Molecule

Sunitinib

AlkaPlorer ID: AK322504

Synonym: None

IUPAC Name: N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide

Structure

SMILES: CCN(CC)CCN=C(O)C1=C(C)NC(/C=C2\C(O)=NC3=CC=C(F)C=C23)=C1C

InChI: InChI=1S/C22H27FN4O2/c1-5-27(6-2)10-9-24-22(29)20-13(3)19(25-14(20)4)12-17-16-11-15(23)7-8-18(16)26-21(17)28/h7-8,11-12,25H,5-6,9-10H2,1-4H3,(H,24,29)(H,26,28)/b17-12-

InChIKey: WINHZLLDWRZWRT-ATVHPVEESA-N

Reference

Gentisyl Alcohol Derivatives from the Marine-Derived Fungus <i>Penicillium terrestre</i>

PubChem CID: 5329102

CAS: 326914-13-0

LOTUS: LTS0010688

NPASS: NPC476118

Source

Species	Genus	Family	Order	Class	Phylum	Kingdom	Domain
Salvia scapiformis	Salvia	Lamiaceae	Lamiales	Magnoliopsida	Streptophyta	Viridiplantae	Eukaryota
Penicillium terrestre	Penicillium	Aspergillaceae	Eurotiales	Eurotiomycetes	Ascomycota	Fungi	Eukaryota

