| Bos taurus |
Progesterone receptor |
IC50 |
nan |
None |
None |
| Bos taurus |
Progesterone receptor |
Ki |
nan |
None |
None |
| Canis lupus familiaris |
Canis familiaris |
ED50 |
0.04 |
mg.kg-1 |
10.1021/jm00345a002 |
| Canis lupus familiaris |
Canis familiaris |
ED50 |
0.3 |
mg.kg-1 |
10.1021/jm00027a007 |
| Canis lupus familiaris |
Canis familiaris |
ED50 |
0.42 |
mg.kg-1 |
10.1021/jm00345a002 |
| Canis lupus familiaris |
Canis familiaris |
ED50 |
0.93 |
mg.kg-1 |
10.1021/jm00402a039 |
| Canis lupus familiaris |
Canis familiaris |
Inhibition |
41.0 |
% |
10.1021/jm00027a007 |
| Canis lupus familiaris |
MDCK |
logPapp |
-8.9 |
None |
10.1021/jm901846t |
| Cavia porcellus |
Cavia porcellus |
Inhibition |
44.0 |
% |
10.1021/jm000169n |
| Cavia porcellus |
Cavia porcellus |
Inhibition |
44.0 |
% |
10.1021/jm010217j |
| Cavia porcellus |
Histamine H2 receptor |
IC50 |
1.05 |
ug.mL-1 |
10.1016/0960-894X(96)00313-7 |
| Cavia porcellus |
Histamine H2 receptor |
IC50 |
3400.0 |
nM |
10.1021/jm00027a007 |
| Cavia porcellus |
Histamine H2 receptor |
Inhibition |
44.0 |
% |
10.1021/jm00027a007 |
| Cavia porcellus |
Histamine H2 receptor |
Kb |
166.0 |
nM |
10.1021/jm00161a005 |
| Cavia porcellus |
Histamine H2 receptor |
KB |
6.3e-08 |
None |
10.1021/jm00163a001 |
| Cavia porcellus |
Histamine H2 receptor |
Kd |
64.57 |
nM |
10.1021/jm00091a012 |
| Cavia porcellus |
Histamine H2 receptor |
Kd |
169.82 |
nM |
10.1016/s0960-894x(03)00235-x |
| Cavia porcellus |
Histamine H2 receptor |
Ki |
53.7 |
nM |
10.1021/jm00090a013 |
| Cavia porcellus |
Histamine H2 receptor |
Ki |
501.19 |
nM |
10.1021/jm00345a002 |
| Cavia porcellus |
Histamine H2 receptor |
-Log KB |
7.05 |
% |
10.1021/jm00398a028 |
| Cavia porcellus |
Histamine H2 receptor |
-Log KB |
7.32 |
None |
10.1021/jm00345a002 |
| Cavia porcellus |
Histamine H2 receptor |
pKB |
7.2 |
None |
10.1021/jm00090a013 |
| Cavia porcellus |
Histamine H2 receptor |
Relative potency |
631.0 |
% |
10.1021/jm00090a013 |
| Cavia porcellus |
Histamine H3 receptor |
KB |
1.2e-06 |
None |
10.1021/jm00163a001 |
| Cavia porcellus |
Leukotriene C4 synthase |
IC50 |
nan |
None |
None |
| Cavia porcellus |
Leukotriene C4 synthase |
Ki |
nan |
None |
None |
| Cavia porcellus |
Serotonin 4 (5-HT4) receptor |
IC50 |
nan |
None |
None |
| Cavia porcellus |
Serotonin 4 (5-HT4) receptor |
Ki |
nan |
None |
None |
| Cryptosporidium parvum |
Cryptosporidium parvum |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Entamoeba histolytica |
Entamoeba histolytica |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Helicobacter pylori |
Helicobacter pylori |
MIC |
100.0 |
ug.mL-1 |
10.1016/0960-894X(96)00313-7 |
| Helicobacter pylori |
Helicobacter pylori |
MIC |
1600.0 |
ug.mL-1 |
10.1021/jm000169n |
| Helicobacter pylori |
Helicobacter pylori |
MIC |
1600.0 |
ug.mL-1 |
10.1021/jm010217j |
| Homo sapiens |
Acetylcholinesterase |
AC50 |
950.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Acetylcholinesterase |
EC30 |
1.8 |
uM |
10.1021/jm00057a007 |
| Homo sapiens |
Acetylcholinesterase |
IC50 |
650.0 |
nM |
10.1021/jm00057a007 |
| Homo sapiens |
Acetylcholinesterase |
IC50 |
2300.0 |
nM |
10.1021/jm00084a015 |
| Homo sapiens |
Acetylcholinesterase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Acetylcholinesterase |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A2a receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A2a receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A2a receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Adenosine A3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Adenosine A3 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Adenosine A3 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1a adrenergic receptor |
AC50 |
18690.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-1d adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-1d adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2a adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2a adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2b adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2b adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2b adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Alpha-2c adrenergic receptor |
AC50 |
17000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Alpha-2c adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Alpha-2c adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Androgen Receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Angiotensin II type 2 (AT-2) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Angiotensin II type 2 (AT-2) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-1 adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-1 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-1 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-2 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-2 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Beta-3 adrenergic receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Beta-3 adrenergic receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Beta-3 adrenergic receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Bile salt export pump |
AC50 |
51000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bile salt export pump |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Bile salt export pump |
IC50 |
1000000.0 |
nM |
10.1124/dmd.111.040758 |
| Homo sapiens |
Bradykinin B1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bradykinin B2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Bradykinin B2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Bradykinin B2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Caco-2 |
logPapp |
-6.31 |
None |
10.1016/j.bmc.2009.08.022 |
| Homo sapiens |
Caco-2 |
logPapp |
-6.2 |
None |
10.1016/j.bmc.2011.03.011 |
| Homo sapiens |
Caco-2 |
Papp |
0.2 |
ucm/s |
10.1021/jm401905m |
| Homo sapiens |
Caco-2 |
Papp |
0.23 |
ucm/s |
10.1016/j.ejmech.2015.06.031 |
| Homo sapiens |
Caco-2 |
Papp |
0.4 |
ucm/s |
10.1016/j.ejmech.2014.02.003 |
| Homo sapiens |
Caco-2 |
Papp |
0.5 |
ucm/s |
10.1021/jm401838x |
| Homo sapiens |
Caco-2 |
Papp |
0.6 |
10'-6 cm/s |
10.1016/j.bmc.2010.10.052 |
| Homo sapiens |
Caco-2 |
Papp |
0.6 |
ucm/s |
10.1016/j.ejmech.2012.01.033 |
| Homo sapiens |
Caco-2 |
Papp |
0.7 |
10'-6 cm/s |
10.1021/jm101067y |
| Homo sapiens |
Caco-2 |
Papp |
1.2 |
ucm/s |
10.1021/jm401905m |
| Homo sapiens |
Caco-2 |
Papp |
1.5 |
10'6cm/s |
10.1016/j.bmcl.2010.12.079 |
| Homo sapiens |
Caco-2 |
Papp |
1.5 |
cm/s |
10.1016/j.bmcl.2010.08.117 |
| Homo sapiens |
Caco-2 |
Papp |
2.6 |
ucm/s |
10.1016/j.ejmech.2014.02.003 |
| Homo sapiens |
Caco-2 |
Papp |
3.1 |
ucm/s |
10.1016/j.ejmech.2015.06.031 |
| Homo sapiens |
Caco-2 |
Papp |
3.8 |
ucm/s |
10.1021/jm401838x |
| Homo sapiens |
Caco-2 |
permeability |
0.3 |
10'-6 cm/s |
10.1128/aac.00246-07 |
| Homo sapiens |
Caco-2 |
permeability |
5.6 |
10'-6 cm/s |
10.1128/aac.00246-07 |
| Homo sapiens |
Caco-2 |
permeability |
nan |
None |
10.1016/j.bmc.2011.03.011 |
| Homo sapiens |
Caco-2 |
Ratio |
1.0 |
None |
10.1016/j.bmc.2010.10.052 |
| Homo sapiens |
Caco-2 |
Ratio |
6.6 |
None |
10.1016/j.ejmech.2014.02.003 |
| Homo sapiens |
Caco-2 |
Ratio |
7.2 |
None |
10.1021/jm401838x |
| Homo sapiens |
Caco-2 |
Ratio |
13.5 |
None |
10.1016/j.ejmech.2015.06.031 |
| Homo sapiens |
Calcitonin receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Calcitonin receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Canalicular multispecific organic anion transporter 1 |
Activity |
52.0 |
% |
10.1021/jm7015683 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 1 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Canalicular multispecific organic anion transporter 2 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Cannabinoid CB1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cannabinoid CB1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cannabinoid CB1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase II |
IC50 |
nan |
None |
None |
| Homo sapiens |
Carbonic anhydrase II |
Ki |
nan |
None |
None |
| Homo sapiens |
Caspase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Caspase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cathepsin G |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cathepsin G |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 2 |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 4 |
Ki |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
C-C chemokine receptor type 5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin A receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cholecystokinin A receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin A receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Cholecystokinin B receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Chromobox protein homolog 1 |
Potency |
89125.1 |
nM |
None |
| Homo sapiens |
Corticotropin releasing factor receptor 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Corticotropin releasing factor receptor 2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-1 |
AC50 |
13080.1 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-1 |
AC50 |
16209.9 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-2 |
AC50 |
14174.2 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Cyclooxygenase-2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cyclooxygenase-2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cysteinyl leukotriene receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cysteinyl leukotriene receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 1A2 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 1A2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2A6 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2A6 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2C19 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C19 |
Potency |
39810.7 |
nM |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2C9 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2C9 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2D6 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 2D6 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2E1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2E1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 2J2 |
IC50 |
50000.0 |
nM |
10.1124/dmd.112.048264 |
| Homo sapiens |
Cytochrome P450 3A4 |
AC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
IC50 |
50000.0 |
nM |
10.1021/jm021012t |
| Homo sapiens |
Cytochrome P450 3A4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Cytochrome P450 3A4 |
Inhibition |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
Cytochrome P450 3A4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Delta opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Delta opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Delta opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
DNA polymerase iota |
Potency |
89125.1 |
nM |
None |
| Homo sapiens |
Dopamine D1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D1 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D2 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D3 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D3 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D3 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine D4 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine D4 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine D4 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Dopamine transporter |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Dopamine transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Dopamine transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Endoplasmic reticulum-associated amyloid beta-peptide-binding protein |
