| Acinetobacter baumannii |
Acinetobacter baumannii |
GI |
nan |
None |
10.1016/j.bmc.2013.06.013 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Inhibition |
7.52 |
% |
10.6019/CHEMBL4513156 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
Inhibition |
18.82 |
% |
10.6019/CHEMBL4513141 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
20000.0 |
nM |
10.6019/CHEMBL4513161 |
| Acinetobacter baumannii |
Acinetobacter baumannii |
MIC |
nan |
None |
10.1016/j.ejmech.2019.04.067 |
| Agaricus bisporus |
Tyrosinase |
IC50 |
1000000.0 |
nM |
10.1016/j.ejmech.2015.10.033 |
| Agaricus bisporus |
Tyrosinase |
KSV |
1.7 |
10'3/M |
10.1016/j.ejmech.2015.10.033 |
| Artemia |
Artemia |
LD50 |
1074.75 |
ug ml-1 |
10.1016/j.ejmech.2011.11.014 |
| Arthrobacter sp. |
Arthrobacter sp. |
MIC |
150.0 |
ug.mL-1 |
10.1007/s00044-013-0488-5 |
| Aspergillus niger |
Aspergillus niger |
-logMIC |
2.04 |
None |
10.1007/s00044-011-9662-9 |
| Aspergillus niger |
Aspergillus niger |
-logMIC |
2.04 |
None |
10.1007/s00044-011-9705-2 |
| Bacillus spizizenii |
Bacillus spizizenii |
MIC |
nan |
None |
10.1016/j.ejmech.2019.01.062 |
| Bacillus spizizenii |
Bacillus spizizenii |
MIC90 |
nan |
None |
10.1016/j.ejmech.2017.12.089 |
| Bacillus subtilis |
4'-phosphopantetheinyl transferase ffp |
Potency |
50118.7 |
nM |
None |
| Bacillus subtilis |
Bacillus subtilis |
IZ |
nan |
None |
10.1016/j.bmcl.2008.07.087 |
| Bacillus subtilis |
Bacillus subtilis |
-logMIC |
1.74 |
None |
10.1007/s00044-011-9662-9 |
| Bacillus subtilis |
Bacillus subtilis |
-logMIC |
1.74 |
None |
10.1007/s00044-011-9705-2 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
150.0 |
ug.mL-1 |
10.1007/s00044-013-0488-5 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
nan |
None |
10.1016/j.bmc.2008.03.062 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
nan |
None |
10.1016/j.bmcl.2008.07.087 |
| Bacillus subtilis |
Bacillus subtilis |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Bacteria |
Cell membrane |
Activity |
nan |
None |
10.1039/d2md00251e |
| Bordetella bronchiseptica |
Bordetella bronchiseptica |
DIZ |
nan |
None |
10.1016/j.ejmech.2011.11.014 |
| Bos taurus |
Progesterone receptor |
IC50 |
nan |
None |
None |
| Bos taurus |
Progesterone receptor |
Ki |
nan |
None |
None |
| Candida albicans |
Candida albicans |
Inhibition |
0.98 |
% |
10.6019/CHEMBL4513156 |
| Candida albicans |
Candida albicans |
Inhibition |
3.95 |
% |
10.6019/CHEMBL4513141 |
| Candida albicans |
Candida albicans |
-logMIC |
2.34 |
None |
10.1007/s00044-011-9662-9 |
| Candida albicans |
Candida albicans |
-logMIC |
2.34 |
None |
10.1007/s00044-011-9705-2 |
| Candida albicans |
Candida albicans |
MIC |
20000.0 |
nM |
10.6019/CHEMBL4513161 |
| Candida albicans |
Candida albicans |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Candida albicans |
Candida albicans |
MIC |
nan |
None |
10.1016/j.bmcl.2013.11.024 |
| Candida albicans |
Candida albicans |
MIC |
nan |
None |
10.1016/j.bmcl.2014.05.018 |
| Candida albicans |
Candida albicans |
MIC90 |
nan |
None |
10.1021/acs.jmedchem.7b00793 |
| Canis lupus familiaris |
MDCK |
CC50 |
nan |
None |
10.1039/C5MD00178A |
| Canis lupus familiaris |
MDCK |
MCC |
nan |
None |
10.1039/C5MD00178A |
| Cavia porcellus |
Cavia porcellus |
AUC |
18.22 |
None |
10.1128/aac.00196-08 |
| Cavia porcellus |
Histamine H1 receptor |
pKb |
nan |
None |
10.1016/j.bmc.2008.10.042 |
| Cavia porcellus |
Leukotriene C4 synthase |
IC50 |
nan |
None |
None |
| Cavia porcellus |
Leukotriene C4 synthase |
Ki |
nan |
None |
None |
| Cavia porcellus |
Serotonin 4 (5-HT4) receptor |
IC50 |
nan |
None |
None |
| Cavia porcellus |
Serotonin 4 (5-HT4) receptor |
Ki |
nan |
None |
None |
| Chlorocebus sabaeus |
Vero |
Activity |
100.0 |
uM |
10.1016/j.bmcl.2022.128604 |
| Chlorocebus sabaeus |
Vero |
Activity |
nan |
None |
10.1016/j.ejmech.2010.04.017 |
| Chlorocebus sabaeus |
Vero |
Activity |
nan |
None |
10.1016/j.ejmech.2011.06.037 |
| Chlorocebus sabaeus |
Vero |
CC50 |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.080 |
| Chlorocebus sabaeus |
Vero |
CC50 |
50.0 |
ug.mL-1 |
10.1021/jm300123s |
| Chlorocebus sabaeus |
Vero |
CC50 |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.041 |
| Chlorocebus sabaeus |
Vero |
CC50 |
125.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.07.023 |
| Chlorocebus sabaeus |
Vero |
CC50 |
125.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.05.057 |
| Chlorocebus sabaeus |
Vero |
CC50 |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.090 |
| Chlorocebus sabaeus |
Vero |
CC50 |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.07.025 |
| Chlorocebus sabaeus |
Vero |
CC50 |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.07.057 |
| Chlorocebus sabaeus |
Vero |
CC50 |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.01.042 |
| Chlorocebus sabaeus |
Vero |
CC50 |
50000.0 |
nM |
10.1016/j.ejmech.2020.112859 |
| Chlorocebus sabaeus |
Vero |
CC50 |
256000.0 |
nM |
10.1016/j.bmc.2019.04.017 |
| Chlorocebus sabaeus |
Vero |
CC50 |
256000.0 |
nM |
10.1016/j.ejmech.2018.09.049 |
| Chlorocebus sabaeus |
Vero |
CC50 |
455730.0 |
nM |
10.1016/j.bmcl.2010.06.096 |
| Chlorocebus sabaeus |
Vero |
CC50 |
455730.0 |
nM |
10.1016/j.bmcl.2011.01.122 |
| Chlorocebus sabaeus |
Vero |
CC50 |
455730.0 |
nM |
10.1016/j.bmcl.2011.07.062 |
| Chlorocebus sabaeus |
Vero |
CC50 |
455800.0 |
nM |
10.1007/s00044-011-9638-9 |
| Chlorocebus sabaeus |
Vero |
CC50 |
455800.0 |
nM |
10.1016/j.ejmech.2008.02.031 |
| Chlorocebus sabaeus |
Vero |
CC50 |
500000.0 |
nM |
10.1016/j.bmcl.2010.08.127 |
| Chlorocebus sabaeus |
Vero |
CC50 |
500000.0 |
nM |
10.1016/j.bmcl.2011.04.072 |
| Chlorocebus sabaeus |
Vero |
CC50 |
1459850.0 |
nM |
10.1016/j.bmcl.2011.08.076 |
| Chlorocebus sabaeus |
Vero |
CC50 |
6282800.0 |
nM |
10.1016/j.ejmech.2010.11.023 |
| Chlorocebus sabaeus |
Vero |
CC50 |
7000000.0 |
nM |
10.1016/j.bmcl.2016.05.053 |
| Chlorocebus sabaeus |
Vero |
CC50 |
7300000.0 |
nM |
10.1016/j.bmcl.2019.07.025 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.bmc.2012.09.019 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.bmc.2014.12.060 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.bmc.2019.01.022 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.bmc.2022.116777 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.ejmech.2014.07.051 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.ejmech.2017.05.044 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.ejmech.2019.111595 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1016/j.ejmech.2021.113398 |
| Chlorocebus sabaeus |
Vero |
CC50 |
nan |
None |
10.1021/acsmedchemlett.7b00299 |
| Chlorocebus sabaeus |
Vero |
IC50 |
6.25 |
ug.mL-1 |
10.1016/j.bmcl.2017.05.050 |
| Chlorocebus sabaeus |
Vero |
IC50 |
12.0 |
ug.mL-1 |
10.1007/s00044-012-0074-2 |
| Chlorocebus sabaeus |
Vero |
IC50 |
62.5 |
ug.mL-1 |
10.1016/j.bmcl.2009.10.034 |
| Chlorocebus sabaeus |
Vero |
IC50 |
62.5 |
ug.mL-1 |
10.1016/j.bmcl.2009.12.045 |
| Chlorocebus sabaeus |
Vero |
IC50 |
62.5 |
ug.mL-1 |
10.1016/j.bmcl.2012.06.047 |
| Chlorocebus sabaeus |
Vero |
IC50 |
62.5 |
ug.mL-1 |
10.1016/j.bmcl.2012.10.059 |
| Chlorocebus sabaeus |
Vero |
IC50 |
62.5 |
ug.mL-1 |
10.1016/j.bmcl.2012.12.069 |
| Chlorocebus sabaeus |
Vero |
IC50 |
62.5 |
ug.mL-1 |
10.1016/j.ejmech.2014.03.085 |
| Chlorocebus sabaeus |
Vero |
IC50 |
62.5 |
ug.mL-1 |
10.1021/jm060339h |
| Chlorocebus sabaeus |
Vero |
IC50 |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2022.117006 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100.0 |
ug.mL-1 |
10.1021/np400497f |
| Chlorocebus sabaeus |
Vero |
IC50 |
200.0 |
ug.mL-1 |
10.1016/j.bmc.2007.08.064 |
| Chlorocebus sabaeus |
Vero |
IC50 |
200.0 |
ug.mL-1 |
10.1016/j.bmc.2018.07.034 |
| Chlorocebus sabaeus |
Vero |
IC50 |
256.0 |
ug.mL-1 |
10.1021/acs.jmedchem.7b00582 |
| Chlorocebus sabaeus |
Vero |
IC50 |
500.0 |
ug.mL-1 |
10.1016/j.ejmech.2009.01.017 |
| Chlorocebus sabaeus |
Vero |
IC50 |
1000.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.02.012 |
| Chlorocebus sabaeus |
Vero |
IC50 |
1000.0 |
ug.mL-1 |
10.1016/s0960-894x(00)00058-5 |
| Chlorocebus sabaeus |
Vero |
IC50 |
1000.0 |
ug.mL-1 |
10.1021/jm020891g |
| Chlorocebus sabaeus |
Vero |
IC50 |
39800.0 |
nM |
10.1016/j.bmc.2007.05.053 |
| Chlorocebus sabaeus |
Vero |
IC50 |
50000.0 |
nM |
10.1016/j.bmc.2016.12.038 |
| Chlorocebus sabaeus |
Vero |
IC50 |
50000.0 |
nM |
10.1021/acs.jnatprod.9b01095 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100000.0 |
nM |
10.1016/j.bmcl.2013.06.069 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100000.0 |
nM |
10.1016/j.bmcl.2013.11.024 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100000.0 |
nM |
10.1016/j.ejmech.2010.09.048 |
| Chlorocebus sabaeus |
Vero |
IC50 |
100000.0 |
nM |
10.1016/j.ejmech.2013.01.017 |
| Chlorocebus sabaeus |
Vero |
IC50 |
128000.0 |
nM |
10.1007/s00044-007-9073-0 |
| Chlorocebus sabaeus |
Vero |
IC50 |
128000.0 |
nM |
10.1016/j.bmc.2012.02.025 |
| Chlorocebus sabaeus |
Vero |
IC50 |
128000.0 |
nM |
10.1016/j.bmcl.2013.09.013 |
| Chlorocebus sabaeus |
Vero |
IC50 |
128000.0 |
nM |
10.1021/jm900003c |
| Chlorocebus sabaeus |
Vero |
IC50 |
128000.0 |
nM |
10.1021/jm900513a |
| Chlorocebus sabaeus |
Vero |
IC50 |
130500.0 |
nM |
10.1016/j.ejmech.2010.05.035 |
| Chlorocebus sabaeus |
Vero |
IC50 |
200000.0 |
nM |
10.1016/j.ejmech.2014.04.077 |
| Chlorocebus sabaeus |
Vero |
IC50 |
450000.0 |
nM |
10.1007/s00044-011-9646-9 |
| Chlorocebus sabaeus |
Vero |
IC50 |
450000.0 |
nM |
10.1007/s00044-012-0112-0 |
| Chlorocebus sabaeus |
Vero |
IC50 |
450000.0 |
nM |
10.1016/j.ejmech.2013.11.004 |
| Chlorocebus sabaeus |
Vero |
IC50 |
450000.0 |
nM |
10.1016/j.ejmech.2015.03.013 |
| Chlorocebus sabaeus |
Vero |
IC50 |
454700.0 |
nM |
10.1016/j.bmcl.2005.11.004 |
| Chlorocebus sabaeus |
Vero |
IC50 |
455690.0 |
nM |
10.1016/j.bmcl.2021.127810 |
| Chlorocebus sabaeus |
Vero |
IC50 |
455770.0 |
nM |
10.1016/j.bmcl.2007.01.037 |
| Chlorocebus sabaeus |
Vero |
IC50 |
455800.0 |
nM |
10.1016/j.bmc.2007.11.016 |
| Chlorocebus sabaeus |
Vero |
IC50 |
455800.0 |
nM |
10.1016/j.bmc.2007.11.050 |
| Chlorocebus sabaeus |
Vero |
IC50 |
455800.0 |
nM |
10.1016/j.bmcl.2007.11.110 |
| Chlorocebus sabaeus |
Vero |
IC50 |
455800.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Chlorocebus sabaeus |
Vero |
IC50 |
455800.0 |
nM |
10.1016/j.ejmech.2009.09.033 |
| Chlorocebus sabaeus |
Vero |
IC50 |
455800.0 |
nM |
10.1021/jm700999n |
| Chlorocebus sabaeus |
Vero |
IC50 |
456000.0 |
nM |
10.1016/j.ejmech.2011.09.035 |
| Chlorocebus sabaeus |
Vero |
IC50 |
7000000.0 |
nM |
10.1021/jm020891g |
| Chlorocebus sabaeus |
Vero |
IC50 |
nan |
None |
10.1016/j.bmcl.2012.05.096 |
| Chlorocebus sabaeus |
Vero |
IC50 |
nan |
None |
10.1016/j.bmcl.2014.05.018 |
| Chlorocebus sabaeus |
Vero |
IC50 |
nan |
None |
10.1016/j.ejmech.2013.09.039 |
| Chlorocebus sabaeus |
Vero |
IC50 |
nan |
None |
10.1021/acsmedchemlett.5b00176 |
| Chlorocebus sabaeus |
Vero |
IC50 |
nan |
None |
10.1021/jm4003878 |
| Chlorocebus sabaeus |
Vero |
IC50 |
nan |
None |
10.1021/np400391p |
| Chlorocebus sabaeus |
Vero |
Maximal non-toxic dose 50 |
32.0 |
ug ml-1 |
10.1021/jm0602662 |
| Chlorocebus sabaeus |
Vero |
MCC |
nan |
None |
10.1039/C5MD00178A |
| Chlorocebus sabaeus |
Vero |
MIC |
128000.0 |
nM |
10.1021/jm901112f |
| Chlorocebus sabaeus |
Vero |
MIC |
128000.0 |
nM |
10.1021/jm901273n |
| Chlorocebus sabaeus |
Vero |
MNCC |
6.25 |
ug ml-1 |
10.1016/j.bmc.2016.09.044 |
| Chlorocebus sabaeus |
Vero |
MNTD50 |
32.0 |
ug ml-1 |
10.1021/jm701560p |
| Chlorocebus sabaeus |
Vero |
MTD50 |
32.0 |
ug ml-1 |
10.1016/s0960-894x(98)00248-0 |
| Chlorocebus sabaeus |
Vero |
MTD50 |
32.0 |
ug ml-1 |
10.1016/s0960-894x(98)00526-5 |
| Chlorocebus sabaeus |
Vero |
MTD50 |
32.0 |
ug ml-1 |
10.1016/s0960-894x(99)00510-7 |
| Chlorocebus sabaeus |
Vero |
PI |
128.0 |
None |
10.1021/jm0602662 |
| Chlorocebus sabaeus |
Vero |
Selective index |
20000.0 |
None |
10.1016/j.bmcl.2005.03.065 |
| Chlorocebus sabaeus |
Vero |
Survival |
98.0 |
% |
10.1016/j.ejmech.2018.03.042 |
| Chlorocebus sabaeus |
Vero |
Survival |
100.0 |
% |
10.1016/j.ejmech.2014.06.019 |
| Chlorocebus sabaeus |
Vero |
Survival |
100.0 |
% |
10.1016/j.ejmech.2015.06.056 |
| Citrobacter koseri |
Citrobacter koseri |
GI |
nan |
None |
10.1016/j.bmc.2013.06.013 |
| Cricetulus griseus |
CHO |
CC50 |
256000.0 |
nM |
10.1016/j.ejmech.2019.111678 |
| Cricetulus griseus |
CHO |
IC50 |
100000.0 |
nM |
10.1016/j.bmc.2017.12.047 |
| Cricetulus griseus |
CHO |
IC50 |
nan |
None |
10.1021/acs.jmedchem.1c00707 |
| Cryptococcus neoformans |
Cryptococcus neoformans |
Inhibition |
-55.93 |
% |
10.6019/CHEMBL4513156 |
| Cryptococcus neoformans |
Cryptococcus neoformans |
Inhibition |
-3.6 |
% |
10.6019/CHEMBL4513141 |
| Cryptococcus neoformans |
Cryptococcus neoformans |
MIC |
20000.0 |
nM |
10.6019/CHEMBL4513161 |
| Electrophorus electricus |
Acetylcholinesterase |
Inhibition |
5.8 |
% |
10.1016/j.bmc.2020.115470 |
| Enterobacter cloacae |
Enterobacter cloacae |
GI |
nan |
None |
10.1016/j.bmc.2013.06.013 |
| Enterococcus faecalis |
Enterococcus faecalis |
GI |
nan |
None |
10.1016/j.bmc.2013.06.013 |
| Enterococcus faecalis |
Enterococcus faecalis |
IZ |
nan |
None |
10.1016/j.bmcl.2008.07.087 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1016/j.bmcl.2008.07.087 |
| Enterococcus faecalis |
Enterococcus faecalis |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Enterococcus faecium |
Enterococcus faecium |
IC50 |
nan |
None |
10.1016/j.ejmech.2019.07.052 |
| Enterococcus faecium |
Enterococcus faecium |
IC50 |
nan |
None |
10.1021/np2006555 |
| Enterococcus faecium |
Enterococcus faecium |
MIC90 |
nan |
None |
10.1021/acs.jmedchem.7b00793 |
| Escherichia coli |
3-oxoacyl-[acyl-carrier-protein] synthase 3 |
IC50 |
1000000.0 |
nM |
10.1016/j.bmc.2019.02.043 |
| Escherichia coli |
DNA gyrase |
IC50 |
1000000.0 |
nM |
10.1016/j.bmc.2019.02.043 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1016/j.ejmech.2009.01.017 |
| Escherichia coli |
Escherichia coli |
Activity |
nan |
None |
10.1128/aac.00453-10 |
| Escherichia coli |
Escherichia coli |
DIZ |
nan |
None |
10.1016/j.ejmech.2011.11.014 |
| Escherichia coli |
Escherichia coli |
GI |
nan |
None |
10.1016/j.bmc.2013.06.013 |
| Escherichia coli |
Escherichia coli |
IC50 |
nan |
None |
10.1016/j.ejmech.2019.07.052 |
| Escherichia coli |
Escherichia coli |
Inhibition |
0.87 |
% |
10.6019/CHEMBL4513141 |
| Escherichia coli |
Escherichia coli |
Inhibition |
20.51 |
% |
10.6019/CHEMBL4513156 |
| Escherichia coli |
Escherichia coli |
Inhibition |
nan |
% |
10.1016/j.bmc.2018.07.034 |
| Escherichia coli |
Escherichia coli |
-logMIC |
1.74 |
None |
10.1007/s00044-011-9662-9 |
| Escherichia coli |
Escherichia coli |
-logMIC |
1.74 |
None |
10.1007/s00044-011-9705-2 |
| Escherichia coli |
Escherichia coli |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| Escherichia coli |
Escherichia coli |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| Escherichia coli |
Escherichia coli |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Escherichia coli |
Escherichia coli |
MIC |
2520.0 |
ug.mL-1 |
10.1007/s00044-013-0488-5 |
| Escherichia coli |
Escherichia coli |
MIC |
20000.0 |
nM |
10.6019/CHEMBL4513161 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.bmc.2008.03.062 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.bmcl.2013.11.024 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.bmcl.2014.05.018 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.ejmech.2019.01.062 |
| Escherichia coli |
Escherichia coli |
MIC |
nan |
None |
10.1016/j.ejmech.2019.04.067 |
| Escherichia coli |
Escherichia coli |
MIC90 |
nan |
None |
10.1016/j.ejmech.2017.12.089 |
| Escherichia coli |
Escherichia coli |
MIC90 |
nan |
None |
10.1021/acs.jmedchem.7b00793 |
| Escherichia coli K-12 |
Phospho-N-acetylmuramoyl-pentapeptide-transferase |
IC50 |
nan |
ug.mL-1 |
10.1016/s0960-894x(03)00597-3 |
| Escherichia coli (strain K12) |
Formamidopyrimidine-DNA glycosylase |
Activity |
nan |
None |
None |
| Escherichia coli (strain K12) |
Formamidopyrimidine-DNA glycosylase |
IC50 |
50000.0 |
nM |
None |
| Homo sapiens |
A549 |
Activity |
3091.0 |
ug ml-1 |
10.1016/j.bmcl.2009.09.095 |
| Homo sapiens |
A549 |
IC50 |
450000.0 |
nM |
10.1007/s00044-012-0112-0 |
| Homo sapiens |
A549 |
IC50 |
450000.0 |
nM |
10.1016/j.ejmech.2013.11.004 |
| Homo sapiens |
A549 |
IC50 |
450000.0 |
nM |
10.1016/j.ejmech.2015.03.013 |
| Homo sapiens |
Acetylcholinesterase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Acetylcholinesterase |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A2a receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A2a receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A2a receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A3 receptor |
AC50 |
32673.8 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A3 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A3 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1d adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-1d adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2b adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2b adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2b adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2c adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2c adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2c adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Angiotensin II type 2 (AT-2) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Angiotensin II type 2 (AT-2) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
ARPE-19 |
Activity |
nan |
None |
10.1016/j.bmcl.2017.07.019 |
| Homo sapiens |
Beta-1 adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-1 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-1 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-2 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-3 adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-3 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-3 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Bile salt export pump |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Bile salt export pump |
IC50 |
135000.0 |
nM |
10.1093/toxsci/kfq269 |
| Homo sapiens |
Bile salt export pump |
IC50 |
1000000.0 |
nM |
10.1124/dmd.111.040758 |
| Homo sapiens |
Bile salt export pump |
IC50 |
1000000.0 |
nM |
10.1124/dmd.112.047068 |
| Homo sapiens |
Bradykinin B1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bradykinin B2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bradykinin B2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Bradykinin B2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Bromodomain adjacent to zinc finger domain protein 2B |
Potency |
89125.1 |
nM |
None |
| Homo sapiens |
Calcitonin receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Calcitonin receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Canalicular multispecific organic anion transporter 1 |
Activity |
96.0 |
% |
10.1021/jm7015683 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 1 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 2 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Cannabinoid CB1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cannabinoid CB1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cannabinoid CB1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cannabinoid CB1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase II |
IC50 |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase II |
Ki |
nan |
None |
None |
| Homo sapiens |
Caspase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Caspase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cathepsin G |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cathepsin G |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 2 |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 4 |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin A receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cholecystokinin A receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin A receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin B receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Corticotropin releasing factor receptor 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Corticotropin releasing factor receptor 2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cysteinyl leukotriene receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cysteinyl leukotriene receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
AC50 |
6309.57 |
nM |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 1A2 |
Ki |
56000.0 |
nM |
10.2174/138920005774330639 |
| Homo sapiens |
Cytochrome P450 1A2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
Kinact |
0.11 |
min-1 |
10.2174/138920005774330639 |
| Homo sapiens |
Cytochrome P450 2A6 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2A6 |
Ki |
60000.0 |
nM |
10.2174/138920005774330639 |
| Homo sapiens |
Cytochrome P450 2A6 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2A6 |
Kinact |
0.13 |
min-1 |
10.2174/138920005774330639 |
| Homo sapiens |
Cytochrome P450 2C19 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
Ki |
10000.0 |
nM |
10.2174/138920005774330639 |
| Homo sapiens |
Cytochrome P450 2C19 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
Kinact |
0.09 |
min-1 |
10.2174/138920005774330639 |
| Homo sapiens |
Cytochrome P450 2C19 |
Ratio IC50 |
5.0 |
None |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2C8 |
Ki |
170000.0 |
nM |
10.2174/138920005774330639 |
| Homo sapiens |
Cytochrome P450 2C8 |
Ki |
374000.0 |
nM |
10.2174/138920005774330639 |
| Homo sapiens |
Cytochrome P450 2C8 |
Kinact |
0.012 |
min-1 |
10.2174/138920005774330639 |
| Homo sapiens |
Cytochrome P450 2C8 |
Kinact |
0.042 |
min-1 |
10.2174/138920005774330639 |
| Homo sapiens |
Cytochrome P450 2C9 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
FC |
1.0 |
None |
10.1016/j.bmcl.2016.06.088 |
| Homo sapiens |
Cytochrome P450 2C9 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2C9 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
AC50 |
12589.25 |
nM |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
FC |
1.0 |
None |
10.1016/j.bmcl.2016.06.088 |
| Homo sapiens |
Cytochrome P450 2D6 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
Potency |
12589.3 |
nM |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
Ratio IC50 |
5.0 |
None |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2E1 |
Activity |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2E1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2E1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
AC50 |
3981.07 |
nM |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
FC |
1.0 |
None |
10.1016/j.bmcl.2016.06.088 |
| Homo sapiens |
Cytochrome P450 3A4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
Ki |
36000.0 |
nM |
10.2174/138920005774330639 |
| Homo sapiens |
Cytochrome P450 3A4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
Kinact |
0.08 |
min-1 |
10.2174/138920005774330639 |
| Homo sapiens |
Cytochrome P450 3A4 |
Potency |
3981.1 |
nM |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
Potency |
15848.9 |
nM |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
Ratio IC50 |
5.0 |
None |
10.1021/tx300075j |
| Homo sapiens |
Delta opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Delta opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Delta opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
DNA-(apurinic or apyrimidinic site) lyase |
Potency |
1000.0 |
nM |
None |
| Homo sapiens |
Dopamine D1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D3 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D3 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D4 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D4 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D4 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Endonuclease 8-like 1 |
Activity |
80.64 |
% |
None |
| Homo sapiens |
Endonuclease 8-like 1 |
IC50 |
50000.0 |
nM |
None |
| Homo sapiens |
Endonuclease III-like protein 1 |
Activity |
97.95 |
% |
None |
| Homo sapiens |
Endonuclease III-like protein 1 |
IC50 |
50000.0 |
nM |
None |
| Homo sapiens |
Endothelin receptor ET-A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Endothelin receptor ET-A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-A |
Ki |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-B |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Equilibrative nucleoside transporter 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor beta |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor beta |
IC50 |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor beta |
Ki |
nan |
None |
None |
| Homo sapiens |
Gastric inhibitory polypeptide receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Geminin |
Potency |
794.3 |
nM |
None |
| Homo sapiens |
Ghrelin receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucagon receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Glucocorticoid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Glutaminase kidney isoform, mitochondrial |
Potency |
31622.8 |
nM |
None |
| Homo sapiens |
HCT-116 |
IC50 |
nan |
None |
10.1016/j.ejmech.2013.06.042 |
| Homo sapiens |
HCT-116 |
IC50 |
nan |
None |
10.1016/j.ejmech.2013.10.069 |
| Homo sapiens |
HCT-8 |
Activity |
1.95 |
% |
10.1016/j.bmc.2013.06.013 |
| Homo sapiens |
HCT-8 |
Activity |
8.56 |
% |
10.1016/j.bmc.2013.06.013 |
| Homo sapiens |
HCT-8 |
Activity |
15.01 |
% |
10.1016/j.bmc.2013.06.013 |
| Homo sapiens |
HCT-8 |
Activity |
17.9 |
% |
10.1016/j.bmc.2013.06.013 |
| Homo sapiens |
HCT-8 |
Activity |
38.48 |
% |
10.1016/j.bmc.2013.06.013 |
| Homo sapiens |
HCT-8 |
Activity |
44.12 |
% |
10.1016/j.bmc.2013.06.013 |
| Homo sapiens |
HCT-8 |
Activity |
71.5 |
% |
10.1016/j.bmc.2013.06.013 |
| Homo sapiens |
HCT-8 |
Activity |
nan |
None |
10.1016/j.bmc.2013.06.013 |
| Homo sapiens |
HCT-8 |
EC50 |
100000.0 |
nM |
10.1016/j.bmc.2009.12.055 |
| Homo sapiens |
HEK293 |
CC50 |
20000.0 |
nM |
10.6019/CHEMBL4513161 |
| Homo sapiens |
HEK293 |
Inhibition |
nan |
% |
10.1016/j.ejmech.2018.07.047 |
| Homo sapiens |
HEK293 |
LC50 |
200.0 |
ug.mL-1 |
10.1016/j.bmc.2008.10.042 |
| Homo sapiens |
HEK293 |
LC50 |
576.0 |
ug.mL-1 |
10.1016/j.ejmech.2007.06.012 |
| Homo sapiens |
HEK293 |
MIC |
120000.0 |
nM |
10.1016/j.bmc.2019.02.043 |
| Homo sapiens |
HEK-293T |
Activity |
nan |
None |
10.1016/j.bmcl.2012.10.060 |
| Homo sapiens |
HEK-293T |
GI |
nan |
None |
10.1016/j.bmcl.2013.01.031 |
| Homo sapiens |
HEK-293T |
MNTD50 |
32.0 |
ug ml-1 |
10.1016/j.bmcl.2019.01.004 |
| Homo sapiens |
HEL |
MCC |
nan |
None |
10.1039/C5MD00178A |
| Homo sapiens |
HeLa |
MCC |
nan |
None |
10.1039/C5MD00178A |
| Homo sapiens |
HepG2 |
Activity |
10.0 |
% |
10.1016/j.bmcl.2012.02.091 |
| Homo sapiens |
HepG2 |
Activity |
56.13 |
% |
10.1007/s00044-010-9405-3 |
| Homo sapiens |
HepG2 |
Activity |
91.31 |
% |
10.1007/s00044-010-9405-3 |
| Homo sapiens |
HepG2 |
Activity |
99.73 |
% |
10.1007/s00044-010-9405-3 |
| Homo sapiens |
HepG2 |
Activity |
125.47 |
% |
10.1007/s00044-010-9405-3 |
| Homo sapiens |
HepG2 |
Activity |
128.56 |
% |
10.1007/s00044-010-9405-3 |
| Homo sapiens |
HepG2 |
Activity |
200.0 |
ug ml-1 |
10.1016/j.ejmech.2016.09.083 |
| Homo sapiens |
HepG2 |
Activity |
nan |
None |
10.1007/s00044-010-9405-3 |
| Homo sapiens |
HepG2 |
CC50 |
nan |
None |
10.1016/j.ejmech.2011.10.054 |
| Homo sapiens |
HepG2 |
CC50 |
nan |
None |
10.1016/j.ejmech.2014.07.051 |
| Homo sapiens |
HepG2 |
CC50 |
nan |
None |
10.1016/j.ejmech.2015.07.039 |
| Homo sapiens |
HepG2 |
GI |
3.51 |
% |
10.1016/j.bmcl.2011.12.022 |
| Homo sapiens |
HepG2 |
IC50 |
250000.0 |
nM |
10.1016/j.bmc.2014.05.064 |
| Homo sapiens |
HepG2 |
IC50 |
250000.0 |
nM |
10.1016/j.bmc.2014.12.019 |
| Homo sapiens |
HepG2 |
IC50 |
250000.0 |
nM |
10.1016/j.ejmech.2019.111578 |
| Homo sapiens |
HepG2 |
IC50 |
1000000.0 |
nM |
10.1016/j.ejmech.2011.07.052 |
| Homo sapiens |
HepG2 |
IC50 |
1000000.0 |
nM |
10.1016/j.ejmech.2011.09.054 |
| Homo sapiens |
HepG2 |
IC50 |
5000000.0 |
nM |
10.1016/j.ejmech.2018.04.017 |
| Homo sapiens |
HepG2 |
IC50 |
nan |
None |
10.1016/j.bmc.2013.12.016 |
| Homo sapiens |
HepG2 |
IC50 |
nan |
None |
10.1016/j.bmc.2014.12.019 |
| Homo sapiens |
HepG2 |
IC50 |
nan |
None |
10.1016/j.bmcl.2012.11.052 |
| Homo sapiens |
HepG2 |
IC50 |
nan |
None |
10.1016/j.ejmech.2019.111578 |
| Homo sapiens |
HepG2 |
LC50 |
105000.0 |
nM |
10.1016/j.ejmech.2018.01.071 |
| Homo sapiens |
HepG2 |
LC50 |
200000.0 |
nM |
10.1016/j.ejmech.2018.01.071 |
| Homo sapiens |
HERG |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
HERG |
IC50 |
nan |
None |
None |
| Homo sapiens |
HERG |
Inhibition |
nan |
% |
10.1016/j.bmc.2019.01.022 |
| Homo sapiens |
HERG |
Ki |
nan |
None |
None |
| Homo sapiens |
HERG |
Potency |
35481.3 |
nM |
None |
| Homo sapiens |
Histamine H1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Histamine H1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H2 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Histamine H2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histone acetyltransferase GCN5 |
Potency |
15848.9 |
nM |
None |
| Homo sapiens |
Histone deacetylase 6 |
Inhibition |
3.37 |
% |
10.6019/CHEMBL4808148 |
| Homo sapiens |
Histone deacetylase 6 |
Inhibition |
25.98 |
% |
10.6019/CHEMBL4808148 |
| Homo sapiens |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Potency |
22387.2 |
nM |
None |
| Homo sapiens |
HMG-CoA reductase |
IC50 |
nan |
None |
None |
| Homo sapiens |
HMG-CoA reductase |
Ki |
nan |
None |
None |
| Homo sapiens |
Homo sapiens |
Activity |
0.8 |
% |
10.1016/j.ejmech.2009.11.034 |
| Homo sapiens |
Homo sapiens |
Activity |
13.3 |
% |
10.1128/aac.01204-07 |
| Homo sapiens |
Homo sapiens |
AUC |
10350.0 |
ng.hr.mL-1 |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
AUC |
16340.0 |
ng.hr.mL-1 |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
AUC |
19780.0 |
ng.hr.mL-1 |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
AUC |
22900.0 |
ng.hr.mL-1 |
10.1371/journal.pmed.0030466 |
| Homo sapiens |
Homo sapiens |
AUC |
38050.0 |
ng.hr.mL-1 |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
AUC |
42190.0 |
ng.hr.mL-1 |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
AUC |
42240.0 |
ng.hr.mL-1 |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
CL |
7.4 |
L/hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
CL |
7.79 |
L/hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
CL |
8.03 |
L/hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
CL |
16.07 |
L/hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
CL |
19.17 |
L/hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
CL |
30.05 |
L/hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
Cmax |
10062.71 |
nM |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
Cmax |
29094.36 |
nM |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
Cmax |
32813.18 |
nM |
10.1371/journal.pmed.0030466 |
| Homo sapiens |
Homo sapiens |
Cmax |
35948.67 |
nM |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
Cmax |
40761.27 |
nM |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
Cmax |
41709.2 |
nM |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
Cmax |
60376.26 |
nM |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
DILI_Concern |
nan |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
DILI_severity_class |
8.0 |
None |
10.1016/j.drudis.2016.02.015 |
| Homo sapiens |
Homo sapiens |
Drug uptake |
0.4 |
ug ml-1 |
10.1128/aac.01302-08 |
| Homo sapiens |
Homo sapiens |
T1/2 |
0.9 |
hr |
10.1128/aac.00185-07 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.0 |
hr |
10.1007/s00044-012-0101-3 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.06 |
hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.15 |
hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.165 |
hr |
10.1002/jps.2600630804 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.178 |
hr |
10.1002/jps.2600630804 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.35 |
hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.39 |
hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
T1/2 |
1.76 |
hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.0 |
hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.2 |
hr |
10.1128/aac.00185-07 |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.467 |
hr |
10.1002/jps.2600630804 |
| Homo sapiens |
Homo sapiens |
T1/2 |
2.73 |
hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
T1/2 |
3.23 |
hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
T1/2 |
3.267 |
hr |
10.1002/jps.2600630804 |
| Homo sapiens |
Homo sapiens |
T1/2 |
3.59 |
hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
T1/2 |
3.84 |
hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
T1/2 |
6.04 |
hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
T1/2 |
20.0 |
hr |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Homo sapiens |
TIME |
5.611e-06 |
hr |
10.1128/aac.01204-07 |
| Homo sapiens |
Homo sapiens |
Vdss |
0.67 |
L.kg-1 |
10.1016/j.ejmech.2009.06.004 |
| Homo sapiens |
Interleukin-8 receptor A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor A |
Ki |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor B |
IC50 |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor B |
Ki |
nan |
None |
None |
| Homo sapiens |
Kappa opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Kappa opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Kappa opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Leukocyte common antigen |
IC50 |
nan |
None |
None |
| Homo sapiens |
Leukocyte common antigen |
Ki |
nan |
None |
None |
| Homo sapiens |
Leukocyte elastase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Leukocyte elastase |
Ki |
nan |
None |
None |
| Homo sapiens |
Liver |
CLH |
nan |
None |
10.1021/acs.jmedchem.7b00793 |
| Homo sapiens |
Liver |
t1/2 |
nan |
None |
10.1021/acs.jmedchem.7b00793 |
| Homo sapiens |
Liver microsomes |
Activity |
nan |
None |
10.1021/tx300075j |
| Homo sapiens |
Liver microsomes |
Stability |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Lysine-specific demethylase 4D-like |
Potency |
7079.5 |
nM |
None |
| Homo sapiens |
Lysine-specific demethylase 4D-like |
Potency |
35481.3 |
nM |
None |
| Homo sapiens |
Macrophage migration inhibitory factor |
IC50 |
400000.0 |
nM |
10.1016/j.bmcl.2021.128445 |
| Homo sapiens |
MAP kinase ERK1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK1 |
Ki |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK2 |
Ki |
nan |
None |
None |
| Homo sapiens |
MAP kinase p38 alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase p38 alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase 9 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase 9 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 3 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Melanocortin receptor 3 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 3 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 4 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Melanocortin receptor 4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Monoamine oxidase A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Monoamine oxidase A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Monoamine oxidase A |
Ki |
nan |
None |
None |
| Homo sapiens |
Motilin receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
MRC5 |
Activity |
293.0 |
ug ml-1 |
10.1016/j.bmcl.2009.09.095 |
| Homo sapiens |
MRC5 |
Activity |
nan |
None |
10.1016/j.bmc.2010.10.060 |
| Homo sapiens |
MRC5 |
Activity |
nan |
None |
10.1016/j.ejmech.2011.02.062 |
| Homo sapiens |
MRC5 |
CC50 |
10.0 |
ug.mL-1 |
10.1016/j.bmc.2015.07.053 |
| Homo sapiens |
MRC5 |
CC50 |
nan |
None |
10.1016/j.ejmech.2017.06.061 |
| Homo sapiens |
MRC5 |
IC50 |
nan |
None |
10.1016/j.ejmech.2022.114831 |
| Homo sapiens |
MRC5 |
IC50 |
nan |
None |
10.1021/acs.jnatprod.5b00266 |
| Homo sapiens |
MRC5 |
IC90 |
nan |
None |
10.1021/acs.jnatprod.5b00266 |
| Homo sapiens |
MT4 |
CC50 |
100000.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Homo sapiens |
Multidrug resistance-associated protein 4 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Mu opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Mu opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Mu opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Myeloperoxidase |
Activity |
64.0 |
% |
10.1021/acsmedchemlett.6b00417 |
| Homo sapiens |
Myeloperoxidase |
Activity |
98.0 |
% |
10.1021/acsmedchemlett.6b00417 |
| Homo sapiens |
Myeloperoxidase |
IC50 |
4700.0 |
nM |
10.1021/acsmedchemlett.6b00417 |
| Homo sapiens |
Myeloperoxidase |
IC50 |
5000.0 |
nM |
10.1021/acsmedchemlett.6b00417 |
| Homo sapiens |
Myeloperoxidase |
Inhibition |
61.0 |
% |
10.1021/acsmedchemlett.6b00417 |
| Homo sapiens |
Neurokinin 1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neurokinin 1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neurokinin 1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurokinin 2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neurokinin 2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Neuronal acetylcholine receptor protein alpha-4 subunit |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurotensin receptor 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
N-glycosylase/DNA lyase |
Activity |
1.0 |
% |
None |
| Homo sapiens |
N-glycosylase/DNA lyase |
IC50 |
50000.0 |
nM |
None |
| Homo sapiens |
N-glycosylase/DNA lyase |
Inhibition |
nan |
% |
None |
| Homo sapiens |
Norepinephrine transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Norepinephrine transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Norepinephrine transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
PBMC |
Activity |
12.4 |
% |
10.1016/j.bmcl.2005.11.005 |
| Homo sapiens |
PBMC |
IC50 |
87.08 |
ug.mL-1 |
10.1016/j.bmc.2007.05.053 |
| Homo sapiens |
PBMC |
IC50 |
100.0 |
ug.mL-1 |
10.1016/j.bmc.2007.05.053 |
| Homo sapiens |
PBMC |
IC50 |
169.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.04.009 |
| Homo sapiens |
PBMC |
IC50 |
4670000.0 |
nM |
10.1016/j.ejmech.2011.07.052 |
| Homo sapiens |
PBMC |
IC50 |
4670000.0 |
nM |
10.1016/j.ejmech.2011.09.054 |
| Homo sapiens |
PBMC |
Survival |
95.0 |
% |
10.1016/j.bmc.2007.05.053 |
| Homo sapiens |
P-glycoprotein 1 |
Ratio |
nan |
None |
10.1016/j.bmcl.2016.11.010 |
| Homo sapiens |
Phosphodiesterase 3A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 4D |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 5A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Phosphodiesterase 5A |
Ki |
nan |
None |
None |
| Homo sapiens |
Plasma |
fCmax |
76.56 |
uM |
10.1124/dmd.111.040758 |
| Homo sapiens |
Plasma |
Ratio |
0.22 |
None |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Plasma |
Ratio |
1.35 |
None |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Plasma |
Ratio |
3.22 |
None |
10.1515/dmdi.2011.016 |
| Homo sapiens |
Platelet activating factor receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Platelet activating factor receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Pregnane X receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Progesterone receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Protein kinase C alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
Protein kinase C alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 1a (5-HT1a) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 1a (5-HT1a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 3a (5-HT3a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 7 (5-HT7) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Serum albumin |
pKa |
0.05 |
None |
10.1021/acs.jmedchem.0c00046 |
| Homo sapiens |
Serum albumin |
pKa |
nan |
None |
10.1021/acs.jmedchem.0c00046 |
| Homo sapiens |
Serum albumin |
PPB |
6.8 |
% |
10.1021/acs.jmedchem.0c00046 |
| Homo sapiens |
Serum albumin |
PPB |
10.9 |
% |
10.1021/acs.jmedchem.0c00046 |
| Homo sapiens |
SH-SY5Y |
IC50 |
nan |
None |
10.1016/j.ejmech.2011.07.052 |
| Homo sapiens |
Sigma opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Sigma opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Inhibition |
29.9 |
% |
10.1021/jm300212s |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B1 |
Inhibition |
88.4 |
% |
10.1124/mol.112.084152 |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
Inhibition |
18.7 |
% |
10.1021/jm300212s |
| Homo sapiens |
Solute carrier organic anion transporter family member 1B3 |
Inhibition |
98.94 |
% |
10.1124/mol.112.084152 |
| Homo sapiens |
Solute carrier organic anion transporter family member 2B1 |
Inhibition |
23.8 |
% |
10.1021/jm300212s |
| Homo sapiens |
THP-1 |
Activity |
40.0 |
