4	%	10.1016/j.ejmech.2011.07.045
Homo sapiens	A549	Activity	86.7	%	10.1016/j.bmcl.2014.09.056
Homo sapiens	A549	Activity	88.0	%	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	Activity	92.35	%	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	Activity	nan	None	10.1016/j.bmc.2015.12.001
Homo sapiens	A549	Activity	nan	None	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	Activity	nan	None	10.1016/j.ejmech.2020.112185
Homo sapiens	A549	Activity	nan	None	10.1021/acs.jmedchem.8b01612
Homo sapiens	A549	Activity	nan	None	10.1021/jm401117t
Homo sapiens	A549	Drug uptake	2.3	uM	10.1016/j.bmcl.2013.08.008
Homo sapiens	A549	Drug uptake	271.0	uM	10.1016/j.bmcl.2013.08.008
Homo sapiens	A549	EC50	18700.0	nM	10.1021/acs.jmedchem.7b00515
Homo sapiens	A549	FC	1.0	None	10.1016/j.ejmech.2009.01.035
Homo sapiens	A549	FC	5.0	None	10.1016/j.ejmech.2017.12.022
Homo sapiens	A549	FC	22.0	None	10.1016/j.ejmech.2017.12.022
Homo sapiens	A549	FC	26.0	None	10.1016/j.ejmech.2017.12.022
Homo sapiens	A549	FC	61.0	None	10.1016/j.ejmech.2017.12.022
Homo sapiens	A549	GI50	2860.0	nM	10.1016/j.bmc.2016.08.002
Homo sapiens	A549	GI50	7940.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	A549	GI50	7940.0	nM	10.1016/j.bmcl.2019.04.029
Homo sapiens	A549	GI50	9300.0	nM	10.1021/acs.jmedchem.6b01774
Homo sapiens	A549	IC50	7.0	nM	10.1016/j.ejmech.2020.112388
Homo sapiens	A549	IC50	130.0	nM	10.1016/j.bmc.2015.04.065
Homo sapiens	A549	IC50	1260.0	nM	10.1016/j.bmc.2018.03.025
Homo sapiens	A549	IC50	2110.0	nM	10.1016/j.bmcl.2019.08.022
Homo sapiens	A549	IC50	2170.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	A549	IC50	2640.0	nM	10.1016/j.bmcl.2021.128503
Homo sapiens	A549	IC50	2650.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	A549	IC50	2690.0	nM	10.1016/j.ejmech.2021.113984
Homo sapiens	A549	IC50	2860.0	nM	10.1016/j.bmcl.2015.08.026
Homo sapiens	A549	IC50	2960.0	nM	10.1016/j.ejmech.2018.11.059
Homo sapiens	A549	IC50	3530.0	nM	10.1016/j.bmcl.2021.127987
Homo sapiens	A549	IC50	4626.0	nM	10.1016/j.ejmech.2013.05.026
Homo sapiens	A549	IC50	5000.0	nM	10.1016/j.bmcl.2017.02.023
Homo sapiens	A549	IC50	5740.0	nM	10.1021/acsmedchemlett.8b00270
Homo sapiens	A549	IC50	5760.0	nM	10.1016/j.bmc.2015.12.001
Homo sapiens	A549	IC50	7000.0	nM	10.1016/j.ejmech.2009.01.035
Homo sapiens	A549	IC50	8270.0	nM	10.1016/j.ejmech.2018.01.081
Homo sapiens	A549	IC50	8280.0	nM	10.1016/j.ejmech.2015.10.045
Homo sapiens	A549	IC50	8400.0	nM	10.1021/acs.jmedchem.5b00354
Homo sapiens	A549	IC50	8510.0	nM	10.1007/s00044-013-0734-x
Homo sapiens	A549	IC50	9280.0	nM	10.1016/j.bmcl.2016.02.009
Homo sapiens	A549	IC50	9860.0	nM	10.1016/j.bmc.2017.03.039
Homo sapiens	A549	IC50	9860.0	nM	10.1016/j.ejmech.2015.09.031
Homo sapiens	A549	IC50	10000.0	nM	10.1016/j.bmc.2016.04.046
Homo sapiens	A549	IC50	10000.0	nM	10.1016/j.bmcl.2018.12.020
Homo sapiens	A549	IC50	10000.0	nM	10.1016/j.ejmech.2019.111888
Homo sapiens	A549	IC50	10000.0	nM	10.1021/ml4002437
Homo sapiens	A549	IC50	10070.0	nM	10.1016/j.bmc.2018.11.009
Homo sapiens	A549	IC50	10070.0	nM	10.1016/j.ejmech.2017.03.083
Homo sapiens	A549	IC50	10080.0	nM	10.1016/j.ejmech.2011.11.015
Homo sapiens	A549	IC50	10210.0	nM	10.1021/jm201591k
Homo sapiens	A549	IC50	10450.0	nM	10.1016/j.bmc.2018.02.023
Homo sapiens	A549	IC50	10500.0	nM	10.1016/j.bmcl.2020.127003
Homo sapiens	A549	IC50	11020.0	nM	10.1016/j.bmcl.2015.08.076
Homo sapiens	A549	IC50	11080.0	nM	10.1021/acs.jmedchem.8b01612
Homo sapiens	A549	IC50	11670.0	nM	10.1016/j.bmc.2014.10.038
Homo sapiens	A549	IC50	11800.0	nM	10.1016/j.bmc.2012.05.034
Homo sapiens	A549	IC50	12080.0	nM	10.1016/j.ejmech.2017.07.005
Homo sapiens	A549	IC50	12170.0	nM	10.1016/j.bmc.2014.10.038
Homo sapiens	A549	IC50	12920.0	nM	10.1016/j.bmc.2013.09.027
Homo sapiens	A549	IC50	13260.0	nM	10.1016/j.ejmech.2022.114231
Homo sapiens	A549	IC50	13320.0	nM	10.1016/j.bmc.2016.01.003
Homo sapiens	A549	IC50	13590.0	nM	10.1016/j.ejmech.2008.01.009
Homo sapiens	A549	IC50	14471.16	nM	10.6019/CHEMBL1201861
Homo sapiens	A549	IC50	14803.0	nM	10.1016/j.bmc.2019.06.001
Homo sapiens	A549	IC50	15580.0	nM	10.1016/j.ejmech.2014.02.032
Homo sapiens	A549	IC50	15580.0	nM	10.1021/jm400463q
Homo sapiens	A549	IC50	15590.0	nM	10.1016/j.ejmech.2021.113300
Homo sapiens	A549	IC50	15790.0	nM	10.1016/j.ejmech.2020.112185
Homo sapiens	A549	IC50	17900.0	nM	10.1016/j.bmc.2019.02.044
Homo sapiens	A549	IC50	20000.0	nM	10.1016/j.ejmech.2019.111607
Homo sapiens	A549	IC50	20300.0	nM	10.1016/j.bmcl.2013.07.049
Homo sapiens	A549	IC50	21170.0	nM	10.1016/j.ejmech.2017.06.023
Homo sapiens	A549	IC50	21170.0	nM	10.1016/j.ejmech.2018.01.090
Homo sapiens	A549	IC50	21170.0	nM	10.1016/j.ejmech.2019.06.015
Homo sapiens	A549	IC50	21900.0	nM	10.1016/j.bmcl.2017.08.063
Homo sapiens	A549	IC50	22500.0	nM	10.1016/j.bmcl.2017.03.094
Homo sapiens	A549	IC50	24250.0	nM	10.1016/j.ejmech.2016.04.026
Homo sapiens	A549	IC50	36210.0	nM	10.1016/j.bmc.2017.03.032
Homo sapiens	A549	IC50	37930.0	nM	10.1016/j.bmc.2010.04.046
Homo sapiens	A549	IC50	39700.0	nM	10.1016/j.ejmech.2016.01.045
Homo sapiens	A549	IC50	50000.0	nM	10.1021/acs.jmedchem.2c00272
Homo sapiens	A549	IC50	nan	None	10.1016/j.ejmech.2013.03.013
Homo sapiens	A549	IC50	nan	None	10.1016/j.ejmech.2013.06.055
Homo sapiens	A549	IG50	21.17	uM	10.1016/j.bmcl.2017.02.027
Homo sapiens	A549	Inhibition	63.0	%	10.1016/j.ejmech.2009.01.035
Homo sapiens	A549	Ratio	112.0	None	10.1016/j.ejmech.2018.11.029
Homo sapiens	A549	TGI	34.31	%	10.1021/acs.jmedchem.8b01612
Homo sapiens	A673	IC50	8676.11	nM	10.6019/CHEMBL1201861
Homo sapiens	A704	IC50	100509.47	nM	10.6019/CHEMBL1201861
Homo sapiens	ABC-1	IC50	12340.99	nM	10.6019/CHEMBL1201861
Homo sapiens	ACHN	IC50	331.4	nM	10.6019/CHEMBL1201861
Homo sapiens	ACN	IC50	580.76	nM	10.6019/CHEMBL1201861
Homo sapiens	Actin-related protein 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Actin-related protein 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Activin receptor type-1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Activin receptor type-1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Activin receptor type-1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Activin receptor type-1	Ki	3981.07	nM	None
Homo sapiens	Activin receptor type-1B	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Activin receptor type-1B	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Activin receptor type-1B	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Activin receptor type-2A	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Activin receptor type-2A	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Activin receptor type-2B	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Activin receptor type-2B	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Activin receptor type-2B	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Acyl-CoA dehydrogenase family member 10	Kd	33795.0	nM	10.1126/science.aan4368
Homo sapiens	Acyl-CoA dehydrogenase family member 11	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Adaptor-associated kinase	Kd	3000.0	nM	10.1021/acs.jmedchem.1c00302
Homo sapiens	Adaptor-associated kinase	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Adaptor-associated kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Adaptor-associated kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Adaptor-associated kinase	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Adenine phosphoribosyltransferase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Adenosine A1 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Adenosine A2a receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Adenosine A3 receptor	AC50	25000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Adenosine kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Adenylate kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	ADP/ATP translocase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	ADP/ATP translocase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	AGS	IC50	5496.18	nM	10.6019/CHEMBL1201861
Homo sapiens	ALK tyrosine kinase receptor	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	ALK tyrosine kinase receptor	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	ALK tyrosine kinase receptor	Ki	1258.93	nM	None
Homo sapiens	ALL-PO	IC50	5225.87	nM	10.6019/CHEMBL1201861
Homo sapiens	Alpha-1a adrenergic receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Alpha-2b adrenergic receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Alpha-2c adrenergic receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	AM-38	IC50	8162.8	nM	10.6019/CHEMBL1201861
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	nan	None	10.1038/nbt1068
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Ki	3981.07	nM	None
Homo sapiens	AMP-activated protein kinase, alpha-2 subunit	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	AMP-activated protein kinase, alpha-2 subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	AMP-activated protein kinase, alpha-2 subunit	Thermal melting change	-0.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	AMP-activated protein kinase, gamma-1 subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	AMP-activated protein kinase, gamma-2 subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	AN3-CA	IC50	22608.37	nM	10.6019/CHEMBL1201861
Homo sapiens	Ankyrin repeat and protein kinase domain-containing protein 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ankyrin repeat and protein kinase domain-containing protein 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Arachidonate 15-lipoxygenase, type II	Potency	19952.6	nM	None
Homo sapiens	ASPC1	IC50	6730.0	nM	10.1016/j.bmc.2018.11.009
Homo sapiens	ASPC1	IC50	32360.48	nM	10.6019/CHEMBL1201861
Homo sapiens	ATN-1	IC50	5411.84	nM	10.6019/CHEMBL1201861
Homo sapiens	ATP-binding cassette sub-family G member 2	Activity	66.0	%	10.1016/j.ejmech.2018.10.026
Homo sapiens	ATP-binding cassette sub-family G member 2	Activity	nan	None	10.1124/mol.65.6.1485
Homo sapiens	ATP-binding cassette sub-family G member 2	EC50	300.0	nM	10.1016/j.ejmech.2022.114231
Homo sapiens	ATP-binding cassette sub-family G member 2	IC50	400.0	nM	10.1124/mol.65.6.1485
Homo sapiens	ATP-binding cassette sub-family G member 2	IC50	500.0	nM	10.1016/j.ejmech.2022.114346
Homo sapiens	ATP-binding cassette sub-family G member 2	IC50	1100.0	nM	10.1016/j.bmcl.2009.11.004
Homo sapiens	ATP-binding cassette sub-family G member 2	IC50	1260.0	nM	10.1016/j.bmcl.2009.11.004
Homo sapiens	ATP-binding cassette sub-family G member 2	IC50	3190.0	nM	10.1016/j.bmc.2013.10.007
Homo sapiens	ATP-binding cassette sub-family G member 2	Inhibition	nan	%	10.1016/j.ejmech.2018.10.026
Homo sapiens	ATP-dependent RNA helicase DDX1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	ATP-dependent RNA helicase DDX3X	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	ATP-dependent RNA helicase DDX42	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	AU565	IC50	869.6	nM	10.6019/CHEMBL1201861
Homo sapiens	BALL-1	IC50	297.42	nM	10.6019/CHEMBL1201861
Homo sapiens	BB30-HNC	IC50	1689.72	nM	10.6019/CHEMBL1201861
Homo sapiens	BB49-HNC	IC50	19920.05	nM	10.6019/CHEMBL1201861
Homo sapiens	BB65-RCC	IC50	2807.13	nM	10.6019/CHEMBL1201861
Homo sapiens	BCPAP	IC50	3082.95	nM	10.6019/CHEMBL1201861
Homo sapiens	BE-13	IC50	1506.71	nM	10.6019/CHEMBL1201861
Homo sapiens	Becker	IC50	19854.67	nM	10.6019/CHEMBL1201861
Homo sapiens	Bel-7402	IC50	11210.0	nM	10.1016/j.ejmech.2020.112661
Homo sapiens	BEN	IC50	16515.46	nM	10.6019/CHEMBL1201861
Homo sapiens	Beta-1 adrenergic receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Beta-2 adrenergic receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Beta-secretase 1	IC50	20000.0	nM	10.1021/acs.jmedchem.6b00078
Homo sapiens	BFTC-905	IC50	5658.78	nM	10.6019/CHEMBL1201861
Homo sapiens	BFTC-909	IC50	9182.97	nM	10.6019/CHEMBL1201861
Homo sapiens	BHT-101	IC50	16243.89	nM	10.6019/CHEMBL1201861
Homo sapiens	BHY	IC50	975.48	nM	10.6019/CHEMBL1201861
Homo sapiens	Bile salt export pump	IC50	10900.0	nM	10.1002/hep.27206
Homo sapiens	Bile salt export pump	IC50	10900.0	nM	10.1093/toxsci/kfq269
Homo sapiens	Bile salt export pump	IC50	10900.0	nM	10.1093/toxsci/kft176
Homo sapiens	BMP-2-inducible protein kinase	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	BMP-2-inducible protein kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	BMP-2-inducible protein kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	BMP-2-inducible protein kinase	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Bone morphogenetic protein receptor type-1A	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Bone morphogenetic protein receptor type-1A	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Bone morphogenetic protein receptor type-1A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Bone morphogenetic protein receptor type-1B	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Bone morphogenetic protein receptor type-1B	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Bone morphogenetic protein receptor type-2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Bone morphogenetic protein receptor type-2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Bone morphogenetic protein receptor type-2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	BPH-1	IC50	491.16	nM	10.6019/CHEMBL1201861
Homo sapiens	Bradykinin B2 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Brain glycogen phosphorylase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Breakpoint cluster region protein	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Bromodomain-containing protein 4	Delta TM	0.5444	C	None
Homo sapiens	BR serine/threonine-protein kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	BR serine/threonine-protein kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	BR serine/threonine-protein kinase 1	Ki	3162.28	nM	None
Homo sapiens	BR serine/threonine-protein kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	BR serine/threonine-protein kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	BT-20	IC50	2267.44	nM	10.6019/CHEMBL1201861
Homo sapiens	BT-474	Activity	nan	None	10.1016/j.ejmech.2011.10.051
Homo sapiens	BT-474	EC50	300.0	nM	10.1016/j.bmcl.2008.11.023
Homo sapiens	BT-474	IC50	360.0	nM	10.1016/j.bmcl.2013.12.079
Homo sapiens	BT-474	IC50	360.0	nM	10.1016/j.bmcl.2016.08.007
Homo sapiens	BT-474	IC50	365.0	nM	10.1016/j.bmcl.2020.127045
Homo sapiens	BT-474	IC50	938.14	nM	10.6019/CHEMBL1201861
Homo sapiens	BT-549	IC50	1587.47	nM	10.6019/CHEMBL1201861
Homo sapiens	BT-549	IC50	6560.0	nM	10.1016/j.ejmech.2018.01.081
Homo sapiens	BV-173	IC50	186.55	nM	10.6019/CHEMBL1201861
Homo sapiens	BXPC-3	IC50	31372.92	nM	10.6019/CHEMBL1201861
Homo sapiens	C2BBe1	IC50	3644.07	nM	10.6019/CHEMBL1201861
Homo sapiens	C32	IC50	9633.4	nM	10.6019/CHEMBL1201861
Homo sapiens	C-33-A	IC50	34685.72	nM	10.6019/CHEMBL1201861
Homo sapiens	C3A	IC50	12578.53	nM	10.6019/CHEMBL1201861
Homo sapiens	C8166	IC50	3465.21	nM	10.6019/CHEMBL1201861
Homo sapiens	Ca9-22	IC50	588.64	nM	10.6019/CHEMBL1201861
Homo sapiens	CAKI-1	IC50	6009.85	nM	10.6019/CHEMBL1201861
Homo sapiens	CAL-120	IC50	6451.62	nM	10.6019/CHEMBL1201861
Homo sapiens	CAL-12T	IC50	2018.61	nM	10.6019/CHEMBL1201861
Homo sapiens	CAL-27	IC50	289.08	nM	10.6019/CHEMBL1201861
Homo sapiens	CAL-33	IC50	370.9	nM	10.6019/CHEMBL1201861
Homo sapiens	CAL-39	IC50	596.3	nM	10.6019/CHEMBL1201861
Homo sapiens	CAL-51	IC50	10087.7	nM	10.6019/CHEMBL1201861
Homo sapiens	CAL-54	IC50	311.23	nM	10.6019/CHEMBL1201861
Homo sapiens	CAL-62	IC50	7398.66	nM	10.6019/CHEMBL1201861
Homo sapiens	CAL-72	IC50	268.73	nM	10.6019/CHEMBL1201861
Homo sapiens	CAL-85-1	IC50	21930.49	nM	10.6019/CHEMBL1201861
Homo sapiens	Calu-3	IC50	985.0	nM	10.1016/j.bmcl.2020.127045
Homo sapiens	Calu-3	IC50	1600.0	nM	10.1021/jm301365e
Homo sapiens	Calu-3	IC50	4520.0	nM	10.1016/j.bmcl.2021.128503
Homo sapiens	Calu-3	IC50	6655.68	nM	10.6019/CHEMBL1201861
Homo sapiens	Calu-6	IC50	17678.21	nM	10.6019/CHEMBL1201861
Homo sapiens	CAMA-1	IC50	12163.26	nM	10.6019/CHEMBL1201861
Homo sapiens	CaM kinase I alpha	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase I alpha	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase I alpha	Kd	nan	None	10.1038/nbt1068
Homo sapiens	CaM kinase I alpha	Ki	6309.57	nM	None
Homo sapiens	CaM kinase I delta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase I delta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase I delta	Kd	nan	None	10.1038/nbt1068
Homo sapiens	CaM kinase I delta	Ki	2511.89	nM	None
Homo sapiens	CaM kinase I delta	Thermal melting change	0.4	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM kinase I gamma	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase I gamma	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase I gamma	Kd	nan	None	10.1038/nbt1068
Homo sapiens	CaM kinase I gamma	Thermal melting change	1.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM kinase II alpha	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase II alpha	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase II alpha	Kd	nan	None	10.1038/nbt1068
Homo sapiens	CaM kinase II alpha	Ki	3981.07	nM	None
Homo sapiens	CaM kinase II alpha	Thermal melting change	0.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM kinase II beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase II beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase II beta	Kd	nan	None	10.1038/nbt1068
Homo sapiens	CaM kinase II beta	Ki	7943.28	nM	None
Homo sapiens	CaM kinase II beta	Thermal melting change	0.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM kinase II delta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase II delta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase II delta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	CaM kinase II delta	Kd	nan	None	10.1038/nbt1068
Homo sapiens	CaM kinase II delta	Ki	2511.89	nM	None
Homo sapiens	CaM kinase II delta	Thermal melting change	0.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM kinase II gamma	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase II gamma	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase II gamma	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	CaM kinase II gamma	Kd	nan	None	10.1038/nbt1068
Homo sapiens	CaM kinase II gamma	Ki	3162.28	nM	None
Homo sapiens	CaM kinase II gamma	Thermal melting change	0.4	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM kinase IV	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase IV	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase IV	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	CaM kinase IV	Thermal melting change	0.6	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM-kinase kinase alpha	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	CaM-kinase kinase alpha	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	CaM-kinase kinase alpha	Kd	nan	None	10.1038/nbt1068
Homo sapiens	CaM-kinase kinase beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	CaM-kinase kinase beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	CaM-kinase kinase beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	CaM-kinase kinase beta	Kd	nan	None	10.1038/nbt1068
Homo sapiens	CaM-kinase kinase beta	Ki	2511.89	nM	None
Homo sapiens	CaM-kinase kinase beta	Thermal melting change	0.7	degrees C	10.1073/pnas.0708800104
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Ki	5011.87	nM	None
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Thermal melting change	1.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	cAMP-dependent protein kinase, gamma catalytic subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	cAMP-dependent protein kinase type II-alpha regulatory subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Canalicular multispecific organic anion transporter 1	Activity	74.0	%	10.1021/jm7015683
Homo sapiens	Canalicular multispecific organic anion transporter 1	IC50	133000.0	nM	10.1093/toxsci/kft176
Homo sapiens	Canalicular multispecific organic anion transporter 2	IC50	133000.0	nM	10.1093/toxsci/kft176
Homo sapiens	Cannabinoid CB1 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	CAPAN-1	IC50	883.29	nM	10.6019/CHEMBL1201861
Homo sapiens	Capan-2	IC50	9401.09	nM	10.6019/CHEMBL1201861
Homo sapiens	CaR-1	IC50	3610.48	nM	10.6019/CHEMBL1201861
Homo sapiens	CAS-1	IC50	30785.94	nM	10.6019/CHEMBL1201861
Homo sapiens	Casein kinase I alpha	IC50	50000.0	nM	10.1038/nchembio.117
Homo sapiens	Casein kinase I alpha	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I alpha	Ki	5011.87	nM	None
Homo sapiens	Casein kinase I delta	Delta TM	1.051	C	None
Homo sapiens	Casein kinase I delta	Kd	3200.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I delta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I delta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I delta	Ki	7943.28	nM	None
Homo sapiens	Casein kinase I epsilon	Kd	430.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I epsilon	Kd	430.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I epsilon	Kd	2000.0	nM	10.1038/nbt1068
Homo sapiens	Casein kinase I epsilon	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I gamma 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I gamma 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I gamma 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I gamma 1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Casein kinase I gamma 1	Ki	6309.57	nM	None
Homo sapiens	Casein kinase I gamma 1	Thermal melting change	0.5	degrees C	10.1073/pnas.0708800104
Homo sapiens	Casein kinase I gamma 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I gamma 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I gamma 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I gamma 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Casein kinase I gamma 2	Ki	7943.28	nM	None
Homo sapiens	Casein kinase I gamma 2	Thermal melting change	-0.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	Casein kinase II alpha	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase II alpha	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase II alpha	Ki	6309.57	nM	None
Homo sapiens	Casein kinase II alpha (prime)	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase II alpha (prime)	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase II alpha (prime)	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I isoform alpha-like	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I isoform alpha-like	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I isoform gamma-3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I isoform gamma-3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I isoform gamma-3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I isoform gamma-3	Ki	6309.57	nM	None
Homo sapiens	Casein kinase I isoform gamma-3	Thermal melting change	0.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	Ca-Ski	IC50	31317.72	nM	10.6019/CHEMBL1201861
Homo sapiens	CCRF-CEM	GI50	5010.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	CCRF-CEM	GI50	5010.0	nM	10.1016/j.bmcl.2019.04.029
Homo sapiens	CCRF-CEM	IC50	1411.1	nM	10.6019/CHEMBL1201861
Homo sapiens	Cell division cycle 2-like protein kinase 6	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cell division cycle 2-like protein kinase 6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cell division cycle 7-related protein kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cell division cycle 7-related protein kinase	Ki	1258.93	nM	None
Homo sapiens	Cell division protein kinase 8	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cell division protein kinase 8	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cell division protein kinase 8	Ki	3981.07	nM	None
Homo sapiens	CFPAC-1	IC50	2438.64	nM	10.6019/CHEMBL1201861
Homo sapiens	cGMP-dependent protein kinase 1 beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	cGMP-dependent protein kinase 1 beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	cGMP-dependent protein kinase 1 beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	cGMP-dependent protein kinase 1 beta	Ki	1995.26	nM	None
Homo sapiens	cGMP-dependent protein kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	cGMP-dependent protein kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	cGMP-dependent protein kinase 2	Ki	1584.89	nM	None
Homo sapiens	CGTH-W-1	IC50	5385.84	nM	10.6019/CHEMBL1201861
Homo sapiens	ChaGo-K-1	IC50	9105.79	nM	10.6019/CHEMBL1201861
Homo sapiens	Chaperone activity of bc1 complex-like, mitochondrial	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Chaperone activity of bc1 complex-like, mitochondrial	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Chaperone activity of bc1 complex-like, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	CHL-1	IC50	208.51	nM	10.6019/CHEMBL1201861
Homo sapiens	Cholecystokinin A receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Cholecystokinin B receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	CHP-212	IC50	50524.23	nM	10.6019/CHEMBL1201861
Homo sapiens	Chromodomain-helicase-DNA-binding protein 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Citron Rho-interacting kinase	Kd	1300.0	nM	10.1038/nbt1358
Homo sapiens	Citron Rho-interacting kinase	Kd	1300.0	nM	10.1038/nbt.1990
Homo sapiens	Citron Rho-interacting kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	c-Jun N-terminal kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	c-Jun N-terminal kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	c-Jun N-terminal kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	c-Jun N-terminal kinase 1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	c-Jun N-terminal kinase 1	Ki	3162.28	nM	None
Homo sapiens	c-Jun N-terminal kinase 2	Kd	1400.0	nM	10.1038/nbt1068
Homo sapiens	c-Jun N-terminal kinase 2	Kd	1700.0	nM	10.1038/nbt.1990
Homo sapiens	c-Jun N-terminal kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	c-Jun N-terminal kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	c-Jun N-terminal kinase 2	Ki	2511.89	nM	None
Homo sapiens	c-Jun N-terminal kinase 3	Kd	2300.0	nM	10.1038/nbt1068
Homo sapiens	c-Jun N-terminal kinase 3	Kd	3200.0	nM	10.1038/nbt1358
Homo sapiens	c-Jun N-terminal kinase 3	Kd	3200.0	nM	10.1038/nbt.1990
Homo sapiens	c-Jun N-terminal kinase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	c-Jun N-terminal kinase 3	Ki	794.33	nM	None
Homo sapiens	CL97	IC50	10000.0	nM	10.1016/j.ejmech.2019.111607
Homo sapiens	CNE	IC50	23500.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	COLO-320-HSR	IC50	15530.66	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-668	IC50	7439.67	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-678	IC50	1734.44	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-679	IC50	39970.83	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-680N	IC50	3004.95	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-684	IC50	753.01	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-741	IC50	23956.48	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-792	IC50	8749.46	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-800	IC50	22765.29	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-824	IC50	27219.48	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-829	IC50	7664.63	nM	10.6019/CHEMBL1201861
Homo sapiens	COR-L105	IC50	662.53	nM	10.6019/CHEMBL1201861
Homo sapiens	COR-L23	IC50	51020.78	nM	10.6019/CHEMBL1201861
Homo sapiens	COR-L88	IC50	882.26	nM	10.6019/CHEMBL1201861
Homo sapiens	CP50-MEL-B	IC50	34659.23	nM	10.6019/CHEMBL1201861
Homo sapiens	CP66-MEL	IC50	45714.34	nM	10.6019/CHEMBL1201861
Homo sapiens	CTB-1	IC50	424.4	nM	10.6019/CHEMBL1201861
Homo sapiens	CTV-1	IC50	1308.0	nM	10.6019/CHEMBL1201861
Homo sapiens	CW-2	IC50	15142.15	nM	10.6019/CHEMBL1201861
Homo sapiens	CWR22R	IC50	14000.0	nM	10.1021/acs.jmedchem.9b02008
Homo sapiens	CWR22R	IC50	50346.14	nM	10.6019/CHEMBL1201861
Homo sapiens	Cyclin-dependent kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 1	Ki	7943.28	nM	None
Homo sapiens	Cyclin-dependent kinase 12	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 13	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 13	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 2	Delta TM	1.137	C	None
Homo sapiens	Cyclin-dependent kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Cyclin-dependent kinase 2	Ki	6309.57	nM	None
Homo sapiens	Cyclin-dependent kinase 2	Thermal melting change	0.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	Cyclin-dependent kinase 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 5	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 5	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Cyclin-dependent kinase 5	Ki	7943.28	nM	None
Homo sapiens	Cyclin-dependent kinase 6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 6	Thermal melting change	0.6	degrees C	10.1073/pnas.0708800104
Homo sapiens	Cyclin-dependent kinase 7	Kd	610.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 7	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 7	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 7	Ki	3981.07	nM	None
Homo sapiens	Cyclin-dependent kinase 9	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 9	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 9	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 9	Ki	1584.89	nM	None
Homo sapiens	Cyclin-dependent kinase-like 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase-like 1	Thermal melting change	0.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	Cyclin-dependent kinase-like 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase-like 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase-like 5	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclooxygenase-2	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Cysteine--tRNA ligase, cytoplasmic	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cytochrome c1, heme protein, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cytochrome P450 3A4	Activity	nan	None	None
Homo sapiens	D-247MG	IC50	23793.87	nM	10.6019/CHEMBL1201861
Homo sapiens	D-263MG	IC50	19017.17	nM	10.6019/CHEMBL1201861
Homo sapiens	D283 Med	IC50	16420.87	nM	10.6019/CHEMBL1201861
Homo sapiens	D-336MG	IC50	10700.48	nM	10.6019/CHEMBL1201861
Homo sapiens	D-392MG	IC50	8662.14	nM	10.6019/CHEMBL1201861
Homo sapiens	D-423MG	IC50	38486.9	nM	10.6019/CHEMBL1201861
Homo sapiens	D-502MG	IC50	17980.83	nM	10.6019/CHEMBL1201861
Homo sapiens	D-542MG	IC50	3442.22	nM	10.6019/CHEMBL1201861
Homo sapiens	D-566MG	IC50	9018.1	nM	10.6019/CHEMBL1201861
Homo sapiens	Daoy	IC50	12454.23	nM	10.6019/CHEMBL1201861
Homo sapiens	DB	IC50	60.96	nM	10.6019/CHEMBL1201861
Homo sapiens	DBTRG-05MG	IC50	632.28	nM	10.6019/CHEMBL1201861