Potency |
3162.3 |
nM |
None |
| Homo sapiens |
Endothelin receptor ET-A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Endothelin receptor ET-A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-A |
Ki |
nan |
None |
None |
| Homo sapiens |
Endothelin receptor ET-B |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Epidermal growth factor receptor erbB1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Equilibrative nucleoside transporter 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor beta |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Estrogen receptor beta |
IC50 |
nan |
None |
None |
| Homo sapiens |
Estrogen receptor beta |
Ki |
nan |
None |
None |
| Homo sapiens |
Gastric inhibitory polypeptide receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Ghrelin receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucagon receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Glucocorticoid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Glucocorticoid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Hepatocyte |
CL |
2.9 |
mL.min-1.kg-1 |
10.1016/j.ejmech.2008.07.027 |
| Homo sapiens |
Hepatocyte |
logCL |
0.4624 |
None |
10.1016/j.ejmech.2008.07.027 |
| Homo sapiens |
HERG |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
HERG |
IC50 |
nan |
None |
None |
| Homo sapiens |
HERG |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Histamine H1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H2 receptor |
AC50 |
227.5 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H2 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Histamine H2 receptor |
Kd |
63.0 |
nM |
10.1007/s00044-004-0012-z |
| Homo sapiens |
Histamine H2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Histamine H3 receptor |
AC50 |
4800.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histamine H3 receptor |
AC50 |
18499.9 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Histone acetyltransferase GCN5 |
Potency |
17782.8 |
nM |
None |
| Homo sapiens |
Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 |
Potency |
11220.2 |
nM |
None |
| Homo sapiens |
HMG-CoA reductase |
IC50 |
nan |
None |
None |
| Homo sapiens |
HMG-CoA reductase |
Ki |
nan |
None |
None |
| Homo sapiens |
Homo sapiens |
% absorbed |
50.0 |
% |
10.1021/jm001020e |
| Homo sapiens |
Homo sapiens |
Activity |
nan |
None |
None |
| Homo sapiens |
Homo sapiens |
CL |
0.153 |
mL.min-1.kg-1 |
10.1124/dmd.112.049312 |
| Homo sapiens |
Homo sapiens |
CL |
0.161 |
mL.min-1.kg-1 |
10.1124/dmd.112.049312 |
| Homo sapiens |
Homo sapiens |
CL |
2.2 |
mL.min-1.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
CL |
9.6 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
CL |
9.6 |
mL.min-1.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
CL_renal |
7.4 |
mL.min-1.kg-1 |
10.1021/jm900403j |
| Homo sapiens |
Homo sapiens |
CL_renal |
7.4 |
mL.min-1.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
F |
50.0 |
% |
10.1021/jm901846t |
| Homo sapiens |
Homo sapiens |
Fa |
0.65 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
F_fraction |
0.6 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Fg |
1.02 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Fh |
0.9 |
None |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Vdss |
1.2 |
L.kg-1 |
10.1021/jm901371v |
| Homo sapiens |
Homo sapiens |
Vdss |
1.3 |
L.kg-1 |
10.1016/j.ejmech.2009.06.004 |
| Homo sapiens |
Hypoxia-inducible factor 1 alpha |
Potency |
3981.1 |
nM |
None |
| Homo sapiens |
Interleukin-8 receptor A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor A |
Ki |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor B |
IC50 |
nan |
None |
None |
| Homo sapiens |
Interleukin-8 receptor B |
Ki |
nan |
None |
None |
| Homo sapiens |
Kappa opioid receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Kappa opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Kappa opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Leukocyte common antigen |
IC50 |
nan |
None |
None |
| Homo sapiens |
Leukocyte common antigen |
Ki |
nan |
None |
None |
| Homo sapiens |
Leukocyte elastase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Leukocyte elastase |
Ki |
nan |
None |
None |
| Homo sapiens |
Liver microsomes |
Activity |
nan |
None |
10.1021/tx300075j |
| Homo sapiens |
Liver microsomes |
Stability |
nan |
% |
10.1021/tx300075j |
| Homo sapiens |
MAP kinase ERK1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK1 |
Ki |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase ERK2 |
Ki |
nan |
None |
None |
| Homo sapiens |
MAP kinase p38 alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
MAP kinase p38 alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase-1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase-1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase 9 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Matrix metalloproteinase 9 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 3 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Melanocortin receptor 3 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 3 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 4 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Melanocortin receptor 4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Melanocortin receptor 5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Menin/Histone-lysine N-methyltransferase MLL |
Potency |
39810.7 |
nM |
None |
| Homo sapiens |
Monoamine oxidase A |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Monoamine oxidase A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Monoamine oxidase A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Monoamine oxidase A |
Ki |
nan |
None |
None |
| Homo sapiens |
Motilin receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Multidrug and toxin extrusion protein 1 |
IC50 |
8300.0 |
nM |
10.1021/jm301302s |
| Homo sapiens |
Multidrug and toxin extrusion protein 1 |
Inhibition |
29.0 |
% |
10.1021/jm301302s |
| Homo sapiens |
Multidrug resistance-associated protein 4 |
IC50 |
133000.0 |
nM |
10.1093/toxsci/kft176 |
| Homo sapiens |
Mu opioid receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Mu opioid receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Mu opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Mu opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
AC50 |
5000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
AC50 |
8600.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
AC50 |
2550.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
AC50 |
5562.6 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
AC50 |
8600.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M3 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M4 |
Ki |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Muscarinic acetylcholine receptor M5 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurokinin 1 receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neurokinin 1 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neurokinin 1 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurokinin 2 receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neurokinin 2 receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Neuronal acetylcholine receptor protein alpha-4 subunit |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Neuropeptide Y receptor type 2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Neurotensin receptor 1 |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Norepinephrine transporter |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Norepinephrine transporter |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Norepinephrine transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Norepinephrine transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Nuclear factor NF-kappa-B p105 subunit |
Potency |
707.9 |
nM |
None |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
-2.4 |
nM/mg*min |
10.1021/jm021012t |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
0.0 |
% |
10.1021/jm021012t |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
nan |
None |
10.1016/s0378-5173(03)00372-7 |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
nan |
None |
10.1021/acs.jmedchem.9b00720 |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
nan |
None |
10.1023/a:1007692622216 |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
nan |
None |
10.1023/a:1025001131513 |
| Homo sapiens |
P-glycoprotein 1 |
Activity |
nan |
None |
None |
| Homo sapiens |
P-glycoprotein 1 |
IC50 |
50000.0 |
nM |
10.1021/jm021012t |
| Homo sapiens |
P-glycoprotein 1 |
Inhibition |
0.0 |
% |
10.1021/jm021012t |
| Homo sapiens |
P-glycoprotein 1 |
% maximum response |
2.92 |
% |
None |
| Homo sapiens |
P-glycoprotein 1 |
Papp |
14.4 |
nm/s |
None |
| Homo sapiens |
P-glycoprotein 1 |
Papp |
19.5 |
nm/s |
None |
| Homo sapiens |
P-glycoprotein 1 |
Ratio_ATPase activity |
1.23 |
None |
None |
| Homo sapiens |
P-glycoprotein 1 |
Ratio_Papp |
1.35 |
None |
None |
| Homo sapiens |
Phosphodiesterase 3A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 4A |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 4D |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Phosphodiesterase 5A |
IC50 |
nan |
None |
None |
| Homo sapiens |
Phosphodiesterase 5A |
Ki |
nan |
None |
None |
| Homo sapiens |
Plasma |
fCmax |
2.703 |
uM |
10.1124/dmd.111.040758 |
| Homo sapiens |
Platelet activating factor receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Platelet activating factor receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Potassium-transporting ATPase |
IC50 |
40.0 |
nM |
10.1021/jm00117a018 |
| Homo sapiens |
Potassium-transporting ATPase alpha chain 2 |
Inhibition |
100.0 |
% |
10.1021/jm00117a018 |
| Homo sapiens |
Prelamin-A/C |
Potency |
79.4 |
nM |
None |
| Homo sapiens |
Progesterone receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Protein kinase C alpha |
IC50 |
nan |
None |
None |
| Homo sapiens |
Protein kinase C alpha |
Ki |
nan |
None |
None |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Receptor protein-tyrosine kinase erbB-2 |
Ki |
nan |
None |
None |
| Homo sapiens |
Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serine/threonine protein phosphatase 2B catalytic subunit, alpha isoform |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 1a (5-HT1a) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 1a (5-HT1a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2a (5-HT2a) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2b (5-HT2b) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 2c (5-HT2c) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin 3a (5-HT3a) receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin 6 (5-HT6) receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Serotonin transporter |
AC50 |
9260.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
AC50 |
10999.9 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Serotonin transporter |
IC50 |
nan |
None |
None |
| Homo sapiens |
Serotonin transporter |
Ki |
nan |
None |
None |
| Homo sapiens |
Serum albumin |
Log K' |
0.1 |
None |
10.1021/jm010960b |
| Homo sapiens |