% |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
Activity |
41.0 |
% |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
Activity |
48.0 |
% |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
Activity |
50.0 |
% |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
Activity |
50.0 |
uM |
10.1016/j.ejmech.2020.112772 |
| Homo sapiens |
THP-1 |
Activity |
57.0 |
% |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
Activity |
67.0 |
% |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
Activity |
68.0 |
% |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
Activity |
74.0 |
% |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
Activity |
83.0 |
% |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
Activity |
84.0 |
% |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
Activity |
85.0 |
% |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
Activity |
90.0 |
% |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
Activity |
2145.0 |
ug ml-1 |
10.1016/j.bmcl.2009.09.095 |
| Homo sapiens |
THP-1 |
Cmax |
1.09 |
ug/10^6 cells |
10.1128/aac.00153-08 |
| Homo sapiens |
THP-1 |
Cmax |
1.31 |
ug/10^6 cells |
10.1128/aac.00153-08 |
| Homo sapiens |
THP-1 |
IC20 |
100.0 |
uM |
10.1016/j.bmc.2017.12.047 |
| Homo sapiens |
THP-1 |
IC50 |
25.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111713 |
| Homo sapiens |
THP-1 |
IC50 |
100000.0 |
nM |
10.1016/j.bmcl.2021.128236 |
| Homo sapiens |
THP-1 |
IC50 |
547000.0 |
nM |
10.1016/j.ejmech.2018.02.067 |
| Homo sapiens |
THP-1 |
IC50 |
3649000.0 |
nM |
10.1021/jm101510d |
| Homo sapiens |
THP-1 |
IC50 |
nan |
None |
10.1021/acs.jnatprod.5b00266 |
| Homo sapiens |
THP-1 |
IC90 |
nan |
None |
10.1021/acs.jnatprod.5b00266 |
| Homo sapiens |
THP-1 |
Kel |
0.034 |
/hr |
10.1128/aac.00153-08 |
| Homo sapiens |
THP-1 |
Kel |
0.369 |
/hr |
10.1128/aac.00153-08 |
| Homo sapiens |
Thromboxane A2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Thromboxane-A synthase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Thromboxane-A synthase |
Ki |
nan |
None |
None |
| Homo sapiens |
Type-1 angiotensin II receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Tyrosine-protein kinase FYN |
IC50 |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase FYN |
Ki |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase LCK |
IC50 |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase LCK |
Ki |
nan |
None |
None |
| Homo sapiens |
U-937 |
IC50 |
nan |
None |
10.1021/np800778b |
| Homo sapiens |
Vascular endothelial growth factor receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vascular endothelial growth factor receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasoactive intestinal polypeptide receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vasoactive intestinal polypeptide receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasopressin V1a receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vasopressin V1a receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vasopressin V1a receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasopressin V2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Influenza A virus |
Influenza A virus |
EC50 |
nan |
None |
10.1039/C5MD00178A |
| Klebsiella aerogenes |
Klebsiella aerogenes |
DIZ |
nan |
None |
10.1016/j.ejmech.2011.11.014 |
| Klebsiella aerogenes |
Klebsiella aerogenes |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
GI |
nan |
None |
10.1016/j.bmc.2013.06.013 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
IC50 |
nan |
None |
10.1016/j.ejmech.2019.07.052 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Inhibition |
6.54 |
% |
10.6019/CHEMBL4513141 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
Inhibition |
18.82 |
% |
10.6019/CHEMBL4513156 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
20000.0 |
nM |
10.6019/CHEMBL4513161 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
nan |
None |
10.1016/j.bmcl.2014.05.018 |
| Klebsiella pneumoniae |
Klebsiella pneumoniae |
MIC |
nan |
None |
10.1016/j.ejmech.2019.04.067 |
| Klebsiella sp. |
Klebsiella sp. |
MIC |
250.0 |
ug.mL-1 |
10.1007/s00044-013-0488-5 |
| Leishmania donovani |
Leishmania donovani |
IC50 |
218750.0 |
nM |
10.6019/CHEMBL3392926 |
| Leishmania donovani |
Leishmania donovani |
IC50 |
656260.0 |
nM |
10.6019/CHEMBL3392926 |
| Leishmania donovani |
Leishmania donovani |
IC50 |
729180.0 |
nM |
10.6019/CHEMBL3392926 |
| Listeria monocytogenes |
Listeria monocytogenes |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Mesocricetus auratus |
BHK-21 |
CC50 |
nan |
None |
10.1016/j.ejmech.2011.10.054 |
| Micrococcus luteus |
Micrococcus luteus |
DIZ |
nan |
None |
10.1016/j.ejmech.2011.11.014 |
| Morganella morganii |
Morganella morganii |
GI |
nan |
None |
10.1016/j.bmc.2013.06.013 |
| Morganella morganii |
Morganella morganii |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Mus musculus |
J774 |
IC50 |
nan |
None |
10.1016/j.bmcl.2018.03.021 |
| Mus musculus |
J774.A1 |
Activity |
90.3 |
% |
10.1016/j.ejmech.2018.01.071 |
| Mus musculus |
J774.A1 |
Activity |
97.3 |
% |
10.1016/j.ejmech.2018.01.071 |
| Mus musculus |
J774.A1 |
Activity |
98.2 |
% |
10.1016/j.ejmech.2018.01.071 |
| Mus musculus |
J774.A1 |
Activity |
98.5 |
% |
10.1016/j.ejmech.2018.01.071 |
| Mus musculus |
J774.A1 |
Activity |
98.7 |
% |
10.1016/j.ejmech.2018.01.071 |
| Mus musculus |
J774.A1 |
Activity |
99.5 |
% |
10.1016/j.ejmech.2018.01.071 |
| Mus musculus |
J774.A1 |
CC50 |
nan |
None |
10.1016/j.ejmech.2019.07.052 |
| Mus musculus |
J774.A1 |
IC50 |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2022.117006 |
| Mus musculus |
J774.A1 |
IC50 |
nan |
None |
10.1016/j.bmc.2019.07.045 |
| Mus musculus |
Monoamine oxidase A |
Activity |
nan |
None |
10.1021/jm800656v |
| Mus musculus |
Monoamine oxidase B |
Activity |
nan |
None |
10.1021/jm800656v |
| Mus musculus |
Mus musculus |
Activity |
nan |
None |
10.1016/j.ejmech.2009.05.009 |
| Mus musculus |
Mus musculus |
AUC |
4550.0 |
ng.hr.mL-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
CL |
4.43 |
ml/hr |
10.1128/aac.00153-08 |
| Mus musculus |
Mus musculus |
CL |
63.9 |
ml/hr |
10.1128/aac.00153-08 |
| Mus musculus |
Mus musculus |
Cmax |
22312.96 |
nM |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cmax |
280005833.45 |
nM |
10.1021/jm050765n |
| Mus musculus |
Mus musculus |
Cp |
0.253 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cp |
0.74 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cp |
1.92 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cp |
2.17 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cp |
2.28 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Cp |
3.06 |
ug ml-1 |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Drug uptake |
1.64 |
ug ml-1 |
10.1128/aac.00897-07 |
| Mus musculus |
Mus musculus |
Drug uptake |
13.12 |
ug ml-1 |
10.1128/aac.00897-07 |
| Mus musculus |
Mus musculus |
F |
80.0 |
% |
10.1021/jm050765n |
| Mus musculus |
Mus musculus |
IC50 |
nan |
None |
10.1016/j.ejmech.2016.07.039 |
| Mus musculus |
Mus musculus |
Inhibition |
12.16 |
% |
10.1016/j.bmc.2016.09.012 |
| Mus musculus |
Mus musculus |
Inhibition |
45.9 |
% |
10.1016/j.bmcl.2010.06.125 |
| Mus musculus |
Mus musculus |
Inhibition |
nan |
% |
10.1016/j.ejmech.2016.08.034 |
| Mus musculus |
Mus musculus |
LD50 |
100.0 |
mg.kg-1 |
10.1016/j.bmcl.2016.03.107 |
| Mus musculus |
Mus musculus |
LD50 |
133.0 |
mg.kg-1 |
10.1016/j.bmc.2016.06.020 |
| Mus musculus |
Mus musculus |
LD50 |
133.0 |
mg.kg-1 |
10.1016/j.bmcl.2014.05.006 |
| Mus musculus |
Mus musculus |
LD50 |
133.0 |
mg.kg-1 |
10.1016/j.bmcl.2017.05.013 |
| Mus musculus |
Mus musculus |
LD50 |
133.0 |
mg.kg-1 |
10.1016/j.ejmech.2015.05.007 |
| Mus musculus |
Mus musculus |
LD50 |
151.0 |
mg.kg-1 |
10.1016/j.bmc.2016.06.020 |
| Mus musculus |
Mus musculus |
LD50 |
151.0 |
mg.kg-1 |
10.1016/j.bmcl.2014.05.006 |
| Mus musculus |
Mus musculus |
LD50 |
151.0 |
mg.kg-1 |
10.1016/j.bmcl.2017.05.013 |
| Mus musculus |
Mus musculus |
LD50 |
151.0 |
mg.kg-1 |
10.1016/j.ejmech.2015.05.007 |
| Mus musculus |
Mus musculus |
MTD |
1000.0 |
mg Kg-1 |
10.1016/j.ejmech.2009.05.009 |
| Mus musculus |
Mus musculus |
Survival |
100.0 |
% |
10.1016/j.ejmech.2011.06.037 |
| Mus musculus |
Mus musculus |
Survival |
100.0 |
% |
10.1021/jm00143a011 |
| Mus musculus |
Mus musculus |
T1/2 |
1.0 |
hr |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
T1/2 |
nan |
None |
10.1021/jm050765n |
| Mus musculus |
Mus musculus |
Tmax |
0.25 |
hr |
10.1371/journal.pmed.0030466 |
| Mus musculus |
Mus musculus |
Tmax |
nan |
None |
10.1021/jm050765n |
| Mus musculus |
Mus musculus |
Vz |
41.34 |
ml |
10.1128/aac.00153-08 |
| Mus musculus |
Mus musculus |
Vz |
16667.78 |
ml |
10.1128/aac.00153-08 |
| Mus musculus |
NIH3T3 |
LC50 |
nan |
None |
10.1016/j.ejmech.2019.05.013 |
| Mus musculus |
Nitric oxide synthase, inducible |
IC50 |
nan |
None |
None |
| Mus musculus |
Nitric oxide synthase, inducible |
Ki |
nan |
None |
None |
| Mus musculus |
Nuclear receptor ROR-gamma |
Potency |
14125.4 |
nM |
None |
| Mus musculus |
Peritoneal macrophage |
Activity |
200.0 |
ug ml-1 |
10.1016/j.ejmech.2016.09.083 |
| Mus musculus |
Plasma |
Cmax |
17281.61 |
nM |
10.1128/aac.00153-08 |
| Mus musculus |
Plasma |
Cmax |
23625.49 |
nM |
10.1128/aac.00153-08 |
| Mus musculus |
RAW264.7 |
Activity |
nan |
None |
10.1016/j.bmc.2017.12.044 |
| Mus musculus |
RAW264.7 |
Activity |
nan |
None |
10.1016/j.ejmech.2017.12.088 |
| Mus musculus |
RAW264.7 |
CC50 |
150000.0 |
nM |
10.1016/j.ejmech.2020.112908 |
| Mus musculus |
RAW264.7 |
CC50 |
nan |
None |
10.1016/j.ejmech.2019.111812 |
| Mus musculus |
RAW264.7 |
GI |
93.21 |
% |
10.1016/j.bmc.2017.03.053 |
| Mus musculus |
RAW264.7 |
GI |
nan |
None |
10.1016/j.bmc.2015.03.004 |
| Mus musculus |
RAW264.7 |
GI |
nan |
None |
10.1016/j.bmc.2017.11.031 |
| Mus musculus |
RAW264.7 |
GI |
nan |
None |
10.1016/j.bmcl.2017.01.026 |
| Mus musculus |
RAW264.7 |
GI |
nan |
None |
10.1016/j.ejmech.2014.02.028 |
| Mus musculus |
RAW264.7 |
GI |
nan |
None |
10.1016/j.ejmech.2018.07.046 |
| Mus musculus |
RAW264.7 |
GI50 |
3000.0 |
ug.mL-1 |
10.1016/j.bmc.2015.04.001 |
| Mus musculus |
RAW264.7 |
GI50 |
21900000.0 |
nM |
10.1039/C3MD00251A |
| Mus musculus |
RAW264.7 |
GI50 |
nan |
None |
10.1016/j.ejmech.2018.07.046 |
| Mus musculus |
RAW264.7 |
GI50 |
nan |
None |
10.1021/acs.jmedchem.6b00031 |
| Mus musculus |
RAW264.7 |
IC50 |
400.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.04.009 |
| Mus musculus |
RAW264.7 |
IC50 |
nan |
None |
10.1016/j.ejmech.2022.114831 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.bmc.2014.01.030 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.bmc.2014.05.038 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.bmc.2014.06.041 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.bmc.2014.10.016 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.bmc.2015.02.032 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.bmc.2016.01.011 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.bmc.2016.01.059 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.ejmech.2014.09.028 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.ejmech.2014.12.046 |
| Mus musculus |
RAW264.7 |
Inhibition |
nan |
% |
10.1016/j.ejmech.2015.06.032 |
| Mus musculus |
Serum |
AUC |
16640.0 |
ng.hr.mL-1 |
10.1128/aac.00153-08 |
| Mus musculus |
Serum |
AUC |
55340.0 |
ng.hr.mL-1 |
10.1128/aac.00153-08 |
| Mus musculus |
Serum |
T1/2 |
3.91 |
hr |
10.1128/aac.00153-08 |
| Mus musculus |
Serum |
T1/2 |
18.62 |
hr |
10.1128/aac.00153-08 |
| Mus musculus |
Tyrosinase |
Inhibition |
97.0 |
% |
10.1016/j.ejmech.2015.10.033 |
| Mus musculus |
Tyrosinase |
Inhibition |
100.0 |
% |
10.1016/j.ejmech.2015.10.033 |
| Mus musculus |
Tyrosinase |
Inhibition |
102.0 |
% |
10.1016/j.ejmech.2015.10.033 |
| Mus musculus |
Tyrosinase |
Inhibition |
104.0 |
% |
10.1016/j.ejmech.2015.10.033 |
| Mycobacterium |
Mycobacterium |
MIC50 |
1400.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycobacterium |
Mycobacterium |
MIC90 |
4700.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycobacterium avium |
Mycobacterium avium |
Activity |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Mycobacterium avium |
Mycobacterium avium |
Activity |
nan |
None |
10.1021/np970182j |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2014.05.006 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.107 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2016.04.017 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
1.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00596-1 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
1.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00597-3 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
3.13 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
3.13 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.bmcl.2013.04.021 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.bmcl.2013.12.054 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
6.25 |
ug.mL-1 |
10.1039/C8MD00056E |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.bmcl.2007.02.024 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.bmcl.2013.12.054 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.084 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.085 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.04.021 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
25.0 |
ug.mL-1 |
10.1021/jm070638m |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
32.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00248-0 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
32.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00526-5 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
32.0 |
ug.mL-1 |
10.1016/s0960-894x(99)00510-7 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00972 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm0602662 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
32.0 |
ug.mL-1 |
10.1021/jm701560p |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.083 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
730.0 |
nM |
10.1016/j.bmc.2016.06.020 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
730.0 |
nM |
10.1016/j.ejmech.2015.05.007 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
23000.0 |
nM |
10.1016/j.bmcl.2012.11.052 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
46000.0 |
nM |
10.1016/j.bmcl.2012.11.052 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
62500.0 |
nM |
10.1039/D1MD00239B |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
116000.0 |
nM |
10.1016/j.bmcl.2016.05.053 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
200000.0 |
nM |
10.1016/j.ejmech.2012.07.044 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2007.01.051 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2007.02.021 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2009.04.008 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2009.12.055 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2010.10.017 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2013.12.016 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2014.05.064 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2014.12.019 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2015.10.029 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2017.01.016 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2017.01.045 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.bmcl.2017.10.050 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2008.06.027 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2010.02.037 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2010.09.040 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2011.07.052 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2011.09.054 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2012.01.060 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2012.07.044 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2012.08.016 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2016.11.041 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2018.04.017 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2019.111578 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2021.113668 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1016/s0960-894x(02)00697-2 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
250000.0 |
nM |
10.1039/C4MD00301B |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
500000.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
nan |
ug.mL-1 |
10.1016/s0960-894x(00)00159-1 |
| Mycobacterium avium |
Mycobacterium avium |
MIC |
nan |
None |
10.1016/j.bmc.2013.10.011 |
| Mycobacterium avium |
Mycobacterium avium |
MIC90 |
100.0 |
nM |
10.1016/j.ejmech.2017.06.061 |
| Mycobacterium avium |
Mycobacterium avium |
MIC>99 |
250.0 |
uM |
10.1016/j.bmc.2017.08.010 |
| Mycobacterium avium |
Mycobacterium avium |
MIC>99 |
250.0 |
uM |
10.1016/j.ejmech.2017.02.058 |
| Mycobacterium avium |
Mycobacterium avium |
MIC>99 |
250.0 |
uM |
10.1021/acs.jmedchem.5b00608 |
| Mycobacterium avium |
Mycobacterium avium |
MIC>99 |
250.0 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium avium complex sp. |
Mycobacterium avium complex sp. |
MIC |
256.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.083 |
| Mycobacterium avium complex sp. |
Mycobacterium avium complex sp. |
MIC=>90 |
3646.0 |
uM |
10.1016/j.bmc.2015.03.018 |
| Mycobacterium avium subsp. paratuberculosis |
Mycobacterium avium subsp. paratuberculosis |
MIC |
990.0 |
nM |
10.1021/jm401735w |
| Mycobacterium avium subsp. paratuberculosis |
Mycobacterium avium subsp. paratuberculosis |
MIC50 |
100.0 |
nM |
10.1016/j.ejmech.2013.03.023 |
| Mycobacterium avium subsp. paratuberculosis |
Mycobacterium avium subsp. paratuberculosis |
MIC=>90 |
1823.0 |
uM |
10.1016/j.bmc.2015.03.018 |
| Mycobacterium gordonae |
Mycobacterium gordonae |
MIC |
32.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00248-0 |
| Mycobacterium gordonae |
Mycobacterium gordonae |
MIC |
32.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00526-5 |
| Mycobacterium gordonae |
Mycobacterium gordonae |
MIC |
32.0 |
ug.mL-1 |
10.1016/s0960-894x(99)00510-7 |
| Mycobacterium gordonae |
Mycobacterium gordonae |
MIC |
116000.0 |
nM |
10.1016/j.bmcl.2016.05.053 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
Activity |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
IC50 |
nan |
None |
10.1021/np900281r |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
6.25 |
ug.mL-1 |
10.1021/jm00150a006 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.084 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.085 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
8.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00596-1 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
8.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00597-3 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
12.5 |
ug.mL-1 |
10.1007/s00044-012-0458-3 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2010.07.020 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.080 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
12.5 |
ug.mL-1 |
10.1021/jm070638m |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
3900.0 |
nM |
10.1039/D1MD00239B |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
467000.0 |
nM |
10.1016/j.bmcl.2016.05.053 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
nan |
None |
10.1016/j.bmc.2013.10.011 |
| Mycobacterium intracellulare |
Mycobacterium intracellulare |
MIC |
nan |
None |
10.1021/np900281r |
| Mycobacterium kansasii |
Mycobacterium kansasii |
IC90 |
72900.0 |
nM |
10.1016/j.bmc.2012.10.007 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
1.56 |
ug.mL-1 |
10.1021/jm00150a006 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00596-1 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
2.0 |
ug.mL-1 |
10.1016/s0960-894x(03)00597-3 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.001 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.bmcl.2013.04.021 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
12.5 |
ug.mL-1 |
10.1039/C8MD00056E |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
2000.0 |
nM |
10.1016/j.bmc.2007.01.051 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
2000.0 |
nM |
10.1016/j.bmc.2013.12.016 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
2000.0 |
nM |
10.1016/j.bmc.2014.05.064 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
2000.0 |
nM |
10.1016/j.bmc.2014.12.019 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
2000.0 |
nM |
10.1016/j.ejmech.2008.06.027 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
2000.0 |
nM |
10.1016/j.ejmech.2010.09.040 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
2000.0 |
nM |
10.1016/j.ejmech.2011.07.052 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
2000.0 |
nM |
10.1016/j.ejmech.2011.09.054 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
2000.0 |
nM |
10.1016/s0960-894x(02)00697-2 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
3860.0 |
nM |
10.1021/ml5003458 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.bmc.2007.01.051 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.bmc.2007.02.021 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.bmc.2009.04.008 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.bmc.2009.12.055 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.bmc.2013.12.016 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.bmc.2014.05.064 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.bmc.2014.12.019 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.bmc.2015.10.029 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.bmc.2017.01.016 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.bmc.2017.01.045 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2008.06.027 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2010.09.040 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2011.07.052 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2011.09.054 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2012.01.060 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2012.07.044 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2012.08.016 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2016.11.041 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2019.111578 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2021.113668 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1016/s0960-894x(02)00697-2 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
4000.0 |
nM |
10.1039/C4MD00301B |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.bmc.2007.02.021 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.bmc.2009.04.008 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.bmc.2010.10.017 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.bmc.2015.10.029 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.bmc.2017.01.016 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.bmc.2017.01.045 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.bmcl.2017.10.050 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.ejmech.2010.02.037 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.ejmech.2012.01.060 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.ejmech.2016.11.041 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.ejmech.2018.04.017 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.ejmech.2019.111578 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
8000.0 |
nM |
10.1016/j.ejmech.2021.113668 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
9100.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
11000.0 |
nM |
10.1016/j.bmcl.2013.12.054 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
11000.0 |
nM |
10.1039/C5MD00178A |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
11400.0 |
nM |
10.1016/j.bmc.2014.11.014 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
16000.0 |
nM |
10.1016/j.bmc.2017.01.045 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
29170.0 |
nM |
10.1016/j.bmc.2013.08.029 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
29200.0 |
nM |
10.1016/j.bmc.2013.08.030 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
29200.0 |
nM |
10.1016/j.bmcl.2016.05.053 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
91000.0 |
nM |
10.1016/j.bmcl.2012.11.052 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
182300.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
200000.0 |
nM |
10.1016/j.ejmech.2012.07.044 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2007.01.051 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2007.02.021 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2009.04.008 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2009.12.055 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2010.10.017 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2013.12.016 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2014.05.064 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2014.12.019 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2015.10.029 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2017.01.016 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.bmc.2017.01.045 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.bmcl.2017.10.050 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2008.06.027 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2010.02.037 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2010.09.040 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2011.07.052 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2011.09.054 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2012.01.060 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2012.07.044 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2012.08.016 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2016.11.041 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2018.04.017 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2019.111578 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/j.ejmech.2021.113668 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1016/s0960-894x(02)00697-2 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
250000.0 |
nM |
10.1039/C4MD00301B |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC |
nan |
None |
10.1016/j.bmc.2013.10.011 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
2.0 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
4.0 |
uM |
10.1016/j.bmc.2017.08.010 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
4.0 |
uM |
10.1016/j.ejmech.2017.02.058 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
4.0 |
uM |
10.1021/acs.jmedchem.5b00608 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
4.0 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
250.0 |
uM |
10.1016/j.bmc.2017.08.010 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
250.0 |
uM |
10.1016/j.ejmech.2017.02.058 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
250.0 |
uM |
10.1021/acs.jmedchem.5b00608 |
| Mycobacterium kansasii |
Mycobacterium kansasii |
MIC>99 |
250.0 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium leprae |
Mycobacterium leprae |
Inhibition |
29.0 |
% |
10.1016/j.bmc.2019.04.032 |
| Mycobacterium marinum |
Mycobacterium marinum |
Activity |
1.8 |
deltalog10CFU/ml |
10.1016/j.bmc.2016.01.059 |
| Mycobacterium marinum |
Mycobacterium marinum |
log(activity) |
2.5 |
None |
10.1016/j.ejmech.2017.12.088 |
| Mycobacterium marinum |
Mycobacterium marinum |
log(activity) |
2.6 |
None |
10.1016/j.bmc.2017.11.031 |
| Mycobacterium marinum |
Mycobacterium marinum |
log(activity) |
2.8 |
None |
10.1016/j.bmc.2017.03.053 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
16.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00248-0 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
16.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00526-5 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
16.0 |
ug.mL-1 |
10.1016/s0960-894x(99)00510-7 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm0602662 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm701560p |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
8000.0 |
nM |
10.1021/ml5003458 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
116000.0 |
nM |
10.1016/j.bmcl.2016.05.053 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
467000.0 |
nM |
10.1016/j.bmc.2013.08.029 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
467000.0 |
nM |
10.1016/j.bmc.2013.08.030 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC |
1000000.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC50 |
2.8 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycobacterium marinum |
Mycobacterium marinum |
MIC90 |
9.2 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycobacterium scrofulaceum |
Mycobacterium scrofulaceum |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycobacterium scrofulaceum |
Mycobacterium scrofulaceum |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium scrofulaceum |
Mycobacterium scrofulaceum |
MIC |
116000.0 |
nM |
10.1016/j.bmcl.2016.05.053 |
| Mycobacterium smegmatis |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.bmc.2014.06.041 |
| Mycobacterium smegmatis |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.bmc.2014.10.016 |
| Mycobacterium smegmatis |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.bmc.2015.02.032 |
| Mycobacterium smegmatis |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.bmc.2015.03.004 |
| Mycobacterium smegmatis |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.ejmech.2015.06.032 |
| Mycobacterium smegmatis |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.ejmech.2016.08.034 |
| Mycobacterium smegmatis (strain ATCC 700084 / mc(2)155) |
DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.ejmech.2016.06.042 |
| Mycobacterium szulgai |
Mycobacterium szulgai |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycobacterium tuberculosis |
2,3-dihydroxybenzoate-AMP ligase |
Ki app |
nan |
None |
10.1021/jm061068d |
| Mycobacterium tuberculosis |
ATP-dependent Clp protease ATP-binding subunit ClpC1 |
Kd |
nan |
None |
10.1021/acs.jnatprod.9b01095 |
| Mycobacterium tuberculosis |
Dihydrofolate reductase |
Ki |
1.0 |
nM |
10.1128/aac.00453-10 |
| Mycobacterium tuberculosis |
Enoyl-[acyl-carrier-protein] reductase |
IC50 |
8290.0 |
nM |
10.1016/j.bmc.2019.02.043 |
| Mycobacterium tuberculosis |
Enoyl-[acyl-carrier-protein] reductase |
Inhibition |
100.0 |
% |
10.1021/acs.jmedchem.0c00007 |
| Mycobacterium tuberculosis |
Enoyl-[acyl-carrier-protein] reductase |
Inhibition |
nan |
% |
10.1016/j.ejmech.2018.04.017 |
| Mycobacterium tuberculosis |
Enoyl-[acyl-carrier-protein] reductase |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2018.07.047 |
| Mycobacterium tuberculosis |
Enoyl-[acyl-carrier-protein] reductase |
MIC99 |
0.07 |
uM |
10.1016/j.bmcl.2020.127576 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
-6.0 |
% |
10.1039/C5MD00589B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
0.0 |
CFU |
10.1016/j.ejmech.2015.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
0.005 |
ug ml-1 |
10.1021/jm00226a016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
0.25 |
ug ml-1 |
10.1128/aac.00753-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.0 |
CFU |
10.1016/j.ejmech.2019.05.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.1 |
deltalog10CFU/ml |
10.1016/j.bmc.2016.01.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.1 |
log10CFU |
10.1016/j.ejmech.2018.11.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.22 |
log10CFU |
10.1039/C4MD00288A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.76 |
log10CFU |
10.1016/j.ejmech.2019.111595 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.76 |
log10CFU |
10.1016/j.ejmech.2020.112075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.76 |
log10CFU |
10.1016/j.ejmech.2022.114145 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.76 |
log10CFU |
10.1021/acs.jmedchem.1c00263 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.929 |
log10CFU |
10.1016/j.ejmech.2018.09.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
1.929 |
log10CFU |
10.1021/acs.jmedchem.0c00500 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.0 |
deltalog10CFU |
10.1039/C5MD00589B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.19 |
ug ml-1 |
10.1515/dmdi.2011.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.44 |
log10CFU |
10.1016/j.ejmech.2016.11.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.5 |
log10CFU |
10.1016/j.ejmech.2018.11.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.59 |
log10CFU |
10.1039/C4MD00288A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
2.66 |
log10CFU |
10.1039/C4MD00288A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
3.2 |
log CFU |
10.1021/jm049972y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
3.38 |
log10CFU |
10.1039/C4MD00288A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
4.0 |
10^-5No_unit |
10.1021/acs.jmedchem.2c00227 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
4.0 |
log10CFU |
10.1016/j.ejmech.2020.112772 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
4.0 |
RLU |
10.1016/j.bmcl.2011.07.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
4.68 |
deltalog10CFU |
10.1021/acs.jmedchem.1c00263 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
4.71 |
None |
10.1016/j.bmc.2007.11.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
5.0 |
log10CFU |
10.1016/j.ejmech.2020.112409 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
5.34 |
log10CFU |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
5.5 |
log CFU |
10.1021/jm049972y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
5.86 |
None |
10.1016/j.bmc.2007.11.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
6.7 |
log10CFU |
10.1016/j.ejmech.2018.11.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
12.0 |
CFU |
10.1016/j.ejmech.2015.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
20.9 |
% |
10.1128/aac.01124-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
29.0 |
% |
10.1021/acs.jmedchem.2c00227 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
50.0 |
mg/L |
10.1128/aac.00185-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
70.0 |
% |
10.1128/aac.00897-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
72.7 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
78.5 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
80.6 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
83.1 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
84.37 |
% |
10.1016/j.ejmech.2009.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
85.4 |
% |
10.1128/aac.01124-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
85.5 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
86.4 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
87.6 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
88.0 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
88.4 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
88.8 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
89.3 |
% |
10.1128/aac.00964-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
89.6 |
% |
10.1016/j.bmcl.2012.10.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
89.6 |
% |
10.1016/j.ejmech.2009.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
89.65 |
% |
10.1016/j.ejmech.2010.08.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
94.7 |
% |
10.1016/j.ejmech.2009.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
95.0 |
% |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
95.85 |
% |
10.1016/j.ejmech.2009.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
95.85 |
% |
10.1016/j.ejmech.2010.08.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
96.0 |
% |
10.1016/j.ejmech.2009.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
96.1 |
% |
10.1128/aac.01124-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
98.0 |
% |
10.1021/jm100165w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
98.0 |
% |
10.1039/C5MD00131E |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
98.42 |
% |
10.1016/j.bmcl.2012.10.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
98.42 |
% |
10.1016/j.ejmech.2009.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
98.42 |
% |
10.1016/j.ejmech.2010.08.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
98.99 |
% |
10.1016/j.ejmech.2009.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
99.0 |
% |
10.1016/j.bmcl.2020.127558 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
99.01 |
% |
10.1016/j.ejmech.2009.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
99.9 |
% |
10.1016/j.bmc.2007.08.064 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
100.0 |
% |
10.1016/j.ejmech.2018.01.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
130.0 |
log10CFU |
10.1016/j.ejmech.2021.113603 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
185.0 |
mg |
10.1126/science.1106753 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmc.2007.02.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmc.2009.04.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmc.2016.03.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmcl.2010.05.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmcl.2011.08.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.bmcl.2012.10.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.ejmech.2012.04.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.ejmech.2014.02.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.ejmech.2016.07.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.ejmech.2017.03.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.ejmech.2018.02.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.ejmech.2019.111713 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.ejmech.2020.112772 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1016/j.ejmech.2022.114404 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acs.jmedchem.0c01374 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acs.jmedchem.1c02122 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acs.jmedchem.6b00415 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acs.jmedchem.8b01533 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acs.jmedchem.9b00010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/acsmedchemlett.7b00287 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/jm00202a020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/jm900358q |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1021/np970182j |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1039/C4MD00288A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1039/C5MD00178A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1128/aac.00196-08 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1128/aac.00453-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1128/aac.00661-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1128/aac.00753-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1128/aac.00898-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1128/aac.01145-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Activity |
nan |
None |
10.1128/aac.01486-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
AUC |
10520.0 |
ng.hr.mL-1 |
10.1515/dmdi.2011.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
0.0 |
/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
1.1 |
10^3/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
1.1 |
10^5/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
1.2 |
10^3/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
1.2 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
1.22 |
10^5/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
1.3 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
1.32 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
1.4 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
1.45 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
1.6 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
1.7 |
10^5/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
2.0 |
10^2/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
2.4 |
10^2/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
2.4 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
2.5 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
3.1 |
10^3/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
3.4 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
3.6 |
10^3/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
4.8 |
10^3/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
4.8 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
5.6 |
10^2/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
7.0 |
10^3/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