Properties Information

Molecule Weight: 398.48200000000014

TPSA？: 84.21

MolLogP？: 4.559240000000004

Number of H-Donors: 3

Number of H-Acceptors: 3

RingCount: 3

Activities Information

Organism	Target Name	Standard Type	Standard Value	Standard Units	doi
Bos taurus	Beta-adrenergic receptor kinase 1	IC50	130000.0	nM	10.1021/acs.jmedchem.0c01522
Chikungunya virus	Chikungunya virus	EC50	4600.0	nM	10.1021/acs.jmedchem.0c01467
Chlorocebus sabaeus	Vero	CC50	11900.0	nM	10.1021/acs.jmedchem.0c01467
Chlorocebus sabaeus	Vero	GI	10.0	%	10.1016/j.ejmech.2012.06.005
Cricetulus griseus	CHO	GI50	2030.0	nM	10.1021/acs.jmedchem.6b00200
dengue virus type 1	dengue virus type 1	EC50	200.0	nM	10.1021/acs.jmedchem.0c01467
dengue virus type 2	dengue virus type 2	EC50	200.0	nM	10.1021/acs.jmedchem.0c01467
dengue virus type 2	dengue virus type 2	EC50	510.0	nM	10.1016/j.bmcl.2020.127284
dengue virus type 2	dengue virus type 2	EC50	1350.0	nM	10.1021/acs.jmedchem.9b00136
dengue virus type 2	dengue virus type 2	EC50	1962.0	nM	10.1016/j.ejmech.2019.05.010
dengue virus type 2	dengue virus type 2	EC90	2.71	uM	10.1021/acs.jmedchem.9b00136
dengue virus type 3	dengue virus type 3	EC50	200.0	nM	10.1021/acs.jmedchem.0c01467
dengue virus type 4	dengue virus type 4	EC50	200.0	nM	10.1021/acs.jmedchem.0c01467
Ebolavirus	Ebolavirus	EC50	470.0	nM	10.1021/acs.jmedchem.0c01467
Gallus gallus	Chorioallantoic membrane	Activity	nan	None	10.1016/j.bmcl.2017.12.066
Gallus gallus	Chorioallantoic membrane	Activity	nan	None	10.1016/j.ejmech.2018.03.018
Gallus gallus	Chorioallantoic membrane	Activity	nan	None	10.1016/j.ejmech.2019.06.094
Gallus gallus	Chorioallantoic membrane	IC50	1.3	nM	10.1016/j.bmc.2014.04.049
Gallus gallus	Chorioallantoic membrane	IC50	1300.0	nM	10.1016/j.bmc.2016.11.026
Gallus gallus	Chorioallantoic membrane	IC50	1300.0	nM	10.1016/j.bmcl.2018.07.039
Gallus gallus	Chorioallantoic membrane	IC50	1300.0	nM	10.1021/ml4004793
Gallus gallus	Myosin light chain kinase, smooth muscle	Kd	23.0	nM	10.1038/nbt1358
Gallus gallus	Tyrosine-protein kinase SRC	IC50	555.0	nM	10.1021/jm4004076
Hepacivirus hominis	Hepatitis C virus	EC50	1200.0	nM	10.1021/acs.jmedchem.0c01467
Homo sapiens	143B	Activity	0.909	None	10.1073/pnas.0707498104
Homo sapiens	26S protease regulatory subunit 6B	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	3-phosphoinositide dependent protein kinase-1	Kd	3500.0	nM	10.1038/nbt1358
Homo sapiens	3-phosphoinositide dependent protein kinase-1	Kd	3500.0	nM	10.1038/nbt.1990
Homo sapiens	3-phosphoinositide dependent protein kinase-1	Kd	3500.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	3-phosphoinositide dependent protein kinase-1	Thermal melting change	2.9	degrees C	10.1073/pnas.0708800104
Homo sapiens	5637	Activity	1.184	None	10.1073/pnas.0707498104
Homo sapiens	639-V	Activity	1.049	None	10.1073/pnas.0707498104
Homo sapiens	647-V	Activity	0.952	None	10.1073/pnas.0707498104
Homo sapiens	697	IC50	614.25	nM	10.6019/CHEMBL1201861
Homo sapiens	769-P	Activity	1.102	None	10.1073/pnas.0707498104
Homo sapiens	8305C	Activity	0.951	None	10.1073/pnas.0707498104
Homo sapiens	8505C	Activity	0.905	None	10.1073/pnas.0707498104
Homo sapiens	8-MG-BA	IC50	6515.07	nM	10.6019/CHEMBL1201861
Homo sapiens	A101D	IC50	2783.04	nM	10.6019/CHEMBL1201861
Homo sapiens	A2058	Activity	1.118	None	10.1073/pnas.0707498104
Homo sapiens	A253 cell line	IC50	275450.52	nM	10.6019/CHEMBL1201861
Homo sapiens	A2780	Activity	1.001	None	10.1073/pnas.0707498104
Homo sapiens	A-375	Activity	1.051	None	10.1073/pnas.0707498104
Homo sapiens	A-375	IC50	5400.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	A-375	IC50	11580.0	nM	10.1016/j.bmcl.2012.03.061
Homo sapiens	A388	IC50	28007.35	nM	10.6019/CHEMBL1201861
Homo sapiens	A3-KAW	IC50	1625.46	nM	10.6019/CHEMBL1201861
Homo sapiens	A-427	Activity	0.842	None	10.1073/pnas.0707498104
Homo sapiens	A-431	Activity	0.986	None	10.1073/pnas.0707498104
Homo sapiens	A-431	IC50	nan	None	10.1016/j.bmc.2014.04.049
Homo sapiens	A-431	IC50	nan	None	10.1016/j.bmc.2015.03.061
Homo sapiens	A-431	IC50	nan	None	10.1016/j.bmc.2016.11.026
Homo sapiens	A-431	IC50	nan	None	10.1016/j.bmcl.2018.07.039
Homo sapiens	A498	IC50	1200.0	nM	10.1016/j.bmcl.2022.129041
Homo sapiens	A498	IC50	1250.0	nM	10.1016/j.ejmech.2020.112752
Homo sapiens	A498	IC50	4300.0	nM	10.1016/j.bmcl.2013.02.061
Homo sapiens	A498	IC50	7981.0	nM	10.1021/acsmedchemlett.7b00192
Homo sapiens	A498	IC50	719937.93	nM	10.6019/CHEMBL1201861
Homo sapiens	A4-Fuk	IC50	1341.41	nM	10.6019/CHEMBL1201861
Homo sapiens	A549	Activity	0.812	None	10.1073/pnas.0707498104
Homo sapiens	A549	Activity	2.4	%	10.1016/j.ejmech.2018.11.023
Homo sapiens	A549	Activity	15.81	%	10.1039/C1MD00105A
Homo sapiens	A549	Activity	16.0	%	10.1016/j.ejmech.2018.11.023
Homo sapiens	A549	Activity	35.0	%	10.1016/j.ejmech.2018.11.023
Homo sapiens	A549	Activity	37.4	%	10.1016/j.ejmech.2011.07.045
Homo sapiens	A549	Activity	38.0	%	10.1016/j.ejmech.2018.11.023
Homo sapiens	A549	Activity	45.0	%	10.1016/j.ejmech.2018.11.023
Homo sapiens	A549	Activity	47.0	%	10.1016/j.ejmech.2018.11.023
Homo sapiens	A549	Activity	56.0	%	10.1016/j.ejmech.2019.03.012
Homo sapiens	A549	Activity	66.0	%	10.1016/j.ejmech.2019.03.012
Homo sapiens	A549	Activity	102.5	%	10.1016/j.ejmech.2011.07.045
Homo sapiens	A549	Activity	135.0	%	10.1016/j.ejmech.2019.03.012
Homo sapiens	A549	IC50	2440.0	nM	10.1016/j.bmcl.2013.03.099
Homo sapiens	A549	IC50	2440.0	nM	10.1016/j.bmcl.2016.08.060
Homo sapiens	A549	IC50	3060.0	nM	10.1016/j.ejmech.2020.112359
Homo sapiens	A549	IC50	5730.0	nM	10.1039/d2md00442a
Homo sapiens	A549	IC50	6610.0	nM	10.1007/s00044-012-0170-3
Homo sapiens	A549	IC50	6610.0	nM	10.1016/j.bmcl.2011.03.031
Homo sapiens	A549	IC50	7900.0	nM	10.1016/j.ejmech.2020.113102
Homo sapiens	A549	IC50	7930.0	nM	10.1016/j.bmcl.2015.05.017
Homo sapiens	A549	IC50	9100.0	nM	10.1016/j.bmcl.2016.02.063
Homo sapiens	A549	IC50	10140.0	nM	10.1016/j.ejmech.2020.112359
Homo sapiens	A549	IC50	11000.0	nM	10.1016/j.ejmech.2018.11.023
Homo sapiens	A549	IC50	11000.0	nM	10.1016/j.ejmech.2019.03.012
Homo sapiens	A549	IC50	12350.0	nM	10.1016/j.bmcl.2012.03.061
Homo sapiens	A549	IC50	14400.0	nM	10.1016/j.bmcl.2016.06.077
Homo sapiens	A549	IC50	18500.0	nM	10.1016/j.ejmech.2011.10.009
Homo sapiens	A549	IC50	18580.0	nM	10.1039/C1MD00105A
Homo sapiens	A549	IC50	22100.0	nM	10.1016/j.ejmech.2019.111719
Homo sapiens	A549	IC50	nan	None	10.1016/j.ejmech.2019.06.054
Homo sapiens	A704	IC50	17990.43	nM	10.6019/CHEMBL1201861
Homo sapiens	ABC-1	Activity	1.025	None	10.1073/pnas.0707498104
Homo sapiens	Acetylcholinesterase	IC50	5870.0	nM	10.1021/acs.jmedchem.6b00078
Homo sapiens	ACHN	Activity	0.811	None	10.1073/pnas.0707498104
Homo sapiens	ACHN	IC50	2500.0	nM	10.1021/np300573m
Homo sapiens	ACHN	IC50	5700.0	nM	10.1016/j.bmcl.2013.02.061
Homo sapiens	ACN	IC50	58168.68	nM	10.6019/CHEMBL1201861
Homo sapiens	Actin-related protein 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Actin-related protein 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Activin receptor type-1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Activin receptor type-1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Activin receptor type-1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Activin receptor type-1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Activin receptor type-1B	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Activin receptor type-1B	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Activin receptor type-1B	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Activin receptor type-1B	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Activin receptor type-2A	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Activin receptor type-2A	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Activin receptor type-2A	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Activin receptor type-2B	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Activin receptor type-2B	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Activin receptor type-2B	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Activin receptor type-2B	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Acyl-CoA dehydrogenase family member 11	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Adaptor-associated kinase	IC50	45.0	nM	10.1021/acs.jmedchem.0c01467
Homo sapiens	Adaptor-associated kinase	IC50	47.4	nM	10.1021/acs.jmedchem.9b00136
Homo sapiens	Adaptor-associated kinase	Kd	11.0	nM	10.1021/acs.jmedchem.1c00302
Homo sapiens	Adaptor-associated kinase	Kd	11.0	nM	10.1021/acs.jmedchem.9b00136
Homo sapiens	Adaptor-associated kinase	Kd	11.0	nM	10.1038/nbt1358
Homo sapiens	Adaptor-associated kinase	Kd	11.0	nM	10.1038/nbt.1990
Homo sapiens	Adaptor-associated kinase	Kd	11.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Adaptor-associated kinase	Kd	35.0	nM	10.1021/acs.jmedchem.0c01467
Homo sapiens	Adaptor-associated kinase	Kd	130.0	nM	10.1038/nbt1068
Homo sapiens	Adaptor-associated kinase	Kd	363.0	nM	10.1126/science.aan4368
Homo sapiens	Adenine phosphoribosyltransferase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Adenosine A1 receptor	AC50	6400.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Adenosine A2a receptor	AC50	5300.1	nM	10.1038/s41467-023-40064-9
Homo sapiens	Adenosine A3 receptor	AC50	8400.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Adenosine kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Adenylate kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	ADP/ATP translocase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	ADP/ATP translocase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	AGS	Activity	1.175	None	10.1073/pnas.0707498104
Homo sapiens	ALK tyrosine kinase receptor	IC50	54.64	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	ALK tyrosine kinase receptor	IC50	2300.0	nM	10.1016/j.bmc.2010.01.011
Homo sapiens	ALK tyrosine kinase receptor	Kd	170.0	nM	10.1038/nbt1358
Homo sapiens	ALK tyrosine kinase receptor	Kd	170.0	nM	10.1038/nbt.1990
Homo sapiens	ALK tyrosine kinase receptor	Kd	170.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	ALK tyrosine kinase receptor	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	ALL-PO	IC50	79.89	nM	10.6019/CHEMBL1201861
Homo sapiens	Alpha-1a adrenergic receptor	AC50	185.3	nM	10.1038/s41467-023-40064-9
Homo sapiens	Alpha-1a adrenergic receptor	AC50	420.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Alpha-1a adrenergic receptor	AC50	920.9	nM	10.1038/s41467-023-40064-9
Homo sapiens	Alpha-1a adrenergic receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Alpha-2a adrenergic receptor	AC50	9472.6	nM	10.1038/s41467-023-40064-9
Homo sapiens	Alpha-2a adrenergic receptor	AC50	23999.9	nM	10.1038/s41467-023-40064-9
Homo sapiens	Alpha-2a adrenergic receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Alpha-2b adrenergic receptor	AC50	4374.9	nM	10.1038/s41467-023-40064-9
Homo sapiens	Alpha-2c adrenergic receptor	AC50	1766.3	nM	10.1038/s41467-023-40064-9
Homo sapiens	AM-38	IC50	197528.13	nM	10.6019/CHEMBL1201861
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	IC50	158.0	nM	10.1016/j.ejmech.2020.112316
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Inhibition	50.0	%	10.1016/j.ejmech.2020.112316
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	19.0	nM	10.1038/nbt1358
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	19.0	nM	10.1038/nbt.1990
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	19.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	52.0	nM	10.1038/nbt1068
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	52.0	nM	10.1073/pnas.0707498104
Homo sapiens	AMP-activated protein kinase, alpha-1 subunit	Kd	1079.0	nM	10.1126/science.aan4368
Homo sapiens	AMP-activated protein kinase, alpha-2 subunit	IC50	61.7	nM	10.1016/j.ejmech.2020.112316
Homo sapiens	AMP-activated protein kinase, alpha-2 subunit	Inhibition	46.0	%	10.1016/j.ejmech.2020.112316
Homo sapiens	AMP-activated protein kinase, alpha-2 subunit	Kd	89.0	nM	10.1038/nbt1358
Homo sapiens	AMP-activated protein kinase, alpha-2 subunit	Kd	89.0	nM	10.1038/nbt.1990
Homo sapiens	AMP-activated protein kinase, alpha-2 subunit	Kd	89.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	AMP-activated protein kinase, alpha-2 subunit	Thermal melting change	7.4	degrees C	10.1073/pnas.0708800104
Homo sapiens	AMP-activated protein kinase, gamma-1 subunit	Kd	1140.0	nM	10.1126/science.aan4368
Homo sapiens	AMP-activated protein kinase, gamma-2 subunit	Kd	1734.0	nM	10.1126/science.aan4368
Homo sapiens	Ankyrin repeat and protein kinase domain-containing protein 1	Kd	310.0	nM	10.1038/nbt1358
Homo sapiens	Ankyrin repeat and protein kinase domain-containing protein 1	Kd	310.0	nM	10.1038/nbt.1990
Homo sapiens	Ankyrin repeat and protein kinase domain-containing protein 1	Kd	310.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	ARH-77	IC50	7535.97	nM	10.6019/CHEMBL1201861
Homo sapiens	ASPC1	Activity	1.046	None	10.1073/pnas.0707498104
Homo sapiens	ATN-1	IC50	3671.14	nM	10.6019/CHEMBL1201861
Homo sapiens	ATP-binding cassette sub-family G member 2	IC50	3000.0	nM	10.1016/j.ejmech.2022.114346
Homo sapiens	ATP-dependent RNA helicase DDX1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	ATP-dependent RNA helicase DDX3X	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	ATP-dependent RNA helicase DDX42	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	ATP-dependent RNA helicase DHX30	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	AU565	Activity	1.244	None	10.1073/pnas.0707498104
Homo sapiens	BB30-HNC	IC50	2223.75	nM	10.6019/CHEMBL1201861
Homo sapiens	BB49-HNC	IC50	3705.08	nM	10.6019/CHEMBL1201861
Homo sapiens	BB65-RCC	IC50	18416.21	nM	10.6019/CHEMBL1201861
Homo sapiens	BC-3	IC50	12465.08	nM	10.6019/CHEMBL1201861
Homo sapiens	BCPAP	Activity	0.814	None	10.1073/pnas.0707498104
Homo sapiens	Bcr/Abl fusion protein	EC50	1000.0	nM	10.1021/acs.jmedchem.6b00087
Homo sapiens	Bcr/Abl fusion protein	EC50	nan	None	10.1021/acs.jmedchem.6b00087
Homo sapiens	BE-13	IC50	3231.11	nM	10.6019/CHEMBL1201861
Homo sapiens	BEAS-2B	IC50	6090.0	nM	10.1039/d2md00442a
Homo sapiens	Becker	IC50	645339.8	nM	10.6019/CHEMBL1201861
Homo sapiens	BEN	Activity	0.986	None	10.1073/pnas.0707498104
Homo sapiens	Beta-1 adrenergic receptor	AC50	6000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Beta-2 adrenergic receptor	AC50	8000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	BFTC-905	Activity	0.93	None	10.1073/pnas.0707498104
Homo sapiens	BFTC-909	Activity	1.131	None	10.1073/pnas.0707498104
Homo sapiens	BHT-101	Activity	1.152	None	10.1073/pnas.0707498104
Homo sapiens	Bile acid receptor FXR	AC50	3300.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Bile acid receptor FXR	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Bile salt export pump	AC50	34000.1	nM	10.1038/s41467-023-40064-9
Homo sapiens	Bile salt export pump	IC50	45810.0	nM	10.1124/dmd.112.047068
Homo sapiens	BL-41	IC50	2912.22	nM	10.6019/CHEMBL1201861
Homo sapiens	BL-70	IC50	1118.46	nM	10.6019/CHEMBL1201861
Homo sapiens	BMP-2-inducible protein kinase	Kd	5.5	nM	10.1038/nbt1358
Homo sapiens	BMP-2-inducible protein kinase	Kd	5.5	nM	10.1038/nbt.1990
Homo sapiens	BMP-2-inducible protein kinase	Kd	5.5	nM	10.1182/blood-2009-05-222034
Homo sapiens	BMP-2-inducible protein kinase	Kd	38.0	nM	10.1038/nbt1068
Homo sapiens	BMP-2-inducible protein kinase	Kd	38.0	nM	10.1073/pnas.0707498104
Homo sapiens	BMP-2-inducible protein kinase	Kd	87.0	nM	10.1126/science.aan4368
Homo sapiens	BOKU	IC50	171831.27	nM	10.6019/CHEMBL1201861
Homo sapiens	Bone morphogenetic protein receptor type-1A	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Bone morphogenetic protein receptor type-1A	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Bone morphogenetic protein receptor type-1A	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Bone morphogenetic protein receptor type-1A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Bone morphogenetic protein receptor type-1B	Kd	2400.0	nM	10.1038/nbt.1990
Homo sapiens	Bone morphogenetic protein receptor type-1B	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Bone morphogenetic protein receptor type-1B	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Bone morphogenetic protein receptor type-2	Kd	570.0	nM	10.1021/acsmedchemlett.3c00127
Homo sapiens	Bone morphogenetic protein receptor type-2	Kd	570.0	nM	10.1038/nbt1358
Homo sapiens	Bone morphogenetic protein receptor type-2	Kd	570.0	nM	10.1038/nbt.1990
Homo sapiens	Bone morphogenetic protein receptor type-2	Kd	570.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Bone morphogenetic protein receptor type-2	Kd	2608.0	nM	10.1126/science.aan4368
Homo sapiens	Bradykinin B2 receptor	AC50	2500.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Brain glycogen phosphorylase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Breakpoint cluster region protein	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Bromodomain-containing protein 7	Kd	11000.0	nM	10.1021/acs.jmedchem.9b01980
Homo sapiens	Bromodomain-containing protein 9	Kd	17000.0	nM	10.1021/acs.jmedchem.9b01980
Homo sapiens	BR serine/threonine-protein kinase 1	Kd	3500.0	nM	10.1038/nbt1358
Homo sapiens	BR serine/threonine-protein kinase 1	Kd	3500.0	nM	10.1038/nbt.1990
Homo sapiens	BR serine/threonine-protein kinase 1	Kd	3500.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	BR serine/threonine-protein kinase 2	Kd	1100.0	nM	10.1038/nbt1358
Homo sapiens	BR serine/threonine-protein kinase 2	Kd	1100.0	nM	10.1038/nbt.1990
Homo sapiens	BR serine/threonine-protein kinase 2	Kd	1100.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	BT-474	Activity	1.31	None	10.1073/pnas.0707498104
Homo sapiens	BT-474	EC50	900.0	nM	10.1021/acsmedchemlett.8b00596
Homo sapiens	BT-474	IC50	653346.75	nM	10.6019/CHEMBL1201861
Homo sapiens	BT-549	Activity	1.154	None	10.1073/pnas.0707498104
Homo sapiens	BT-549	IC50	2200.0	nM	10.1016/j.bmcl.2019.126710
Homo sapiens	BT-549	IC50	3500.0	nM	10.1016/j.bmcl.2019.126710
Homo sapiens	BT-549	IC50	15500.0	nM	10.1016/j.bmcl.2016.06.077
Homo sapiens	BV-173	IC50	2336.6	nM	10.6019/CHEMBL1201861
Homo sapiens	BXPC-3	Activity	0.836	None	10.1073/pnas.0707498104
Homo sapiens	BXPC-3	EC50	2500.0	nM	10.1021/acsmedchemlett.8b00596
Homo sapiens	BXPC-3	IC50	3630.0	nM	10.1016/j.bmcl.2013.08.037
Homo sapiens	C2BBe1	IC50	208215.17	nM	10.6019/CHEMBL1201861
Homo sapiens	C32	Activity	0.973	None	10.1073/pnas.0707498104
Homo sapiens	C-33-A	Activity	1.079	None	10.1073/pnas.0707498104
Homo sapiens	C8166	IC50	968734.91	nM	10.6019/CHEMBL1201861
Homo sapiens	CA46	IC50	7580.12	nM	10.6019/CHEMBL1201861
Homo sapiens	Caco-2	Activity	1.029	None	10.1073/pnas.0707498104
Homo sapiens	CAKI-1	Activity	0.876	None	10.1073/pnas.0707498104
Homo sapiens	CAKI-1	GI50	630.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	CAKI-1	IC50	4930.0	nM	10.1016/j.ejmech.2020.112752
Homo sapiens	CAKI-1	TGI	85.0	%	10.1016/j.bmcl.2017.06.071
Homo sapiens	CAL-120	Activity	1.134	None	10.1073/pnas.0707498104
Homo sapiens	CAL-12T	Activity	1.004	None	10.1073/pnas.0707498104
Homo sapiens	CAL-148	Activity	0.842	None	10.1073/pnas.0707498104
Homo sapiens	CAL-148	IC50	1861288.0	nM	10.6019/CHEMBL1201861
Homo sapiens	CAL-51	Activity	1.061	None	10.1073/pnas.0707498104
Homo sapiens	CAL-54	Activity	0.94	None	10.1073/pnas.0707498104
Homo sapiens	CAL-62	Activity	0.971	None	10.1073/pnas.0707498104
Homo sapiens	CAL-85-1	Activity	0.902	None	10.1073/pnas.0707498104
Homo sapiens	Calu-1	Activity	0.936	None	10.1073/pnas.0707498104
Homo sapiens	Calu-3	Activity	0.944	None	10.1073/pnas.0707498104
Homo sapiens	Calu-6	IC50	322909.47	nM	10.6019/CHEMBL1201861
Homo sapiens	Calu-6	TGI	nan	None	10.1016/j.bmc.2011.12.058
Homo sapiens	CaM kinase I alpha	Kd	970.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase I alpha	Kd	970.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase I alpha	Kd	970.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	CaM kinase I alpha	Kd	2000.0	nM	10.1038/nbt1068
Homo sapiens	CaM kinase I delta	Kd	510.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase I delta	Kd	510.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase I delta	Kd	510.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	CaM kinase I delta	Kd	1100.0	nM	10.1038/nbt1068
Homo sapiens	CaM kinase I delta	Thermal melting change	2.4	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM kinase I gamma	Kd	440.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase I gamma	Kd	440.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase I gamma	Kd	990.0	nM	10.1038/nbt1068
Homo sapiens	CaM kinase I gamma	Thermal melting change	7.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM kinase II alpha	Kd	80.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase II alpha	Kd	80.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase II alpha	Kd	80.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	CaM kinase II alpha	Kd	370.0	nM	10.1038/nbt1068
Homo sapiens	CaM kinase II alpha	Kd	370.0	nM	10.1073/pnas.0707498104
Homo sapiens	CaM kinase II alpha	Thermal melting change	5.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM kinase II beta	Kd	1400.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase II beta	Kd	1400.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase II beta	Kd	1400.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	CaM kinase II beta	Kd	3200.0	nM	10.1038/nbt1068
Homo sapiens	CaM kinase II beta	Thermal melting change	2.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM kinase II delta	Kd	420.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase II delta	Kd	420.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase II delta	Kd	420.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	CaM kinase II delta	Kd	1100.0	nM	10.1038/nbt1068
Homo sapiens	CaM kinase II delta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	CaM kinase II delta	Thermal melting change	2.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM kinase II gamma	Kd	440.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	CaM kinase II gamma	Kd	690.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase II gamma	Kd	690.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase II gamma	Kd	690.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	CaM kinase II gamma	Kd	760.0	nM	10.1038/nbt1068
Homo sapiens	CaM kinase II gamma	Kd	760.0	nM	10.1073/pnas.0707498104
Homo sapiens	CaM kinase II gamma	Kd	898.0	nM	10.1126/science.aan4368
Homo sapiens	CaM kinase II gamma	Thermal melting change	5.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM kinase IV	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	CaM kinase IV	Kd	890.0	nM	10.1038/nbt1358
Homo sapiens	CaM kinase IV	Kd	890.0	nM	10.1038/nbt.1990
Homo sapiens	CaM kinase IV	Kd	890.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	CaM kinase IV	Kd	2970.0	nM	10.1126/science.aan4368
Homo sapiens	CaM kinase IV	Thermal melting change	6.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	CaM-kinase kinase alpha	Kd	420.0	nM	10.1038/nbt1358
Homo sapiens	CaM-kinase kinase alpha	Kd	420.0	nM	10.1038/nbt.1990
Homo sapiens	CaM-kinase kinase alpha	Kd	420.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	CaM-kinase kinase alpha	Kd	900.0	nM	10.1038/nbt1068
Homo sapiens	CaM-kinase kinase beta	Kd	1500.0	nM	10.1038/nbt1358
Homo sapiens	CaM-kinase kinase beta	Kd	1500.0	nM	10.1038/nbt.1990
Homo sapiens	CaM-kinase kinase beta	Kd	1500.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	CaM-kinase kinase beta	Kd	5800.0	nM	10.1038/nbt1068
Homo sapiens	CaM-kinase kinase beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	CaM-kinase kinase beta	Thermal melting change	6.8	degrees C	10.1073/pnas.0708800104
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	cAMP-dependent protein kinase alpha-catalytic subunit	Thermal melting change	9.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	cAMP-dependent protein kinase beta-1 catalytic subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	cAMP-dependent protein kinase, gamma catalytic subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	cAMP-dependent protein kinase type II-alpha regulatory subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cannabinoid CB1 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	CAPAN-1	Activity	1.238	None	10.1073/pnas.0707498104
Homo sapiens	Capan-2	Activity	1.242	None	10.1073/pnas.0707498104
Homo sapiens	CaR-1	Activity	0.974	None	10.1073/pnas.0707498104
Homo sapiens	CAS-1	IC50	322440.62	nM	10.6019/CHEMBL1201861
Homo sapiens	Casein kinase I alpha	IC50	1.0	nM	10.1038/nchembio.117
Homo sapiens	Casein kinase I alpha	Kd	99.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I alpha	Kd	550.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Casein kinase I alpha	Kd	7339.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I delta	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Casein kinase I delta	Kd	15.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I delta	Kd	15.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I delta	Kd	15.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Casein kinase I delta	Kd	869.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I epsilon	Kd	13.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I epsilon	Kd	13.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I epsilon	Kd	13.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Casein kinase I epsilon	Kd	848.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I epsilon	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Casein kinase I gamma 1	Kd	930.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I gamma 1	Kd	930.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I gamma 1	Kd	930.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Casein kinase I gamma 1	Kd	3374.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I gamma 1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Casein kinase I gamma 1	Thermal melting change	4.5	degrees C	10.1073/pnas.0708800104
Homo sapiens	Casein kinase I gamma 2	Kd	110.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I gamma 2	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I gamma 2	Kd	110.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Casein kinase I gamma 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I gamma 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Casein kinase I gamma 2	Thermal melting change	4.9	degrees C	10.1073/pnas.0708800104
Homo sapiens	Casein kinase II alpha	Kd	81.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase II alpha	Kd	81.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Casein kinase II alpha	Kd	900.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase II alpha (prime)	Kd	160.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase II alpha (prime)	Kd	370.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase II alpha (prime)	Kd	370.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Casein kinase II alpha (prime)	Kd	3201.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I isoform alpha-like	Kd	550.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I isoform alpha-like	Kd	550.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I isoform gamma-3	Kd	240.0	nM	10.1038/nbt1358
Homo sapiens	Casein kinase I isoform gamma-3	Kd	240.0	nM	10.1038/nbt.1990
Homo sapiens	Casein kinase I isoform gamma-3	Kd	240.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Casein kinase I isoform gamma-3	Kd	2946.0	nM	10.1126/science.aan4368
Homo sapiens	Casein kinase I isoform gamma-3	Thermal melting change	4.9	degrees C	10.1073/pnas.0708800104
Homo sapiens	CCF-STTG1	Activity	0.929	None	10.1073/pnas.0707498104
Homo sapiens	CCRF-CEM	IC50	14416.94	nM	10.6019/CHEMBL1201861
Homo sapiens	Cell division cycle 2-like protein kinase 6	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cell division cycle 2-like protein kinase 6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cell division cycle 2-like protein kinase 6	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Cell division cycle 7-related protein kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cell division protein kinase 8	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cell division protein kinase 8	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cell division protein kinase 8	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	CESS	IC50	7104.38	nM	10.6019/CHEMBL1201861
Homo sapiens	CFPAC-1	Activity	0.868	None	10.1073/pnas.0707498104
Homo sapiens	cGMP-dependent protein kinase 1 beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	cGMP-dependent protein kinase 1 beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	cGMP-dependent protein kinase 1 beta	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	cGMP-dependent protein kinase 1 beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	cGMP-dependent protein kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	cGMP-dependent protein kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	cGMP-dependent protein kinase 2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	CGTH-W-1	IC50	30.94	nM	10.6019/CHEMBL1201861
Homo sapiens	ChaGo-K-1	Activity	0.771	None	10.1073/pnas.0707498104
Homo sapiens	Chaperone activity of bc1 complex-like, mitochondrial	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Chaperone activity of bc1 complex-like, mitochondrial	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Chaperone activity of bc1 complex-like, mitochondrial	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Chaperone activity of bc1 complex-like, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cholecystokinin A receptor	AC50	6699.9	nM	10.1038/s41467-023-40064-9
Homo sapiens	Cholecystokinin B receptor	AC50	10000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Choline-phosphate cytidylyltransferase A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	CHP-126	IC50	591933.32	nM	10.6019/CHEMBL1201861
Homo sapiens	Chromodomain-helicase-DNA-binding protein 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Citron Rho-interacting kinase	Kd	3900.0	nM	10.1038/nbt1358
Homo sapiens	Citron Rho-interacting kinase	Kd	3900.0	nM	10.1038/nbt.1990
Homo sapiens	Citron Rho-interacting kinase	Kd	3900.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Citron Rho-interacting kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	c-Jun N-terminal kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	c-Jun N-terminal kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	c-Jun N-terminal kinase 1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	c-Jun N-terminal kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	c-Jun N-terminal kinase 1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	c-Jun N-terminal kinase 2	Kd	2400.0	nM	10.1038/nbt.1990
Homo sapiens	c-Jun N-terminal kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	c-Jun N-terminal kinase 2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	c-Jun N-terminal kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	c-Jun N-terminal kinase 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	c-Jun N-terminal kinase 3	Kd	4300.0	nM	10.1038/nbt.1990
Homo sapiens	c-Jun N-terminal kinase 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	c-Jun N-terminal kinase 3	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	c-Jun N-terminal kinase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	c-Jun N-terminal kinase 3	Kd	nan	None	10.1038/nbt1068
Homo sapiens	CMK	IC50	1955.17	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO 205	Activity	1.318	None	10.1073/pnas.0707498104
Homo sapiens	COLO 205	IC50	4000.0	nM	10.1016/j.bmc.2010.05.021
Homo sapiens	COLO 205	IC50	8000.0	nM	10.1016/j.bmcl.2017.07.029
Homo sapiens	COLO 320	Activity	1.157	None	10.1073/pnas.0707498104
Homo sapiens	COLO 320DM	AC50	1.464	None	10.1073/pnas.0707498104
Homo sapiens	COLO-320-HSR	IC50	12156.49	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-668	IC50	30791.97	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-684	IC50	90456.22	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-800	IC50	606515.33	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-824	IC50	273365.03	nM	10.6019/CHEMBL1201861
Homo sapiens	COLO-829	IC50	359086.75	nM	10.6019/CHEMBL1201861
Homo sapiens	COR-L23	Activity	0.874	None	10.1073/pnas.0707498104
Homo sapiens	COR-L279	IC50	9390.9	nM	10.6019/CHEMBL1201861
Homo sapiens	COR-L88	IC50	16001.2	nM	10.6019/CHEMBL1201861
Homo sapiens	CP66-MEL	IC50	531468.01	nM	10.6019/CHEMBL1201861
Homo sapiens	CP67-MEL	IC50	132542.98	nM	10.6019/CHEMBL1201861
Homo sapiens	CPC-N	IC50	8291.99	nM	10.6019/CHEMBL1201861
Homo sapiens	CTB-1	IC50	13729.43	nM	10.6019/CHEMBL1201861
Homo sapiens	CTV-1	IC50	1727.51	nM	10.6019/CHEMBL1201861
Homo sapiens	CW-2	IC50	383859.65	nM	10.6019/CHEMBL1201861
Homo sapiens	Cyclin-dependent kinase 1	Inhibition	nan	%	10.1021/acs.jmedchem.5b01582
Homo sapiens	Cyclin-dependent kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 10	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 12	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 13	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 13	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 2	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Cyclin-dependent kinase 2	Kd	10000.0	nM	10.1021/jm200222m
Homo sapiens	Cyclin-dependent kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Cyclin-dependent kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Cyclin-dependent kinase 2	Thermal melting change	-0.8	degrees C	10.1073/pnas.0708800104
Homo sapiens	Cyclin-dependent kinase 3	Kd	1024.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 3	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Cyclin-dependent kinase 4	Kd	2000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 4	Kd	6200.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 5	Kd	6900.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 5	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Cyclin-dependent kinase 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 5	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Cyclin-dependent kinase 6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 6	Thermal melting change	2.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	Cyclin-dependent kinase 7	Kd	330.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 7	Kd	330.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 7	Kd	330.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Cyclin-dependent kinase 7	Kd	1202.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase 9	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Cyclin-dependent kinase 9	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase 9	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Cyclin-dependent kinase 9	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclin-dependent kinase-like 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase-like 1	Thermal melting change	0.5	degrees C	10.1073/pnas.0708800104
Homo sapiens	Cyclin-dependent kinase-like 2	Kd	1100.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase-like 2	Kd	1100.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Cyclin-dependent kinase-like 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase-like 3	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Cyclin-dependent kinase-like 5	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Cyclin-dependent kinase-like 5	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Cyclin-dependent kinase-like 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cyclooxygenase-2	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Cysteine--tRNA ligase, cytoplasmic	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cytochrome c1, heme protein, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Cytochrome P450 3A4	Activity	nan	None	None
Homo sapiens	D-247MG	IC50	103799.28	nM	10.6019/CHEMBL1201861
Homo sapiens	D-263MG	IC50	200070.54	nM	10.6019/CHEMBL1201861
Homo sapiens	D283 Med	IC50	16848.86	nM	10.6019/CHEMBL1201861
Homo sapiens	D-336MG	IC50	292957.93	nM	10.6019/CHEMBL1201861
Homo sapiens	D-502MG	IC50	984380.98	nM	10.6019/CHEMBL1201861
Homo sapiens	DAN-G	Activity	1.036	None	10.1073/pnas.0707498104
Homo sapiens	Daoy	Activity	1.132	None	10.1073/pnas.0707498104
Homo sapiens	Daudi	IC50	8235.46	nM	10.6019/CHEMBL1201861
Homo sapiens	DB	IC50	311668.15	nM	10.6019/CHEMBL1201861
Homo sapiens	dCTP pyrophosphatase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Death-associated protein kinase 1	Kd	120.0	nM	10.1038/nbt1358
Homo sapiens	Death-associated protein kinase 1	Kd	120.0	nM	10.1038/nbt.1990
Homo sapiens	Death-associated protein kinase 1	Kd	120.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Death-associated protein kinase 2	Kd	150.0	nM	10.1038/nbt1358
Homo sapiens	Death-associated protein kinase 2	Kd	150.0	nM	10.1038/nbt.1990
Homo sapiens	Death-associated protein kinase 2	Kd	150.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Death-associated protein kinase 2	Kd	470.0	nM	10.1038/nbt1068
Homo sapiens	Death-associated protein kinase 2	Kd	470.0	nM	10.1073/pnas.0707498104
Homo sapiens	Death-associated protein kinase 3	Kd	22.0	nM	10.1038/nbt1358
Homo sapiens	Death-associated protein kinase 3	Kd	22.0	nM	10.1038/nbt.1990
Homo sapiens	Death-associated protein kinase 3	Kd	22.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Death-associated protein kinase 3	Kd	100.0	nM	10.1038/nbt1358
Homo sapiens	Death-associated protein kinase 3	Kd	300.0	nM	10.1038/nbt1068
Homo sapiens	Death-associated protein kinase 3	Kd	300.0	nM	10.1073/pnas.0707498104
Homo sapiens	Death-associated protein kinase 3	Thermal melting change	0.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	DEL	IC50	2084.82	nM	10.6019/CHEMBL1201861
Homo sapiens	Delta(24)-sterol reductase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Delta opioid receptor	AC50	1700.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Deoxycytidine kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	DG-75	IC50	6430.69	nM	10.6019/CHEMBL1201861
Homo sapiens	Discoidin domain-containing receptor 2	Kd	2900.0	nM	10.1038/nbt.1990