Sigma opioid receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Sigma opioid receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Sodium channel protein type V alpha subunit |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Solute carrier family 22 member 1 |
Activity |
21.7 |
uM |
10.1124/mol.63.3.489 |
| Homo sapiens |
Solute carrier family 22 member 1 |
Drug uptake |
600.0 |
pmol/mg |
10.1021/jm400966v |
| Homo sapiens |
Solute carrier family 22 member 1 |
FC |
18.0 |
None |
10.1021/jm400966v |
| Homo sapiens |
Solute carrier family 22 member 1 |
Inhibition |
28.8 |
% |
10.1021/jm8003152 |
| Homo sapiens |
Solute carrier family 22 member 2 |
Activity |
nan |
None |
10.1038/nrd3028 |
| Homo sapiens |
Solute carrier family 22 member 2 |
Drug uptake |
22.0 |
pmol/mg |
10.1021/jm400966v |
| Homo sapiens |
Solute carrier family 22 member 2 |
FC |
1.6 |
None |
10.1021/jm400966v |
| Homo sapiens |
Solute carrier family 22 member 8 |
Km |
234000.0 |
nM |
10.1124/jpet.105.094052 |
| Homo sapiens |
Thrombin |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Thromboxane A2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Thromboxane-A synthase |
IC50 |
nan |
None |
None |
| Homo sapiens |
Thromboxane-A synthase |
Ki |
nan |
None |
None |
| Homo sapiens |
Thyroid stimulating hormone receptor |
Potency |
7943.3 |
nM |
None |
| Homo sapiens |
Type-1 angiotensin II receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Tyrosine-protein kinase FYN |
IC50 |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase FYN |
Ki |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase LCK |
IC50 |
nan |
None |
None |
| Homo sapiens |
Tyrosine-protein kinase LCK |
Ki |
nan |
None |
None |
| Homo sapiens |
Ubiquitin carboxyl-terminal hydrolase 1 |
Potency |
17782.8 |
nM |
None |
| Homo sapiens |
Vascular endothelial growth factor receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vascular endothelial growth factor receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasoactive intestinal polypeptide receptor 1 |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vasoactive intestinal polypeptide receptor 1 |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasopressin V1a receptor |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Homo sapiens |
Vasopressin V1a receptor |
IC50 |
nan |
None |
None |
| Homo sapiens |
Vasopressin V1a receptor |
Ki |
nan |
None |
None |
| Homo sapiens |
Vasopressin V2 receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Leishmania amazonensis |
Leishmania amazonensis |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Leishmania donovani |
Leishmania donovani |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Leishmania infantum |
Leishmania infantum |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Leishmania major |
Leishmania major |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Leishmania mexicana |
Leishmania mexicana |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Mus musculus |
Monoamine oxidase A |
Activity |
nan |
None |
10.1021/jm800656v |
| Mus musculus |
Mus musculus |
Permeability |
nan |
None |
10.1021/jm990968+ |
| Mus musculus |
Nitric oxide synthase, inducible |
IC50 |
nan |
None |
None |
| Mus musculus |
Nitric oxide synthase, inducible |
Ki |
nan |
None |
None |
| Mus musculus |
P-glycoprotein 1 |
IC50 |
50000.0 |
nM |
10.1021/jm021012t |
| Mus musculus |
P-glycoprotein 3 |
IC50 |
50000.0 |
nM |
10.1021/jm021012t |
| Oryctolagus cuniculus |
Angiotensin-converting enzyme |
IC50 |
nan |
None |
None |
| Oryctolagus cuniculus |
Angiotensin-converting enzyme |
Ki |
nan |
None |
None |
| Oryctolagus cuniculus |
Arachidonate 15-lipoxygenase |
IC50 |
nan |
None |
None |
| Oryctolagus cuniculus |
Arachidonate 15-lipoxygenase |
Ki |
nan |
None |
None |
| Plasmodium falciparum |
Plasmodium falciparum |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Plasmodium falciparum |
Plasmodium falciparum |
Potency |
19011.5 |
nM |
None |
| Pneumocystis carinii |
Pneumocystis carinii |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Rattus norvegicus |
Aldose reductase |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Aldose reductase |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1a adrenergic receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1a adrenergic receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1b adrenergic receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Alpha-1b adrenergic receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Androgen Receptor |
AC50 |
30000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Androgen Receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Androgen Receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Bile salt export pump |
IC50 |
1000000.0 |
nM |
10.1124/dmd.111.040758 |
| Rattus norvegicus |
Cyclooxygenase-1 |
AC50 |
7782.7 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
GABA receptor alpha-1 subunit |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
GABA receptor alpha-1 subunit |
AC50 |
16339.9 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Glutamate (NMDA) receptor subunit zeta 1 |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Glycine receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Glycine receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Insulin receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Insulin receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Muscarinic acetylcholine receptor M1 |
Potency |
15848.9 |
nM |
None |
| Rattus norvegicus |
Nitric-oxide synthase, brain |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Nitric-oxide synthase, brain |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Peripheral myelin protein 22 |
Potency |
20.3 |
nM |
None |
| Rattus norvegicus |
Plasma |
Fu |
0.95 |
None |
10.1021/jm901371v |
| Rattus norvegicus |
Plasma |
logFu |
0.85 |
None |
10.1016/j.ejmech.2009.06.004 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
-1.23 |
None |
10.1021/jm00398a028 |
| Rattus norvegicus |
Rattus norvegicus |
Activity |
0.0586 |
None |
10.1021/jm00398a028 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
33000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
34000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
35000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
41700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
42200.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
42700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALB |
43300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.3 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.4 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.5 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.6 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALBGLOB |
1.7 |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
349.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
358.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
373.17 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
378.5 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
392.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
395.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
562.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
621.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
642.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
677.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
741.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
783.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
785.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
793.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
802.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
835.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
839.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
849.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
852.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
872.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
881.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
885.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
906.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
907.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
918.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
924.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
929.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
931.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
944.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
955.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
966.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
967.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
970.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1000.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1036.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1059.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALP |
1082.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
29.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
31.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
32.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
32.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
32.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
32.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
33.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
33.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
33.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
34.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
35.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
36.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
36.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
36.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
37.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
38.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
38.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
41.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
42.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
43.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
49.17 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
50.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
53.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
54.17 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
ALT |
57.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
17.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
18.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
18.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
19.8 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
20.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
21.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
21.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
APTT |
23.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
60.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
60.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
61.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
61.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
61.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
62.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
62.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
63.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
63.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
63.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
63.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
64.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