7.5 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
7.6 |
10^3/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
7.9 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
8.0 |
10^4/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
25.0 |
/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
40.0 |
/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
CFU |
55.0 |
/ml |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Concentration |
0.1 |
ug ml-1 |
10.1021/jm00131a002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Concentration |
0.5 |
ug ml-1 |
10.1021/jm00131a002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Concentration |
1.0 |
ug ml-1 |
10.1021/jm00131a002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Concentration |
50.0 |
ug ml-1 |
10.1021/jm00131a002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Concentration |
100.0 |
ug ml-1 |
10.1021/jm00131a002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Concentration |
150.0 |
ug ml-1 |
10.1021/jm00131a002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC50 |
130.0 |
nM |
10.1016/j.bmcl.2012.12.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC50 |
180.0 |
nM |
10.1016/j.bmcl.2014.01.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC50 |
190.0 |
nM |
10.1016/j.bmcl.2012.12.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC90 |
0.03 |
mg/ml |
10.1016/j.ejmech.2009.05.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC90 |
0.03 |
ug ml-1 |
10.1016/j.bmcl.2004.09.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC90 |
0.03 |
ug ml-1 |
10.1016/j.bmcl.2005.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC90 |
0.03 |
ug ml-1 |
10.1016/j.bmcl.2016.06.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC90 |
0.2 |
uM |
10.1016/j.bmcl.2012.12.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC90 |
0.29 |
uM |
10.1016/j.bmcl.2014.01.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC90 |
5.0 |
uM |
10.1016/j.bmcl.2012.12.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC90/MIC |
1.2 |
None |
10.1016/j.bmcl.2004.09.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC99 |
0.42 |
mg/ml |
10.1016/j.ejmech.2009.05.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC99 |
0.42 |
ug ml-1 |
10.1016/j.bmcl.2004.09.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC99 |
0.42 |
ug ml-1 |
10.1016/j.bmcl.2005.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
EC99 |
0.42 |
ug ml-1 |
10.1016/j.bmcl.2016.06.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
ED99 |
0.95 |
mg kg-1 |
10.1128/aac.01423-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Emax |
25.0 |
mg kg-1 |
10.1128/aac.01423-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.2 |
None |
10.1016/j.bmc.2016.09.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.2 |
None |
10.1016/j.ejmech.2014.12.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.25 |
None |
10.1016/j.bmcl.2016.11.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.4 |
None |
10.1016/j.ejmech.2020.112035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.4 |
None |
10.1016/j.ejmech.2020.112402 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.5 |
None |
10.1016/j.bmc.2016.07.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.5 |
None |
10.1016/j.ejmech.2019.112010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
1.5 |
None |
10.1021/acs.jnatprod.9b00475 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
2.5 |
None |
10.1016/j.ejmech.2020.112402 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
8.0 |
None |
10.1021/jm500833f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
30.0 |
None |
10.1039/C9MD00006B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
200.0 |
None |
10.1016/j.ejmech.2020.112772 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
FC |
257.08 |
None |
10.1039/C5MD00131E |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
0.0 |
% |
10.1016/j.bmc.2012.09.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
1.47 |
% |
10.1016/j.bmc.2016.09.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
7.22 |
% |
10.1016/j.bmc.2016.09.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
9.77 |
% |
10.1016/j.ejmech.2011.12.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
10.0 |
% |
10.1016/j.bmc.2012.05.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
29.38 |
% |
10.1016/j.ejmech.2011.12.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
37.0 |
% |
10.1016/j.ejmech.2013.03.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
38.0 |
% |
10.1021/acs.jmedchem.0c00007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
48.79 |
% |
10.1016/j.bmc.2016.09.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
51.39 |
% |
10.1016/j.ejmech.2011.12.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
55.0 |
% |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
76.4 |
% |
10.1016/j.ejmech.2013.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
82.3 |
% |
10.1016/j.ejmech.2013.03.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
85.0 |
% |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
90.0 |
% |
10.1016/j.bmc.2017.12.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
92.8 |
% |
10.1016/j.ejmech.2013.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
94.2 |
% |
10.1021/np9000569 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
95.0 |
% |
10.1007/s00044-012-0451-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
95.0 |
% |
10.1016/j.bmcl.2013.06.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
95.0 |
% |
10.1016/j.ejmech.2011.07.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
95.0 |
% |
10.1016/j.ejmech.2011.07.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
95.0 |
% |
10.1016/j.ejmech.2012.01.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
95.0 |
% |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
97.0 |
% |
10.1016/j.bmcl.2016.11.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
97.3 |
% |
10.1016/j.ejmech.2013.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
97.7 |
% |
10.1016/j.ejmech.2013.03.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
98.0 |
% |
10.1016/j.ejmech.2011.12.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
98.0 |
% |
10.1016/j.ejmech.2013.03.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1007/s00044-011-9808-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1007/s00044-012-0026-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1007/s00044-012-0041-y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1007/s00044-012-0073-3 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1007/s00044-012-0129-4 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1007/s00044-012-0322-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1007/s00044-013-0576-6 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1016/j.bmcl.2011.06.040 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1016/j.bmcl.2012.04.070 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1016/j.ejmech.2011.09.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1016/j.ejmech.2013.03.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1016/j.ejmech.2013.05.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1016/j.ejmech.2013.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.0 |
% |
10.1016/j.ejmech.2014.02.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
99.3 |
% |
10.1016/j.bmc.2009.02.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.bmc.2012.05.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.bmc.2012.09.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.bmc.2016.09.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.bmcl.2020.127351 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.ejmech.2011.12.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.ejmech.2013.03.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.ejmech.2013.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
100.0 |
% |
10.1016/j.ejmech.2018.03.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
nan |
None |
10.1016/j.bmc.2013.07.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
nan |
None |
10.1016/j.bmc.2016.02.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
nan |
None |
10.1016/j.ejmech.2013.12.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI |
nan |
None |
10.1021/acs.jmedchem.6b00031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI50 |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2014.03.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI50 |
10.0 |
nM |
10.1016/j.ejmech.2013.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI99 |
0.04 |
ug ml-1 |
10.1016/j.ejmech.2014.03.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
GI99 |
0.06 |
ug ml-1 |
10.1016/j.ejmech.2014.03.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
4.0 |
None |
10.1016/j.bmc.2009.02.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
5.0 |
None |
10.1016/j.bmc.2009.02.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
7.0 |
None |
10.1016/j.bmc.2009.02.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
8.0 |
None |
10.1016/j.bmc.2009.02.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
10.0 |
None |
10.1016/j.bmc.2009.02.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
11.0 |
None |
10.1016/j.bmc.2009.02.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
12.0 |
None |
10.1016/j.bmc.2009.02.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
16.0 |
None |
10.1016/j.ejmech.2012.04.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
20.0 |
None |
10.1016/j.ejmech.2012.04.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
25.0 |
None |
10.1016/j.ejmech.2012.04.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
40.0 |
None |
10.1016/j.ejmech.2012.04.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
48.0 |
None |
10.1016/j.ejmech.2012.04.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
65.0 |
None |
10.1016/j.ejmech.2012.04.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Growth_index |
90.0 |
None |
10.1016/j.ejmech.2012.04.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0013 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0014 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0019 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0023 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0023 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0024 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0025 |
ug.mL-1 |
10.1016/j.bmcl.2015.11.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0025 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.056 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.0025 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.04 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.05 |
ug.mL-1 |
10.1021/np9000703 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.18 |
ug.mL-1 |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.63 |
ug.mL-1 |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
0.69 |
ug.mL-1 |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
1.851 |
ug.mL-1 |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
4.0 |
ug.mL-1 |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
40.0 |
nM |
10.1016/j.ejmech.2014.02.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
70.0 |
nM |
10.1016/j.bmcl.2011.08.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
90.0 |
nM |
10.1016/j.bmcl.2011.08.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
100.0 |
nM |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
100.0 |
nM |
10.1016/j.ejmech.2019.111812 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
100.0 |
nM |
10.1016/j.ejmech.2020.113021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
100.0 |
ug.mL-1 |
10.1016/j.bmc.2007.01.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
110.0 |
nM |
10.1016/j.ejmech.2019.07.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
120.0 |
nM |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
131.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
150.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
180.0 |
nM |
10.1016/j.bmc.2016.09.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
180.0 |
nM |
10.1016/j.bmcl.2017.05.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
180.0 |
nM |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
180.0 |
nM |
10.1016/j.ejmech.2014.08.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
190.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
204.0 |
nM |
10.1021/acs.jmedchem.2c01493 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
210.0 |
nM |
10.1016/j.bmcl.2019.03.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
210.0 |
nM |
10.1016/j.bmcl.2019.03.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
220.0 |
nM |
10.1016/j.bmc.2015.07.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
250.0 |
nM |
10.1016/j.ejmech.2019.07.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
300.0 |
nM |
10.1016/j.ejmech.2010.07.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
330.0 |
nM |
10.1016/j.bmc.2015.03.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
350.0 |
nM |
10.1016/j.bmc.2020.115797 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
360.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
400.0 |
nM |
10.1016/j.bmc.2020.115797 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
540.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
650.0 |
nM |
10.1016/j.bmc.2015.07.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
2040.0 |
nM |
10.1016/j.bmcl.2016.09.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
15000.0 |
nM |
10.1016/j.ejmech.2011.02.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
45570.0 |
nM |
10.1016/j.bmcl.2005.07.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
200000.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
59579931.56 |
nM |
10.1016/j.ejmech.2009.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
nan |
None |
10.1016/j.bmc.2012.01.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC50 |
nan |
None |
10.1021/np900281r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.0078 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.055 |
ug.mL-1 |
10.1021/np400002p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.074 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.075 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.075 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.056 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.11 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2012.11.097 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
0.29 |
ug.mL-1 |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
110.0 |
nM |
10.1016/j.ejmech.2014.02.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
190.0 |
nM |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
200.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
200.0 |
nM |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
210.0 |
nM |
10.1016/j.bmcl.2011.04.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
210.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
240.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
290.0 |
nM |
10.1016/j.bmc.2016.09.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
290.0 |
nM |
10.1016/j.bmcl.2017.05.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
290.0 |
nM |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
290.0 |
nM |
10.1016/j.ejmech.2014.08.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
470.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
600.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC90 |
200000.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC99 |
0.13 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IC99 |
130.0 |
nM |
10.1016/j.ejmech.2014.02.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
0.0 |
% |
10.1021/jm100165w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
10.0 |
% |
10.1016/j.bmc.2016.03.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
49.7 |
% |
10.1021/jm030479g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
59.1 |
% |
10.1021/jm030479g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
64.0 |
% |
10.1016/j.ejmech.2012.08.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
68.7 |
% |
10.1021/jm030479g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
84.0 |
% |
10.1016/j.bmcl.2012.05.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
84.0 |
% |
10.1016/j.ejmech.2015.03.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
90.0 |
% |
10.1016/j.bmc.2016.09.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
90.0 |
% |
10.1016/j.bmcl.2006.06.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
92.0 |
% |
10.1016/j.ejmech.2012.08.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
92.0 |
% |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
92.9 |
% |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
93.0 |
% |
10.1016/j.ejmech.2015.03.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
93.9 |
% |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
94.0 |
% |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.0 |
% |
10.1016/j.bmc.2017.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.0 |
% |
10.1016/j.bmcl.2004.05.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.0 |
% |
10.1016/j.ejmech.2009.11.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.0 |
% |
10.1016/j.ejmech.2010.04.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.0 |
% |
10.1016/j.ejmech.2011.03.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.0 |
% |
10.1016/j.ejmech.2011.08.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
95.0 |
% |
10.1016/j.ejmech.2013.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
96.0 |
% |
10.1016/j.bmcl.2006.06.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1007/s00044-011-9950-4 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1007/s00044-012-0351-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1007/s00044-013-0472-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1007/s00044-013-0839-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.bmc.2009.02.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.bmc.2009.04.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.bmc.2015.11.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.bmc.2017.09.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.bmcl.2013.01.079 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.bmcl.2014.05.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.bmcl.2016.06.038 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2007.06.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2010.01.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2011.06.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2012.03.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2012.05.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2014.02.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2014.06.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2014.07.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2014.07.100 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2016.02.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2020.112358 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2020.112886 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.0 |
% |
10.1039/d2md00076h |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.18 |
% |
10.1016/j.ejmech.2019.05.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
99.98 |
% |
10.1016/j.ejmech.2011.06.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1007/s00044-012-9971-7 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1016/j.bmc.2016.03.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1016/j.bmcl.2015.07.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1016/j.bmcl.2021.128261 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1016/j.ejmech.2015.06.056 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1016/j.ejmech.2022.114831 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1021/jm0703901 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1021/jm100165w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
100.0 |
% |
10.1021/jm100568q |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
nan |
% |
10.1007/s00044-013-0472-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
nan |
% |
10.1016/j.bmc.2015.03.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
nan |
% |
10.1016/j.bmc.2020.115579 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
nan |
% |
10.1016/j.bmcl.2010.08.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
nan |
% |
10.1016/j.ejmech.2014.03.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
nan |
% |
10.1016/j.ejmech.2015.03.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
nan |
% |
10.1021/acsmedchemlett.9b00515 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
nan |
% |
10.1021/jm5003606 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Inhibition |
nan |
% |
10.1039/C5MD00178A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IZ |
21.0 |
mm |
10.1016/j.bmcl.2011.02.103 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IZ |
31.0 |
mm |
10.1016/j.ejmech.2021.113266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
IZ |
nan |
None |
10.1016/j.ejmech.2017.07.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
0.87 |
None |
10.1016/j.bmcl.2013.12.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
1.0 |
None |
10.1038/35016103 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
1.22 |
None |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
1.3 |
None |
10.1128/aac.00185-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
1.4 |
None |
10.1038/35016103 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
1.75 |
mg |
10.1126/science.1106753 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
2.0 |
None |
10.1016/j.bmcl.2011.12.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
2.16 |
None |
10.1021/np800572r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
2.2 |
None |
10.1128/aac.00379-08 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
2.59 |
None |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
2.66 |
None |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
2.8 |
None |
10.1016/j.bmcl.2013.02.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.0 |
None |
10.1016/j.bmcl.2011.12.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.05 |
mg |
10.1126/science.1106753 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.14 |
None |
10.1128/aac.00897-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.33 |
None |
10.1128/aac.00379-08 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.38 |
None |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.63 |
None |
10.1016/j.bmc.2012.03.058 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
3.68 |
None |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.0 |
None |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.434 |
None |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.47 |
None |
10.1128/aac.00379-08 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.595 |
None |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.62 |
None |
10.1016/j.ejmech.2010.05.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.71 |
None |
10.1016/j.ejmech.2008.02.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.71 |
None |
10.1016/j.ejmech.2009.05.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.71 |
None |
10.1016/j.ejmech.2009.09.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.92 |
None |
10.1021/jm800545k |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.944 |
None |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
4.96 |
None |
10.1016/j.ejmech.2009.05.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.01 |
None |
10.1021/jm5003606 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.04 |
None |
10.1128/aac.00379-08 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.33 |
None |
10.1021/np800572r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.41 |
None |
10.1016/j.bmc.2012.03.058 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.45 |
None |
10.1016/j.ejmech.2010.05.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.58 |
None |
10.1016/j.ejmech.2009.05.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.61 |
None |
10.1021/jm800545k |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.751 |
None |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.8 |
None |
10.1128/aac.00897-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.86 |
None |
10.1016/j.ejmech.2008.02.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
5.86 |
None |
10.1016/j.ejmech.2009.09.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10cfu |
6.702 |
None |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
3.5 |
None |
10.1021/jm050948+ |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
3.88 |
None |
10.1021/jm050765n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
3.98 |
None |
10.1016/j.bmcl.2007.09.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
4.11 |
None |
10.1021/jm060339h |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
4.7 |
None |
10.1128/aac.00898-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
4.71 |
None |
10.1016/j.bmc.2007.11.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
4.71 |
None |
10.1016/j.bmcl.2007.11.110 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
4.71 |
None |
10.1021/jm700999n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
4.9 |
None |
10.1128/aac.00898-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
5.12 |
None |
10.1021/jm060339h |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
5.86 |
None |
10.1016/j.bmc.2007.11.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
5.86 |
None |
10.1016/j.bmcl.2007.11.110 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log10 cfu |
5.86 |
None |
10.1021/jm700999n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-1.94 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-1.88 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-1.68 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-1.41 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-1.34 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-1.32 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-0.57 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
-0.43 |
None |
10.1128/aac.01204-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
0.21 |
None |
10.1016/j.bmc.2014.12.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
1.88 |
None |
10.1016/j.ejmech.2012.02.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml |
2.89 |
None |
10.1128/aac.00185-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml/day |
0.67 |
None |
10.1016/j.ejmech.2012.02.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log10CFU/ml/day |
0.9 |
None |
10.1128/aac.00185-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(1/MIC) |
-0.041 |
None |
10.1021/jm00226a007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(1/MIC) |
0.0 |
None |
10.1016/j.ejmech.2013.10.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(1/MIC) |
1.7 |
None |
10.1016/j.ejmech.2013.10.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.0 |
None |
10.1016/j.bmc.2017.11.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.0 |
None |
10.1016/j.ejmech.2020.112178 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.0 |
None |
10.1021/acs.jmedchem.6b00674 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.1 |
None |
10.1016/j.bmc.2017.11.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.2 |
None |
10.1016/j.bmc.2017.03.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.2 |
None |
10.1016/j.ejmech.2017.12.088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.4 |
None |
10.1016/j.ejmech.2017.12.088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.5 |
None |
10.1016/j.ejmech.2020.112178 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.7 |
None |
10.1016/j.bmc.2017.12.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
1.9 |
None |
10.1016/j.bmc.2017.03.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
2.5 |
None |
10.1016/j.ejmech.2020.112178 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
2.6 |
None |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
2.6 |
None |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
2.7 |
None |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
2.7 |
None |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
log(activity) |
4.22 |
None |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Log CFU |
6.38 |
None |
10.1016/j.bmcl.2005.07.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
-logMIC |
6.447 |
None |
10.1007/s00044-012-0385-3 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
0.1 |
ug ml-1 |
10.1016/j.bmcl.2004.09.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
0.1 |
ug ml-1 |
10.1016/j.bmcl.2005.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
0.12 |
ug ml-1 |
10.1128/aac.00753-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
0.3 |
uM |
10.1016/j.ejmech.2018.02.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
0.57 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
0.99 |
uM |
10.1021/acs.jnatprod.9b01095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
1.6 |
ug ml-1 |
10.1016/j.bmcl.2004.09.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
1.6 |
ug ml-1 |
10.1016/j.bmcl.2005.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
1.75 |
uM |
10.1007/s00044-011-9788-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
4.0 |
uM |
10.1021/acs.jnatprod.9b01095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
nan |
None |
10.1016/j.bmcl.2005.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
nan |
None |
10.1016/j.ejmech.2018.02.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC |
nan |
None |
10.1021/np800778b |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC90 |
nan |
None |
10.1016/j.ejmech.2011.10.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC90 |
nan |
None |
10.1016/j.ejmech.2015.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MBC99.9 |
3.2 |
uM |
10.1021/acsmedchemlett.0c00588 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.bmc.2011.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2008.04.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2017.06.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.01 |
ug.mL-1 |
10.1016/j.ejmech.2020.112175 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.01 |
ug.mL-1 |
10.1021/jm401468w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.013 |
ug.mL-1 |
10.1021/jm401468w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.014 |
ug.mL-1 |
10.1016/j.bmcl.2018.05.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.bmc.2013.09.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0156 |
ug.mL-1 |
10.1128/aac.00185-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.016 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00972 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.018 |
ug.mL-1 |
10.1021/jm000350w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.019 |
ug.mL-1 |
10.1016/j.ejmech.2022.114145 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.bmc.2009.04.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.bmcl.2010.02.081 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.bmcl.2010.05.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.bmcl.2014.07.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.bmcl.2014.09.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2013.10.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2014.06.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2015.06.056 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1021/jm9708745 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1039/C7MD00350A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1039/C7MD00366H |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.02 |
ug.mL-1 |
10.1039/d2md00401a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.023 |
ug.mL-1 |
10.1021/np900021h |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.023 |
ug.mL-1 |
10.1021/np900082h |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0234 |
ug.mL-1 |
10.1021/np200429b |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmc.2007.01.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmc.2008.10.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmc.2010.09.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmcl.2005.08.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmcl.2007.07.089 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmcl.2008.11.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmcl.2017.07.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.bmcl.2019.01.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.ejmech.2006.08.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.ejmech.2010.04.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.ejmech.2011.06.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1016/s0960-894x(00)00648-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.025 |
ug.mL-1 |
10.1021/ml4002248 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmc.2008.05.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmc.2019.07.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmc.2022.116777 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.100 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2010.08.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2011.07.068 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2014.02.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2017.08.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2009.05.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2011.10.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2015.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2017.07.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.070 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2019.04.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2020.112996 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2021.113580 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00500 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1021/jm201608g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1021/jm4012033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1021/jm500432n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1021/jm500853v |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1021/np400391p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1038/35016103 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1039/d1md00387a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.03 |
ug.mL-1 |
10.1128/aac.00643-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.031 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.031 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00972 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.034 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0366 |
ug.mL-1 |
10.1016/j.ejmech.2021.113398 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.038 |
ug.mL-1 |
10.1016/j.bmc.2018.03.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.038 |
ug.mL-1 |
10.1016/j.ejmech.2020.112409 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.039 |
ug.mL-1 |
10.1016/j.bmcl.2018.07.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.039 |
ug.mL-1 |
10.1016/j.ejmech.2020.112075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.039 |
ug.mL-1 |
10.1016/j.ejmech.2021.113603 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.039 |
ug.mL-1 |
10.1021/acsmedchemlett.7b00299 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1016/s0960-894x(03)00241-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00500 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1021/np0004404 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1021/np020055+ |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1021/np0204489 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1021/np030067a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1021/np030429e |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1021/np030519j |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1021/np0503202 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.04 |
ug.mL-1 |
10.1021/np800805f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.041 |
ug.mL-1 |
10.1128/aac.00897-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.043 |
ug.mL-1 |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.045 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0469 |
ug.mL-1 |
10.1021/acs.jnatprod.5b00961 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.047 |
ug.mL-1 |
10.1021/acs.jnatprod.8b00869 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.047 |
ug.mL-1 |
10.1021/acs.jnatprod.9b00947 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.048 |
ug.mL-1 |
10.1128/aac.00897-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.049 |
ug.mL-1 |
10.1016/j.ejmech.2019.06.038 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1007/s00044-011-9948-y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmc.2008.05.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmc.2009.06.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmc.2015.04.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmc.2015.04.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmc.2016.01.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2005.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2005.08.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2007.10.083 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2009.04.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.100 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2010.09.137 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2011.05.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2011.09.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2012.04.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2013.04.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2015.07.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2017.07.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2017.08.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.bmcl.2018.05.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2014.07.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2014.09.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.090 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2019.112010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1016/s0960-894x(00)00058-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/jm00150a006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/jm020452h |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/jm020891g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/jm060339h |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/jm070638m |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/jm201608g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/np010006h |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/np0205598 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/np049757k |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/np060164e |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/np070293a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/np070629g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/np5001494 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1021/np9003189 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1128/aac.01288-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.05 |
ug.mL-1 |
10.1128/aac.01486-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.056 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1007/s00044-012-0222-8 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmc.2013.09.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmc.2019.04.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.bmcl.2015.12.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2010.07.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2011.10.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2015.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2017.06.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00360 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1021/jm4012033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1021/jm500432n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1021/np2000667 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1038/35016103 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00453-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.00753-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.bmcl.2011.12.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.bmcl.2012.08.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.bmcl.2014.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.0625 |