Homo sapiens	dCTP pyrophosphatase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Death-associated protein kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Death-associated protein kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Death-associated protein kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Death-associated protein kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Death-associated protein kinase 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Death-associated protein kinase 3	Kd	5700.0	nM	10.1038/nbt1358
Homo sapiens	Death-associated protein kinase 3	Kd	5700.0	nM	10.1038/nbt.1990
Homo sapiens	Death-associated protein kinase 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Death-associated protein kinase 3	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Death-associated protein kinase 3	Ki	1258.93	nM	None
Homo sapiens	Death-associated protein kinase 3	Thermal melting change	3.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	DEL	IC50	877.65	nM	10.6019/CHEMBL1201861
Homo sapiens	Delta(24)-sterol reductase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Delta opioid receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Deoxycytidine kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Detroit 562	IC50	2698.45	nM	10.6019/CHEMBL1201861
Homo sapiens	Discoidin domain-containing receptor 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Discoidin domain-containing receptor 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Discoidin domain-containing receptor 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	DJM-1	IC50	10173.24	nM	10.6019/CHEMBL1201861
Homo sapiens	DK-MG	IC50	7832.01	nM	10.6019/CHEMBL1201861
Homo sapiens	DLD-1	Activity	65.7	%	10.1016/j.ejmech.2011.07.045
Homo sapiens	DLD-1	Activity	87.0	%	10.1016/j.ejmech.2011.07.045
Homo sapiens	DLD-1	IC50	nan	None	10.1016/j.ejmech.2013.03.013
Homo sapiens	DMS-114	IC50	7296.31	nM	10.6019/CHEMBL1201861
Homo sapiens	DMS-273	IC50	12863.3	nM	10.6019/CHEMBL1201861
Homo sapiens	DMS-79	IC50	2692.84	nM	10.6019/CHEMBL1201861
Homo sapiens	DNA-dependent protein kinase	IC50	50000.0	nM	10.1038/nchembio.117
Homo sapiens	DnaJ homolog subfamily A member 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	DNA replication licensing factor MCM4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	DNA topoisomerase II alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	DNA topoisomerase II beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	DOHH-2	IC50	1000.21	nM	10.6019/CHEMBL1201861
Homo sapiens	DOK	IC50	93.62	nM	10.6019/CHEMBL1201861
Homo sapiens	Dopamine D1 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Dopamine D2 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Dopamine D3 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Dopamine transporter	AC50	12000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	DoTc2-4510	IC50	442.12	nM	10.6019/CHEMBL1201861
Homo sapiens	DSH1	IC50	566.88	nM	10.6019/CHEMBL1201861
Homo sapiens	DU-145	IC50	219.04	nM	10.6019/CHEMBL1201861
Homo sapiens	DU-145	IC50	7300.0	nM	10.1021/acs.jmedchem.9b02008
Homo sapiens	DU-145	IC50	8630.0	nM	10.1016/j.ejmech.2017.07.005
Homo sapiens	DU-145	IC50	42170.0	nM	10.1016/j.bmc.2010.04.046
Homo sapiens	DU-145	IC50	100000.0	nM	10.1016/j.bmc.2019.06.001
Homo sapiens	DU-145	IC50	100000.0	nM	10.1016/j.ejmech.2013.06.055
Homo sapiens	DU-4475	IC50	2990.52	nM	10.6019/CHEMBL1201861
Homo sapiens	Dual serine/threonine and tyrosine protein kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Ki	3162.28	nM	None
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Ki	3981.07	nM	None
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Thermal melting change	0.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 5	Inhibition	86.8	%	10.1016/j.bmc.2018.02.022
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 5	Kd	600.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Thermal melting change	0.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 7	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase CLK2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity protein kinase CLK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase CLK2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity protein kinase CLK2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Dual specificity protein kinase CLK2	Ki	6309.57	nM	None
Homo sapiens	Dual specificity protein kinase CLK2	Thermal melting change	0.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	Dual specificity protein kinase CLK3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity protein kinase CLK3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase CLK3	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Dual specificity protein kinase CLK3	Thermal melting change	0.8	degrees C	10.1073/pnas.0708800104
Homo sapiens	Dual specificity protein kinase CLK4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity protein kinase CLK4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase CLK4	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Dual specificity protein kinase CLK4	Ki	6309.57	nM	None
Homo sapiens	Dual specificity protein kinase TTK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity protein kinase TTK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase TTK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity protein kinase TTK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Dual specificity testis-specific protein kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity testis-specific protein kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity testis-specific protein kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	Ki	5011.87	nM	None
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Ki	2511.89	nM	None
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 3	Ki	5011.87	nM	None
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 4	Ki	7943.28	nM	None
Homo sapiens	Dual specificty protein kinase CLK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificty protein kinase CLK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificty protein kinase CLK1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificty protein kinase CLK1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Dual specificty protein kinase CLK1	Thermal melting change	0.7	degrees C	10.1073/pnas.0708800104
Homo sapiens	Dynamin-like 120 kDa protein, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	ECa-109 cell line	IC50	26470.0	nM	10.1016/j.ejmech.2020.112737
Homo sapiens	ECC10	IC50	352.96	nM	10.6019/CHEMBL1201861
Homo sapiens	EC-GI-10	IC50	788.52	nM	10.6019/CHEMBL1201861
Homo sapiens	EFM-19	IC50	56948.82	nM	10.6019/CHEMBL1201861
Homo sapiens	EFO-21	IC50	9587.35	nM	10.6019/CHEMBL1201861
Homo sapiens	EFO-27	IC50	454.74	nM	10.6019/CHEMBL1201861
Homo sapiens	EGI-1	IC50	8600.88	nM	10.6019/CHEMBL1201861
Homo sapiens	EKVX	IC50	2049.39	nM	10.6019/CHEMBL1201861
Homo sapiens	Electron transfer flavoprotein subunit beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Elongation factor Tu, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	EM-2	IC50	1030.16	nM	10.6019/CHEMBL1201861
Homo sapiens	Endothelin receptor ET-A	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	EOL1	IC50	5.166	nM	10.6019/CHEMBL1201861
Homo sapiens	Ephrin type-A receptor 1	Kd	4000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 1	Kd	4000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-A receptor 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-A receptor 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 2	Ki	3162.28	nM	None
Homo sapiens	Ephrin type-A receptor 3	Kd	5500.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 3	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-A receptor 4	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 5	Kd	1500.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-A receptor 5	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 6	Inhibition	46.0	%	10.1021/acs.jmedchem.6b01774
Homo sapiens	Ephrin type-A receptor 6	Inhibition	84.9	%	10.1016/j.bmc.2018.02.022
Homo sapiens	Ephrin type-A receptor 6	Kd	590.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 6	Kd	590.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 6	Kd	1400.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 7	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 7	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 7	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-A receptor 7	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 8	Kd	1800.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 8	Kd	1800.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 8	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ephrin type-B receptor 1	Kd	1300.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 1	Kd	7300.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-B receptor 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-B receptor 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-B receptor 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-B receptor 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-B receptor 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-B receptor 4	IC50	1000.0	nM	10.1038/nchembio.117
Homo sapiens	Ephrin type-B receptor 4	Kd	2500.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-B receptor 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-B receptor 4	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ephrin type-B receptor 6	Kd	3200.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Epidermal growth factor receptor	IC50	0.637	nM	10.1016/j.ejmech.2016.04.026
Homo sapiens	Epidermal growth factor receptor	IC50	2.6	nM	10.1016/j.bmc.2015.12.001
Homo sapiens	Epidermal growth factor receptor	IC50	6.2	nM	10.1021/acs.jmedchem.5b01073
Homo sapiens	Epidermal growth factor receptor	IC50	8.7	nM	10.1021/jm400822z
Homo sapiens	Epidermal growth factor receptor	IC50	22.0	nM	10.1016/j.bmc.2016.05.063
Homo sapiens	Epidermal growth factor receptor	Inhibition	nan	%	10.1021/jm201591k
Homo sapiens	Epidermal growth factor receptor erbB1	AC50	3.8	nM	10.1038/s41467-023-40064-9
Homo sapiens	Epidermal growth factor receptor erbB1	Activity	100.0	%	10.1016/j.ejmech.2021.113786
Homo sapiens	Epidermal growth factor receptor erbB1	Activity	nan	None	10.1021/acs.jmedchem.9b01566
Homo sapiens	Epidermal growth factor receptor erbB1	Activity	nan	None	10.1021/jm4012388
Homo sapiens	Epidermal growth factor receptor erbB1	EC50	2162.0	nM	10.1021/acs.jmedchem.6b01626
Homo sapiens	Epidermal growth factor receptor erbB1	EC50	10733.0	nM	10.1021/acs.jmedchem.6b01626
Homo sapiens	Epidermal growth factor receptor erbB1	FC	0.347	None	10.1016/j.bmc.2020.115889
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.1	nM	10.1016/j.ejmech.2013.05.026
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.1	nM	10.1016/j.ejmech.2014.02.032
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.1	nM	10.1016/j.ejmech.2021.113786
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.1	nM	10.1021/jm400463q
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.15	nM	10.1016/j.bmcl.2017.02.023
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.17	nM	10.1016/j.bmcl.2017.02.023
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.2	nM	10.1016/j.ejmech.2013.05.026
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.2	nM	10.1016/j.ejmech.2014.02.032
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.2	nM	10.1021/jm400463q
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.32	nM	10.1016/j.ejmech.2021.113786
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.45	nM	10.1016/j.bmc.2014.10.038
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.45	nM	10.1016/j.ejmech.2014.11.010
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.47	nM	10.1016/j.ejmech.2018.11.029
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.5	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.5	nM	10.1021/acsmedchemlett.8b00270
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.509	nM	10.1016/j.bmc.2016.05.063
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.585	nM	10.1016/j.ejmech.2016.04.026
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.6	nM	10.1016/j.bmcl.2013.08.008
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.769	nM	10.1016/j.bmc.2019.06.001
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.9	nM	10.1021/acs.jmedchem.2c01041
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	0.96	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1016/j.bmcl.2003.10.010
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1016/j.bmcl.2011.01.119
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1016/j.bmcl.2011.10.103
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1016/j.bmcl.2013.12.079
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1016/j.bmcl.2016.08.007
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1016/j.bmcl.2020.127045
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1021/acs.jmedchem.5b01082
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1021/acs.jmedchem.6b01626
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1021/acs.jmedchem.7b00316
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1021/acs.jmedchem.7b00515
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1021/jm500007h
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1021/jm901132v
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.0	nM	10.1038/nchembio.117
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.268	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.3	nM	10.1016/j.bmc.2015.12.001
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.4	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.43	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.5	nM	10.1016/j.ejmech.2018.01.090
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.6	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.9	nM	10.1016/j.bmc.2020.115897
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1.9	nM	10.1016/j.ejmech.2022.114502
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	2.1	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	2.2	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	2.21	nM	10.1016/j.ejmech.2017.07.005
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	2.3	nM	10.1016/j.ejmech.2018.01.081
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	2.6	nM	10.1016/j.bmc.2016.01.003
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3.0	nM	10.1021/acs.jmedchem.6b00883
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3.0	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3.1	nM	10.1021/acs.jmedchem.9b01617
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3.1	nM	10.1021/jm050936o
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3.1	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3.2	nM	10.1016/j.ejmech.2018.01.090
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3.22	nM	10.1016/j.bmcl.2017.02.027
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3.22	nM	10.1016/j.bmcl.2017.08.035
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3.22	nM	10.1016/j.ejmech.2017.06.023
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3.25	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3.7	nM	10.1016/j.bmc.2018.12.032
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3.8	nM	10.1021/acs.jmedchem.2c01041
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	4.0	nM	10.1016/j.bmc.2017.10.030
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	4.0	nM	10.1016/j.bmc.2021.116039
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	4.0	nM	10.1021/acs.jmedchem.6b01774
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	4.0	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	4.2	nM	10.1016/j.bmc.2011.06.022
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	5.0	nM	10.1021/acs.jmedchem.6b00995
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	5.4	nM	10.1016/j.bmc.2007.03.055
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	5.8	nM	10.1021/acs.jmedchem.8b01612
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	6.5	nM	10.1021/acs.jmedchem.5b01073
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	6.7	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	7.0	nM	10.1021/acs.jmedchem.6b00618
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	7.3	nM	10.1016/j.ejmech.2012.01.021
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	8.0	nM	10.1021/acs.jmedchem.6b00995
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	8.43	nM	10.1016/j.ejmech.2022.114231
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	9.0	nM	10.1016/j.bmcl.2018.06.043
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	9.6	nM	10.1016/j.bmc.2016.10.006
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	10.6	nM	10.1016/j.bmc.2017.03.032
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	11.0	nM	10.1016/j.ejmech.2016.12.014
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	11.5	nM	10.1016/j.ejmech.2018.06.061
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	11.75	nM	10.1016/j.bmcl.2022.129104
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	11.8	nM	10.1016/j.bmcl.2016.02.009
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	12.0	nM	10.1016/j.bmcl.2017.09.048
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	12.0	nM	10.1016/j.bmcl.2018.12.020
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	12.5	nM	10.1016/j.ejmech.2018.06.061
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	13.0	nM	10.1039/C5MD00208G
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	14.0	nM	10.1021/acs.jmedchem.6b00883
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	14.2	nM	10.1016/j.ejmech.2019.111966
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	14.4	nM	10.1021/jm050936o
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	15.0	nM	10.1021/acs.jmedchem.9b00350
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	15.5	nM	10.1016/j.bmc.2018.11.009
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	15.5	nM	10.1016/j.ejmech.2016.01.045
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	15.5	nM	10.1016/j.ejmech.2017.03.083
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	15.5	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	17.1	nM	10.1016/j.ejmech.2021.113300
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	18.0	nM	10.1016/j.ejmech.2020.112062
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	20.0	nM	10.1016/j.bmcl.2014.03.072
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	20.0	nM	10.1016/j.ejmech.2007.09.018
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	20.0	nM	10.1016/j.ejmech.2011.11.015
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	20.0	nM	10.1021/jm1000198
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	20.0	nM	10.1021/jm100607r
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	21.0	nM	10.1016/j.bmc.2009.11.035
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	22.0	nM	10.1016/j.ejmech.2015.08.027
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	22.0	nM	10.1016/j.ejmech.2015.09.031
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	22.0	nM	10.1021/jm800829v
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	22.5	nM	10.1016/j.bmc.2016.01.003
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	23.0	nM	10.1016/j.bmcl.2006.06.054
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	23.0	nM	10.1016/j.bmcl.2013.07.049
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	23.0	nM	10.1016/j.ejmech.2017.12.022
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	23.0	nM	10.1016/s0960-894x(01)00344-4
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	25.0	nM	10.1016/j.bmcl.2013.12.079
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	25.0	nM	10.1016/j.bmcl.2016.02.009
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	25.0	nM	10.1016/j.bmcl.2016.08.007
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	25.0	nM	10.1016/j.bmcl.2020.127045
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	26.0	nM	10.1016/j.ejmech.2015.07.030
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	26.0	nM	10.1016/j.ejmech.2019.03.004
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	27.0	nM	10.1016/j.ejmech.2018.05.006
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	29.0	nM	10.1021/acs.jmedchem.9b00722
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	29.16	nM	10.1016/j.ejmech.2021.113865
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	29.6	nM	10.1016/j.bmc.2018.02.023
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	31.0	nM	10.1016/j.ejmech.2020.112185
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1016/j.bmc.2009.12.048
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1016/j.bmc.2016.10.006
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1016/j.bmcl.2006.02.025
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1016/j.bmcl.2008.11.023
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1016/j.bmcl.2009.05.060
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1016/j.bmcl.2017.09.048
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1016/j.bmcl.2022.129045
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1016/j.ejmech.2010.02.056
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1016/j.ejmech.2012.10.017
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1016/j.ejmech.2020.113016
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1016/j.ejmech.2020.113019
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1016/j.ejmech.2021.113218
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1021/acs.jmedchem.0c01467
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1021/acs.jmedchem.1c00302
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	33.0	nM	10.1021/jm400072p
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	37.0	nM	10.1016/j.bmc.2020.115657
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	39.0	nM	10.1016/j.bmcl.2007.08.061
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	39.9	nM	10.1016/j.bmcl.2013.08.008
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	45.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	54.0	nM	10.1016/j.bmcl.2006.02.025
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	60.0	nM	10.1016/j.ejmech.2018.11.029
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	62.0	nM	10.1016/j.ejmech.2022.114661
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	62.0	nM	10.1021/jm400822z
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	70.0	nM	10.1016/j.bmcl.2011.01.137
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	70.0	nM	10.1039/C0MD00183J
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	72.0	nM	10.1016/j.ejmech.2012.06.055
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	76.0	nM	10.1016/j.bmc.2016.04.046
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	76.0	nM	10.1016/j.bmc.2017.03.039
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	76.0	nM	10.1021/jm5014659
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	80.0	nM	10.1016/j.bmcl.2006.06.054
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	83.0	nM	10.1016/j.bmcl.2019.04.029
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	100.0	nM	10.1021/acs.jmedchem.2c01041
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	100.0	nM	10.1021/acs.jmedchem.5b01082
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	127.0	nM	10.1016/j.bmc.2016.05.063
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	127.9	nM	10.1016/j.ejmech.2018.01.090
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	129.7	nM	10.1016/j.ejmech.2018.06.061
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	148.7	nM	10.1021/acs.jmedchem.8b01612
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	166.0	nM	10.1016/j.bmcl.2021.127987
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	173.0	nM	10.1016/j.bmc.2016.04.046
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	173.0	nM	10.1016/j.bmc.2017.03.039
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	185.0	nM	10.1021/acs.jmedchem.7b00316
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	188.0	nM	10.1021/acs.jmedchem.6b01626
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	190.0	nM	10.1021/acs.jmedchem.7b00515
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	280.0	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	296.4	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	378.4	nM	10.1016/j.ejmech.2021.113300
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	380.0	nM	10.1016/j.ejmech.2015.03.004
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	390.0	nM	10.1021/acs.jnatprod.9b00659
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	460.0	nM	10.1016/j.bmcl.2018.12.020
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	498.0	nM	10.1016/j.bmcl.2013.08.008
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	515.0	nM	10.1016/s0960-894x(02)00598-x
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	639.0	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	777.1	nM	10.1016/j.ejmech.2019.111966
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	823.3	nM	10.1016/j.bmc.2018.11.009
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	823.3	nM	10.1016/j.ejmech.2017.03.083
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	823.7	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	832.3	nM	10.1016/j.ejmech.2016.01.045
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	832.3	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	845.0	nM	10.1039/C5MD00208G
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	941.0	nM	10.1016/j.ejmech.2013.05.026
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	941.0	nM	10.1016/j.ejmech.2014.02.032
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	941.0	nM	10.1021/jm400463q
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1000.0	nM	10.1016/j.bmc.2017.10.030
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1000.0	nM	10.1016/j.bmc.2021.116039
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1013.0	nM	10.1016/j.ejmech.2016.04.026
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1080.0	nM	10.1016/j.bmc.2012.05.034
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1100.0	nM	10.1016/j.bmc.2013.09.027
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1100.0	nM	10.1021/acs.jmedchem.6b00995
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1202.0	nM	10.1016/j.bmc.2017.03.032
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1730.0	nM	10.1021/jm5014659
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1740.0	nM	10.1016/j.bmc.2020.115373
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	1900.0	nM	10.1021/acs.jmedchem.6b00995
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	2000.0	nM	10.1016/j.ejmech.2018.01.090
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	2753.0	nM	10.1016/j.bmc.2007.03.055
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	2815.0	nM	10.1021/jm1000198
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	2815.0	nM	10.1021/jm100607r
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	2874.7	nM	10.1016/j.bmc.2018.02.023
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3100.0	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3170.0	nM	10.1021/acs.jnatprod.9b00659
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	3300.0	nM	10.1021/jm400822z
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	4000.0	nM	10.1021/ml4002437
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	4000.0	nM	10.1039/C3MD00118K
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	4270.0	nM	10.1016/j.ejmech.2015.09.031
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	4990.0	nM	10.1021/acs.jnatprod.9b00659
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	5000.0	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	6746.0	nM	10.1021/acs.jmedchem.9b00722
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	7680.0	nM	10.1016/j.bmcl.2017.09.048
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	10000.0	nM	10.1016/j.bmc.2016.05.063
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	10480.0	nM	10.1021/ml4002437
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	10620.0	nM	10.1016/j.ejmech.2015.09.031
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	12720.0	nM	10.1016/j.ejmech.2015.09.031
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	13980.0	nM	10.1039/C3MD00118K
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	15500.0	nM	10.1016/j.bmcl.2021.128238
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	22800.0	nM	10.1016/j.bmcl.2017.09.048
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	0.94	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	3.3	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	8.0	%	10.1016/j.ejmech.2018.11.029
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	18.0	%	10.1016/j.ejmech.2018.11.029
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	28.3	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	35.0	%	10.1016/j.bmcl.2004.02.001
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	46.0	%	10.1016/j.ejmech.2018.11.029
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	46.4	%	10.1021/jm201507x
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	55.66	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	61.0	%	10.1016/j.ejmech.2019.111966
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	65.4	%	10.1016/j.bmcl.2006.05.010
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	66.98	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	77.36	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	80.0	%	10.1016/j.ejmech.2019.06.015
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	82.48	%	10.1016/j.bmcl.2017.08.035
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	88.68	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	90.0	%	10.1021/acs.jmedchem.6b00883
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	93.2	%	10.1021/acs.jmedchem.6b01774
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	96.0	%	10.1016/j.bmcl.2013.08.008
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	96.0	%	10.1016/j.ejmech.2018.11.029
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	98.0	%	10.1016/j.ejmech.2019.111966
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	98.37	%	10.1016/j.bmc.2010.04.046
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	98.5	%	10.1016/j.bmc.2014.09.029
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	98.5	%	10.1016/j.ejmech.2013.03.013
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	99.6	%	10.1016/j.ejmech.2012.01.021