64.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
65.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
65.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
65.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
66.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
66.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
67.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
68.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
69.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
69.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
70.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
70.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
70.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
80.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
81.83 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
82.17 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
86.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
90.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
AST |
93.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BASO |
0.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BASOLE |
0.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.6 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.62 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.64 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.66 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.68 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.7 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.74 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.78 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.8 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.84 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.86 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.88 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.9 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.92 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.94 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.96 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
0.98 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILDIR |
1.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
1.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
1.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
1.8 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BILI |
2.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
84.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
88.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
94.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
96.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
98.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
100.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
102.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
108.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
114.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
144.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
146.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
146.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
148.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
150.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
154.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
156.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
156.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
158.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
160.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
162.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
163.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
164.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
166.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
166.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
168.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
170.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
172.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
174.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
176.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
178.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
BUN |
180.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
103.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
104.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
105.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
106.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
107.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
108.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
109.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CALCIUM |
110.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
99.0 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
99.17 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
100.33 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
101.33 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHLORIDE |
102.0 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
503.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
642.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
646.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
652.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
664.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
672.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
680.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
680.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
686.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
692.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
696.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
704.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
708.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
710.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
711.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
728.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
730.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
732.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
742.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
752.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
756.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
764.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
768.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
772.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
784.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
786.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
792.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
800.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
808.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
816.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
822.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
842.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
844.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
846.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CHOL |
924.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
245.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
258.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
268.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
273.5 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
304.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CK |
330.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
101.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
102.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
102.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
102.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.2 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.6 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
103.8 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.0 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Cl |
104.4 |
meq/L |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CL |
1.4 |
mL.min-1.kg-1 |
10.1124/dmd.112.049312 |
| Rattus norvegicus |
Rattus norvegicus |
CL |
1.556 |
mL.min-1.kg-1 |
10.1124/dmd.112.049312 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
21330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
27330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
28000000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
30330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
31000000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CO2 |
34330000.0 |
nM |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
1.8 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
1.9 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.2 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
2.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
3.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
4.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
CREAT |
5.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
ED50 |
2.4 |
mg.kg-1 |
10.1021/jm00163a053 |
| Rattus norvegicus |
Rattus norvegicus |
ED50 |
3.6 |
mg.kg-1 |
10.1021/jm00163a053 |
| Rattus norvegicus |
Rattus norvegicus |
ED50 |
9.1 |
mg.kg-1 |
10.1021/jm00117a018 |
| Rattus norvegicus |
Rattus norvegicus |
ED50 |
30.5 |
mg.kg-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
ED50 |
100.0 |
mg.kg-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
ED50 |
109.0 |
nmol |
10.1007/s00044-004-0012-z |
| Rattus norvegicus |
Rattus norvegicus |
ED50 |
nan |
mg.kg-1 |
10.1021/jm00163a053 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
0.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
23.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
49.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
61.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
64.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOS |
82.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.17 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
0.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
EOSLE |
1.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2090.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2150.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2162.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2168.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2172.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2208.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2214.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2238.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2240.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2254.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2258.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2270.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2274.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2288.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2296.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2300.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2316.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2328.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2332.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2342.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2344.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2350.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2382.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2388.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2392.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2410.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2422.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2434.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