ug.mL-1 |
10.1016/j.ejmech.2012.03.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.063 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.07 |
ug.mL-1 |
10.1128/aac.01486-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.072 |
ug.mL-1 |
10.1016/j.bmc.2022.117006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.074 |
ug.mL-1 |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.075 |
ug.mL-1 |
10.1016/j.bmcl.2007.02.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.075 |
ug.mL-1 |
10.1016/j.bmcl.2015.11.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.075 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.075 |
ug.mL-1 |
10.1016/j.ejmech.2017.06.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.075 |
ug.mL-1 |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.078 |
ug.mL-1 |
10.1016/j.ejmech.2019.01.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.08 |
ug.mL-1 |
10.1016/j.bmc.2012.03.058 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.08 |
ug.mL-1 |
10.1016/j.bmc.2019.115050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.08 |
ug.mL-1 |
10.1016/j.ejmech.2011.10.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.08 |
ug.mL-1 |
10.1016/j.ejmech.2015.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.088 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.09 |
ug.mL-1 |
10.1016/s0960-894x(03)00111-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.094 |
ug.mL-1 |
10.1021/acs.jnatprod.5b00826 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.094 |
ug.mL-1 |
10.1021/acs.jnatprod.6b00973 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.094 |
ug.mL-1 |
10.1021/np5005328 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.098 |
ug.mL-1 |
10.1016/j.bmc.2013.06.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.098 |
ug.mL-1 |
10.1016/j.ejmech.2018.05.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1007/s00044-011-9664-7 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmc.2019.04.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2006.06.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2008.09.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2011.05.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2012.10.056 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2013.07.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2013.11.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2014.02.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2014.05.006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2015.08.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.107 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2016.04.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2016.04.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2016.04.088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2016.05.085 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2016.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2017.05.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2017.10.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2018.03.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2019.01.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.040 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2020.127434 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2023.129189 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2011.06.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2012.04.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2013.10.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2015.03.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2015.10.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2015.10.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2018.07.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1021/acs.jnatprod.0c01212 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm000149l |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm070638m |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1021/np070174v |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1021/np900342b |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1039/C8MD00056E |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1039/C8MD00212F |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1128/aac.01458-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.1 |
ug.mL-1 |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.11 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.bmc.2016.10.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.12 |
ug.mL-1 |
10.1016/j.ejmech.2019.07.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1007/s00044-012-0351-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmc.2011.01.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmc.2011.02.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.bmcl.2014.09.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2014.02.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1016/j.ejmech.2020.112440 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00360 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1021/jm701560p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1021/np050554l |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.15 |
ug.mL-1 |
10.1016/j.ejmech.2020.112768 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.16 |
ug.mL-1 |
10.1039/C9MD00057G |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.19 |
ug.mL-1 |
10.1016/j.ejmech.2011.10.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.19 |
ug.mL-1 |
10.1016/j.ejmech.2015.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.19 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1007/s00044-011-9728-8 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1007/s00044-011-9950-4 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1007/s00044-012-0026-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1007/s00044-012-0041-y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1007/s00044-012-0060-8 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1007/s00044-012-0073-3 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1007/s00044-012-0129-4 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1007/s00044-012-0322-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1007/s00044-013-0472-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1007/s00044-013-0839-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmc.2007.08.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmc.2007.08.064 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmc.2012.04.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2004.09.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2005.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2005.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2007.09.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2007.11.091 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2009.02.101 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2014.05.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2016.01.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.bmcl.2021.127819 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2007.08.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2009.03.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2009.07.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2011.06.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2011.09.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2011.10.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2012.03.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2013.03.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2013.05.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2014.06.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2015.03.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2015.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2016.08.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2017.07.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2019.01.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2019.05.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1016/j.ejmech.2021.113266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1021/jm800038g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1021/jm950956y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1021/np9700681 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1128/aac.00643-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.2 |
ug.mL-1 |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.23 |
ug.mL-1 |
10.1021/np100632g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.23 |
ug.mL-1 |
10.1021/np200593d |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.24 |
ug.mL-1 |
10.1016/j.ejmech.2014.06.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.24 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.24 |
ug.mL-1 |
10.1021/acsmedchemlett.9b00515 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-011-9573-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-011-9646-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-012-0092-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-012-0112-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-012-0340-3 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-012-0431-1 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1007/s00044-013-0576-6 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2009.06.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2010.05.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2013.10.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmc.2019.07.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.073 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.084 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.085 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2006.12.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2008.10.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2012.01.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.bmcl.2014.09.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2007.11.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2009.05.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2009.06.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2010.01.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2010.08.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2013.11.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2015.03.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2020.112045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/s0960-894x(98)00248-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/s0960-894x(98)00526-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1016/s0960-894x(99)00510-7 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1021/acsmedchemlett.1c00431 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm0602662 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm401468w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1021/jm701560p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00643-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.25 |
ug.mL-1 |
10.1128/aac.00661-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.3 |
ug.mL-1 |
10.1016/j.bmc.2015.11.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.3 |
ug.mL-1 |
10.1016/j.ejmech.2016.07.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.3 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.312 |
ug.mL-1 |
10.1039/C7MD00366H |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.313 |
ug.mL-1 |
10.1039/C7MD00350A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.32 |
ug.mL-1 |
10.1016/j.ejmech.2010.05.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.36 |
ug.mL-1 |
10.1007/s00044-013-0787-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.36 |
ug.mL-1 |
10.1016/j.ejmech.2014.09.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.36 |
ug.mL-1 |
10.1016/j.ejmech.2014.10.079 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.36 |
ug.mL-1 |
10.1016/j.ejmech.2017.03.015 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.36 |
ug.mL-1 |
10.1021/jm800545k |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1007/s00044-012-0043-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.bmcl.2011.10.064 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.bmcl.2012.08.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.bmcl.2014.05.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2010.09.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2013.09.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.4 |
ug.mL-1 |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.41 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.41 |
ug.mL-1 |
10.1039/C8MD00212F |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.43 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.44 |
ug.mL-1 |
10.1016/j.bmcl.2015.09.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.48 |
ug.mL-1 |
10.1016/j.bmc.2019.01.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.48 |
ug.mL-1 |
10.1039/C6MD00085A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.49 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2008.02.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2009.04.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmc.2011.11.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.bmcl.2007.07.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2018.07.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2018.12.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.07.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.5 |
ug.mL-1 |
10.1128/aac.00661-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.56 |
ug.mL-1 |
10.1016/j.ejmech.2020.112609 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.56 |
ug.mL-1 |
10.1016/j.ejmech.2021.113266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.6 |
ug.mL-1 |
10.1007/s00044-013-0485-8 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.6 |
ug.mL-1 |
10.1016/j.bmc.2019.115050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.625 |
ug.mL-1 |
10.1007/s00044-013-0815-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.625 |
ug.mL-1 |
10.1016/j.ejmech.2021.113293 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.63 |
ug.mL-1 |
10.1007/s00044-007-9000-4 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.63 |
ug.mL-1 |
10.1021/np500538c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.65 |
ug.mL-1 |
10.1007/s00044-007-9036-5 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.65 |
ug.mL-1 |
10.1016/j.bmcl.2006.07.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.65 |
ug.mL-1 |
10.1016/j.ejmech.2009.02.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.68 |
ug.mL-1 |
10.1016/j.ejmech.2011.04.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.7 |
ug.mL-1 |
10.1007/s00044-012-0451-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.7 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.7 |
ug.mL-1 |
10.1016/j.ejmech.2011.03.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.7 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.7 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.7 |
ug.mL-1 |
10.1016/j.ejmech.2011.08.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.7 |
ug.mL-1 |
10.1016/j.ejmech.2012.01.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.7 |
ug.mL-1 |
10.1016/j.ejmech.2013.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.72 |
ug.mL-1 |
10.1039/C6MD00593D |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.75 |
ug.mL-1 |
10.1007/s00044-010-9402-6 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.75 |
ug.mL-1 |
10.1016/j.bmcl.2011.06.040 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.75 |
ug.mL-1 |
10.1016/j.bmcl.2011.10.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.75 |
ug.mL-1 |
10.1016/j.ejmech.2008.09.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.75 |
ug.mL-1 |
10.1016/j.ejmech.2009.09.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.75 |
ug.mL-1 |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.75 |
ug.mL-1 |
10.1016/j.ejmech.2017.07.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.bmcl.2011.12.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.78 |
ug.mL-1 |
10.1016/j.ejmech.2018.10.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.8 |
nM |
10.1007/s00044-011-9813-z |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.8 |
nM |
10.1016/j.ejmech.2010.08.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.8 |
ug.mL-1 |
10.1007/s00044-013-0485-8 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.8 |
ug.mL-1 |
10.1016/j.bmcl.2016.11.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
0.98 |
ug.mL-1 |
10.1016/j.bmcl.2018.01.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2016.10.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2019.115050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.12.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.06.076 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.09.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.10.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.09.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.0 |
ug.mL-1 |
10.1128/aac.00661-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.1 |
ug.mL-1 |
10.1016/j.bmc.2011.11.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.2 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.25 |
ug.mL-1 |
10.1016/j.ejmech.2021.113266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.3 |
ug.mL-1 |
10.1016/j.bmc.2019.115050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.3 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.4 |
ug.mL-1 |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.4 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.45 |
nM |
10.1016/j.bmc.2016.02.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.5 |
ug.mL-1 |
10.1007/s00044-012-0074-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2009.11.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2006.06.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2009.04.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2012.01.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2013.04.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.56 |
ug.mL-1 |
10.1021/jm060339h |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.6 |
ug.mL-1 |
10.1016/j.bmcl.2020.127655 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.6 |
ug.mL-1 |
10.1016/j.bmcl.2021.127984 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1.6 |
ug.mL-1 |
10.1016/j.ejmech.2021.113266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2013.09.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2019.07.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.02.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.10.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1021/np050554l |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00086-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.0 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.04 |
nM |
10.1007/s00044-011-9662-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.04 |
nM |
10.1007/s00044-011-9705-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.379 |
ug.mL-1 |
10.1016/j.ejmech.2020.112075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.38 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.46 |
ug.mL-1 |
10.1016/j.ejmech.2022.114145 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.5 |
ug.mL-1 |
10.1128/aac.01486-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2.7 |
ug.mL-1 |
10.1007/s00044-013-0485-8 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.1 |
ug.mL-1 |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.1 |
ug.mL-1 |
10.1016/j.ejmech.2020.112106 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.1 |
ug.mL-1 |
10.1021/np2000667 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.12 |
ug.mL-1 |
10.1016/j.ejmech.2019.02.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.13 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.2 |
ug.mL-1 |
10.1039/C9MD00057G |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3.78 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmc.2011.01.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmc.2011.02.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmc.2016.10.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.08.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.07.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.03.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.09.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00360 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1021/np050554l |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4.0 |
ug.mL-1 |
10.1128/aac.00661-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
5.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.083 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
5.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.01.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
5.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00972 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
5.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b01578 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.25 |
ug.mL-1 |
10.1007/s00044-012-0351-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.25 |
ug.mL-1 |
10.1007/s00044-013-0815-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2015.06.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2018.03.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2020.112666 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
6.25 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7.0 |
nM |
10.1021/jm401268f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.02.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7.9 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2015.03.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1021/acs.jnatprod.2c00360 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1021/jm201608g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.0 |
ug.mL-1 |
10.1128/aac.00287-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8.5 |
ug.mL-1 |
10.1016/j.ejmech.2010.05.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.bmcl.2021.127924 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112409 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113398 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113603 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114145 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c00500 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c02153 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
nM |
10.1021/acs.jnatprod.0c00804 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1007/s00044-012-0451-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.bmcl.2011.12.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.08.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2012.01.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.11.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2014.10.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2015.06.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2018.08.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2020.112106 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12.5 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
15.0 |
nM |
10.1016/j.bmc.2017.12.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
15.0 |
nM |
10.1021/jm401268f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116529 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.073 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.084 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.bmcl.2005.01.085 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1021/jm701560p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00643-09 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16.0 |
ug.mL-1 |
10.1128/aac.00661-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
17.5 |
ug.mL-1 |
10.1021/np400391p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
19.2 |
ug.mL-1 |
10.1039/C9MD00057G |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
20.0 |
nM |
10.1016/s0960-894x(98)00126-7 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
20.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.12.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
20.0 |
ug.mL-1 |
10.1021/acs.jmedchem.8b00281 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.ejmech.2014.10.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1021/acs.jmedchem.6b00031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1021/acsmedchemlett.1c00431 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25.0 |
ug.mL-1 |
10.1021/jm070638m |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
27.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.05.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
27.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
29.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
30.0 |
nM |
10.1021/ml5001728 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
30.0 |
nM |
10.1021/ml5003458 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
30.0 |
nM |
10.1021/ml500531p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmc.2021.116529 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.bmcl.2014.09.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.03.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
nM |
10.1039/C6MD00231E |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.bmcl.2011.09.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.07.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.01.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.06.038 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40.0 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00330 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45.57 |
ug.mL-1 |
10.1021/jm800545k |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
nM |
10.1007/s00044-011-9770-6 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
nM |
10.1021/jm4012033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
50.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.0 |
nM |
10.1016/j.ejmech.2019.111935 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.0 |
nM |
10.1016/j.ejmech.2020.112967 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.0 |
nM |
10.1021/ml5001728 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
60.0 |
nM |
10.1021/ml500531p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmc.2022.116777 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.bmcl.2019.07.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.03.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.07.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2021.113580 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64.0 |
ug.mL-1 |
10.1039/d1md00387a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
70.0 |
nM |
10.1039/C9MD00347A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
90.0 |
nM |
10.1021/jm401735w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1016/j.bmcl.2009.11.105 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1021/jm5002937 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1021/ml5003458 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
nM |
10.1039/C9MD00347A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.bmc.2008.05.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.bmc.2015.04.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.100 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm00150a006 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100.0 |
ug.mL-1 |
10.1371/journal.pmed.0030466 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.ejmech.2011.03.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
120.0 |
nM |
10.1016/j.ejmech.2017.06.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.bmc.2019.01.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.bmc.2019.04.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.07.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.04.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.090 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.09.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.11.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.07.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111678 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128.0 |
ug.mL-1 |
10.1021/jm201608g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
140.0 |
nM |
10.1016/j.bmcl.2014.07.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
140.0 |
nM |
10.1021/acs.jmedchem.1c00707 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
145.0 |
nM |
10.1016/j.ejmech.2011.07.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
146.0 |
nM |
10.1016/j.ejmech.2014.04.077 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
150.0 |
nM |
10.1021/jm000350w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
156.0 |
nM |
10.1021/jm500571f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
160.0 |
nM |
10.1016/j.ejmech.2016.11.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
160.0 |
nM |
10.1016/s0960-894x(98)00126-7 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
170.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
170.0 |
nM |
10.1021/np100282k |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
nM |
10.1016/j.bmc.2019.06.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
nM |
10.1016/j.bmc.2021.116426 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
nM |
10.1016/j.bmcl.2013.06.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
nM |
10.1016/j.bmcl.2013.08.101 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
nM |
10.1016/j.ejmech.2014.07.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
nM |
10.1016/j.ejmech.2015.04.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
nM |
10.1016/j.ejmech.2018.02.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
nM |
10.1021/acs.jnatprod.2c01003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
nM |
10.1021/jm5002937 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
217.0 |
nM |
10.1016/j.ejmech.2013.01.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
220.0 |
nM |
10.1016/j.bmc.2011.12.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
220.0 |
nM |
10.1016/j.bmcl.2013.11.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
220.0 |
nM |
10.1021/acsmedchemlett.9b00343 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
220.0 |
nM |
10.1021/jm5005978 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
230.0 |
nM |
10.1016/j.bmc.2010.08.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
230.0 |
nM |
10.1021/jm5005978 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
240.0 |
nM |
10.1016/j.bmc.2010.08.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
240.0 |
nM |
10.1016/j.bmcl.2013.11.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
250.0 |
nM |
10.1016/j.bmc.2010.08.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
250.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
256.0 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01833 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
256.0 |
ug.mL-1 |
10.1128/aac.01577-08 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
269.0 |
nM |
10.1016/j.ejmech.2019.06.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
270.0 |
nM |
10.1016/j.bmc.2019.01.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
280.0 |
nM |
10.1016/j.bmc.2011.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
280.0 |
nM |
10.1016/j.bmcl.2015.12.083 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
290.0 |
nM |
10.1016/j.ejmech.2010.11.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
290.0 |
nM |
10.1021/np0498354 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
290.0 |
nM |
10.1021/np050036a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
290.0 |
nM |
10.1021/np0601197 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
290.0 |
nM |
10.1021/np070010e |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
300.0 |
nM |
10.1016/j.bmcl.2016.03.066 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
300.0 |
nM |
10.1021/acs.jnatprod.6b00839 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
300.0 |
nM |
10.1021/jm5002937 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
300.0 |
nM |
10.1039/C9MD00347A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
300.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
310.0 |
nM |
10.1016/j.bmc.2016.09.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
310.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
310.0 |
nM |
10.1016/j.bmc.2018.04.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
310.0 |
nM |
10.1016/j.bmcl.2012.12.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
310.0 |
nM |
10.1016/j.bmcl.2017.05.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
310.0 |
nM |
10.1016/j.ejmech.2014.08.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
310.0 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
310.0 |
nM |
10.1016/j.ejmech.2017.11.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
312.0 |
nM |
10.1021/jm500571f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
313.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
340.0 |
nM |
10.1021/acsmedchemlett.7b00356 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
350.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
350.0 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
350.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
357.0 |
nM |
10.1007/s00044-012-0385-3 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.bmc.2007.11.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.bmc.2007.11.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.bmc.2009.06.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.bmc.2011.04.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.bmcl.2007.09.095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.bmcl.2012.02.091 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.bmcl.2014.02.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.bmcl.2021.127810 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.bmcl.2022.128604 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.ejmech.2008.02.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.ejmech.2009.09.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.ejmech.2009.09.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.ejmech.2009.09.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.ejmech.2009.09.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.ejmech.2010.10.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.ejmech.2012.04.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.ejmech.2019.01.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.ejmech.2019.05.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.ejmech.2020.112035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.ejmech.2020.112402 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1016/j.ejmech.2020.112699 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1021/jm020891g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1021/jm700999n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
360.0 |
nM |
10.1021/np900650c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
370.0 |
nM |
10.1016/j.bmcl.2009.12.062 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
370.0 |
nM |
10.1016/j.bmcl.2011.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
370.0 |
nM |
10.1021/jm201023g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
370.0 |
nM |
10.1021/jm300125e |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
370.0 |
nM |
10.1021/np800702c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
390.0 |
nM |
10.1016/j.bmc.2010.08.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
390.0 |
nM |
10.1016/j.ejmech.2009.05.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
390.0 |
nM |
10.1039/C9MD00006B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
390.0 |
nM |
10.1039/C9MD00347A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.bmc.2012.08.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.bmc.2017.03.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.bmcl.2009.10.107 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.bmcl.2010.04.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.bmcl.2010.10.080 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.bmcl.2011.03.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.bmcl.2011.05.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.bmcl.2011.12.119 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.ejmech.2011.07.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.ejmech.2011.07.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.ejmech.2011.09.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.ejmech.2012.10.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.ejmech.2013.06.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.ejmech.2013.10.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.ejmech.2013.11.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.ejmech.2015.06.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1016/j.ejmech.2020.112178 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1021/acs.jmedchem.6b00674 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
400.0 |
nM |
10.1021/jm901273n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
430.0 |
nM |
10.1021/jm900003c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
437.0 |
nM |
10.1021/jm2003624 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
440.0 |
nM |
10.1016/j.bmc.2007.05.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
440.0 |
nM |
10.1021/acsmedchemlett.9b00343 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
450.0 |
nM |
10.1016/j.bmc.2013.11.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
450.0 |
nM |
10.1016/j.bmcl.2013.11.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
450.0 |
nM |
10.1016/j.ejmech.2013.08.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
450.0 |
nM |
10.1021/jm5005978 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
450.0 |
nM |
10.1021/jm900003c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
460.0 |
nM |
10.1021/acs.jnatprod.9b01095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.bmc.2007.02.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.bmc.2009.04.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.bmc.2009.12.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.bmc.2010.10.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.bmc.2013.12.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.bmc.2014.05.064 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.bmc.2014.12.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.bmc.2015.10.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.bmc.2017.01.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.bmc.2017.01.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.bmcl.2017.10.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2008.06.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2010.09.040 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2012.01.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2012.07.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2012.08.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2016.11.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2018.04.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2019.111578 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/j.ejmech.2021.113668 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1016/s0960-894x(02)00697-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1021/acs.jnatprod.1c00232 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1021/jm00226a007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1021/jm500497v |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1021/jm900003c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1021/jm901112f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1021/jm901273n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1021/ml5001933 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1039/C4MD00301B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1039/C7MD00146K |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
500.0 |
nM |
10.1128/aac.00055-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
512.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
560.0 |
nM |
10.1016/j.ejmech.2011.09.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
580.0 |
nM |