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	99.75	%	10.1016/j.bmcl.2023.129265
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	99.83	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	100.0	%	10.1016/j.bmcl.2019.08.022
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	100.0	%	10.1016/j.ejmech.2012.10.017
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	100.0	%	10.1021/jm800829v
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	101.0	%	10.1016/j.ejmech.2016.04.026
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	105.7	%	10.1016/j.bmc.2018.02.022
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.bmc.2009.11.035
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.bmc.2013.07.032
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.bmc.2016.05.063
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.bmc.2018.02.022
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.bmcl.2013.08.008
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.bmcl.2016.04.032
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.bmcl.2017.02.023
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.ejmech.2014.02.032
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.ejmech.2016.01.045
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.ejmech.2017.06.023
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.ejmech.2018.01.090
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.ejmech.2018.11.029
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.ejmech.2019.06.015
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.ejmech.2021.113173
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.ejmech.2021.113300
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1021/acs.jmedchem.2c01041
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1021/acs.jmedchem.9b00722
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1021/acs.jmedchem.9b01566
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1021/jm201591k
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1021/jm301365e
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1021/jm4012388
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1021/jm901558p
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1021/ml4002437
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	0.52	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	0.52	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	0.54	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	0.54	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	0.57	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	0.57	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	0.94	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	0.94	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	0.98	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	0.98	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	1.0	nM	10.1016/j.bmcl.2019.05.025
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	1.0	nM	10.1021/acs.jmedchem.9b00350
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	1.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	1.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	1.1	nM	10.1021/acs.jmedchem.9b01566
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	1.1	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	1.1	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	1.4	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	1.4	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	1.8	nM	10.1038/nbt1068
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	2.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	2.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	2.4	nM	10.1021/jm8010542
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	2.4	nM	10.1039/C5MD00208G
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	10.9	nM	10.1021/jm8010542
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	10.9	nM	10.1039/C5MD00208G
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	35.3	nM	10.1021/jm8010542
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	40.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	413.0	nM	10.1126/science.aan4368
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	470.0	nM	10.1021/acs.jmedchem.1c00649
Homo sapiens	Epidermal growth factor receptor erbB1	Ki	0.4	nM	10.1016/j.chembiol.2005.04.011
Homo sapiens	Epidermal growth factor receptor erbB1	Potency	3.2	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	Potency	1122.0	nM	None
Homo sapiens	Epidermal growth factor receptor erbB1	Ratio	505.3	None	10.1016/j.bmc.2007.03.055
Homo sapiens	Epidermal growth factor receptor erbB1	Ratio IC50	3.2	None	10.1016/j.ejmech.2021.113786
Homo sapiens	Epidermal growth factor receptor erbB1	Ratio IC50	12.5	None	10.1016/j.bmcl.2013.08.008
Homo sapiens	Epidermal growth factor receptor erbB1	TIME	0.1667	hr	10.1016/j.ejmech.2017.07.023
Homo sapiens	Epithelial discoidin domain-containing receptor 1	Inhibition	98.1	%	10.1016/j.bmc.2018.02.022
Homo sapiens	Epithelial discoidin domain-containing receptor 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Epithelial discoidin domain-containing receptor 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Epithelial discoidin domain-containing receptor 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	EPLC-272H	IC50	1855.49	nM	10.6019/CHEMBL1201861
Homo sapiens	ES1	IC50	4960.35	nM	10.6019/CHEMBL1201861
Homo sapiens	ES3	IC50	24002.28	nM	10.6019/CHEMBL1201861
Homo sapiens	ES4	IC50	3822.86	nM	10.6019/CHEMBL1201861
Homo sapiens	ES5	IC50	33729.2	nM	10.6019/CHEMBL1201861
Homo sapiens	ES6	IC50	40455.19	nM	10.6019/CHEMBL1201861
Homo sapiens	ES7	IC50	50164.37	nM	10.6019/CHEMBL1201861
Homo sapiens	ES8	IC50	17859.26	nM	10.6019/CHEMBL1201861
Homo sapiens	ESS-1	IC50	43555.81	nM	10.6019/CHEMBL1201861
Homo sapiens	Estrogen receptor alpha	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	ETK-1	IC50	662.59	nM	10.6019/CHEMBL1201861
Homo sapiens	Eukaryotic peptide chain release factor GTP-binding subunit ERF3B	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Eukaryotic translation initiation factor 2-alpha kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Eukaryotic translation initiation factor 2-alpha kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Eukaryotic translation initiation factor 2-alpha kinase 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Eukaryotic translation initiation factor 2-alpha kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	EW-1	IC50	27355.4	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-11	IC50	4132.61	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-13	IC50	225.1	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-16	IC50	3955.77	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-18	IC50	2354.71	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-22	IC50	30196.89	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-24	IC50	35633.46	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-3	IC50	46.04	nM	10.6019/CHEMBL1201861
Homo sapiens	Exosome RNA helicase MTR4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	FaDu	IC50	50.0	nM	10.1021/jm301365e
Homo sapiens	FaDu	IC50	604.69	nM	10.6019/CHEMBL1201861
Homo sapiens	Ferrochelatase, mitochondrial	Kd	6682.0	nM	10.1126/science.aan4368
Homo sapiens	Fibroblast	Growth Rate	0.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast	Growth Rate	1.0	None	10.6019/CHEMBL4689842
Homo sapiens	Fibroblast growth factor receptor 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Fibroblast growth factor receptor 1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Fibroblast growth factor receptor 1	Ki	3981.07	nM	None
Homo sapiens	Fibroblast growth factor receptor 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Fibroblast growth factor receptor 3	Delta TM	0.4556	C	None
Homo sapiens	Fibroblast growth factor receptor 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 3	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Fibroblast growth factor receptor 3	Ki	1995.26	nM	None
Homo sapiens	Fibroblast growth factor receptor 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Focal adhesion kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Focal adhesion kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Focal adhesion kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Focal adhesion kinase 1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Focal adhesion kinase 1	Ki	1584.89	nM	None
Homo sapiens	FTC-133	IC50	11308.14	nM	10.6019/CHEMBL1201861
Homo sapiens	G-361	IC50	12912.89	nM	10.6019/CHEMBL1201861
Homo sapiens	G-401	IC50	23046.18	nM	10.6019/CHEMBL1201861
Homo sapiens	G-402	IC50	41080.93	nM	10.6019/CHEMBL1201861
Homo sapiens	GAK	IC50	21498.97	nM	10.6019/CHEMBL1201861
Homo sapiens	GAMG	IC50	6506.2	nM	10.6019/CHEMBL1201861
Homo sapiens	GB-1	IC50	26187.91	nM	10.6019/CHEMBL1201861
Homo sapiens	GCIY	IC50	1301.32	nM	10.6019/CHEMBL1201861
Homo sapiens	GCT	IC50	6533.87	nM	10.6019/CHEMBL1201861
Homo sapiens	Geminin	Potency	13335.9	nM	None
Homo sapiens	Geminin	Potency	29855.4	nM	None
Homo sapiens	General transcription and DNA repair factor IIH helicase subunit XPD	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ghrelin receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	GI-1	IC50	21170.0	nM	10.6019/CHEMBL1201861
Homo sapiens	GI-ME-N	IC50	16903.23	nM	10.6019/CHEMBL1201861
Homo sapiens	Glucocorticoid receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Glycine--tRNA ligase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Glycogen synthase kinase-3 alpha	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Glycogen synthase kinase-3 alpha	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Glycogen synthase kinase-3 alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Glycogen synthase kinase-3 alpha	Ki	6309.57	nM	None
Homo sapiens	Glycogen synthase kinase-3 beta	Delta TM	2.442	C	None
Homo sapiens	Glycogen synthase kinase-3 beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Glycogen synthase kinase-3 beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Glycogen synthase kinase-3 beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Glycogen synthase kinase-3 beta	Ki	6309.57	nM	None
Homo sapiens	Glycogen synthase kinase-3 beta	Thermal melting change	0.9	degrees C	10.1073/pnas.0708800104
Homo sapiens	GMS-10	IC50	33300.45	nM	10.6019/CHEMBL1201861
Homo sapiens	GOTO	IC50	11520.57	nM	10.6019/CHEMBL1201861
Homo sapiens	GP5d	IC50	16218.7	nM	10.6019/CHEMBL1201861
Homo sapiens	G-protein coupled receptor kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	G protein-coupled receptor kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	G protein-coupled receptor kinase 5	Ki	3981.07	nM	None
Homo sapiens	G protein-coupled receptor kinase 6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	G protein-coupled receptor kinase 7	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	GR-ST	IC50	4431.8	nM	10.6019/CHEMBL1201861
Homo sapiens	GT3TKB	IC50	12632.67	nM	10.6019/CHEMBL1201861
Homo sapiens	GTP-binding nuclear protein Ran	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Guanine nucleotide-binding protein G(i) subunit alpha-2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	H4	IC50	30465.44	nM	10.6019/CHEMBL1201861
Homo sapiens	H9	IC50	137.2	nM	10.6019/CHEMBL1201861
Homo sapiens	HAL-01	IC50	734.71	nM	10.6019/CHEMBL1201861
Homo sapiens	HC-1	IC50	2940.12	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC1187	IC50	5710.32	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC1395	IC50	48743.21	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC1419	IC50	7468.33	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC1569	IC50	47165.84	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC1806	IC50	337.51	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC1937	IC50	4379.93	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC1954	IC50	11435.99	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC2218	IC50	50.59	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC 2998	IC50	5718.77	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC38	IC50	10971.61	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC70	IC50	2008.15	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC827	Activity	nan	None	10.1021/acs.jmedchem.1c01671
Homo sapiens	HCC827	CC50	26.0	nM	10.1021/acs.jmedchem.9b00722
Homo sapiens	HCC827	EC50	14.0	nM	10.1021/acs.jmedchem.7b00515
Homo sapiens	HCC827	IC50	1.6	nM	10.1016/j.ejmech.2018.01.090
Homo sapiens	HCC827	IC50	1.6	nM	10.1016/j.ejmech.2019.06.015
Homo sapiens	HCC827	IC50	1.69	nM	10.1016/j.ejmech.2021.113984
Homo sapiens	HCC827	IC50	2.0	nM	10.1016/j.bmcl.2017.02.023
Homo sapiens	HCC827	IC50	6.0	nM	10.1016/j.ejmech.2017.03.083
Homo sapiens	HCC827	IC50	6.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	HCC827	IC50	9.9	nM	10.1016/j.bmc.2017.03.032
Homo sapiens	HCC827	IC50	10.0	nM	10.1016/j.ejmech.2019.111888
Homo sapiens	HCC827	IC50	33.3	nM	10.1016/j.bmc.2018.03.025
Homo sapiens	HCC827	TGI	nan	None	10.1021/acs.jmedchem.9b00722
Homo sapiens	HCE-4	IC50	10112.19	nM	10.6019/CHEMBL1201861
Homo sapiens	HCE-T	IC50	279.79	nM	10.6019/CHEMBL1201861
Homo sapiens	HCT-116	GI50	7940.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	HCT-116	IC50	5980.0	nM	10.1016/j.ejmech.2018.01.081
Homo sapiens	HCT-116	IC50	10000.0	nM	10.1021/jm301365e
Homo sapiens	HCT-116	IC50	19820.0	nM	10.1016/j.ejmech.2019.111665
Homo sapiens	HCT-116	IC50	21550.0	nM	10.1016/j.bmc.2019.02.044
Homo sapiens	HCT-116	IC50	25418.57	nM	10.6019/CHEMBL1201861
Homo sapiens	HCT-116	IC50	66900.0	nM	10.1016/j.bmc.2012.09.034
Homo sapiens	HCT-116	IC50	nan	None	10.1016/j.ejmech.2013.03.013
Homo sapiens	HCT-116	Inhibition	nan	%	10.1016/j.ejmech.2019.111665
Homo sapiens	HCT-15	GI50	5010.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	HCT-15	IC50	34127.04	nM	10.6019/CHEMBL1201861
Homo sapiens	HDLM-2	IC50	6014.89	nM	10.6019/CHEMBL1201861
Homo sapiens	HD-MY-Z	IC50	5685.81	nM	10.6019/CHEMBL1201861
Homo sapiens	HEC-1	IC50	10408.14	nM	10.6019/CHEMBL1201861
Homo sapiens	HEK-293T	CC50	52030.0	nM	10.1016/j.bmcl.2015.03.022
Homo sapiens	HEK-293T	Growth Rate	0.0	None	10.6019/CHEMBL4689842
Homo sapiens	HEL	IC50	7375.21	nM	10.6019/CHEMBL1201861
Homo sapiens	HeLa	EC50	nan	None	10.1021/jm500873e
Homo sapiens	HeLa	GI50	1520.0	nM	10.1016/j.bmc.2016.08.002
Homo sapiens	HeLa	IC50	1480.0	nM	10.1016/j.bmcl.2018.05.004
Homo sapiens	HeLa	IC50	1520.0	nM	10.1016/j.bmcl.2015.08.026
Homo sapiens	HeLa	IC50	2260.0	nM	10.1016/j.bmcl.2015.03.022
Homo sapiens	HeLa	IC50	2670.0	nM	10.1016/j.bmcl.2014.03.072
Homo sapiens	HeLa	IC50	4300.0	nM	10.1016/j.ejmech.2018.03.076
Homo sapiens	HeLa	IC50	15400.0	nM	10.1016/j.bmcl.2015.08.076
Homo sapiens	HeLa	IC50	18300.0	nM	10.1016/j.bmcl.2017.03.094
Homo sapiens	HeLa	IC50	23920.0	nM	10.1016/j.ejmech.2020.112737
Homo sapiens	HeLa	IC50	39320.0	nM	10.1016/j.bmcl.2021.128503
Homo sapiens	HeLa	IC50	45590.0	nM	10.1016/j.ejmech.2010.03.001
Homo sapiens	HeLa	IC50	108300.0	nM	10.1016/j.bmc.2012.09.034
Homo sapiens	H-EMC-SS	IC50	45769.27	nM	10.6019/CHEMBL1201861
Homo sapiens	Heme oxygenase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	HEp-2	CC50	100000.0	nM	10.1021/acs.jmedchem.0c01467
Homo sapiens	Hepatocyte growth factor receptor	Inhibition	28.18	%	10.1016/j.bmc.2010.04.046
Homo sapiens	Hepatocyte growth factor receptor	Inhibition	nan	%	10.1016/j.bmc.2013.07.032
Homo sapiens	Hepatocyte growth factor receptor	Kd	3500.0	nM	10.1038/nbt.1990
Homo sapiens	Hepatocyte growth factor receptor	Kd	4372.0	nM	10.1126/science.aan4368
Homo sapiens	Hepatocyte growth factor receptor	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Hepatocyte growth factor receptor	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Hepatocyte growth factor receptor	Ki	2511.89	nM	None
Homo sapiens	HepG2	Activity	42.08	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	HepG2	Activity	45.24	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	HepG2	Activity	45.36	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	HepG2	Activity	47.62	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	HepG2	Activity	48.69	%	10.1016/j.ejmech.2017.07.005
Homo sapiens	HepG2	Activity	75.0	%	10.1021/jm501177w
Homo sapiens	HepG2	IC50	120.0	nM	10.1016/j.bmc.2015.04.065
Homo sapiens	HepG2	IC50	6420.0	nM	10.1016/j.bmcl.2014.03.072
Homo sapiens	HepG2	IC50	6420.0	nM	10.1016/j.ejmech.2012.05.039
Homo sapiens	HepG2	IC50	6600.0	nM	10.1021/acs.jnatprod.8b00821
Homo sapiens	HepG2	IC50	7520.0	nM	10.1016/j.bmcl.2016.04.032
Homo sapiens	HepG2	IC50	10000.0	nM	10.1016/j.bmcl.2015.06.076
Homo sapiens	HepG2	IC50	10000.0	nM	10.1016/j.ejmech.2020.113102
Homo sapiens	HepG2	IC50	10000.0	nM	10.1021/jm301365e
Homo sapiens	HepG2	IC50	15900.0	nM	10.1016/j.bmcl.2017.03.094
Homo sapiens	HepG2	IC50	18220.0	nM	10.1016/j.ejmech.2015.10.045
Homo sapiens	HepG2	IC50	18360.0	nM	10.1016/j.bmc.2019.02.044
Homo sapiens	HepG2	IC50	24190.0	nM	10.1016/j.ejmech.2020.112737
Homo sapiens	HepG2	IC50	29790.0	nM	10.1016/j.bmc.2019.06.001
Homo sapiens	HepG2	IC50	29790.0	nM	10.1016/j.ejmech.2013.06.055
Homo sapiens	HepG2	IC50	29790.0	nM	10.1016/j.ejmech.2017.07.005
Homo sapiens	HepG2	IC50	33900.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	HepG2	IC50	50000.0	nM	10.1016/j.bmc.2016.04.046
Homo sapiens	HepG2	IC50	nan	None	10.1016/j.bmcl.2015.08.026
Homo sapiens	HERG	AC50	1600.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	HERG	IC50	nan	None	10.1021/acsmedchemlett.8b00270
Homo sapiens	HGC-27	IC50	12440.0	nM	10.1016/j.ejmech.2019.03.030
Homo sapiens	HGC-27	IC50	20139.42	nM	10.6019/CHEMBL1201861
Homo sapiens	HH	IC50	2498.54	nM	10.6019/CHEMBL1201861
Homo sapiens	Histamine H1 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Histamine H2 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Histamine H3 receptor	AC50	9900.1	nM	10.1038/s41467-023-40064-9
Homo sapiens	Histone deacetylase	IC50	nan	None	10.1016/j.bmc.2012.05.034
Homo sapiens	Histone deacetylase	Inhibition	nan	%	10.1016/j.ejmech.2021.113173
Homo sapiens	Histone deacetylase 1	IC50	nan	None	10.1016/j.bmc.2016.10.006
Homo sapiens	Histone deacetylase 6	IC50	nan	None	10.1016/j.bmc.2016.10.006
Homo sapiens	Histone deacetylase 6	Inhibition	8.19	%	10.6019/CHEMBL4808148
Homo sapiens	Histone deacetylase 6	Inhibition	11.42	%	10.6019/CHEMBL4808148
Homo sapiens	HL-60	IC50	4122.41	nM	10.6019/CHEMBL1201861
Homo sapiens	HL-60	IC50	54500.0	nM	10.1016/j.bmc.2012.05.034
Homo sapiens	HLE	IC50	18314.77	nM	10.6019/CHEMBL1201861
Homo sapiens	HMV-2 cell line	IC50	98582.42	nM	10.6019/CHEMBL1201861
Homo sapiens	HN	IC50	517.38	nM	10.6019/CHEMBL1201861
Homo sapiens	HN5	EC50	10.0	nM	10.1016/j.bmcl.2008.11.023
Homo sapiens	HO-1-N-1	IC50	509.25	nM	10.6019/CHEMBL1201861
Homo sapiens	Homeodomain-interacting protein kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Homeodomain-interacting protein kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Homeodomain-interacting protein kinase 2	Ki	3162.28	nM	None
Homo sapiens	Homeodomain-interacting protein kinase 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Homeodomain-interacting protein kinase 4	Inhibition	82.8	%	10.1016/j.bmc.2018.02.022
Homo sapiens	Homeodomain-interacting protein kinase 4	Kd	310.0	nM	10.1038/nbt.1990
Homo sapiens	Homeodomain-interacting protein kinase 4	Ki	1258.93	nM	None
Homo sapiens	Homo sapiens	Activity	nan	None	10.1002/hep.27206
Homo sapiens	Homo sapiens	AUC	2402.14	ng.hr.mL-1	10.1093/toxsci/kft176
Homo sapiens	Homo sapiens	Cmax	356.0	nM	10.1002/hep.27206
Homo sapiens	Homo sapiens	Css	0.224	uM	10.1093/toxsci/kft176
Homo sapiens	Homo sapiens	DILI_Concern	nan	None	10.1016/j.drudis.2016.02.015
Homo sapiens	Homo sapiens	DILI_severity_class	4.0	None	10.1016/j.drudis.2016.02.015
Homo sapiens	Homo sapiens	F	60.0	%	10.1016/j.bmc.2007.08.060
Homo sapiens	Homo sapiens	Ratio	0.021	None	10.1093/toxsci/kft176
Homo sapiens	Homo sapiens	Ratio	0.049	None	10.1093/toxsci/kft176
Homo sapiens	Homo sapiens	T1/2	28.0	hr	10.1016/j.bmcl.2006.06.054
Homo sapiens	Homo sapiens	T1/2	37.0	hr	10.1016/j.bmcl.2006.06.054
Homo sapiens	HOP-62	GI50	10000.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	HOP-62	IC50	21278.41	nM	10.6019/CHEMBL1201861
Homo sapiens	HOP-92	GI50	7940.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	HOP-92	IC50	24724.98	nM	10.6019/CHEMBL1201861
Homo sapiens	Hormonally up-regulated neu tumor-associated kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	HOS	IC50	11868.34	nM	10.6019/CHEMBL1201861
Homo sapiens	HPAF-II	IC50	9225.18	nM	10.6019/CHEMBL1201861
Homo sapiens	Hs-578T	GI	20.0	%	10.1016/j.bmcl.2017.04.053
Homo sapiens	Hs-578T	GI	20.0	%	10.1039/C6MD00329J
Homo sapiens	Hs-578T	GI50	10000.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Hs-578T	IC50	27529.94	nM	10.6019/CHEMBL1201861
Homo sapiens	HSC-2	IC50	165.57	nM	10.6019/CHEMBL1201861
Homo sapiens	HSC-3	IC50	1543.8	nM	10.6019/CHEMBL1201861
Homo sapiens	HSC-4	IC50	61.53	nM	10.6019/CHEMBL1201861
Homo sapiens	HT	IC50	21433.09	nM	10.6019/CHEMBL1201861
Homo sapiens	HT-1080	IC50	33390.05	nM	10.6019/CHEMBL1201861
Homo sapiens	HT1197	IC50	40286.93	nM	10.6019/CHEMBL1201861
Homo sapiens	HT-1376	IC50	3205.06	nM	10.6019/CHEMBL1201861
Homo sapiens	HT-144	IC50	29336.22	nM	10.6019/CHEMBL1201861
Homo sapiens	HT-29	GI50	3980.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	HT-29	IC50	3360.0	nM	10.1016/j.ejmech.2012.05.039
Homo sapiens	HT-29	IC50	3630.0	nM	10.1016/j.bmc.2014.10.038
Homo sapiens	HT-29	IC50	3630.0	nM	10.1016/j.ejmech.2014.11.010
Homo sapiens	HT-29	IC50	5210.0	nM	10.1016/j.bmc.2014.10.038
Homo sapiens	HT-29	IC50	5210.0	nM	10.1016/j.ejmech.2014.11.010
Homo sapiens	HT-29	IC50	8190.0	nM	10.1016/j.bmc.2017.03.039
Homo sapiens	HT-29	IC50	8190.0	nM	10.1016/j.ejmech.2015.09.031
Homo sapiens	HT-29	IC50	9800.0	nM	10.1016/j.bmc.2009.12.048
Homo sapiens	HT-29	IC50	16930.0	nM	10.1016/j.ejmech.2010.03.001
Homo sapiens	HT-29	IC50	22882.26	nM	10.6019/CHEMBL1201861
Homo sapiens	HT-29	IC50	110300.0	nM	10.1016/j.bmc.2012.09.034
Homo sapiens	HT-29	IC50	nan	None	10.1016/j.bmcl.2011.01.137
Homo sapiens	HT-29	IC50	nan	None	10.1039/C0MD00183J
Homo sapiens	HT-3	IC50	982.41	nM	10.6019/CHEMBL1201861
Homo sapiens	HT55	IC50	15947.82	nM	10.6019/CHEMBL1201861
Homo sapiens	HTC-C3	IC50	2422.67	nM	10.6019/CHEMBL1201861
Homo sapiens	HuCCT-1	IC50	15873.98	nM	10.6019/CHEMBL1201861
Homo sapiens	Huh-7	IC50	10000.0	nM	10.1016/j.ejmech.2020.113102
Homo sapiens	Huh-7	IC50	19742.13	nM	10.6019/CHEMBL1201861
Homo sapiens	HuO-3N1	IC50	56.09	nM	10.6019/CHEMBL1201861
Homo sapiens	HuO9	IC50	22739.58	nM	10.6019/CHEMBL1201861
Homo sapiens	HuP-T3	IC50	26610.16	nM	10.6019/CHEMBL1201861
Homo sapiens	HuP-T4	IC50	2728.18	nM	10.6019/CHEMBL1201861
Homo sapiens	HuTu80	ED50	0.77	ug ml-1	10.1007/s00044-012-0309-2
Homo sapiens	HuTu80	IC50	21433.65	nM	10.6019/CHEMBL1201861
Homo sapiens	HUVEC	GI50	13000.0	nM	10.1021/acs.jmedchem.6b01774
Homo sapiens	IA-LM	IC50	9419.66	nM	10.6019/CHEMBL1201861
Homo sapiens	IGR-1	IC50	36707.5	nM	10.6019/CHEMBL1201861
Homo sapiens	IGROV-1	GI50	200.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	IGROV-1	IC50	2312.37	nM	10.6019/CHEMBL1201861
Homo sapiens	Inactive serine/threonine-protein kinase VRK3	Thermal melting change	0.6	degrees C	10.1073/pnas.0708800104
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	Ki	3981.07	nM	None
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	Ki	3162.28	nM	None
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	Ki	3162.28	nM	None
Homo sapiens	Inosine-5'-monophosphate dehydrogenase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Insulin-like growth factor I receptor	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Insulin-like growth factor I receptor	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Insulin-like growth factor I receptor	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Insulin-like growth factor I receptor	Ki	1258.93	nM	None
Homo sapiens	Insulin receptor	IC50	50000.0	nM	10.1038/nchembio.117
Homo sapiens	Insulin receptor	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Insulin receptor	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Insulin receptor	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Insulin receptor	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Insulin receptor	Ki	5011.87	nM	None
Homo sapiens	Insulin receptor-related protein	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Insulin receptor-related protein	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Interferon-induced, double-stranded RNA-activated protein kinase	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Interferon-induced, double-stranded RNA-activated protein kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Interleukin-1 receptor-associated kinase 1	Kd	69.0	nM	10.1038/nbt.1990
Homo sapiens	Interleukin-1 receptor-associated kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Interleukin-1 receptor-associated kinase 1	Ki	316.23	nM	None
Homo sapiens	Interleukin-1 receptor-associated kinase 3	Kd	1500.0	nM	10.1038/nbt1358
Homo sapiens	Interleukin-1 receptor-associated kinase 3	Kd	1500.0	nM	10.1038/nbt.1990
Homo sapiens	Interleukin-1 receptor-associated kinase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Interleukin-1 receptor-associated kinase 4	Kd	540.0	nM	10.1038/nbt.1990
Homo sapiens	Interleukin-1 receptor-associated kinase 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Interleukin-1 receptor-associated kinase 4	Ki	1000.0	nM	None
Homo sapiens	Ishikawa	EC50	nan	None	10.1021/jm500873e
Homo sapiens	Isoleucine--tRNA ligase, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	IST-MEL1	IC50	61652.64	nM	10.6019/CHEMBL1201861
Homo sapiens	IST-MES1	IC50	3940.29	nM	10.6019/CHEMBL1201861
Homo sapiens	IST-SL1	IC50	20787.86	nM	10.6019/CHEMBL1201861
Homo sapiens	J82	IC50	1457.66	nM	10.6019/CHEMBL1201861
Homo sapiens	JAR	IC50	12336.93	nM	10.6019/CHEMBL1201861
Homo sapiens	JEG-3	IC50	33097.14	nM	10.6019/CHEMBL1201861
Homo sapiens	J-RT3-T3-5	IC50	3754.06	nM	10.6019/CHEMBL1201861
Homo sapiens	JVM-2	IC50	3947.52	nM	10.6019/CHEMBL1201861
Homo sapiens	JVM-3	IC50	2346.43	nM	10.6019/CHEMBL1201861
Homo sapiens	K5	IC50	10339.51	nM	10.6019/CHEMBL1201861
Homo sapiens	K562	Activity	4.64	%	10.1016/j.ejmech.2008.01.009
Homo sapiens	K562	Activity	19.24	%	10.1016/j.ejmech.2008.01.009
Homo sapiens	K562	Activity	76.12	%	10.1016/j.ejmech.2008.01.009
Homo sapiens	K562	GI50	2510.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	K562	IC50	9360.0	nM	10.1016/j.ejmech.2008.01.009
Homo sapiens	K562	IC50	10000.0	nM	10.1021/ml4002437
Homo sapiens	K562	IC50	10839.53	nM	10.6019/CHEMBL1201861
Homo sapiens	K562	IC50	14270.0	nM	10.1016/j.ejmech.2022.114231
Homo sapiens	K562	IC50	nan	None	10.1016/j.ejmech.2013.03.013
Homo sapiens	K562/A02	IC50	32350.0	nM	10.1016/j.ejmech.2022.114231
Homo sapiens	KALS-1	IC50	13852.53	nM	10.6019/CHEMBL1201861
Homo sapiens	Kappa opioid receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	KARPAS-299	IC50	4310.13	nM	10.6019/CHEMBL1201861
Homo sapiens	KARPAS-45	IC50	2124.79	nM	10.6019/CHEMBL1201861
Homo sapiens	Kasumi 1	IC50	366.73	nM	10.6019/CHEMBL1201861
Homo sapiens	KB	ED50	0.33	ug ml-1	10.1007/s00044-012-0309-2
Homo sapiens	KB	IC50	54.0	nM	10.1016/j.ejmech.2021.113218
Homo sapiens	KB	IC50	2800.0	nM	10.1016/j.ejmech.2012.06.055
Homo sapiens	KB 3-1	IC50	80.0	nM	10.1016/s0960-894x(01)00344-4
Homo sapiens	KE-37	IC50	6072.58	nM	10.6019/CHEMBL1201861
Homo sapiens	KG-1	IC50	204.34	nM	10.6019/CHEMBL1201861
Homo sapiens	KGN	IC50	47331.12	nM	10.6019/CHEMBL1201861
Homo sapiens	KINGS-1	IC50	35843.42	nM	10.6019/CHEMBL1201861
Homo sapiens	KLE	IC50	6965.16	nM	10.6019/CHEMBL1201861
Homo sapiens	KM12	GI50	7940.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	KM12	IC50	34047.82	nM	10.6019/CHEMBL1201861
Homo sapiens	KM-H2	IC50	17941.11	nM	10.6019/CHEMBL1201861
Homo sapiens	KMOE-2	IC50	1398.15	nM	10.6019/CHEMBL1201861
Homo sapiens	KNS-42	IC50	18801.53	nM	10.6019/CHEMBL1201861
Homo sapiens	KNS-62	IC50	4908.07	nM	10.6019/CHEMBL1201861
Homo sapiens	KNS-81-FD	IC50	25902.12	nM	10.6019/CHEMBL1201861
Homo sapiens	KOSC-2	IC50	4999.59	nM	10.6019/CHEMBL1201861
Homo sapiens	KP-4	IC50	9488.38	nM	10.6019/CHEMBL1201861
Homo sapiens	KP-N-YN	IC50	5125.91	nM	10.6019/CHEMBL1201861
Homo sapiens	KP-N-YS	IC50	7181.4	nM	10.6019/CHEMBL1201861
Homo sapiens	KS-1	IC50	12283.24	nM	10.6019/CHEMBL1201861
Homo sapiens	KU-19-19	IC50	1085.41	nM	10.6019/CHEMBL1201861
Homo sapiens	KU812 cell line	IC50	2367.79	nM	10.6019/CHEMBL1201861
Homo sapiens	KURAMOCHI	IC50	3860.56	nM	10.6019/CHEMBL1201861
Homo sapiens	KY821	IC50	408.57	nM	10.6019/CHEMBL1201861
Homo sapiens	KYSE-140	IC50	209.96	nM	10.6019/CHEMBL1201861
Homo sapiens	KYSE-150 cell line	IC50	32377.31	nM	10.6019/CHEMBL1201861
Homo sapiens	KYSE-180	IC50	530.62	nM	10.6019/CHEMBL1201861
Homo sapiens	KYSE-270	IC50	498.65	nM	10.6019/CHEMBL1201861
Homo sapiens	KYSE-410	IC50	28277.88	nM	10.6019/CHEMBL1201861
Homo sapiens	KYSE-450	IC50	247.92	nM	10.6019/CHEMBL1201861
Homo sapiens	KYSE-510	IC50	2867.86	nM	10.6019/CHEMBL1201861
Homo sapiens	KYSE-520 cell line	IC50	4880.18	nM	10.6019/CHEMBL1201861
Homo sapiens	KYSE-70 cell line	IC50	8197.61	nM	10.6019/CHEMBL1201861
Homo sapiens	L02	IC50	7140.0	nM	10.1016/j.ejmech.2020.112388
Homo sapiens	L02	IC50	10080.0	nM	10.1016/j.bmcl.2021.128238
Homo sapiens	L02	IC50	13260.0	nM	10.1016/j.ejmech.2020.112737
Homo sapiens	L02	IC50	19800.0	nM	10.1021/acs.jnatprod.8b00821
Homo sapiens	L02	IC50	33170.0	nM	10.1016/j.ejmech.2021.113300
Homo sapiens	L02	IC50	45310.0	nM	10.1016/j.bmcl.2021.128503
Homo sapiens	L02	IC50	nan	None	10.1016/j.bmcl.2017.02.023
Homo sapiens	L132	ED50	1.0	ug ml-1	10.1007/s00044-012-0309-2
Homo sapiens	L-363	IC50	671.94	nM	10.6019/CHEMBL1201861
Homo sapiens	L-428	IC50	6180.37	nM	10.6019/CHEMBL1201861
Homo sapiens	LAMA-84	IC50	1538.15	nM	10.6019/CHEMBL1201861
Homo sapiens	LAN-6	IC50	14252.99	nM	10.6019/CHEMBL1201861
Homo sapiens	LB1047-RCC	IC50	625.29	nM	10.6019/CHEMBL1201861
Homo sapiens	LB2241-RCC	IC50	194.93	nM	10.6019/CHEMBL1201861
Homo sapiens	LB2518-MEL	IC50	20373.91	nM	10.6019/CHEMBL1201861
Homo sapiens	LB373-MEL-D	IC50	16723.22	nM	10.6019/CHEMBL1201861
Homo sapiens	LB771-HNC	IC50	3391.26	nM	10.6019/CHEMBL1201861
Homo sapiens	LB831-BLC	IC50	11255.61	nM	10.6019/CHEMBL1201861
Homo sapiens	LC-2-ad	IC50	36699.02	nM	10.6019/CHEMBL1201861
Homo sapiens	LCLC-103H cell line	IC50	47440.39	nM	10.6019/CHEMBL1201861
Homo sapiens	LCLC-97TM1	IC50	25728.47	nM	10.6019/CHEMBL1201861
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	Ki	2511.89	nM	None
Homo sapiens	Leukocyte tyrosine kinase receptor	Kd	5500.0	nM	10.1038/nbt.1990
Homo sapiens	Leukocyte tyrosine kinase receptor	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Leukocyte tyrosine kinase receptor	Ki	1584.89	nM	None
