Metabolic products of microorganisms. 268. Obscurolides, a novel class of phosphodiesterase inhibitors from streptomyces. II. Minor components belonging to the obscurolide B to D series.

The Journal of Antibiotics
1993.0

Abstract

We previously 2* reported the isolation, structural elucidation and biological properties of new phosphodiesterase inhibitors, the obscurolides A₁ to A4 (1 to 4) from the cultures of Streptomyces viridochromogenes (strain Tü 2580). A careful search for minor components by chemical screening methods 3)4) revealed eight further members of the obscurolide-complex 2) (Scheme 1). They were assigned to the B, C and D series signifying their differences in the polyketide moiety (C-1 to C-8), whereas the subscripts indicated the oxidation level of the functional group at C-4'. In this paper the isolation, physico-chemical and biological characterization of these new compounds are described. All obscurolides were isolated as diastereomeric mixtures at C-7 (A and C series) and C-5 (B series), respectively. Only in the cases of 5/6 and 9/10 could the isomers be separated.

Knowledge Graph

Similar Paper

Metabolic products of microorganisms. 268. Obscurolides, a novel class of phosphodiesterase inhibitors from streptomyces. II. Minor components belonging to the obscurolide B to D series.
The Journal of Antibiotics 1993.0
Metabolic products of microorganisms. 261. Obscurolides, a novel class of phosphodiesterase inhibitors from streptomyces. I. Production, isolation, structural elucidation and biological activity of obscurolides A1 to A4.
The Journal of Antibiotics 1992.0
Streptoglycerides A–D with a Rare 6/5/5 Tricyclic Ring Skeleton from a Marine Actinomycete <i>Streptomyces</i> species
Organic Letters 2018.0
Tartrolone C:  A Novel Insecticidal Macrodiolide Produced by <i>Streptomyces</i> sp. CP1130
Journal of Natural Products 2003.0
Tartrolone C:  A Novel Insecticidal Macrodiolide Produced by <i>Streptomyces</i> sp. CP1130
Journal of Natural Products 2003.0
Microbial Metabolites of Ophiobolin A and Antimicrobial Evaluation of Ophiobolins
Journal of Natural Products 1995.0
Osmanicin, a Polyketide Alkaloid Isolated from Streptomyces osmaniensis CA-244599 Inhibits Elastase in Human Fibroblasts
Molecules 2019.0
Osmanicin, a Polyketide Alkaloid Isolated from Streptomyces osmaniensis CA-244599 Inhibits Elastase in Human Fibroblasts
Molecules 2019.0
Isolation and Structure Determination of Novel Phosphatidylinositol Kinase Inhibitors, Echiguanines A and B, from Streptomyces sp.
Journal of Natural Products 1991.0
Isolation and Structure Determination of Novel Phosphatidylinositol Kinase Inhibitors, Echiguanines A and B, from Streptomyces sp.
Journal of Natural Products 1991.0