10.1016/j.bmc.2019.02.043 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
600.0 |
nM |
10.1016/j.bmc.2009.08.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
600.0 |
nM |
10.1016/j.bmc.2011.09.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
600.0 |
nM |
10.1016/j.bmc.2012.01.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
600.0 |
nM |
10.1016/j.bmc.2015.07.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
600.0 |
nM |
10.1016/j.bmc.2022.116938 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
600.0 |
nM |
10.1021/jm101510d |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
600.0 |
nM |
10.1039/C9MD00347A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
620.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
625.0 |
nM |
10.1021/jm500571f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
640.0 |
nM |
10.1016/j.ejmech.2021.113266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1007/s00044-011-9638-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1016/j.bmc.2014.06.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1016/j.bmc.2014.10.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1016/j.bmc.2015.02.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1016/j.bmc.2015.03.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1016/j.bmc.2016.01.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1016/j.bmc.2016.09.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1016/j.bmc.2017.12.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1016/j.bmcl.2011.03.079 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1016/j.bmcl.2020.127512 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1016/j.ejmech.2015.06.032 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
660.0 |
nM |
10.1016/j.ejmech.2016.06.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
670.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
670.0 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
700.0 |
nM |
10.1016/j.bmcl.2015.10.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
700.0 |
nM |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.bmc.2014.01.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.bmc.2014.05.038 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.bmc.2014.08.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.bmc.2016.01.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.bmc.2016.07.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.bmc.2017.11.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.bmcl.2007.01.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.bmcl.2010.06.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.bmcl.2011.07.062 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.bmcl.2012.10.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.bmcl.2013.01.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.bmcl.2017.01.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.ejmech.2013.08.036 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.ejmech.2014.02.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.ejmech.2014.09.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.ejmech.2014.12.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.ejmech.2016.03.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
720.0 |
nM |
10.1016/j.ejmech.2021.113266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
729.0 |
nM |
10.1021/acsmedchemlett.5b00176 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
729.0 |
nM |
10.1039/C5MD00346F |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
730.0 |
nM |
10.1016/j.bmc.2016.06.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
730.0 |
nM |
10.1016/j.bmc.2019.02.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
730.0 |
nM |
10.1016/j.bmcl.2006.05.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
730.0 |
nM |
10.1016/j.bmcl.2007.04.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
730.0 |
nM |
10.1016/j.bmcl.2011.01.122 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
730.0 |
nM |
10.1016/j.bmcl.2015.11.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
730.0 |
nM |
10.1016/j.ejmech.2015.05.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
730.0 |
nM |
10.1021/acsmedchemlett.5b00367 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
730.0 |
nM |
10.1039/C3MD00251A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
740.0 |
nM |
10.1016/j.bmcl.2022.128604 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
750.0 |
nM |
10.1016/j.bmcl.2009.10.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
780.0 |
nM |
10.1016/j.bmcl.2011.06.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
780.0 |
nM |
10.1016/j.bmcl.2011.07.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
780.0 |
nM |
10.1016/j.ejmech.2017.12.088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
790.0 |
nM |
10.1016/j.bmcl.2017.05.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
800.0 |
nM |
10.1016/j.bmc.2018.04.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
800.0 |
nM |
10.1016/j.bmcl.2013.06.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
810.0 |
nM |
10.1016/j.ejmech.2012.01.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
810.0 |
nM |
10.1016/j.ejmech.2013.11.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
810.0 |
nM |
10.1039/C7MD00146K |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
850.0 |
nM |
10.1016/j.ejmech.2013.11.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
880.0 |
nM |
10.1007/s00044-011-9788-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
880.0 |
nM |
10.1016/j.ejmech.2018.01.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
900.0 |
nM |
10.1016/j.bmcl.2016.05.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
910.0 |
nM |
10.1016/j.bmc.2007.05.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
910.0 |
nM |
10.1016/j.bmc.2014.10.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
910.0 |
nM |
10.1016/j.bmcl.2019.07.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
910.0 |
nM |
10.1016/j.ejmech.2019.111578 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.bmc.2007.01.051 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.bmc.2007.02.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.bmc.2008.12.070 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.bmc.2013.12.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.bmc.2014.05.064 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.bmc.2015.10.029 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.bmc.2017.01.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.bmc.2017.01.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.bmc.2018.07.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.bmcl.2017.10.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2008.06.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2010.02.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2011.09.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2012.01.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2016.02.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2016.11.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2018.04.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2019.111578 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/j.ejmech.2021.113668 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1016/s0960-894x(02)00697-2 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1021/jm00226a007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1039/C4MD00301B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1000.0 |
nM |
10.1039/D1MD00239B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1100.0 |
nM |
10.1021/jm00226a007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1170.0 |
nM |
10.1016/j.ejmech.2015.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1170.0 |
nM |
10.1016/j.ejmech.2017.03.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1200.0 |
nM |
10.1021/acs.jmedchem.9b01457 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1300.0 |
nM |
10.1016/j.ejmech.2011.05.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1400.0 |
nM |
10.1016/j.bmcl.2020.127558 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1400.0 |
nM |
10.1016/j.ejmech.2020.112358 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1400.0 |
nM |
10.1021/np800778b |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1450.0 |
nM |
10.1016/j.bmcl.2016.11.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1450.0 |
nM |
10.1016/j.ejmech.2011.07.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1450.0 |
nM |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1460.0 |
nM |
10.1016/j.bmcl.2005.11.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1460.0 |
nM |
10.1021/acsmedchemlett.5b00324 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1500.0 |
nM |
10.1016/j.bmc.2014.11.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1500.0 |
nM |
10.1016/j.ejmech.2010.04.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1800.0 |
nM |
10.1016/j.bmcl.2010.01.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1800.0 |
nM |
10.1016/j.bmcl.2010.08.127 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1800.0 |
nM |
10.1016/j.bmcl.2011.08.076 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1800.0 |
nM |
10.1016/j.bmcl.2019.07.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1800.0 |
nM |
10.1016/j.bmcl.2020.127192 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1800.0 |
nM |
10.1016/j.ejmech.2017.12.075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1800.0 |
nM |
10.1016/j.ejmech.2018.01.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1800.0 |
nM |
10.1021/acs.jmedchem.8b01356 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1800.0 |
nM |
10.1021/acsmedchemlett.9b00204 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1820.0 |
nM |
10.1016/j.bmc.2014.10.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2000.0 |
nM |
10.1016/j.bmcl.2015.08.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2000.0 |
nM |
10.1016/j.ejmech.2019.111935 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2000.0 |
nM |
10.1016/j.ejmech.2020.112408 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2040.0 |
nM |
10.1016/j.bmcl.2005.07.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2200.0 |
nM |
10.1016/j.ejmech.2020.112859 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2300.0 |
nM |
10.1021/acsmedchemlett.2c00254 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2600.0 |
nM |
10.1016/j.bmcl.2015.04.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2800.0 |
nM |
10.1039/C5MD00178A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2840.0 |
nM |
10.1016/j.ejmech.2018.06.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2900.0 |
nM |
10.1016/j.ejmech.2018.06.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2900.0 |
nM |
10.1021/acs.jnatprod.9b00475 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2900.0 |
nM |
10.1021/np800778b |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2920.0 |
nM |
10.1016/j.ejmech.2022.114454 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2989.0 |
nM |
10.1021/acsmedchemlett.5b00176 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3000.0 |
nM |
10.1016/j.bmcl.2013.12.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3200.0 |
nM |
10.1021/np900281r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3600.0 |
nM |
10.1016/j.ejmech.2013.11.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3600.0 |
nM |
10.1016/j.ejmech.2016.10.014 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3650.0 |
nM |
10.1016/j.bmc.2014.10.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
3650.0 |
nM |
10.1016/j.ejmech.2020.112898 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2019.111935 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
4000.0 |
nM |
10.1016/j.ejmech.2020.112408 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
5000.0 |
nM |
10.1021/jm5002937 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
5250.0 |
nM |
10.1016/j.ejmech.2014.06.075 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7200.0 |
nM |
10.1016/j.bmcl.2017.01.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7250.0 |
nM |
10.1021/jm5005978 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7290.0 |
nM |
10.1016/j.ejmech.2020.112898 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7300.0 |
nM |
10.1016/j.bmc.2012.08.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7300.0 |
nM |
10.1016/j.ejmech.2015.07.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7300.0 |
nM |
10.1016/j.ejmech.2017.03.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7300.0 |
nM |
10.1016/j.ejmech.2020.112699 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7500.0 |
nM |
10.1021/ml5001933 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
7800.0 |
nM |
10.1021/acs.jmedchem.1c00837 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8000.0 |
nM |
10.1016/j.bmc.2010.08.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8000.0 |
nM |
10.1016/j.bmcl.2015.12.083 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8000.0 |
nM |
10.1016/j.ejmech.2013.11.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8000.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8000.0 |
nM |
10.1016/j.ejmech.2019.111935 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8000.0 |
nM |
10.1016/j.ejmech.2020.112408 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
8000.0 |
nM |
10.1039/C7MD00146K |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
9110.0 |
nM |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
10930.0 |
nM |
10.1016/j.ejmech.2020.112967 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
11000.0 |
nM |
10.1016/j.bmcl.2012.11.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
11370.0 |
nM |
10.1016/j.bmcl.2006.05.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
11370.0 |
nM |
10.1016/j.bmcl.2007.04.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
11380.0 |
nM |
10.1016/j.ejmech.2009.05.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
11380.0 |
nM |
10.1016/j.ejmech.2012.04.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
11400.0 |
nM |
10.1016/j.bmcl.2009.10.107 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
11570.0 |
nM |
10.1016/j.bmcl.2009.10.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12500.0 |
nM |
10.1016/j.bmc.2012.01.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12500.0 |
nM |
10.1016/j.bmc.2015.07.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12500.0 |
nM |
10.1016/j.bmc.2018.04.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12500.0 |
nM |
10.1016/j.bmcl.2011.06.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12500.0 |
nM |
10.1016/j.bmcl.2011.07.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12500.0 |
nM |
10.1016/j.ejmech.2010.04.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
12500.0 |
nM |
10.1016/j.ejmech.2020.112178 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
14600.0 |
nM |
10.1016/j.ejmech.2010.09.040 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
15300.0 |
nM |
10.1016/j.bmcl.2013.09.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16000.0 |
nM |
10.1016/j.bmc.2009.12.055 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16000.0 |
nM |
10.1016/j.bmc.2013.12.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16000.0 |
nM |
10.1016/j.bmc.2017.01.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16000.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16000.0 |
nM |
10.1016/j.ejmech.2016.11.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16000.0 |
nM |
10.1039/C3MD00366C |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
16000.0 |
nM |
10.1039/C5MD00178A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
18000.0 |
nM |
10.1021/jm101510d |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
18230.0 |
nM |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
25000.0 |
nM |
10.1016/j.ejmech.2020.112859 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
29000.0 |
nM |
10.1021/jm5002937 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
29170.0 |
nM |
10.1016/j.ejmech.2020.112898 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
29190.0 |
nM |
10.1016/j.bmc.2007.05.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
31200.0 |
nM |
10.1021/acs.jmedchem.1c00837 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32000.0 |
nM |
10.1016/j.bmc.2017.01.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32000.0 |
nM |
10.1016/j.ejmech.2014.05.069 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32000.0 |
nM |
10.1016/j.ejmech.2016.11.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
32000.0 |
nM |
10.1039/C5MD00178A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
36450.0 |
nM |
10.1016/j.ejmech.2021.113932 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
37300.0 |
nM |
10.1021/acs.jmedchem.9b01457 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40000.0 |
nM |
10.1016/j.bmc.2019.01.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
40000.0 |
nM |
10.1016/j.ejmech.2019.06.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
43800.0 |
nM |
10.1016/j.ejmech.2014.04.077 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45570.0 |
nM |
10.1007/s00044-011-9638-9 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45570.0 |
nM |
10.1016/j.bmc.2007.11.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45570.0 |
nM |
10.1016/j.bmc.2007.11.050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45570.0 |
nM |
10.1016/j.bmc.2014.08.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45570.0 |
nM |
10.1016/j.bmcl.2007.09.095 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45570.0 |
nM |
10.1016/j.bmcl.2011.01.122 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45570.0 |
nM |
10.1016/j.ejmech.2008.02.031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45570.0 |
nM |
10.1016/j.ejmech.2009.09.001 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45570.0 |
nM |
10.1016/j.ejmech.2009.09.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45570.0 |
nM |
10.1016/j.ejmech.2011.09.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45570.0 |
nM |
10.1016/j.ejmech.2014.09.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45570.0 |
nM |
10.1021/jm700999n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45600.0 |
nM |
10.1016/j.ejmech.2012.10.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
45600.0 |
nM |
10.1016/j.ejmech.2018.06.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
58300.0 |
nM |
10.1016/j.bmcl.2017.01.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
58300.0 |
nM |
10.1016/j.ejmech.2010.09.040 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
58380.0 |
nM |
10.1016/j.bmc.2007.05.053 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
58400.0 |
nM |
10.1016/j.ejmech.2018.01.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
62500.0 |
nM |
10.1021/acs.jmedchem.1c00837 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64000.0 |
nM |
10.1016/j.ejmech.2016.11.041 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64000.0 |
nM |
10.1039/C3MD00366C |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
64000.0 |
nM |
10.1039/C7MD00146K |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
70000.0 |
nM |
10.1016/j.ejmech.2016.11.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
70000.0 |
nM |
10.1021/acsmedchemlett.5b00324 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
72900.0 |
nM |
10.1016/j.ejmech.2014.04.077 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
80000.0 |
nM |
10.1016/j.ejmech.2018.01.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
90940.0 |
nM |
10.1016/j.bmcl.2005.11.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
91000.0 |
nM |
10.1016/j.bmc.2015.03.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
91140.0 |
nM |
10.1016/j.bmcl.2010.06.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
91140.0 |
nM |
10.1016/j.bmcl.2016.03.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100000.0 |
nM |
10.1016/j.bmcl.2013.11.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100000.0 |
nM |
10.1016/j.ejmech.2020.112859 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
100000.0 |
nM |
10.1021/jm5002937 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
116800.0 |
nM |
10.1016/j.ejmech.2018.01.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128000.0 |
nM |
10.1016/j.bmc.2011.04.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128000.0 |
nM |
10.1016/j.bmcl.2009.12.062 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128000.0 |
nM |
10.1016/j.bmcl.2011.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128000.0 |
nM |
10.1021/acs.jnatprod.2c01003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128000.0 |
nM |
10.1021/acsmedchemlett.7b00356 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128000.0 |
nM |
10.1021/jm900003c |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128000.0 |
nM |
10.1021/jm901273n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
128000.0 |
nM |
10.1128/aac.00055-06 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
145800.0 |
nM |
10.1021/acsmedchemlett.2c00254 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
182000.0 |
nM |
10.1016/j.bmc.2015.03.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
182300.0 |
nM |
10.1016/j.bmcl.2019.02.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
182300.0 |
nM |
10.1016/j.ejmech.2018.06.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
182310.0 |
nM |
10.1016/j.ejmech.2010.10.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200000.0 |
nM |
10.1016/j.bmc.2017.09.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200000.0 |
nM |
10.1016/j.ejmech.2017.07.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
200000.0 |
nM |
10.1021/acsmedchemlett.6b00088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
233000.0 |
nM |
10.1016/j.bmcl.2019.07.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
256000.0 |
nM |
10.1016/j.bmc.2013.11.011 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
291700.0 |
nM |
10.1021/acsmedchemlett.2c00254 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
364670.0 |
nM |
10.1016/j.bmcl.2011.07.062 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
467000.0 |
nM |
10.1016/j.ejmech.2010.11.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
729000.0 |
nM |
10.1021/jm101510d |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
729100.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
729200.0 |
nM |
10.1016/j.ejmech.2018.06.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
1900000.0 |
nM |
10.1021/jm00226a007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
2187500.0 |
nM |
10.1016/j.ejmech.2018.02.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
ug.mL-1 |
10.1016/j.bmcl.2005.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
ug.mL-1 |
10.1016/s0960-894x(00)00159-1 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1007/s00044-013-0472-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1016/j.bmcl.2016.03.107 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1016/j.bmcl.2018.05.049 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1016/j.ejmech.2014.09.028 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1021/acs.jmedchem.6b00031 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1039/C3MD00366C |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1039/D1MD00239B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC |
nan |
None |
10.1128/aac.01486-07 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC100 |
0.04 |
ug ml-1 |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC100 |
0.1 |
ug ml-1 |
10.1016/j.bmc.2014.12.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC100 |
0.12 |
ug ml-1 |
10.1016/j.bmc.2014.12.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC100 |
1.25 |
uM |
10.1021/acs.jnatprod.5b00266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.019 |
ug.mL-1 |
10.1016/j.bmcl.2018.03.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.024 |
ug.mL-1 |
10.1016/j.bmcl.2022.128824 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.024 |
ug.mL-1 |
10.1016/j.bmcl.2022.128871 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.03 |
ug.mL-1 |
10.1021/acs.jnatprod.0c00864 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.07 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.125 |
ug.mL-1 |
10.1021/jm701560p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.25 |
ug.mL-1 |
10.1021/jm030479g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.8 |
ug.mL-1 |
10.1016/j.bmcl.2020.127351 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.8 |
ug.mL-1 |
10.1016/j.bmcl.2021.128261 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.9 |
ug.mL-1 |
10.1016/j.bmcl.2020.127351 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
0.9 |
ug.mL-1 |
10.1016/j.bmcl.2021.128261 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm100165w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
1.0 |
ug.mL-1 |
10.1021/jm100568q |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
4.205 |
ug.mL-1 |
10.1016/j.bmcl.2022.128824 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
4.374 |
ug.mL-1 |
10.1016/j.bmcl.2022.128871 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
30.0 |
nM |
10.1016/j.ejmech.2011.10.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
30.0 |
nM |
10.1016/j.ejmech.2015.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
41.0 |
ug.mL-1 |
10.1021/jm050765n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
60.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
90.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
100.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
100.0 |
nM |
10.1016/j.ejmech.2013.03.023 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
120.0 |
ug.mL-1 |
10.1021/jm050765n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
200.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
330.0 |
nM |
10.1016/j.ejmech.2015.10.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
330.0 |
nM |
10.1021/jm4012774 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
465.0 |
nM |
10.1016/j.ejmech.2011.12.035 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
540.0 |
nM |
10.1016/j.ejmech.2011.11.033 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
1300.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
1600.0 |
nM |
10.1021/acs.jmedchem.1c01383 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
1800.0 |
nM |
10.1021/acsmedchemlett.0c00588 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC50 |
nan |
None |
10.1021/jm051060o |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
0.02 |
uM |
10.1021/acs.jmedchem.6b01358 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
0.03 |
ug ml-1 |
10.1021/jm500833f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
0.03 |
uM |
10.1021/acs.jmedchem.6b01358 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
0.06 |
ug ml-1 |
10.1021/jm500833f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
0.2 |
uM |
10.1039/C5MD00589B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
15.0 |
uM |
10.1039/C5MD00589B |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>80 |
16.0 |
ug ml-1 |
10.1021/jm500833f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC80 |
200.0 |
nM |
10.1016/j.ejmech.2016.09.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC80 |
200.0 |
nM |
10.1016/j.ejmech.2017.05.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC80 |
449.0 |
nM |
10.1021/jm5003606 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC80 |
490.0 |
nM |
10.1016/j.ejmech.2016.09.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC80 |
490.0 |
nM |
10.1016/j.ejmech.2017.05.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC80 |
617.0 |
nM |
10.1021/jm5003606 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=<90 |
0.04 |
ug ml-1 |
10.1016/j.ejmech.2021.113202 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=<90 |
0.04 |
ug ml-1 |
10.1021/acs.jmedchem.7b00582 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=<90 |
0.04 |
ug ml-1 |
10.1021/acs.jmedchem.8b01578 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=<90 |
8.0 |
ug ml-1 |
10.1016/j.ejmech.2021.113202 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=<90 |
16.0 |
ug ml-1 |
10.1016/j.ejmech.2021.113202 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.02 |
ug ml-1 |
10.1016/j.bmcl.2021.127924 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.031 |
ug ml-1 |
10.1016/j.ejmech.2019.111595 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.035 |
ug ml-1 |
10.1016/j.ejmech.2018.09.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.037 |
ug ml-1 |
10.1016/j.ejmech.2018.03.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.037 |
ug ml-1 |
10.1021/acsmedchemlett.7b00068 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.04 |
ug ml-1 |
10.1021/acs.jmedchem.2c00718 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.049 |
ug ml-1 |
10.1016/j.bmcl.2015.10.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.05 |
ug ml-1 |
10.1016/j.ejmech.2015.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.1 |
ug ml-1 |
10.1016/j.ejmech.2016.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.1 |
uM |
10.1016/j.ejmech.2015.05.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.239 |
ug ml-1 |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.36 |
uM |
10.1016/j.ejmech.2017.05.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.438 |
ug ml-1 |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
0.5 |
mg/L |
10.1016/j.bmcl.2015.09.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
1.0 |
mg/L |
10.1016/j.bmcl.2015.09.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
2.04 |
uM |
10.1021/acs.jnatprod.5b00650 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
2.46 |
ug ml-1 |
10.1016/j.ejmech.2020.112420 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
2.5 |
ug ml-1 |
10.1021/acsmedchemlett.7b00068 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
3.64 |
uM |
10.1016/j.ejmech.2019.01.073 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
4.0 |
mg/L |
10.1016/j.bmcl.2015.09.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
4.0 |
ug ml-1 |
10.1016/j.bmcl.2015.10.027 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
4.0 |
ug ml-1 |
10.1016/j.ejmech.2015.09.030 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
8.0 |
ug ml-1 |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
19.47 |
ug ml-1 |
10.1016/j.ejmech.2018.09.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
40.0 |
ug ml-1 |
10.1016/j.ejmech.2018.03.060 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
40.0 |
ug ml-1 |
10.1016/j.ejmech.2018.09.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
40.0 |
ug ml-1 |
10.1016/j.ejmech.2019.111595 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
40.0 |
ug ml-1 |
10.1021/acsmedchemlett.7b00068 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
58.0 |
uM |
10.1016/j.bmc.2015.03.018 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
200.0 |
uM |
10.1016/j.ejmech.2019.01.073 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC=>90 |
291.0 |
uM |
10.1016/j.ejmech.2017.05.044 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.03 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.035 |
ug ml-1 |
10.1016/j.bmcl.2018.07.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.04 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.049 |
ug ml-1 |
10.1021/acsmedchemlett.6b00330 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.0781 |
ug ml-1 |
10.1021/acsmedchemlett.8b00177 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.1 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.277 |
uM |
10.1016/j.ejmech.2018.12.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.284 |
uM |
10.1021/acsmedchemlett.7b00106 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.39 |
ug ml-1 |
10.1016/j.ejmech.2014.01.024 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
0.9 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
1.1 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
4.7 |
uM |
10.1039/C0MD00246A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
34.48 |
uM |
10.1021/acsmedchemlett.7b00106 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
40.0 |
ug ml-1 |
10.1016/j.bmcl.2018.07.046 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
40.0 |
ug ml-1 |
10.1021/acsmedchemlett.8b00177 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
40.0 |
uM |
10.1016/j.ejmech.2018.12.071 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
140.4 |
ug ml-1 |
10.1021/np400145u |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>90 |
291.7 |
uM |
10.1021/acsmedchemlett.7b00106 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.005 |
ug.mL-1 |
10.1021/acs.jmedchem.1c01349 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.025 |
ug.mL-1 |
10.1016/j.bmcl.2007.09.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.03 |
ug.mL-1 |
10.1016/j.bmcl.2016.06.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.03 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.03 |
ug.mL-1 |
10.1021/acs.jmedchem.1c01349 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.03 |
ug.mL-1 |
10.1021/np400497f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.032 |
ug.mL-1 |
10.1016/j.bmcl.2022.128824 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.034 |
ug.mL-1 |
10.1016/j.bmcl.2022.128871 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.04 |
ug.mL-1 |
10.1021/acs.jmedchem.0c01372 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.04 |
ug.mL-1 |
10.1021/acs.jmedchem.2c01064 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.04 |
ug.mL-1 |
10.1021/np400497f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2017.05.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.05 |
ug.mL-1 |
10.1016/j.ejmech.2018.07.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.05 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.06 |
ug.mL-1 |
10.1021/jm300123s |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.0625 |
ug.mL-1 |
10.1016/j.bmcl.2011.12.022 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.07 |
ug.mL-1 |
10.1021/np400497f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.074 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.075 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.091 |
ug.mL-1 |
10.1021/jm300123s |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.11 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.11 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.083 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.11 |
ug.mL-1 |
10.1016/j.ejmech.2022.114404 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.2 |
ug.mL-1 |
10.1007/s00044-011-9718-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.25 |
ug.mL-1 |
10.1016/j.ejmech.2019.111713 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.25 |
ug.mL-1 |
10.1021/jm701560p |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
0.33 |
ug.mL-1 |
10.1016/j.bmcl.2012.05.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
2.19 |
ug.mL-1 |
10.1021/np400497f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
10.0 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
20.0 |
ug.mL-1 |
10.1021/jm300123s |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
25.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.042 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
25.0 |
ug.mL-1 |
10.1016/j.ejmech.2022.114404 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
40.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128824 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
40.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128871 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
90.0 |
nM |
10.1016/j.ejmech.2013.06.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
100.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
110.0 |
nM |
10.1016/j.ejmech.2016.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
128.0 |
ug.mL-1 |
10.1016/j.bmcl.2012.05.096 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.05.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2018.07.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
128.0 |
ug.mL-1 |
10.1021/acsmedchemlett.8b00410 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
200.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
200.0 |
nM |
10.1016/j.bmcl.2011.08.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
200.0 |
nM |
10.1016/j.ejmech.2021.113207 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
200.0 |
nM |
10.1039/C8MD00480C |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
220.0 |
nM |
10.1016/j.bmc.2012.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
220.0 |
nM |
10.1021/acs.jmedchem.7b00793 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
230.0 |
nM |
10.1016/j.ejmech.2012.08.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
230.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
230.0 |
nM |
10.1021/ml200036r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
240.0 |
nM |
10.1016/j.bmc.2016.12.038 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
240.0 |
nM |
10.1021/jm201716n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
280.0 |
nM |
10.1016/j.ejmech.2021.113734 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
280.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
290.0 |
nM |
10.1016/j.ejmech.2021.113734 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
290.0 |
nM |
10.1021/jm4003878 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
300.0 |
nM |
10.1016/j.ejmech.2017.06.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
300.0 |
nM |
10.1016/j.ejmech.2019.111812 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
300.0 |
nM |
10.1016/j.ejmech.2022.114201 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
310.0 |
nM |
10.1016/j.bmcl.2014.01.007 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
310.0 |
nM |
10.1016/j.ejmech.2013.09.061 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
310.0 |
nM |
10.1016/j.ejmech.2019.07.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
350.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
370.0 |
nM |
10.1016/j.bmc.2012.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
390.0 |
nM |
10.1016/j.bmcl.2011.08.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
400.0 |
nM |
10.1007/s00044-007-9073-0 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
400.0 |
nM |
10.1016/j.bmcl.2013.09.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
400.0 |
nM |
10.1016/j.ejmech.2022.114201 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
410.0 |
nM |
10.1016/j.ejmech.2017.05.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
430.0 |
nM |
10.1021/ml200036r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
463.0 |
nM |
10.1021/acs.jnatprod.1c00198 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
550.0 |
nM |
10.1016/j.ejmech.2021.113734 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
620.0 |
nM |
10.1016/j.ejmech.2021.113734 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
625.0 |
nM |
10.1021/acs.jnatprod.5b00266 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
730.0 |
nM |
10.1016/j.bmcl.2012.06.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
730.0 |
nM |
10.1016/j.bmcl.2012.10.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
740.0 |
nM |
10.1007/s00044-012-9971-7 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
780.0 |
nM |
10.1016/j.bmcl.2011.10.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
800.0 |
nM |
10.1016/j.bmcl.2019.02.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
840.0 |
nM |
10.1021/jm900513a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1108.4 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
1800.0 |
nM |
10.1039/d2md00155a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
3200.0 |
nM |
10.1021/acs.jmedchem.1c01383 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
3800.0 |
nM |
10.1021/acsmedchemlett.0c00588 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
5000.0 |
nM |
10.1016/j.ejmech.2017.05.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
5000.0 |
nM |
10.1021/acs.jmedchem.7b01332 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
6300.0 |
nM |
10.1016/j.ejmech.2022.114201 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
8000.0 |
nM |
10.1021/ml200036r |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
9800.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
11230.0 |
nM |
10.1016/j.bmcl.2012.06.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
11230.0 |
nM |
10.1016/j.bmcl.2012.10.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
11580.0 |
nM |
10.1016/j.bmcl.2011.10.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
13000.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