Homo sapiens	LIM domain kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	LIM domain kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	LIM domain kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	LIM domain kinase 1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	LIM domain kinase 1	Ki	3981.07	nM	None
Homo sapiens	LIM domain kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	LIM domain kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	LIM domain kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Liver glycogen phosphorylase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	LK-2	IC50	59570.35	nM	10.6019/CHEMBL1201861
Homo sapiens	LN-405	IC50	35430.75	nM	10.6019/CHEMBL1201861
Homo sapiens	LNCaP-Clone-FGC	IC50	24021.06	nM	10.6019/CHEMBL1201861
Homo sapiens	Long-chain-fatty-acid--CoA ligase 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	LoVo	IC50	59.0	nM	10.1021/acs.jmedchem.0c00507
Homo sapiens	LoVo	IC50	859.06	nM	10.6019/CHEMBL1201861
Homo sapiens	LoVo	Inhibition	60.0	%	10.1016/j.bmcl.2006.06.054
Homo sapiens	LoVo	Inhibition	84.0	%	10.1016/j.bmcl.2006.06.054
Homo sapiens	LOX IMVI	GI50	7940.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	LOX IMVI	IC50	13615.13	nM	10.6019/CHEMBL1201861
Homo sapiens	LS-1034	IC50	8946.52	nM	10.6019/CHEMBL1201861
Homo sapiens	LS-123	IC50	24961.36	nM	10.6019/CHEMBL1201861
Homo sapiens	LS-411N	IC50	11610.07	nM	10.6019/CHEMBL1201861
Homo sapiens	LS-513	IC50	32118.69	nM	10.6019/CHEMBL1201861
Homo sapiens	LU-134-A	IC50	719.09	nM	10.6019/CHEMBL1201861
Homo sapiens	LU-135	IC50	783.03	nM	10.6019/CHEMBL1201861
Homo sapiens	LU-139	IC50	4372.47	nM	10.6019/CHEMBL1201861
Homo sapiens	Lu-65	IC50	166.61	nM	10.6019/CHEMBL1201861
Homo sapiens	LU-99A	IC50	24184.07	nM	10.6019/CHEMBL1201861
Homo sapiens	LXF-289 cell line	IC50	10796.72	nM	10.6019/CHEMBL1201861
Homo sapiens	M059J	IC50	16283.98	nM	10.6019/CHEMBL1201861
Homo sapiens	M14	IC50	25444.74	nM	10.6019/CHEMBL1201861
Homo sapiens	Macrophage colony stimulating factor receptor	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Macrophage colony stimulating factor receptor	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Macrophage colony stimulating factor receptor	Ki	2511.89	nM	None
Homo sapiens	Macrophage colony stimulating factor receptor	Selectivity	0.0	None	10.1038/nbt1358
Homo sapiens	Macrophage-stimulating protein receptor	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Macrophage-stimulating protein receptor	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Macrophage-stimulating protein receptor	Ki	3981.07	nM	None
Homo sapiens	MAP kinase-activated protein kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase-activated protein kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase-activated protein kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase-activated protein kinase 2	Ki	7943.28	nM	None
Homo sapiens	MAP kinase-activated protein kinase 3	Ki	10000.0	nM	None
Homo sapiens	MAP kinase-activated protein kinase 5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase-activated protein kinase 5	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase-activated protein kinase 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase-activated protein kinase 5	Ki	1584.89	nM	None
Homo sapiens	MAP kinase ERK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase ERK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase ERK1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase ERK1	Thermal melting change	-0.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	MAP kinase ERK2	Delta TM	0.5667	C	None
Homo sapiens	MAP kinase ERK2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase ERK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase ERK2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase ERK2	Ki	7943.28	nM	None
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	Inhibition	46.0	%	10.1021/acs.jmedchem.6b01774
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	Inhibition	98.8	%	10.1016/j.bmc.2018.02.022
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	Kd	290.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	Kd	290.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 alpha	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase p38 alpha	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase p38 alpha	Kd	nan	None	10.1038/nbt1068
Homo sapiens	MAP kinase p38 alpha	Ki	501.19	nM	None
Homo sapiens	MAP kinase p38 beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase p38 beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase p38 beta	Kd	nan	None	10.1038/nbt1068
Homo sapiens	MAP kinase p38 beta	Thermal melting change	0.8	degrees C	10.1073/pnas.0708800104
Homo sapiens	MAP kinase p38 delta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 delta	Ki	7943.28	nM	None
Homo sapiens	MAP kinase p38 gamma	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase p38 gamma	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 gamma	Kd	nan	None	10.1038/nbt1068
Homo sapiens	MAP kinase p38 gamma	Ki	6309.57	nM	None
Homo sapiens	MAP kinase signal-integrating kinase 2	Inhibition	46.0	%	10.1021/acs.jmedchem.6b01774
Homo sapiens	MAP kinase signal-integrating kinase 2	Kd	360.0	nM	10.1038/nbt1068
Homo sapiens	MAP kinase signal-integrating kinase 2	Kd	1200.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase signal-integrating kinase 2	Kd	1200.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase signal-integrating kinase 2	Ki	398.11	nM	None
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Ki	7943.28	nM	None
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	Ki	5011.87	nM	None
Homo sapiens	Maternal embryonic leucine zipper kinase	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Maternal embryonic leucine zipper kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Maternal embryonic leucine zipper kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Maternal embryonic leucine zipper kinase	Ki	1584.89	nM	None
Homo sapiens	MC116	IC50	21072.33	nM	10.6019/CHEMBL1201861
Homo sapiens	MCF-10A	IC50	nan	None	10.1016/j.bmcl.2019.08.022
Homo sapiens	MCF7	Activity	16.2	%	10.1016/j.bmcl.2016.12.006
Homo sapiens	MCF7	Activity	30.0	%	10.1016/j.bmcl.2011.01.137
Homo sapiens	MCF7	Activity	70.3	%	10.1016/j.bmcl.2018.11.010
Homo sapiens	MCF7	Activity	72.6	%	10.1016/j.bmcl.2016.12.006
Homo sapiens	MCF7	Activity	73.1	%	10.1016/j.bmcl.2016.12.006
Homo sapiens	MCF7	Activity	89.7	%	10.1016/j.bmcl.2016.12.006
Homo sapiens	MCF7	Activity	nan	None	10.1016/j.ejmech.2011.10.051
Homo sapiens	MCF7	EC50	35000.0	nM	10.1021/jm500873e
Homo sapiens	MCF7	EC50	50000.0	nM	10.1021/jm500873e
Homo sapiens	MCF7	ED50	0.89	ug ml-1	10.1007/s00044-012-0309-2
Homo sapiens	MCF7	GI50	6710.0	nM	10.1016/j.bmc.2016.08.002
Homo sapiens	MCF7	GI50	10000.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	MCF7	GI50	20800.0	nM	10.1016/j.bmcl.2016.12.006
Homo sapiens	MCF7	GI50	30000.0	nM	10.1016/j.bmcl.2018.11.010
Homo sapiens	MCF7	IC50	1000.0	nM	10.1016/j.ejmech.2008.07.023
Homo sapiens	MCF7	IC50	2970.0	nM	10.1016/j.bmcl.2019.08.022
Homo sapiens	MCF7	IC50	3300.0	nM	10.1016/j.bmcl.2015.06.076
Homo sapiens	MCF7	IC50	3300.0	nM	10.1016/j.ejmech.2020.113102
Homo sapiens	MCF7	IC50	3570.0	nM	10.1016/j.bmcl.2021.127987
Homo sapiens	MCF7	IC50	6260.0	nM	10.1016/j.ejmech.2018.11.059
Homo sapiens	MCF7	IC50	6710.0	nM	10.1016/j.bmcl.2015.08.026
Homo sapiens	MCF7	IC50	6770.0	nM	10.1016/j.bmcl.2018.05.004
Homo sapiens	MCF7	IC50	7340.0	nM	10.1016/j.ejmech.2019.03.030
Homo sapiens	MCF7	IC50	10290.0	nM	10.1016/j.bmcl.2015.03.022
Homo sapiens	MCF7	IC50	12050.0	nM	10.1016/j.ejmech.2011.11.015
Homo sapiens	MCF7	IC50	12050.0	nM	10.1016/j.ejmech.2017.07.005
Homo sapiens	MCF7	IC50	13100.0	nM	10.1016/j.ejmech.2016.01.045
Homo sapiens	MCF7	IC50	13240.0	nM	10.1016/j.bmcl.2021.128503
Homo sapiens	MCF7	IC50	15814.5	nM	10.6019/CHEMBL1201861
Homo sapiens	MCF7	IC50	17830.0	nM	10.1016/j.bmcl.2015.08.076
Homo sapiens	MCF7	IC50	20680.0	nM	10.1016/j.bmc.2019.02.044
Homo sapiens	MCF7	IC50	23520.0	nM	10.1016/j.bmc.2019.02.044
Homo sapiens	MCF7	IC50	25370.0	nM	10.1016/j.ejmech.2016.04.026
Homo sapiens	MCF7	IC50	26700.0	nM	10.1016/j.ejmech.2018.01.081
Homo sapiens	MCF7	IC50	69160.0	nM	10.1016/j.ejmech.2010.03.001
Homo sapiens	MCF7	IC50	100000.0	nM	10.1016/j.bmc.2019.06.001
Homo sapiens	MCF7	IC50	nan	None	10.1016/j.ejmech.2013.06.055
Homo sapiens	MCF7	Inhibition	30.0	%	10.1039/C0MD00183J
Homo sapiens	MC-IXC	IC50	2644.53	nM	10.6019/CHEMBL1201861
Homo sapiens	MDA-MB-157	IC50	34819.34	nM	10.6019/CHEMBL1201861
Homo sapiens	MDA-MB-175-VII	IC50	378.88	nM	10.6019/CHEMBL1201861
Homo sapiens	MDA-MB-231	Activity	nan	None	10.1021/acs.jmedchem.6b01489
Homo sapiens	MDA-MB-231	EC50	25000.0	nM	10.1021/jm500873e
Homo sapiens	MDA-MB-231	EC50	50000.0	nM	10.1021/jm500873e
Homo sapiens	MDA-MB-231	GI50	12600.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	MDA-MB-231	GI50	14200.0	nM	10.1021/acs.jmedchem.6b01774
Homo sapiens	MDA-MB-231	GI50	15000.0	nM	10.1021/acs.jmedchem.6b01774
Homo sapiens	MDA-MB-231	IC50	4100.0	nM	10.1016/j.bmcl.2015.06.076
Homo sapiens	MDA-MB-231	IC50	4100.0	nM	10.1016/j.ejmech.2020.113102
Homo sapiens	MDA-MB-231	IC50	6850.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	MDA-MB-231	IC50	7120.0	nM	10.1016/j.bmc.2021.116265
Homo sapiens	MDA-MB-231	IC50	8720.0	nM	10.1016/j.ejmech.2019.03.030
Homo sapiens	MDA-MB-231	IC50	10000.0	nM	10.1021/jm301365e
Homo sapiens	MDA-MB-231	IC50	14520.0	nM	10.1016/j.bmcl.2021.128503
Homo sapiens	MDA-MB-231	IC50	28300.0	nM	10.1016/j.ejmech.2018.03.076
Homo sapiens	MDA-MB-231	IC50	35505.41	nM	10.6019/CHEMBL1201861
Homo sapiens	MDA-MB-231	IC50	36610.0	nM	10.1016/j.ejmech.2008.01.009
Homo sapiens	MDA-MB-231	IC50	37820.0	nM	10.1016/j.ejmech.2016.04.026
Homo sapiens	MDA-MB-231	Selectivity ratio	1700.0	None	10.1021/ml400162g
Homo sapiens	MDA-MB-231	TGI	nan	None	10.1021/acs.jmedchem.6b01774
Homo sapiens	MDA-MB-361	IC50	18558.78	nM	10.6019/CHEMBL1201861
Homo sapiens	MDA-MB-415	IC50	31175.33	nM	10.6019/CHEMBL1201861
Homo sapiens	MDA-MB-453	IC50	52768.69	nM	10.6019/CHEMBL1201861
Homo sapiens	MDA-MB-468	Activity	6.7	%	10.1016/j.bmcl.2016.12.006
Homo sapiens	MDA-MB-468	Activity	49.1	%	10.1016/j.bmcl.2016.12.006
Homo sapiens	MDA-MB-468	Activity	60.3	%	10.1016/j.bmcl.2018.11.010
Homo sapiens	MDA-MB-468	Activity	nan	None	10.1016/j.ejmech.2011.02.057
Homo sapiens	MDA-MB-468	GI50	10.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	MDA-MB-468	GI50	9700.0	nM	10.1016/j.bmcl.2016.12.006
Homo sapiens	MDA-MB-468	GI50	25500.0	nM	10.1016/j.bmcl.2018.11.010
Homo sapiens	MDA-MB-468	IC50	3900.0	nM	10.1016/j.bmcl.2015.06.076
Homo sapiens	MDA-MB-468	IC50	3900.0	nM	10.1016/j.ejmech.2020.113102
Homo sapiens	MDA-MB-468	Inhibition	nan	%	10.1016/j.bmcl.2016.12.006
Homo sapiens	ME-180	IC50	632.9	nM	10.6019/CHEMBL1201861
Homo sapiens	MEG-01	IC50	276.76	nM	10.6019/CHEMBL1201861
Homo sapiens	Melanocortin receptor 3	AC50	25999.8	nM	10.1038/s41467-023-40064-9
Homo sapiens	MEL-HO	IC50	16885.44	nM	10.6019/CHEMBL1201861
Homo sapiens	MEL-JUSO	IC50	50579.08	nM	10.6019/CHEMBL1201861
Homo sapiens	MeWo	IC50	6114.87	nM	10.6019/CHEMBL1201861
Homo sapiens	MFE-280	IC50	18729.35	nM	10.6019/CHEMBL1201861
Homo sapiens	MFH-ino	IC50	18966.87	nM	10.6019/CHEMBL1201861
Homo sapiens	MFM-223	IC50	38943.08	nM	10.6019/CHEMBL1201861
Homo sapiens	MG-63	IC50	30847.76	nM	10.6019/CHEMBL1201861
Homo sapiens	MGC-803	IC50	8190.0	nM	10.1016/j.bmc.2021.116265
Homo sapiens	MGC-803	IC50	8820.0	nM	10.1016/j.ejmech.2019.03.030
Homo sapiens	MGC-803	IC50	26190.0	nM	10.1016/j.ejmech.2020.112661
Homo sapiens	MHH-ES-1	IC50	56575.27	nM	10.6019/CHEMBL1201861
Homo sapiens	MHH-NB-11	IC50	27800.69	nM	10.6019/CHEMBL1201861
Homo sapiens	MHH-PREB-1	IC50	1084.51	nM	10.6019/CHEMBL1201861
Homo sapiens	MIA PaCa-2	Activity	nan	None	10.1016/j.bmc.2010.04.046
Homo sapiens	MIA PaCa-2	ED50	0.51	ug ml-1	10.1007/s00044-012-0309-2
Homo sapiens	MIA PaCa-2	IC50	14968.96	nM	10.6019/CHEMBL1201861
Homo sapiens	MIA PaCa-2	IC50	45800.0	nM	10.1016/j.bmc.2010.04.046
Homo sapiens	MIA PaCa-2	Inhibition	nan	%	10.1016/j.bmc.2010.04.046
Homo sapiens	Microtubule-associated protein tau	Potency	25118.9	nM	None
Homo sapiens	Microtubule-associated protein tau	Potency	35481.3	nM	None
Homo sapiens	Microtubule-associated protein tau	Potency	39810.7	nM	None
Homo sapiens	Microtubule-associated serine/threonine-protein kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Midasin	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Misshapen-like kinase 1	IC50	15000.0	nM	None
Homo sapiens	Misshapen-like kinase 1	Kd	1800.0	nM	10.1038/nbt.1990
Homo sapiens	Misshapen-like kinase 1	Ki	5011.87	nM	None
Homo sapiens	Mitogen-activated protein kinase 15	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase 15	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase 15	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase 4	Kd	3100.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase 4	Kd	3100.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase 6	Kd	1600.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase 6	Kd	1600.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase 6	Thermal melting change	0.8	degrees C	10.1073/pnas.0708800104
Homo sapiens	Mitogen-activated protein kinase 7	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase 7	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase 7	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 10	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 10	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 10	Ki	3162.28	nM	None
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 12	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 13	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 15	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 2	Kd	3300.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 3	Kd	2100.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 4	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Thermal melting change	0.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	Mitogen-activated protein kinase kinase kinase 6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 2	Ki	5011.87	nM	None
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	Ki	1000.0	nM	None
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Ki	1584.89	nM	None
Homo sapiens	Mitotic checkpoint serine/threonine-protein kinase BUB1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mixed lineage kinase 7	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mixed lineage kinase 7	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mixed lineage kinase 7	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mixed lineage kinase 7	Ki	7943.28	nM	None
Homo sapiens	MKN-1	IC50	1219.87	nM	10.6019/CHEMBL1201861
Homo sapiens	MKN-28	IC50	35823.6	nM	10.6019/CHEMBL1201861
Homo sapiens	MKN-45	IC50	12290.0	nM	10.1016/j.bmc.2018.02.023
Homo sapiens	MKN-45	IC50	25631.5	nM	10.6019/CHEMBL1201861
Homo sapiens	MKN-7	IC50	2627.48	nM	10.6019/CHEMBL1201861
Homo sapiens	ML-2	IC50	1640.29	nM	10.6019/CHEMBL1201861
Homo sapiens	MLMA	IC50	11699.71	nM	10.6019/CHEMBL1201861
Homo sapiens	MMAC-SF	IC50	11725.18	nM	10.6019/CHEMBL1201861
Homo sapiens	MN-60	IC50	3049.74	nM	10.6019/CHEMBL1201861
Homo sapiens	Mo	IC50	11954.06	nM	10.6019/CHEMBL1201861
Homo sapiens	MOLT-13	IC50	514.82	nM	10.6019/CHEMBL1201861
Homo sapiens	MOLT-16	IC50	26616.6	nM	10.6019/CHEMBL1201861
Homo sapiens	MOLT-4	ED50	1.0	ug ml-1	10.1007/s00044-012-0309-2
Homo sapiens	MOLT-4	GI50	3980.0	nM	10.1016/j.bmcl.2019.04.029
Homo sapiens	MOLT-4	IC50	15020.0	nM	10.1016/j.ejmech.2008.01.009
Homo sapiens	MOLT-4	IC50	15049.71	nM	10.6019/CHEMBL1201861
Homo sapiens	Monoamine oxidase A	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Motilin receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	MPP-89	IC50	15941.66	nM	10.6019/CHEMBL1201861
Homo sapiens	MS-1	IC50	994.69	nM	10.6019/CHEMBL1201861
Homo sapiens	MSTO-211H	IC50	6511.7	nM	10.6019/CHEMBL1201861
Homo sapiens	Multidrug resistance-associated protein 4	IC50	4600.0	nM	10.1093/toxsci/kft176
Homo sapiens	Multifunctional protein ADE2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mu opioid receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Muscarinic acetylcholine receptor M1	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Muscarinic acetylcholine receptor M2	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Muscarinic acetylcholine receptor M3	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Muscle, skeletal receptor tyrosine protein kinase	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Muscle, skeletal receptor tyrosine protein kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MV4-11	Activity	7.0	%	10.1016/j.ejmech.2011.07.045
Homo sapiens	MV4-11	Activity	92.4	%	10.1016/j.ejmech.2011.07.045
Homo sapiens	MV4-11	IC50	627.7	nM	10.6019/CHEMBL1201861
Homo sapiens	Myelin transcription factor 1	Activity	5.0	%	10.1016/j.ejmech.2012.06.007
Homo sapiens	Myelin transcription factor 1	Activity	6.85	%	10.1016/j.ejmech.2012.06.007
Homo sapiens	Myelin transcription factor 1	IC50	nan	None	10.1016/j.ejmech.2012.06.007
Homo sapiens	Myosin-14	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Myosin IIIA	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Myosin IIIA	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin-IIIB	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Myosin-IIIB	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin light chain kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	myosin light chain kinase 2	Kd	1900.0	nM	10.1038/nbt1358
Homo sapiens	myosin light chain kinase 2	Kd	1900.0	nM	10.1038/nbt.1990
Homo sapiens	myosin light chain kinase 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Myosin light chain kinase family member 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Myosin light chain kinase family member 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin light chain kinase, smooth muscle	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Myosin light chain kinase, smooth muscle	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin light chain kinase, smooth muscle	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Myotonin-protein kinase	Kd	6900.0	nM	10.1038/nbt1358
Homo sapiens	Myotonin-protein kinase	Kd	6900.0	nM	10.1038/nbt.1990
Homo sapiens	Myotonin-protein kinase	Thermal melting change	3.6	degrees C	10.1073/pnas.0708800104
Homo sapiens	MZ1-PC	IC50	41809.98	nM	10.6019/CHEMBL1201861
Homo sapiens	MZ2-MEL	IC50	17132.98	nM	10.6019/CHEMBL1201861
Homo sapiens	MZ7-mel	IC50	39119.89	nM	10.6019/CHEMBL1201861
Homo sapiens	NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	NB10	IC50	4597.81	nM	10.6019/CHEMBL1201861
Homo sapiens	NB12	IC50	6784.04	nM	10.6019/CHEMBL1201861
Homo sapiens	NB13	IC50	7826.67	nM	10.6019/CHEMBL1201861
Homo sapiens	NB14	IC50	38454.36	nM	10.6019/CHEMBL1201861
Homo sapiens	NB17	IC50	58429.33	nM	10.6019/CHEMBL1201861
Homo sapiens	NB5	IC50	1408.94	nM	10.6019/CHEMBL1201861
Homo sapiens	NB6	IC50	64999.85	nM	10.6019/CHEMBL1201861
Homo sapiens	NB69	IC50	614.35	nM	10.6019/CHEMBL1201861
Homo sapiens	NB7	IC50	546.32	nM	10.6019/CHEMBL1201861
Homo sapiens	NBsusSR	IC50	646.52	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1048	IC50	19232.64	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1092	IC50	1308.5	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1155	IC50	3841.59	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1299	Activity	nan	None	10.1021/acs.jmedchem.2c00345
Homo sapiens	NCI-H1299	IC50	3020.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	NCI-H1299	IC50	4050.0	nM	10.1016/j.ejmech.2021.113984
Homo sapiens	NCI-H1299	IC50	6560.0	nM	10.1021/acs.jmedchem.1c00649
Homo sapiens	NCI-H1299	IC50	11664.69	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1299	IC50	40000.0	nM	10.1016/j.ejmech.2022.114502
Homo sapiens	NCI-H1304	IC50	1016.43	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1355	IC50	9940.88	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1395	IC50	31232.84	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1437	IC50	19046.74	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1563	IC50	18712.39	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1573	IC50	17282.56	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1581	IC50	17441.13	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1623	IC50	599.36	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1648	IC50	1106.16	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1650	Activity	83.0	%	10.1016/j.ejmech.2020.112359
Homo sapiens	NCI-H1650	IC50	1334.82	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1650	IC50	2640.0	nM	10.1016/j.bmcl.2021.128503
Homo sapiens	NCI-H1651	IC50	33395.96	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1666	IC50	1747.04	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1693	IC50	2958.97	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1703	IC50	48335.2	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1755	IC50	14995.33	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1770	IC50	722.4	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1792	IC50	8889.03	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1793	IC50	3210.98	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1838	IC50	5020.76	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1975	Activity	0.61	%	10.1016/j.ejmech.2021.113300
Homo sapiens	NCI-H1975	Activity	5.44	%	10.1016/j.ejmech.2021.113300
Homo sapiens	NCI-H1975	Activity	7.78	%	10.1016/j.ejmech.2021.113300
Homo sapiens	NCI-H1975	Activity	18.7	%	10.1016/j.bmc.2018.11.009
Homo sapiens	NCI-H1975	Activity	18.76	%	10.1016/j.ejmech.2021.113300
Homo sapiens	NCI-H1975	Activity	32.7	%	10.1016/j.bmc.2018.11.009
Homo sapiens	NCI-H1975	Activity	33.72	%	10.1016/j.ejmech.2021.113300
Homo sapiens	NCI-H1975	Activity	47.52	%	10.1016/j.ejmech.2021.113300
Homo sapiens	NCI-H1975	Activity	48.7	%	10.1016/j.bmc.2018.11.009
Homo sapiens	NCI-H1975	Activity	55.0	%	10.1016/j.ejmech.2020.112359
Homo sapiens	NCI-H1975	Activity	63.2	%	10.1016/j.bmc.2018.11.009
Homo sapiens	NCI-H1975	Activity	84.3	%	10.1016/j.bmc.2018.11.009
Homo sapiens	NCI-H1975	Activity	86.2	%	10.1016/j.ejmech.2021.113300
Homo sapiens	NCI-H1975	Activity	89.9	%	10.1016/j.bmc.2018.11.009
Homo sapiens	NCI-H1975	Activity	90.6	%	10.1016/j.bmc.2018.11.009
Homo sapiens	NCI-H1975	Activity	93.5	%	10.1016/j.bmc.2018.11.009
Homo sapiens	NCI-H1975	Activity	97.6	%	10.1016/j.bmc.2018.11.009
Homo sapiens	NCI-H1975	Activity	nan	None	10.1016/j.bmcl.2017.02.023
Homo sapiens	NCI-H1975	Activity	nan	None	10.1016/j.ejmech.2013.05.026
Homo sapiens	NCI-H1975	Activity	nan	None	10.1016/j.ejmech.2014.02.032
Homo sapiens	NCI-H1975	Activity	nan	None	10.1016/j.ejmech.2020.113022
Homo sapiens	NCI-H1975	Activity	nan	None	10.1021/jm901558p
Homo sapiens	NCI-H1975	CC50	18755.0	nM	10.1021/acs.jmedchem.9b00722
Homo sapiens	NCI-H1975	EC50	10700.0	nM	10.1021/acs.jmedchem.7b00515
Homo sapiens	NCI-H1975	EC50	11000.0	nM	10.1021/acs.jmedchem.7b00316
Homo sapiens	NCI-H1975	IC50	1230.0	nM	10.1016/j.bmcl.2016.04.032
Homo sapiens	NCI-H1975	IC50	1710.0	nM	10.1016/j.ejmech.2021.113984
Homo sapiens	NCI-H1975	IC50	3102.0	nM	10.1021/acs.jmedchem.0c00507
Homo sapiens	NCI-H1975	IC50	4691.0	nM	10.1016/j.ejmech.2017.03.083
Homo sapiens	NCI-H1975	IC50	4810.0	nM	10.1016/j.ejmech.2020.112185
Homo sapiens	NCI-H1975	IC50	6500.0	nM	10.1016/j.ejmech.2019.111867
Homo sapiens	NCI-H1975	IC50	6917.0	nM	10.1016/j.ejmech.2014.02.032
Homo sapiens	NCI-H1975	IC50	6917.0	nM	10.1021/jm400463q
Homo sapiens	NCI-H1975	IC50	7184.0	nM	10.1016/j.bmc.2018.02.022
Homo sapiens	NCI-H1975	IC50	8260.0	nM	10.1021/jm901558p
Homo sapiens	NCI-H1975	IC50	8580.0	nM	10.1016/j.bmc.2018.02.023
Homo sapiens	NCI-H1975	IC50	8589.0	nM	10.1016/j.ejmech.2013.05.026
Homo sapiens	NCI-H1975	IC50	8710.0	nM	10.1016/j.bmc.2017.03.039
Homo sapiens	NCI-H1975	IC50	8710.0	nM	10.1016/j.ejmech.2015.09.031
Homo sapiens	NCI-H1975	IC50	9020.0	nM	10.1021/jm201591k
Homo sapiens	NCI-H1975	IC50	9100.0	nM	10.1016/j.ejmech.2018.11.029
Homo sapiens	NCI-H1975	IC50	9200.0	nM	10.1016/j.bmc.2021.116265
Homo sapiens	NCI-H1975	IC50	10000.0	nM	10.1016/j.bmc.2018.03.025
Homo sapiens	NCI-H1975	IC50	10000.0	nM	10.1016/j.bmcl.2013.12.079
Homo sapiens	NCI-H1975	IC50	10000.0	nM	10.1016/j.bmcl.2016.08.007
Homo sapiens	NCI-H1975	IC50	10000.0	nM	10.1016/j.bmcl.2018.12.020
Homo sapiens	NCI-H1975	IC50	10000.0	nM	10.1016/j.bmcl.2020.127045
Homo sapiens	NCI-H1975	IC50	10000.0	nM	10.1016/j.ejmech.2019.111607
Homo sapiens	NCI-H1975	IC50	10000.0	nM	10.1021/acs.jnatprod.9b00659
Homo sapiens	NCI-H1975	IC50	10000.0	nM	10.1021/jm301365e
Homo sapiens	NCI-H1975	IC50	10000.0	nM	10.1021/jm5014659
Homo sapiens	NCI-H1975	IC50	10780.0	nM	10.1016/j.ejmech.2021.113300
Homo sapiens	NCI-H1975	IC50	10890.0	nM	10.1016/j.bmc.2018.11.009
Homo sapiens	NCI-H1975	IC50	10890.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	NCI-H1975	IC50	11390.0	nM	10.1039/C3MD00118K
Homo sapiens	NCI-H1975	IC50	12700.0	nM	10.1016/j.ejmech.2017.06.023
Homo sapiens	NCI-H1975	IC50	12700.0	nM	10.1016/j.ejmech.2018.01.090
Homo sapiens	NCI-H1975	IC50	12700.0	nM	10.1016/j.ejmech.2019.06.015
Homo sapiens	NCI-H1975	IC50	13130.0	nM	10.1016/j.bmc.2017.03.032
Homo sapiens	NCI-H1975	IC50	13613.0	nM	10.1021/jm401045n
Homo sapiens	NCI-H1975	IC50	14380.0	nM	10.1016/j.bmc.2016.04.046
Homo sapiens	NCI-H1975	IC50	14707.0	nM	10.1016/j.bmc.2015.04.055
Homo sapiens	NCI-H1975	IC50	15350.0	nM	10.1016/j.bmcl.2017.02.023
Homo sapiens	NCI-H1975	IC50	17790.0	nM	10.1016/j.ejmech.2020.112388
Homo sapiens	NCI-H1975	IC50	18190.0	nM	10.1039/C2MD20078C
Homo sapiens	NCI-H1975	IC50	21461.01	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1975	IC50	26900.0	nM	10.1016/j.ejmech.2016.01.045
Homo sapiens	NCI-H1975	IC50	44600.0	nM	10.1016/j.ejmech.2019.111966
Homo sapiens	NCI-H1975	IC50	78700.0	nM	10.1016/j.ejmech.2019.111867
Homo sapiens	NCI-H1975	IC50	nan	None	10.1016/j.ejmech.2019.111888
Homo sapiens	NCI-H1975	IG50	12.7	uM	10.1016/j.bmcl.2017.02.027
Homo sapiens	NCI-H1975	Ratio IC50	446.0	None	10.1016/j.bmc.2015.04.055
Homo sapiens	NCI-H1975	TGI	8.0	%	10.1021/acsmedchemlett.6b00058
Homo sapiens	NCI-H1975	TGI	8.0	%	10.1021/jm400822z
Homo sapiens	NCI-H1975	TGI	8.0	%	10.1021/jm500973a
Homo sapiens	NCI-H1975	TGI	23.0	%	10.1021/jm301365e
Homo sapiens	NCI-H1975	TGI	27.0	%	10.1016/j.ejmech.2019.111607
Homo sapiens	NCI-H1975	TGI	nan	None	10.1021/jm400463q
Homo sapiens	NCI-H1993	IC50	100.0	nM	10.1021/np2003512
Homo sapiens	NCI-H1993	IC50	13428.51	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1993	IC50	20000.0	nM	10.1021/np2003512
Homo sapiens	NCI-H2009	IC50	2062.14	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2029	IC50	31776.5	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2030	IC50	7336.98	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2052	IC50	45902.7	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2087	IC50	59083.16	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H209	IC50	1772.69	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2122	IC50	33557.45	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2126	IC50	882.83	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2170	IC50	2347.83	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2228	IC50	9110.81	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H226	GI50	15900.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	NCI-H226	IC50	9090.0	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2291	IC50	34247.21	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H23	GI50	15900.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	NCI-H23	IC50	1020.0	nM	10.1016/j.bmcl.2017.10.060
Homo sapiens	NCI-H23	IC50	15843.84	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2342	IC50	10015.47	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2347	IC50	21942.8	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2405	IC50	7083.93	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2452	IC50	34788.23	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H28	IC50	3829.61	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H292	IC50	20.0	nM	10.1021/np2003512
Homo sapiens	NCI-H292	IC50	120.0	nM	10.1021/jm301365e
Homo sapiens	NCI-H292	IC50	162.66	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H292	IC50	190.0	nM	10.1021/np500385b
Homo sapiens	NCI-H292	IC50	410.0	nM	10.1021/np2003512
Homo sapiens	NCI-H322M	GI50	80.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	NCI-H322M	GI50	80.0	nM	10.1016/j.bmcl.2019.04.029
Homo sapiens	NCI-H3255	Activity	nan	None	10.1021/acs.jmedchem.9b01566
Homo sapiens	NCI-H3255	IC50	863.0	nM	10.1021/acs.jmedchem.2c00272
Homo sapiens	NCI-H358	IC50	527.66	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H358	IC50	5680.0	nM	10.1016/j.bmc.2016.01.003
Homo sapiens	NCI-H358	IC50	14660.0	nM	10.1016/j.bmcl.2016.02.009
Homo sapiens	NCI-H441	IC50	3970.14	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H446	IC50	19358.91	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H460	GI50	6310.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	NCI-H460	GI50	6310.0	nM	10.1016/j.bmcl.2019.04.029
Homo sapiens	NCI-H460	IC50	3020.0	nM	10.1016/j.bmcl.2021.128503
Homo sapiens	NCI-H460	IC50	5590.0	nM	10.1016/j.ejmech.2012.05.039
Homo sapiens	NCI-H460	IC50	7600.0	nM	10.1021/np500382k
Homo sapiens	NCI-H460	IC50	57750.73	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H460	Inhibition	19.9	%	10.1016/j.bmc.2018.08.009
Homo sapiens	NCI-H460	Inhibition	22.6	%	10.1016/j.bmc.2018.08.009
Homo sapiens	NCI-H460	Inhibition	41.4	%	10.1016/j.bmc.2018.08.009
Homo sapiens	NCI-H460	Inhibition	44.2	%	10.1016/j.bmc.2018.08.009
Homo sapiens	NCI-H460	Inhibition	47.7	%	10.1016/j.bmc.2018.08.009
Homo sapiens	NCI-H460	Inhibition	51.3	%	10.1016/j.bmc.2018.08.009
Homo sapiens	NCI-H510A	IC50	38645.06	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H520	IC50	32448.17	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H522	GI50	6310.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	NCI-H526	IC50	1438.26	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H596	IC50	26048.73	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H630	IC50	14946.72	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H650	IC50	19750.84	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H661	IC50	8058.67	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H661	IC50	31060.0	nM	10.1016/j.bmc.2010.04.046
Homo sapiens	NCI-H661	IC50	nan	None	10.1016/j.ejmech.2013.03.013