FIBRINO |
2438.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Flow rate |
53.4 |
ml min-1 100g-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Flow rate |
55.4 |
ml min-1 100g-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Flow rate |
82.3 |
ml min-1 100g-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Flow rate |
85.3 |
ml min-1 100g-1 |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
0.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GGT |
1.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1418.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1426.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1460.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1480.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1540.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1573.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1812.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1882.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1902.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1904.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1906.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1928.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1930.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1934.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1942.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1952.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1956.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1966.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1970.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1980.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1984.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1986.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
1988.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2038.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2042.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2046.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2052.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2108.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2116.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2146.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2192.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2202.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2236.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
GLUC |
2244.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
34.53 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
35.28 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
35.4 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.1 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.57 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
36.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
37.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
38.9 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
39.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
40.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
42.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
43.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
43.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
43.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HCT |
45.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
127000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
129000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
131000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
132000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
133000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
134000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
135000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
136000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
136700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
137000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
139000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
140000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
140000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
141000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
142200.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
142700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
144700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
145000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
146000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
147000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
148000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
153000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
153000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
155000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
156000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
HGB |
157000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
-16.8 |
% |
10.1021/jm00091a012 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
3.0 |
% |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
72.0 |
% |
10.1021/jm000169n |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
72.0 |
% |
10.1021/jm00027a007 |
| Rattus norvegicus |
Rattus norvegicus |
Inhibition |
72.0 |
% |
10.1021/jm010217j |
| Rattus norvegicus |
Rattus norvegicus |
LD50 |
nan |
mg.kg-1 |
10.1021/jm00163a053 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
98.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
111.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
111.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
112.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
114.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
120.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
121.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
122.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
126.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
126.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
126.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
127.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
130.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
132.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
141.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
144.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
147.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
148.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
153.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
153.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
154.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
159.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
164.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
164.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
168.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
169.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
174.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
177.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
178.4 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
180.0 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
185.2 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
195.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
205.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
216.6 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
228.8 |
IU.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
312.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
319.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LDH |
426.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
8.67 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
9.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
9.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
10.0 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LIPASE |
10.33 |
U.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
12269.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
12453.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
14230.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
14943.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
15225.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYM |
16689.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
67.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
68.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
72.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
72.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
72.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
73.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
75.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
75.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
76.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
76.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
76.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
77.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
77.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
78.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
79.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
79.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
79.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
80.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
81.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
82.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
82.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
83.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
83.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
89.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
91.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
92.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
LYMLE |
93.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
19.8 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.1 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.5 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
20.6 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.2 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.3 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.5 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.6 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.7 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.8 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
21.9 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.0 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.1 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.3 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.4 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.5 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
22.7 |
pg |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.67 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.8 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
24.97 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
25.02 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
25.53 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCH |
25.9 |
pg |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
34.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
35.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
36.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