100000.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
116800.0 |
nM |
10.1016/j.ejmech.2015.05.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
128000.0 |
nM |
10.1016/j.bmcl.2011.08.054 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
128000.0 |
nM |
10.1016/j.ejmech.2012.08.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
128000.0 |
nM |
10.1021/jm201716n |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
128000.0 |
nM |
10.1021/jm900513a |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
256000.0 |
nM |
10.1016/j.ejmech.2017.05.026 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
467100.0 |
nM |
10.1016/j.ejmech.2015.05.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
512000.0 |
nM |
10.1016/j.bmc.2012.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
nan |
None |
10.1016/j.bmc.2012.02.025 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
nan |
None |
10.1016/j.ejmech.2015.05.020 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
nan |
None |
10.1016/j.ejmech.2016.07.039 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC90 |
nan |
None |
10.1021/acs.jmedchem.7b00793 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC95 |
0.06 |
ug ml-1 |
10.1016/j.bmc.2017.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC95 |
0.1 |
ug ml-1 |
10.1016/j.bmc.2006.12.009 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC95 |
0.1 |
ug ml-1 |
10.1016/j.bmc.2008.06.057 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC95 |
0.25 |
ug ml-1 |
10.1016/j.ejmech.2009.01.017 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC95 |
1.8 |
uM |
10.1016/j.ejmech.2010.09.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC95 |
4.4 |
uM |
10.1016/j.ejmech.2010.09.048 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
0.15 |
uM |
10.1016/j.ejmech.2020.112659 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
0.5 |
uM |
10.1016/j.bmc.2017.08.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
0.5 |
uM |
10.1016/j.ejmech.2017.02.058 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
0.5 |
uM |
10.1021/acs.jmedchem.5b00608 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
0.5 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
1.0 |
uM |
10.1016/j.ejmech.2017.02.058 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
1.0 |
uM |
10.1021/acs.jmedchem.5b00608 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
1.0 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
16.0 |
uM |
10.1016/j.bmc.2017.08.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
16.0 |
uM |
10.1021/acs.jmedchem.5b00608 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
16.0 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
32.0 |
uM |
10.1016/j.bmc.2017.08.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
32.0 |
uM |
10.1021/acs.jmedchem.5b00608 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
32.0 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
64.0 |
uM |
10.1016/j.bmc.2017.08.010 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
64.0 |
uM |
10.1021/acs.jmedchem.5b00608 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC>99 |
64.0 |
uM |
10.1021/acs.jmedchem.9b00912 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.02 |
ug ml-1 |
10.1016/j.bmc.2019.115050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.05 |
ug ml-1 |
10.1016/j.ejmech.2016.09.083 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.05 |
ug ml-1 |
10.1021/jm201023g |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.07 |
ug ml-1 |
10.1016/j.bmc.2019.115050 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.098 |
ug ml-1 |
10.1016/j.bmcl.2016.04.012 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.098 |
ug ml-1 |
10.1016/j.bmcl.2016.10.082 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.098 |
ug ml-1 |
10.1039/C4MD00224E |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.1 |
ug ml-1 |
10.1016/j.bmc.2012.09.019 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.1 |
ug ml-1 |
10.1016/j.bmc.2013.07.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.1 |
ug ml-1 |
10.1016/j.ejmech.2014.07.100 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.1 |
ug ml-1 |
10.1016/j.ejmech.2015.01.013 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.1 |
ug ml-1 |
10.1016/j.ejmech.2015.02.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.1 |
uM |
10.1016/j.ejmech.2021.113843 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.13 |
uM |
10.1021/jm401735w |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.15 |
uM |
10.1016/j.ejmech.2020.112450 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.18 |
uM |
10.1021/acs.jmedchem.7b01347 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.18 |
uM |
10.1021/jm051060o |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.18 |
uM |
10.1021/jm061068d |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.19 |
uM |
10.1016/j.ejmech.2020.112772 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.2 |
ug ml-1 |
10.1007/s00044-011-9942-4 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.2 |
ug ml-1 |
10.1007/s00044-012-0273-x |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.2 |
ug ml-1 |
10.1016/j.bmcl.2012.06.072 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.2 |
ug ml-1 |
10.1016/j.ejmech.2014.03.085 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.2 |
uM |
10.1016/j.ejmech.2020.112450 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.3 |
uM |
10.1021/ml400088y |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.36 |
ug ml-1 |
10.1016/j.bmcl.2013.10.016 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.36 |
ug ml-1 |
10.1016/j.ejmech.2014.01.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.36 |
uM |
10.1016/j.bmcl.2007.11.110 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.36 |
uM |
10.1021/acs.jmedchem.7b01347 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.39 |
uM |
10.1016/j.ejmech.2014.05.005 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.39 |
uM |
10.1039/C4MD00288A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.4 |
uM |
10.1016/j.bmcl.2017.02.021 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.4 |
uM |
10.1039/C0MD00239A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.73 |
uM |
10.1016/j.bmc.2017.12.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.78 |
uM |
10.1016/j.bmcl.2021.128236 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
0.78 |
uM |
10.1039/C4MD00303A |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
1.0 |
ug ml-1 |
10.1016/j.ejmech.2008.10.004 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
1.86 |
uM |
10.1016/j.ejmech.2017.07.059 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
2.5 |
uM |
10.1016/j.bmc.2017.12.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
10.0 |
uM |
10.1016/j.bmc.2017.12.047 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
45.57 |
uM |
10.1016/j.bmcl.2007.11.110 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MIC99 |
nan |
None |
10.1016/j.bmc.2013.07.003 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MST |
29.0 |
day |
10.1039/C5MD00131E |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MST |
30.0 |
day |
10.1016/j.ejmech.2011.06.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MST |
30.0 |
None |
10.1016/j.ejmech.2010.09.063 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MST |
40.0 |
day |
10.1016/j.ejmech.2011.06.037 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
MST |
40.0 |
None |
10.1016/j.ejmech.2010.09.063 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
pMIC |
4.2 |
None |
10.1021/jm049913k |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
1.0 |
None |
10.1016/j.bmcl.2011.08.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
1.0 |
None |
10.1021/jm500833f |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
1.6 |
None |
10.1016/j.ejmech.2018.02.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
3.1 |
None |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
6.25 |
None |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
15.6 |
None |
10.1016/j.bmc.2018.04.045 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
20.0 |
None |
10.1128/aac.00453-10 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
21.0 |
None |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
25.0 |
None |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
31.0 |
None |
10.1021/acs.jmedchem.9b01457 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
50.0 |
None |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
100.0 |
None |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
400.0 |
None |
10.1016/j.ejmech.2016.02.008 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
nan |
None |
10.1016/j.bmcl.2005.03.065 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio |
nan |
None |
10.1016/j.ejmech.2018.02.067 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Ratio IC50 |
1.0 |
None |
10.1016/j.bmcl.2011.08.052 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Selectivity Index |
0.2 |
None |
10.1021/acs.jmedchem.1c01349 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Selectivity ratio |
4.0 |
None |
10.1021/acs.jmedchem.6b01358 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Selectivity ratio |
2500.0 |
None |
10.1016/j.bmc.2018.07.034 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Survival |
100.0 |
% |
10.1016/j.ejmech.2010.09.063 |
| Mycobacterium tuberculosis |
Mycobacterium tuberculosis |
Survival |
100.0 |
% |
10.1016/j.ejmech.2011.06.037 |
| Mycobacterium tuberculosis |
O-acetylserine sulfhydrylase |
Inhibition |
nan |
% |
10.1016/j.bmcl.2013.01.031 |
| Mycobacterium tuberculosis |
Pantothenate synthetase |
IC50 |
25000.0 |
nM |
10.1016/j.bmc.2014.01.030 |
| Mycobacterium tuberculosis |
Pantothenate synthetase |
IC50 |
25000.0 |
nM |
10.1016/j.bmc.2014.05.038 |
| Mycobacterium tuberculosis |
Pantothenate synthetase |
IC50 |
25000.0 |
nM |
10.1016/j.bmc.2016.01.059 |
| Mycobacterium tuberculosis |
Pantothenate synthetase |
Inhibition |
0.0 |
% |
10.1016/j.ejmech.2013.08.036 |
| Mycobacterium tuberculosis H37Rv |
Mycobacterium tuberculosis H37Rv |
MIC50 |
1200.0 |
nM |
10.1016/j.ejmech.2020.112908 |
| Mycobacterium tuberculosis H37Rv |
Mycobacterium tuberculosis H37Rv |
MIC90 |
290.0 |
nM |
10.1016/j.ejmech.2021.113734 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
50000.0 |
nM |
10.1016/j.bmc.2016.01.011 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.bmc.2014.06.041 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.bmc.2014.10.016 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.bmc.2015.03.004 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.ejmech.2015.06.032 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
nan |
None |
10.1016/j.ejmech.2016.08.034 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
DNA gyrase subunit A/DNA gyrase subunit B |
IC50 |
nan |
None |
10.1021/ml500531p |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
FAD-dependent decaprenylphosphoryl-beta-D-ribofuranose 2-oxidase |
MIC |
0.019 |
ug.mL-1 |
10.1021/acs.jmedchem.1c00263 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
Polyketide synthase Pks13 |
MIC=<90 |
0.04 |
ug ml-1 |
10.1021/acs.jmedchem.9b00010 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
Polyketide synthase Pks13 |
MIC=<90 |
8.0 |
ug ml-1 |
10.1021/acs.jmedchem.9b00010 |
| Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
Polyketide synthase Pks13 |
MIC=<90 |
16.0 |
ug ml-1 |
10.1021/acs.jmedchem.9b00010 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
Activity |
2.6 |
None |
10.1016/j.ejmech.2016.07.068 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
Activity |
nan |
None |
10.1016/j.ejmech.2016.07.068 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
Activity |
nan |
None |
10.1021/acs.jmedchem.6b01530 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
Activity |
nan |
None |
10.1039/d2md00251e |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
IC50 |
0.021 |
ug.mL-1 |
10.1016/j.bmc.2023.117212 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
IC50 |
0.036 |
ug.mL-1 |
10.1016/j.bmc.2023.117212 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
IC50 |
3000.0 |
nM |
None |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
Inhibition |
100.0 |
% |
10.1016/j.ejmech.2022.114831 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MBC99.9 |
10.0 |
uM |
10.1021/acsmedchemlett.0c00588 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.015 |
ug.mL-1 |
10.1016/j.ejmech.2017.04.002 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.06 |
ug.mL-1 |
10.1128/aac.01302-08 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.063 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.042 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.1 |
ug.mL-1 |
10.1128/aac.01302-08 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.125 |
ug.mL-1 |
10.1128/aac.01302-08 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
0.4 |
ug.mL-1 |
10.1128/aac.01302-08 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
80.0 |
nM |
10.1021/jm401735w |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
1000.0 |
nM |
10.1039/D1MD00239B |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC |
7300.0 |
nM |
10.1016/j.bmcl.2016.05.053 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC50 |
100.0 |
nM |
10.1016/j.ejmech.2013.03.023 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC90 |
100.0 |
nM |
10.1016/j.ejmech.2017.06.061 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC90 |
6250.0 |
nM |
10.1016/j.ejmech.2016.07.068 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC90 |
12520.0 |
nM |
10.1016/j.bmcl.2019.126671 |
| Mycobacterium tuberculosis variant bovis |
Mycobacterium tuberculosis variant bovis |
MIC99 |
0.1 |
ug ml-1 |
10.1016/j.bmcl.2005.05.119 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
Activity |
25.0 |
% |
10.1021/acs.jmedchem.8b00832 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
FC |
100.0 |
None |
10.1021/acs.jmedchem.8b00777 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
IC50 |
0.0012 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
IC50 |
0.0017 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
IC50 |
0.0023 |
ug.mL-1 |
10.1016/j.bmcl.2015.11.071 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.033 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.037 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.043 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.045 |
ug.mL-1 |
10.1016/j.bmcl.2015.11.071 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
0.1 |
ug.mL-1 |
10.1021/jm070638m |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
410.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
500.0 |
nM |
10.1021/ml5003458 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC |
730.0 |
nM |
10.1039/C3MD00251A |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC50 |
1600.0 |
nM |
10.1021/acs.jmedchem.1c01383 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC90 |
0.0078 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC90 |
0.075 |
ug.mL-1 |
10.1021/acsmedchemlett.6b00077 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC90 |
3200.0 |
nM |
10.1021/acs.jmedchem.1c01383 |
| Mycobacterium tuberculosis variant bovis BCG |
Mycobacterium tuberculosis variant bovis BCG |
MIC95 |
0.4 |
ug ml-1 |
10.1016/j.ejmech.2009.01.017 |
| Mycobacterium tuberculosis variant microti |
Mycobacterium tuberculosis variant microti |
MIC |
22820.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
MIC |
40.0 |
ug.mL-1 |
10.1128/aac.00400-10 |
| Mycobacterium ulcerans |
Mycobacterium ulcerans |
MIC50 |
390.0 |
nM |
10.1016/j.ejmech.2013.03.023 |
| Mycobacterium xenopi |
Mycobacterium xenopi |
MIC |
12.5 |
ug.mL-1 |
10.1007/s00044-012-0458-3 |
| Mycobacterium xenopi |
Mycobacterium xenopi |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2010.07.020 |
| Mycobacterium xenopi |
Mycobacterium xenopi |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.080 |
| Mycobacterium xenopi |
Mycobacterium xenopi |
MIC |
64.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
Activity |
26.0 |
CFU |
10.1016/j.ejmech.2015.07.001 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
Activity |
nan |
None |
10.1016/j.bmcl.2022.128692 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
Activity |
nan |
None |
10.1016/j.ejmech.2017.03.047 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
8000.0 |
nM |
10.1021/acs.jnatprod.9b01095 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
62500.0 |
nM |
10.1039/D1MD00239B |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
291800.0 |
nM |
10.1016/j.ejmech.2015.07.001 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
291800.0 |
nM |
10.1016/j.ejmech.2017.03.047 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
500000.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
nan |
None |
10.1016/j.bmc.2022.116777 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
nan |
None |
10.1016/j.ejmech.2018.08.070 |
| Mycobacteroides abscessus |
Mycobacteroides abscessus |
MIC |
nan |
None |
10.1016/j.ejmech.2020.112996 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
12.5 |
ug.mL-1 |
10.1007/s00044-012-0458-3 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2010.07.020 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.080 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
400.0 |
ug.mL-1 |
10.1128/aac.00590-09 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
500000.0 |
nM |
10.1016/j.bmcl.2014.05.062 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
nan |
None |
10.1016/j.bmc.2013.10.011 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
nan |
None |
10.1016/j.bmc.2022.116777 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
nan |
None |
10.1016/j.ejmech.2018.08.070 |
| Mycobacteroides chelonae |
Mycobacteroides chelonae |
MIC |
nan |
None |
10.1016/j.ejmech.2020.112996 |
| Mycolicibacterium aurum |
Mycolicibacterium aurum |
MIC |
2.0 |
ug.mL-1 |
10.1021/np049706n |
| Mycolicibacterium aurum |
Mycolicibacterium aurum |
MIC |
3.91 |
ug.mL-1 |
10.1016/j.ejmech.2019.111578 |
| Mycolicibacterium aurum |
Mycolicibacterium aurum |
MIC |
6.3 |
ug.mL-1 |
10.1021/jm070638m |
| Mycolicibacterium diernhoferi |
Mycolicibacterium diernhoferi |
MIC |
0.25 |
ug.mL-1 |
10.1021/np2006555 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
0.25 |
ug.mL-1 |
10.1021/np800572r |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
0.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.12.037 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
0.5 |
ug.mL-1 |
10.1021/np049706n |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.bmc.2010.10.060 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
1.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.02.062 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
6.3 |
ug.mL-1 |
10.1021/jm070638m |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
12.5 |
ug.mL-1 |
10.1007/s00044-012-0451-x |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.bmcl.2009.12.045 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.072 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.03.039 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.033 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.049 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2011.08.014 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2012.01.008 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2013.11.002 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
128.0 |
ug.mL-1 |
10.1016/j.ejmech.2019.111882 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
22820.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
29200.0 |
nM |
10.1021/np2003319 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
nan |
None |
10.1016/j.bmc.2010.05.016 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
nan |
None |
10.1016/j.bmc.2013.10.011 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
nan |
None |
10.1016/j.bmc.2022.116777 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
nan |
None |
10.1016/j.ejmech.2018.08.070 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC |
nan |
None |
10.1016/j.ejmech.2020.112996 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC50 |
0.322 |
ug.mL-1 |
10.1016/j.bmc.2013.06.027 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC50 |
100000.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycolicibacterium fortuitum |
Mycolicibacterium fortuitum |
MIC90 |
250.0 |
ug.mL-1 |
10.1016/j.bmc.2013.06.027 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmc.2010.10.060 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
4.0 |
ug.mL-1 |
10.1021/np049706n |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
16.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.02.062 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
128.0 |
ug.mL-1 |
10.1021/np800572r |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
14600.0 |
nM |
10.1021/np2003319 |
| Mycolicibacterium phlei |
Mycolicibacterium phlei |
MIC |
91150.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Activity |
1.2 |
None |
10.1016/j.ejmech.2016.07.068 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Activity |
36.0 |
% |
10.1016/j.ejmech.2006.09.009 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Activity |
nan |
None |
10.1016/j.ejmech.2016.07.068 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Activity |
nan |
None |
10.1128/aac.00453-10 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
GI |
nan |
None |
10.1016/j.ejmech.2012.02.031 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
GI |
nan |
None |
10.1016/j.ejmech.2012.12.012 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
GI50 |
7.94 |
ug.mL-1 |
10.1016/j.ejmech.2014.02.042 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
GI50 |
41630.0 |
nM |
10.1016/j.ejmech.2014.06.075 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
IC50 |
7800.0 |
nM |
10.1016/j.ejmech.2010.07.016 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
IC50 |
9800.0 |
nM |
10.1016/j.ejmech.2015.02.062 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
IC50 |
16000.0 |
nM |
10.1016/j.bmcl.2015.02.052 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
IC50 |
39000.0 |
nM |
10.1016/j.ejmech.2010.07.016 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
IZ |
17.0 |
mm |
10.1016/j.bmcl.2008.07.087 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
IZ |
23.0 |
mm |
10.1016/j.bmc.2008.03.062 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
IZ |
29.0 |
mm |
10.1016/j.ejmech.2012.02.031 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MBC |
nan |
None |
10.1021/np800778b |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
0.05 |
ug.mL-1 |
10.1021/jm00202a020 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.ejmech.2014.08.066 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
0.25 |
ug.mL-1 |
10.1021/np800572r |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
0.8 |
ug.mL-1 |
10.1021/np0102509 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
0.8 |
ug.mL-1 |
10.1021/np020198w |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.0 |
ug.mL-1 |
10.1021/np049706n |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.0 |
ug.mL-1 |
10.1021/np2006555 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
1.5 |
ug.mL-1 |
10.1016/j.ejmech.2006.09.009 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
2.0 |
ug.mL-1 |
10.1016/j.bmc.2008.03.062 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
2.5 |
ug.mL-1 |
10.1016/j.bmc.2008.05.061 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
2.5 |
ug.mL-1 |
10.1016/j.bmc.2015.04.033 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
2.5 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.100 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
2.5 |
ug.mL-1 |
10.1039/C3MD00016H |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
3.13 |
ug.mL-1 |
10.1016/j.bmcl.2022.128650 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmc.2012.02.039 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2008.07.087 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.02.044 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2018.05.049 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.02.062 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2016.12.042 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2017.11.025 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.ejmech.2020.112837 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
4.7 |
ug.mL-1 |
10.1128/aac.00453-10 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
6.1 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
6.25 |
ug.mL-1 |
10.1016/j.ejmech.2016.09.083 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
7.8 |
ug.mL-1 |
10.1039/C8MD00056E |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
8.0 |
ug.mL-1 |
10.1021/np3006277 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
10.0 |
ug.mL-1 |
10.1016/j.ejmech.2015.06.007 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
12.07 |
ug.mL-1 |
10.1016/j.bmcl.2015.05.044 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
12.5 |
ug.mL-1 |
10.1007/s00044-012-0458-3 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2010.07.020 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2018.01.080 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.ejmech.2021.113266 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
12.5 |
ug.mL-1 |
10.1021/jm070638m |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
15.62 |
ug.mL-1 |
10.1016/j.ejmech.2019.111578 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.bmc.2008.05.061 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.bmc.2015.04.033 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
25.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.04.100 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
25.0 |
ug.mL-1 |
10.1039/C3MD00016H |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
25.0 |
ug.mL-1 |
10.1039/C7MD00350A |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
32.0 |
ug.mL-1 |
10.1021/acs.jmedchem.2c00972 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
45.57 |
ug.mL-1 |
10.1021/jm800545k |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
50.0 |
ug.mL-1 |
10.1007/s00044-012-0451-x |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.12.045 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.bmcl.2013.06.072 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.03.039 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.033 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.07.049 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.ejmech.2011.08.014 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.ejmech.2012.01.008 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
50.0 |
ug.mL-1 |
10.1016/j.ejmech.2013.11.002 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
64.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00248-0 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
64.0 |
ug.mL-1 |
10.1016/s0960-894x(98)00526-5 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
64.0 |
ug.mL-1 |
10.1016/s0960-894x(99)00510-7 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm0602662 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
64.0 |
ug.mL-1 |
10.1021/jm701560p |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
300.0 |
ug.mL-1 |
10.1128/aac.00453-10 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
2000.0 |
nM |
10.1016/j.ejmech.2021.113212 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
3900.0 |
nM |
10.1039/D1MD00239B |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
5690.0 |
nM |
10.1016/j.ejmech.2010.11.023 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
10000.0 |
nM |
10.1016/j.ejmech.2012.02.031 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
14600.0 |
nM |
10.1021/np2003319 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
18900.0 |
nM |
10.1016/j.bmcl.2013.11.024 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
25000.0 |
ug.mL-1 |
10.1039/C7MD00366H |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
29000.0 |
nM |
10.1016/j.ejmech.2021.113212 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
29200.0 |
nM |
10.1016/j.bmc.2018.04.045 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
45570.0 |
nM |
10.1016/j.bmc.2007.11.016 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
45570.0 |
nM |
10.1016/j.bmc.2007.11.050 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
45570.0 |
nM |
10.1016/j.bmcl.2007.09.095 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
45570.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
45570.0 |
nM |
10.1016/j.bmcl.2011.07.062 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
45570.0 |
nM |
10.1016/j.ejmech.2008.02.031 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
45570.0 |
nM |
10.1016/j.ejmech.2009.05.010 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
45570.0 |
nM |
10.1016/j.ejmech.2009.09.001 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
45570.0 |
nM |
10.1021/jm700999n |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
117000.0 |
nM |
10.1016/j.bmc.2013.08.029 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
117000.0 |
nM |
10.1016/j.bmc.2013.08.030 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
364670.0 |
nM |
10.1016/j.bmcl.2011.07.062 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
729100.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
nan |
ug.mL-1 |
10.1016/s0960-894x(03)00597-3 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
nan |
None |
10.1021/np800572r |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
nan |
None |
10.1021/np800778b |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC |
nan |
None |
10.1128/aac.00453-10 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC50 |
1.2 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC50 |
1.3 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC50 |
1.4 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC50 |
12.07 |
ug.mL-1 |
10.1016/j.ejmech.2013.10.034 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC50 |
1800.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC>90 |
4.0 |
ug ml-1 |
10.1016/j.ejmech.2015.07.050 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC>90 |
12.7 |
ug ml-1 |
10.1021/np400145u |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
2.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c01349 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
2.5 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
2.7 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
3.1 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
11.78 |
ug.mL-1 |
10.1016/j.ejmech.2013.10.034 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
100.0 |
nM |
10.1016/j.ejmech.2017.06.061 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
6700.0 |
nM |
10.1016/j.bmcl.2004.01.010 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
10000.0 |
nM |
10.1016/j.ejmech.2017.05.026 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC90 |
15000.0 |
nM |
10.1016/j.ejmech.2016.07.068 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC95 |
12.0 |
ug ml-1 |
10.1016/j.bmc.2006.12.009 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC95 |
12.0 |
ug ml-1 |
10.1016/j.bmc.2008.06.057 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC99 |
4.0 |
ug ml-1 |
10.1016/j.bmcl.2014.02.025 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC99 |
45.57 |
uM |
10.1016/j.bmcl.2007.11.110 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
MIC99 |
50.0 |
uM |
10.1039/C4MD00303A |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Ratio |
2.0 |
None |
10.1128/aac.00453-10 |
| Mycolicibacterium smegmatis |
Mycolicibacterium smegmatis |
Selectivity Index |
1.0 |
None |
10.1021/acs.jmedchem.1c01349 |
| Mycolicibacterium vaccae |
Mycolicibacterium vaccae |
MIC |
182300.0 |
nM |
10.1016/j.bmcl.2008.12.088 |
| Mycolicibacter terrae |
Mycolicibacter terrae |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2014.05.006 |
| Mycolicibacter terrae |
Mycolicibacter terrae |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2016.03.107 |
| Mycolicibacter terrae |
Mycolicibacter terrae |
MIC |
0.1 |
ug.mL-1 |
10.1016/j.bmcl.2016.04.017 |
| Mycolicibacter terrae |
Mycolicibacter terrae |
MIC |
730.0 |
nM |
10.1016/j.bmc.2016.06.020 |
| Mycolicibacter terrae |
Mycolicibacter terrae |
MIC |
730.0 |
nM |
10.1016/j.ejmech.2015.05.007 |
| Oryctolagus cuniculus |
Angiotensin-converting enzyme |
IC50 |
nan |
None |
None |
| Oryctolagus cuniculus |
Angiotensin-converting enzyme |
Ki |
nan |
None |
None |
| Oryctolagus cuniculus |
Arachidonate 15-lipoxygenase |
IC50 |
nan |
None |
None |
| Oryctolagus cuniculus |
Arachidonate 15-lipoxygenase |
Ki |
nan |
None |
None |
| Papio hamadryas |
Plasma |
PPB |
94.63 |
% |
10.1021/jm901858n |
| Photinus pyralis |
Luciferin 4-monooxygenase |
Potency |
5011.9 |
nM |
None |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
36460.0 |
nM |
10.6019/CHEMBL3392926 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
246460.0 |
nM |
10.6019/CHEMBL3392926 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
1200000.0 |
nM |
10.1074/jbc.m701813200 |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
1800000.0 |
nM |
10.1074/jbc.m701813200 |
| Plasmodium falciparum |
Plasmodium falciparum |
MIC |
0.1 |
ug.mL-1 |
10.1021/np0602012 |
| Proteus mirabilis |
Proteus mirabilis |
GI |
nan |
None |
10.1016/j.bmc.2013.06.013 |
| Proteus mirabilis |
Proteus mirabilis |
MIC |
200.0 |
ug.mL-1 |
10.1007/s00044-013-0488-5 |
| Proteus vulgaris |
Proteus vulgaris |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
GI |
nan |
None |
10.1016/j.bmc.2013.06.013 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
IC50 |
nan |
None |
10.1016/j.ejmech.2019.07.052 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Inhibition |
1.16 |
% |
10.6019/CHEMBL4513141 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
Inhibition |
12.59 |
% |
10.6019/CHEMBL4513156 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
2850.0 |
nM |
10.1016/j.bmc.2019.02.043 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
20000.0 |
nM |
10.6019/CHEMBL4513161 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1016/j.ejmech.2019.01.062 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC |
nan |
None |
10.1016/j.ejmech.2019.04.067 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
nan |
None |
10.1016/j.ejmech.2017.12.089 |
| Pseudomonas aeruginosa |
Pseudomonas aeruginosa |
MIC90 |
nan |
None |
10.1021/acs.jmedchem.7b00793 |
| Rattus norvegicus |
Aldose reductase |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Aldose reductase |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1a adrenergic receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1a adrenergic receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1b adrenergic receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1b adrenergic receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Androgen Receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Androgen Receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Androgen Receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Bile salt export pump |
IC50 |
1000000.0 |
nM |
10.1124/dmd.111.040758 |
| Rattus norvegicus |
Cyclooxygenase-1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
GABA-A receptor; anion channel |
Inhibition |
nan |
% |
10.1021/jm50001a020 |
| Rattus norvegicus |
GABA receptor alpha-1 subunit |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Gamma-amino-N-butyrate transaminase |
Inhibition |
nan |
% |
10.1021/jm50001a020 |
| Rattus norvegicus |
Glutamate decarboxylase 67 kDa isoform |
Inhibition |
42.0 |
% |
10.1021/jm50001a020 |
| Rattus norvegicus |
Glutamate (NMDA) receptor subunit zeta 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Glycine receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Glycine receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Insulin receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Insulin receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Liver |
Activity |
9.1 |
nmol |
10.1016/j.bmcl.2010.06.125 |
| Rattus norvegicus |
Liver |
Activity |
nan |
None |
10.1016/j.bmcl.2017.01.024 |
| Rattus norvegicus |
Liver microsomes |
Stability |
nan |
% |
10.1016/j.bmcl.2007.09.048 |
| Rattus norvegicus |
Multidrug resistance protein 1a |
Activity |
nan |
None |
10.1124/dmd.30.7.838 |
| Rattus norvegicus |
Nitric-oxide synthase, brain |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Nitric-oxide synthase, brain |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Plasma |
logFu |
1.0 |
None |
10.1016/j.ejmech.2009.06.004 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
1.48 |
g/dl |
10.1016/j.bmcl.2010.06.125 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
1.55 |
g/dl |
10.1016/j.bmcl.2010.06.125 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
8.31 |
U/ml |
10.1016/j.bmcl.2010.06.125 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
40.21 |
U/ml |
10.1016/j.bmcl.2010.06.125 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
151.25 |
U/ml |
10.1016/j.bmcl.2010.06.125 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
33000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
34000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
35000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
36000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
37000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
38000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
41700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
42300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
43200.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
43300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
43700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
49000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.4 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.5 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.6 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.7 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.8 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.9 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
331.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
339.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
349.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
359.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
369.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
384.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
533.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
560.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
587.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
589.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
683.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
722.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
722.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
735.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
751.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
752.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
757.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
760.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
761.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
774.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
780.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
783.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
793.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
797.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
817.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
823.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
823.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
836.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
838.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
862.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
884.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
918.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
930.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
945.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
950.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
962.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
976.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1043.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
6.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
8.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
8.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
10.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
11.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
11.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