Homo sapiens	Discoidin domain-containing receptor 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Discoidin domain-containing receptor 2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Discoidin domain-containing receptor 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	DJM-1	IC50	91562.43	nM	10.6019/CHEMBL1201861
Homo sapiens	DLD-1	Activity	1.088	None	10.1073/pnas.0707498104
Homo sapiens	DLD-1	Activity	52.7	%	10.1016/j.ejmech.2011.07.045
Homo sapiens	DLD-1	Activity	92.9	%	10.1016/j.ejmech.2011.07.045
Homo sapiens	DMS-114	IC50	77138.15	nM	10.6019/CHEMBL1201861
Homo sapiens	DMS-153	IC50	255682.13	nM	10.6019/CHEMBL1201861
Homo sapiens	DMS-79	IC50	288357.2	nM	10.6019/CHEMBL1201861
Homo sapiens	DNA-dependent protein kinase	IC50	50000.0	nM	10.1038/nchembio.117
Homo sapiens	DnaJ homolog subfamily A member 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	DNA polymerase kappa	Potency	13371.4	nM	None
Homo sapiens	DNA replication licensing factor MCM4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	DNA topoisomerase II alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	DNA topoisomerase II beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	DOHH-2	IC50	2334.31	nM	10.6019/CHEMBL1201861
Homo sapiens	Dopamine D1 receptor	AC50	4717.8	nM	10.1038/s41467-023-40064-9
Homo sapiens	Dopamine D1 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Dopamine D2 receptor	AC50	1148.9	nM	10.1038/s41467-023-40064-9
Homo sapiens	Dopamine D3 receptor	AC50	1936.5	nM	10.1038/s41467-023-40064-9
Homo sapiens	Dopamine D4 receptor	AC50	108.5	nM	10.1038/s41467-023-40064-9
Homo sapiens	Dopamine transporter	AC50	3454.7	nM	10.1038/s41467-023-40064-9
Homo sapiens	DSH1	IC50	507141.98	nM	10.6019/CHEMBL1201861
Homo sapiens	DU-145	Activity	0.931	None	10.1073/pnas.0707498104
Homo sapiens	DU-145	IC50	16400.0	nM	10.1016/j.bmcl.2016.06.077
Homo sapiens	DU-4475	IC50	4367.29	nM	10.6019/CHEMBL1201861
Homo sapiens	Dual serine/threonine and tyrosine protein kinase	Kd	1300.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Kd	130.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Kd	130.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Kd	130.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 1	Kd	2580.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Kd	110.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Kd	110.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Kd	1677.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 2	Thermal melting change	2.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 3	Kd	1700.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 3	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 4	Kd	700.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 4	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 5	Kd	46.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 5	Kd	3525.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Kd	5200.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 6	Thermal melting change	3.9	degrees C	10.1073/pnas.0708800104
Homo sapiens	Dual specificity mitogen-activated protein kinase kinase 7	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase CLK2	Kd	20.0	nM	10.1016/j.ejmech.2016.11.003
Homo sapiens	Dual specificity protein kinase CLK2	Kd	20.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity protein kinase CLK2	Kd	20.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase CLK2	Kd	20.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual specificity protein kinase CLK2	Kd	190.0	nM	10.1038/nbt1068
Homo sapiens	Dual specificity protein kinase CLK2	Kd	190.0	nM	10.1073/pnas.0707498104
Homo sapiens	Dual specificity protein kinase CLK2	Kd	922.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity protein kinase CLK2	Thermal melting change	5.9	degrees C	10.1073/pnas.0708800104
Homo sapiens	Dual specificity protein kinase CLK3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity protein kinase CLK3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase CLK3	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual specificity protein kinase CLK3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity protein kinase CLK3	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Dual specificity protein kinase CLK3	Thermal melting change	2.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	Dual specificity protein kinase CLK4	Kd	29.0	nM	10.1016/j.ejmech.2016.11.003
Homo sapiens	Dual specificity protein kinase CLK4	Kd	29.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity protein kinase CLK4	Kd	29.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase CLK4	Kd	29.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual specificity protein kinase CLK4	Kd	80.0	nM	10.1038/nbt1068
Homo sapiens	Dual specificity protein kinase CLK4	Kd	80.0	nM	10.1073/pnas.0707498104
Homo sapiens	Dual specificity protein kinase CLK4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity protein kinase TTK	Kd	63.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity protein kinase TTK	Kd	63.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity protein kinase TTK	Kd	63.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual specificity protein kinase TTK	Kd	230.0	nM	10.1038/nbt1068
Homo sapiens	Dual specificity protein kinase TTK	Kd	230.0	nM	10.1073/pnas.0707498104
Homo sapiens	Dual specificity protein kinase TTK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity testis-specific protein kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity testis-specific protein kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity testis-specific protein kinase 1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual specificity testis-specific protein kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	Kd	200.0	nM	10.1038/nbt.1990
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	Kd	200.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 1A	Kd	3675.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Kd	2300.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Kd	2300.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Kd	2300.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 2	Kd	680.0	nM	10.1038/nbt.1990
Homo sapiens	Dual-specificity tyrosine-phosphorylation regulated kinase 2	Kd	680.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual specificty protein kinase CLK1	Kd	22.0	nM	10.1016/j.ejmech.2016.11.003
Homo sapiens	Dual specificty protein kinase CLK1	Kd	22.0	nM	10.1038/nbt1358
Homo sapiens	Dual specificty protein kinase CLK1	Kd	22.0	nM	10.1038/nbt.1990
Homo sapiens	Dual specificty protein kinase CLK1	Kd	22.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Dual specificty protein kinase CLK1	Kd	100.0	nM	10.1038/nbt1068
Homo sapiens	Dual specificty protein kinase CLK1	Kd	100.0	nM	10.1073/pnas.0707498104
Homo sapiens	Dual specificty protein kinase CLK1	Kd	440.0	nM	10.1126/science.aan4368
Homo sapiens	Dual specificty protein kinase CLK1	Thermal melting change	5.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	Dynamin-like 120 kDa protein, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	EB2	IC50	656710.31	nM	10.6019/CHEMBL1201861
Homo sapiens	EB-3	IC50	29530.89	nM	10.6019/CHEMBL1201861
Homo sapiens	ECC4	IC50	98471.68	nM	10.6019/CHEMBL1201861
Homo sapiens	EC-GI-10	IC50	1951442.26	nM	10.6019/CHEMBL1201861
Homo sapiens	EFM-19	Activity	1.06	None	10.1073/pnas.0707498104
Homo sapiens	EFO-21	Activity	0.994	None	10.1073/pnas.0707498104
Homo sapiens	EGI-1	Activity	1.094	None	10.1073/pnas.0707498104
Homo sapiens	EHEB	IC50	34119.26	nM	10.6019/CHEMBL1201861
Homo sapiens	EKVX	GI50	7900.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	EKVX	IC50	1061717.33	nM	10.6019/CHEMBL1201861
Homo sapiens	Electron transfer flavoprotein subunit beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Elongation factor Tu, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	EM-2	IC50	18567.24	nM	10.6019/CHEMBL1201861
Homo sapiens	Endothelin receptor ET-A	AC50	8300.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	EOL1	IC50	0.001635	nM	10.6019/CHEMBL1201861
Homo sapiens	Ephrin type-A receptor 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-A receptor 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-A receptor 2	Inhibition	nan	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Ephrin type-A receptor 2	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Ephrin type-A receptor 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-A receptor 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-A receptor 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 3	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Ephrin type-A receptor 3	Kd	2100.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 3	Kd	2100.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 3	Kd	2100.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-A receptor 3	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 4	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Ephrin type-A receptor 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 4	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-A receptor 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-A receptor 4	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 5	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Ephrin type-A receptor 5	Kd	1200.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 5	Kd	5900.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 5	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-A receptor 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-A receptor 6	Kd	960.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 6	Kd	960.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 6	Kd	960.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-A receptor 6	Kd	2000.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 7	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Ephrin type-A receptor 7	Kd	710.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-A receptor 7	Kd	710.0	nM	10.1073/pnas.0707498104
Homo sapiens	Ephrin type-A receptor 7	Kd	2400.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 7	Kd	2400.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 7	Kd	2400.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-A receptor 7	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-A receptor 8	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Ephrin type-A receptor 8	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-A receptor 8	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-A receptor 8	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-A receptor 8	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Ephrin type-B receptor 1	Kd	480.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-B receptor 1	Kd	480.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 1	Kd	480.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-B receptor 1	Kd	960.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-B receptor 1	Kd	960.0	nM	10.1073/pnas.0707498104
Homo sapiens	Ephrin type-B receptor 2	Inhibition	nan	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Ephrin type-B receptor 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-B receptor 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-B receptor 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-B receptor 3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-B receptor 3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 3	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-B receptor 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-B receptor 4	IC50	50000.0	nM	10.1038/nchembio.117
Homo sapiens	Ephrin type-B receptor 4	Inhibition	nan	%	10.1021/acs.jmedchem.5b01582
Homo sapiens	Ephrin type-B receptor 4	Kd	2200.0	nM	10.1038/nbt1068
Homo sapiens	Ephrin type-B receptor 4	Kd	3100.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ephrin type-B receptor 4	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-B receptor 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ephrin type-B receptor 6	Kd	850.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ephrin type-B receptor 6	Kd	1000.0	nM	10.1038/nbt.1990
Homo sapiens	Ephrin type-B receptor 6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Epidermal growth factor receptor erbB1	AC50	8600.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	31.8	nM	10.1016/j.ejmech.2019.06.054
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	140.0	nM	10.1021/acs.jmedchem.8b01391
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	172.1	nM	10.1016/j.bmc.2014.04.049
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	172.1	nM	10.1016/j.bmc.2015.03.061
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	172.1	nM	10.1016/j.bmc.2021.116061
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	172.1	nM	10.1016/j.bmcl.2018.07.039
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	18000.0	nM	10.1038/nchembio.117
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	20000.0	nM	10.1021/jm0204183
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	172100.0	nM	10.1016/j.bmc.2010.03.052
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	172100.0	nM	10.1016/j.bmc.2010.05.049
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	172100.0	nM	10.1016/j.bmc.2011.11.058
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	172100.0	nM	10.1016/j.bmc.2012.05.068
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	172100.0	nM	10.1016/j.bmc.2012.12.045
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	172100.0	nM	10.1016/j.bmc.2013.01.040
Homo sapiens	Epidermal growth factor receptor erbB1	IC50	nan	None	10.1016/j.bmc.2016.11.026
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Epidermal growth factor receptor erbB1	Inhibition	nan	%	10.1016/j.ejmech.2018.09.032
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	860.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	2400.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	6788.0	nM	10.1126/science.aan4368
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	6800.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	6800.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	6800.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Epidermal growth factor receptor erbB1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Epithelial discoidin domain-containing receptor 1	Kd	2000.0	nM	10.1016/j.ejmech.2020.112421
Homo sapiens	Epithelial discoidin domain-containing receptor 1	Kd	2000.0	nM	10.1038/nbt1358
Homo sapiens	Epithelial discoidin domain-containing receptor 1	Kd	2000.0	nM	10.1038/nbt.1990
Homo sapiens	Epithelial discoidin domain-containing receptor 1	Kd	2000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Epithelial discoidin domain-containing receptor 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	EPLC-272H	Activity	0.857	None	10.1073/pnas.0707498104
Homo sapiens	Epoxide hydratase	IC50	10000.0	nM	10.1016/j.bmcl.2013.05.011
Homo sapiens	Equilibrative nucleoside transporter 1	AC50	5000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	ES1	IC50	10298.42	nM	10.6019/CHEMBL1201861
Homo sapiens	ES3	IC50	37500.38	nM	10.6019/CHEMBL1201861
Homo sapiens	ES4	IC50	2806.28	nM	10.6019/CHEMBL1201861
Homo sapiens	ES5	IC50	24734.92	nM	10.6019/CHEMBL1201861
Homo sapiens	ES6	IC50	981.06	nM	10.6019/CHEMBL1201861
Homo sapiens	ES7	IC50	177447.89	nM	10.6019/CHEMBL1201861
Homo sapiens	ES8	IC50	146113.1	nM	10.6019/CHEMBL1201861
Homo sapiens	Estrogen receptor alpha	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	ETK-1	IC50	1285.8	nM	10.6019/CHEMBL1201861
Homo sapiens	Eukaryotic translation initiation factor 2-alpha kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Eukaryotic translation initiation factor 2-alpha kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Eukaryotic translation initiation factor 2-alpha kinase 4	Kd	180.0	nM	10.1038/nbt1358
Homo sapiens	Eukaryotic translation initiation factor 2-alpha kinase 4	Kd	180.0	nM	10.1038/nbt.1990
Homo sapiens	Eukaryotic translation initiation factor 2-alpha kinase 4	Kd	180.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Eukaryotic translation initiation factor 5B	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	EVSA-T	Activity	1.017	None	10.1073/pnas.0707498104
Homo sapiens	EVSA-T	IC50	17048.46	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-1	IC50	4679.11	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-11	IC50	34472.54	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-12	IC50	1452216.08	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-13	IC50	55580.14	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-16	IC50	2135.08	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-18	IC50	1720215.75	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-24	IC50	547608.71	nM	10.6019/CHEMBL1201861
Homo sapiens	EW-3	IC50	6432.07	nM	10.6019/CHEMBL1201861
Homo sapiens	Exosome RNA helicase MTR4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ferrochelatase, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Fibroblast growth factor receptor 1	IC50	170.0	nM	10.1073/pnas.0707498104
Homo sapiens	Fibroblast growth factor receptor 1	IC50	1064.0	nM	10.1016/j.bmcl.2012.06.029
Homo sapiens	Fibroblast growth factor receptor 1	IC50	2900.0	nM	10.1021/jm0204183
Homo sapiens	Fibroblast growth factor receptor 1	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Fibroblast growth factor receptor 1	Inhibition	nan	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Fibroblast growth factor receptor 1	Kd	520.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 1	Kd	520.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 1	Kd	520.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Fibroblast growth factor receptor 1	Kd	1800.0	nM	10.1038/nbt1068
Homo sapiens	Fibroblast growth factor receptor 1	Kd	3595.0	nM	10.1126/science.aan4368
Homo sapiens	Fibroblast growth factor receptor 1	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	Fibroblast growth factor receptor 2	Inhibition	61.8	%	10.1039/C1MD00105A
Homo sapiens	Fibroblast growth factor receptor 2	Kd	530.0	nM	10.1038/nbt1068
Homo sapiens	Fibroblast growth factor receptor 2	Kd	530.0	nM	10.1073/pnas.0707498104
Homo sapiens	Fibroblast growth factor receptor 2	Kd	570.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 2	Kd	570.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 2	Kd	570.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Fibroblast growth factor receptor 3	Inhibition	nan	%	10.1021/acs.jmedchem.5b01582
Homo sapiens	Fibroblast growth factor receptor 3	Kd	290.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 3	Kd	290.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 3	Kd	290.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Fibroblast growth factor receptor 3	Kd	300.0	nM	10.1038/nbt1068
Homo sapiens	Fibroblast growth factor receptor 3	Kd	1400.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 3	Kd	1400.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 3	Kd	1400.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Fibroblast growth factor receptor 3	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	Fibroblast growth factor receptor 4	Kd	2100.0	nM	10.1038/nbt.1990
Homo sapiens	Fibroblast growth factor receptor 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Fibroblast growth factor receptor 4	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Focal adhesion kinase 1	IC50	1600.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	Focal adhesion kinase 1	Kd	440.0	nM	10.1038/nbt1358
Homo sapiens	Focal adhesion kinase 1	Kd	440.0	nM	10.1038/nbt.1990
Homo sapiens	Focal adhesion kinase 1	Kd	440.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Focal adhesion kinase 1	Kd	610.0	nM	10.1038/nbt1068
Homo sapiens	Focal adhesion kinase 1	Kd	610.0	nM	10.1073/pnas.0707498104
Homo sapiens	Focal adhesion kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Focal adhesion kinase 1	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	FTC-133	Activity	1.022	None	10.1073/pnas.0707498104
Homo sapiens	G-361	Activity	1.183	None	10.1073/pnas.0707498104
Homo sapiens	G-401	Activity	0.506	None	10.1073/pnas.0707498104
Homo sapiens	G-402	Activity	0.841	None	10.1073/pnas.0707498104
Homo sapiens	GAK	IC50	64656.78	nM	10.6019/CHEMBL1201861
Homo sapiens	GAMG	Activity	0.998	None	10.1073/pnas.0707498104
Homo sapiens	Gamma-secretase	Activity	nan	None	10.1016/j.bmcl.2010.02.110
Homo sapiens	Gamma-secretase	IC50	nan	None	10.1016/j.bmcl.2012.10.016
Homo sapiens	Gamma-secretase	Inhibition	26.0	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Gamma-secretase	Inhibition	53.0	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	GB-1	IC50	710.23	nM	10.6019/CHEMBL1201861
Homo sapiens	GCIY	IC50	392528.84	nM	10.6019/CHEMBL1201861
Homo sapiens	GCT	Activity	0.931	None	10.1073/pnas.0707498104
Homo sapiens	GDM-1	IC50	21941.42	nM	10.6019/CHEMBL1201861
Homo sapiens	General transcription and DNA repair factor IIH helicase subunit XPD	Kd	1225.0	nM	10.1126/science.aan4368
Homo sapiens	Ghrelin receptor	AC50	7200.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	GI-1	IC50	8204.11	nM	10.6019/CHEMBL1201861
Homo sapiens	GI-ME-N	IC50	775148.79	nM	10.6019/CHEMBL1201861
Homo sapiens	GIST430	Activity	nan	None	10.1021/acs.jmedchem.8b01845
Homo sapiens	GIST430	Activity	nan	None	10.1021/acs.jmedchem.9b01229
Homo sapiens	GIST430	GI50	47.0	nM	10.1021/acs.jmedchem.8b01845
Homo sapiens	GIST430	GI50	2000.0	nM	10.1021/acs.jmedchem.9b01229
Homo sapiens	GIST430	TGI	nan	None	10.1021/acs.jmedchem.8b01845
Homo sapiens	GIST48	GI50	47.0	nM	10.1021/acs.jmedchem.9b01229
Homo sapiens	GIST48	GI50	2000.0	nM	10.1021/acs.jmedchem.8b01845
Homo sapiens	GIST882	GI50	64.0	nM	10.1021/acs.jmedchem.8b01845
Homo sapiens	GIST882	GI50	64.0	nM	10.1021/acs.jmedchem.9b01229
Homo sapiens	GISTT1	Activity	0.09	g	10.1021/acs.jmedchem.9b00280
Homo sapiens	GISTT1	GI50	38.0	nM	10.1021/acs.jmedchem.8b01845
Homo sapiens	GISTT1	GI50	38.0	nM	10.1021/acs.jmedchem.9b01229
Homo sapiens	GISTT1	GI50	40.0	nM	10.1021/acs.jmedchem.7b00841
Homo sapiens	GISTT1	GI50	90.0	nM	10.1021/acs.jmedchem.7b00841
Homo sapiens	GISTT1	GI50	5880.0	nM	10.1021/acs.jmedchem.7b00841
Homo sapiens	GISTT1	TGI	93.6	%	10.1021/acs.jmedchem.9b00280
Homo sapiens	Glucocorticoid receptor	AC50	10000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Glucocorticoid receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Glutaminase kidney isoform, mitochondrial	Potency	25118.9	nM	None
Homo sapiens	Glycine--tRNA ligase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Glycogen synthase kinase-3 alpha	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Glycogen synthase kinase-3 alpha	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Glycogen synthase kinase-3 alpha	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Glycogen synthase kinase-3 alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Glycogen synthase kinase-3 beta	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Glycogen synthase kinase-3 beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Glycogen synthase kinase-3 beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Glycogen synthase kinase-3 beta	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Glycogen synthase kinase-3 beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Glycogen synthase kinase-3 beta	Thermal melting change	12.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	GMS-10	Activity	0.82	None	10.1073/pnas.0707498104
Homo sapiens	GOTO	IC50	31608.53	nM	10.6019/CHEMBL1201861
Homo sapiens	GP5d	Activity	1.12	None	10.1073/pnas.0707498104
Homo sapiens	G-protein coupled receptor kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	G protein-coupled receptor kinase 4	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	G protein-coupled receptor kinase 4	Kd	140.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	G protein-coupled receptor kinase 5	IC50	830.0	nM	10.1021/acs.jmedchem.0c01522
Homo sapiens	G protein-coupled receptor kinase 6	Kd	1615.0	nM	10.1126/science.aan4368
Homo sapiens	G protein-coupled receptor kinase 7	Kd	180.0	nM	10.1038/nbt.1990
Homo sapiens	G protein-coupled receptor kinase 7	Kd	180.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	GR-ST	IC50	10220.69	nM	10.6019/CHEMBL1201861
Homo sapiens	GT3TKB	IC50	6607.63	nM	10.6019/CHEMBL1201861
Homo sapiens	GTP-binding nuclear protein Ran	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Guanine nucleotide-binding protein G(i) subunit alpha-2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	H4	Activity	0.842	None	10.1073/pnas.0707498104
Homo sapiens	H4	Activity	40.0	uM	10.1016/j.bmcl.2010.02.110
Homo sapiens	H69AR	IC50	5800.0	nM	10.1016/j.ejmech.2020.112359
Homo sapiens	HAL-01	IC50	2059.46	nM	10.6019/CHEMBL1201861
Homo sapiens	HC-1	IC50	5432.91	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC1187	IC50	18018.75	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC1395	Activity	0.908	None	10.1073/pnas.0707498104
Homo sapiens	HCC1599	IC50	8199.87	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC1806	Activity	1.048	None	10.1073/pnas.0707498104
Homo sapiens	HCC1937	Activity	1.444	None	10.1073/pnas.0707498104
Homo sapiens	HCC1954	Activity	1.218	None	10.1073/pnas.0707498104
Homo sapiens	HCC2157	IC50	314432.99	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC2218	IC50	600384.33	nM	10.6019/CHEMBL1201861
Homo sapiens	HCC38	Activity	1.165	None	10.1073/pnas.0707498104
Homo sapiens	HCC70	Activity	1.143	None	10.1073/pnas.0707498104
Homo sapiens	HCE-4	IC50	3786.42	nM	10.6019/CHEMBL1201861
Homo sapiens	HCE-T	IC50	556276.24	nM	10.6019/CHEMBL1201861
Homo sapiens	HCT-116	Activity	0.924	None	10.1073/pnas.0707498104
Homo sapiens	HCT-116	Activity	14.16	%	10.1016/j.bmcl.2016.08.060
Homo sapiens	HCT-116	Activity	33.36	%	10.1016/j.bmcl.2016.08.060
Homo sapiens	HCT-116	Activity	50.07	%	10.1016/j.bmcl.2016.08.060
Homo sapiens	HCT-116	Activity	nan	None	10.1016/j.bmcl.2016.08.060
Homo sapiens	HCT-116	IC50	2110.0	nM	10.1039/C1MD00105A
Homo sapiens	HCT-116	IC50	4710.0	nM	10.1016/j.bmcl.2013.03.099
Homo sapiens	HCT-116	IC50	4710.0	nM	10.1016/j.bmcl.2016.08.060
Homo sapiens	HCT-116	IC50	5620.0	nM	10.1016/j.ejmech.2018.07.052
Homo sapiens	HCT-116	IC50	6100.0	nM	10.1016/j.ejmech.2011.10.009
Homo sapiens	HCT-116	IC50	10690.0	nM	10.1039/d2md00442a
Homo sapiens	HCT-116	IC50	18350.0	nM	10.1016/j.bmcl.2012.03.061
Homo sapiens	HCT-116	IC50	nan	None	10.1016/j.ejmech.2019.06.094
Homo sapiens	HCT-116	Inhibition	nan	%	10.1021/jm301419d
Homo sapiens	HCT-8	Activity	1.028	None	10.1073/pnas.0707498104
Homo sapiens	HDLM-2	IC50	6321.09	nM	10.6019/CHEMBL1201861
Homo sapiens	HD-MY-Z	IC50	5173.01	nM	10.6019/CHEMBL1201861
Homo sapiens	HEK293	IC50	5000.0	nM	10.1016/j.ejmech.2018.11.023
Homo sapiens	HEK293	IC50	5000.0	nM	10.1016/j.ejmech.2019.03.012
Homo sapiens	HEL	IC50	3480.05	nM	10.6019/CHEMBL1201861
Homo sapiens	HeLa	Activity	1.003	None	10.1073/pnas.0707498104
Homo sapiens	HeLa	Activity	1.051	None	10.1073/pnas.0707498104
Homo sapiens	HeLa	Activity	1.06	None	10.1073/pnas.0707498104
Homo sapiens	HeLa	Activity	1.072	None	10.1073/pnas.0707498104
Homo sapiens	HeLa	Activity	1.073	None	10.1073/pnas.0707498104
Homo sapiens	HeLa	Activity	1.1	None	10.1073/pnas.0707498104
Homo sapiens	HeLa	EC50	10000.0	nM	10.1021/jm201649s
Homo sapiens	HeLa	IC50	7800.0	nM	10.1016/j.ejmech.2018.11.023
Homo sapiens	HeLa	IC50	7800.0	nM	10.1016/j.ejmech.2019.03.012
Homo sapiens	HeLa	IC50	30000.0	nM	10.1016/j.bmcl.2015.05.017
Homo sapiens	HeLa	IC50	30000.0	nM	10.1016/j.ejmech.2020.113102
Homo sapiens	Heme oxygenase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Hepatocyte growth factor receptor	Activity	5.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	Hepatocyte growth factor receptor	Activity	96.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	Hepatocyte growth factor receptor	IC50	2000.0	nM	10.1016/j.bmcl.2008.04.009
Homo sapiens	Hepatocyte growth factor receptor	IC50	5000.0	nM	10.1016/j.bmcl.2009.01.068
Homo sapiens	Hepatocyte growth factor receptor	IC50	5000.0	nM	10.1016/j.bmcl.2009.10.040
Homo sapiens	Hepatocyte growth factor receptor	IC50	10000.0	nM	10.1016/j.bmcl.2008.04.009
Homo sapiens	Hepatocyte growth factor receptor	IC50	20000.0	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Hepatocyte growth factor receptor	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Hepatocyte growth factor receptor	Inhibition	nan	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Hepatocyte growth factor receptor	Inhibition	nan	%	10.1021/acs.jmedchem.5b01582
Homo sapiens	Hepatocyte growth factor receptor	Kd	1200.0	nM	10.1038/nbt.1990
Homo sapiens	Hepatocyte growth factor receptor	Kd	1200.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Hepatocyte growth factor receptor	Kd	4700.0	nM	10.1038/nbt.1990
Homo sapiens	Hepatocyte growth factor receptor	Kd	4700.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Hepatocyte growth factor receptor	Kd	7200.0	nM	10.1038/nbt.1990
Homo sapiens	Hepatocyte growth factor receptor	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Hepatocyte growth factor receptor	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Hepatocyte growth factor receptor	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	HepG2	Activity	5.0	%	10.1021/jm501177w
Homo sapiens	HepG2	Activity	28.0	%	10.1021/jm501177w
Homo sapiens	HepG2	Activity	68.0	%	10.1021/jm501177w
Homo sapiens	HepG2	Activity	75.0	%	10.1021/jm501177w
Homo sapiens	HepG2	IC50	3810.0	nM	10.1016/j.bmc.2010.05.021
Homo sapiens	HepG2	IC50	5610.0	nM	10.1016/j.bmcl.2013.08.037
Homo sapiens	HepG2	IC50	7780.0	nM	10.1016/j.ejmech.2018.07.052
Homo sapiens	HepG2	IC50	13240.0	nM	10.1016/j.bmcl.2012.03.061
Homo sapiens	HepG2	IC50	13600.0	nM	10.1016/j.ejmech.2014.07.071
Homo sapiens	HepG2	IC50	15400.0	nM	10.1016/j.ejmech.2011.10.009
Homo sapiens	HepG2	IC50	16060.0	nM	10.1016/j.bmcl.2015.05.017
Homo sapiens	HepG2	IC50	16060.0	nM	10.1016/j.bmcl.2016.12.029
Homo sapiens	HepG2	IC50	nan	None	10.1016/j.ejmech.2019.06.054
Homo sapiens	HepG2	IC50	nan	None	10.1016/j.ejmech.2019.06.094
Homo sapiens	HERG	AC50	581.7	nM	10.1038/s41467-023-40064-9
Homo sapiens	HERG	IC50	251.19	nM	10.1016/j.vascn.2014.07.002
Homo sapiens	HERG	IC50	500.0	nM	10.1016/j.ejmech.2014.05.051
Homo sapiens	HERG	IC50	500.0	nM	10.1016/j.ejmech.2016.12.038
Homo sapiens	HERG	IC50	7943.28	nM	10.1016/j.vascn.2014.07.002
Homo sapiens	HERG	IC50	10000.0	nM	10.1016/j.vascn.2014.07.002
Homo sapiens	HGC-27	Activity	0.751	None	10.1073/pnas.0707498104
Homo sapiens	HH	IC50	4209.14	nM	10.6019/CHEMBL1201861
Homo sapiens	Histamine H1 receptor	AC50	3300.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Histamine H2 receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Histamine H3 receptor	AC50	880.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Histone deacetylase 6	Inhibition	-2.67	%	10.6019/CHEMBL4808148
Homo sapiens	Histone deacetylase 6	Inhibition	16.34	%	10.6019/CHEMBL4808148
Homo sapiens	Histone-lysine N-methyltransferase, H3 lysine-9 specific 3	Potency	17782.8	nM	None
Homo sapiens	Histone-lysine N-methyltransferase MLL	Potency	70794.6	nM	None
Homo sapiens	HL-60	IC50	3530.0	nM	10.1007/s00044-012-0170-3
Homo sapiens	HL-60	IC50	3530.0	nM	10.1016/j.bmcl.2011.03.031
Homo sapiens	HL-60	IC50	4210.65	nM	10.6019/CHEMBL1201861
Homo sapiens	HL-60	IC50	7000.0	nM	10.1016/j.ejmech.2018.11.023
Homo sapiens	HL-60	IC50	8700.0	nM	10.1016/j.bmcl.2022.129041
Homo sapiens	HL-60	IC50	15500.0	nM	10.1016/j.ejmech.2011.10.009
Homo sapiens	HL-60	IC50	21500.0	nM	10.1016/j.ejmech.2019.111719
Homo sapiens	HLE	Activity	0.945	None	10.1073/pnas.0707498104
Homo sapiens	HMEC-1	IC50	7000.0	nM	10.1016/j.ejmech.2018.11.023
Homo sapiens	HMEC-1	IC50	7000.0	nM	10.1016/j.ejmech.2019.03.012
Homo sapiens	HMEC-1	MAC	3.0	uM	10.1016/j.ejmech.2018.11.023
Homo sapiens	HMEC-1	MAC	3.0	uM	10.1016/j.ejmech.2019.03.012
Homo sapiens	Homeodomain-interacting protein kinase 1	Kd	55.0	nM	10.1038/nbt.1990
Homo sapiens	Homeodomain-interacting protein kinase 1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Homeodomain-interacting protein kinase 2	Kd	31.0	nM	10.1038/nbt.1990
Homo sapiens	Homeodomain-interacting protein kinase 2	Kd	31.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Homeodomain-interacting protein kinase 3	Kd	41.0	nM	10.1038/nbt.1990
Homo sapiens	Homeodomain-interacting protein kinase 3	Kd	41.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Homeodomain-interacting protein kinase 4	Kd	160.0	nM	10.1038/nbt.1990
Homo sapiens	Homeodomain-interacting protein kinase 4	Kd	160.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Homo sapiens	Activity	31.0	%	10.1016/j.ejmech.2017.08.007
Homo sapiens	Homo sapiens	AUC	1063.0	ng.hr.mL-1	10.1124/dmd.111.042853
Homo sapiens	Homo sapiens	CL/F	49.9	L/hr	10.1124/dmd.111.042853
Homo sapiens	Homo sapiens	Cmax	61.23	nM	10.1124/dmd.111.042853
Homo sapiens	Homo sapiens	DILI_Concern	nan	None	10.1016/j.drudis.2016.02.015
Homo sapiens	Homo sapiens	DILI_severity_class	8.0	None	10.1016/j.drudis.2016.02.015
Homo sapiens	Homo sapiens	Survival	7.8	months	10.1016/j.ejmech.2017.08.007
Homo sapiens	Homo sapiens	Survival	9.5	months	10.1016/j.ejmech.2017.08.007
Homo sapiens	Homo sapiens	Survival	11.0	months	10.1016/j.ejmech.2017.08.007
Homo sapiens	Homo sapiens	Survival	26.4	months	10.1016/j.ejmech.2017.08.007
Homo sapiens	Homo sapiens	Survival	29.1	months	10.1016/j.ejmech.2017.08.007
Homo sapiens	Homo sapiens	T1/2	50.9	hr	10.1124/dmd.111.042853
Homo sapiens	Homo sapiens	Tmax	8.0	hr	10.1124/dmd.111.042853
Homo sapiens	HOP-62	IC50	4335.2	nM	10.6019/CHEMBL1201861
Homo sapiens	HOP-92	Activity	0.935	None	10.1073/pnas.0707498104
Homo sapiens	Hormonally up-regulated neu tumor-associated kinase	Kd	500.0	nM	10.1038/nbt.1990
Homo sapiens	Hormonally up-regulated neu tumor-associated kinase	Kd	500.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	HOS	Activity	0.987	None	10.1073/pnas.0707498104
Homo sapiens	HPAC	Activity	1.047	None	10.1073/pnas.0707498104
Homo sapiens	HPAF-II	Activity	1.089	None	10.1073/pnas.0707498104
Homo sapiens	Hs 683	Activity	1.139	None	10.1073/pnas.0707498104
Homo sapiens	HT	IC50	69470.83	nM	10.6019/CHEMBL1201861
Homo sapiens	HT-1080	Activity	1.023	None	10.1073/pnas.0707498104
Homo sapiens	HT-1080	ED75	65.0	mg/kg/day	10.1021/jm061223o
Homo sapiens	HT-144	IC50	28689.95	nM	10.6019/CHEMBL1201861
Homo sapiens	HT-29	Activity	1.16	None	10.1073/pnas.0707498104
Homo sapiens	HT-29	Activity	3.0	%	10.1016/j.ejmech.2018.03.039
Homo sapiens	HT-29	Activity	22.0	%	10.1016/j.ejmech.2018.03.039
Homo sapiens	HT-29	Activity	45.0	%	10.1016/j.ejmech.2018.03.039
Homo sapiens	HT-29	Activity	46.0	%	10.1016/j.ejmech.2018.03.039
Homo sapiens	HT-29	Activity	47.0	%	10.1016/j.ejmech.2018.03.039
Homo sapiens	HT-29	Activity	68.0	%	10.1016/j.ejmech.2018.03.039
Homo sapiens	HT-29	Activity	75.0	%	10.1016/j.ejmech.2018.03.039
Homo sapiens	HT-29	Activity	88.9	%	10.1016/j.ejmech.2014.05.051
Homo sapiens	HT-29	Activity	90.0	%	10.1016/j.ejmech.2018.03.039
Homo sapiens	HT-29	Activity	100.0	%	10.1016/j.ejmech.2018.03.039
Homo sapiens	HT-29	Activity	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	HT-29	Activity	nan	None	10.1021/jm101036c
Homo sapiens	HT-29	GI	10.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	HT-29	GI50	1600.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	HT-29	IC50	330.0	nM	10.1016/j.bmcl.2012.02.068
Homo sapiens	HT-29	IC50	330.0	nM	10.1016/j.ejmech.2012.10.020
Homo sapiens	HT-29	IC50	1300.0	nM	10.1016/j.ejmech.2011.05.017
Homo sapiens	HT-29	IC50	1470.0	nM	10.1016/j.bmcl.2013.08.037
Homo sapiens	HT-29	IC50	1700.0	nM	10.1016/j.bmcl.2016.02.063
Homo sapiens	HT-29	IC50	3800.0	nM	10.1016/j.ejmech.2018.11.023
Homo sapiens	HT-29	IC50	3800.0	nM	10.1016/j.ejmech.2019.03.012
Homo sapiens	HT-29	IC50	4700.0	nM	10.1016/j.bmcl.2015.05.017
Homo sapiens	HT-29	IC50	10140.0	nM	10.1016/j.ejmech.2020.112359
Homo sapiens	HT-29	IC50	10340.0	nM	10.1016/j.ejmech.2020.113083
Homo sapiens	HT-29	IC50	nan	None	10.1016/j.ejmech.2019.06.094
Homo sapiens	HT-29	TGI	53.83	%	10.1021/jm101036c
Homo sapiens	HT-3	Activity	0.975	None	10.1073/pnas.0707498104
Homo sapiens	HTC-C3	Activity	0.689	None	10.1073/pnas.0707498104
Homo sapiens	Huh-7	CC50	246000.0	nM	10.1021/acs.jmedchem.9b00136
Homo sapiens	Huh-7	IC50	3030.0	nM	10.1016/j.ejmech.2018.07.052
Homo sapiens	Huh-7	IC50	4707.0	nM	10.1021/acsmedchemlett.7b00192
Homo sapiens	Huh-7.5	CC50	10000.0	nM	10.1021/acs.jmedchem.0c01467
Homo sapiens	Huntingtin	Potency	35481.3	nM	None
Homo sapiens	HuP-T3	Activity	1.215	None	10.1073/pnas.0707498104
Homo sapiens	HuP-T4	Activity	0.98	None	10.1073/pnas.0707498104
Homo sapiens	HuTu80	IC50	13757.26	nM	10.6019/CHEMBL1201861
Homo sapiens	HUVEC	Activity	43.0	%	10.1021/acs.jmedchem.1c00892
Homo sapiens	HUVEC	Activity	nan	None	10.1016/j.bmcl.2011.09.022
Homo sapiens	HUVEC	Activity	nan	None	10.1016/j.bmcl.2016.02.033
Homo sapiens	HUVEC	Activity	nan	None	10.1021/jm301419d
Homo sapiens	HUVEC	Activity	nan	None	10.1039/C1MD00105A
Homo sapiens	HUVEC	EC50	645.0	nM	10.1016/j.ejmech.2013.03.022
Homo sapiens	HUVEC	IC50	7.0	nM	10.1021/acs.jmedchem.5b01582
Homo sapiens	HUVEC	IC50	11.8	nM	10.1016/j.bmc.2014.04.049
Homo sapiens	HUVEC	IC50	120.0	nM	10.1016/j.bmc.2011.06.013
Homo sapiens	HUVEC	IC50	546.0	nM	10.1021/acsmedchemlett.7b00281
Homo sapiens	HUVEC	IC50	800.0	nM	10.1016/j.ejmech.2016.04.029
Homo sapiens	HUVEC	IC50	1500.0	nM	10.1021/acs.jnatprod.0c00772
Homo sapiens	HUVEC	IC50	2100.0	nM	10.1021/acs.jnatprod.1c00837
Homo sapiens	HUVEC	IC50	2540.0	nM	10.1021/acs.jmedchem.0c01965
Homo sapiens	HUVEC	IC50	2750.0	nM	10.1007/s00044-012-0170-3
Homo sapiens	HUVEC	IC50	2750.0	nM	10.1016/j.bmcl.2011.03.031
Homo sapiens	HUVEC	IC50	3000.0	nM	10.1016/j.bmcl.2017.12.066
Homo sapiens	HUVEC	IC50	3000.0	nM	10.1021/acs.jmedchem.5b01582
Homo sapiens	HUVEC	IC50	3200.0	nM	10.1016/j.ejmech.2018.10.045
Homo sapiens	HUVEC	IC50	3630.0	nM	10.1016/j.ejmech.2019.06.094
Homo sapiens	HUVEC	IC50	3900.0	nM	10.1007/s00044-012-0170-3
Homo sapiens	HUVEC	IC50	4040.0	nM	10.1007/s00044-012-0170-3
Homo sapiens	HUVEC	IC50	4040.0	nM	10.1016/j.bmcl.2011.03.031
Homo sapiens	HUVEC	IC50	6360.0	nM	10.1016/j.ejmech.2018.03.018
Homo sapiens	HUVEC	IC50	6370.0	nM	10.1016/j.ejmech.2020.113083