388500.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
393300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
395700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
396000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
401000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCHC |
404300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
56.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
56.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
58.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
58.6 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
58.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
59.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
60.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
61.82 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
62.8 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.0 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.03 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.1 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.3 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.52 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.7 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.8 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
63.9 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.2 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.4 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.47 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.5 |
fL |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MCV |
64.73 |
fL |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
0.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
32.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
42.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
160.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
162.67 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONO |
303.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
0.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
0.17 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
0.33 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
1.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
1.17 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
1.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
1.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
2.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
MONOLE |
3.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
6.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
7.0 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
7.17 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
7.67 |
% |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
10.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
11.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
12.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
12.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
13.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
14.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
15.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
16.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
17.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
18.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
18.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
18.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
18.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
19.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
19.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
19.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
21.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
24.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTLE |
26.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
970.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1061.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1084.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1138.33 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1162.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
NEUTSG |
1274.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
66.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
69.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
71.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
72.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
74.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
75.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
76.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
77.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
78.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
79.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
80.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
82.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
83.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
84.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
85.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
86.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
87.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
113.8 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
116.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
121.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
125.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
126.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOS |
150.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1292.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1326.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1328.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1336.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1340.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1342.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1368.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1372.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1378.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1382.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1384.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1408.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1412.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1426.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1428.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1438.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1460.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1474.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1484.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1488.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1492.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1514.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1516.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1520.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1526.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1528.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1556.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1594.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PHOSLPD |
1696.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1010000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1037000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1062000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1063000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1100000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1119000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1120000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1130000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1143000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1151000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1162000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1165000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1167000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1168000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1173000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1174000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1180000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1180670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1184000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1187000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1188000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1198000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1204000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1209000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1218000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1224000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1233000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1234330.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1250830.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1254000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1259000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1272000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1274000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1282000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1299000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1304000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PLAT |
1360670.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
3.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
3.7 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
3.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
3.9 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.1 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
4.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.43 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
6.46 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
7.08 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
7.11 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
POTASSIUM |
7.13 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
53000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
54000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
55000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
56000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
56000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
57000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
57700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
58000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
58300.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
60000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
60000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
61000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
61000.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
62000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
62700.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
PROT |
63000.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
11.9 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.0 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.1 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.2 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.3 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.4 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.5 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.6 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
PT |
12.7 |