12.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
14.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
15.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
15.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
18.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
19.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
19.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
20.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
23.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
23.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
23.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
26.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
27.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
27.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
28.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
28.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
29.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
30.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
33.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
33.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
39.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
47.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
50.5 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
52.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
14.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
14.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
15.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
16.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
17.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
17.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
18.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
18.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
18.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
18.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
18.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
25.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
32.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
40.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
43.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
44.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
44.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
46.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
48.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
49.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
52.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
53.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
55.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
55.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
56.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
56.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
57.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
58.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
58.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
60.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
61.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
62.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
64.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
66.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
66.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
68.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
70.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
73.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
74.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
83.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
85.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
88.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
92.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
95.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AUC |
197090.0 |
ng.hr.mL-1 |
10.1016/j.bmcl.2012.02.091 |
| Rattus norvegicus |
Rattus norvegicus |
AUC |
684000.0 |
ng.hr.mL-1 |
10.1016/j.bmcl.2012.02.091 |
| Rattus norvegicus |
Rattus norvegicus |
BASO |
0.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.02 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.04 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.06 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.08 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.14 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.24 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.28 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.4 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.42 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.52 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.525 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.58 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.6 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.62 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.64 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.66 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.68 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.74 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.8 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
1.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
1.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
1.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
3.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
4.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
78.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
82.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
88.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
90.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
94.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
96.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
100.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
140.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
143.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
148.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
153.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
156.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
160.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
162.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
166.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
166.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
170.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
172.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
178.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
184.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
190.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
192.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
194.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
195.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
196.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
202.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
204.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
226.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
99.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
100.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
101.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
102.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
103.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
104.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
105.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
106.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
107.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
108.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
109.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
101.67 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
102.33 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
102.67 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
103.17 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
103.83 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
470.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
538.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
586.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
602.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
636.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
644.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
664.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
686.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
688.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
700.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
704.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
706.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
710.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
713.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
714.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
728.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
732.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
736.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
748.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
760.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
760.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
762.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
764.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
782.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
784.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
786.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
792.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
800.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
800.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
802.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
808.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
814.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
816.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
858.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
936.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
235.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
246.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
281.83 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
463.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
472.83 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
505.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
102.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
105.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
106.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
106.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CL |
0.21 |
mL.min-1.kg-1 |
10.1016/j.bmcl.2012.02.091 |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
98439.55 |
nM |
10.1021/acs.jmedchem.5b00391 |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
381580.87 |
nM |
10.1016/j.bmcl.2012.02.091 |
| Rattus norvegicus |
Rattus norvegicus |
Cmax |
2174420.3 |
nM |
10.1016/j.bmcl.2012.02.091 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
23670000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
24670000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
25000000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
25670000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
26000000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
26170000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.1 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.6 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.8 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.9 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
4.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
4.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
5.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
6.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
0.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
23.5 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
46.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
46.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
53.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.17 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
2.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
F |
17.36 |
% |
10.1016/j.bmcl.2012.02.091 |
| Rattus norvegicus |
Rattus norvegicus |
F |
65.0 |
% |
10.1021/acs.jmedchem.5b00391 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
1960.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2128.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2178.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2182.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2186.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2214.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2218.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2228.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2234.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2242.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2250.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2262.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2274.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2278.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2282.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2286.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2292.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2294.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2300.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2304.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2310.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2322.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2348.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2350.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2364.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2398.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2422.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2452.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
0.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
0.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
0.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.5 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1550.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1616.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1730.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1785.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1883.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1892.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1910.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1952.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1956.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1976.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2004.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2006.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2030.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2042.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2054.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2086.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2088.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2092.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2096.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2100.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2108.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2110.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2122.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2125.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2132.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2154.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2172.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2218.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2224.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2226.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2238.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2252.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2272.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2273.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
33.43 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
33.8 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
34.97 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.03 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.72 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
41.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
42.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
44.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
44.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
46.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
125500.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
128000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
130000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
131700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
133000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
134000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
134000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
135000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
136000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
137000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
137200.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
138000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
139000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
140000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
140300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
144000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
145000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
147000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
151000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
155000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
12.0 |
% |
10.1021/jm00399a021 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
14.0 |
% |
10.1021/jm00399a021 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
16.0 |
% |
10.1021/jm00399a021 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
19.0 |
% |
10.1021/jm00399a021 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
22.0 |
% |
10.1021/jm00399a021 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
51.62 |
% |
10.1016/j.bmcl.2010.06.125 |
| Rattus norvegicus |
Rattus norvegicus |
Kel |
0.24 |
/hr |
10.1016/j.bmcl.2012.02.091 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
73.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
75.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
77.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
81.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
87.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
92.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
92.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
93.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
93.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
95.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
101.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
102.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
108.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
113.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
115.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
123.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
140.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
156.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
160.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
175.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
177.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
177.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
185.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
190.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
191.17 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
195.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
197.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
202.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
202.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
203.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
203.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
211.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
221.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
231.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
237.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
244.83 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
268.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
9.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
10.17 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
10.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
10.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
11.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
12.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
10225.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
10642.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
12797.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
12954.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
13139.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
13245.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
68.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
70.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
70.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
72.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
73.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
73.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
74.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
74.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
75.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
75.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
76.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
76.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
76.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
79.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
79.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
80.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
80.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
80.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
82.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
83.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
84.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
85.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
85.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
86.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
86.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
86.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
86.5 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
87.5 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
91.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
16.6 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
18.6 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
18.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
19.1 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
19.7 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.1 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.3 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.2 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.4 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.5 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.7 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.8 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.1 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.2 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.4 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.6 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.8 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
23.27 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
23.4 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
23.67 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
23.8 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.35 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
33.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
363000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
371700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
373500.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
375700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
376700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
379000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
50.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
55.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
56.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
57.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
58.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
58.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
59.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
59.8 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.8 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.33 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.73 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.47 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.72 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.47 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.8 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
65.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
65.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
319.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
465.5 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
507.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
520.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
527.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
0.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
1.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
1.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.17 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
4.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
5.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
5.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
5.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
6.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
6.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
7.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
8.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
10.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
11.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
4.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
7.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
8.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
9.17 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
9.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
10.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
10.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
10.5 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
10.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
11.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
11.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
11.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
12.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
12.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
13.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
13.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
17.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
19.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
19.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
19.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
19.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
20.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
22.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
22.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
23.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
26.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
28.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
647.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
779.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1242.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1313.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1492.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1614.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
67.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
69.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
72.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
73.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
76.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
77.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
78.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
79.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
80.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
81.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
82.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
83.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
84.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
85.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
86.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
88.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
89.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
90.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
92.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
93.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
95.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
97.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
98.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
100.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
101.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
102.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
114.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
117.2 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
120.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
124.5 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
127.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
141.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1082.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1142.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1232.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1278.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1338.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1348.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1360.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1370.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1376.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1386.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1390.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1404.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1406.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1408.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1418.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1422.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1454.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1470.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1482.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1502.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1510.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1512.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1518.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1528.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1540.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1586.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1630.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1634.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1022000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1026170.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1063000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1065670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1130000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1146000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1154000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1157330.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1160000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1172000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1186000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1190000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1192000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1207000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1209000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1214000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1219000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1239670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1253000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1254000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1257000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1260000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1268000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1270670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1274000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1276000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1288000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1301000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1312000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1333000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1340000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1342000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1380000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1389670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1395000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1408000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1528000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
3.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
3.7 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
3.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
3.9 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.1 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.3 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.5 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.9 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.1 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
5.97 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.35 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.52 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.62 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.76 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
7.15 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PPB |
nan |
% |
10.1016/j.bmcl.2007.09.048 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
54000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
55000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
56000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
57000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
57700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
58000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
58300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
59000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
60000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
61000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
61500.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
62000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
63000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
67700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
14.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5170000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5420000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5660000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5760000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5870000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6000000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6100000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6166000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6174000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6184000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6190000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6218000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6224000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6228000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6254000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6262000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6266000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6272000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6298000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6338000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6418000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6440000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6464000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6492000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6564000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6616000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6782000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6974000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7066000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7074000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7408000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7712000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7800000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7818000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7906000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
0.0 |
/100WBC |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
0.17 |
/100WBC |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
0.33 |
/100WBC |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
3.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
3.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
3.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
3.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
8.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
138.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
138.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
143.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
143.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
143.8 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
144.23 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
144.27 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
145.17 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
146.0 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
146.23 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
0.3167 |
hr |
10.1021/acs.jmedchem.5b00391 |
| Rattus norvegicus |
Rattus norvegicus |
T1/2 |
2.88 |
hr |
10.1016/j.bmcl.2012.02.091 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
211.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
212.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
215.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
217.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
217.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
217.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
218.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
219.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
219.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
219.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
219.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
220.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
220.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
221.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
221.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
221.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
222.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
225.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
228.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
229.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
234.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
244.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
247.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