Homo sapiens	NCI-H69	IC50	3901.78	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H720	IC50	26.92	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H727	IC50	3385.84	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H747	IC50	17529.72	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H810	IC50	10159.68	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H82	IC50	540.5	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-N87	IC50	1000.0	nM	10.1016/j.bmcl.2013.12.079
Homo sapiens	NCI-N87	IC50	1000.0	nM	10.1016/j.bmcl.2016.08.007
Homo sapiens	NCI-N87	IC50	1000.0	nM	10.1016/j.bmcl.2020.127045
Homo sapiens	NCI-N87	IC50	19599.24	nM	10.6019/CHEMBL1201861
Homo sapiens	NEC8	IC50	22507.78	nM	10.6019/CHEMBL1201861
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Nerve growth factor receptor Trk-A	Ki	2511.89	nM	None
Homo sapiens	Neuronal acetylcholine receptor protein alpha-4 subunit	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Neuropeptide Y receptor type 1	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	Ki	3981.07	nM	None
Homo sapiens	NH-12	IC50	3941.87	nM	10.6019/CHEMBL1201861
Homo sapiens	NKM-1	IC50	1325.97	nM	10.6019/CHEMBL1201861
Homo sapiens	NMC-G1	IC50	38722.2	nM	10.6019/CHEMBL1201861
Homo sapiens	no-10	IC50	53282.5	nM	10.6019/CHEMBL1201861
Homo sapiens	no-11	IC50	15966.25	nM	10.6019/CHEMBL1201861
Homo sapiens	NOMO-1	IC50	5231.76	nM	10.6019/CHEMBL1201861
Homo sapiens	Non-receptor tyrosine-protein kinase TNK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Non-receptor tyrosine-protein kinase TNK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Non-receptor tyrosine-protein kinase TNK1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Norepinephrine transporter	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	NOS-1	IC50	7258.28	nM	10.6019/CHEMBL1201861
Homo sapiens	NT-3 growth factor receptor	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	NT-3 growth factor receptor	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	NT-3 growth factor receptor	Ki	1258.93	nM	None
Homo sapiens	NTERA-2-cl-D1	IC50	3449.57	nM	10.6019/CHEMBL1201861
Homo sapiens	NUAK family SNF1-like kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	NUAK family SNF1-like kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	NUAK family SNF1-like kinase 2	Kd	4600.0	nM	10.1038/nbt.1990
Homo sapiens	NUAK family SNF1-like kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	NUAK family SNF1-like kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Nuclear factor NF-kappa-B p65 subunit	IC50	55.0	nM	10.1016/j.ejmech.2020.112062
Homo sapiens	Nuclear factor NF-kappa-B p65 subunit	Inhibition	nan	%	10.1021/acs.jmedchem.6b01774
Homo sapiens	Nucleolar GTP-binding protein 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	NUGC-3	IC50	401.81	nM	10.6019/CHEMBL1201861
Homo sapiens	NY	IC50	2372.7	nM	10.6019/CHEMBL1201861
Homo sapiens	OAW-28	IC50	3594.26	nM	10.6019/CHEMBL1201861
Homo sapiens	OAW-42	IC50	1278.25	nM	10.6019/CHEMBL1201861
Homo sapiens	Obg-like ATPase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	OC-314	IC50	22884.48	nM	10.6019/CHEMBL1201861
Homo sapiens	OCI-AML2	IC50	9869.6	nM	10.6019/CHEMBL1201861
Homo sapiens	OCUB-M	IC50	25445.6	nM	10.6019/CHEMBL1201861
Homo sapiens	OE19	IC50	11936.73	nM	10.6019/CHEMBL1201861
Homo sapiens	OE33	IC50	21604.62	nM	10.6019/CHEMBL1201861
Homo sapiens	OMC-1	IC50	1998.88	nM	10.6019/CHEMBL1201861
Homo sapiens	ONS-76	IC50	37130.92	nM	10.6019/CHEMBL1201861
Homo sapiens	OS-RC-2	IC50	7498.94	nM	10.6019/CHEMBL1201861
Homo sapiens	OVCAR-3	GI50	5010.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	OVCAR-3	IC50	2855.94	nM	10.6019/CHEMBL1201861
Homo sapiens	OVCAR-4	GI50	7940.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	OVCAR-4	IC50	7153.5	nM	10.6019/CHEMBL1201861
Homo sapiens	OVCAR-5	IC50	34218.21	nM	10.6019/CHEMBL1201861
Homo sapiens	OVCAR-8	Activity	nan	None	10.1021/acs.jmedchem.2c00345
Homo sapiens	OVCAR-8	GI50	10000.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	OVCAR-8	IC50	18927.56	nM	10.6019/CHEMBL1201861
Homo sapiens	P12-Ichikawa	IC50	328.06	nM	10.6019/CHEMBL1201861
Homo sapiens	P30-OHK	IC50	4819.29	nM	10.6019/CHEMBL1201861
Homo sapiens	PA-1	IC50	21278.73	nM	10.6019/CHEMBL1201861
Homo sapiens	PANC-03-27	IC50	1701.39	nM	10.6019/CHEMBL1201861
Homo sapiens	PANC-08-13	IC50	22011.9	nM	10.6019/CHEMBL1201861
Homo sapiens	PANC-1	IC50	40420.0	nM	10.1016/j.bmc.2010.04.046
Homo sapiens	PANC-1	IC50	69320.0	nM	10.1016/j.ejmech.2010.03.001
Homo sapiens	PANC-1	INH	11.3	uM	10.1021/acsmedchemlett.0c00159
Homo sapiens	Panc1005	IC50	3720.72	nM	10.6019/CHEMBL1201861
Homo sapiens	Panel breast (Carcinoma cell lines)	GI50	7810.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel breast (Carcinoma cell lines)	LC50	63100.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel breast (Carcinoma cell lines)	TGI	25100.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel CNS (Carcinoma cell lines)	GI50	8140.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel CNS (Carcinoma cell lines)	LC50	39800.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel CNS (Carcinoma cell lines)	TGI	20000.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel colon (Carcinoma cell lines)	GI50	7020.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel colon (Carcinoma cell lines)	LC50	63100.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel colon (Carcinoma cell lines)	TGI	31600.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel leukemia (Carcinoma cell lines)	GI50	3540.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel leukemia (Carcinoma cell lines)	LC50	31600.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel leukemia (Carcinoma cell lines)	TGI	12600.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel melanoma (Carcinoma cell lines)	GI50	5280.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel melanoma (Carcinoma cell lines)	LC50	31600.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel melanoma (Carcinoma cell lines)	TGI	12600.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel NCI-60 (60 carcinoma cell lines)	GI50	3240.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel NCI-60 (60 carcinoma cell lines)	GI50	3240.0	nM	10.1016/j.ejmech.2019.111970
Homo sapiens	Panel NCI-60 (60 carcinoma cell lines)	LC50	50100.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel NCI-60 (60 carcinoma cell lines)	TGI	20000.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel ovarian (Carcinoma cell lines)	GI50	6630.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel ovarian (Carcinoma cell lines)	LC50	63100.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel ovarian (Carcinoma cell lines)	TGI	25100.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel prostate (Carcinoma cell lines)	GI50	1650.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel prostate (Carcinoma cell lines)	LC50	63100.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel prostate (Carcinoma cell lines)	TGI	20000.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel renal (Carcinoma cell lines)	GI50	2670.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel renal (Carcinoma cell lines)	LC50	39800.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	Panel renal (Carcinoma cell lines)	TGI	15900.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	PAS domain-containing serine/threonine-protein kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	PAS domain-containing serine/threonine-protein kinase	Ki	1584.89	nM	None
Homo sapiens	PC-14	IC50	333.41	nM	10.6019/CHEMBL1201861
Homo sapiens	PC-3	GI50	800.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	PC-3	IC50	2800.0	nM	10.1007/s00044-013-0734-x
Homo sapiens	PC-3	IC50	2833.17	nM	10.6019/CHEMBL1201861
Homo sapiens	PC-3	IC50	5300.0	nM	10.1021/acs.jmedchem.9b02008
Homo sapiens	PC-3	IC50	7400.0	nM	10.1016/j.bmcl.2011.01.137
Homo sapiens	PC-3	IC50	7400.0	nM	10.1039/C0MD00183J
Homo sapiens	PC-3	IC50	7990.0	nM	10.1016/j.ejmech.2019.03.030
Homo sapiens	PC-3	IC50	8920.0	nM	10.1016/j.bmc.2021.116265
Homo sapiens	PC-3	IC50	15100.0	nM	10.1016/j.ejmech.2008.01.009
Homo sapiens	PC-3	IC50	22860.0	nM	10.1016/j.bmc.2010.04.046
Homo sapiens	PC-9	Activity	64.0	%	10.1016/j.ejmech.2020.112359
Homo sapiens	PC-9	Activity	83.0	%	10.1016/j.ejmech.2020.112359
Homo sapiens	PC-9	EC50	17.0	nM	10.1016/j.bmcl.2010.12.036
Homo sapiens	PC-9	EC50	7000.0	nM	10.1016/j.bmcl.2010.12.036
Homo sapiens	PC-9	IC50	6.1	nM	10.1016/j.bmcl.2018.12.020
Homo sapiens	PC-9	IC50	14.0	nM	10.1021/jm301365e
Homo sapiens	PC-9	IC50	17.0	nM	10.1016/j.ejmech.2020.112185
Homo sapiens	PC-9	IC50	100.0	nM	10.1016/j.ejmech.2019.111607
Homo sapiens	PC-9	IC50	100.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	PC-9	IC50	31320.0	nM	10.1016/j.ejmech.2020.112388
Homo sapiens	PC-9	TGI	142.0	%	10.1021/jm400822z
Homo sapiens	PDZ-binding kinase	Ki	10000.0	nM	None
Homo sapiens	PDZ-binding kinase	Thermal melting change	0.6	degrees C	10.1073/pnas.0708800104
Homo sapiens	Peregrin	Delta TM	0.4566	C	None
Homo sapiens	Peripheral plasma membrane protein CASK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Peroxisomal acyl-coenzyme A oxidase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Peroxisomal acyl-coenzyme A oxidase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	PFSK-1	IC50	6734.78	nM	10.6019/CHEMBL1201861
Homo sapiens	P-glycoprotein 1	EC50	1000.0	nM	10.1016/j.ejmech.2022.114231
Homo sapiens	P-glycoprotein 1	IC50	19970.0	nM	10.1016/j.ejmech.2022.114231
Homo sapiens	P-glycoprotein 1	Inhibition	nan	%	10.1016/j.ejmech.2022.114231
Homo sapiens	P-glycoprotein 1	Ratio IC50	4.89	None	10.1016/j.ejmech.2022.114231
Homo sapiens	Phenylalanine--tRNA ligase beta subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Phosphatidylethanolamine-binding protein 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing beta polypeptide	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing subunit gamma	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-4-phosphate 5-kinase type-1 gamma	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 gamma	Kd	7500.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 gamma	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Phosphodiesterase 3A	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Phosphodiesterase 4D	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Phosphofructokinase platelet type	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Phosphorylase kinase gamma subunit 1	Kd	3700.0	nM	10.1038/nbt1358
Homo sapiens	Phosphorylase kinase gamma subunit 1	Kd	3700.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphorylase kinase gamma subunit 1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	2700.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	6400.0	nM	10.1038/nbt1068
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Phosphorylase kinase gamma subunit 2	Ki	3162.28	nM	None
Homo sapiens	PI3-kinase p110-alpha subunit	IC50	50000.0	nM	10.1038/nchembio.117
Homo sapiens	PI3-kinase p110-alpha subunit	IC50	nan	None	10.1016/j.ejmech.2018.01.081
Homo sapiens	PI3-kinase p110-alpha subunit	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	PI3-kinase p110-alpha subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PI3-kinase p110-beta subunit	IC50	50000.0	nM	10.1038/nchembio.117
Homo sapiens	PI3-kinase p110-beta subunit	IC50	nan	None	10.1016/j.ejmech.2018.01.081
Homo sapiens	PI3-kinase p110-beta subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PI3-kinase p110-delta subunit	IC50	50000.0	nM	10.1038/nchembio.117
Homo sapiens	PI3-kinase p110-delta subunit	IC50	nan	None	10.1016/j.ejmech.2018.01.081
Homo sapiens	PI3-kinase p110-delta subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PI3-kinase p110-gamma subunit	IC50	50000.0	nM	10.1038/nchembio.117
Homo sapiens	PI3-kinase p110-gamma subunit	IC50	nan	None	10.1016/j.ejmech.2018.01.081
Homo sapiens	PI3-kinase p110-gamma subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PI4-kinase beta subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Platelet-derived growth factor receptor alpha	Inhibition	54.0	%	10.1016/j.bmc.2018.02.022
Homo sapiens	Platelet-derived growth factor receptor alpha	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Platelet-derived growth factor receptor alpha	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Platelet-derived growth factor receptor alpha	Ki	1995.26	nM	None
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Platelet-derived growth factor receptor beta	Ki	1995.26	nM	None
Homo sapiens	PLC-PRF-5	IC50	4000.0	nM	10.1021/acs.jnatprod.8b00821
Homo sapiens	Pregnane X receptor	AC50	20000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Pregnane X receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Prelamin-A/C	Potency	0.8	nM	None
Homo sapiens	Probable ATP-dependent RNA helicase DDX6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Progesterone receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Protein kinase C alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C alpha	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Protein kinase C beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C delta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C delta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C delta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C delta	Ki	7943.28	nM	None
Homo sapiens	Protein kinase C epsilon	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C epsilon	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C eta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C eta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C gamma	Ki	7943.28	nM	None
Homo sapiens	Protein kinase C iota	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C iota	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C iota	Ki	5011.87	nM	None
Homo sapiens	Protein kinase C mu	Kd	3500.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C mu	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C nu	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C nu	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C nu	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C nu	Ki	1258.93	nM	None
Homo sapiens	Protein kinase C theta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C theta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C theta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C theta	Ki	2511.89	nM	None
Homo sapiens	Protein kinase C zeta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C zeta	Ki	7943.28	nM	None
Homo sapiens	Protein kinase N1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase N1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase N1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase N2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase N2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase N2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase N2	Ki	7943.28	nM	None
Homo sapiens	Protein tyrosine kinase 2 beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Protein tyrosine kinase 2 beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein tyrosine kinase 2 beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein tyrosine kinase 2 beta	Ki	1584.89	nM	None
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	Ki	1995.26	nM	None
Homo sapiens	PSN1	IC50	38991.9	nM	10.6019/CHEMBL1201861
Homo sapiens	Putative heat shock protein HSP 90-beta 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Putative uncharacterized serine/threonine-protein kinase SgK110	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Pyridoxal kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	QIMR-WIL	IC50	2759.52	nM	10.6019/CHEMBL1201861
Homo sapiens	Quinone reductase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ramos-2G6-4C10	IC50	621.46	nM	10.6019/CHEMBL1201861
Homo sapiens	Ras-related protein Rab-10	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ras-related protein Rab-27A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ras-related protein Rab-6A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	RCC10RGB	IC50	4012.46	nM	10.6019/CHEMBL1201861
Homo sapiens	RCM-1	IC50	6077.19	nM	10.6019/CHEMBL1201861
Homo sapiens	RD	IC50	14481.27	nM	10.6019/CHEMBL1201861
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 3	Kd	2664.0	nM	10.1126/science.aan4368
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	AC50	25.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	24.0	nM	10.1016/j.ejmech.2016.12.014
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	97.0	nM	10.1021/acs.jmedchem.0c00870
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	151.0	nM	10.1016/j.bmcl.2018.12.020
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	240.0	nM	10.1016/j.bmcl.2003.10.010
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	240.0	nM	10.1016/j.bmcl.2011.01.119
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	240.0	nM	10.1016/j.bmcl.2011.10.103
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	240.0	nM	10.1021/jm901132v
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	280.0	nM	10.1016/j.bmcl.2013.12.079
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	281.0	nM	10.1016/j.bmcl.2016.08.007
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	281.0	nM	10.1016/j.bmcl.2020.127045
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	343.0	nM	10.1021/acs.jmedchem.6b00883
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	343.0	nM	10.1021/acs.jmedchem.9b01617
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	343.0	nM	10.1021/jm050936o
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	599.0	nM	10.1021/jm050936o
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	1000.0	nM	10.1021/jm5014659
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	1604.0	nM	10.1016/s0960-894x(02)00598-x
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	1830.0	nM	10.1016/j.ejmech.2016.04.026
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	2700.0	nM	10.1016/j.bmcl.2008.11.023
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	3700.0	nM	10.1016/j.bmc.2016.10.006
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	9420.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	nan	None	10.1016/j.bmc.2016.10.006
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	nan	None	10.1016/j.ejmech.2018.06.061
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	IC50	nan	None	10.1021/acs.jmedchem.8b01612
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Inhibition	46.0	%	10.1021/acs.jmedchem.6b01774
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Inhibition	81.11	%	10.1016/j.bmc.2010.04.046
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Inhibition	nan	%	10.1021/jm901558p
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Kd	1100.0	nM	10.1038/nbt1068
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Kd	3500.0	nM	10.1038/nbt1358
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Kd	3500.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Ki	25.12	nM	None
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	IC50	476.0	nM	10.1021/acs.jmedchem.6b00883
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	IC50	nan	None	10.1016/j.ejmech.2016.04.026
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	Inhibition	46.0	%	10.1021/acs.jmedchem.6b01774
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	Inhibition	103.9	%	10.1016/j.bmc.2018.02.022
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	Kd	410.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	Ki	158.49	nM	None
Homo sapiens	Receptor tyrosine-protein kinase erbB-3	Kd	790.0	nM	10.1038/nbt.1990
Homo sapiens	RERF-LC-MS	IC50	42508.71	nM	10.6019/CHEMBL1201861
Homo sapiens	RH-1	IC50	1411.36	nM	10.6019/CHEMBL1201861
Homo sapiens	RH-18	IC50	13296.24	nM	10.6019/CHEMBL1201861
Homo sapiens	Rho-associated protein kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Rho-associated protein kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Rho-associated protein kinase 1	Ki	6309.57	nM	None
Homo sapiens	Rho-associated protein kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Rho-associated protein kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Rho-associated protein kinase 2	Ki	6309.57	nM	None
Homo sapiens	Rhodopsin kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ribosomal protein S6 kinase 1	Ki	5011.87	nM	None
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Ki	3981.07	nM	None
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Thermal melting change	1.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Thermal melting change	5.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	1200.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Ki	1584.89	nM	None
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Ki	1995.26	nM	None
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	RKO	IC50	17074.82	nM	10.6019/CHEMBL1201861
Homo sapiens	RKO	Inhibition	nan	%	10.1016/j.bmcl.2014.09.056
Homo sapiens	RMG-I	IC50	5659.42	nM	10.6019/CHEMBL1201861
Homo sapiens	RNA cytidine acetyltransferase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	RO82-W-1	IC50	43615.34	nM	10.6019/CHEMBL1201861
Homo sapiens	RPMI-2650	IC50	72175.02	nM	10.6019/CHEMBL1201861
Homo sapiens	RPMI-7951	IC50	11634.84	nM	10.6019/CHEMBL1201861
Homo sapiens	RPMI-8226	Activity	80.92	pg/ml	10.1016/j.ejmech.2020.112062
Homo sapiens	RPMI-8226	IC50	9113.04	nM	10.6019/CHEMBL1201861
Homo sapiens	RPMI-8866	IC50	2084.81	nM	10.6019/CHEMBL1201861
Homo sapiens	RS4-11	IC50	568.59	nM	10.6019/CHEMBL1201861
Homo sapiens	RT-112	IC50	5902.45	nM	10.6019/CHEMBL1201861
Homo sapiens	RVH-421	IC50	25816.07	nM	10.6019/CHEMBL1201861
Homo sapiens	RXF 393	GI50	5010.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	RXF 393	IC50	2130.36	nM	10.6019/CHEMBL1201861
Homo sapiens	S-117	IC50	43695.84	nM	10.6019/CHEMBL1201861
Homo sapiens	S-adenosylmethionine synthase isoform type-2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	SAOS-2	IC50	23518.16	nM	10.6019/CHEMBL1201861
Homo sapiens	SAS	IC50	1516.22	nM	10.6019/CHEMBL1201861
Homo sapiens	SBC-1	IC50	307.79	nM	10.6019/CHEMBL1201861
Homo sapiens	SBC-5	IC50	55130.6	nM	10.6019/CHEMBL1201861
Homo sapiens	SCC-15	IC50	525.68	nM	10.6019/CHEMBL1201861
Homo sapiens	SCC-25	IC50	1523.22	nM	10.6019/CHEMBL1201861
Homo sapiens	SCC-4	IC50	2217.76	nM	10.6019/CHEMBL1201861
Homo sapiens	SCC-9	IC50	11815.07	nM	10.6019/CHEMBL1201861
Homo sapiens	SCH	IC50	29883.07	nM	10.6019/CHEMBL1201861
Homo sapiens	Septin-9	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase 10	Inhibition	46.0	%	10.1021/acs.jmedchem.6b01774
Homo sapiens	Serine/threonine-protein kinase 10	Inhibition	80.8	%	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 10	Kd	470.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 10	Kd	470.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 10	Kd	870.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 10	Kd	5236.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase 10	Thermal melting change	0.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase 11	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 11	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 11	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase 16	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 16	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 16	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase 16	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 16	Thermal melting change	3.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase 17A	Kd	2000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 17A	Kd	2000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 17A	Kd	2900.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 17A	Ki	3981.07	nM	None
Homo sapiens	Serine/threonine-protein kinase 17A	Thermal melting change	0.6	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase 17B	Kd	3800.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 17B	Kd	3800.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 17B	Kd	6500.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 2	Inhibition	72.7	%	10.1016/j.bmc.2018.02.022
Homo sapiens	Serine/threonine-protein kinase 2	Kd	920.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 2	Kd	920.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 2	Kd	1100.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase 2	Ki	398.11	nM	None
Homo sapiens	Serine/threonine-protein kinase 2	Thermal melting change	7.8	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase 24	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 24	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 24	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase 25	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 25	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 25	Thermal melting change	nan	None	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase 32A	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 32B	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 32B	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 32C	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 32C	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 33	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 33	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 35	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 36	Kd	5700.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 36	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 36	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 38	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 38	Thermal melting change	0.5	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase 38-like	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 38-like	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 38-like	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase AKT	Inhibition	nan	%	10.1016/j.ejmech.2014.02.032
Homo sapiens	Serine/threonine-protein kinase AKT	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase AKT	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase AKT	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase AKT	Ki	7943.28	nM	None
Homo sapiens	Serine/threonine-protein kinase AKT2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase AKT2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase AKT2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase AKT2	Ki	7943.28	nM	None
Homo sapiens	Serine/threonine-protein kinase AKT3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase AKT3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase AKT3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase AKT3	Ki	10000.0	nM	None
Homo sapiens	Serine/threonine-protein kinase A-Raf	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Delta TM	0.1745	C	None
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Ki	3162.28	nM	None
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Ki	6309.57	nM	None
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	2000.0	nM	10.1021/jm500007h
Homo sapiens	Serine/threonine-protein kinase B-raf	IC50	30000.0	nM	None
Homo sapiens	Serine/threonine-protein kinase B-raf	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase B-raf	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase B-raf	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Chk1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Chk1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Chk1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Chk1	Ki	6309.57	nM	None
Homo sapiens	Serine/threonine-protein kinase Chk2	Kd	800.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Chk2	Ki	630.96	nM	None
Homo sapiens	Serine/threonine-protein kinase Chk2	Thermal melting change	3.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Ki	6309.57	nM	None
Homo sapiens	Serine/threonine-protein kinase D2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase D2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase D2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase D2	Ki	2511.89	nM	None
Homo sapiens	Serine/threonine-protein kinase DCLK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase DCLK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase DCLK1	Ki	10000.0	nM	None
Homo sapiens	Serine/threonine-protein kinase DCLK2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase DCLK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase DCLK3	Kd	2900.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase DCLK3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase EEF2K	Ki	3981.07	nM	None
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase GAK	IC50	420.0	nM	10.1021/acs.jmedchem.9b00350
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	7.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	13.0	nM	10.1016/j.bmcl.2019.05.025
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	13.0	nM	10.1021/acs.jmedchem.1c00302
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	13.0	nM	10.1021/acs.jmedchem.8b01213
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	13.0	nM	10.1021/acs.jmedchem.9b00350
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	13.0	nM	10.1021/jm501759m
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	13.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	13.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	951.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase ICK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase ICK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase ILK-1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase LATS1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase LATS1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase LATS1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase LATS2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase LATS2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MAK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MARK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MARK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Ki	10000.0	nM	None
Homo sapiens	Serine/threonine-protein kinase MRCK beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MRCK beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MRCK beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase MRCK gamma	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MRCK gamma	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MRCK gamma	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase MST1	Thermal melting change	1.6	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase MST2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MST2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MST2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase MST2	Ki	7943.28	nM	None