Homo sapiens	HUVEC	IC50	6460.0	nM	10.1016/j.ejmech.2019.06.094
Homo sapiens	HUVEC	IC50	9920.0	nM	10.1021/acsmedchemlett.7b00281
Homo sapiens	HUVEC	IC50	nan	None	10.1016/j.ejmech.2019.06.054
Homo sapiens	HUVEC	IC90	1000.0	nM	10.1016/j.bmcl.2011.09.022
Homo sapiens	HUVEC	Inhibition	nan	%	10.1016/j.bmc.2015.03.085
Homo sapiens	HUVEC	Inhibition	nan	%	10.1016/j.bmcl.2011.09.022
Homo sapiens	HUVEC	Inhibition	nan	%	10.1021/acsmedchemlett.7b00192
Homo sapiens	HUVEC	Inhibition	nan	%	10.1021/jm301419d
Homo sapiens	IA-LM	IC50	184193.16	nM	10.6019/CHEMBL1201861
Homo sapiens	IGR-1	Activity	1.214	None	10.1073/pnas.0707498104
Homo sapiens	IGROV-1	Activity	1.02	None	10.1073/pnas.0707498104
Homo sapiens	IM-9	IC50	1350.0	nM	10.1007/s00044-012-0170-3
Homo sapiens	IM-9	IC50	1350.0	nM	10.1016/j.bmcl.2011.03.031
Homo sapiens	IM-9	IC50	1678948.53	nM	10.6019/CHEMBL1201861
Homo sapiens	IMR-5	IC50	7548.76	nM	10.6019/CHEMBL1201861
Homo sapiens	IMR-90	Activity	1.035	None	10.1073/pnas.0707498104
Homo sapiens	Inactive serine/threonine-protein kinase VRK3	Thermal melting change	nan	None	10.1073/pnas.0708800104
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	Kd	520.0	nM	10.1038/nbt.1990
Homo sapiens	Inhibitor of nuclear factor kappa B kinase alpha subunit	Kd	520.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Inhibitor of nuclear factor kappa B kinase beta subunit	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	Kd	620.0	nM	10.1038/nbt1358
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	Kd	620.0	nM	10.1038/nbt.1990
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	Kd	620.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Inhibitor of nuclear factor kappa B kinase epsilon subunit	Kd	1731.0	nM	10.1126/science.aan4368
Homo sapiens	Inosine-5'-monophosphate dehydrogenase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Insulin-like growth factor I receptor	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Insulin-like growth factor I receptor	Inhibition	nan	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Insulin-like growth factor I receptor	Kd	2600.0	nM	10.1038/nbt1358
Homo sapiens	Insulin-like growth factor I receptor	Kd	2600.0	nM	10.1038/nbt.1990
Homo sapiens	Insulin-like growth factor I receptor	Kd	2600.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Insulin-like growth factor I receptor	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Insulin receptor	IC50	3200.0	nM	10.1038/nchembio.117
Homo sapiens	Insulin receptor	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Insulin receptor	Kd	180.0	nM	10.1038/nbt1068
Homo sapiens	Insulin receptor	Kd	180.0	nM	10.1073/pnas.0707498104
Homo sapiens	Insulin receptor	Kd	500.0	nM	10.1038/nbt1358
Homo sapiens	Insulin receptor	Kd	500.0	nM	10.1038/nbt.1990
Homo sapiens	Insulin receptor	Kd	500.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Insulin receptor	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Insulin receptor-related protein	Kd	430.0	nM	10.1038/nbt1358
Homo sapiens	Insulin receptor-related protein	Kd	430.0	nM	10.1038/nbt.1990
Homo sapiens	Insulin receptor-related protein	Kd	430.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Integrin alpha-V/beta-3	Drug uptake	2.9	nmol	10.1021/acs.jmedchem.6b01266
Homo sapiens	Integrin alpha-V/beta-3	Drug uptake	5.72	nmol	10.1021/acs.jmedchem.6b01266
Homo sapiens	Integrin alpha-V/beta-3	Drug uptake	95.3	pmol/min	10.1021/acs.jmedchem.6b01266
Homo sapiens	Integrin alpha-V/beta-3	Inhibition	nan	%	10.1021/acs.jmedchem.6b01266
Homo sapiens	Integrin alpha-V/beta-3	log(activity)	1.98	None	10.1021/acs.jmedchem.6b01266
Homo sapiens	Interferon-induced, double-stranded RNA-activated protein kinase	Kd	670.0	nM	10.1038/nbt1358
Homo sapiens	Interferon-induced, double-stranded RNA-activated protein kinase	Kd	670.0	nM	10.1038/nbt.1990
Homo sapiens	Interferon-induced, double-stranded RNA-activated protein kinase	Kd	670.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Interleukin-1 receptor-associated kinase 1	Kd	14.0	nM	10.1038/nbt.1990
Homo sapiens	Interleukin-1 receptor-associated kinase 1	Kd	14.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Interleukin-1 receptor-associated kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Interleukin-1 receptor-associated kinase 3	Kd	940.0	nM	10.1038/nbt1358
Homo sapiens	Interleukin-1 receptor-associated kinase 3	Kd	940.0	nM	10.1038/nbt.1990
Homo sapiens	Interleukin-1 receptor-associated kinase 3	Kd	940.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Interleukin-1 receptor-associated kinase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Interleukin-1 receptor-associated kinase 4	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Interleukin-1 receptor-associated kinase 4	Kd	66.0	nM	10.1038/nbt.1990
Homo sapiens	Interleukin-1 receptor-associated kinase 4	Kd	2625.0	nM	10.1126/science.aan4368
Homo sapiens	IPC-298	Activity	1.143	None	10.1073/pnas.0707498104
Homo sapiens	Ishikawa	Activity	0.948	None	10.1073/pnas.0707498104
Homo sapiens	Ishikawa	Activity	1.003	None	10.1073/pnas.0707498104
Homo sapiens	Ishikawa	Activity	14.3	uM	10.1016/j.ejmech.2018.10.045
Homo sapiens	Isoleucine--tRNA ligase, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	IST-MEL1	IC50	12869.45	nM	10.6019/CHEMBL1201861
Homo sapiens	IST-MES1	IC50	13672.93	nM	10.6019/CHEMBL1201861
Homo sapiens	IST-SL1	IC50	8024.17	nM	10.6019/CHEMBL1201861
Homo sapiens	IST-SL2	IC50	6125.19	nM	10.6019/CHEMBL1201861
Homo sapiens	J82	Activity	1.0	None	10.1073/pnas.0707498104
Homo sapiens	JAR	IC50	3988.32	nM	10.6019/CHEMBL1201861
Homo sapiens	JIYOYE	IC50	26274.19	nM	10.6019/CHEMBL1201861
Homo sapiens	J-RT3-T3-5	IC50	6079.09	nM	10.6019/CHEMBL1201861
Homo sapiens	Jurkat	IC50	1000.0	nM	10.1021/acs.jmedchem.8b01714
Homo sapiens	Jurkat	IC50	8500.0	nM	10.1016/j.ejmech.2019.111719
Homo sapiens	JVM-2	IC50	28289.82	nM	10.6019/CHEMBL1201861
Homo sapiens	JVM-3	IC50	1600617.87	nM	10.6019/CHEMBL1201861
Homo sapiens	K052	IC50	2402.02	nM	10.6019/CHEMBL1201861
Homo sapiens	K5	IC50	12298.52	nM	10.6019/CHEMBL1201861
Homo sapiens	K562	EC50	7030.0	nM	10.1016/j.ejmech.2020.112316
Homo sapiens	K562	EC50	7230.0	nM	10.1016/j.ejmech.2020.112316
Homo sapiens	K562	EC50	12500.0	nM	10.1016/j.ejmech.2020.112316
Homo sapiens	K562	GI50	1000.0	nM	10.1021/acs.jmedchem.6b00200
Homo sapiens	K562	IC50	2410.0	nM	10.1007/s00044-012-0170-3
Homo sapiens	K562	IC50	2410.0	nM	10.1016/j.bmcl.2011.03.031
Homo sapiens	K562	IC50	5800.0	nM	10.1016/j.bmcl.2022.129041
Homo sapiens	K562	IC50	11870.23	nM	10.6019/CHEMBL1201861
Homo sapiens	K562	IC50	14000.0	nM	10.1016/j.bmcl.2017.07.029
Homo sapiens	K562	IC50	21900.0	nM	10.1016/j.ejmech.2011.10.009
Homo sapiens	K562	Inhibition	61.0	%	10.1016/j.ejmech.2020.112316
Homo sapiens	KALS-1	IC50	16593.13	nM	10.6019/CHEMBL1201861
Homo sapiens	Kappa opioid receptor	AC50	10342.8	nM	10.1038/s41467-023-40064-9
Homo sapiens	KARPAS-299	IC50	2113.13	nM	10.6019/CHEMBL1201861
Homo sapiens	KARPAS-422	IC50	7572.06	nM	10.6019/CHEMBL1201861
Homo sapiens	KARPAS-45	IC50	2494.46	nM	10.6019/CHEMBL1201861
Homo sapiens	Kasumi 1	IC50	16.0	nM	10.1016/j.bmc.2010.05.021
Homo sapiens	Kasumi 1	IC50	166607.38	nM	10.6019/CHEMBL1201861
Homo sapiens	KB	GI	10.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	KE-37	IC50	4061.58	nM	10.6019/CHEMBL1201861
Homo sapiens	KG-1	IC50	6028.78	nM	10.6019/CHEMBL1201861
Homo sapiens	KGN	IC50	2603.39	nM	10.6019/CHEMBL1201861
Homo sapiens	KHOS/NP	Activity	0.899	None	10.1073/pnas.0707498104
Homo sapiens	KINGS-1	IC50	102588.21	nM	10.6019/CHEMBL1201861
Homo sapiens	KLE	IC50	29619.03	nM	10.6019/CHEMBL1201861
Homo sapiens	KM12	IC50	350.14	nM	10.6019/CHEMBL1201861
Homo sapiens	KM-H2	Activity	1.272	None	10.1073/pnas.0707498104
Homo sapiens	KM-H2	IC50	44957.74	nM	10.6019/CHEMBL1201861
Homo sapiens	KMOE-2	IC50	8194.2	nM	10.6019/CHEMBL1201861
Homo sapiens	KMS-12-PE	IC50	22273.95	nM	10.6019/CHEMBL1201861
Homo sapiens	KNS-42	IC50	327343.8	nM	10.6019/CHEMBL1201861
Homo sapiens	KNS-81-FD	IC50	850390.79	nM	10.6019/CHEMBL1201861
Homo sapiens	KP-4	Activity	1.408	None	10.1073/pnas.0707498104
Homo sapiens	KP-N-RT-BM-1	IC50	136501.69	nM	10.6019/CHEMBL1201861
Homo sapiens	KP-N-YS	IC50	14289.44	nM	10.6019/CHEMBL1201861
Homo sapiens	KS-1	IC50	1692.47	nM	10.6019/CHEMBL1201861
Homo sapiens	KU-19-19	Activity	1.017	None	10.1073/pnas.0707498104
Homo sapiens	KU812 cell line	IC50	6694.2	nM	10.6019/CHEMBL1201861
Homo sapiens	KURAMOCHI	IC50	93087.14	nM	10.6019/CHEMBL1201861
Homo sapiens	KY821	IC50	2797.58	nM	10.6019/CHEMBL1201861
Homo sapiens	KYSE-140	Activity	0.896	None	10.1073/pnas.0707498104
Homo sapiens	KYSE-180	Activity	1.099	None	10.1073/pnas.0707498104
Homo sapiens	KYSE-270	Activity	1.047	None	10.1073/pnas.0707498104
Homo sapiens	KYSE-410	Activity	0.889	None	10.1073/pnas.0707498104
Homo sapiens	KYSE-450	Activity	1.016	None	10.1073/pnas.0707498104
Homo sapiens	KYSE-510	Activity	0.882	None	10.1073/pnas.0707498104
Homo sapiens	L-363	IC50	4806.21	nM	10.6019/CHEMBL1201861
Homo sapiens	L-428	IC50	18015.08	nM	10.6019/CHEMBL1201861
Homo sapiens	L-540	IC50	66545.24	nM	10.6019/CHEMBL1201861
Homo sapiens	LAMA-84	IC50	2695.45	nM	10.6019/CHEMBL1201861
Homo sapiens	LAN-6	IC50	14245.73	nM	10.6019/CHEMBL1201861
Homo sapiens	LB1047-RCC	IC50	1816.24	nM	10.6019/CHEMBL1201861
Homo sapiens	LB2241-RCC	IC50	238478.22	nM	10.6019/CHEMBL1201861
Homo sapiens	LB2518-MEL	IC50	528801.96	nM	10.6019/CHEMBL1201861
Homo sapiens	LB373-MEL-D	IC50	540755.91	nM	10.6019/CHEMBL1201861
Homo sapiens	LB647-SCLC	IC50	161260.81	nM	10.6019/CHEMBL1201861
Homo sapiens	LB771-HNC	IC50	333074.77	nM	10.6019/CHEMBL1201861
Homo sapiens	LB831-BLC	IC50	32384.31	nM	10.6019/CHEMBL1201861
Homo sapiens	LB996-RCC	IC50	4121.68	nM	10.6019/CHEMBL1201861
Homo sapiens	LC-1F	IC50	43368.22	nM	10.6019/CHEMBL1201861
Homo sapiens	LC-2-ad	IC50	1114.07	nM	10.6019/CHEMBL1201861
Homo sapiens	LC4-1	IC50	4380.7	nM	10.6019/CHEMBL1201861
Homo sapiens	LCLC-97TM1	Activity	1.265	None	10.1073/pnas.0707498104
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	IC50	15.0	nM	10.1016/j.bmcl.2013.04.086
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	IC50	28.0	nM	10.1016/j.bmcl.2013.05.054
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	Kd	76.0	nM	10.1038/nbt.1990
Homo sapiens	Leucine-rich repeat serine/threonine-protein kinase 2	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	Leukocyte tyrosine kinase receptor	Kd	1800.0	nM	10.1038/nbt1358
Homo sapiens	Leukocyte tyrosine kinase receptor	Kd	1800.0	nM	10.1038/nbt.1990
Homo sapiens	Leukocyte tyrosine kinase receptor	Kd	1800.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	LIM domain kinase 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	LIM domain kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	LIM domain kinase 1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	LIM domain kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	LIM domain kinase 1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	LIM domain kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	LIM domain kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	LIM domain kinase 2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	LIM domain kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Liver glycogen phosphorylase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Liver microsome	T1/2	0.735	hr	10.1021/jm501284e
Homo sapiens	Liver microsomes	T1/2	0.5	hr	10.1021/jm401067s
Homo sapiens	LK-2	Activity	1.0	None	10.1073/pnas.0707498104
Homo sapiens	LN-405	Activity	0.844	None	10.1073/pnas.0707498104
Homo sapiens	LNCaP	IC50	12610.0	nM	10.1016/j.bmcl.2016.05.019
Homo sapiens	LNCaP-Clone-FGC	IC50	882124.32	nM	10.6019/CHEMBL1201861
Homo sapiens	Long-chain-fatty-acid--CoA ligase 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	LOUCY	IC50	11987.49	nM	10.6019/CHEMBL1201861
Homo sapiens	LoVo	Activity	0.693	None	10.1073/pnas.0707498104
Homo sapiens	LOX IMVI	IC50	16255.98	nM	10.6019/CHEMBL1201861
Homo sapiens	LP-1	IC50	9780.83	nM	10.6019/CHEMBL1201861
Homo sapiens	LS-1034	IC50	154318.55	nM	10.6019/CHEMBL1201861
Homo sapiens	LS-123	IC50	9681.61	nM	10.6019/CHEMBL1201861
Homo sapiens	LS174T	Activity	0.976	None	10.1073/pnas.0707498104
Homo sapiens	LS-411N	IC50	377461.28	nM	10.6019/CHEMBL1201861
Homo sapiens	LS-513	IC50	55877.51	nM	10.6019/CHEMBL1201861
Homo sapiens	LU-134-A	IC50	52334.88	nM	10.6019/CHEMBL1201861
Homo sapiens	LU-135	Activity	1.055	None	10.1073/pnas.0707498104
Homo sapiens	LU-139	IC50	264810.11	nM	10.6019/CHEMBL1201861
Homo sapiens	LU-165	IC50	401593.35	nM	10.6019/CHEMBL1201861
Homo sapiens	Lu-65	IC50	192987.03	nM	10.6019/CHEMBL1201861
Homo sapiens	LU-99A	Activity	0.929	None	10.1073/pnas.0707498104
Homo sapiens	LXF-289 cell line	IC50	2729.89	nM	10.6019/CHEMBL1201861
Homo sapiens	LXR-alpha	AC50	10000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	LXR-alpha	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	LXR-beta	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	M059J	Activity	1.113	None	10.1073/pnas.0707498104
Homo sapiens	M14	Activity	0.811	None	10.1073/pnas.0707498104
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	2.0	%	10.1016/j.bmc.2010.01.056
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	37.0	%	10.1016/j.bmc.2010.01.056
Homo sapiens	Macrophage colony stimulating factor receptor	Activity	90.0	%	10.1016/j.bmc.2010.01.056
Homo sapiens	Macrophage colony stimulating factor receptor	IC50	35.0	nM	10.1021/jm901132v
Homo sapiens	Macrophage colony stimulating factor receptor	IC50	82.5	nM	10.1021/acs.jmedchem.0c02247
Homo sapiens	Macrophage colony stimulating factor receptor	IC50	82.5	nM	10.1021/acs.jmedchem.1c01184
Homo sapiens	Macrophage colony stimulating factor receptor	IC50	155.0	nM	10.1016/j.bmc.2010.01.056
Homo sapiens	Macrophage colony stimulating factor receptor	Inhibition	99.2	%	10.1016/j.ejmech.2020.112316
Homo sapiens	Macrophage colony stimulating factor receptor	Inhibition	99.8	%	10.1016/j.ejmech.2020.112316
Homo sapiens	Macrophage colony stimulating factor receptor	Inhibition	nan	%	10.1016/j.bmc.2010.01.056
Homo sapiens	Macrophage colony stimulating factor receptor	Kd	2.0	nM	10.1038/nbt1358
Homo sapiens	Macrophage colony stimulating factor receptor	Kd	2.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Macrophage colony stimulating factor receptor	Kd	2.5	nM	10.1038/nbt.1990
Homo sapiens	Macrophage colony stimulating factor receptor	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	Macrophage colony stimulating factor receptor	logIC50	2.18	None	10.1016/j.bmc.2010.01.056
Homo sapiens	Macrophage-stimulating protein receptor	Inhibition	nan	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Macrophage-stimulating protein receptor	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Macrophage-stimulating protein receptor	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Macrophage-stimulating protein receptor	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase-activated protein kinase 2	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	MAP kinase-activated protein kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase-activated protein kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase-activated protein kinase 2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MAP kinase-activated protein kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase-activated protein kinase 5	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	MAP kinase-activated protein kinase 5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase-activated protein kinase 5	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase-activated protein kinase 5	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MAP kinase-activated protein kinase 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase ERK1	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	MAP kinase ERK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase ERK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase ERK1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MAP kinase ERK1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase ERK1	Thermal melting change	0.9	degrees C	10.1073/pnas.0708800104
Homo sapiens	MAP kinase ERK2	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	MAP kinase ERK2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase ERK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase ERK2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MAP kinase ERK2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	Kd	3900.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase-interacting serine/threonine-protein kinase MNK1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MAP kinase p38 alpha	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	MAP kinase p38 alpha	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase p38 alpha	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 alpha	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MAP kinase p38 alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase p38 alpha	Kd	nan	None	10.1038/nbt1068
Homo sapiens	MAP kinase p38 beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase p38 beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 beta	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MAP kinase p38 beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MAP kinase p38 beta	Kd	nan	None	10.1038/nbt1068
Homo sapiens	MAP kinase p38 beta	Thermal melting change	0.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	MAP kinase p38 delta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 delta	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MAP kinase p38 gamma	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase p38 gamma	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase p38 gamma	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MAP kinase p38 gamma	Kd	nan	None	10.1038/nbt1068
Homo sapiens	MAP kinase signal-integrating kinase 2	Kd	5700.0	nM	10.1038/nbt.1990
Homo sapiens	MAP kinase signal-integrating kinase 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	MAP kinase signal-integrating kinase 2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MAP kinase signal-integrating kinase 2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Kd	310.0	nM	10.1038/nbt1358
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Kd	310.0	nM	10.1038/nbt.1990
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Kd	310.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Kd	320.0	nM	10.1038/nbt1068
Homo sapiens	MAP/microtubule affinity-regulating kinase 2	Kd	3013.0	nM	10.1126/science.aan4368
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	Kd	3600.0	nM	10.1038/nbt1358
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	Kd	3600.0	nM	10.1038/nbt.1990
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	Kd	3600.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MAP/microtubule affinity-regulating kinase 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Maternal embryonic leucine zipper kinase	Kd	350.0	nM	10.1038/nbt1358
Homo sapiens	Maternal embryonic leucine zipper kinase	Kd	350.0	nM	10.1038/nbt.1990
Homo sapiens	Maternal embryonic leucine zipper kinase	Kd	350.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Maternal embryonic leucine zipper kinase	Kd	1353.0	nM	10.1126/science.aan4368
Homo sapiens	MC116	IC50	4430.81	nM	10.6019/CHEMBL1201861
Homo sapiens	MC-CAR	IC50	8335.8	nM	10.6019/CHEMBL1201861
Homo sapiens	MCF-10A	IC50	nan	None	10.1016/j.bmcl.2016.06.077
Homo sapiens	MCF7	Activity	1.068	None	10.1073/pnas.0707498104
Homo sapiens	MCF7	EC50	960.0	nM	10.1021/acsmedchemlett.8b00596
Homo sapiens	MCF7	GI	10.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	MCF7	GI50	2000.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	MCF7	IC50	27.1	nM	10.1016/j.bmc.2014.04.049
Homo sapiens	MCF7	IC50	29.3	nM	10.1016/j.bmc.2014.04.049
Homo sapiens	MCF7	IC50	80.0	nM	10.1016/j.ejmech.2018.11.023
Homo sapiens	MCF7	IC50	80.0	nM	10.1016/j.ejmech.2019.03.012
Homo sapiens	MCF7	IC50	6290.0	nM	10.1016/j.bmcl.2013.03.099
Homo sapiens	MCF7	IC50	6290.0	nM	10.1016/j.bmcl.2016.08.060
Homo sapiens	MCF7	IC50	6800.0	nM	10.1016/j.ejmech.2019.111719
Homo sapiens	MCF7	IC50	10500.0	nM	10.1016/j.ejmech.2014.07.071
Homo sapiens	MCF7	IC50	23760.0	nM	10.1016/j.bmcl.2016.05.019
Homo sapiens	MCF7	IC50	25400.0	nM	10.1016/j.ejmech.2020.113102
Homo sapiens	MCF7	IC50	25410.0	nM	10.1016/j.bmcl.2015.05.017
Homo sapiens	MCF7	IC50	25410.0	nM	10.1016/j.bmcl.2016.12.029
Homo sapiens	MCF7	IC50	100000.0	nM	10.1016/j.ejmech.2020.112359
Homo sapiens	MCF7	Inhibition	94.0	%	10.1016/j.bmcl.2015.05.017
Homo sapiens	MCF7	Inhibition	nan	%	10.1016/j.ejmech.2018.10.045
Homo sapiens	MC-IXC	Activity	0.9	None	10.1073/pnas.0707498104
Homo sapiens	MDA-MB-134-VI	IC50	1607819.19	nM	10.6019/CHEMBL1201861
Homo sapiens	MDA-MB-157	Activity	1.059	None	10.1073/pnas.0707498104
Homo sapiens	MDA-MB-231	Activity	1.583	None	10.1073/pnas.0707498104
Homo sapiens	MDA-MB-231	EC50	1000.0	nM	10.1021/acs.jmedchem.6b00087
Homo sapiens	MDA-MB-231	IC50	22.3	nM	10.1016/j.bmc.2014.04.049
Homo sapiens	MDA-MB-231	IC50	2600.0	nM	10.1016/j.bmcl.2019.126710
Homo sapiens	MDA-MB-231	IC50	3700.0	nM	10.1016/j.bmcl.2019.126710
Homo sapiens	MDA-MB-231	IC50	3700.0	nM	10.1016/j.ejmech.2011.05.017
Homo sapiens	MDA-MB-231	IC50	4510.0	nM	10.1007/s00044-012-0170-3
Homo sapiens	MDA-MB-231	IC50	4510.0	nM	10.1016/j.bmcl.2011.03.031
Homo sapiens	MDA-MB-231	IC50	6000.0	nM	10.1016/j.bmcl.2017.03.018
Homo sapiens	MDA-MB-231	IC50	6980.0	nM	10.1016/j.ejmech.2017.07.033
Homo sapiens	MDA-MB-231	IC50	7400.0	nM	10.1016/j.bmcl.2016.06.077
Homo sapiens	MDA-MB-231	IC50	7400.0	nM	10.1016/j.ejmech.2016.04.025
Homo sapiens	MDA-MB-231	IC50	32000.0	nM	10.1016/j.bmcl.2017.07.029
Homo sapiens	MDA-MB-231	IC50	nan	None	10.1016/j.ejmech.2019.06.054
Homo sapiens	MDA-MB-231	TGI	84.0	%	10.1016/j.bmcl.2017.06.071
Homo sapiens	MDA-MB-361	Activity	1.364	None	10.1073/pnas.0707498104
Homo sapiens	MDA-MB-415	Activity	1.226	None	10.1073/pnas.0707498104
Homo sapiens	MDA-MB-435	GI50	2000.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	MDA-MB-435	IC50	9.7	nM	10.1016/j.bmc.2014.04.049
Homo sapiens	MDA-MB-435	IC50	9300.0	nM	10.1016/j.bmcl.2016.02.063
Homo sapiens	MDA-MB-435	Inhibition	nan	%	10.1016/j.bmcl.2013.04.031
Homo sapiens	MDA-MB-435	Inhibition	nan	%	10.1021/ml4004793
Homo sapiens	MDA-MB-453	Activity	0.947	None	10.1073/pnas.0707498104
Homo sapiens	MDA-MB-468	Activity	1.127	None	10.1073/pnas.0707498104
Homo sapiens	MDA-MB-468	IC50	6.1	nM	10.1016/j.bmc.2014.04.049
Homo sapiens	ME-180	Activity	1.011	None	10.1073/pnas.0707498104
Homo sapiens	MEG-01	IC50	1835.63	nM	10.6019/CHEMBL1201861
Homo sapiens	Melanocortin receptor 3	AC50	7799.9	nM	10.1038/s41467-023-40064-9
Homo sapiens	MEL-HO	Activity	0.96	None	10.1073/pnas.0707498104
Homo sapiens	MEL-JUSO	Activity	0.945	None	10.1073/pnas.0707498104
Homo sapiens	Membrane-associated progesterone receptor component 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Menin/Histone-lysine N-methyltransferase MLL	Potency	6309.6	nM	None
Homo sapiens	MeWo	Activity	1.109	None	10.1073/pnas.0707498104
Homo sapiens	MFE-280	Activity	1.184	None	10.1073/pnas.0707498104
Homo sapiens	MFE-296	Activity	0.844	None	10.1073/pnas.0707498104
Homo sapiens	MFH-ino	IC50	150608.09	nM	10.6019/CHEMBL1201861
Homo sapiens	MFM-223	IC50	1294064.09	nM	10.6019/CHEMBL1201861
Homo sapiens	MG-63	Activity	0.92	None	10.1073/pnas.0707498104
Homo sapiens	MHH-CALL-2	IC50	5767.19	nM	10.6019/CHEMBL1201861
Homo sapiens	MHH-NB-11	IC50	20552.08	nM	10.6019/CHEMBL1201861
Homo sapiens	MHH-PREB-1	IC50	5323.12	nM	10.6019/CHEMBL1201861
Homo sapiens	MIA PaCa-2	Activity	0.991	None	10.1073/pnas.0707498104
Homo sapiens	Microtubule-associated serine/threonine-protein kinase 1	Kd	200.0	nM	10.1038/nbt.1990
Homo sapiens	Microtubule-associated serine/threonine-protein kinase 1	Kd	200.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Midasin	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Misshapen-like kinase 1	Kd	29.0	nM	10.1038/nbt.1990
Homo sapiens	Misshapen-like kinase 1	Kd	29.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase 15	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase 15	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase 15	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase 15	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase 4	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase 6	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase 6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase 6	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase 6	Thermal melting change	2.4	degrees C	10.1073/pnas.0708800104
Homo sapiens	Mitogen-activated protein kinase 7	Kd	9900.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase 7	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase 7	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase 7	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 10	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 10	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 10	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	Kd	1300.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	Kd	1300.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	Kd	1300.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase 11	Kd	3097.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 12	Kd	100.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 13	Kd	95.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 13	Kd	95.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase 15	Kd	1300.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 15	Kd	1300.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase 2	Kd	57.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 2	Kd	57.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase 2	Kd	2387.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 3	Kd	220.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 3	Kd	220.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase 3	Kd	3264.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 4	Kd	3300.0	nM	10.1038/nbt1068
Homo sapiens	Mitogen-activated protein kinase kinase kinase 4	Kd	4800.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 4	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Mitogen-activated protein kinase kinase kinase 5	Thermal melting change	-0.6	degrees C	10.1073/pnas.0708800104
Homo sapiens	Mitogen-activated protein kinase kinase kinase 6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 6	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase 6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7	Kd	93.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 7	Kd	93.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	Kd	3400.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	Kd	3400.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase 9	Kd	3400.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 1	Kd	16.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 1	Kd	16.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 1	Kd	16.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 1	Kd	249.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 2	Kd	33.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 3	Kd	180.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 3	Kd	180.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 3	Kd	180.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 3	Kd	528.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	Kd	140.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	Kd	140.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 4	Kd	268.0	nM	10.1126/science.aan4368
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	41.0	nM	10.1038/nbt1358
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	41.0	nM	10.1038/nbt.1990
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	41.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	77.0	nM	10.1038/nbt1068
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	77.0	nM	10.1073/pnas.0707498104
Homo sapiens	Mitogen-activated protein kinase kinase kinase kinase 5	Kd	1194.0	nM	10.1126/science.aan4368
Homo sapiens	Mitotic checkpoint serine/threonine-protein kinase BUB1	Kd	3507.0	nM	10.1126/science.aan4368
Homo sapiens	Mixed lineage kinase 7	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Mixed lineage kinase 7	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Mixed lineage kinase 7	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Mixed lineage kinase 7	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	MKN-28	Activity	1.097	None	10.1073/pnas.0707498104
Homo sapiens	MKN-45	Activity	1.445	None	10.1073/pnas.0707498104
Homo sapiens	MKN-45	IC50	9250.0	nM	10.1016/j.ejmech.2020.113083
Homo sapiens	MKN-7	Activity	1.14	None	10.1073/pnas.0707498104
Homo sapiens	MKN-74	Activity	0.799	None	10.1073/pnas.0707498104
Homo sapiens	ML-2	IC50	2635.12	nM	10.6019/CHEMBL1201861
Homo sapiens	MLMA	IC50	16990.75	nM	10.6019/CHEMBL1201861
Homo sapiens	MMAC-SF	IC50	6109.49	nM	10.6019/CHEMBL1201861
Homo sapiens	MN-60	IC50	7540.88	nM	10.6019/CHEMBL1201861
Homo sapiens	Mo	IC50	999979.72	nM	10.6019/CHEMBL1201861
Homo sapiens	MOG-G-UVW	Activity	0.857	None	10.1073/pnas.0707498104
Homo sapiens	MOLM-13	Activity	-1.1	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	-0.6	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	-0.5	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	0.24	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	0.4	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	0.5	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	0.9	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	1.14	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	1.3	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	2.6	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	3.2	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	3.32	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	3.7	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	3.98	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	4.19	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	4.2	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	5.3	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	5.58	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	6.13	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	6.3	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	9.3	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	9.47	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	16.42	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	19.36	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	23.49	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	24.17	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	25.9	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	26.6	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	31.1	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	41.02	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	44.27	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	49.02	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	63.75	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	65.44	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	70.77	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	92.46	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	Activity	nan	None	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	EC50	14.3	nM	10.1016/j.ejmech.2020.112316
Homo sapiens	MOLM-13	GI50	54.0	nM	10.1021/acs.jmedchem.9b01229
Homo sapiens	MOLM-13	IC50	17.7	nM	10.1016/j.ejmech.2014.07.108
Homo sapiens	MOLM-13	IC50	69.6	nM	10.1021/acs.jmedchem.0c02247
Homo sapiens	MOLM-13	IC50	nan	None	10.1016/j.bmc.2010.05.021
Homo sapiens	MOLT-16	IC50	631.32	nM	10.6019/CHEMBL1201861
Homo sapiens	MOLT-4	IC50	3398.38	nM	10.6019/CHEMBL1201861
Homo sapiens	Monoamine oxidase A	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	MONO-MAC-6	IC50	33.8	nM	10.6019/CHEMBL1201861
Homo sapiens	MONO-MAC-6	IC50	5700.0	nM	10.1016/j.ejmech.2019.111719
Homo sapiens	Motilin receptor	AC50	7300.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	MPP-89	IC50	42058.56	nM	10.6019/CHEMBL1201861
Homo sapiens	MRK-nu-1	IC50	104990.83	nM	10.6019/CHEMBL1201861
Homo sapiens	MS-1	IC50	3837.78	nM	10.6019/CHEMBL1201861
Homo sapiens	MSTO-211H	Activity	0.953	None	10.1073/pnas.0707498104
Homo sapiens	MSTO-211H	IC50	31867.8	nM	10.6019/CHEMBL1201861
Homo sapiens	Multifunctional protein ADE2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Mu opioid receptor	AC50	4900.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Mu opioid receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Muscarinic acetylcholine receptor M1	AC50	2049.4	nM	10.1038/s41467-023-40064-9
Homo sapiens	Muscarinic acetylcholine receptor M2	AC50	7188.9	nM	10.1038/s41467-023-40064-9
Homo sapiens	Muscarinic acetylcholine receptor M2	AC50	10000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Muscarinic acetylcholine receptor M2	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Muscarinic acetylcholine receptor M3	AC50	1612.4	nM	10.1038/s41467-023-40064-9
Homo sapiens	Muscarinic acetylcholine receptor M4	AC50	10000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Muscarinic acetylcholine receptor M5	AC50	10000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Muscle, skeletal receptor tyrosine protein kinase	Kd	490.0	nM	10.1038/nbt1358
Homo sapiens	Muscle, skeletal receptor tyrosine protein kinase	Kd	490.0	nM	10.1038/nbt.1990
Homo sapiens	Muscle, skeletal receptor tyrosine protein kinase	Kd	490.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	MV4-11	Activity	0.29	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	0.32	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	0.5	%	10.1016/j.ejmech.2011.07.045
Homo sapiens	MV4-11	Activity	1.03	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	1.22	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	1.4	%	10.1016/j.ejmech.2011.07.045
Homo sapiens	MV4-11	Activity	1.71	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	2.53	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	2.68	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	2.69	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	2.79	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	3.91	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	5.86	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	6.58	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	8.55	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	9.64	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	12.8	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	13.27	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	26.11	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	32.53	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	60.29	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	66.78	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	68.1	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	80.1	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	89.41	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	98.36	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	Activity	nan	None	10.1016/j.bmcl.2009.07.024
Homo sapiens	MV4-11	Activity	nan	None	10.1021/jm9007533
Homo sapiens	MV4-11	GI50	1.0	nM	10.1021/acs.jmedchem.6b00200
Homo sapiens	MV4-11	IC50	0.2722	nM	10.6019/CHEMBL1201861
Homo sapiens	MV4-11	IC50	3.0	nM	10.1021/jm300042x
Homo sapiens	MV4-11	IC50	4.3	nM	10.1021/jm9007533
Homo sapiens	MV4-11	IC50	4.3	nM	10.1182/blood-2009-05-222034
Homo sapiens	MV4-11	IC50	8.0	nM	10.1021/acs.jmedchem.0c00696
Homo sapiens	MV4-11	IC50	9.0	nM	10.1016/j.bmc.2010.05.021
Homo sapiens	MV4-11	IC50	9.0	nM	10.1016/j.bmcl.2010.08.025
Homo sapiens	MV4-11	IC50	10.0	nM	10.1016/j.bmcl.2018.06.026
Homo sapiens	MV4-11	IC50	24.3	nM	10.1016/j.ejmech.2014.07.108
Homo sapiens	MV4-11	IC50	31.5	nM	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	IC50	38.5	nM	10.1016/j.ejmech.2016.12.038
Homo sapiens	MV4-11	IC50	54.0	nM	10.1021/acs.jmedchem.8b01714
Homo sapiens	MV4-11	Inhibition	nan	%	10.1021/jm9007533
Homo sapiens	MV4-11	Inhibition	nan	%	10.1182/blood-2009-05-222034
Homo sapiens	MV4-11	MED	10.0	mg/kg/day	10.1016/j.ejmech.2016.12.038
Homo sapiens	MV4-11	TGI	29.9	%	10.1021/acs.jmedchem.0c02247
Homo sapiens	MV4-11	TGI	81.01	%	10.1016/j.ejmech.2016.12.038
Homo sapiens	Myelin transcription factor 1	Activity	5.0	%	10.1016/j.ejmech.2012.06.007
Homo sapiens	Myelin transcription factor 1	IC50	nan	None	10.1016/j.ejmech.2012.06.007
Homo sapiens	Myosin-10	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Myosin-14	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Myosin IIIA	Kd	3100.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin IIIA	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Myosin IIIA	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Myosin-IIIB	Kd	4500.0	nM	10.1038/nbt1358
Homo sapiens	Myosin-IIIB	Kd	4500.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin-IIIB	Kd	4500.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Myosin light chain kinase	Kd	23.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin light chain kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	myosin light chain kinase 2	Kd	49.0	nM	10.1038/nbt1358
Homo sapiens	myosin light chain kinase 2	Kd	49.0	nM	10.1038/nbt.1990
Homo sapiens	myosin light chain kinase 2	Kd	49.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	myosin light chain kinase 2	Kd	57.0	nM	10.1038/nbt1068
Homo sapiens	myosin light chain kinase 2	Kd	57.0	nM	10.1073/pnas.0707498104
Homo sapiens	Myosin light chain kinase family member 4	Kd	15.0	nM	10.1038/nbt1358
Homo sapiens	Myosin light chain kinase family member 4	Kd	15.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin light chain kinase family member 4	Kd	15.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Myosin light chain kinase, smooth muscle	Kd	23.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Myosin light chain kinase, smooth muscle	Kd	280.0	nM	10.1038/nbt1358
Homo sapiens	Myosin light chain kinase, smooth muscle	Kd	280.0	nM	10.1038/nbt.1990