251.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
255.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
283.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
294.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
307.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
314.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
361.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
372.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
374.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Tissue Severity Score |
nan |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Tissue Severity Score |
nan |
None |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
Tmax |
2.0 |
hr |
10.1016/j.bmcl.2012.02.091 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
418.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
478.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
496.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
528.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
546.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
578.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
588.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
618.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
622.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
630.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
696.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
712.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
746.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
772.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
780.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
900.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
904.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
906.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
916.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
948.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
980.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1004.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1016.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1046.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1054.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1102.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1140.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1192.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1256.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1302.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1312.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1440.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
UI |
3.75 |
None |
10.1016/j.bmcl.2010.06.125 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
14.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
20.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
20.8 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
21.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
39.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
Vd |
0.026 |
l |
10.1016/j.bmcl.2012.02.091 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
4140.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
5130.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
6070.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
6130.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
6730.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7150.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7570.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8090.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8210.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8250.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8530.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8590.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8700.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8720.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8920.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9630.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9690.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10160.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10180.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10600.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10810.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10980.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11530.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11830.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11840.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
12640.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
13080.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
13700.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
14080.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
14370.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
14600.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
14940.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
14970.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
15010.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
15160.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
15370.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
17260.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
18120.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
0.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
13.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
15.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
15.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
15.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Serotonin 1a (5-HT1a) receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1a (5-HT1a) receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1b (5-HT1b) receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1b (5-HT1b) receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Voltage-gated L-type calcium channel alpha-1C subunit |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Voltage-gated N-type calcium channel alpha-1B subunit |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Salmonella enterica subsp. enterica serovar Typhi |
Salmonella typhi |
DIZ |
nan |
None |
10.1016/j.ejmech.2011.11.014 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
Activity |
nan |
None |
10.1016/j.ejmech.2017.06.061 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
Activity |
nan |
None |
10.1016/j.ejmech.2018.01.071 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
FC |
1.1 |
None |
10.1016/j.ejmech.2018.01.071 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
FC |
1.2 |
None |
10.1016/j.ejmech.2018.01.071 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
FC |
1.3 |
None |
10.1016/j.ejmech.2018.01.071 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
FC |
1.4 |
None |
10.1016/j.ejmech.2018.01.071 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
FC |
1.5 |
None |
10.1016/j.ejmech.2018.01.071 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
FC |
1.6 |
None |
10.1016/j.ejmech.2018.01.071 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
FC |
1.9 |
None |
10.1016/j.ejmech.2018.01.071 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
FC |
2.0 |
None |
10.1016/j.ejmech.2018.01.071 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
FC |
3.7 |
None |
10.1016/j.ejmech.2018.01.071 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
FC |
4.0 |
None |
10.1016/j.ejmech.2018.01.071 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Salmonella enterica subsp. enterica serovar Typhimurium |
Salmonella typhimurium |
MIC90 |
nan |
None |
10.1016/j.ejmech.2017.12.089 |
| Severe acute respiratory syndrome coronavirus 2 |
Replicase polyprotein 1ab |
Inhibition |
12.72 |
% |
10.6019/CHEMBL4495564 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
19952.62 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
20000.0 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
0.12 |
% |
10.6019/CHEMBL4495565 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
22.5 |
% |
10.21203/rs.3.rs-23951/v1 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition index |
0.2337 |
None |
10.1101/2020.04.03.023846 |
| Shigella sp. |
Shigella sp. |
MIC |
300.0 |
ug.mL-1 |
10.1007/s00044-013-0488-5 |
| Staphylococcus aureus |
Staphylococcus aureus |
DIZ |
nan |
None |
10.1016/j.ejmech.2011.11.014 |
| Staphylococcus aureus |
Staphylococcus aureus |
GI |
nan |
None |
10.1016/j.bmc.2013.06.013 |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
nan |
None |
10.1016/j.ejmech.2019.07.052 |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
nan |
None |
10.1021/np2006555 |
| Staphylococcus aureus |
Staphylococcus aureus |
IC50 |
nan |
None |
10.1021/np900281r |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
8.75 |
% |
10.6019/CHEMBL4513141 |
| Staphylococcus aureus |
Staphylococcus aureus |
Inhibition |
27.38 |
% |
10.6019/CHEMBL4513156 |
| Staphylococcus aureus |
Staphylococcus aureus |
-logMIC |
2.04 |
None |
10.1007/s00044-011-9662-9 |
| Staphylococcus aureus |
Staphylococcus aureus |
-logMIC |
2.04 |
None |
10.1007/s00044-011-9705-2 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.07.043 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.02.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1260.0 |
nM |
10.1016/j.bmc.2019.02.043 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
1420.0 |
nM |
10.1016/j.bmc.2019.02.043 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
20000.0 |
nM |
10.6019/CHEMBL4513161 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
100000.0 |
ug.mL-1 |
10.1016/j.bmcl.2007.02.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmcl.2012.08.003 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmcl.2013.11.024 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.bmcl.2014.05.018 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.ejmech.2019.01.062 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1016/j.ejmech.2019.04.067 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1021/np800572r |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC |
nan |
None |
10.1021/np900281r |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
nan |
None |
10.1016/j.ejmech.2017.12.089 |
| Staphylococcus aureus |
Staphylococcus aureus |
MIC90 |
nan |
None |
10.1021/acs.jmedchem.7b00793 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
4.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.07.043 |
| Staphylococcus epidermidis |
Staphylococcus epidermidis |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Staphylococcus hominis |
Staphylococcus hominis |
GI |
nan |
None |
10.1016/j.bmc.2013.06.013 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
IC50 |
nan |
None |
10.1016/j.ejmech.2019.07.052 |
| Streptococcus pneumoniae |
Streptococcus pneumoniae |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Streptococcus pyogenes |
Streptococcus pyogenes |
MIC |
100.0 |
ug.mL-1 |
10.1021/jm0703901 |
| Trypanosoma brucei rhodesiense |
Trypanosoma brucei rhodesiense |
IC50 |
656260.0 |
nM |
10.6019/CHEMBL3392926 |
| Trypanosoma brucei rhodesiense |
Trypanosoma brucei rhodesiense |
IC50 |
729180.0 |
nM |
10.6019/CHEMBL3392926 |
| Trypanosoma cruzi |
Trypanosoma cruzi |
IC50 |
150000.0 |
nM |
10.1016/j.ejmech.2012.10.047 |
| Trypanosoma cruzi |
Trypanosoma cruzi |
IC50 |
382820.0 |
nM |
10.6019/CHEMBL3392926 |
| Trypanosoma cruzi |
Trypanosoma cruzi |
IC50 |
656260.0 |
nM |
10.6019/CHEMBL3392926 |
| Yersinia pseudotuberculosis |
Yersinia pseudotuberculosis |
MIC99 |
nan |
None |
10.1021/jm061068d |
| None |
ADMET |
Activity |
20.9 |
g |
10.1016/j.ejmech.2020.112075 |
| None |
ADMET |
Activity |
20.9 |
g |
10.1016/j.ejmech.2022.114145 |
| None |
ADMET |
Activity |
21.3 |
g |
10.1021/acs.jmedchem.0c00500 |
| None |
ADMET |
Activity |
23.1 |
% |
10.1016/j.bmcl.2010.01.031 |
| None |
ADMET |
Activity |
24.66 |
g |
10.1016/j.ejmech.2021.113603 |
| None |
ADMET |
Activity |
31.7 |
% |
10.1016/j.bmcl.2010.01.031 |
| None |
ADMET |
Activity |
95.5 |
% |
10.1016/j.bmcl.2010.01.031 |
| None |
ADMET |
Activity |
98.5 |
% |
10.1016/j.bmcl.2010.01.031 |
| None |
ADMET |
Activity |
99.3 |
% |
10.1016/j.bmcl.2010.01.031 |
| None |
ADMET |
Activity |
nan |
None |
10.1016/j.ejmech.2010.04.017 |
| None |
ADMET |
Activity |
nan |
None |
10.1016/j.ejmech.2011.06.037 |
| None |
ADMET |
CC50 |
199.0 |
ug.mL-1 |
10.1007/s00044-012-0043-9 |
| None |
ADMET |
CC50 |
1470000.0 |
nM |
10.1016/j.bmcl.2013.09.027 |
| None |
ADMET |
CC50 |
5833500.0 |
nM |
10.1016/j.bmcl.2010.01.031 |
| None |
ADMET |
CC50 |
nan |
None |
10.1016/j.ejmech.2015.07.039 |
| None |
ADMET |
CC50 |
nan |
None |
10.1039/C5MD00178A |
| None |
ADMET |
CL |
7.4 |
mL.min-1.kg-1 |
10.1124/dmd.108.020479 |
| None |
ADMET |
CLH |
nan |
None |
10.1021/acsmedchemlett.7b00299 |
| None |
ADMET |
Cmax |
0.29 |
ug |
10.1128/aac.00153-08 |
| None |
ADMET |
Cmax |
0.56 |
ug |
10.1128/aac.00153-08 |
| None |
ADMET |
delta logD |
0.0 |
None |
10.1021/jm0000564 |
| None |
ADMET |
Drugexcretion |
3.6 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
9.25 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
9.44 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
10.07 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
10.4 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
10.6 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
10.68 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
11.2 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
11.32 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
11.4 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
11.6 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
12.2 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
12.5 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
12.7 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
12.7 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
12.82 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
13.0 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
13.1 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
13.18 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
13.38 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
13.5 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
14.26 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
16.5 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
16.8 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
17.0 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
17.1 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
17.18 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
17.2 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
17.3 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
17.9 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
18.5 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
20.0 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
20.23 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
21.24 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
26.6 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
26.76 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
27.1 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
27.3 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
27.92 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
28.0 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
28.41 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
28.7 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
29.0 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
29.6 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
30.44 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
32.0 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
32.27 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
32.59 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
33.2 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
33.6 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
33.69 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
33.7 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
34.76 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
36.2 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
37.21 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
37.75 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
38.1 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
38.5 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
38.71 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
38.8 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
39.4 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
39.7 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
39.9 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
40.5 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
42.1 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
42.3 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
43.3 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
43.4 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
44.45 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
45.9 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
48.1 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
49.9 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
50.1 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
51.7 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
51.8 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
57.7 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
59.9 |
mg |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
95.4 |
% |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
95.6 |
% |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
96.9 |
% |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
97.0 |
% |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
97.9 |
% |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
98.0 |
% |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
98.8 |
% |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
99.6 |
% |
10.1002/jps.2600630804 |
| None |
ADMET |
Drugexcretion |
101.0 |
% |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug metabolism |
1.4 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug metabolism |
2.9 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug metabolism |
6.9 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug metabolism |
13.9 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug metabolism |
14.2 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug metabolism |
18.1 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug metabolism |
21.3 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug metabolism |
27.1 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug metabolism |
32.3 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug metabolism |
34.3 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug metabolism |
43.8 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug metabolism |
48.4 |
%molar |
10.1002/jps.2600630804 |
| None |
ADMET |
Drug uptake |
0.02 |
ug/g |
10.1021/jm901858n |
| None |
ADMET |
Drug uptake |
0.31 |
ug ml-1 |
10.1021/jm901858n |
| None |
ADMET |
Drug uptake |
1.9 |
ug ml-1 |
10.1021/jm901858n |
| None |
ADMET |
Drug uptake |
nan |
None |
10.1021/acs.jmedchem.6b00415 |
| None |
ADMET |
F |
80.0 |
% |
10.1021/jm0000564 |
| None |
ADMET |
GI50 |
nan |
None |
10.1021/acs.jmedchem.6b00031 |
| None |
ADMET |
HC50 |
nan |
None |
10.1039/C4MD00303A |
| None |
ADMET |
I50 |
nan |
None |
10.1016/j.ejmech.2014.02.065 |
| None |
ADMET |
I50 |
nan |
None |
10.1016/j.ejmech.2014.03.024 |
| None |
ADMET |
IC50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2015.12.049 |
| None |
ADMET |
IC50 |
100000.0 |
nM |
10.1016/j.ejmech.2013.01.017 |
| None |
ADMET |
IC50 |
100000.0 |
nM |
10.1021/jm401735w |
| None |
ADMET |
IC50 |
400000.0 |
nM |
10.1016/j.ejmech.2012.10.047 |
| None |
ADMET |
IC50 |
nan |
None |
10.1016/j.bmcl.2016.04.017 |
| None |
ADMET |
IC50 |
nan |
None |
10.1016/j.ejmech.2011.11.033 |
| None |
ADMET |
IC50 |
nan |
None |
10.1016/j.ejmech.2011.12.035 |
| None |
ADMET |
IC50 |
nan |
None |
10.1016/j.ejmech.2013.06.010 |
| None |
ADMET |
IC50 |
nan |
None |
10.1016/j.ejmech.2013.06.042 |
| None |
ADMET |
IC50 |
nan |
None |
10.1016/j.ejmech.2013.10.069 |
| None |
ADMET |
IC50 |
nan |
None |
10.1016/j.ejmech.2013.12.057 |
| None |
ADMET |
Inhibition |
nan |
% |
10.1016/j.bmcl.2016.04.012 |
| None |
ADMET |
MRT |
1.8 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
PPB |
0.0 |
% |
10.1021/acs.jmedchem.0c00046 |
| None |
ADMET |
Selectivity Index |
nan |
None |
10.1016/j.bmc.2022.116777 |
| None |
ADMET |
Selectivity Index |
nan |
None |
10.1016/j.bmcl.2021.128236 |
| None |
ADMET |
Survival |
103.0 |
% |
10.1016/j.ejmech.2015.10.033 |
| None |
ADMET |
Survival |
nan |
None |
10.1016/j.ejmech.2019.06.038 |
| None |
ADMET |
t1/2 |
nan |
None |
10.1021/acsmedchemlett.7b00299 |
| None |
ADMET |
T1/2 |
1.0 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
TI |
nan |
None |
10.1016/j.ejmech.2013.06.010 |
| None |
ADMET |
TI |
nan |
None |
10.1016/j.ejmech.2017.06.061 |
| None |
ADMET |
TI |
nan |
None |
10.1039/C4MD00303A |
| None |
ADMET |
Vdss |
0.82 |
L.kg-1 |
10.1124/dmd.108.020479 |
| None |
BMDM |
CC50 |
20.0 |
ug.mL-1 |
10.1016/j.bmcl.2022.128692 |
| None |
Erythrocyte |
HC10 |
20.0 |
uM |
10.6019/CHEMBL4513161 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Index Value |
12.7 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Active |
5.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Marginal |
0.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Index Value |
8.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1021/tx1000865 |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1021/tx900326k |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1124/dmd.110.035113 |
| None |
Hepatotoxicity |
HepSE_bilirubinemia |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholecystitis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholelithiasis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cirrhosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_Combined Scores |
2.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_elevated liver function tests |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic failure |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic necrosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatitis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatomegaly |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_jaundice |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver disease |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver fatty |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver function tests abnormal |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
LDH Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LDH Increase - Index Value |
10.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LDH Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LTKB_BD DILI severity score |
8.0 |
None |
10.1016/j.drudis.2011.05.007 |
| None |
Hepatotoxicity |
SGOT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Index Value |
38.7 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Index Value |
34.7 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Lipid bilayer |
Activity |
nan |
None |
10.1016/j.ejmech.2016.07.068 |
| None |
NON-PROTEIN TARGET |
Activity |
nan |
None |
10.1016/j.ejmech.2010.03.031 |
| None |
NON-PROTEIN TARGET |
fAUC/MIC |
800.0 |
None |
10.1016/j.bmcl.2013.07.006 |
| None |
NON-PROTEIN TARGET |
fCmax/MIC |
400.0 |
None |
10.1016/j.bmcl.2013.07.006 |
| None |
NON-PROTEIN TARGET |
fT>MIC |
60.0 |
% |
10.1016/j.bmcl.2013.07.006 |
| None |
NON-PROTEIN TARGET |
Fu |
1.0 |
None |
10.1124/dmd.108.020479 |
| None |
NON-PROTEIN TARGET |
GI |
nan |
None |
10.1016/j.ejmech.2011.02.047 |
| None |
NON-PROTEIN TARGET |
GI |
nan |
None |
10.1016/j.ejmech.2016.06.042 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (acute) |
26.7 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (animal toxicity known) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (benign tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (granulomatous hepatitis) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (mechanism) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
51.2 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
60.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (time to onset) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
IC50 |
0.0023 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.056 |
| None |
NON-PROTEIN TARGET |
IC50 |
2600.0 |
nM |
10.1016/j.ejmech.2012.12.012 |
| None |
NON-PROTEIN TARGET |
IC50 |
218750.0 |
nM |
10.6019/CHEMBL3392926 |
| None |
NON-PROTEIN TARGET |
IC50 |
450000.0 |
nM |
10.1016/j.ejmech.2016.05.025 |
| None |
NON-PROTEIN TARGET |
IC50 |
602300.0 |
nM |
10.6019/CHEMBL3392926 |
| None |
NON-PROTEIN TARGET |
IC50 |
656260.0 |
nM |
10.6019/CHEMBL3392926 |
| None |
NON-PROTEIN TARGET |
IC50 |
nan |
None |
10.1016/j.bmcl.2016.11.003 |
| None |
NON-PROTEIN TARGET |
IC50 |
nan |
None |
10.1016/j.ejmech.2016.07.039 |
| None |
NON-PROTEIN TARGET |
IC90 |
0.045 |
ug.mL-1 |
10.1016/j.bmcl.2016.02.056 |
| None |
NON-PROTEIN TARGET |
MIC |
0.04 |
ug.mL-1 |
10.1016/j.bmcl.2009.09.095 |
| None |
NON-PROTEIN TARGET |
MIC |
0.04 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| None |
NON-PROTEIN TARGET |
MIC |
1.56 |
ug.mL-1 |
10.1016/j.bmcl.2010.12.084 |
| None |
NON-PROTEIN TARGET |
MIC |
12.5 |
ug.mL-1 |
10.1016/j.bmc.2014.11.014 |
| None |
NON-PROTEIN TARGET |
MIC |
760.0 |
nM |
10.1021/jm401735w |
| None |
NON-PROTEIN TARGET |
MIC |
45570.0 |
nM |
10.1016/j.bmcl.2010.06.096 |
| None |
NON-PROTEIN TARGET |
MIC |
91140.0 |
nM |
10.1016/j.bmcl.2010.06.096 |
| None |
NON-PROTEIN TARGET |
MIC50 |
100.0 |
nM |
10.1016/j.ejmech.2013.03.023 |
| None |
NON-PROTEIN TARGET |
RatioAUC/MIC |
63.0 |
None |
10.1128/aac.00185-07 |
| None |
NON-PROTEIN TARGET |
RatioAUC/MIC |
1300.0 |
None |
10.1016/j.bmcl.2013.07.006 |
| None |
NON-PROTEIN TARGET |
Selectivity Index |
nan |
None |
10.1021/acs.jmedchem.6b00031 |
| None |
NON-PROTEIN TARGET |
%T>MIC |
80.0 |
% |
10.1016/j.bmcl.2013.07.006 |
| None |
No relevant target |
Activity |
0.0 |
mol/mol |
10.1016/j.ejmech.2016.07.039 |
| None |
No relevant target |
Activity |
91.3 |
% |
10.1016/j.bmc.2020.115470 |
| None |
No relevant target |
CLogP |
0.58 |
None |
10.1016/j.bmcl.2005.07.011 |
| None |
No relevant target |
Drug metabolism |
nan |
None |
10.1016/j.bmcl.2017.07.019 |
| None |
No relevant target |
IC50 |
22900.0 |
nM |
10.1016/j.bmc.2020.115470 |
| None |
No relevant target |
IC50 |
nan |
None |
10.1016/j.bmcl.2015.11.071 |
| None |
No relevant target |
Kinetic_solubility |
nan |
None |
10.1016/j.ejmech.2012.08.047 |
| None |
No relevant target |
Kinetic_solubility |
nan |
None |
10.1021/acs.jmedchem.1c00707 |
| None |
No relevant target |
LogD |
-0.7 |
None |
10.1021/jm0000564 |
| None |
No relevant target |
LogD |
nan |
None |
10.1021/jm901858n |
| None |
No relevant target |
LogD7.4 |
-0.57 |
None |
10.6019/CHEMBL3301361 |
| None |
No relevant target |
log K |
-0.7432 |
None |
10.1016/j.bmcl.2013.12.054 |
| None |
No relevant target |
log K |
-0.743 |
None |
10.1039/C5MD00178A |
| None |
No relevant target |
log K |
nan |
None |
10.1016/j.bmcl.2012.11.052 |
| None |
No relevant target |
log K |
nan |
None |
10.1016/j.bmcl.2013.04.021 |
| None |
No relevant target |
LogP |
-2.322 |
None |
10.1016/j.ejmech.2013.10.029 |
| None |
No relevant target |
LogP |
-1.137 |
None |
10.1021/jm00226a007 |
| None |
No relevant target |
LogP |
-0.851 |
None |
10.1016/j.ejmech.2014.04.077 |
| None |
No relevant target |
LogP |
-0.822 |
None |
10.1016/j.ejmech.2013.10.029 |
| None |
No relevant target |
LogP |
0.64 |
None |
10.1016/j.bmc.2018.07.049 |
| None |
No relevant target |
LogP |
nan |
None |
10.1016/j.ejmech.2016.07.039 |
| None |
No relevant target |
-log(solubility) |
3.23 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
-log(solubility) |
3.54 |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
-log(solubility) |
nan |
None |
10.1016/j.bmcl.2015.02.013 |
| None |
No relevant target |
pKa |
1.8 |
None |
10.1016/j.ejmech.2018.03.042 |
| None |
No relevant target |
pKa |
nan |
None |
10.1021/jm0000564 |
| None |
No relevant target |
Rm |
0.372 |
None |
10.1021/jm00226a007 |
| None |
No relevant target |
solubility |
nan |
None |
10.1039/C8MD00056E |
| None |
No relevant target |
Solubility |
nan |
None |
10.1016/j.bmcl.2007.09.048 |
| None |
No relevant target |
Stability |
nan |
% |
10.1128/aac.00086-07 |
| None |
Nucleic Acid |
Activity |
8.0 |
None |
10.1016/j.ejmech.2011.11.014 |
| None |
Nucleic Acid |
Activity |
50.8 |
% |
10.1016/j.ejmech.2011.11.014 |
| None |
Nucleic Acid |
Activity |
51.0 |
None |
10.1016/j.ejmech.2011.11.014 |
| None |
Nucleic Acid |
Activity |
77.1 |
% |
10.1016/j.ejmech.2011.11.014 |
| None |
Nucleic Acid |
Activity |
nan |
None |
10.1016/j.ejmech.2011.11.014 |
| None |
Nucleic Acid |
Kb |
1.42 |
10'4/M |
10.1016/j.ejmech.2011.11.014 |
| None |
Nucleic Acid |
Kb |
1.6 |
10'4/M |
10.1016/j.ejmech.2011.11.014 |
| None |
Nucleic Acid |
Kb |
2.03 |
10'4/M |
10.1016/j.ejmech.2011.11.014 |
| None |
Phospholipidosis |
Phospholipidosis |
nan |
None |
10.1080/15376510701857262 |
| None |
Radical scavenging activity |
TAC |
90.0 |
% |
10.1016/j.bmc.2013.06.013 |
| None |
Unchecked |
Ac50 |
0.7079 |
uM |
None |
| None |
Unchecked |
Ac50 |
3.162 |
uM |
None |
| None |
Unchecked |
AC50 |
707.9 |
nM |
None |
| None |
Unchecked |
AC50 |
3162.3 |
nM |
None |
| None |
Unchecked |
Activity |
nan |
None |
10.1021/acs.jmedchem.6b00031 |
| None |
Unchecked |
Average IC90 |
0.294 |
uM |
None |
| None |
Unchecked |
Average IC90 |
0.32 |
uM |
None |
| None |
Unchecked |
Average IC90 |
0.46 |
uM |
None |
| None |
Unchecked |
Average IC90 |
37.61 |
uM |
None |
| None |
Unchecked |
CC50 |
100.0 |
ug.mL-1 |
10.1016/j.bmcl.2017.07.008 |
| None |
Unchecked |
GI |
nan |
None |
10.1016/j.ejmech.2012.12.012 |
| None |
Unchecked |
Hepatotoxicity (acute) |
91.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (association with vascular disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (choleostasis) |
11.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (chronic liver disease) |
3.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cirrhosis) |
4.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (comment) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cytolytic) |
61.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (malignant tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (severe hepatitis) |
40.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (steatosis) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (successful reintroduction) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
IC50 |
71.68 |
ug.mL-1 |
10.1016/j.ejmech.2020.112835 |
| None |
Unchecked |
IC50 |
3900.0 |
nM |
10.1016/j.bmc.2020.115470 |
| None |
Unchecked |
IC50 |
5000.0 |
nM |
10.1021/jm00399a021 |
| None |
Unchecked |
IC50 |
10000.0 |
nM |
10.1021/jm00399a021 |
| None |
Unchecked |
IC50 |
25000.0 |
nM |
10.1016/j.bmc.2016.09.012 |
| None |
Unchecked |
IC50 |
25000.0 |
nM |
10.1016/j.bmc.2017.11.031 |
| None |
Unchecked |
IC50 |
25000.0 |
nM |
10.1016/j.ejmech.2017.12.088 |
| None |
Unchecked |
IC50 |
100000.0 |
nM |
10.1021/jm00399a021 |
| None |
Unchecked |
IC50 |
1000000.0 |
nM |
10.1016/j.ejmech.2021.113568 |
| None |
Unchecked |
IC50 |
nan |
None |
10.1016/j.bmc.2014.12.060 |
| None |
Unchecked |
IC50 |
nan |
None |
10.1016/j.bmc.2015.02.032 |
| None |
Unchecked |
IC50 |
nan |
None |
10.1016/j.bmcl.2017.01.026 |
| None |
Unchecked |
IC50 |
nan |
None |
10.1016/j.ejmech.2014.12.046 |
| None |
Unchecked |
IC50 |
nan |
None |
10.1016/j.ejmech.2016.06.042 |
| None |
Unchecked |
IC50 |
nan |
None |
10.1021/acs.jmedchem.7b00793 |
| None |
Unchecked |
IC50 |
nan |
None |
10.1021/ml5001728 |
| None |
Unchecked |
IC50 |
nan |
None |
None |
| None |
Unchecked |
Inhibition |
-39.0 |
% |
10.1016/j.bmcl.2011.06.040 |
| None |
Unchecked |
Inhibition |
0.0 |
% |
10.1016/j.bmc.2014.05.064 |
| None |
Unchecked |
Inhibition |
0.0 |
% |
10.1016/j.bmc.2014.12.060 |
| None |
Unchecked |
Inhibition |
0.0 |
% |
10.1016/j.ejmech.2019.111578 |
| None |
Unchecked |
Inhibition |
78.5 |
% |
10.1016/j.bmc.2014.12.060 |
| None |
Unchecked |
Inhibition |
95.0 |
% |
10.1016/j.bmcl.2009.12.045 |
| None |
Unchecked |
Inhibition |
99.0 |
% |
10.1016/j.bmc.2020.115470 |
| None |
Unchecked |
Inhibition |
99.0 |
% |
10.1016/j.ejmech.2019.111644 |
| None |
Unchecked |
Inhibition |
nan |
% |
10.1016/j.bmc.2012.12.012 |
| None |
Unchecked |
Inhibition |
nan |
% |
10.1016/j.bmc.2015.04.033 |
| None |
Unchecked |
Inhibition |
nan |
% |
10.1016/j.bmc.2017.12.047 |
| None |
Unchecked |
Inhibition |
nan |
% |
10.1016/j.bmcl.2017.01.026 |
| None |
Unchecked |
Ki |
nan |
None |
None |
| None |
Unchecked |
MIC |
2.46 |
ug.mL-1 |
10.1021/acs.jmedchem.1c00263 |
| None |
Unchecked |
MIC |
10.0 |
ug.mL-1 |
10.1021/acs.jmedchem.1c00263 |
| None |
Unchecked |
MIC |
2300.0 |
nM |
10.1016/j.ejmech.2020.112179 |
| None |
Unchecked |
MIC |
72900.0 |
nM |
10.1016/j.ejmech.2020.112179 |
| None |
Unchecked |
MIC |
145800.0 |
nM |
10.1016/j.ejmech.2020.112179 |
| None |
Unchecked |
MIC |
291700.0 |
nM |
10.1016/j.ejmech.2020.112179 |
| None |
Unchecked |
MIC100 |
0.25 |
ug ml-1 |
10.1016/j.ejmech.2020.112420 |
| None |
Unchecked |
MIC=>90 |
0.019 |
ug ml-1 |
10.1016/j.ejmech.2020.112538 |
| None |
Unchecked |
MIC=>90 |
0.052 |
ug ml-1 |
10.1016/j.ejmech.2020.112538 |
| None |
Unchecked |
MIC=>90 |
2.264 |
ug ml-1 |
10.1016/j.ejmech.2020.112538 |
| None |
Unchecked |
MIC=>90 |
10.0 |
ug ml-1 |
10.1016/j.ejmech.2020.112538 |
| None |
Unchecked |
MIC90 |
290.0 |
nM |
10.1021/acs.jmedchem.6b00415 |
| None |
Unchecked |
MIC>99 |
0.15 |
uM |
10.1021/acs.jmedchem.0c01374 |
| None |
Unchecked |
Potency |
3162.3 |
nM |
None |
| None |
Unchecked |
Potency |
19952.6 |
nM |
None |
| None |
Unchecked |
Ratio |
0.8 |
None |
10.1016/j.bmcl.2022.128692 |
| None |
Unchecked |
Ratio |
0.84 |
None |
10.1016/j.bmcl.2022.128692 |
| None |
Unchecked |
Ratio |
0.86 |
None |
10.1016/j.bmcl.2022.128692 |
| None |
Unchecked |
Ratio |
0.9 |
None |
10.1016/j.bmcl.2022.128692 |
| None |
Unchecked |
Ratio |
1.0 |
None |
10.1016/j.bmcl.2016.06.082 |
| None |
Unchecked |
Ratio |
1.0 |
None |
10.1016/j.ejmech.2009.05.009 |
| None |
Unchecked |
Ratio |
8.0 |
None |
10.1021/ml5001933 |
| None |
Unchecked |
Ratio |
128.0 |
None |
10.1021/jm701560p |
| None |
Unchecked |
Ratio |
320.0 |
None |
10.1016/j.bmcl.2019.01.004 |
| None |
Unchecked |
Ratio |
660.0 |
None |
10.1016/j.bmcl.2013.07.006 |
| None |
Unchecked |
Ratio |
1000.0 |
None |
10.1016/j.bmc.2007.08.064 |
| None |
Unchecked |
Ratio |
7325.0 |
None |
10.1016/j.bmcl.2009.09.095 |
| None |
Unchecked |
Ratio |
20000.0 |
None |
10.1016/j.bmcl.2011.04.072 |
| None |
Unchecked |
Ratio |
53613.0 |
None |
10.1016/j.bmcl.2009.09.095 |
| None |
Unchecked |
Ratio |
77277.0 |
None |
10.1016/j.bmcl.2009.09.095 |
| None |
Unchecked |
Ratio IC50 |
200.0 |
None |
None |
| None |
Unchecked |
Ratio IC50 |
nan |
None |
10.1016/j.ejmech.2013.12.057 |
| None |
Unchecked |
Selectivity Index |
2.0 |
None |
10.1016/j.ejmech.2019.111678 |
| None |
Unchecked |
Selectivity Index |
6.0 |
None |
10.1016/j.bmc.2015.07.053 |
| None |
Unchecked |
Selectivity Index |
6.25 |
None |
10.1016/j.bmc.2009.12.055 |
| None |
Unchecked |
Selectivity Index |
8.0 |
None |
10.1007/s00044-012-0074-2 |
| None |
Unchecked |
Selectivity Index |
9.0 |
None |
10.1016/j.ejmech.2012.10.047 |
| None |
Unchecked |
Selectivity Index |
22.7 |
None |
10.1016/j.ejmech.2020.112859 |
| None |
Unchecked |
Selectivity Index |
31.3 |
None |
10.1016/j.bmc.2014.05.064 |
| None |
Unchecked |
Selectivity Index |
31.3 |
None |
10.1016/j.bmc.2014.12.019 |
| None |
Unchecked |
Selectivity Index |
31.3 |
None |
10.1016/j.ejmech.2019.111578 |
| None |
Unchecked |
Selectivity Index |
35.0 |
None |
10.1016/j.bmc.2017.12.047 |
| None |
Unchecked |
Selectivity Index |
96.0 |
None |
10.1016/j.bmcl.2013.09.027 |
| None |
Unchecked |
Selectivity Index |
109.0 |
None |
10.1021/acs.jnatprod.9b01095 |
| None |
Unchecked |
Selectivity Index |
119.0 |
None |
10.1016/j.ejmech.2018.01.071 |
| None |
Unchecked |
Selectivity Index |
125.0 |
None |
10.1016/j.bmc.2015.07.053 |
| None |
Unchecked |
Selectivity Index |
200.0 |
None |
10.1016/j.bmc.2009.12.055 |
| None |
Unchecked |
Selectivity Index |
208.0 |
None |
10.1016/j.bmc.2016.12.038 |
| None |
Unchecked |
Selectivity Index |
250.0 |
None |
10.1016/j.bmc.2014.05.064 |
| None |
Unchecked |
Selectivity Index |
250.0 |
None |
10.1016/j.bmc.2014.12.019 |
| None |
Unchecked |
Selectivity Index |
250.0 |
None |
10.1016/j.ejmech.2019.111578 |
| None |
Unchecked |
Selectivity Index |
320.0 |
None |
10.1007/s00044-007-9073-0 |
| None |
Unchecked |
Selectivity Index |
320.0 |
None |
10.1016/j.bmcl.2013.09.013 |
| None |
Unchecked |
Selectivity Index |
499.0 |
None |
10.1007/s00044-012-0043-9 |
| None |
Unchecked |
Selectivity Index |
500.0 |
None |
10.1016/j.bmcl.2013.06.069 |
| None |
Unchecked |
Selectivity Index |
512.0 |
None |
10.1016/j.bmcl.2019.07.041 |
| None |
Unchecked |
Selectivity Index |
625.0 |
None |
10.1016/j.ejmech.2018.04.017 |
| None |
Unchecked |
Selectivity Index |
686.0 |
None |
10.1016/j.ejmech.2014.04.077 |
| None |
Unchecked |
Selectivity Index |
769.23 |
None |
10.1021/jm401735w |
| None |
Unchecked |
Selectivity Index |
830.0 |
None |
10.1021/jm300123s |
| None |
Unchecked |
Selectivity Index |
1000.0 |
None |
10.1016/j.ejmech.2012.10.047 |
| None |
Unchecked |
Selectivity Index |
1024.0 |
None |
10.1016/j.ejmech.2019.07.057 |
| None |
Unchecked |
Selectivity Index |
1333.3 |
None |
10.1016/j.bmcl.2015.11.071 |
| None |
Unchecked |
Selectivity Index |
1666.0 |
None |
10.1016/j.bmcl.2015.12.049 |
| None |
Unchecked |
Selectivity Index |
2000.0 |
None |
10.1016/j.bmc.2018.07.034 |
| None |
Unchecked |
Selectivity Index |
2222.2 |
None |
10.1016/j.bmcl.2015.11.071 |
| None |
Unchecked |
Selectivity Index |
2560.0 |
None |
10.1016/j.ejmech.2017.11.090 |
| None |
Unchecked |
Selectivity Index |
2564.1 |
None |
10.1016/j.bmcl.2016.02.043 |
| None |
Unchecked |
Selectivity Index |
2735.0 |
None |
10.1016/j.ejmech.2018.02.067 |
| None |
Unchecked |
Selectivity Index |
3030.3 |
None |
10.1016/j.bmcl.2016.02.043 |
| None |
Unchecked |
Selectivity Index |
3282.0 |
None |
10.1016/j.ejmech.2019.01.042 |
| None |
Unchecked |
Selectivity Index |
3333.0 |
None |
10.1021/np400497f |
| None |
Unchecked |
Selectivity Index |
4000.0 |
None |
10.1016/j.bmcl.2017.07.008 |
| None |
Unchecked |
Selectivity Index |
4096.0 |
None |
10.1016/j.bmc.2019.04.017 |
| None |
Unchecked |
Selectivity Index |
4096.0 |
None |
10.1016/j.ejmech.2018.09.049 |
| None |
Unchecked |
Selectivity Index |
5000.0 |
None |
10.1016/j.ejmech.2018.04.017 |
| None |
Unchecked |
Selectivity Index |
6081.0 |
None |
10.1021/jm101510d |
| None |
Unchecked |
Selectivity Index |
6400.0 |
None |
10.1021/acs.jmedchem.7b00582 |
| None |
Unchecked |
Selectivity Index |
8000.0 |
None |
10.1016/j.bmcl.2019.07.025 |
| None |
Unchecked |
Selectivity Index |
21665.0 |
None |
10.1016/j.ejmech.2010.11.023 |
| None |
Unchecked |
Selectivity Index |
30000.0 |
None |
10.1039/C3MD00251A |
| None |
Unchecked |
Selectivity Index |
40000.0 |
None |
10.1016/j.bmcl.2014.02.012 |
| None |
Unchecked |
Selectivity Index |
40000.0 |
None |
10.1016/j.bmcl.2016.06.082 |
| None |
Unchecked |
Selectivity Index |
60000.0 |
None |
10.1016/j.bmc.2015.04.001 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.bmc.2014.12.060 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.bmc.2019.07.045 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.bmcl.2010.08.046 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.bmcl.2012.11.052 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.bmcl.2018.03.021 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.ejmech.2011.07.052 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.ejmech.2011.11.033 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.ejmech.2014.02.065 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.ejmech.2014.03.024 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.ejmech.2016.07.039 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.ejmech.2018.04.017 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.ejmech.2019.05.013 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.ejmech.2019.07.052 |
| None |
Unchecked |
Selectivity Index |
nan |
None |
10.1016/j.ejmech.2019.111812 |
| None |
Unchecked |
Selectivity ratio |
500.0 |
None |
10.1039/C7MD00350A |
| None |
Unchecked |
Selectivity ratio |
1000.0 |
None |
10.1039/C7MD00366H |