Homo sapiens	Serine/threonine-protein kinase MST4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MST4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MST4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase MST4	Thermal melting change	0.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase MST4	Thermal melting change	1.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase mTOR	IC50	50000.0	nM	10.1038/nchembio.117
Homo sapiens	Serine/threonine-protein kinase mTOR	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase N3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Nek1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Nek1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Nek1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Nek11	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase NEK2	Ki	7943.28	nM	None
Homo sapiens	Serine/threonine-protein kinase NEK2	Thermal melting change	1.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase Nek3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Nek3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Nek4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Nek4	Ki	6309.57	nM	None
Homo sapiens	Serine/threonine-protein kinase Nek5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Nek5	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK6	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase NEK6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK6	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase NEK6	Thermal melting change	-0.4	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase NEK7	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase NEK7	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK7	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase NEK9	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase NEK9	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK9	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase NEK9	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase NIM1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine protein kinase NLK	Kd	4200.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine protein kinase NLK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine protein kinase NLK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase OSR1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase OSR1	Thermal melting change	0.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PAK 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK 1	Ki	10000.0	nM	None
Homo sapiens	Serine/threonine-protein kinase PAK 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PAK 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 3	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PAK 4	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK 4	Ki	5011.87	nM	None
Homo sapiens	Serine/threonine-protein kinase PAK 4	Thermal melting change	1.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PAK6	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PAK6	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK6	Thermal melting change	0.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PAK7	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK7	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK7	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK7	Thermal melting change	0.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Thermal melting change	-0.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PFTAIRE-1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PFTAIRE-1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PFTAIRE-2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PIM1	Ki	1995.26	nM	None
Homo sapiens	Serine/threonine-protein kinase PIM1	Thermal melting change	3.4	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PIM2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PIM2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PIM2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PIM2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PIM2	Ki	794.33	nM	None
Homo sapiens	Serine/threonine-protein kinase PIM2	Thermal melting change	0.6	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PIM3	Kd	5800.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PIM3	Kd	5800.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PIM3	Ki	1258.93	nM	None
Homo sapiens	Serine/threonine-protein kinase PIM3	Thermal melting change	-0.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PLK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PLK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PLK1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PLK1	Ki	7943.28	nM	None
Homo sapiens	Serine/threonine-protein kinase PLK1	Thermal melting change	1.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PLK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PLK3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PLK3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PLK3	Ki	7943.28	nM	None
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PLK4	Ki	3981.07	nM	None
Homo sapiens	Serine/threonine-protein kinase PLK4	Thermal melting change	0.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PRKX	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PRKX	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PRKX	Ki	1584.89	nM	None
Homo sapiens	Serine/threonine-protein kinase PRP4 homolog	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RAF	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase RAF	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase receptor R3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase receptor R3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIO1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase RIO1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIO2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIO2	Thermal melting change	2.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase RIO3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase RIO3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIPK2	IC50	3.8	nM	None
Homo sapiens	Serine/threonine-protein kinase RIPK2	Inhibition	46.0	%	10.1021/acs.jmedchem.6b01774
Homo sapiens	Serine/threonine-protein kinase RIPK2	Kd	530.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase RIPK2	Kd	530.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIPK2	Kd	800.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase RIPK2	Kd	903.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase SBK1	Kd	560.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Sgk2	Ki	7943.28	nM	None
Homo sapiens	Serine/threonine-protein kinase Sgk3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SIK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase SIK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SIK2	Inhibition	46.0	%	10.1021/acs.jmedchem.6b01774
Homo sapiens	Serine/threonine-protein kinase SIK2	Kd	2100.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase SIK2	Kd	2100.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SIK2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase SIK2	Ki	316.23	nM	None
Homo sapiens	Serine/threonine-protein kinase SIK3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SIK3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase SRPK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase SRPK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SRPK1	Ki	7943.28	nM	None
Homo sapiens	Serine/threonine-protein kinase SRPK2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase SRPK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SRPK3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TAO1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TAO1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase TAO1	Ki	6309.57	nM	None
Homo sapiens	Serine/threonine-protein kinase TAO2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TAO2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase TAO3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TAO3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase TBK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TBK1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase TBK1	Ki	3162.28	nM	None
Homo sapiens	Serine/threonine-protein kinase TNNI3K	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase TNNI3K	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase tousled-like 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase tousled-like 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase tousled-like 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase tousled-like 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase ULK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase ULK1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase ULK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase ULK3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase ULK3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase VRK1	Thermal melting change	0.5	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase VRK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase VRK2	Thermal melting change	0.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase WEE1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase WEE1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase WEE1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serotonin 1a (5-HT1a) receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 2a (5-HT2a) receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 2b (5-HT2b) receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 2c (5-HT2c) receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 3a (5-HT3a) receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin transporter	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	SF-126	IC50	28743.51	nM	10.6019/CHEMBL1201861
Homo sapiens	SF-268	IC50	17696.89	nM	10.6019/CHEMBL1201861
Homo sapiens	SF-295	GI50	2000.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	SF-295	IC50	10990.17	nM	10.6019/CHEMBL1201861
Homo sapiens	SF-539	IC50	42552.94	nM	10.6019/CHEMBL1201861
Homo sapiens	SGC-7901	IC50	10260.0	nM	10.1016/j.ejmech.2012.05.039
Homo sapiens	SGC-7901	IC50	29010.0	nM	10.1016/j.ejmech.2020.112737
Homo sapiens	SH-4	IC50	6588.44	nM	10.6019/CHEMBL1201861
Homo sapiens	SHP77	IC50	7866.53	nM	10.6019/CHEMBL1201861
Homo sapiens	SH-SY5Y	IC50	18210.0	nM	10.1016/j.ejmech.2017.07.005
Homo sapiens	SH-SY5Y	IC50	18216.0	nM	10.1016/j.bmc.2019.06.001
Homo sapiens	Signal recognition particle receptor subunit alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	SiHa	IC50	20371.18	nM	10.6019/CHEMBL1201861
Homo sapiens	SJRH30	IC50	94066.69	nM	10.6019/CHEMBL1201861
Homo sapiens	SJSA-1	IC50	52895.17	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-BR-3	IC50	0.174	ug.mL-1	10.1016/s0960-894x(02)00598-x
Homo sapiens	SK-BR-3	IC50	2518.0	nM	10.1016/j.bmcl.2018.12.020
Homo sapiens	SK-BR-3	IC50	4920.0	nM	10.1016/j.ejmech.2016.04.026
Homo sapiens	SKG-IIIa	IC50	7453.81	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-HEP1	IC50	6717.53	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-HEP1	IC50	10100.0	nM	10.1016/j.ejmech.2018.01.081
Homo sapiens	SK-LMS-1	IC50	78325.64	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-LU-1	IC50	3606.45	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-MEL-1	IC50	510.99	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-MEL-2	IC50	32052.01	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-MEL-24	IC50	337.87	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-MEL-28	GI50	320.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	SK-MEL-28	IC50	6209.67	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-MEL-28	IC50	20000.0	nM	10.1021/jm500007h
Homo sapiens	SK-MEL3	IC50	26982.76	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-MEL-30	IC50	207070.64	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-MES-1	IC50	3646.14	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-N-AS	IC50	21561.86	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-N-DZ	IC50	1369.47	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-NEP-1	IC50	989.44	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-N-FI	IC50	22307.41	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-OV-3	IC50	4460.42	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-OV-3	IC50	24500.0	nM	10.1016/j.ejmech.2020.112640
Homo sapiens	SK-PN-DW	IC50	13842.73	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-UT-1	IC50	10257.37	nM	10.6019/CHEMBL1201861
Homo sapiens	SMMC-7721	IC50	9200.0	nM	10.1021/acs.jnatprod.8b00821
Homo sapiens	SMMC-7721	IC50	33120.0	nM	10.1016/j.ejmech.2010.03.001
Homo sapiens	SN12C	IC50	13380.78	nM	10.6019/CHEMBL1201861
Homo sapiens	SNB-75	GI50	6310.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	SNB-75	IC50	57826.66	nM	10.6019/CHEMBL1201861
Homo sapiens	SNF-related serine/threonine-protein kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	SNU1	IC50	283.32	nM	10.6019/CHEMBL1201861
Homo sapiens	SNU-387	IC50	40823.79	nM	10.6019/CHEMBL1201861
Homo sapiens	SNU-423	IC50	55193.93	nM	10.6019/CHEMBL1201861
Homo sapiens	SNU-449	IC50	1222.08	nM	10.6019/CHEMBL1201861
Homo sapiens	SNU-5	IC50	28.19	nM	10.6019/CHEMBL1201861
Homo sapiens	SNU-638	IC50	7560.0	nM	10.1016/j.ejmech.2018.01.081
Homo sapiens	SNU-C2B	IC50	4346.86	nM	10.6019/CHEMBL1201861
Homo sapiens	SPS1/STE20-related protein kinase YSK4	Kd	240.0	nM	10.1038/nbt.1990
Homo sapiens	SR	GI50	3160.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	STE20-related kinase adapter protein alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	STE20/SPS1-related proline-alanine-rich protein kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	1800.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	4300.0	nM	10.1016/j.ejmech.2011.02.057
Homo sapiens	Stem cell growth factor receptor	Kd	4300.0	nM	10.1038/nbt1358
Homo sapiens	Stem cell growth factor receptor	Kd	4300.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	5500.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	10000.0	nM	10.1016/j.ejmech.2011.02.057
Homo sapiens	Stem cell growth factor receptor	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Stem cell growth factor receptor	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Stem cell growth factor receptor	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Stem cell growth factor receptor	Ki	1000.0	nM	None
Homo sapiens	Structural maintenance of chromosomes protein 1A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Structural maintenance of chromosomes protein 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	SW1088	IC50	1296.07	nM	10.6019/CHEMBL1201861
Homo sapiens	SW 1116	IC50	2060.09	nM	10.6019/CHEMBL1201861
Homo sapiens	SW13	IC50	5532.65	nM	10.6019/CHEMBL1201861
Homo sapiens	SW1417	IC50	42302.96	nM	10.6019/CHEMBL1201861
Homo sapiens	SW1463	IC50	3261.92	nM	10.6019/CHEMBL1201861
Homo sapiens	SW1573	IC50	29350.86	nM	10.6019/CHEMBL1201861
Homo sapiens	SW1710	IC50	24150.62	nM	10.6019/CHEMBL1201861
Homo sapiens	SW1783	IC50	17641.45	nM	10.6019/CHEMBL1201861
Homo sapiens	SW1990	IC50	5622.85	nM	10.6019/CHEMBL1201861
Homo sapiens	SW1990	Inhibition	nan	%	10.1016/j.bmcl.2015.01.060
Homo sapiens	SW48	IC50	1366.18	nM	10.6019/CHEMBL1201861
Homo sapiens	SW480	IC50	12500.0	nM	10.1016/j.ejmech.2017.06.023
Homo sapiens	SW480	IC50	12500.0	nM	10.1016/j.ejmech.2018.01.090
Homo sapiens	SW480	IC50	12500.0	nM	10.1016/j.ejmech.2019.06.015
Homo sapiens	SW480	IG50	12.5	uM	10.1016/j.bmcl.2017.02.027
Homo sapiens	SW-620	IC50	5.0	ug.mL-1	10.1016/s0960-894x(02)00598-x
Homo sapiens	SW-620	IC50	10000.0	nM	10.1021/jm901558p
Homo sapiens	SW-620	IC50	28200.0	nM	10.1021/ml4002437
Homo sapiens	SW-620	IC50	29364.1	nM	10.6019/CHEMBL1201861
Homo sapiens	SW626	IC50	37041.73	nM	10.6019/CHEMBL1201861
Homo sapiens	SW684	IC50	47008.1	nM	10.6019/CHEMBL1201861
Homo sapiens	SW756	IC50	43824.15	nM	10.6019/CHEMBL1201861
Homo sapiens	SW780	IC50	47635.06	nM	10.6019/CHEMBL1201861
Homo sapiens	SW837	IC50	9848.2	nM	10.6019/CHEMBL1201861
Homo sapiens	SW872	IC50	40203.1	nM	10.6019/CHEMBL1201861
Homo sapiens	SW900	IC50	10822.81	nM	10.6019/CHEMBL1201861
Homo sapiens	SW948	IC50	38894.86	nM	10.6019/CHEMBL1201861
Homo sapiens	SW 954	IC50	1340.48	nM	10.6019/CHEMBL1201861
Homo sapiens	SW 962	IC50	10620.42	nM	10.6019/CHEMBL1201861
Homo sapiens	SW982	IC50	18407.48	nM	10.6019/CHEMBL1201861
Homo sapiens	T-24	IC50	14600.0	nM	10.1016/j.ejmech.2020.112661
Homo sapiens	T-24	IC50	31736.17	nM	10.6019/CHEMBL1201861
Homo sapiens	T47D	IC50	41019.23	nM	10.6019/CHEMBL1201861
Homo sapiens	T84	IC50	24976.52	nM	10.6019/CHEMBL1201861
Homo sapiens	T98G	IC50	37863.55	nM	10.6019/CHEMBL1201861
Homo sapiens	TCC-SUP	IC50	4110.5	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-1	IC50	3591.69	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-10	IC50	6048.33	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-11	IC50	7049.67	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-12	IC50	821.11	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-5	IC50	20748.25	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-6	IC50	764.31	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-8	IC50	2636.53	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-9	IC50	5015.25	nM	10.6019/CHEMBL1201861
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	Ki	1584.89	nM	None
Homo sapiens	Testis-specific serine/threonine-protein kinase 2	Ki	1584.89	nM	None
Homo sapiens	TGBC11TKB	IC50	8461.64	nM	10.6019/CHEMBL1201861
Homo sapiens	TGBC1TKB	IC50	14661.5	nM	10.6019/CHEMBL1201861
Homo sapiens	TGBC24TKB	IC50	2029.61	nM	10.6019/CHEMBL1201861
Homo sapiens	TGF-beta receptor type I	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	TGF-beta receptor type I	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	TGF-beta receptor type I	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	TGF-beta receptor type II	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	TGF-beta receptor type II	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	TGF-beta receptor type II	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Thromboxane A2 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Thyroid hormone receptor-associated protein 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	TI-73	IC50	312.75	nM	10.6019/CHEMBL1201861
Homo sapiens	TK-10	GI50	100.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	TK-10	IC50	515.11	nM	10.6019/CHEMBL1201861
Homo sapiens	TP53-regulating kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	6900.0	nM	10.1038/nbt.1990
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	nan	None	10.1038/nbt1068
Homo sapiens	TRAF2- and NCK-interacting kinase	Thermal melting change	-1.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	Transcription intermediary factor 1-alpha	Delta TM	0.074	C	None
Homo sapiens	Transient receptor potential cation channel subfamily M member 6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	TYK-nu	IC50	19837.82	nM	10.6019/CHEMBL1201861
Homo sapiens	Type-1 angiotensin II receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine kinase non-receptor protein 2	IC50	2300.0	nM	None
Homo sapiens	Tyrosine kinase non-receptor protein 2	IC50	20000.0	nM	10.1021/acs.jmedchem.1c01030
Homo sapiens	Tyrosine kinase non-receptor protein 2	Inhibition	77.0	%	10.1021/acs.jmedchem.1c01030
Homo sapiens	Tyrosine kinase non-receptor protein 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine kinase non-receptor protein 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine kinase non-receptor protein 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine kinase non-receptor protein 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine kinase non-receptor protein 2	Ki	3162.28	nM	None
Homo sapiens	Tyrosine-protein kinase ABL	Delta TM	4.064	C	None
Homo sapiens	Tyrosine-protein kinase ABL	IC50	1200.0	nM	10.1038/nchembio.117
Homo sapiens	Tyrosine-protein kinase ABL	Inhibition	nan	%	10.1016/j.ejmech.2013.03.013
Homo sapiens	Tyrosine-protein kinase ABL	Kd	230.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	360.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	400.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	460.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	480.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	520.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	680.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	780.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	1100.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	2200.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	2700.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	4700.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase ABL	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Ki	630.96	nM	None
Homo sapiens	Tyrosine-protein kinase ABL2	Inhibition	38.6	%	10.1016/j.bmc.2018.02.022
Homo sapiens	Tyrosine-protein kinase ABL2	Kd	1600.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase ABL2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase BLK	Kd	1200.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase BLK	Kd	1200.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase BLK	Ki	1000.0	nM	None
Homo sapiens	Tyrosine-protein kinase BMX	Activity	nan	None	10.1016/j.bmcl.2008.07.062
Homo sapiens	Tyrosine-protein kinase BMX	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase BMX	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase BMX	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase BRK	IC50	980.0	nM	None
Homo sapiens	Tyrosine-protein kinase BRK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase BRK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase BRK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase BRK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase BRK	Ki	1995.26	nM	None
Homo sapiens	Tyrosine-protein kinase BTK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase BTK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase BTK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase BTK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase BTK	Ki	1258.93	nM	None
Homo sapiens	Tyrosine-protein kinase CSK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase CSK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase CSK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase CSK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase CTK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase CTK	Ki	1995.26	nM	None
Homo sapiens	Tyrosine-protein kinase FER	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FER	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FER	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase FER	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase FER	Ki	1584.89	nM	None
Homo sapiens	Tyrosine-protein kinase FES	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FES	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FES	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase FES	Ki	1995.26	nM	None
Homo sapiens	Tyrosine-protein kinase FGR	Kd	2600.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FGR	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FGR	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase FGR	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase FRK	Kd	2000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FRK	Kd	2000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FRK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase FRK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase FRK	Ki	251.19	nM	None
Homo sapiens	Tyrosine-protein kinase FYN	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FYN	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FYN	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase FYN	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase FYN	Ki	794.33	nM	None
Homo sapiens	Tyrosine-protein kinase HCK	IC50	110.0	nM	10.1038/nchembio.117
Homo sapiens	Tyrosine-protein kinase HCK	Kd	4400.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase HCK	Kd	4400.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase HCK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase HCK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase HCK	Ki	2511.89	nM	None
Homo sapiens	Tyrosine-protein kinase ITK/TSK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ITK/TSK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ITK/TSK	Ki	1584.89	nM	None
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase JAK1	Thermal melting change	1.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	Tyrosine-protein kinase JAK2	Activity	nan	None	10.1074/jbc.c600277200
Homo sapiens	Tyrosine-protein kinase JAK2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase JAK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase JAK2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase JAK2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase JAK2	Ki	1584.89	nM	None
Homo sapiens	Tyrosine-protein kinase JAK3	IC50	1000.0	nM	10.1021/acs.jmedchem.6b00883
Homo sapiens	Tyrosine-protein kinase JAK3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase JAK3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase JAK3	Ki	1584.89	nM	None
Homo sapiens	Tyrosine-protein kinase LCK	Kd	630.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase LCK	Kd	630.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase LCK	Kd	1100.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase LCK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase LCK	Ki	398.11	nM	None
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	990.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	990.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase Lyn	Ki	158.49	nM	None
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	1000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	1000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	1100.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	1100.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2900.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	3000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	3000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	3100.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	3500.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	5100.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Ki	2511.89	nM	None
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	1700.0	nM	10.1038/nchembio.117
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase receptor RET	Ki	1258.93	nM	None
Homo sapiens	Tyrosine-protein kinase receptor Tie-1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor Tie-1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Ki	1995.26	nM	None
Homo sapiens	Tyrosine-protein kinase receptor UFO	Kd	1800.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor UFO	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor UFO	Ki	1584.89	nM	None
Homo sapiens	Tyrosine-protein kinase SRC	IC50	1100.0	nM	10.1038/nchembio.117
Homo sapiens	Tyrosine-protein kinase SRC	Inhibition	nan	%	10.1016/j.ejmech.2012.06.055
Homo sapiens	Tyrosine-protein kinase SRC	Inhibition	nan	%	10.1016/j.ejmech.2013.03.013
Homo sapiens	Tyrosine-protein kinase SRC	Kd	3800.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase SRC	Kd	3800.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase SRC	Kd	5000.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase SRC	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase SRC	Ki	1995.26	nM	None
Homo sapiens	Tyrosine-protein kinase Srms	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase Srms	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase Srms	Ki	1584.89	nM	None
Homo sapiens	Tyrosine-protein kinase SYK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase SYK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase SYK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase SYK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase SYK	Ki	1584.89	nM	None
Homo sapiens	Tyrosine-protein kinase TEC	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase TEC	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TEC	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase TIE-2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase TIE-2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TIE-2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase TXK	Kd	6000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase TXK	Kd	6000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TYK2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase TYK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TYK2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase TYK2	Ki	1995.26	nM	None
Homo sapiens	Tyrosine-protein kinase YES	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase YES	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase YES	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase YES	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase YES	Potency	1373.4	nM	None
Homo sapiens	Tyrosine-protein kinase YES	Potency	1729.1	nM	None
Homo sapiens	Tyrosine-protein kinase ZAP-70	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ZAP-70	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosyl-DNA phosphodiesterase 1	Potency	5309.1	nM	None
Homo sapiens	Tyrosyl-tRNA synthetase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	U-118-MG	IC50	12244.13	nM	10.6019/CHEMBL1201861
Homo sapiens	U-251	GI50	10000.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	U-251	IC50	10800.0	nM	10.1021/np500382k
Homo sapiens	U-251	IC50	18734.69	nM	10.6019/CHEMBL1201861
Homo sapiens	U-266	IC50	18864.94	nM	10.6019/CHEMBL1201861
Homo sapiens	U2OS	Growth Rate	0.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	Growth Rate	1.0	None	10.6019/CHEMBL4689842
Homo sapiens	U2OS	IC50	26375.72	nM	10.6019/CHEMBL1201861
Homo sapiens	U5 small nuclear ribonucleoprotein 200 kDa helicase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	U-87 MG	IC50	22400.0	nM	10.1016/j.ejmech.2019.111966
Homo sapiens	U-87 MG	IC50	26743.84	nM	10.6019/CHEMBL1201861
Homo sapiens	U-937	IC50	nan	None	10.1016/j.ejmech.2013.03.013
Homo sapiens	UACC-257	GI50	6310.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	UACC-257	IC50	27380.36	nM	10.6019/CHEMBL1201861
Homo sapiens	UACC-62	GI50	5010.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	UACC-62	IC50	23583.26	nM	10.6019/CHEMBL1201861
Homo sapiens	UACC-893	IC50	27663.12	nM	10.6019/CHEMBL1201861
Homo sapiens	UMC-11	IC50	15752.26	nM	10.6019/CHEMBL1201861