Homo sapiens	Myosin light chain kinase, smooth muscle	Kd	280.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Myosin light chain kinase, smooth muscle	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Myotonin-protein kinase	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Myotonin-protein kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Myotonin-protein kinase	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Myotonin-protein kinase	Thermal melting change	2.7	degrees C	10.1073/pnas.0708800104
Homo sapiens	MZ1-PC	IC50	7303.89	nM	10.6019/CHEMBL1201861
Homo sapiens	MZ2-MEL	IC50	15225.11	nM	10.6019/CHEMBL1201861
Homo sapiens	MZ7-mel	IC50	59766.18	nM	10.6019/CHEMBL1201861
Homo sapiens	NAD-dependent deacetylase sirtuin 1	Inhibition	10.0	%	10.1021/jm901055u
Homo sapiens	NAD-dependent deacetylase sirtuin 2	IC50	122700.0	nM	10.1021/jm901055u
Homo sapiens	NAD-dependent deacetylase sirtuin 3	Inhibition	26.4	%	10.1021/jm901055u
Homo sapiens	NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	NALM-6	IC50	2904.73	nM	10.6019/CHEMBL1201861
Homo sapiens	NB1	IC50	1961.17	nM	10.6019/CHEMBL1201861
Homo sapiens	NB10	IC50	1602160.0	nM	10.6019/CHEMBL1201861
Homo sapiens	NB13	IC50	9799.94	nM	10.6019/CHEMBL1201861
Homo sapiens	NB14	IC50	10927.65	nM	10.6019/CHEMBL1201861
Homo sapiens	NB17	IC50	60544.58	nM	10.6019/CHEMBL1201861
Homo sapiens	NB5	IC50	80719.32	nM	10.6019/CHEMBL1201861
Homo sapiens	NB6	IC50	101286.69	nM	10.6019/CHEMBL1201861
Homo sapiens	NB69	Activity	0.905	None	10.1073/pnas.0707498104
Homo sapiens	NB69	IC50	290226.31	nM	10.6019/CHEMBL1201861
Homo sapiens	NB7	IC50	27922.87	nM	10.6019/CHEMBL1201861
Homo sapiens	NCCIT	IC50	8717.45	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1048	Activity	0.941	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1092	IC50	342184.82	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1155	IC50	130531.69	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H128	IC50	13072.31	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1299	Activity	1.066	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1299	EC50	1540.0	nM	10.1021/acsmedchemlett.8b00596
Homo sapiens	NCI-H1304	IC50	8206.61	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1355	IC50	7458.04	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1395	IC50	486680.57	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1417	IC50	1837567.56	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1436	IC50	613542.78	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1437	Activity	1.141	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1522	IC50	779702.16	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1563	Activity	0.901	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1573	Activity	0.895	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1581	Activity	0.956	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1581	IC50	18086.59	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1623	Activity	0.969	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1648	IC50	9138.34	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1650	Activity	0.896	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1650	IC50	29017.58	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1651	Activity	0.91	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1666	Activity	1.035	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1693	Activity	0.873	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1694	IC50	13114.4	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1703	Activity	0.365	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1734	Activity	1.046	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1755	Activity	0.957	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1770	IC50	14536.94	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1792	Activity	0.886	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1793	Activity	0.812	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1838	IC50	101554.95	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H187	IC50	231956.07	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1882	IC50	17983.42	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1963	IC50	403364.25	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H1975	Activity	0.749	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H1975	EC50	1000.0	nM	10.1021/acs.jmedchem.6b00087
Homo sapiens	NCI-H2009	Activity	0.945	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H2029	Activity	1.168	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H2030	Activity	1.127	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H2081	IC50	228219.53	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2087	Activity	0.82	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H209	IC50	8116.52	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2107	IC50	11598.42	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2122	Activity	0.888	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H2126	IC50	104941.07	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2141	IC50	38084.3	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2170	Activity	0.552	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H2171	IC50	123449.6	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2196	Activity	0.941	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H2196	IC50	108550.34	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2228	Activity	0.852	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H226	IC50	139254.61	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H23	Activity	0.915	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H23	IC50	31106.26	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H2342	Activity	1.026	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H2347	Activity	0.748	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H2405	Activity	0.796	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H2452	Activity	1.198	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H322M	IC50	116336.87	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H345	IC50	295123.82	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H358	Activity	0.951	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H441	Activity	1.035	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H446	IC50	27494.64	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H460	Activity	0.86	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H460	IC50	2700.0	nM	10.1016/j.ejmech.2011.05.017
Homo sapiens	NCI-H460	IC50	4000.0	nM	10.1016/j.bmc.2010.05.021
Homo sapiens	NCI-H460	IC50	4310.0	nM	10.1016/j.ejmech.2014.05.051
Homo sapiens	NCI-H460	TGI	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	NCI-H510A	IC50	24127.78	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H520	Activity	0.89	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H522	Activity	0.849	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H524	IC50	58569.55	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H526	IC50	1010.0	nM	10.1016/j.ejmech.2014.05.051
Homo sapiens	NCI-H526	IC50	55135.4	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H596	Activity	0.809	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H630	Activity	1.023	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H64	IC50	1239989.26	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H647	Activity	1.01	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H661	Activity	1.013	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H69	IC50	200770.41	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H716	IC50	133966.8	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H719	IC50	16916.14	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H720	IC50	231837.57	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H727	Activity	1.041	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H727	IC50	10120.0	nM	10.1021/acsmedchemlett.7b00192
Homo sapiens	NCI-H747	IC50	28919.47	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H748	IC50	479317.88	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H810	Activity	1.079	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H82	IC50	7378.5	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-H838	Activity	0.91	None	10.1073/pnas.0707498104
Homo sapiens	NCI-H889	IC50	351121.04	nM	10.6019/CHEMBL1201861
Homo sapiens	NCI-N87	Activity	1.145	None	10.1073/pnas.0707498104
Homo sapiens	NEC8	IC50	12688.74	nM	10.6019/CHEMBL1201861
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	100.0	nM	10.1016/j.ejmech.2020.112421
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	100.0	nM	10.1038/nbt1358
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	100.0	nM	10.1038/nbt.1990
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	100.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	220.0	nM	10.1038/nbt1068
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	220.0	nM	10.1073/pnas.0707498104
Homo sapiens	Nerve growth factor receptor Trk-A	Kd	1940.0	nM	10.1126/science.aan4368
Homo sapiens	Neuronal acetylcholine receptor protein alpha-4 subunit	AC50	7300.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Neuropeptide Y receptor type 1	AC50	6900.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	Kd	590.0	nM	10.1038/nbt1358
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	Kd	590.0	nM	10.1038/nbt.1990
Homo sapiens	Neurotrophic tyrosine kinase receptor type 2	Kd	590.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	NH-12	IC50	43935.91	nM	10.6019/CHEMBL1201861
Homo sapiens	NH-6	Activity	0.961	None	10.1073/pnas.0707498104
Homo sapiens	Nitric-oxide synthase, endothelial	Inhibition	nan	%	10.1016/j.bmcl.2011.09.022
Homo sapiens	NKM-1	IC50	98.52	nM	10.6019/CHEMBL1201861
Homo sapiens	NMC-G1	IC50	27182.16	nM	10.6019/CHEMBL1201861
Homo sapiens	no-10	IC50	21026.45	nM	10.6019/CHEMBL1201861
Homo sapiens	no-11	IC50	7775.57	nM	10.6019/CHEMBL1201861
Homo sapiens	NOMO-1	IC50	4336.99	nM	10.6019/CHEMBL1201861
Homo sapiens	Non-receptor tyrosine-protein kinase TNK1	Kd	680.0	nM	10.1038/nbt1358
Homo sapiens	Non-receptor tyrosine-protein kinase TNK1	Kd	680.0	nM	10.1038/nbt.1990
Homo sapiens	Non-receptor tyrosine-protein kinase TNK1	Kd	680.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Non-receptor tyrosine-protein kinase TNK1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Norepinephrine transporter	AC50	1755.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	NOS-1	IC50	15.3	nM	10.6019/CHEMBL1201861
Homo sapiens	NT-3 growth factor receptor	Kd	5100.0	nM	10.1038/nbt1358
Homo sapiens	NT-3 growth factor receptor	Kd	5100.0	nM	10.1038/nbt.1990
Homo sapiens	NT-3 growth factor receptor	Kd	5100.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	NTERA-2-cl-D1	IC50	17857.2	nM	10.6019/CHEMBL1201861
Homo sapiens	NUAK family SNF1-like kinase 1	IC50	48.0	nM	10.1021/acs.jmedchem.0c00533
Homo sapiens	NUAK family SNF1-like kinase 1	Kd	48.0	nM	10.1038/nbt1358
Homo sapiens	NUAK family SNF1-like kinase 1	Kd	48.0	nM	10.1038/nbt.1990
Homo sapiens	NUAK family SNF1-like kinase 1	Kd	48.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	NUAK family SNF1-like kinase 2	Kd	150.0	nM	10.1038/nbt1358
Homo sapiens	NUAK family SNF1-like kinase 2	Kd	150.0	nM	10.1038/nbt.1990
Homo sapiens	NUAK family SNF1-like kinase 2	Kd	150.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	NUAK family SNF1-like kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Nuclear receptor subfamily 1 group I member 3	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Nuclear receptor subfamily 2 group C member 2	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Nucleolar GTP-binding protein 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	NUGC-3	Activity	0.75	None	10.1073/pnas.0707498104
Homo sapiens	NUGC-4	Activity	1.0	None	10.1073/pnas.0707498104
Homo sapiens	OAW-28	Activity	0.951	None	10.1073/pnas.0707498104
Homo sapiens	OAW-42	Activity	0.926	None	10.1073/pnas.0707498104
Homo sapiens	Obg-like ATPase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	OCI-AML2	IC50	1368.51	nM	10.6019/CHEMBL1201861
Homo sapiens	OCI-AML-5	IC50	14.0	nM	10.1021/acs.jmedchem.0c00696
Homo sapiens	OCUB-M	IC50	8565.08	nM	10.6019/CHEMBL1201861
Homo sapiens	OE19	Activity	1.055	None	10.1073/pnas.0707498104
Homo sapiens	OE33	Activity	1.069	None	10.1073/pnas.0707498104
Homo sapiens	OMC-1	IC50	73153.43	nM	10.6019/CHEMBL1201861
Homo sapiens	ONS-76	IC50	9810.16	nM	10.6019/CHEMBL1201861
Homo sapiens	OPM-2	IC50	3059.54	nM	10.6019/CHEMBL1201861
Homo sapiens	OS-RC-2	IC50	4873.1	nM	10.6019/CHEMBL1201861
Homo sapiens	OV-1063	Activity	0.858	None	10.1073/pnas.0707498104
Homo sapiens	OVCAR-3	GI50	3200.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	OVCAR-4	IC50	8503.51	nM	10.6019/CHEMBL1201861
Homo sapiens	OVCAR-5	Activity	1.092	None	10.1073/pnas.0707498104
Homo sapiens	OVCAR-8	Activity	0.893	None	10.1073/pnas.0707498104
Homo sapiens	P30-OHK	IC50	151373.0	nM	10.6019/CHEMBL1201861
Homo sapiens	P31-FUJ	IC50	1224725.48	nM	10.6019/CHEMBL1201861
Homo sapiens	PA-1	Activity	0.973	None	10.1073/pnas.0707498104
Homo sapiens	PANC-1	Activity	1.158	None	10.1073/pnas.0707498104
Homo sapiens	PAS domain-containing serine/threonine-protein kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	PBMC	IC50	46300.0	nM	10.1016/j.ejmech.2019.111719
Homo sapiens	PC-14	Activity	0.841	None	10.1073/pnas.0707498104
Homo sapiens	PC-3	Activity	1.014	None	10.1073/pnas.0707498104
Homo sapiens	PC-3	GI	10.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	PC-3	IC50	25100.0	nM	10.1016/j.ejmech.2011.10.009
Homo sapiens	PC-3	IC50	nan	None	10.1016/j.ejmech.2019.06.094
Homo sapiens	PC-9	Activity	0.846	None	10.1073/pnas.0707498104
Homo sapiens	PC-9	IC50	10970.0	nM	10.1016/j.bmcl.2012.03.061
Homo sapiens	PDZ-binding kinase	Thermal melting change	0.4	degrees C	10.1073/pnas.0708800104
Homo sapiens	Peripheral plasma membrane protein CASK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Peroxisomal acyl-coenzyme A oxidase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Peroxisomal acyl-coenzyme A oxidase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Peroxisome proliferator-activated receptor alpha	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	PF-382	IC50	3445.7	nM	10.6019/CHEMBL1201861
Homo sapiens	P-glycoprotein 1	Ratio	4.183	None	10.1021/acs.jmedchem.0c02011
Homo sapiens	Phenylalanine--tRNA ligase beta subunit	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Phosphatidylethanolamine-binding protein 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing beta polypeptide	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing beta polypeptide	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing subunit gamma	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing subunit gamma	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha	Kd	5400.0	nM	10.1038/nbt1358
Homo sapiens	Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha	Kd	5400.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha	Kd	5400.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Phosphatidylinositol-4-phosphate 5-kinase type-1 gamma	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 beta	Kd	39.0	nM	10.1038/nbt1358
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 beta	Kd	39.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 beta	Kd	39.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 gamma	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Phosphatidylinositol-5-phosphate 4-kinase type-2 gamma	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Phosphodiesterase 3A	AC50	17999.9	nM	10.1038/s41467-023-40064-9
Homo sapiens	Phosphodiesterase 4D	AC50	9800.1	nM	10.1038/s41467-023-40064-9
Homo sapiens	Phosphofructokinase platelet type	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Phosphorylase kinase gamma subunit 1	Kd	5.5	nM	10.1038/nbt1358
Homo sapiens	Phosphorylase kinase gamma subunit 1	Kd	5.5	nM	10.1038/nbt.1990
Homo sapiens	Phosphorylase kinase gamma subunit 1	Kd	5.5	nM	10.1182/blood-2009-05-222034
Homo sapiens	Phosphorylase kinase gamma subunit 1	Kd	70.0	nM	10.1038/nbt1068
Homo sapiens	Phosphorylase kinase gamma subunit 1	Kd	70.0	nM	10.1073/pnas.0707498104
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	5.9	nM	10.1038/nbt1358
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	5.9	nM	10.1038/nbt.1990
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	5.9	nM	10.1182/blood-2009-05-222034
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	39.0	nM	10.1038/nbt1068
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	39.0	nM	10.1073/pnas.0707498104
Homo sapiens	Phosphorylase kinase gamma subunit 2	Kd	661.0	nM	10.1126/science.aan4368
Homo sapiens	Phosphorylase kinase gamma subunit 2	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	PI3-kinase p110-alpha subunit	IC50	11000.0	nM	10.1038/nchembio.117
Homo sapiens	PI3-kinase p110-alpha subunit	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	PI3-kinase p110-alpha subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PI3-kinase p110-alpha subunit	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	PI3-kinase p110-beta subunit	IC50	50000.0	nM	10.1038/nchembio.117
Homo sapiens	PI3-kinase p110-beta subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PI3-kinase p110-beta subunit	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	PI3-kinase p110-delta subunit	IC50	12000.0	nM	10.1038/nchembio.117
Homo sapiens	PI3-kinase p110-delta subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PI3-kinase p110-delta subunit	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	PI3-kinase p110-gamma subunit	IC50	13000.0	nM	10.1038/nchembio.117
Homo sapiens	PI3-kinase p110-gamma subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PI3-kinase p110-gamma subunit	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	PI4-kinase beta subunit	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PI4-kinase beta subunit	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	PITSLRE serine/threonine-protein kinase CDC2L2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Plasma	Stability	102.3	%	10.1021/acs.jmedchem.6b01266
Homo sapiens	Platelet-derived growth factor receptor	IC50	80.0	nM	10.1016/j.bmcl.2012.02.068
Homo sapiens	Platelet-derived growth factor receptor alpha	GI50	30.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Platelet-derived growth factor receptor alpha	GI50	631.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Platelet-derived growth factor receptor alpha	IC50	6.9	nM	10.1021/acs.jmedchem.0c02167
Homo sapiens	Platelet-derived growth factor receptor alpha	IC50	27.3	nM	10.1021/acs.jmedchem.0c02247
Homo sapiens	Platelet-derived growth factor receptor alpha	IC50	130.0	nM	10.1016/j.ejmech.2016.12.038
Homo sapiens	Platelet-derived growth factor receptor alpha	Inhibition	68.4	%	10.1016/j.bmcl.2014.11.070
Homo sapiens	Platelet-derived growth factor receptor alpha	Inhibition	71.4	%	10.1016/j.bmc.2018.09.027
Homo sapiens	Platelet-derived growth factor receptor alpha	Inhibition	71.4	%	10.1016/j.bmcl.2014.10.078
Homo sapiens	Platelet-derived growth factor receptor alpha	Inhibition	71.4	%	10.1021/acs.jmedchem.0c02254
Homo sapiens	Platelet-derived growth factor receptor alpha	Inhibition	93.0	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Platelet-derived growth factor receptor alpha	Inhibition	94.0	%	10.1016/j.ejmech.2017.04.039
Homo sapiens	Platelet-derived growth factor receptor alpha	Kd	0.79	nM	10.1038/nbt1358
Homo sapiens	Platelet-derived growth factor receptor alpha	Kd	0.79	nM	10.1038/nbt.1990
Homo sapiens	Platelet-derived growth factor receptor alpha	Kd	0.79	nM	10.1182/blood-2009-05-222034
Homo sapiens	Platelet-derived growth factor receptor beta	GI50	114.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	2.0	nM	10.1021/acs.jmedchem.6b01266
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	2.0	nM	10.1021/jm0204183
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	3.9	nM	10.1021/acs.jmedchem.0c02167
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	9.0	nM	10.1021/jm101036c
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	10.5	nM	10.1021/acs.jmedchem.0c02247
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	10.6	nM	10.1016/j.bmcl.2013.08.037
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	17.0	nM	10.1016/j.bmcl.2010.08.025
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	55.0	nM	10.1021/jm901132v
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	83.1	nM	10.1016/j.bmc.2014.04.049
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	83.1	nM	10.1016/j.bmc.2015.03.061
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	83.1	nM	10.1016/j.bmc.2016.11.026
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	83.1	nM	10.1016/j.bmc.2021.116061
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	83.1	nM	10.1016/j.bmcl.2018.07.039
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	12200.0	nM	10.1016/j.bmc.2010.03.052
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	12200.0	nM	10.1016/j.bmc.2010.05.049
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	12200.0	nM	10.1016/j.bmc.2011.11.058
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	83100.0	nM	10.1016/j.bmc.2012.05.068
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	83100.0	nM	10.1016/j.bmc.2012.12.045
Homo sapiens	Platelet-derived growth factor receptor beta	IC50	83100.0	nM	10.1016/j.bmc.2013.01.040
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	70.6	%	10.1016/j.bmc.2018.09.027
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	70.6	%	10.1016/j.bmcl.2014.10.078
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	70.6	%	10.1021/acs.jmedchem.0c02254
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	75.7	%	10.1016/j.ejmech.2018.09.032
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	76.1	%	10.1016/j.ejmech.2021.113333
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	80.2	%	10.1016/j.bmcl.2014.11.070
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	82.1	%	10.1016/j.bmcl.2012.09.043
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	82.1	%	10.1016/j.ejmech.2012.09.021
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	90.6	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Platelet-derived growth factor receptor beta	Inhibition	97.0	%	10.1016/j.ejmech.2017.04.039
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	0.075	nM	10.1038/nbt1358
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	0.075	nM	10.1038/nbt.1990
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	0.075	nM	10.1182/blood-2009-05-222034
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	0.2	nM	10.1073/pnas.0707498104
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	0.21	nM	10.1038/nbt1068
Homo sapiens	Platelet-derived growth factor receptor beta	Kd	4.0	nM	10.1126/science.aan4368
Homo sapiens	Platelet-derived growth factor receptor beta	Ki	8.0	nM	10.1016/j.ejmech.2014.05.051
Homo sapiens	Pregnane X receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Prelamin-A/C	Potency	7079.5	nM	None
Homo sapiens	Probable ATP-dependent RNA helicase DDX6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Progesterone receptor	AC50	1700.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Protein delta homolog 1	Kd	100.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Protein delta homolog 1	Ki	6.3	nM	10.1021/acs.jmedchem.8b00370
Homo sapiens	Protein kinase C alpha	Kd	6000.0	nM	10.1038/nbt1068
Homo sapiens	Protein kinase C alpha	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Protein kinase C alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C beta	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Protein kinase C beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C delta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C delta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C delta	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Protein kinase C delta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C epsilon	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C epsilon	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C epsilon	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Protein kinase C eta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C eta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C eta	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Protein kinase C iota	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C iota	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C mu	Kd	310.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C mu	Kd	310.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C mu	Kd	310.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Protein kinase C nu	Kd	280.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C nu	Kd	280.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C nu	Kd	280.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Protein kinase C nu	Kd	1645.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C theta	Kd	4300.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase C theta	Kd	4300.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase C theta	Kd	4300.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Protein kinase C theta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase C zeta	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Protein kinase C zeta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase N1	Kd	710.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase N1	Kd	710.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase N1	Kd	710.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Protein kinase N1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein kinase N2	Kd	1300.0	nM	10.1038/nbt1358
Homo sapiens	Protein kinase N2	Kd	1300.0	nM	10.1038/nbt.1990
Homo sapiens	Protein kinase N2	Kd	1300.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Protein kinase N2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein tyrosine kinase 2 beta	Kd	82.0	nM	10.1038/nbt1358
Homo sapiens	Protein tyrosine kinase 2 beta	Kd	82.0	nM	10.1038/nbt.1990
Homo sapiens	Protein tyrosine kinase 2 beta	Kd	82.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Protein tyrosine kinase 2 beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Protein tyrosine kinase 2 beta	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Activity	99.6	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Activity	100.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Kd	26.0	nM	10.1038/nbt1358
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Kd	26.0	nM	10.1038/nbt.1990
Homo sapiens	Proto-oncogene tyrosine-protein kinase MER	Kd	26.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Proto-oncogene tyrosine-protein kinase ROS	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	PSN1	IC50	1506.76	nM	10.6019/CHEMBL1201861
Homo sapiens	Putative heat shock protein HSP 90-beta 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Putative uncharacterized serine/threonine-protein kinase SgK110	Kd	1900.0	nM	10.1038/nbt.1990
Homo sapiens	Putative uncharacterized serine/threonine-protein kinase SgK110	Kd	1900.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Pyridoxal kinase	Kd	6021.0	nM	10.1126/science.aan4368
Homo sapiens	QIMR-WIL	IC50	3633.91	nM	10.6019/CHEMBL1201861
Homo sapiens	Quinone reductase 2	Kd	4022.0	nM	10.1126/science.aan4368
Homo sapiens	Rab-like protein 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Raji	IC50	19956.54	nM	10.6019/CHEMBL1201861
Homo sapiens	Ramos-2G6-4C10	IC50	11265.02	nM	10.6019/CHEMBL1201861
Homo sapiens	Ras-related protein Rab-10	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ras-related protein Rab-27A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ras-related protein Rab-6A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	RCC10RGB	IC50	366741.78	nM	10.6019/CHEMBL1201861
Homo sapiens	RCC4	IC50	4000.0	nM	10.1016/j.bmcl.2017.03.018
Homo sapiens	RCM-1	Activity	0.83	None	10.1073/pnas.0707498104
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 1	Kd	370.0	nM	10.1021/acs.jmedchem.2c01518
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 1	Kd	370.0	nM	10.1038/nbt1358
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 1	Kd	370.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 1	Kd	370.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 4	Kd	2100.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor-interacting serine/threonine-protein kinase 4	Kd	2100.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Inhibition	nan	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Inhibition	nan	%	10.1016/j.ejmech.2018.09.032
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Receptor protein-tyrosine kinase erbB-2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor protein-tyrosine kinase erbB-4	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Receptor tyrosine-protein kinase erbB-3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Receptor tyrosine-protein kinase erbB-3	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	REH	IC50	12649.81	nM	10.6019/CHEMBL1201861
Homo sapiens	RERF-LC-MS	Activity	0.983	None	10.1073/pnas.0707498104
Homo sapiens	Retinoic acid receptor alpha	AC50	3000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Retinoic acid receptor alpha	AC50	10000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Retinoic acid receptor beta	AC50	3000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Retinoic acid receptor beta	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Retinoic acid receptor gamma	AC50	10000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Retinoic acid receptor gamma	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	RH-1	IC50	187317.12	nM	10.6019/CHEMBL1201861
Homo sapiens	Rho-associated protein kinase 1	Kd	460.0	nM	10.1038/nbt.1990
Homo sapiens	Rho-associated protein kinase 1	Kd	460.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Rho-associated protein kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Rho-associated protein kinase 2	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Rho-associated protein kinase 2	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	Rho-associated protein kinase 2	Kd	140.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Rho-associated protein kinase 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Rhodopsin kinase	Kd	290.0	nM	10.1038/nbt.1990
Homo sapiens	Rhodopsin kinase	Kd	290.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase 1	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Ribosomal protein S6 kinase 1	Kd	48.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase 1	Kd	200.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Ribosomal protein S6 kinase alpha 1	IC50	131.3	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	96.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	140.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	580.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	2675.0	nM	10.1126/science.aan4368
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	5000.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 1	Kd	5000.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	17.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	17.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	28.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	58.0	nM	10.1038/nbt1068
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	58.0	nM	10.1073/pnas.0707498104
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	1700.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	8400.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 2	Kd	8400.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 3	IC50	183.9	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	55.0	nM	10.1038/nbt1068
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	55.0	nM	10.1073/pnas.0707498104
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	580.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	580.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	1696.0	nM	10.1126/science.aan4368
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Kd	2000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Thermal melting change	7.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	Ribosomal protein S6 kinase alpha 3	Thermal melting change	8.6	degrees C	10.1073/pnas.0708800104
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	96.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	96.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	140.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	572.0	nM	10.1126/science.aan4368
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	2000.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	2000.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 4	Kd	5000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	17.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	28.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	28.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	250.0	nM	10.1038/nbt1068
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	250.0	nM	10.1073/pnas.0707498104
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	1122.0	nM	10.1126/science.aan4368
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	1700.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	1700.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 5	Kd	8400.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	2400.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	2400.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	2400.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Ribosomal protein S6 kinase alpha 6	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	RKO	IC50	44125.24	nM	10.6019/CHEMBL1201861
Homo sapiens	RL	IC50	890094.82	nM	10.6019/CHEMBL1201861
Homo sapiens	RL95-2	IC50	2111.37	nM	10.6019/CHEMBL1201861
Homo sapiens	RNA cytidine acetyltransferase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	RO82-W-1	Activity	0.952	None	10.1073/pnas.0707498104
Homo sapiens	RPMI-6666	IC50	3541.71	nM	10.6019/CHEMBL1201861
Homo sapiens	RPMI-7951	Activity	0.81	None	10.1073/pnas.0707498104
Homo sapiens	RPMI-8226	IC50	7507.39	nM	10.6019/CHEMBL1201861
Homo sapiens	RPMI 8402	IC50	2336.18	nM	10.6019/CHEMBL1201861
Homo sapiens	RPMI-8866	IC50	75234.81	nM	10.6019/CHEMBL1201861
Homo sapiens	RS4-11	IC50	2179.24	nM	10.6019/CHEMBL1201861
Homo sapiens	RT-112	Activity	0.681	None	10.1073/pnas.0707498104
Homo sapiens	RT-4	Activity	1.033	None	10.1073/pnas.0707498104
Homo sapiens	RVH-421	Activity	1.059	None	10.1073/pnas.0707498104
Homo sapiens	RXF 393	IC50	11483.43	nM	10.6019/CHEMBL1201861
Homo sapiens	S-117	Activity	1.043	None	10.1073/pnas.0707498104
Homo sapiens	S-adenosylmethionine synthase isoform type-2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	SAOS-2	Activity	0.945	None	10.1073/pnas.0707498104
Homo sapiens	SBC-1	IC50	738121.17	nM	10.6019/CHEMBL1201861
Homo sapiens	SBC-3	Activity	1.075	None	10.1073/pnas.0707498104
Homo sapiens	SBC-5	Activity	0.992	None	10.1073/pnas.0707498104
Homo sapiens	SCaBER	Activity	0.917	None	10.1073/pnas.0707498104
Homo sapiens	SCC-15	IC50	127049.15	nM	10.6019/CHEMBL1201861
Homo sapiens	SCC-3	IC50	2828.91	nM	10.6019/CHEMBL1201861
Homo sapiens	SCCH-26	Activity	1.098	None	10.1073/pnas.0707498104
Homo sapiens	SCH	Activity	1.025	None	10.1073/pnas.0707498104
Homo sapiens	SCH	IC50	32848.46	nM	10.6019/CHEMBL1201861
Homo sapiens	SCLC-21H	Activity	1.033	None	10.1073/pnas.0707498104
Homo sapiens	SCLC-21H	IC50	1214121.44	nM	10.6019/CHEMBL1201861
Homo sapiens	Septin-9	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine-protein kinase ATR	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase 10	Kd	19.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 10	Kd	19.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 10	Kd	19.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 10	Kd	640.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 10	Kd	3965.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase 10	Thermal melting change	11.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase 11	Kd	38.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 11	Kd	38.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 11	Kd	38.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 11	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase 16	Kd	250.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 16	Kd	250.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 16	Kd	250.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 16	Kd	360.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 16	Kd	360.0	nM	10.1073/pnas.0707498104
Homo sapiens	Serine/threonine-protein kinase 16	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase 16	Thermal melting change	3.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase 17A	Kd	1.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 17A	Kd	1.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 17A	Kd	1.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 17A	Kd	21.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 17A	Kd	21.0	nM	10.1073/pnas.0707498104
Homo sapiens	Serine/threonine-protein kinase 17A	Thermal melting change	8.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase 17B	Kd	110.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 17B	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 17B	Kd	110.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 17B	Kd	220.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 17B	Kd	220.0	nM	10.1073/pnas.0707498104
Homo sapiens	Serine/threonine-protein kinase 2	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Serine/threonine-protein kinase 2	Kd	56.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 2	Kd	56.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 2	Kd	56.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 2	Kd	81.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 2	Kd	81.0	nM	10.1073/pnas.0707498104