s |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5360000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5580000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5610000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5710000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5760000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5852000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5880000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
5962000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6032000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6050000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6060000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6072000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6088000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6112000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6138000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6144000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6160000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6164000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6172000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6180000.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6214000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6276000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6294000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6314000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6322000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6390000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6394000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6432000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6442000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6464000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6780000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6860000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
6872000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7206000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7470000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7698000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7792000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBC |
7974000.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
0.0 |
/100WBC |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RBCNUC |
0.33 |
/100WBC |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
1.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
2.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
3.7 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
3.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
4.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
5.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.5 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.8 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
6.9 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.0 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.1 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.2 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.3 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.4 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
RETIRBC |
7.6 |
% |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
139.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
140.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.4 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.6 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
141.8 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.0 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.2 |
mEq.L-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.22 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
142.75 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
144.53 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
145.5 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
145.6 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
SODIUM |
147.4 |
mEq.L-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
210.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
211.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
211.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
213.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
213.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
214.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
216.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
216.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
216.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
216.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
218.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
226.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
228.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
228.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
230.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
231.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
232.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
234.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
237.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
260.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
264.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
264.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
265.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
305.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
309.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
314.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
314.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
379.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
381.6 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
385.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TERMBW |
391.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Tissue Severity Score |
nan |
None |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
Tissue Severity Score |
nan |
None |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
222.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
288.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
302.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
432.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
448.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
460.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
478.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
480.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
508.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
528.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
554.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
574.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
678.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
786.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
800.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
824.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
830.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
858.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
900.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
924.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
960.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1036.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1040.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1072.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1074.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1248.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1254.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1256.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1424.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
TRIG |
1520.0 |
ug.mL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
13.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
13.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
15.5 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
16.7 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
23.0 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
URATE |
27.3 |
ug.mL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7140.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7410.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7510.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7540.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
7600.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8120.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8160.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8210.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8430.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8500.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8750.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8760.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8770.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
8870.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9080.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9190.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9390.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9530.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9630.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9740.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9900.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
9990.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10070.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10120.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10420.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10470.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
10960.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11120.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11200.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11220.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11770.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
11970.0 |
cells.uL-1 |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
13400.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
13900.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
15430.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
16080.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
16600.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WBC |
18070.0 |
cells.uL-1 |
10.6019/CHEMBL3885881 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
0.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
1.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
2.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
8.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
9.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
10.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.1 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
11.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.0 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
12.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
13.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
13.8 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.2 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
14.7 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
15.4 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
15.5 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
15.9 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Rattus norvegicus |
WEIGHT |
16.3 |
g |
10.6019/CHEMBL3885861 |
| Rattus norvegicus |