Homo sapiens	UMP-CMP kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	UMUC3	IC50	11742.08	nM	10.6019/CHEMBL1201861
Homo sapiens	Uncharacterized aarF domain-containing protein kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Uncharacterized aarF domain-containing protein kinase 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Uncharacterized aarF domain-containing protein kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Uncharacterized aarF domain-containing protein kinase 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Uncharacterized protein FLJ45252	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	UO-31	GI50	1260.0	nM	10.1016/j.bmcl.2016.05.047
Homo sapiens	UO-31	IC50	10268.57	nM	10.6019/CHEMBL1201861
Homo sapiens	VA-ES-BJ	IC50	6304.62	nM	10.6019/CHEMBL1201861
Homo sapiens	Vascular endothelial growth factor receptor	IC50	nan	None	10.1016/j.ejmech.2018.06.061
Homo sapiens	Vascular endothelial growth factor receptor 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Vascular endothelial growth factor receptor 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Vascular endothelial growth factor receptor 1	Ki	398.11	nM	None
Homo sapiens	Vascular endothelial growth factor receptor 2	AC50	2500.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	48.5	nM	10.1016/j.bmc.2018.02.023
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	1900.0	nM	10.1038/nchembio.117
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	10000.0	nM	10.1016/j.bmc.2007.03.055
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	14800.0	nM	10.1016/j.bmcl.2011.01.137
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	14800.0	nM	10.1039/C0MD00183J
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	nan	None	10.1016/j.bmc.2015.12.001
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	6.0	%	10.1016/j.bmc.2007.03.055
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	12.0	%	10.1016/j.bmc.2007.03.055
Homo sapiens	Vascular endothelial growth factor receptor 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Vascular endothelial growth factor receptor 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Vascular endothelial growth factor receptor 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Vascular endothelial growth factor receptor 2	Ki	1995.26	nM	None
Homo sapiens	Vascular endothelial growth factor receptor 2	Ratio	1.0	None	10.1016/j.bmc.2007.03.055
Homo sapiens	Vascular endothelial growth factor receptor 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Vascular endothelial growth factor receptor 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Vascular endothelial growth factor receptor 3	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Vascular endothelial growth factor receptor 3	Ki	6309.57	nM	None
Homo sapiens	Vasopressin V1a receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Vasopressin V2 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Very long-chain specific acyl-CoA dehydrogenase, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	VHL/EGFR	Activity	nan	None	10.1021/acs.jmedchem.1c00649
Homo sapiens	VHL/PARP1	Activity	nan	None	10.1021/acs.jmedchem.1c00649
Homo sapiens	Vitamin D receptor	Potency	89125.1	nM	None
Homo sapiens	VM-CUB-1	IC50	8170.29	nM	10.6019/CHEMBL1201861
Homo sapiens	VMRC-RCZ	IC50	10674.89	nM	10.6019/CHEMBL1201861
Homo sapiens	Wee1-like protein kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	WM-115	IC50	19677.44	nM	10.6019/CHEMBL1201861
Homo sapiens	WM 266-4	IC50	17420.0	nM	10.1016/j.ejmech.2019.111665
Homo sapiens	YAPC	IC50	32040.73	nM	10.6019/CHEMBL1201861
Homo sapiens	YH-13	IC50	10305.66	nM	10.6019/CHEMBL1201861
Homo sapiens	YKG-1	IC50	21654.52	nM	10.6019/CHEMBL1201861
Homo sapiens	ZR-75-30	IC50	26229.66	nM	10.6019/CHEMBL1201861
Mus musculus	B16-F10	ED50	0.91	ug ml-1	10.1007/s00044-012-0309-2
Mus musculus	BaF3	IC50	10.6	nM	10.1021/acs.jmedchem.2c01041
Mus musculus	BaF3	IC50	12.5	nM	10.1021/acs.jmedchem.2c01041
Mus musculus	BaF3	IC50	21.8	nM	10.1021/acs.jmedchem.2c01041
Mus musculus	BaF3	IC50	53.6	nM	10.1021/acs.jmedchem.2c01041
Mus musculus	BaF3	IC50	54.2	nM	10.1021/acs.jmedchem.2c01041
Mus musculus	BaF3	IC50	1757.0	nM	10.1021/acs.jmedchem.2c01041
Mus musculus	BaF3	IC50	2779.2	nM	10.1021/acs.jmedchem.2c01041
Mus musculus	BaF3	IC50	6981.5	nM	10.1021/acs.jmedchem.2c01041
Mus musculus	Ehrlich	Activity	nan	None	10.1016/j.ejmech.2017.12.022
Mus musculus	Ehrlich	TGI	70.02	%	10.1016/j.ejmech.2017.12.022
Mus musculus	L929	GI	25.95	%	10.1021/acs.jmedchem.8b01612
Mus musculus	L929	IC50	1980.0	nM	10.1021/acs.jmedchem.8b01612
Mus musculus	Lewis lung carcinoma cell line	Activity	nan	None	10.1021/acs.jmedchem.0c00151
Mus musculus	Lewis lung carcinoma cell line	TGI	30.0	%	10.1021/acs.jmedchem.0c00151
Mus musculus	Liver	Stability	90.0	%	10.1016/j.ejmech.2014.11.010
Mus musculus	Mus musculus	Activity	1.77	pg/ml	10.1016/j.bmcl.2021.128238
Mus musculus	Mus musculus	Activity	2.17	pg/ml	10.1016/j.bmcl.2021.128238
Mus musculus	Mus musculus	Activity	2.39	pg/ml	10.1016/j.bmcl.2021.128238
Mus musculus	Mus musculus	Activity	3.39	ug/mg	10.1016/j.bmcl.2021.128238
Mus musculus	Mus musculus	Activity	8.92	nmol/ml	10.1016/j.bmcl.2021.128238
Mus musculus	Mus musculus	Activity	9.7	g	10.1016/j.bmcl.2021.128238
Mus musculus	Mus musculus	Activity	19.4	g	10.1016/j.bmc.2018.08.009
Mus musculus	Mus musculus	Activity	19.6	g	10.1016/j.bmc.2018.08.009
Mus musculus	Mus musculus	Activity	19.9	g	10.1016/j.bmc.2018.08.009
Mus musculus	Mus musculus	Activity	nan	None	10.1016/j.bmc.2015.12.001
Mus musculus	Mus musculus	Activity	nan	None	10.1016/j.bmc.2018.08.009
Mus musculus	Mus musculus	Activity	nan	None	10.1016/j.bmc.2019.115254
Mus musculus	Mus musculus	Activity	nan	None	10.1016/j.bmcl.2021.128238
Mus musculus	Mus musculus	Activity	nan	None	10.1021/acs.jmedchem.6b01489
Mus musculus	Mus musculus	Activity	nan	None	10.1021/jm401117t
Mus musculus	Mus musculus	Activity	nan	None	10.1021/ml4002437
Mus musculus	Mus musculus	AUC	35171.82	ng.hr.mL-1	10.1016/j.bmcl.2006.06.054
Mus musculus	Mus musculus	AUC	38389.57	ng.hr.mL-1	10.1016/j.bmcl.2006.06.054
Mus musculus	Mus musculus	Cmax	6700.0	nM	10.1016/j.bmcl.2006.06.054
Mus musculus	Mus musculus	Cmax	8100.0	nM	10.1016/j.bmcl.2006.06.054
Mus musculus	Mus musculus	Concentration	5.7	uM	10.1016/s0960-894x(01)00344-4
Mus musculus	Mus musculus	Concentration	6.8	uM	10.1016/s0960-894x(01)00344-4
Mus musculus	Mus musculus	Concentration	38.0	uM	10.1016/s0960-894x(01)00344-4
Mus musculus	Mus musculus	Cp	0.01	uM	10.1016/j.bmcl.2006.06.054
Mus musculus	Mus musculus	Cp	0.13	uM	10.1016/j.bmcl.2006.06.054
Mus musculus	Mus musculus	Cp	0.15	uM	10.1016/j.bmcl.2006.06.054
Mus musculus	Mus musculus	Cp	0.26	uM	10.1016/j.bmcl.2006.06.054
Mus musculus	Mus musculus	Fu	0.03	None	10.1016/j.bmcl.2006.06.054
Mus musculus	Mus musculus	Inhibition	nan	%	10.1021/acs.jmedchem.6b00883
Mus musculus	NIH3T3	IC50	540.0	nM	10.1016/j.bmcl.2009.05.060
Mus musculus	Serine/threonine-protein kinase MST2	Kd	nan	None	10.1038/nbt1068
Mus musculus	ULK3 kinase	Kd	1400.0	nM	10.1038/nbt1068
Mycobacterium tuberculosis	Mycobacterium tuberculosis	Activity	nan	None	10.1016/j.bmcl.2019.07.012
Mycobacterium tuberculosis	Mycobacterium tuberculosis	Ratio	1.05	None	10.1016/j.bmcl.2019.07.012
Mycobacterium tuberculosis	Mycobacterium tuberculosis	Ratio	1.08	None	10.1016/j.bmcl.2019.07.012
Mycobacterium tuberculosis	Mycobacterium tuberculosis	Ratio	1.09	None	10.1016/j.bmcl.2019.07.012
Mycobacterium tuberculosis	Serine/threonine-protein kinase pknB	Kd	10000.0	nM	10.1038/nbt.1990
Plasmodium falciparum	Calcium-dependent protein kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Plasmodium falciparum	Plasmodium falciparum	Potency	535.8	nM	None
Plasmodium falciparum	Plasmodium falciparum	Potency	1694.4	nM	None
Plasmodium falciparum (isolate 3D7)	Cell division control protein 2 homolog	Kd	10000.0	nM	10.1038/nbt.1990
Rattus norvegicus	Androgen Receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Rattus norvegicus	Blood	AUC	14260.9	ng.hr.mL-1	10.1021/acs.jmedchem.5b01073
Rattus norvegicus	Blood	Fu	0.033	None	10.1021/acs.jmedchem.5b01073
Rattus norvegicus	Brain	AUC	2523.7	ng.hr.mL-1	10.1021/acs.jmedchem.5b01073
Rattus norvegicus	Brain	Fu	0.0039	None	10.1021/acs.jmedchem.5b01073
Rattus norvegicus	Cerebrospinal fluid	AUC	41.56	ng.hr.mL-1	10.1021/acs.jmedchem.5b01073
Rattus norvegicus	Cyclooxygenase-1	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Rattus norvegicus	GABA receptor alpha-1 subunit	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Rattus norvegicus	Glutamate (NMDA) receptor subunit zeta 1	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Rattus norvegicus	Liver	IC50	nan	None	10.1002/hep.27206
Rattus norvegicus	Peripheral myelin protein 22	Potency	36125.4	nM	None
Rattus norvegicus	Plasma	Fu	0.033	None	10.1016/j.bmcl.2006.06.054
Rattus norvegicus	Rattus norvegicus	ALB	33000.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALB	34000.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALB	36000.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALB	36300.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALB	38000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALB	38000.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALB	39000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALB	40000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALB	42000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALBGLOB	2.4	None	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALBGLOB	2.5	None	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALBGLOB	2.6	None	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALBGLOB	2.7	None	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALBGLOB	2.8	None	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	264.0	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALP	296.0	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALP	348.0	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALP	361.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALP	369.0	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALP	417.83	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALP	1061.5	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1162.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1266.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1267.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1287.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1338.6	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1407.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1488.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1548.6	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1562.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1581.8	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1590.6	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1618.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1643.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1687.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALP	1878.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	35.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	39.6	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	41.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	42.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	42.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	44.5	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	44.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALT	47.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALT	48.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	50.0	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALT	51.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	52.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	52.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALT	53.8	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	55.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	ALT	56.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	56.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	58.6	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	59.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	71.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	ALT	76.8	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	67.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	71.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	71.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	72.8	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	73.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	73.8	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	75.8	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	77.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	78.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	78.6	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	80.8	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	82.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	82.8	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	83.0	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	AST	86.17	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	AST	87.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AST	93.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	AST	94.0	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	AST	107.33	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	AST	118.0	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	AST	126.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	AUC	143.01	ng.hr.mL-1	10.1016/j.bmcl.2006.06.054
Rattus norvegicus	Rattus norvegicus	AUC	490.6	ng.hr.mL-1	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	AUC	500.8	ng.hr.mL-1	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	AUC	2356.79	ng.hr.mL-1	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	AUC	2371.1	ng.hr.mL-1	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	AUMC	1261.5	hr2.ng/ml	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	AUMC	5903.9	hr2.ng/ml	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	AUMCt	1098.0	hr2.ng/ml	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	AUMCt	5649.7	hr2.ng/ml	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	BASOLE	0.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILDIR	0.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILDIR	0.02	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILDIR	0.04	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILDIR	0.08	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILDIR	0.1	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILDIR	0.12	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILDIR	0.16	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILDIR	0.18	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILDIR	0.24	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILDIR	0.28	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILDIR	0.3	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	0.1	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	0.18	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	0.2	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	0.22	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	0.48	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	0.58	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	0.66	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	0.72	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	0.74	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	0.76	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	0.78	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	0.92	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	1.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BILI	3.7	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	BILI	4.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	BILI	4.3	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	BILI	5.5	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	BUN	105.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	108.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	112.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	113.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	114.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	116.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	123.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	126.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	130.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	135.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	148.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	152.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	153.3	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	BUN	160.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	163.3	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	BUN	166.7	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	BUN	173.3	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	BUN	177.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	BUN	180.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	BUN	229.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	C0	714.8	ng/ml	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	CALCIUM	96.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CALCIUM	97.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CALCIUM	98.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CALCIUM	99.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CALCIUM	101.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CALCIUM	103.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CALCIUM	105.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CALCIUM	106.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CALCIUM	107.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CALCIUM	108.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHLORIDE	98.17	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CHLORIDE	100.33	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CHLORIDE	104.83	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CHLORIDE	108.0	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CHLORIDE	108.67	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CHOL	668.3	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CHOL	790.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	796.7	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CHOL	798.3	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CHOL	816.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	853.3	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CHOL	854.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	872.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	890.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CHOL	908.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	912.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	930.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	936.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	953.3	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CHOL	960.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	970.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	980.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	996.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	1046.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	1112.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CHOL	1264.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CK	299.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CK	307.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CK	340.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CK	383.17	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CK	392.83	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CK	512.0	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	Cl	99.8	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	100.8	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	101.1	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	101.5	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	102.1	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	102.2	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	103.1	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	103.6	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	103.8	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	103.9	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	104.2	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	104.3	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	104.4	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	104.7	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Cl	105.2	meq/L	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CL	33.81	mL.min-1.kg-1	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	CL	68.0	mL.min-1.kg-1	10.1016/j.bmcl.2006.06.054
Rattus norvegicus	Rattus norvegicus	CL	70.31	mL.min-1.kg-1	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	Cmax	1390.21	nM	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	Cmax	2691.82	nM	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	CO2	35670000.0	nM	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CO2	36330000.0	nM	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CO2	37330000.0	nM	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CO2	38000000.0	nM	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CO2	38830000.0	nM	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CO2	39000000.0	nM	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CREAT	1.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CREAT	2.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	CREAT	6.8	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CREAT	7.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CREAT	7.2	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	CREAT	7.3	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	EOSLE	0.2	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	EOSLE	0.5	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	EOSLE	0.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	EOSLE	0.8	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	EOSLE	1.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	F	47.4	%	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	F	56.0	%	10.1016/j.bmcl.2006.06.054
Rattus norvegicus	Rattus norvegicus	GGT	0.9	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GGT	1.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GGT	1.1	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GGT	1.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GGT	1.3	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GGT	1.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1380.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	GLUC	1533.3	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	GLUC	1565.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	GLUC	1570.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	GLUC	1640.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	GLUC	1650.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	GLUC	1746.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1776.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1782.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1822.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1825.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1840.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1882.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1884.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1892.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1894.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1926.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1930.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1946.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	1994.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	GLUC	2100.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	36.1	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	36.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	37.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	37.2	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	37.3	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	37.4	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	38.5	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	39.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	39.9	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	40.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	40.1	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	40.5	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	40.7	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HCT	42.62	%	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	HCT	45.2	%	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	HCT	46.2	%	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	HCT	46.33	%	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	HCT	46.77	%	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	HCT	46.82	%	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	HGB	121000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HGB	122000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HGB	123000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HGB	124000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HGB	125000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HGB	126000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HGB	128000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HGB	129000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HGB	130700.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	HGB	131000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HGB	132000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HGB	134000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	HGB	138300.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	HGB	139300.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	HGB	142000.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	HGB	142300.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	HGB	142700.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LDH	142.6	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	145.5	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	160.6	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	169.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	178.6	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	183.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	184.6	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	188.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	191.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	200.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	200.6	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	210.6	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	215.2	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	220.4	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	236.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	272.0	IU.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LDH	373.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LDH	423.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LDH	426.17	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LDH	426.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LDH	519.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LDH	875.0	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LIPASE	4.0	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LIPASE	4.83	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LIPASE	5.33	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LIPASE	10.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LIPASE	11.67	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LIPASE	16.0	U.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	LYMLE	59.8	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	66.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	66.2	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	68.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	74.2	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	74.4	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	75.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	76.2	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	76.4	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	77.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	78.4	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	78.5	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	79.4	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	80.2	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	LYMLE	83.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCH	20.37	pg	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCH	20.55	pg	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCH	20.6	pg	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCH	20.7	pg	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCH	20.73	pg	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCH	20.8	pg	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCH	20.8	pg	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCH	20.9	pg	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCH	21.0	pg	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCH	21.1	pg	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCH	21.17	pg	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCH	21.3	pg	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCH	21.4	pg	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCH	21.47	pg	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCH	21.5	pg	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCHC	32.1	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCHC	32.3	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCHC	32.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCHC	33.1	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCHC	33.2	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCHC	33.4	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCHC	33.5	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCHC	33.8	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCHC	296000.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCHC	303800.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCHC	306200.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCHC	307000.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCHC	308300.