Homo sapiens	Serine/threonine-protein kinase 2	Kd	3184.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase 2	Thermal melting change	6.5	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase 24	Kd	63.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 24	Kd	63.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 24	Kd	63.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 24	Kd	4084.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase 25	Kd	290.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 25	Kd	290.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 25	Kd	290.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 25	Thermal melting change	nan	None	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase 32A	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 32B	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 32B	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 32B	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 32C	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 32C	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 32C	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 33	Kd	17.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 33	Kd	17.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 33	Kd	17.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 35	Kd	1300.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 35	Kd	1300.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 36	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 36	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 36	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 36	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 38	Kd	410.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 38	Kd	410.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 38	Thermal melting change	5.6	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase 38-like	Kd	970.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase 38-like	Kd	970.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase 38-like	Kd	970.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase 38-like	Kd	1500.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase 38-like	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase AKT	IC50	10000.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	Serine/threonine-protein kinase AKT	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase AKT	Inhibition	nan	%	10.1021/acs.jmedchem.9b00280
Homo sapiens	Serine/threonine-protein kinase AKT	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase AKT	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase AKT	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase AKT	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase AKT2	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase AKT2	Kd	2700.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase AKT2	Kd	2700.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase AKT2	Kd	2700.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase AKT2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase AKT3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase AKT3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase AKT3	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase AKT3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase A-Raf	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Aurora-A	IC50	1837.0	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Kd	1700.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Kd	1700.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Kd	1700.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Kd	6600.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase Aurora-A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Aurora-B	IC50	1500.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Kd	380.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Kd	380.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Kd	380.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase Aurora-B	Kd	1817.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Kd	220.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Kd	220.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Kd	220.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Kd	310.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase Aurora-C	Kd	310.0	nM	10.1073/pnas.0707498104
Homo sapiens	Serine/threonine-protein kinase B-raf	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase B-raf	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase B-raf	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase B-raf	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Chk1	IC50	77.27	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Serine/threonine-protein kinase Chk1	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase Chk1	Kd	300.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Chk1	Kd	300.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Chk1	Kd	300.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase Chk1	Kd	3294.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Chk1	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	Serine/threonine-protein kinase Chk2	IC50	16.84	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Serine/threonine-protein kinase Chk2	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase Chk2	Kd	7.1	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase Chk2	Kd	10.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Chk2	Thermal melting change	12.9	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Kd	410.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Kd	410.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Kd	410.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Kd	640.0	nM	10.1073/pnas.0707498104
Homo sapiens	Serine/threonine-protein kinase c-TAK1	Kd	2567.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase D2	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase D2	Kd	380.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase D2	Kd	380.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase D2	Kd	380.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase D2	Kd	1125.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase DCLK1	Kd	370.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase DCLK1	Kd	370.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase DCLK1	Kd	370.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase DCLK2	Kd	2700.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase DCLK2	Kd	2700.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase DCLK2	Kd	2700.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase DCLK3	Kd	110.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase DCLK3	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase DCLK3	Kd	110.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE1	Kd	600.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE1	Kd	600.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase/endoribonuclease IRE2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	20.0	nM	10.1021/acs.jmedchem.1c00302
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	20.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	20.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	20.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	120.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	120.0	nM	10.1073/pnas.0707498104
Homo sapiens	Serine/threonine-protein kinase GAK	Kd	1287.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase ICK	Kd	470.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase ICK	Kd	470.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase ICK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase ILK-1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase LATS1	Kd	630.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase LATS1	Kd	630.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase LATS1	Kd	630.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase LATS1	Kd	743.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase LATS2	Kd	460.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase LATS2	Kd	460.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase LATS2	Kd	460.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase MAK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MAK	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase MARK1	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase MARK1	Kd	1200.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MARK1	Kd	1200.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MARK1	Kd	1200.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase MRCK-A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase MRCK beta	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MRCK beta	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MRCK beta	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase MRCK beta	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase MRCK gamma	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MRCK gamma	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MRCK gamma	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase MRCK gamma	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	19.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	19.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	19.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	100.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	100.0	nM	10.1073/pnas.0707498104
Homo sapiens	Serine/threonine-protein kinase MST1	Kd	1329.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase MST1	Thermal melting change	0.5	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase MST2	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase MST2	Kd	56.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MST2	Kd	56.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MST2	Kd	56.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase MST2	Kd	2403.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase MST4	Kd	340.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase MST4	Kd	340.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase MST4	Kd	340.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase MST4	Kd	2234.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase MST4	Thermal melting change	-0.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase MST4	Thermal melting change	4.7	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase mTOR	IC50	50000.0	nM	10.1038/nchembio.117
Homo sapiens	Serine/threonine-protein kinase mTOR	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase N3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Nek1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Nek1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Nek1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase Nek1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Nek11	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK2	IC50	12000.0	nM	10.1074/jbc.m609721200
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	500.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	500.0	nM	10.1073/pnas.0707498104
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	1400.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	1400.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	1400.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase NEK2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase NEK2	Thermal melting change	-0.4	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase Nek3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Nek3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase Nek4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Nek5	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase Nek5	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Nek5	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase NEK6	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase NEK6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK6	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase NEK6	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase NEK6	Thermal melting change	3.4	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase NEK7	Kd	4100.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase NEK7	Kd	4100.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK7	Kd	4100.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase NEK7	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase NEK9	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase NEK9	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NEK9	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase NEK9	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase NEK9	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase NIM1	Kd	850.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase NIM1	Kd	850.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine protein kinase NLK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine protein kinase NLK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine protein kinase NLK	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine protein kinase NLK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase OSR1	Kd	530.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase OSR1	Kd	530.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase OSR1	Thermal melting change	3.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PAK 1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK 1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PAK 1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK 2	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase PAK 2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PAK 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PAK 3	Kd	16.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK 3	Kd	16.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 3	Kd	16.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PAK 3	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK 4	IC50	569.2	nM	10.1016/j.bmc.2017.04.047
Homo sapiens	Serine/threonine-protein kinase PAK 4	IC50	569.2	nM	10.1016/j.ejmech.2021.113334
Homo sapiens	Serine/threonine-protein kinase PAK 4	Kd	2300.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK 4	Kd	2300.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK 4	Kd	2300.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PAK 4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PAK 4	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK 4	Ki	500.0	nM	10.1016/j.bmc.2017.04.047
Homo sapiens	Serine/threonine-protein kinase PAK 4	Thermal melting change	3.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PAK6	Kd	2400.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK6	Kd	2400.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK6	Kd	2400.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PAK6	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK6	Ki	500.0	nM	10.1016/j.bmc.2017.04.047
Homo sapiens	Serine/threonine-protein kinase PAK6	Thermal melting change	3.5	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PAK7	Kd	640.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PAK7	Kd	640.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PAK7	Kd	640.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PAK7	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PAK7	Ki	500.0	nM	10.1016/j.bmc.2017.04.047
Homo sapiens	Serine/threonine-protein kinase PAK7	Thermal melting change	1.7	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	130.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	130.0	nM	10.1073/pnas.0707498104
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	150.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	150.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	150.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Kd	2353.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-1	Thermal melting change	-0.2	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-2	Kd	1200.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-2	Kd	1200.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-2	Kd	1200.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-2	Kd	2880.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-3	Kd	1700.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-3	Kd	1700.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-3	Kd	1700.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PCTAIRE-3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PFTAIRE-1	Kd	270.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PFTAIRE-1	Kd	270.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PFTAIRE-1	Kd	270.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PFTAIRE-2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PFTAIRE-2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PIM1	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PIM1	Thermal melting change	2.3	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PIM2	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase PIM2	Kd	5000.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PIM2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PIM2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PIM2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PIM2	Thermal melting change	0.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PIM3	Kd	2400.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PIM3	Kd	2400.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PIM3	Kd	2400.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PIM3	Thermal melting change	7.1	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PLK1	IC50	10000.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	Serine/threonine-protein kinase PLK1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PLK1	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PLK1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PLK1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PLK1	Thermal melting change	1.5	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PLK2	Kd	4700.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PLK2	Kd	4700.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PLK3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PLK3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PLK3	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	190.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	190.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	190.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	380.0	nM	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	380.0	nM	10.1073/pnas.0707498104
Homo sapiens	Serine/threonine-protein kinase PLK4	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PLK4	Thermal melting change	1.6	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase PRKX	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase PRKX	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PRKX	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase PRKX	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase PRP4 homolog	Kd	390.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase PRP4 homolog	Kd	390.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase RAF	IC50	10000.0	nM	10.1016/j.bmcl.2013.05.011
Homo sapiens	Serine/threonine-protein kinase RAF	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase RAF	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase RAF	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RAF	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase receptor R3	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase receptor R3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase receptor R3	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase RIO1	Kd	35.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase RIO1	Kd	35.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIO1	Kd	35.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase RIO2	Kd	49.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIO2	Kd	49.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase RIO2	Kd	200.0	nM	10.1021/acs.jmedchem.2c00271
Homo sapiens	Serine/threonine-protein kinase RIO2	Thermal melting change	6.0	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase RIO3	Kd	3800.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase RIO3	Kd	3800.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIO3	Kd	3800.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase RIPK2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase RIPK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase RIPK2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase RIPK2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase RIPK2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Serine/threonine-protein kinase SBK1	Kd	200.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase Sgk1	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Serine/threonine-protein kinase Sgk3	Kd	220.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SIK1	Kd	3200.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase SIK1	Kd	3200.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SIK1	Kd	3200.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase SIK2	Kd	580.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase SIK2	Kd	580.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SIK2	Kd	580.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase SIK2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase SIK3	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SIK3	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase SIK3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase SRPK1	Kd	250.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase SRPK1	Kd	250.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SRPK1	Kd	250.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase SRPK2	Kd	190.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase SRPK2	Kd	190.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SRPK2	Kd	190.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase SRPK3	Kd	59.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase SRPK3	Kd	59.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase TAO1	Kd	890.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TAO1	Kd	890.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase TAO1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase TAO1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase TAO2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TAO2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase TAO3	Kd	210.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TAO3	Kd	210.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase TAO3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase TBK1	Kd	120.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TBK1	Kd	120.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase TBK1	Kd	1502.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase TNNI3K	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase TNNI3K	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase TNNI3K	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase tousled-like 1	Kd	740.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase tousled-like 1	Kd	740.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase tousled-like 1	Kd	740.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase tousled-like 2	Kd	330.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase tousled-like 2	Kd	330.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase tousled-like 2	Kd	330.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase ULK1	Kd	23.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase ULK1	Kd	23.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase ULK1	Kd	2170.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase ULK2	Kd	13.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase ULK2	Kd	13.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase ULK3	Kd	42.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase ULK3	Kd	42.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase ULK3	Kd	1125.0	nM	10.1126/science.aan4368
Homo sapiens	Serine/threonine-protein kinase VRK1	Thermal melting change	6.8	degrees C	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase VRK2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase VRK2	Thermal melting change	nan	None	10.1073/pnas.0708800104
Homo sapiens	Serine/threonine-protein kinase WEE1	Kd	1100.0	nM	10.1038/nbt1358
Homo sapiens	Serine/threonine-protein kinase WEE1	Kd	1100.0	nM	10.1038/nbt.1990
Homo sapiens	Serine/threonine-protein kinase WEE1	Kd	1100.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Serine/threonine-protein kinase WEE1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Serotonin 1a (5-HT1a) receptor	AC50	7134.9	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 1a (5-HT1a) receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 2a (5-HT2a) receptor	AC50	95.9	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 2a (5-HT2a) receptor	AC50	4700.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 2a (5-HT2a) receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 2b (5-HT2b) receptor	AC50	158.2	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 2b (5-HT2b) receptor	AC50	5200.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 2b (5-HT2b) receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 2c (5-HT2c) receptor	AC50	2245.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 3a (5-HT3a) receptor	AC50	3304.5	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 5a (5-HT5a) receptor	AC50	10000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 6 (5-HT6) receptor	AC50	2391.6	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin 7 (5-HT7) receptor	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Serotonin transporter	AC50	510.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	SF-126	IC50	3061.98	nM	10.6019/CHEMBL1201861
Homo sapiens	SF-268	IC50	3328.69	nM	10.6019/CHEMBL1201861
Homo sapiens	SF-295	Activity	0.811	None	10.1073/pnas.0707498104
Homo sapiens	SF-539	IC50	106449.32	nM	10.6019/CHEMBL1201861
Homo sapiens	SH-4	IC50	5483.7	nM	10.6019/CHEMBL1201861
Homo sapiens	SHP77	Activity	0.726	None	10.1073/pnas.0707498104
Homo sapiens	SHP77	IC50	51267.81	nM	10.6019/CHEMBL1201861
Homo sapiens	SIG-M5	IC50	1370.09	nM	10.6019/CHEMBL1201861
Homo sapiens	Signal recognition particle receptor subunit alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	SiHa	Activity	1.014	None	10.1073/pnas.0707498104
Homo sapiens	SIMA	IC50	316661.06	nM	10.6019/CHEMBL1201861
Homo sapiens	SISO	Activity	1.025	None	10.1073/pnas.0707498104
Homo sapiens	SJSA-1	IC50	7660.61	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-BR-3	Activity	1.235	None	10.1073/pnas.0707498104
Homo sapiens	SK-CO-1	Activity	0.811	None	10.1073/pnas.0707498104
Homo sapiens	SKG-IIIa	Activity	1.083	None	10.1073/pnas.0707498104
Homo sapiens	SK-HEP1	Activity	1.024	None	10.1073/pnas.0707498104
Homo sapiens	SK-LMS-1	IC50	3833.38	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-LU-1	Activity	0.632	None	10.1073/pnas.0707498104
Homo sapiens	SKM-1	IC50	113679.83	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-MEL-1	IC50	138129.55	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-MEL-2	IC50	42640.52	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-MEL-28	Activity	5.09	%	10.1039/d2md00442a
Homo sapiens	SK-MEL-28	Activity	17.92	%	10.1039/d2md00442a
Homo sapiens	SK-MEL-28	Activity	76.33	%	10.1039/d2md00442a
Homo sapiens	SK-MEL-28	IC50	4130.0	nM	10.1039/d2md00442a
Homo sapiens	SK-MEL3	Activity	1.178	None	10.1073/pnas.0707498104
Homo sapiens	SK-MEL-30	Activity	0.925	None	10.1073/pnas.0707498104
Homo sapiens	SK-MES-1	Activity	0.833	None	10.1073/pnas.0707498104
Homo sapiens	SK-MES-1	Activity	0.993	None	10.1073/pnas.0707498104
Homo sapiens	SK-MM-2	IC50	5478.2	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-N-AS	Activity	1.056	None	10.1073/pnas.0707498104
Homo sapiens	SK-N-DZ	IC50	4670.99	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-NEP-1	Activity	0.855	None	10.1073/pnas.0707498104
Homo sapiens	SK-NEP-1	IC50	2602.37	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-N-FI	IC50	17691.26	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-N-SH	Activity	1.006	None	10.1073/pnas.0707498104
Homo sapiens	SK-OV-3	Activity	0.859	None	10.1073/pnas.0707498104
Homo sapiens	SK-OV-3	EC50	1360.0	nM	10.1021/acsmedchemlett.8b00596
Homo sapiens	SK-OV-3	IC50	9210.0	nM	10.1016/j.bmcl.2015.05.017
Homo sapiens	SK-PN-DW	IC50	8609.85	nM	10.6019/CHEMBL1201861
Homo sapiens	SK-UT-1	IC50	49882.54	nM	10.6019/CHEMBL1201861
Homo sapiens	SMMC-7721	IC50	6470.0	nM	10.1016/j.ejmech.2011.05.017
Homo sapiens	SNB-19	GI50	10000.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	SNB-75	IC50	127392.26	nM	10.6019/CHEMBL1201861
Homo sapiens	SNF-related serine/threonine-protein kinase	Kd	640.0	nM	10.1038/nbt.1990
Homo sapiens	SNG-M	Activity	1.367	None	10.1073/pnas.0707498104
Homo sapiens	SNU1	Activity	0.975	None	10.1073/pnas.0707498104
Homo sapiens	SNU1	IC50	13344.96	nM	10.6019/CHEMBL1201861
Homo sapiens	SNU-16	Activity	0.931	None	10.1073/pnas.0707498104
Homo sapiens	SNU-16	IC50	1464.86	nM	10.6019/CHEMBL1201861
Homo sapiens	SNU-398	Activity	1.005	None	10.1073/pnas.0707498104
Homo sapiens	SNU-449	Activity	1.101	None	10.1073/pnas.0707498104
Homo sapiens	SNU-5	Activity	0.894	None	10.1073/pnas.0707498104
Homo sapiens	SNU-5	IC50	1501043.78	nM	10.6019/CHEMBL1201861
Homo sapiens	SNU-C1	IC50	67427.57	nM	10.6019/CHEMBL1201861
Homo sapiens	SNU-C2B	IC50	149036.76	nM	10.6019/CHEMBL1201861
Homo sapiens	Sodium channel protein type V alpha subunit	AC50	26999.8	nM	10.1038/s41467-023-40064-9
Homo sapiens	Sodium channel protein type V alpha subunit	IC50	15848.93	nM	10.1016/j.vascn.2014.07.002
Homo sapiens	Sodium channel protein type V alpha subunit	IC50	39810.72	nM	10.1016/j.vascn.2014.07.002
Homo sapiens	Solute carrier family 22 member 1	IC50	6100.0	nM	10.1021/acs.jmedchem.6b01317
Homo sapiens	SPS1/STE20-related protein kinase YSK4	Kd	17.0	nM	10.1038/nbt.1990
Homo sapiens	SPS1/STE20-related protein kinase YSK4	Kd	17.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	SR	IC50	1545.72	nM	10.6019/CHEMBL1201861
Homo sapiens	ST486	IC50	6347.1	nM	10.6019/CHEMBL1201861
Homo sapiens	STE20-related kinase adapter protein alpha	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	STE20/SPS1-related proline-alanine-rich protein kinase	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	STE20/SPS1-related proline-alanine-rich protein kinase	Kd	140.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Stem cell growth factor receptor	GI50	1.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	2.0	nM	10.1021/acs.jmedchem.6b00200
Homo sapiens	Stem cell growth factor receptor	GI50	4.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	4.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	5.0	nM	10.1021/acs.jmedchem.6b00902
Homo sapiens	Stem cell growth factor receptor	GI50	5.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	5.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	6.0	nM	10.1021/acs.jmedchem.6b00200
Homo sapiens	Stem cell growth factor receptor	GI50	6.0	nM	10.1021/acs.jmedchem.6b00902
Homo sapiens	Stem cell growth factor receptor	GI50	6.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	6.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	7.0	nM	10.1021/acs.jmedchem.6b00902
Homo sapiens	Stem cell growth factor receptor	GI50	7.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	9.0	nM	10.1021/acs.jmedchem.6b00200
Homo sapiens	Stem cell growth factor receptor	GI50	10.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	11.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	12.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	14.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	18.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	20.0	nM	10.1021/acs.jmedchem.6b00200
Homo sapiens	Stem cell growth factor receptor	GI50	20.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	21.0	nM	10.1021/acs.jmedchem.6b00902
Homo sapiens	Stem cell growth factor receptor	GI50	23.0	nM	10.1021/acs.jmedchem.6b00200
Homo sapiens	Stem cell growth factor receptor	GI50	24.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	27.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	35.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	53.0	nM	10.1021/acs.jmedchem.6b00200
Homo sapiens	Stem cell growth factor receptor	GI50	78.0	nM	10.1021/acs.jmedchem.6b00200
Homo sapiens	Stem cell growth factor receptor	GI50	93.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	98.0	nM	10.1021/acs.jmedchem.7b00841
Homo sapiens	Stem cell growth factor receptor	GI50	110.0	nM	10.1021/acs.jmedchem.6b00902
Homo sapiens	Stem cell growth factor receptor	GI50	172.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	214.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	271.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	315.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	384.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	398.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	420.0	nM	10.1021/acs.jmedchem.6b00902
Homo sapiens	Stem cell growth factor receptor	GI50	430.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	510.0	nM	10.1021/acs.jmedchem.6b00200
Homo sapiens	Stem cell growth factor receptor	GI50	584.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	638.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	696.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	704.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	GI50	782.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Stem cell growth factor receptor	GI50	1380.0	nM	10.1021/acs.jmedchem.6b00200
Homo sapiens	Stem cell growth factor receptor	GI50	1720.0	nM	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	IC50	0.7	nM	10.1021/jm4004076
Homo sapiens	Stem cell growth factor receptor	IC50	1.1	nM	10.1021/acs.jmedchem.7b00841
Homo sapiens	Stem cell growth factor receptor	IC50	2.8	nM	10.1021/acs.jmedchem.0c02247
Homo sapiens	Stem cell growth factor receptor	IC50	8.0	nM	10.1021/jm201198w
Homo sapiens	Stem cell growth factor receptor	IC50	8.9	nM	10.1016/j.bmcl.2013.08.037
Homo sapiens	Stem cell growth factor receptor	IC50	10.0	nM	10.1021/jm901132v
Homo sapiens	Stem cell growth factor receptor	IC50	13.1	nM	10.1016/j.bmc.2010.05.021
Homo sapiens	Stem cell growth factor receptor	IC50	15.0	nM	10.1016/j.bmcl.2010.08.025
Homo sapiens	Stem cell growth factor receptor	IC50	35.0	nM	10.1021/jm101036c
Homo sapiens	Stem cell growth factor receptor	IC50	48.0	nM	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	IC50	48.0	nM	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	IC50	80.0	nM	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	IC50	99.6	nM	10.1021/acs.jmedchem.7b00841
Homo sapiens	Stem cell growth factor receptor	IC50	124.9	nM	10.1021/acs.jmedchem.7b00841
Homo sapiens	Stem cell growth factor receptor	IC50	264.0	nM	10.1021/jm4004076
Homo sapiens	Stem cell growth factor receptor	IC50	350.0	nM	10.1016/j.ejmech.2016.12.038
Homo sapiens	Stem cell growth factor receptor	IC50	616.8	nM	10.1021/acs.jmedchem.7b00841
Homo sapiens	Stem cell growth factor receptor	IC50	3021.0	nM	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	5.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	5.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	6.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	6.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	7.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	7.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	8.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	8.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	9.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	9.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	12.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	12.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	16.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	16.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	28.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	28.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	32.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	32.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	36.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	36.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	41.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	41.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	43.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	43.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	47.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	47.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	48.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	48.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	49.4	%	10.1016/j.bmc.2018.09.027
Homo sapiens	Stem cell growth factor receptor	Inhibition	49.4	%	10.1021/acs.jmedchem.0c02254
Homo sapiens	Stem cell growth factor receptor	Inhibition	51.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	51.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	52.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	52.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	56.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	56.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	60.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	60.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	65.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	65.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	73.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	73.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	76.0	%	10.1016/j.ejmech.2017.04.039
Homo sapiens	Stem cell growth factor receptor	Inhibition	80.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	80.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	81.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	81.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	82.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	82.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	84.8	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Stem cell growth factor receptor	Inhibition	85.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	85.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	90.1	%	10.1016/j.bmc.2010.05.021