Serotonin 1a (5-HT1a) receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1a (5-HT1a) receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1b (5-HT1b) receptor |
IC50 |
nan |
None |
None |
| Rattus norvegicus |
Serotonin 1b (5-HT1b) receptor |
Ki |
nan |
None |
None |
| Rattus norvegicus |
Voltage-gated L-type calcium channel alpha-1C subunit |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Rattus norvegicus |
Voltage-gated N-type calcium channel alpha-1B subunit |
AC50 |
10000.0 |
nM |
10.1038/s41467-023-40064-9 |
| Saccharomyces cerevisiae |
Saccharomyces cerevisiae |
Potency |
14581.0 |
nM |
None |
| Severe acute respiratory syndrome coronavirus 2 |
Replicase polyprotein 1ab |
Inhibition |
26.81 |
% |
10.6019/CHEMBL4495564 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Hit score |
0.2229 |
None |
10.1101/2020.04.21.054387 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
19952.62 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
IC50 |
20000.0 |
nM |
10.6019/CHEMBL4651402 |
| Severe acute respiratory syndrome coronavirus 2 |
SARS-CoV-2 |
Inhibition |
-0.26 |
% |
10.6019/CHEMBL4495565 |
| Toxoplasma gondii |
Toxoplasma gondii |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Trichomonas vaginalis |
Trichomonas vaginalis |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Trypanosoma brucei |
6-phospho-1-fructokinase |
Potency |
37933.0 |
nM |
None |
| Trypanosoma brucei |
Trypanosoma brucei |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Trypanosoma brucei brucei |
Trypanosoma brucei brucei |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Trypanosoma brucei rhodesiense |
Trypanosoma brucei rhodesiense |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| Trypanosoma cruzi |
Trypanosoma cruzi |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| None |
ADMET |
B(DPB) |
3.9 |
% |
10.1021/jm040760a |
| None |
ADMET |
Biotransformation |
nan |
None |
10.1038/s41586-019-1291-3 |
| None |
ADMET |
CL |
3.0 |
mL.min-1.g-1 |
10.6019/CHEMBL3301361 |
| None |
ADMET |
CL |
3.0 |
uL.min-1.(10^6cells)-1 |
10.6019/CHEMBL3301361 |
| None |
ADMET |
CL |
9.6 |
mL.min-1.kg-1 |
10.1124/dmd.108.020479 |
| None |
ADMET |
delta logD |
-0.84 |
None |
10.1021/jm0000564 |
| None |
ADMET |
Drug excretion |
1.5 |
% |
10.1124/dmd.112.049312 |
| None |
ADMET |
Drug excretion |
5.0 |
% |
10.1124/dmd.112.049312 |
| None |
ADMET |
eLog D |
-0.5 |
None |
10.1021/jm0200409 |
| None |
ADMET |
F |
79.0 |
% |
10.1021/jm0000564 |
| None |
ADMET |
Fraction ionised |
0.922 |
None |
10.1021/jm0200409 |
| None |
ADMET |
Fu |
0.289 |
None |
10.1021/jm0200409 |
| None |
ADMET |
Fu |
0.85 |
None |
10.1021/jm0200409 |
| None |
ADMET |
Fu |
0.85 |
None |
10.1021/jm030408h |
| None |
ADMET |
log10(%HIA +10) |
1.798 |
None |
10.1016/j.ejmech.2010.11.005 |
| None |
ADMET |
LogP app |
-6.05 |
None |
10.1016/j.bmc.2007.03.040 |
| None |
ADMET |
LogP app |
-5.52 |
None |
10.1016/j.bmc.2007.03.040 |
| None |
ADMET |
log Pe |
-8.02 |
None |
10.1021/jm300460c |
| None |
ADMET |
log Pe |
-8.02 |
None |
10.1021/ml400462j |
| None |
ADMET |
Log Pe |
-4.6 |
cm s-1 |
10.1021/jm001020e |
| None |
ADMET |
Log Pe |
-4.5 |
cm s-1 |
10.1021/jm001020e |
| None |
ADMET |
Log Pn |
-3.0 |
None |
10.1021/jm00398a028 |
| None |
ADMET |
MRT |
2.1 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
Papp |
0.18 |
ucm/s |
10.1021/jm501719e |
| None |
ADMET |
Papp |
0.2 |
10'-6 cm/s |
10.1021/acs.jmedchem.9b00720 |
| None |
ADMET |
Papp |
0.24 |
ucm/s |
10.1021/jm5015742 |
| None |
ADMET |
Papp |
0.27 |
cm s-1 |
10.1021/jm049661n |
| None |
ADMET |
Papp |
1.6 |
ucm/s |
10.1021/jm501719e |
| None |
ADMET |
Papp |
1.7 |
10'-6 cm/s |
10.1021/acs.jmedchem.9b00720 |
| None |
ADMET |
Papp |
3.0 |
10^-6 cm/s |
10.1016/j.bmc.2007.03.040 |
| None |
ADMET |
Papp |
nan |
None |
10.1021/jm049661n |
| None |
ADMET |
permeability |
0.04 |
10^-6 cm/s |
10.1016/j.ejmech.2020.113112 |
| None |
ADMET |
permeability |
0.273 |
10'-4 cm/s |
10.1021/jm901846t |
| None |
ADMET |
permeability |
2.0 |
% |
10.1016/j.bmc.2010.05.001 |
| None |
ADMET |
permeability |
55.0 |
nm/s |
10.1016/j.bmc.2010.05.001 |
| None |
ADMET |
PPB |
28.95 |
% |
10.6019/CHEMBL3301361 |
| None |
ADMET |
Ratio |
8.5 |
None |
10.1021/acs.jmedchem.9b00720 |
| None |
ADMET |
Ratio |
8.9 |
None |
10.1021/jm501719e |
| None |
ADMET |
T1/2 |
2.1 |
hr |
10.1124/dmd.108.020479 |
| None |
ADMET |
Vdss |
1.2 |
L.kg-1 |
10.1124/dmd.108.020479 |
| None |
ADMET |
Vdss |
1.3 |
L.kg-1 |
10.1021/jm0200409 |
| None |
ADMET |
Vdss |
1.3 |
L.kg-1 |
10.1021/jm030408h |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Index Value |
1.1 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Alkaline Phosphatase Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Active |
0.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Marginal |
0.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Composite Activity - Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Index Value |
0.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
GGT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1021/tx1000865 |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1021/tx900326k |
| None |
Hepatotoxicity |
Hepatotoxicity |
nan |
None |
10.1124/dmd.110.035113 |
| None |
Hepatotoxicity |
HepSE_bilirubinemia |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholecystitis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cholelithiasis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_cirrhosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_Combined Scores |
4.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_elevated liver function tests |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic failure |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatic necrosis |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatitis |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_hepatomegaly |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_jaundice |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver disease |
1.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver fatty |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
HepSE_liver function tests abnormal |
0.0 |
None |
10.1371/journal.pcbi.1002310 |
| None |
Hepatotoxicity |
LDH Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LDH Increase - Index Value |
0.3 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LDH Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
LTKB_BD DILI severity score |
5.0 |
None |
10.1016/j.drudis.2011.05.007 |
| None |
Hepatotoxicity |
SGOT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Index Value |
1.2 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGOT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Activity Score |
nan |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Index Value |
1.0 |
None |
10.2174/1570163043334794 |
| None |
Hepatotoxicity |
SGPT Increase - Number of Reports |
4.0 |
None |
10.2174/1570163043334794 |
| None |
NON-PROTEIN TARGET |
Fu |
0.95 |
None |
10.1124/dmd.108.020479 |
| None |
NON-PROTEIN TARGET |
Fu |
1.0 |
None |
10.1021/jm401963n |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (acute) |
0.0 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (animal toxicity known) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (benign tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (granulomatous hepatitis) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (mechanism) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
18.6 |
% |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (moderate) |
37.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
Hepatotoxicity (time to onset) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
NON-PROTEIN TARGET |
IC50 |
nan |
None |
10.1016/j.bmc.2010.01.068 |
| None |
No relevant target |
Daq |
7.3 |
10'-6cm2/s |
10.1021/jm901846t |
| None |
No relevant target |
LogD |
-1.44 |
None |
10.1021/jm0000564 |
| None |
No relevant target |
LogD |
-1.1 |
None |
10.1021/jm001020e |
| None |
No relevant target |
LogD |
-0.99 |
None |
10.1021/jm8005228 |
| None |
No relevant target |
LogD |
-0.91 |
None |
10.1021/jm8005228 |
| None |
No relevant target |
LogD |
-0.32 |
None |
10.1021/jf102525e |
| None |
No relevant target |
LogD |
-0.29 |
None |
10.1021/jm0100990 |
| None |
No relevant target |
LogD7.4 |
-0.95 |
None |
10.6019/CHEMBL3301361 |
| None |
No relevant target |
LogD7.4 |
-0.48 |
None |
10.1021/jm040760a |
| None |
No relevant target |
LogP |
0.27 |
None |
10.1016/j.bmc.2007.03.040 |
| None |
No relevant target |
LogP |
0.27 |
None |
10.1021/jf102525e |
| None |
No relevant target |
LogP |
0.6 |
None |
10.1021/jm021012t |
| None |
No relevant target |
LogP |
1.06 |
None |
10.1021/jm801441s |
| None |
No relevant target |
LogP |
1.28 |
None |
10.1021/jm801441s |
| None |
No relevant target |
LogP |
1.28 |
None |
10.1021/jm901846t |
| None |
No relevant target |
logPapp |
-6.05 |
None |
10.1021/jf102525e |
| None |
No relevant target |
Log Pn |
0.27 |
None |
10.1021/jm00398a028 |
| None |
No relevant target |
Papp |
0.14 |
10'-6 cm/s |
10.1016/j.bmcl.2014.07.016 |
| None |
No relevant target |
pKa |
0.88 |
None |
10.1021/jf102525e |
| None |
No relevant target |
pKa |
2.11 |
None |
10.1021/jm901846t |
| None |
No relevant target |
pKa |
8.2 |
None |
10.1021/jm0000564 |
| None |
No relevant target |
pKa |
8.31 |
None |
10.1007/s11095-013-1232-z |
| None |
No relevant target |
pKa |
8.47 |
None |
10.1016/j.ejmech.2009.06.004 |
| None |
No relevant target |
pKa |
8.47 |
None |
10.1021/jm0200409 |
| None |
No relevant target |
pKa |
8.47 |
None |
10.1021/jm030408h |
| None |
No relevant target |
pKa |
8.48 |
None |
10.1021/jm040760a |
| None |
No relevant target |
Solubility |
33.7 |
ug.mL-1 |
10.1016/j.bmcl.2015.03.016 |
| None |
No relevant target |
Solubility |
990.0 |
ug.mL-1 |
10.1016/j.bmc.2010.08.003 |
| None |
Unchecked |
Ac50 |
1.0 |
uM |
None |
| None |
Unchecked |
Ac50 |
1.122 |
uM |
None |
| None |
Unchecked |
Ac50 |
4.467 |
uM |
None |
| None |
Unchecked |
Ac50 |
28.18 |
uM |
None |
| None |
Unchecked |
Ac50 |
31.62 |
uM |
None |
| None |
Unchecked |
AC50 |
1000.0 |
nM |
None |
| None |
Unchecked |
AC50 |
1122.0 |
nM |
None |
| None |
Unchecked |
AC50 |
1130.0 |
nM |
None |
| None |
Unchecked |
AC50 |
4466.8 |
nM |
None |
| None |
Unchecked |
AC50 |
28183.8 |
nM |
None |
| None |
Unchecked |
AC50 |
31622.8 |
nM |
None |
| None |
Unchecked |
Hepatotoxicity (acute) |
21.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (association with vascular disease) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (choleostasis) |
15.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (chronic liver disease) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cirrhosis) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (comment) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (cytolytic) |
12.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (malignant tumour) |
0.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (severe hepatitis) |
2.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (steatosis) |
1.0 |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
Hepatotoxicity (successful reintroduction) |
nan |
None |
10.1016/s0399-8320(04)95062-2 |
| None |
Unchecked |
IC50 |
nan |
None |
None |
| None |
Unchecked |
Ki |
nan |
None |
None |
| None |
Unchecked |
Potency |
35481.3 |
nM |
None |
| None |
Unchecked |
Ratio |
14.0 |
None |
10.1021/jm00345a002 |
| None |
Unchecked |
Slope |
0.76 |
None |
10.1021/jm00345a002 |
| None |
Unchecked |
Slope |
1.6 |
None |
10.1021/jm00345a002 |