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCHC	308700.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCV	62.6	fL	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCV	62.9	fL	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCV	63.0	fL	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCV	63.1	fL	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCV	63.4	fL	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCV	64.1	fL	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCV	64.3	fL	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCV	64.4	fL	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCV	64.5	fL	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCV	64.6	fL	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCV	64.9	fL	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MCV	66.37	fL	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCV	67.23	fL	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCV	67.62	fL	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCV	68.57	fL	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCV	70.05	fL	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MCV	70.3	fL	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	MONOLE	2.4	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MONOLE	2.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MONOLE	3.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MONOLE	3.2	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MONOLE	3.4	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MONOLE	3.5	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MONOLE	3.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MONOLE	4.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	MRT	2.4	hr	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	MRT	2.49	hr	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	MRT(t)	2.12	hr	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	MRT(t)	2.4	hr	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	NEUTLE	12.8	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	15.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	15.8	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	16.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	17.2	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	17.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	18.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	18.8	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	20.4	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	21.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	21.4	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	21.8	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	27.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	28.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	29.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	NEUTLE	35.8	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	74.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	82.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	84.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	86.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	87.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	88.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	89.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	91.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	92.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	95.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	96.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	100.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOS	103.7	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	PHOS	108.7	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	PHOS	110.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	PHOS	110.3	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	PHOS	110.7	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	PHOS	118.7	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1396.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1410.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1428.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1448.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1454.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1460.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1474.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1482.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1486.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1495.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1508.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1528.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1530.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1588.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1660.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PHOSLPD	1862.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1035000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1074000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1078000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1098000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1108000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1109000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1118000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1129000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1160000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1167000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1170000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1197000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1249000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1265000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1290000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PLAT	1325000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	POTASSIUM	3.5	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	POTASSIUM	3.8	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	POTASSIUM	3.9	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	POTASSIUM	4.0	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	POTASSIUM	4.1	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	POTASSIUM	4.2	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	POTASSIUM	4.3	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	POTASSIUM	4.4	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	POTASSIUM	5.57	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	POTASSIUM	6.03	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	POTASSIUM	6.17	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	POTASSIUM	6.33	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	POTASSIUM	6.7	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	POTASSIUM	6.72	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	PROT	53000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PROT	53700.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	PROT	54000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PROT	55000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PROT	56300.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	PROT	57000.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	PROT	59700.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	PROT	60700.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	PROT	63000.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	PROT	63200.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	RBC	5772000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	5792000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	5820000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	5870000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	5880000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	5892000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	5910000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	5926000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	6012000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	6090000.0	cells.uL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	RBC	6102000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	6110000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	6198000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	6236000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	6256000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	6320000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	6350000.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RBC	6590000.0	cells.uL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	RBC	6650000.0	cells.uL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	RBC	6900000.0	cells.uL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	RBC	6930000.0	cells.uL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	RBC	6960000.0	cells.uL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	RETIRBC	7.6	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RETIRBC	8.1	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RETIRBC	8.2	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RETIRBC	8.8	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RETIRBC	8.9	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RETIRBC	9.0	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RETIRBC	9.1	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RETIRBC	9.2	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RETIRBC	9.3	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RETIRBC	9.4	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	RETIRBC	9.7	%	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	138.0	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	SODIUM	139.67	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	SODIUM	140.7	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	141.0	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	SODIUM	141.3	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	141.5	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	141.6	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	141.8	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	141.9	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	142.1	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	142.5	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	142.6	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	142.8	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	142.9	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	143.1	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	143.2	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	143.4	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	143.6	mEq.L-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	SODIUM	146.67	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	SODIUM	148.67	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	SODIUM	151.33	mEq.L-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	T1/2	2.17	hr	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	T1/2	2.39	hr	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	T1/2	7.0	hr	10.1016/j.bmcl.2006.06.054
Rattus norvegicus	Rattus norvegicus	TERMBW	204.0	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	210.0	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	210.3	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	210.7	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	211.6	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	212.3	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	212.6	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	212.8	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	213.7	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	214.3	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	214.5	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	215.0	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	215.5	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	216.0	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TERMBW	223.4	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Tissue Severity Score	nan	None	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	Tissue Severity Score	nan	None	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	Tmax	0.033	hr	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	Tmax	1.0	hr	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	TRIG	290.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	300.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	314.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	390.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	396.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	399.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	428.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	467.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	497.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	565.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	642.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	650.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	673.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	694.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	782.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	TRIG	1227.0	ug.mL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	URATE	0.0	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	URATE	0.167	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	URATE	0.333	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	URATE	0.833	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	URATE	2.3	ug.mL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	Vd	6.678	L.kg-1	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	Vd	13.24	L.kg-1	10.1021/acs.jmedchem.6b01489
Rattus norvegicus	Rattus norvegicus	Vdss	5.8	L.kg-1	10.1016/j.bmcl.2006.06.054
Rattus norvegicus	Rattus norvegicus	Vdss	8.0	L.kg-1	10.1016/j.bmcl.2006.06.054
Rattus norvegicus	Rattus norvegicus	WBC	7880.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	8090.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	8180.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	8190.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	8470.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	8660.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	8710.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	9180.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	9320.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	9470.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	9530.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	9740.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	10110.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	10150.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	10230.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	12730.0	cells.uL-1	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WBC	12830.0	cells.uL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	WBC	13220.0	cells.uL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	WBC	13430.0	cells.uL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	WBC	13950.0	cells.uL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	WBC	14500.0	cells.uL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	WBC	14790.0	cells.uL-1	10.6019/CHEMBL3885881
Rattus norvegicus	Rattus norvegicus	WEIGHT	0.9	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	1.0	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	1.8	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	1.9	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	2.0	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	8.6	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	8.9	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	9.0	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	9.1	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	9.2	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	9.4	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	9.5	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	9.6	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	9.7	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	10.2	g	10.6019/CHEMBL3885861
Rattus norvegicus	Rattus norvegicus	WEIGHT	10.6	g	10.6019/CHEMBL3885861
Rattus norvegicus	Tubulin alpha-1 chain	Kd	410.0	nM	10.1038/nbt1358
Saccharomyces cerevisiae	Saccharomyces cerevisiae	IZ	2.0	mm	10.1016/j.ejmech.2010.07.050
Saccharomyces cerevisiae	Saccharomyces cerevisiae	IZ	9.0	mm	10.1016/j.ejmech.2010.07.050
Severe acute respiratory syndrome coronavirus 2	Replicase polyprotein 1ab	Inhibition	19.63	%	10.6019/CHEMBL4495564
Severe acute respiratory syndrome coronavirus 2	SARS-CoV-2	Hit score	0.178	None	10.1101/2020.04.21.054387
Severe acute respiratory syndrome coronavirus 2	SARS-CoV-2	IC50	19952.62	nM	10.6019/CHEMBL4651402
Severe acute respiratory syndrome coronavirus 2	SARS-CoV-2	IC50	20000.0	nM	10.6019/CHEMBL4651402
Severe acute respiratory syndrome coronavirus 2	SARS-CoV-2	Inhibition	9.07	%	10.6019/CHEMBL4495565
Severe acute respiratory syndrome coronavirus 2	SARS-CoV-2	Inhibition	18.82	%	10.21203/rs.3.rs-23951/v1
Severe acute respiratory syndrome coronavirus 2	SARS-CoV-2	Inhibition index	0.2901	None	10.1101/2020.04.03.023846
Staphylococcus aureus	Quinolone resistance protein norA	FC	8.0	None	10.1021/acs.jmedchem.6b01439
Staphylococcus aureus	Quinolone resistance protein norA	FC	16.0	None	10.1021/acs.jmedchem.6b01439
Staphylococcus aureus	Quinolone resistance protein norA	IC50	9700.0	nM	10.1021/acs.jmedchem.6b01439
Staphylococcus aureus	Quinolone resistance protein norA	Inhibition	94.2	%	10.1021/acs.jmedchem.6b01439
Staphylococcus aureus	Staphylococcus aureus	Activity	nan	None	10.1021/acs.jmedchem.6b01439
Staphylococcus aureus	Staphylococcus aureus	GI	nan	None	10.1021/acs.jmedchem.6b01439
Toxoplasma gondii	Toxoplasma gondii	IC50	20000.0	nM	10.1021/acs.jmedchem.1c01569
Trypanosoma cruzi	Cruzipain	IC50	88000.0	nM	10.1021/jm100254w
Trypanosoma cruzi	Cruzipain	IC50	148000.0	nM	10.1021/jm100254w
Vaccinia virus	Vaccinia virus	EC50	4900.0	nM	10.1021/acs.jmedchem.0c01467
None	ADMET	Activity	nan	None	10.1016/j.ejmech.2020.113022
None	ADMET	Activity	nan	None	10.1021/acs.jmedchem.8b01612
None	ADMET	Activity	nan	None	10.1124/dmd.112.050054
None	ADMET	AUC	7722.0	ng.hr.mL-1	10.1016/j.ejmech.2020.112640
None	ADMET	AUC	7803.0	ng.hr.mL-1	10.1016/j.ejmech.2020.112640
None	ADMET	CC50	280600.0	nM	10.1016/j.bmcl.2014.03.072
None	ADMET	CL	12.0	mL.min-1.kg-1	10.1124/dmd.108.020479
None	ADMET	CL	21.83	mL.min-1.kg-1	10.1016/j.ejmech.2020.112640
None	ADMET	Drug uptake	2.4	uM	10.1016/j.ejmech.2018.11.029
None	ADMET	Drug uptake	271.0	uM	10.1016/j.ejmech.2018.11.029
None	ADMET	IC50	1601.0	nM	10.1016/j.ejmech.2013.05.026
None	ADMET	IC50	10000.0	nM	10.1021/jm201591k
None	ADMET	IC50	12710.0	nM	10.1016/j.ejmech.2014.02.032
None	ADMET	IC50	12710.0	nM	10.1021/jm400463q
None	ADMET	IC50	13940.0	nM	10.1021/jm400463q
None	ADMET	IC50	30000.0	nM	10.1021/jm500873e
None	ADMET	IC50	55080.0	nM	10.1039/C2MD20078C
None	ADMET	IC50	77000.0	nM	10.1124/dmd.112.050054
None	ADMET	Kp	1.85	None	10.1016/j.ejmech.2020.112640
None	ADMET	K(p,uu,brain)	0.02	None	10.1021/acs.jmedchem.6b00618
None	ADMET	K(p,uu,brain)	0.021	None	10.1021/acs.jmedchem.5b01073
None	ADMET	K(p,uu,CSF)	0.088	None	10.1021/acs.jmedchem.5b01073
None	ADMET	K(p,uu,CSF)	0.09	None	10.1021/acs.jmedchem.6b00618
None	ADMET	MRT	4.54	hr	10.1016/j.ejmech.2020.112640
None	ADMET	MRT	32.0	hr	10.1124/dmd.108.020479
None	ADMET	Papp	4.2	10'-6 cm/s	10.1021/acs.jmedchem.5b01073
None	ADMET	Papp	8.3	10'-6 cm/s	10.1021/acs.jmedchem.5b01073
None	ADMET	Ratio	3.0	None	10.1021/acs.jmedchem.5b01073
None	ADMET	Ratio	18.0	None	10.1021/acs.jmedchem.5b01073
None	ADMET	Ratio IC50	2.0	None	10.1016/j.ejmech.2021.113984
None	ADMET	T1/2	0.3752	hr	10.1016/j.ejmech.2020.112640
None	ADMET	T1/2	0.6667	hr	10.1021/acs.jmedchem.6b00883
None	ADMET	T1/2	1.683	hr	10.1021/acs.jmedchem.6b00883
None	ADMET	T1/2	3.75	hr	10.1021/acs.jmedchem.6b00883
None	ADMET	T1/2	3.85	hr	10.1016/j.ejmech.2020.112640
None	ADMET	T1/2	34.0	hr	10.1124/dmd.108.020479
None	ADMET	TI	0.45	None	10.1016/j.bmc.2013.10.007
None	ADMET	TI	0.8	None	10.1016/j.ejmech.2018.10.026
None	ADMET	Vdss	5.93	L.kg-1	10.1016/j.ejmech.2020.112640
None	ADMET	Vdss	23.0	L.kg-1	10.1124/dmd.108.020479
None	DNA	K	2.41	10^5/M	10.1016/j.ejmech.2020.112640
None	Hepatotoxicity	Hepatotoxicity	nan	None	10.1021/tx900326k
None	Hepatotoxicity	Hepatotoxicity	nan	None	10.1124/dmd.110.035113
None	Hepatotoxicity	HepSE_bilirubinemia	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_cholecystitis	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_cholelithiasis	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_cirrhosis	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_Combined Scores	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_elevated liver function tests	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_hepatic failure	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_hepatic necrosis	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_hepatitis	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_hepatomegaly	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_jaundice	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_liver disease	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_liver fatty	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_liver function tests abnormal	0.0	None	10.1371/journal.pcbi.1002310
None	Molecular identity unknown	Activity	nan	None	10.1016/j.bmc.2013.10.007
None	NON-PROTEIN TARGET	Activity	nan	None	10.1021/jm100607r
None	NON-PROTEIN TARGET	EC50	nan	None	10.1021/jm500873e
None	NON-PROTEIN TARGET	Fu	0.089	None	10.1124/dmd.108.020479
None	NON-PROTEIN TARGET	Fu	0.322	None	10.1016/j.bmcl.2013.08.008
None	NON-PROTEIN TARGET	GI	nan	None	10.1016/j.bmc.2013.07.032
None	NON-PROTEIN TARGET	IC50	1.5	nM	10.1021/jm301365e
None	NON-PROTEIN TARGET	IC50	5.81	nM	10.1021/jm401045n
None	NON-PROTEIN TARGET	IC50	6.0	nM	10.1016/j.ejmech.2013.05.026
None	NON-PROTEIN TARGET	IC50	6.0	nM	10.1016/j.ejmech.2014.02.032
None	NON-PROTEIN TARGET	IC50	6.0	nM	10.1021/jm400463q
None	NON-PROTEIN TARGET	IC50	8.0	nM	10.1021/jm201591k
None	NON-PROTEIN TARGET	IC50	10.8	nM	10.1021/jm8010542
None	NON-PROTEIN TARGET	IC50	12.0	nM	10.1016/j.bmcl.2013.07.049
None	NON-PROTEIN TARGET	IC50	12.0	nM	10.1021/jm1000198
None	NON-PROTEIN TARGET	IC50	13.0	nM	10.1016/j.ejmech.2016.01.045
None	NON-PROTEIN TARGET	IC50	13.0	nM	10.1021/jm100607r
None	NON-PROTEIN TARGET	IC50	33.0	nM	10.1016/j.bmc.2015.04.055
None	NON-PROTEIN TARGET	IC50	41.0	nM	10.1039/C2MD20078C
None	NON-PROTEIN TARGET	IC50	63.0	nM	10.1016/j.bmc.2016.05.063
None	NON-PROTEIN TARGET	IC50	530.0	nM	10.1016/j.ejmech.2016.04.026
None	NON-PROTEIN TARGET	IC50	990.0	nM	10.1016/j.bmcl.2013.12.079
None	NON-PROTEIN TARGET	IC50	1240.0	nM	10.1016/j.bmc.2016.05.063
None	NON-PROTEIN TARGET	IC50	2200.0	nM	10.1016/j.bmcl.2015.03.022
None	NON-PROTEIN TARGET	IC50	3308.0	nM	10.1016/j.bmc.2016.09.001
None	NON-PROTEIN TARGET	IC50	4160.0	nM	10.1016/j.bmcl.2016.04.032
None	NON-PROTEIN TARGET	IC50	5000.0	nM	None
None	NON-PROTEIN TARGET	IC50	5360.0	nM	10.1039/C3MD00118K
None	NON-PROTEIN TARGET	IC50	10000.0	nM	10.1016/j.bmcl.2015.06.076
None	NON-PROTEIN TARGET	IC50	10890.0	nM	10.1016/j.bmc.2016.09.001
None	NON-PROTEIN TARGET	IC50	13940.0	nM	10.1016/j.ejmech.2014.02.032
None	NON-PROTEIN TARGET	IC50	16330.0	nM	10.1016/j.bmc.2016.05.063
None	NON-PROTEIN TARGET	IC50	18210.0	nM	10.1016/j.ejmech.2013.06.055
None	NON-PROTEIN TARGET	IC50	20000.0	nM	10.1021/jm500007h
None	NON-PROTEIN TARGET	IC50	21000.0	nM	10.1021/np500385b
None	NON-PROTEIN TARGET	IC50	23760.0	nM	10.1016/j.bmc.2016.09.001
None	NON-PROTEIN TARGET	IC50	26190.0	nM	10.1016/j.ejmech.2015.10.045
None	NON-PROTEIN TARGET	IC50	29430.0	nM	10.1016/j.bmc.2016.09.001
None	NON-PROTEIN TARGET	IC50	nan	None	10.1016/j.bmcl.2011.01.137
None	NON-PROTEIN TARGET	IC50	nan	None	10.1039/C0MD00183J
None	NON-PROTEIN TARGET	ID50	28.0	nM	None
None	NON-PROTEIN TARGET	ID50	206.0	nM	None
None	NON-PROTEIN TARGET	Inhibition	nan	%	10.1016/j.bmcl.2014.09.056
None	NON-PROTEIN TARGET	Potency	472.8	nM	None
None	NON-PROTEIN TARGET	Potency	2728.2	nM	None
None	NON-PROTEIN TARGET	Ratio IC50/EC50	0.857	None	10.1021/jm500873e
None	NON-PROTEIN TARGET	Ratio IC50/EC50	1.2	None	10.1021/jm500873e
None	NON-PROTEIN TARGET	TGI	142.0	%	10.1021/acsmedchemlett.6b00058
None	NON-PROTEIN TARGET	TGI	nan	None	10.1021/jm301365e
None	No relevant target	Activity	160.1	nm	10.1021/jm100254w
None	No relevant target	Activity	250.0	uM	10.1021/jm100254w
None	No relevant target	Activity	nan	None	10.1016/j.ejmech.2018.11.029
None	No relevant target	LogD	2.41	None	10.1021/acsmedchemlett.8b00270
None	No relevant target	LogP	3.2	None	10.1016/j.ejmech.2009.12.043
None	No relevant target	pKa	5.5	None	10.1124/dmd.112.050278
None	No relevant target	pKa	7.2	None	10.1016/j.bmcl.2006.06.054
None	No relevant target	solubility	nan	None	10.1021/acs.jmedchem.6b01774
None	No relevant target	Solubility	2.1	ug.mL-1	10.1016/j.bmcl.2013.07.049
None	No relevant target	Solubility	4000.0	nM	10.1016/j.bmcl.2006.06.054
None	No relevant target	Solubility	10000.0	nM	10.1021/acsmedchemlett.8b00270
None	No relevant target	Solubility	1400000.0	nM	10.1021/acsmedchemlett.8b00270
None	No relevant target	t1/2	nan	None	10.1016/j.ejmech.2018.11.029
None	Unchecked	Ac50	1.413	uM	None
None	Unchecked	Ac50	2.512	uM	None
None	Unchecked	Ac50	2.818	uM	None
None	Unchecked	Ac50	7.079	uM	None
None	Unchecked	Ac50	7.689	uM	None
None	Unchecked	Ac50	9.68	uM	None
None	Unchecked	Ac50	12.19	uM	None
None	Unchecked	Ac50	15.85	uM	None
None	Unchecked	AC50	1412.5	nM	None
None	Unchecked	AC50	2511.9	nM	None
None	Unchecked	AC50	2818.4	nM	None
None	Unchecked	AC50	7079.5	nM	None
None	Unchecked	AC50	15848.9	nM	None
None	Unchecked	AC50	15850.0	nM	None
None	Unchecked	Activity	30.0	%	10.1021/acsmedchemlett.8b00270
None	Unchecked	Activity	nan	None	10.1016/j.ejmech.2010.07.050
None	Unchecked	Activity	nan	None	10.1016/j.ejmech.2022.114231
None	Unchecked	EC50	14.0	nM	10.1021/acs.jmedchem.6b01626
None	Unchecked	GI50	7810.0	nM	10.1016/j.bmcl.2016.05.047
None	Unchecked	IC50	15.0	nM	10.1021/acs.jmedchem.0c00870
None	Unchecked	IC50	15.0	nM	10.1021/jm400072p
None	Unchecked	IC50	190.0	nM	10.1038/nchembio.117
None	Unchecked	IC50	590.2	nM	None
None	Unchecked	IC50	990.0	nM	10.1016/j.bmcl.2016.08.007
None	Unchecked	IC50	1400.0	nM	10.1021/acs.jmedchem.9b00350
None	Unchecked	IC50	1500.0	nM	10.1038/nchembio.117
None	Unchecked	IC50	1794.0	nM	10.1021/acs.jmedchem.0c00870
None	Unchecked	IC50	2421.4	nM	None
None	Unchecked	IC50	2882.0	nM	10.1021/acs.jmedchem.0c00870
None	Unchecked	IC50	3118.0	nM	None
None	Unchecked	IC50	4389.6	nM	None
None	Unchecked	IC50	5000.0	nM	10.1016/j.ejmech.2019.111607
None	Unchecked	IC50	6480.0	nM	10.1016/j.bmc.2018.02.023
None	Unchecked	IC50	7253.0	nM	None
None	Unchecked	IC50	8200.0	nM	10.1016/j.bmcl.2017.03.094
None	Unchecked	IC50	9680.0	nM	10.1021/acs.jmedchem.8b00035
None	Unchecked	IC50	9700.0	nM	10.1021/acs.jmedchem.6b01774
None	Unchecked	IC50	10000.0	nM	10.1016/j.ejmech.2020.113102
None	Unchecked	IC50	10000.0	nM	10.1021/acsmedchemlett.8b00270
None	Unchecked	IC50	10000.0	nM	None
None	Unchecked	IC50	17640.0	nM	10.1016/j.bmc.2017.03.032
None	Unchecked	IC50	18400.0	nM	10.1016/j.bmcl.2021.128238
None	Unchecked	IC50	20000.0	nM	10.1021/acs.jmedchem.9b00350
None	Unchecked	IC50	20000.0	nM	None
None	Unchecked	IC50	23000.0	nM	10.1016/j.bmcl.2019.07.012
None	Unchecked	IC50	23000.0	nM	10.1021/acs.jmedchem.9b00350
None	Unchecked	IC50	23800.0	nM	10.1016/j.bmc.2018.11.009
None	Unchecked	IC50	23800.0	nM	10.1016/j.ejmech.2017.03.083
None	Unchecked	IC50	23800.0	nM	10.1016/j.ejmech.2020.112640
None	Unchecked	IC50	28600.0	nM	10.1016/j.ejmech.2019.111966
None	Unchecked	IC50	30780.0	nM	10.1016/j.ejmech.2017.07.005
None	Unchecked	IC50	38760.0	nM	10.1016/j.ejmech.2021.113589
None	Unchecked	IC50	40780.0	nM	10.1016/j.bmcl.2021.127987
None	Unchecked	IC50	42950.0	nM	10.1016/j.ejmech.2021.113589
None	Unchecked	IC50	50000.0	nM	10.1021/acs.jmedchem.9b00350
None	Unchecked	IC50	51180.0	nM	10.1016/j.ejmech.2021.113589
None	Unchecked	IC50	100000.0	nM	10.1016/j.bmcl.2017.08.035
None	Unchecked	IC50	nan	None	10.1016/j.ejmech.2018.06.061
None	Unchecked	IC50	nan	None	10.1016/j.ejmech.2020.112661
None	Unchecked	IC50	nan	None	10.1016/j.ejmech.2022.114231
None	Unchecked	INH	2.8	uM	10.1021/acsmedchemlett.0c00159
None	Unchecked	INH	3.3	uM	10.1021/acsmedchemlett.0c00159
None	Unchecked	INH	5.4	uM	10.1021/acsmedchemlett.0c00159
None	Unchecked	INH	13.2	uM	10.1021/acsmedchemlett.0c00159
None	Unchecked	INH	14.9	uM	10.1021/acsmedchemlett.0c00159
None	Unchecked	Inhibition	51.3	%	10.1021/acs.jmedchem.6b01774
None	Unchecked	Inhibition	nan	%	10.1016/j.ejmech.2014.02.032
None	Unchecked	Inhibition	nan	%	10.1021/acs.jmedchem.6b01774
None	Unchecked	Inhibition	nan	%	10.1021/acs.jmedchem.9b00722
None	Unchecked	Kd	0.8	nM	10.1021/acs.jmedchem.9b01566
None	Unchecked	Kd	30000.0	nM	10.1126/science.aan4368
None	Unchecked	LC50	63100.0	nM	10.1016/j.bmcl.2016.05.047
None	Unchecked	Potency	3317.3	nM	None
None	Unchecked	Potency	4176.3	nM	None
None	Unchecked	Potency	14818.0	nM	None
None	Unchecked	Potency	17782.8	nM	None
None	Unchecked	Potency	18818.0	nM	None
None	Unchecked	Potency	25118.9	nM	None
None	Unchecked	Potency	29565.9	nM	None
None	Unchecked	Potency	33173.4	nM	None
None	Unchecked	Potency	36125.4	nM	None
None	Unchecked	Potency	37221.2	nM	None
None	Unchecked	Ratio EC50	0.2	None	10.1021/acs.jmedchem.7b00515
None	Unchecked	RatioGI50	0.9	None	10.1021/acs.jmedchem.6b01774
None	Unchecked	RatioGI50	1.2	None	10.1016/j.bmcl.2018.11.010
None	Unchecked	RatioGI50	1.4	None	10.1021/acs.jmedchem.6b01774
None	Unchecked	RatioGI50	3.1	None	10.1021/acs.jmedchem.6b01774
None	Unchecked	RatioGI50	4.7	None	10.1021/acs.jmedchem.6b01774
None	Unchecked	Ratio IC50	0.009	None	10.1016/j.bmc.2017.03.032
None	Unchecked	Ratio IC50	0.019	None	10.1016/j.bmc.2018.11.009
None	Unchecked	Ratio IC50	0.019	None	10.1016/j.ejmech.2017.03.083
None	Unchecked	Ratio IC50	0.02	None	10.1021/jm400822z
None	Unchecked	Ratio IC50	0.1	None	10.1016/j.bmc.2018.11.009
None	Unchecked	Ratio IC50	0.1	None	10.1021/acs.jmedchem.7b00515
None	Unchecked	Ratio IC50	0.88	None	10.1016/j.bmc.2017.03.039
None	Unchecked	Ratio IC50	4.5	None	10.1016/j.bmcl.2017.08.063
None	Unchecked	Ratio IC50	nan	None	10.1016/j.ejmech.2020.112661
None	Unchecked	Ratio IC50	nan	None	10.1016/j.ejmech.2022.114231
None	Unchecked	Ratio Ki	50.0	None	10.1016/j.chembiol.2005.04.011
None	Unchecked	Selectivity ratio	0.019	None	10.1016/j.ejmech.2020.112640
None	Unchecked	TGI	25100.0	nM	10.1016/j.bmcl.2016.05.047