Homo sapiens	Stem cell growth factor receptor	Inhibition	93.0	%	10.1021/acs.jmedchem.8b01845
Homo sapiens	Stem cell growth factor receptor	Inhibition	93.0	%	10.1021/acs.jmedchem.9b01229
Homo sapiens	Stem cell growth factor receptor	Inhibition	98.3	%	10.1016/j.ejmech.2020.112316
Homo sapiens	Stem cell growth factor receptor	Inhibition	nan	%	10.1021/acs.jmedchem.9b00280
Homo sapiens	Stem cell growth factor receptor	Kd	0.21	nM	10.1038/nbt1358
Homo sapiens	Stem cell growth factor receptor	Kd	0.21	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	0.21	nM	10.1182/blood-2009-05-222034
Homo sapiens	Stem cell growth factor receptor	Kd	0.28	nM	10.1038/nbt1358
Homo sapiens	Stem cell growth factor receptor	Kd	0.28	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	0.28	nM	10.1182/blood-2009-05-222034
Homo sapiens	Stem cell growth factor receptor	Kd	0.37	nM	10.1016/j.ejmech.2011.02.057
Homo sapiens	Stem cell growth factor receptor	Kd	0.37	nM	10.1038/nbt1358
Homo sapiens	Stem cell growth factor receptor	Kd	0.37	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	0.37	nM	10.1182/blood-2009-05-222034
Homo sapiens	Stem cell growth factor receptor	Kd	0.41	nM	10.1038/nbt1358
Homo sapiens	Stem cell growth factor receptor	Kd	0.41	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	0.41	nM	10.1182/blood-2009-05-222034
Homo sapiens	Stem cell growth factor receptor	Kd	0.7	nM	10.1073/pnas.0707498104
Homo sapiens	Stem cell growth factor receptor	Kd	0.71	nM	10.1038/nbt1068
Homo sapiens	Stem cell growth factor receptor	Kd	1.3	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	2.2	nM	10.1182/blood-2009-05-222034
Homo sapiens	Stem cell growth factor receptor	Kd	43.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	110.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	380.0	nM	10.1016/j.ejmech.2011.02.057
Homo sapiens	Stem cell growth factor receptor	Kd	380.0	nM	10.1038/nbt1358
Homo sapiens	Stem cell growth factor receptor	Kd	380.0	nM	10.1038/nbt.1990
Homo sapiens	Stem cell growth factor receptor	Kd	380.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Stem cell growth factor receptor	Ki	4.0	nM	10.1016/j.ejmech.2014.05.051
Homo sapiens	Stem cell growth factor receptor	Selectivity	0.0174	None	10.1038/nbt1358
Homo sapiens	Structural maintenance of chromosomes protein 1A	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Structural maintenance of chromosomes protein 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	SU-DHL-1	IC50	4801.74	nM	10.6019/CHEMBL1201861
Homo sapiens	SUP-T1	IC50	181296.9	nM	10.6019/CHEMBL1201861
Homo sapiens	SW1088	Activity	0.744	None	10.1073/pnas.0707498104
Homo sapiens	SW13	Activity	1.009	None	10.1073/pnas.0707498104
Homo sapiens	SW1417	Activity	1.119	None	10.1073/pnas.0707498104
Homo sapiens	SW1463	Activity	1.27	None	10.1073/pnas.0707498104
Homo sapiens	SW1573	Activity	0.787	None	10.1073/pnas.0707498104
Homo sapiens	SW1710	Activity	1.116	None	10.1073/pnas.0707498104
Homo sapiens	SW1783	Activity	0.873	None	10.1073/pnas.0707498104
Homo sapiens	SW1990	Activity	1.053	None	10.1073/pnas.0707498104
Homo sapiens	SW48	Activity	1.054	None	10.1073/pnas.0707498104
Homo sapiens	SW480	IC50	nan	None	10.1016/j.ejmech.2019.06.094
Homo sapiens	SW-620	Activity	1.119	None	10.1073/pnas.0707498104
Homo sapiens	SW-620	GI50	1300.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	SW-620	IC50	6250.0	nM	10.1016/j.ejmech.2018.07.052
Homo sapiens	SW684	IC50	895464.88	nM	10.6019/CHEMBL1201861
Homo sapiens	SW756	Activity	1.033	None	10.1073/pnas.0707498104
Homo sapiens	SW780	Activity	0.892	None	10.1073/pnas.0707498104
Homo sapiens	SW837	Activity	1.033	None	10.1073/pnas.0707498104
Homo sapiens	SW872	IC50	8347.58	nM	10.6019/CHEMBL1201861
Homo sapiens	SW900	Activity	0.865	None	10.1073/pnas.0707498104
Homo sapiens	SW948	Activity	1.0	None	10.1073/pnas.0707498104
Homo sapiens	SW 954	IC50	6275.17	nM	10.6019/CHEMBL1201861
Homo sapiens	SW 962	IC50	20429.26	nM	10.6019/CHEMBL1201861
Homo sapiens	SW982	IC50	4553.07	nM	10.6019/CHEMBL1201861
Homo sapiens	SW982	IC50	41200.0	nM	10.1016/j.ejmech.2019.111719
Homo sapiens	T-24	Activity	1.059	None	10.1073/pnas.0707498104
Homo sapiens	T-24	IC50	2440.0	nM	10.1016/j.bmcl.2013.08.037
Homo sapiens	T47D	Activity	0.917	None	10.1073/pnas.0707498104
Homo sapiens	T84	Activity	0.84	None	10.1073/pnas.0707498104
Homo sapiens	T98G	Activity	0.84	None	10.1073/pnas.0707498104
Homo sapiens	TALL-1	IC50	8183.84	nM	10.6019/CHEMBL1201861
Homo sapiens	Tankyrase-2	Kd	8900.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	TCO-1	Activity	0.912	None	10.1073/pnas.0707498104
Homo sapiens	TE-1	IC50	20410.37	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-10	IC50	2343.84	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-11	IC50	1839.85	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-12	IC50	804.55	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-15	IC50	507.61	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-441-T	IC50	94973.98	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-5	IC50	177295.71	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-6	IC50	107684.43	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-8	IC50	2370.38	nM	10.6019/CHEMBL1201861
Homo sapiens	TE-9	IC50	37040.1	nM	10.6019/CHEMBL1201861
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	Kd	6300.0	nM	10.1038/nbt1358
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	Kd	6300.0	nM	10.1038/nbt.1990
Homo sapiens	Testis-specific serine/threonine-protein kinase 1	Kd	6300.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	TGBC1TKB	IC50	12001.96	nM	10.6019/CHEMBL1201861
Homo sapiens	TGBC24TKB	IC50	160923.65	nM	10.6019/CHEMBL1201861
Homo sapiens	TGF-beta receptor type I	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	TGF-beta receptor type I	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	TGF-beta receptor type I	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	TGF-beta receptor type I	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	TGF-beta receptor type II	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	TGF-beta receptor type II	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	TGF-beta receptor type II	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	TGF-beta receptor type II	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	TGW	Activity	1.024	None	10.1073/pnas.0707498104
Homo sapiens	TGW	IC50	13327.57	nM	10.6019/CHEMBL1201861
Homo sapiens	THP-1	IC50	45.7	nM	10.1016/j.ejmech.2014.07.108
Homo sapiens	THP-1	IC50	500.0	nM	10.1016/j.bmc.2010.05.021
Homo sapiens	THP-1	IC50	1000.0	nM	10.1021/acs.jmedchem.8b01714
Homo sapiens	THP-1	IC50	14900.0	nM	10.1016/j.ejmech.2019.111719
Homo sapiens	THP-1	IC50	191743.4	nM	10.6019/CHEMBL1201861
Homo sapiens	Thromboxane A2 receptor	AC50	9100.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Thyroid hormone receptor-associated protein 3	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	TK-10	GI50	6300.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	TK-10	IC50	30126.01	nM	10.6019/CHEMBL1201861
Homo sapiens	TP53-regulating kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	TRAF2- and NCK-interacting kinase	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	25.0	nM	10.1038/nbt1068
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	25.0	nM	10.1038/nbt1358
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	25.0	nM	10.1038/nbt.1990
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	25.0	nM	10.1039/C5MD00090D
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	25.0	nM	10.1073/pnas.0707498104
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	25.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	TRAF2- and NCK-interacting kinase	Kd	387.0	nM	10.1126/science.aan4368
Homo sapiens	TRAF2- and NCK-interacting kinase	Thermal melting change	0.7	degrees C	10.1073/pnas.0708800104
Homo sapiens	Transient receptor potential cation channel subfamily M member 6	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	TT	IC50	40.0	nM	10.1016/j.ejmech.2014.05.051
Homo sapiens	TUR	IC50	1053110.03	nM	10.6019/CHEMBL1201861
Homo sapiens	TYK-nu	Activity	0.813	None	10.1073/pnas.0707498104
Homo sapiens	Type-1 angiotensin II receptor	AC50	4300.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine- and threonine-specific cdc2-inhibitory kinase	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine kinase non-receptor protein 2	IC50	7830.0	nM	10.1021/acs.jmedchem.1c01030
Homo sapiens	Tyrosine kinase non-receptor protein 2	Inhibition	33.0	%	10.1021/acs.jmedchem.1c01030
Homo sapiens	Tyrosine kinase non-receptor protein 2	Kd	2200.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine kinase non-receptor protein 2	Kd	8900.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine kinase non-receptor protein 2	Kd	8900.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine kinase non-receptor protein 2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase ABL	Activity	73.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	Tyrosine-protein kinase ABL	Activity	99.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	Tyrosine-protein kinase ABL	Activity	100.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	Tyrosine-protein kinase ABL	IC50	410.0	nM	10.1038/nchembio.117
Homo sapiens	Tyrosine-protein kinase ABL	IC50	504.0	nM	10.1021/jm4004076
Homo sapiens	Tyrosine-protein kinase ABL	IC50	1613.0	nM	10.1021/jm4004076
Homo sapiens	Tyrosine-protein kinase ABL	IC50	50000.0	nM	10.1016/j.bmc.2010.01.011
Homo sapiens	Tyrosine-protein kinase ABL	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Tyrosine-protein kinase ABL	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Tyrosine-protein kinase ABL	Kd	55.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	74.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	76.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	120.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	140.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	140.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	140.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase ABL	Kd	150.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	180.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	210.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Kd	240.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	270.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	370.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	530.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Kd	720.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Kd	730.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	830.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	830.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase ABL	Kd	870.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Kd	870.0	nM	10.1073/pnas.0707498104
Homo sapiens	Tyrosine-protein kinase ABL	Kd	890.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	890.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	890.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase ABL	Kd	950.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	950.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase ABL	Kd	1000.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Kd	1000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	1000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase ABL	Kd	1200.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	1200.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase ABL	Kd	2300.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Kd	2800.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL	Kd	2800.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase ABL	Kd	3600.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase ABL	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase ABL	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	Tyrosine-protein kinase ABL2	Kd	1000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ABL2	Kd	1000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ABL2	Kd	1000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase ABL2	Kd	1200.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ABL2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase ABL2	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	Tyrosine-protein kinase BLK	Kd	65.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase BLK	Kd	65.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase BLK	Kd	65.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase BMX	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase BMX	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase BMX	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase BMX	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase BRK	Kd	4600.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase BRK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase BRK	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase BRK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase BRK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase BTK	Inhibition	91.3	%	10.1016/j.ejmech.2020.112316
Homo sapiens	Tyrosine-protein kinase BTK	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Tyrosine-protein kinase BTK	Kd	2100.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase BTK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase BTK	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase BTK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase BTK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase CSK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase CSK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase CSK	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase CSK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase CSK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase CTK	Kd	7700.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase CTK	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase FER	Kd	1100.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FER	Kd	1100.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FER	Kd	1100.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase FER	Kd	1400.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase FER	Kd	1999.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase FES	Kd	960.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FES	Kd	960.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FES	Kd	960.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase FES	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase FGR	Kd	270.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FGR	Kd	270.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FGR	Kd	270.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase FGR	Kd	290.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase FGR	Kd	290.0	nM	10.1073/pnas.0707498104
Homo sapiens	Tyrosine-protein kinase FGR	Kd	1518.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase FRK	Kd	530.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FRK	Kd	530.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FRK	Kd	530.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase FRK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase FRK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase FYN	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Tyrosine-protein kinase FYN	Kd	520.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase FYN	Kd	520.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase FYN	Kd	520.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase FYN	Kd	3900.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase FYN	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase FYN	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	Tyrosine-protein kinase HCK	IC50	190.0	nM	10.1038/nchembio.117
Homo sapiens	Tyrosine-protein kinase HCK	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Tyrosine-protein kinase HCK	Kd	880.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase HCK	Kd	880.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase HCK	Kd	880.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase HCK	Kd	1943.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase HCK	Kd	3300.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase ITK/TSK	Kd	13.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ITK/TSK	Kd	13.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ITK/TSK	Kd	13.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase JAK1	Inhibition	98.1	%	10.1016/j.ejmech.2020.112316
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	9.0	nM	10.1073/pnas.0707498104
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	9.2	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	49.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	49.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	49.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	475.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	6000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase JAK1	Kd	6000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase JAK1	Thermal melting change	5.5	degrees C	10.1073/pnas.0708800104
Homo sapiens	Tyrosine-protein kinase JAK2	Kd	410.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase JAK2	Kd	410.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase JAK2	Kd	410.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase JAK2	Kd	940.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase JAK2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase JAK3	Kd	1200.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase JAK3	Kd	1200.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase JAK3	Kd	1200.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase LCK	IC50	8.9	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Tyrosine-protein kinase LCK	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Tyrosine-protein kinase LCK	Kd	230.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase LCK	Kd	230.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase LCK	Kd	230.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase LCK	Kd	1200.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase LCK	Kd	1464.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase LCK	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	Tyrosine-protein kinase Lyn	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	270.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	270.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	270.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	540.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	540.0	nM	10.1073/pnas.0707498104
Homo sapiens	Tyrosine-protein kinase Lyn	Kd	1416.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	0.7	nM	10.1021/acs.jmedchem.0c02247
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	0.8	nM	10.1021/acs.jmedchem.0c02247
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	1.4	nM	10.1021/acs.jmedchem.0c02247
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	2.5	nM	10.1016/j.ejmech.2016.12.038
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	2.5	nM	10.1021/acs.jmedchem.0c02167
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	3.0	nM	10.1016/j.bmcl.2010.08.025
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	4.7	nM	10.1016/j.bmc.2021.116422
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	5.0	nM	10.1021/acs.jmedchem.0c02167
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	6.5	nM	10.1016/j.bmc.2010.05.021
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	8.0	nM	10.1021/jm201198w
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	9.9	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	12.0	nM	10.1016/j.ejmech.2016.12.038
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	16.0	nM	10.1016/j.bmcl.2010.08.025
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	21.0	nM	10.1021/jm901132v
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	25.0	nM	10.1016/j.ejmech.2020.112205
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	30.0	nM	10.1016/j.bmc.2021.116596
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	30.0	nM	10.1016/j.ejmech.2019.111710
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	31.0	nM	10.1021/acs.jmedchem.9b01229
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	34.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	50.0	nM	10.1016/j.bmc.2021.116596
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	50.0	nM	10.1016/j.ejmech.2019.111710
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	50.0	nM	10.1021/acs.jmedchem.0c00696
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	250.0	nM	10.1016/j.bmc.2021.116596
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	250.0	nM	10.1016/j.ejmech.2019.111710
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	250.0	nM	10.1021/acs.jmedchem.0c00696
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	550.0	nM	10.1016/j.bmc.2010.01.011
Homo sapiens	Tyrosine-protein kinase receptor FLT3	IC50	nan	None	10.1016/j.bmcl.2010.08.025
Homo sapiens	Tyrosine-protein kinase receptor FLT3	INH	8.2	nM	10.1021/acs.jmedchem.8b01714
Homo sapiens	Tyrosine-protein kinase receptor FLT3	INH	105.0	nM	10.1021/acs.jmedchem.8b01714
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	29.0	%	10.1021/acs.jmedchem.8b01714
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	70.0	%	10.1021/acs.jmedchem.8b01714
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	78.8	%	10.1016/j.bmc.2010.05.021
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	82.0	%	10.1021/acs.jmedchem.8b01714
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	92.3	%	10.1016/j.bmcl.2018.06.026
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	94.8	%	10.1016/j.bmcl.2018.06.026
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	96.0	%	10.1021/acs.jmedchem.8b01714
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	100.0	%	10.1016/j.bmcl.2012.10.016
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	nan	%	10.1021/acs.jmedchem.5b01582
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Tyrosine-protein kinase receptor FLT3	K	0.0613	/min	10.1016/j.bmc.2014.10.006
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.22	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.22	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.41	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.43	nM	10.1021/acs.jmedchem.8b01714
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.47	nM	10.1021/jm9007533
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.47	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.47	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.8	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.8	nM	10.1073/pnas.0707498104
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.99	nM	10.1021/acs.jmedchem.8b01714
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.99	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	0.99	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.3	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.3	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.3	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.4	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.4	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	2.4	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	4.3	nM	10.1021/acs.jmedchem.8b01714
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	4.3	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	4.3	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	4.3	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	11.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Kd	nan	None	10.1021/acs.jmedchem.8b01714
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	Tyrosine-protein kinase receptor FLT3	Ratio	10.0	None	10.1021/acs.jmedchem.8b01714
Homo sapiens	Tyrosine-protein kinase receptor FLT3	T1/2	0.1883	hr	10.1016/j.bmc.2014.10.006
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	1.0	nM	10.1038/nchembio.117
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	5.0	nM	10.1021/acs.jmedchem.0c02167
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	220.0	nM	10.1021/jm501464c
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	224.0	nM	10.1021/jm501464c
Homo sapiens	Tyrosine-protein kinase receptor RET	IC50	1300.0	nM	10.1016/j.bmc.2010.01.011
Homo sapiens	Tyrosine-protein kinase receptor RET	Inhibition	76.7	%	10.1016/j.ejmech.2018.09.032
Homo sapiens	Tyrosine-protein kinase receptor RET	Inhibition	84.8	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Tyrosine-protein kinase receptor RET	Inhibition	97.0	%	10.1016/j.bmc.2018.09.027
Homo sapiens	Tyrosine-protein kinase receptor RET	Inhibition	97.0	%	10.1021/acs.jmedchem.0c02254
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	5.8	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	5.8	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	8.7	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	8.7	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	12.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	12.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	13.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	19.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	19.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	19.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor RET	Kd	33.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase receptor RET	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	Tyrosine-protein kinase receptor Tie-1	Kd	3900.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor Tie-1	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor Tie-1	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Activity	9.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Activity	99.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Kd	49.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Kd	49.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor TYRO3	Kd	49.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor UFO	Activity	99.9	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	Tyrosine-protein kinase receptor UFO	Activity	100.0	%	10.1016/j.ejmech.2012.06.005
Homo sapiens	Tyrosine-protein kinase receptor UFO	IC50	9.0	nM	10.1016/j.bmcl.2017.06.071
Homo sapiens	Tyrosine-protein kinase receptor UFO	IC50	9.0	nM	10.1021/acs.jmedchem.5b01273
Homo sapiens	Tyrosine-protein kinase receptor UFO	Kd	9.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase receptor UFO	Kd	9.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase receptor UFO	Kd	9.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase receptor UFO	Ki	nan	None	10.1016/j.ejmech.2014.05.051
Homo sapiens	Tyrosine-protein kinase SRC	IC50	152.8	nM	10.1016/j.ejmech.2011.07.001
Homo sapiens	Tyrosine-protein kinase SRC	IC50	400.0	nM	10.1038/nchembio.117
Homo sapiens	Tyrosine-protein kinase SRC	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Tyrosine-protein kinase SRC	Inhibition	nan	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Tyrosine-protein kinase SRC	Inhibition	nan	%	10.1021/acs.jmedchem.5b01582
Homo sapiens	Tyrosine-protein kinase SRC	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Tyrosine-protein kinase SRC	Kd	2100.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase SRC	Kd	2100.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase SRC	Kd	2100.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase SRC	Kd	3100.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase SRC	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase Srms	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase Srms	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase Srms	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase SYK	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Tyrosine-protein kinase SYK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase SYK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase SYK	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase SYK	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase SYK	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase TEC	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase TEC	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TEC	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase TEC	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase TIE-2	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase TIE-2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TIE-2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase TIE-2	Kd	nan	None	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase TXK	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase TXK	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TXK	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase TYK2	Kd	360.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TYK2	Kd	360.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase TYK2	Kd	1600.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase TYK2	Kd	1600.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase TYK2	Kd	1600.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase TYK2	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase YES	Kd	120.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase YES	Kd	120.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase YES	Kd	120.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosine-protein kinase YES	Kd	240.0	nM	10.1038/nbt1068
Homo sapiens	Tyrosine-protein kinase YES	Kd	758.0	nM	10.1126/science.aan4368
Homo sapiens	Tyrosine-protein kinase YES	Potency	48.7	nM	None
Homo sapiens	Tyrosine-protein kinase ZAP-70	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Tyrosine-protein kinase ZAP-70	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Tyrosine-protein kinase ZAP-70	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Tyrosyl-tRNA synthetase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	U-251	Inhibition	nan	%	10.1021/ml4004793
Homo sapiens	U-266	IC50	34278.15	nM	10.6019/CHEMBL1201861
Homo sapiens	U373 MG	Activity	1.055	None	10.1073/pnas.0707498104
Homo sapiens	U5 small nuclear ribonucleoprotein 200 kDa helicase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	U-698-M	IC50	189794.52	nM	10.6019/CHEMBL1201861
Homo sapiens	U-87 MG	IC50	440400.7	nM	10.6019/CHEMBL1201861
Homo sapiens	U-87 MG	Inhibition	nan	%	10.1021/jm201649s
Homo sapiens	U-937	IC50	5000.0	nM	10.1016/j.bmc.2010.05.021
Homo sapiens	U-937	IC50	13700.0	nM	10.1016/j.ejmech.2019.111719
Homo sapiens	UACC-257	GI50	4000.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	UACC-257	IC50	108945.85	nM	10.6019/CHEMBL1201861
Homo sapiens	UACC-812	Activity	1.301	None	10.1073/pnas.0707498104
Homo sapiens	Ubiquitin carboxyl-terminal hydrolase 1	Potency	89125.1	nM	None
Homo sapiens	UMC-11	Activity	0.902	None	10.1073/pnas.0707498104
Homo sapiens	UMP-CMP kinase	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	UMUC3	Activity	0.97	None	10.1073/pnas.0707498104
Homo sapiens	Uncharacterized aarF domain-containing protein kinase 1	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Uncharacterized aarF domain-containing protein kinase 4	Kd	10000.0	nM	10.1038/nbt1358
Homo sapiens	Uncharacterized aarF domain-containing protein kinase 4	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Uncharacterized aarF domain-containing protein kinase 4	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Uncharacterized aarF domain-containing protein kinase 5	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	Uncharacterized protein FLJ45252	Kd	431.0	nM	10.1126/science.aan4368
Homo sapiens	UO-31	Activity	0.867	None	10.1073/pnas.0707498104
Homo sapiens	VA-ES-BJ	IC50	9999.33	nM	10.6019/CHEMBL1201861
Homo sapiens	Vascular endothelial growth factor receptor 1	IC50	1.0	nM	10.1016/j.bmcl.2012.06.029
Homo sapiens	Vascular endothelial growth factor receptor 1	IC50	15.0	nM	10.1021/acs.jmedchem.5b01582
Homo sapiens	Vascular endothelial growth factor receptor 1	IC50	90.5	nM	10.1021/acs.jmedchem.0c02247
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	66.0	%	10.1016/j.ejmech.2018.09.032
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	66.6	%	10.1016/j.bmcl.2014.11.070
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	74.2	%	10.1016/j.ejmech.2017.04.039
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	74.8	%	10.1016/j.bmc.2018.09.027
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	74.8	%	10.1021/acs.jmedchem.0c02254
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	86.4	%	10.1016/j.ejmech.2021.113333
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	87.1	%	10.1016/j.bmcl.2012.09.043
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	87.1	%	10.1016/j.ejmech.2012.09.021
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	88.0	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	96.1	%	10.1016/j.ejmech.2020.112316
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	nan	%	10.1016/j.ejmech.2013.03.022
Homo sapiens	Vascular endothelial growth factor receptor 1	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Vascular endothelial growth factor receptor 1	Kd	1.8	nM	10.1038/nbt1358
Homo sapiens	Vascular endothelial growth factor receptor 1	Kd	1.8	nM	10.1038/nbt.1990
Homo sapiens	Vascular endothelial growth factor receptor 1	Kd	1.8	nM	10.1182/blood-2009-05-222034
Homo sapiens	Vascular endothelial growth factor receptor 1	Ki	2.0	nM	10.1016/j.ejmech.2014.05.051
Homo sapiens	Vascular endothelial growth factor receptor 2	AC50	15.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Vascular endothelial growth factor receptor 2	Activity	66.0	%	10.1016/j.ejmech.2018.11.023
Homo sapiens	Vascular endothelial growth factor receptor 2	Activity	70.0	%	10.1016/j.ejmech.2018.11.023
Homo sapiens	Vascular endothelial growth factor receptor 2	Activity	79.0	%	10.1016/j.ejmech.2018.11.023
Homo sapiens	Vascular endothelial growth factor receptor 2	Activity	80.0	%	10.1016/j.ejmech.2018.11.023
Homo sapiens	Vascular endothelial growth factor receptor 2	Activity	135.0	%	10.1016/j.ejmech.2018.11.023
Homo sapiens	Vascular endothelial growth factor receptor 2	GI50	33.0	nM	10.1021/acs.jmedchem.8b00938
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	0.4	nM	10.1021/acs.jmedchem.0c02167
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	4.0	nM	10.1016/j.bmcl.2013.08.037
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	4.7	nM	10.1016/j.ejmech.2018.09.032
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	5.5	nM	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	5.7	nM	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	8.0	nM	10.1021/jm201198w
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	8.75	nM	10.1021/acs.jmedchem.5b01582
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	9.0	nM	10.1016/j.ejmech.2010.09.002
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	10.0	nM	None
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	10.2	nM	10.1021/acs.jmedchem.5b01582
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	12.0	nM	10.1016/j.ejmech.2011.10.009
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	15.0	nM	10.1021/jm101036c
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18.0	nM	10.1016/j.bmcl.2007.01.089
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18.0	nM	10.1016/j.ejmech.2015.12.016
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18.0	nM	10.1021/jm050458h
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18.9	nM	10.1016/j.bmc.2014.04.049
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18.9	nM	10.1016/j.bmc.2015.03.061
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18.9	nM	10.1016/j.bmc.2016.11.026
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18.9	nM	10.1016/j.bmc.2021.116061
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18.9	nM	10.1016/j.bmcl.2018.07.039
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18.9	nM	10.1021/ml4004793
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	22.0	nM	10.1021/jm050458h
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	22.6	nM	10.1016/j.bmc.2010.05.021
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	25.0	nM	10.1016/j.bmcl.2008.04.009
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	27.0	nM	10.1073/pnas.0707498104
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	29.2	nM	10.1016/j.ejmech.2019.06.054
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	30.0	nM	10.1016/j.bmcl.2008.04.009
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	37.0	nM	10.1016/j.bmcl.2012.06.029
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	38.0	nM	10.1021/jm901132v
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	39.0	nM	10.1016/j.ejmech.2015.08.012
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	40.0	nM	10.1016/j.ejmech.2014.07.071
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	53.0	nM	10.1016/j.bmcl.2010.08.025
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	54.0	nM	10.1016/j.ejmech.2018.03.018
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	65.0	nM	10.1016/j.ejmech.2018.10.045
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	70.0	nM	10.1016/j.ejmech.2012.04.007
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	75.0	nM	10.1016/j.ejmech.2020.112752
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	75.9	nM	10.1021/acs.jmedchem.0c02247
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	80.0	nM	10.1016/j.ejmech.2015.10.053
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	80.0	nM	10.1016/j.ejmech.2019.02.050
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	80.0	nM	10.1016/j.ejmech.2019.06.070
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	80.0	nM	10.1021/acs.jmedchem.6b01266
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	80.0	nM	10.1021/acs.jmedchem.7b01091
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	80.0	nM	10.1021/jm0204183
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	95.0	nM	10.1038/nchembio.117
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	98.0	nM	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	139.0	nM	10.1021/jm101036c
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	140.0	nM	10.1016/j.ejmech.2016.04.029
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	147.0	nM	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	185.0	nM	10.1016/j.bmcl.2009.01.068
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	461.0	nM	10.1016/j.ejmech.2020.112316
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18900.0	nM	10.1016/j.bmc.2010.03.052
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18900.0	nM	10.1016/j.bmc.2010.05.049
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18900.0	nM	10.1016/j.bmc.2011.11.058
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18900.0	nM	10.1016/j.bmc.2012.05.068
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18900.0	nM	10.1016/j.bmc.2012.12.045
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	18900.0	nM	10.1016/j.bmc.2013.01.040
Homo sapiens	Vascular endothelial growth factor receptor 2	IC50	83200.0	nM	10.1016/j.ejmech.2020.113083
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	74.6	%	10.1016/j.bmc.2010.05.021
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	76.0	%	10.1021/jm300667v
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	81.8	%	10.1016/j.bmcl.2014.11.070
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	82.1	%	10.1021/np070421v
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	89.7	%	10.1016/j.bmcl.2012.09.043
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	89.7	%	10.1016/j.ejmech.2012.09.021
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	92.74	%	10.1016/j.ejmech.2018.03.018
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	94.2	%	10.1016/j.bmcl.2011.11.003
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	100.0	%	10.1016/j.bmcl.2014.03.042
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	100.0	%	10.1016/j.ejmech.2020.112316
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	102.3	%	10.1016/j.ejmech.2019.06.054
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	nan	%	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	nan	%	10.1016/j.bmcl.2011.09.022
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	nan	%	10.1016/j.bmcl.2017.12.066
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	nan	%	10.1016/j.ejmech.2013.03.022
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	nan	%	10.1016/j.ejmech.2016.04.029
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	nan	%	10.1016/j.ejmech.2017.09.015
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	nan	%	10.1016/j.ejmech.2018.03.018
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	nan	%	10.1016/j.ejmech.2018.11.023
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	nan	%	10.1021/acs.jmedchem.6b01266
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Vascular endothelial growth factor receptor 2	Inhibition	nan	%	10.1021/acs.jnatprod.9b00648
Homo sapiens	Vascular endothelial growth factor receptor 2	Kd	0.2	nM	10.1073/pnas.0707498104
Homo sapiens	Vascular endothelial growth factor receptor 2	Kd	0.23	nM	10.1038/nbt1068
Homo sapiens	Vascular endothelial growth factor receptor 2	Kd	1.5	nM	10.1038/nbt1358
Homo sapiens	Vascular endothelial growth factor receptor 2	Kd	1.5	nM	10.1038/nbt.1990
Homo sapiens	Vascular endothelial growth factor receptor 2	Kd	1.5	nM	10.1182/blood-2009-05-222034
Homo sapiens	Vascular endothelial growth factor receptor 2	Kd	30.0	nM	10.1021/ml500394m
Homo sapiens	Vascular endothelial growth factor receptor 2	Ki	2.9	nM	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	Ki	9.0	nM	10.1016/j.bmcl.2012.02.068
Homo sapiens	Vascular endothelial growth factor receptor 2	Ki	9.0	nM	10.1016/j.ejmech.2012.10.020
Homo sapiens	Vascular endothelial growth factor receptor 2	Ki	9.0	nM	10.1016/j.ejmech.2014.05.051
Homo sapiens	Vascular endothelial growth factor receptor 2	Ki	nan	None	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	Ratio IC50	20.0	None	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	T1/2	0.08333	hr	10.1016/j.bmc.2011.08.002
Homo sapiens	Vascular endothelial growth factor receptor 2	TIME	0.04833	hr	10.1021/ml500394m
Homo sapiens	Vascular endothelial growth factor receptor 3	IC50	8.9	nM	10.1016/j.bmc.2010.05.021
Homo sapiens	Vascular endothelial growth factor receptor 3	IC50	24.0	nM	10.1021/acs.jmedchem.5b01582
Homo sapiens	Vascular endothelial growth factor receptor 3	Inhibition	81.3	%	10.1016/j.bmc.2010.05.021
Homo sapiens	Vascular endothelial growth factor receptor 3	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
Homo sapiens	Vascular endothelial growth factor receptor 3	Kd	35.0	nM	10.1038/nbt1068
Homo sapiens	Vascular endothelial growth factor receptor 3	Kd	35.0	nM	10.1073/pnas.0707498104
Homo sapiens	Vascular endothelial growth factor receptor 3	Kd	50.0	nM	10.1038/nbt1358
Homo sapiens	Vascular endothelial growth factor receptor 3	Kd	50.0	nM	10.1038/nbt.1990
Homo sapiens	Vascular endothelial growth factor receptor 3	Kd	50.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	Vascular endothelial growth factor receptor 3	Ki	17.0	nM	10.1016/j.ejmech.2014.05.051
Homo sapiens	Vasopressin V1a receptor	AC50	10000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Vasopressin V2 receptor	AC50	5400.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Very long-chain specific acyl-CoA dehydrogenase, mitochondrial	Kd	30000.0	nM	10.1126/science.aan4368
Homo sapiens	VM-CUB-1	Activity	0.981	None	10.1073/pnas.0707498104
Homo sapiens	VMRC-LCP	Activity	1.04	None	10.1073/pnas.0707498104
Homo sapiens	VMRC-MELG	Activity	1.0	None	10.1073/pnas.0707498104
Homo sapiens	VMRC-RCZ	Activity	0.772	None	10.1073/pnas.0707498104
Homo sapiens	Voltage-gated L-type calcium channel	IC50	33400.0	nM	10.1038/srep02100
Homo sapiens	Voltage-gated L-type calcium channel alpha-1C subunit	AC50	50000.0	nM	10.1038/s41467-023-40064-9
Homo sapiens	Voltage-gated L-type calcium channel alpha-1C subunit	IC50	79432.82	nM	10.1016/j.vascn.2014.07.002
Homo sapiens	Voltage-gated L-type calcium channel alpha-1C subunit	IC50	199526.23	nM	10.1016/j.vascn.2014.07.002
Homo sapiens	Voltage-gated potassium channel, IKs; KCNQ1(Kv7.1)/KCNE1(MinK)	IC50	63095.73	nM	10.1016/j.vascn.2014.07.002
Homo sapiens	Voltage-gated potassium channel, IKs; KCNQ1(Kv7.1)/KCNE1(MinK)	pIC50	nan	None	10.1016/j.vascn.2014.07.002
Homo sapiens	Voltage-gated potassium channel subunit Kv4.3	IC50	50118.72	nM	10.1016/j.vascn.2014.07.002
Homo sapiens	Wee1-like protein kinase 2	Kd	10000.0	nM	10.1038/nbt.1990
Homo sapiens	Wee1-like protein kinase 2	Kd	10000.0	nM	10.1182/blood-2009-05-222034
Homo sapiens	WI-38	IC50	8560.0	nM	10.1016/j.ejmech.2011.05.017
Homo sapiens	WI-38 VA13	Activity	0.935	None	10.1073/pnas.0707498104
Homo sapiens	WiDr	Activity	1.095	None	10.1073/pnas.0707498104
Homo sapiens	WSU-NHL	IC50	375216.05	nM	10.6019/CHEMBL1201861
Homo sapiens	YAPC	Activity	0.801	None	10.1073/pnas.0707498104
Homo sapiens	YKG-1	Activity	0.916	None	10.1073/pnas.0707498104
Homo sapiens	YT	IC50	193369.91	nM	10.6019/CHEMBL1201861
Homo sapiens	ZR-75-1	Activity	1.04	None	10.1073/pnas.0707498104
Homo sapiens	ZR-75-1	IC50	5870.0	nM	10.1016/j.ejmech.2020.112359
Homo sapiens	ZR-75-1	IC50	18900.0	nM	10.1016/j.ejmech.2020.112359
Homo sapiens	ZR-75-30	Activity	1.095	None	10.1073/pnas.0707498104
Macaca fascicularis	Cynomolgus monkey	AUC	1099.0	ng.hr.mL-1	10.1124/dmd.111.042853
Macaca fascicularis	Cynomolgus monkey	AUC	1453.0	ng.hr.mL-1	10.1124/dmd.111.042853
Macaca fascicularis	Cynomolgus monkey	Cmax	208.29	nM	10.1124/dmd.111.042853
Macaca fascicularis	Cynomolgus monkey	Cmax	230.88	nM	10.1124/dmd.111.042853
Macaca fascicularis	Cynomolgus monkey	T1/2	16.0	hr	10.1124/dmd.111.042853
Macaca fascicularis	Cynomolgus monkey	T1/2	18.0	hr	10.1124/dmd.111.042853
Macaca fascicularis	Cynomolgus monkey	Tmax	4.0	hr	10.1124/dmd.111.042853
Macaca fascicularis	Cynomolgus monkey	Tmax	5.0	hr	10.1124/dmd.111.042853
Mus musculus	4T1	IC50	16.0	nM	10.1016/j.bmc.2014.04.049
Mus musculus	B16-F10	IC50	15350.0	nM	10.1039/d2md00442a
Mus musculus	BaF3	Activity	87.0	%	10.1021/acs.jmedchem.8b00938
Mus musculus	BaF3	GI50	1.3	nM	10.1039/d2md00067a
Mus musculus	BaF3	GI50	2.3	nM	10.1039/d2md00067a
Mus musculus	BaF3	GI50	4.3	nM	10.1039/d2md00067a
Mus musculus	BaF3	GI50	6.5	nM	10.1039/d2md00067a
Mus musculus	BaF3	GI50	6.9	nM	10.1039/d2md00067a
Mus musculus	BaF3	GI50	8.7	nM	10.1039/d2md00067a
Mus musculus	BaF3	GI50	19.38	nM	10.1039/d2md00067a
Mus musculus	BaF3	GI50	67.8	nM	10.1039/d2md00067a
Mus musculus	BaF3	GI50	1010.0	nM	10.1021/acs.jmedchem.9b00280
Mus musculus	BaF3	GI50	1600.0	nM	10.1021/acs.jmedchem.6b00902
Mus musculus	BaF3	GI50	2780.0	nM	10.1021/acs.jmedchem.6b00200
Mus musculus	BaF3	GI50	4789.0	nM	10.1021/acs.jmedchem.8b00938
Mus musculus	BaF3	IC50	2.3	nM	10.1021/acs.jmedchem.5b01582
Mus musculus	BaF3	IC50	35.0	nM	10.1021/acs.jmedchem.5b01582
Mus musculus	BaF3	IC50	238.0	nM	10.1021/acs.jmedchem.5b01582
Mus musculus	BaF3	IC50	297.0	nM	10.1021/acs.jmedchem.5b01582
Mus musculus	BaF3	IC50	1154.0	nM	10.1021/acs.jmedchem.5b01582
Mus musculus	BaF3	IC50	1289.0	nM	10.1021/acs.jmedchem.5b01582
Mus musculus	BaF3	IC50	1469.0	nM	10.1021/acs.jmedchem.5b01582
Mus musculus	BaF3	IC50	1561.0	nM	10.1021/acs.jmedchem.5b01582
Mus musculus	BaF3	IC50	3846.0	nM	10.1021/acs.jmedchem.5b01582
Mus musculus	BaF3	IC50	5124.0	nM	10.1021/acs.jmedchem.5b01582
Mus musculus	BaF3	IC50	7177.0	nM	10.1021/acs.jmedchem.5b01582
Mus musculus	BaF3	IC50	10000.0	nM	10.1021/acs.jmedchem.5b01582
Mus musculus	BaF3	TGI	100.0	%	10.1021/acs.jmedchem.8b00938
Mus musculus	Beta-TC6	Activity	93.35	%	None
Mus musculus	G protein-coupled receptor kinase 5	Activity	53.2	%	None
Mus musculus	Liver	T1/2	0.1833	hr	10.1021/jm401067s
Mus musculus	Liver	T1/2	0.205	hr	10.1021/jm501284e
Mus musculus	Mast/stem cell growth factor receptor Kit	GI50	3.0	nM	10.1021/acs.jmedchem.9b00280
Mus musculus	Mus musculus	Activity	-24.1	%	10.1016/j.ejmech.2014.05.051
Mus musculus	Mus musculus	Activity	12.3	%	10.1016/j.ejmech.2014.05.051
Mus musculus	Mus musculus	Activity	80.0	%	10.1016/j.bmc.2017.05.028
Mus musculus	Mus musculus	Activity	nan	None	10.1016/j.bmcl.2009.06.022
Mus musculus	Mus musculus	Activity	nan	None	10.1016/j.ejmech.2014.05.051
Mus musculus	Mus musculus	Activity	nan	None	10.1021/acs.jmedchem.1c00892
Mus musculus	Mus musculus	Activity	nan	None	10.1021/ml4004793
Mus musculus	Mus musculus	AUC	438.33	ng.hr.mL-1	10.1182/blood-2009-05-222034
Mus musculus	Mus musculus	Cmax	320.0	nM	10.1182/blood-2009-05-222034
Mus musculus	Mus musculus	Cpss	1378.0	ng/ml	10.1021/jm201198w
Mus musculus	Mus musculus	ED50	9.0	mg.kg-1	10.1021/jm050458h
Mus musculus	Mus musculus	ED50	11.0	mg.kg-1	10.1021/jm050458h
Mus musculus	Mus musculus	Inhibition	0.0	%	10.1016/j.bmcl.2012.06.029
Mus musculus	Mus musculus	Inhibition	78.0	%	10.1016/j.bmcl.2017.06.071
Mus musculus	Mus musculus	Inhibition	nan	%	10.1021/acs.jmedchem.6b01266
Mus musculus	Mus musculus	MTD	30.0	mg kg-1	10.1016/j.bmc.2014.04.049
Mus musculus	Mus musculus	MTD	80.0	mg kg-1	10.1016/j.bmc.2011.12.058
Mus musculus	Mus musculus	MTD	80.0	mg/kg/day	10.1016/j.ejmech.2016.12.038
Mus musculus	Mus musculus	Tmax	1.2	hr	10.1182/blood-2009-05-222034
Mus musculus	N-terminal kinase-like protein	Activity	58.2	%	None
Mus musculus	Platelet-derived growth factor receptor	IC50	7.0	nM	10.1021/jm0204183
Mus musculus	Platelet-derived growth factor receptor	IC50	8.0	nM	10.1021/jm0204183
Mus musculus	Platelet-derived growth factor receptor	IC50	10.0	nM	10.1021/jm0204183
Mus musculus	Platelet-derived growth factor receptor	IC50	83.0	nM	10.1021/jm0204183
Mus musculus	Serine/threonine-protein kinase MST2	Kd	160.0	nM	10.1038/nbt1068
Mus musculus	ULK3 kinase	Kd	110.0	nM	10.1038/nbt1068
Mus musculus	Vascular endothelial growth factor receptor 2	IC50	73.0	nM	10.1021/acs.jmedchem.5b01582
Mycobacterium tuberculosis	Serine/threonine-protein kinase pknB	Kd	87.0	nM	10.1038/nbt.1990
Plasmodium falciparum	Calcium-dependent protein kinase 1	Kd	1300.0	nM	10.1038/nbt.1990
Plasmodium falciparum	Plasmodium falciparum	Potency	2133.1	nM	None
Plasmodium falciparum	Plasmodium falciparum	Potency	2685.5	nM	None
Plasmodium falciparum (isolate 3D7)	Cell division control protein 2 homolog	Kd	10000.0	nM	10.1038/nbt.1990
Rattus norvegicus	AMP-activated protein kinase, AMPK	IC50	62.0	nM	10.1016/j.ejmech.2022.114846
Rattus norvegicus	Androgen Receptor	AC50	5900.0	nM	10.1038/s41467-023-40064-9
Rattus norvegicus	Cyclooxygenase-1	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Rattus norvegicus	GABA receptor alpha-1 subunit	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Rattus norvegicus	Glutamate (NMDA) receptor subunit zeta 1	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Rattus norvegicus	Liver microsome	T1/2	0.4417	hr	10.1021/jm501284e
Rattus norvegicus	Peripheral myelin protein 22	Potency	10181.5	nM	None
Rattus norvegicus	Plasma	Stability	97.3	%	10.1021/acs.jmedchem.6b01266
Rattus norvegicus	Rattus norvegicus	AUC	7202.0	ng.hr.mL-1	10.1124/dmd.111.042853
Rattus norvegicus	Rattus norvegicus	AUC	11848.0	ng.hr.mL-1	10.1124/dmd.111.042853
Rattus norvegicus	Rattus norvegicus	AUC	23994.0	ng.hr.mL-1	10.1124/dmd.111.042853
Rattus norvegicus	Rattus norvegicus	CL	13.0	mL.min-1.kg-1	10.1124/dmd.111.042853
Rattus norvegicus	Rattus norvegicus	Cmax	2416.68	nM	10.1124/dmd.111.042853
Rattus norvegicus	Rattus norvegicus	Cmax	3144.45	nM	10.1124/dmd.111.042853
Rattus norvegicus	Rattus norvegicus	Cmax	4574.88	nM	10.1124/dmd.111.042853
Rattus norvegicus	Rattus norvegicus	T1/2	7.2	hr	10.1124/dmd.111.042853
Rattus norvegicus	Rattus norvegicus	T1/2	7.4	hr	10.1124/dmd.111.042853
Rattus norvegicus	Rattus norvegicus	T1/2	8.0	hr	10.1124/dmd.111.042853
Rattus norvegicus	Rattus norvegicus	Tmax	3.0	hr	10.1124/dmd.111.042853
Rattus norvegicus	Rattus norvegicus	Tmax	4.0	hr	10.1124/dmd.111.042853
Rattus norvegicus	Rattus norvegicus	Vdss	3.361	L.kg-1	10.1124/dmd.111.042853
Rattus norvegicus	Thoracic aorta	Inhibition	nan	%	10.1016/j.bmc.2015.03.085
Rattus norvegicus	Tubulin alpha-1 chain	Kd	10000.0	nM	10.1038/nbt1358
Rattus norvegicus	Voltage-gated L-type calcium channel alpha-1C subunit	AC50	30000.0	nM	10.1038/s41467-023-40064-9
Severe acute respiratory syndrome coronavirus 2	Replicase polyprotein 1ab	Inhibition	5.088	%	10.6019/CHEMBL4495564
Severe acute respiratory syndrome coronavirus 2	SARS-CoV-2	Hit score	0.1025	None	10.1101/2020.04.21.054387
Severe acute respiratory syndrome coronavirus 2	SARS-CoV-2	IC50	19952.62	nM	10.6019/CHEMBL4651402
Severe acute respiratory syndrome coronavirus 2	SARS-CoV-2	IC50	20000.0	nM	10.6019/CHEMBL4651402
Severe acute respiratory syndrome coronavirus 2	SARS-CoV-2	Inhibition	-2.05	%	10.21203/rs.3.rs-23951/v1
Severe acute respiratory syndrome coronavirus 2	SARS-CoV-2	Inhibition	-0.17	%	10.6019/CHEMBL4495565
West Nile virus	West Nile virus	EC50	550.0	nM	10.1021/acs.jmedchem.0c01467
Zika virus	Zika virus	EC50	510.0	nM	10.1021/acs.jmedchem.0c01467
None	ADMET	Activity	1.003	None	10.1073/pnas.0707498104
None	ADMET	Activity	1.019	None	10.1073/pnas.0707498104
None	ADMET	Activity	nan	None	10.1021/acs.jmedchem.0c02247
None	ADMET	Activity	nan	None	10.1021/acs.jmedchem.8b01714
None	ADMET	Activity	nan	None	10.1021/acs.jmedchem.9b00280
None	ADMET	Activity	nan	None	None
None	ADMET	CLH	13.0	uM/min.mg	10.1021/acs.jmedchem.1c00742
None	ADMET	CLH	53.0	uM/min.mg	10.1021/acs.jmedchem.1c00742
None	ADMET	Compound recovery	0.2	%	10.1124/dmd.111.042853
None	ADMET	Compound recovery	0.3	%	10.1124/dmd.111.042853
None	ADMET	Compound recovery	0.5	%	10.1124/dmd.111.042853
None	ADMET	Compound recovery	0.6	%	10.1124/dmd.111.042853
None	ADMET	Compound recovery	5.8	%	10.1124/dmd.111.042853
None	ADMET	Compound recovery	6.4	%	10.1124/dmd.111.042853
None	ADMET	Compound recovery	8.8	%	10.1124/dmd.111.042853
None	ADMET	Compound recovery	9.2	%	10.1124/dmd.111.042853
None	ADMET	Compound recovery	11.5	%	10.1124/dmd.111.042853
None	ADMET	Compound recovery	13.6	%	10.1124/dmd.111.042853
None	ADMET	Compound recovery	22.6	%	10.1124/dmd.111.042853
None	ADMET	EC50	10000.0	nM	10.1021/jm201649s
None	ADMET	FC	0.77	None	None
None	ADMET	Fu	0.007	None	10.1021/acs.jmedchem.0c02011
None	ADMET	Fu	0.009	None	10.1021/acs.jmedchem.0c02011
None	ADMET	GI50	2480.0	nM	10.1021/acs.jmedchem.6b00200
None	ADMET	IC50	5850.0	nM	10.1016/j.ejmech.2014.05.051
None	ADMET	IC50	8000.0	nM	10.1016/j.bmcl.2016.02.033
None	ADMET	IC50	19930.0	nM	10.1016/j.ejmech.2014.05.051
None	ADMET	IC50	23000.0	nM	10.1016/j.bmcl.2016.05.019
None	ADMET	IC50	23000.0	nM	10.1016/j.ejmech.2016.04.025
None	ADMET	IC50	50000.0	nM	10.1016/j.ejmech.2011.10.009
None	ADMET	IC50	75600.0	nM	10.1016/j.ejmech.2014.07.071
None	ADMET	K(p,uu,brain)	0.414	None	10.1021/acs.jmedchem.0c02011
None	ADMET	LD50	48.9	uM	10.1021/jm0204183
None	ADMET	Ratio	0.481	None	10.1021/acs.jmedchem.0c02011
None	ADMET	Ratio IC50	18.2	None	10.1021/acsmedchemlett.7b00281
None	ADMET	Selectivity Index	3.9	None	10.1021/acs.jmedchem.0c01965
None	ADMET	Stability	13.0	min	10.1016/j.bmcl.2017.12.026
None	ADMET	Stability	30.0	min	10.1016/j.bmcl.2017.12.026
None	ADMET	Stability	46.0	min	10.1016/j.bmcl.2017.12.026
None	ADMET	T1/2	0.2167	hr	10.1016/j.bmc.2017.12.020
None	ADMET	T1/2	0.2167	hr	10.1016/j.bmc.2018.08.020
None	ADMET	T1/2	0.2167	hr	None
None	ADMET	T1/2	0.4167	hr	10.1021/acs.jmedchem.1c00742
None	ADMET	T1/2	0.4633	hr	10.1021/acs.jmedchem.1c00742
None	ADMET	T1/2	0.4667	hr	None
None	ADMET	T1/2	0.5	hr	10.1016/j.bmc.2017.12.020
None	ADMET	T1/2	0.5667	hr	10.1016/j.bmc.2018.08.020
None	ADMET	T1/2	0.7667	hr	10.1016/j.bmc.2017.12.020
None	ADMET	T1/2	1.25	hr	10.1016/j.bmc.2018.08.020
None	ADMET	T1/2	1.25	hr	None
None	BC1 cell line	IC50	7248.12	nM	10.6019/CHEMBL1201861
None	COLO	Activity	0.777	None	10.1073/pnas.0707498104
None	COLO	Activity	0.844	None	10.1073/pnas.0707498104
None	COLO	Activity	0.874	None	10.1073/pnas.0707498104
None	COLO	Activity	0.897	None	10.1073/pnas.0707498104
None	COLO	Activity	0.919	None	10.1073/pnas.0707498104
None	COLO	Activity	0.929	None	10.1073/pnas.0707498104
None	COLO	Activity	0.934	None	10.1073/pnas.0707498104
None	COLO	Activity	0.964	None	10.1073/pnas.0707498104
None	COLO	Activity	0.974	None	10.1073/pnas.0707498104
None	COLO	Activity	0.985	None	10.1073/pnas.0707498104
None	COLO	Activity	0.993	None	10.1073/pnas.0707498104
None	COLO	Activity	1.074	None	10.1073/pnas.0707498104
None	COLO	Activity	1.176	None	10.1073/pnas.0707498104
None	COLO	Activity	1.269	None	10.1073/pnas.0707498104
None	Hepatotoxicity	HepSE_bilirubinemia	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_cholecystitis	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_cholelithiasis	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_cirrhosis	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_Combined Scores	2.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_elevated liver function tests	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_hepatic failure	1.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_hepatic necrosis	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_hepatitis	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_hepatomegaly	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_jaundice	1.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_liver disease	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_liver fatty	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	HepSE_liver function tests abnormal	0.0	None	10.1371/journal.pcbi.1002310
None	Hepatotoxicity	LTKB_BD DILI severity score	8.0	None	10.1016/j.drudis.2011.05.007
None	Molecular identity unknown	Activity	13.9	%	10.1016/j.ejmech.2016.07.019
None	Molecular identity unknown	Activity	18.3	%	10.1016/j.ejmech.2016.07.019
None	Molecular identity unknown	Activity	67.6	%	10.1016/j.ejmech.2016.07.019
None	NON-PROTEIN TARGET	Activity	0.54	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.613	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.676	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.687	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.697	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.718	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.729	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.737	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.745	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.759	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.779	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.788	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.79	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.792	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.793	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.802	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.804	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.806	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.807	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.815	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.825	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.833	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.834	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.837	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.842	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.845	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.846	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.85	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.855	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.857	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.858	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.859	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.864	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.866	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.869	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.875	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.881	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.889	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.89	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.892	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.896	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.898	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.9	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.902	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.903	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.909	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.912	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.914	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.916	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.917	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.924	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.927	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.93	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.933	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.935	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.936	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.937	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.938	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.939	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.94	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.943	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.944	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.945	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.946	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.951	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.952	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.953	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.955	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.956	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.958	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.959	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.961	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.965	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.968	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.972	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.974	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.977	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.979	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.98	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.981	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.983	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.984	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.985	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.987	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.988	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.989	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.99	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.991	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	0.996	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.0	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.006	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.01	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.011	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.013	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.017	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.024	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.025	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.027	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.028	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.031	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.032	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.033	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.034	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.035	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.04	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.044	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.045	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.047	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.048	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.052	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.054	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.056	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.059	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.071	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.074	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.076	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.077	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.081	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.084	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.085	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.092	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.093	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.096	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.107	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.108	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.109	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.11	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.112	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.113	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.118	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.119	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.12	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.121	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.124	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.126	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.13	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.134	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.135	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.138	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.139	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.144	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.153	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.154	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.157	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.16	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.164	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.168	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.17	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.176	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.184	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.193	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.196	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.204	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.205	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.218	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.223	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.228	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.236	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.256	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.267	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.271	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.282	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.299	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.305	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.31	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.315	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.322	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.344	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.351	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.356	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.544	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.616	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	1.624	None	10.1073/pnas.0707498104
None	NON-PROTEIN TARGET	Activity	nan	None	10.1016/j.bmcl.2009.06.022
None	NON-PROTEIN TARGET	Activity	nan	None	10.1021/jm201198w
None	NON-PROTEIN TARGET	EC50	1000.0	nM	10.1021/acs.jmedchem.6b00087
None	NON-PROTEIN TARGET	EC50	11000.0	nM	10.1016/j.ejmech.2015.11.006
None	NON-PROTEIN TARGET	EC50	13000.0	nM	10.1016/j.ejmech.2015.11.006
None	NON-PROTEIN TARGET	GI50	1.0	nM	10.1021/acs.jmedchem.6b00200
None	NON-PROTEIN TARGET	GI50	5.0	nM	10.1021/acs.jmedchem.6b00200
None	NON-PROTEIN TARGET	GI50	41.0	nM	10.1021/acs.jmedchem.6b00200
None	NON-PROTEIN TARGET	GI50	110.0	nM	10.1021/acs.jmedchem.6b00200
None	NON-PROTEIN TARGET	GI50	870.0	nM	10.1021/acs.jmedchem.6b00200
None	NON-PROTEIN TARGET	GI50	1100.0	nM	10.1021/acs.jmedchem.6b00200
None	NON-PROTEIN TARGET	GI50	1200.0	nM	10.1021/acs.jmedchem.6b00200
None	NON-PROTEIN TARGET	GI50	1700.0	nM	10.1021/acs.jmedchem.6b00200
None	NON-PROTEIN TARGET	GI50	2010.0	nM	10.1021/acs.jmedchem.6b00200
None	NON-PROTEIN TARGET	IC50	3.0	nM	10.1016/j.ejmech.2014.05.051
None	NON-PROTEIN TARGET	IC50	30.0	nM	10.1021/jm201198w
None	NON-PROTEIN TARGET	IC50	36.8	nM	10.1016/j.ejmech.2014.07.108
None	NON-PROTEIN TARGET	IC50	100.0	nM	10.1016/j.bmcl.2012.02.068
None	NON-PROTEIN TARGET	IC50	100.0	nM	10.1016/j.ejmech.2012.10.020
None	NON-PROTEIN TARGET	IC50	220.0	nM	10.1016/j.bmc.2010.01.011
None	NON-PROTEIN TARGET	IC50	830.0	nM	10.1016/j.ejmech.2014.05.051
None	NON-PROTEIN TARGET	IC50	1000.0	nM	10.1016/j.bmc.2010.05.021
None	NON-PROTEIN TARGET	IC50	1100.0	nM	10.1021/jm201198w
None	NON-PROTEIN TARGET	IC50	1200.0	nM	10.1016/j.bmc.2010.01.011
None	NON-PROTEIN TARGET	IC50	1300.0	nM	10.1016/j.bmc.2010.05.049
None	NON-PROTEIN TARGET	IC50	1300.0	nM	10.1016/j.bmc.2015.03.061
None	NON-PROTEIN TARGET	IC50	2300.0	nM	10.1021/jm800861c
None	NON-PROTEIN TARGET	IC50	2670.0	nM	10.1016/j.ejmech.2014.05.051
None	NON-PROTEIN TARGET	IC50	3030.0	nM	10.1016/j.bmcl.2016.11.089
None	NON-PROTEIN TARGET	IC50	4100.0	nM	10.1021/jm800861c
None	NON-PROTEIN TARGET	IC50	4620.0	nM	10.1016/j.ejmech.2016.09.005
None	NON-PROTEIN TARGET	IC50	4780.0	nM	10.1016/j.bmcl.2013.08.037
None	NON-PROTEIN TARGET	IC50	4950.0	nM	10.1016/j.ejmech.2016.09.005
None	NON-PROTEIN TARGET	IC50	5620.0	nM	10.1016/j.bmcl.2016.11.089
None	NON-PROTEIN TARGET	IC50	6250.0	nM	10.1016/j.bmcl.2016.11.089
None	NON-PROTEIN TARGET	IC50	7400.0	nM	10.1016/j.ejmech.2016.09.009
None	NON-PROTEIN TARGET	IC50	7440.0	nM	10.1016/j.ejmech.2016.07.019
None	NON-PROTEIN TARGET	IC50	7970.0	nM	10.1016/j.bmcl.2016.05.019
None	NON-PROTEIN TARGET	IC50	10400.0	nM	10.1016/j.ejmech.2016.09.009
None	NON-PROTEIN TARGET	IC50	12600.0	nM	10.1016/j.ejmech.2016.09.009
None	NON-PROTEIN TARGET	IC50	14400.0	nM	10.1016/j.ejmech.2016.07.019
None	NON-PROTEIN TARGET	IC50	14400.0	nM	10.1016/j.ejmech.2016.09.009
None	NON-PROTEIN TARGET	IC50	14940.0	nM	10.1016/j.bmcl.2015.05.017
None	NON-PROTEIN TARGET	IC50	15500.0	nM	10.1016/j.ejmech.2016.04.025
None	NON-PROTEIN TARGET	IC50	15500.0	nM	10.1016/j.ejmech.2016.09.009
None	NON-PROTEIN TARGET	IC50	15540.0	nM	10.1016/j.ejmech.2016.07.019
None	NON-PROTEIN TARGET	IC50	16300.0	nM	10.1016/j.ejmech.2016.09.009
None	NON-PROTEIN TARGET	IC50	16380.0	nM	10.1016/j.ejmech.2016.07.019
None	NON-PROTEIN TARGET	IC50	16400.0	nM	10.1016/j.ejmech.2016.04.025
None	NON-PROTEIN TARGET	IC50	16860.0	nM	10.1039/C1MD00105A
None	NON-PROTEIN TARGET	IC50	18600.0	nM	10.1039/C1MD00105A
None	NON-PROTEIN TARGET	IC50	19600.0	nM	10.1016/j.ejmech.2016.04.025
None	NON-PROTEIN TARGET	IC50	19600.0	nM	10.1016/j.ejmech.2016.07.019
None	NON-PROTEIN TARGET	IC50	23800.0	nM	10.1016/j.ejmech.2016.07.019
None	NON-PROTEIN TARGET	IC50	25200.0	nM	10.1016/j.ejmech.2016.09.009
None	NON-PROTEIN TARGET	IC50	55600.0	nM	10.1016/j.bmcl.2016.02.063
None	NON-PROTEIN TARGET	IC50	59750.0	nM	10.1016/j.bmcl.2016.05.019
None	NON-PROTEIN TARGET	IC50	nan	None	10.1016/j.ejmech.2016.07.019
None	NON-PROTEIN TARGET	Inhibition	nan	%	10.1016/j.bmcl.2013.04.031
None	NON-PROTEIN TARGET	MSD	32.0	day	10.1021/jm201198w
None	NON-PROTEIN TARGET	MSD	36.0	day	10.1021/jm201198w
None	NON-PROTEIN TARGET	Survival	2.6	%	10.1039/C6MD00170J
None	NON-PROTEIN TARGET	Survival	9.8	%	10.1039/C6MD00170J
None	NON-PROTEIN TARGET	Survival	54.2	%	10.1039/C6MD00170J
None	NON-PROTEIN TARGET	Survival	73.74	%	10.1039/C6MD00170J
None	No relevant target	CHI	51.0	None	10.1016/j.bmcl.2018.06.026
None	No relevant target	CHI	55.0	None	10.1016/j.bmcl.2018.06.026
None	No relevant target	CHI	57.0	None	10.1016/j.bmcl.2018.06.026
None	No relevant target	CHI	98.0	None	10.1016/j.bmcl.2018.06.026
None	No relevant target	LogD	2.51	None	10.1021/acs.jmedchem.6b01266
None	No relevant target	LogD7.4	2.26	None	10.6019/CHEMBL3301361
None	No relevant target	Retention_time	4.0	min	10.1124/dmd.111.042853
None	No relevant target	Solubility	350.0	ug.mL-1	10.1021/acs.jmedchem.0c01522
None	No relevant target	Solubility	364.0	ug.mL-1	10.1021/jm0204183
None	No relevant target	Solubility	2582.0	ug.mL-1	10.1021/jm0204183
None	No relevant target	Solubility	38000.0	nM	10.6019/CHEMBL3301361
None	No relevant target	Solubility	120000.0	nM	10.1016/j.bmcl.2018.06.026
None	No relevant target	t1/2	nan	None	10.1021/acs.jmedchem.8b01714
None	Unchecked	Activity	0.06	g	10.1021/acs.jmedchem.9b00280
None	Unchecked	Activity	0.64	g	10.1021/acs.jmedchem.9b00280
None	Unchecked	Activity	1.37	g	10.1021/acs.jmedchem.9b00280
None	Unchecked	Activity	1.87	g	10.1021/acs.jmedchem.9b00280
None	Unchecked	Activity	nan	None	10.1021/acs.jmedchem.0c02247
None	Unchecked	Activity	nan	None	10.1021/acs.jmedchem.6b01266
None	Unchecked	EC50	300.0	nM	10.1021/acsmedchemlett.8b00596
None	Unchecked	EC50	4890.0	nM	10.1016/j.ejmech.2020.112316
None	Unchecked	GI50	3.0	nM	10.1021/acs.jmedchem.6b00902
None	Unchecked	GI50	12.0	nM	10.1021/acs.jmedchem.9b00280
None	Unchecked	GI50	19.0	nM	10.1021/acs.jmedchem.9b00280
None	Unchecked	GI50	28.0	nM	10.1021/acs.jmedchem.9b00280
None	Unchecked	GI50	59.0	nM	10.1021/acs.jmedchem.9b00280
None	Unchecked	GI50	89.0	nM	10.1021/acs.jmedchem.9b00280
None	Unchecked	GI50	389.0	nM	10.1021/acs.jmedchem.9b00280
None	Unchecked	GI50	740.0	nM	10.1021/acs.jmedchem.9b00280
None	Unchecked	GI50	nan	None	10.1021/acs.jmedchem.7b00841
None	Unchecked	IC50	1.0	nM	10.1038/nchembio.117
None	Unchecked	IC50	1.4	nM	10.1016/j.ejmech.2016.12.038
None	Unchecked	IC50	3.0	nM	10.1073/pnas.0707498104
None	Unchecked	IC50	8.0	nM	10.1021/jm201198w
None	Unchecked	IC50	9.6	nM	10.1021/jm201649s
None	Unchecked	IC50	45.0	nM	10.1016/j.ejmech.2020.112316
None	Unchecked	IC50	50.0	nM	10.1021/jm0204183
None	Unchecked	IC50	80.0	nM	10.1016/j.bmcl.2012.02.068
None	Unchecked	IC50	110.0	nM	10.1038/nchembio.117
None	Unchecked	IC50	134.0	nM	10.1021/jm4004076
None	Unchecked	IC50	185.0	nM	10.1016/j.bmcl.2009.10.040
None	Unchecked	IC50	1000.0	nM	10.1016/j.bmc.2010.01.056
None	Unchecked	IC50	13600.0	nM	10.1021/jm201649s
None	Unchecked	IC50	16900.0	nM	10.1016/j.ejmech.2020.112752
None	Unchecked	IC50	nan	None	10.1016/j.bmc.2016.11.026
None	Unchecked	IC50	nan	None	10.1021/acs.jmedchem.0c01522
None	Unchecked	Inhibition	30.0	%	10.1021/acs.jmedchem.6b01266
None	Unchecked	Inhibition	33.0	%	10.1021/acs.jmedchem.6b01266
None	Unchecked	Inhibition	51.8	%	10.1016/j.ejmech.2020.112316
None	Unchecked	Inhibition	nan	%	10.1016/j.bmc.2016.11.026
None	Unchecked	Inhibition	nan	%	10.1016/j.bmcl.2010.02.110
None	Unchecked	Inhibition	nan	%	10.1016/j.bmcl.2011.09.022
None	Unchecked	Inhibition	nan	%	10.1021/acs.jmedchem.6b01266
None	Unchecked	Inhibition	nan	%	10.1021/acs.jmedchem.7b01091
None	Unchecked	Kd	0.99	nM	10.1182/blood-2009-05-222034
None	Unchecked	Kd	130.0	nM	10.1073/pnas.0707498104
None	Unchecked	Kd	1430.0	nM	10.1126/science.aan4368
None	Unchecked	Kd	3110.0	nM	10.1126/science.aan4368
None	Unchecked	Kd	10000.0	nM	10.1182/blood-2009-05-222034
None	Unchecked	Kd	30000.0	nM	10.1126/science.aan4368
None	Unchecked	logIC50	3.08	None	10.1016/j.bmc.2010.01.056
None	Unchecked	Potency	32196.8	nM	None
None	Unchecked	Ratio	10.0	None	10.1021/jm9007533
None	Unchecked	Ratio IC50	0.6	None	10.1021/jm800861c
None	Unchecked	Ratio IC50	3.0	None	10.1021/acs.jmedchem.0c02247
None	Unchecked	Ratio IC50	7.7	None	10.1016/j.bmc.2010.01.056
None	Unchecked	Ratio IC50	150.0	None	10.1021/acs.jmedchem.0c01522
None	Unchecked	TGI	75.6	%	10.1021/acs.jmedchem.9b00280
None	Unchecked	TGI	96.7	%	10.1021/acs.jmedchem.9b00280