Structure of brassicicolin A: a novel isocyanide antibiotic from the phylloplane fungus Alternaria brassicicola

The Journal of Organic Chemistry
1988.0

Abstract

Studies of the secondary metabolites produced in culture by the plant pathogenic phylloplane fungus Alternaria brassicicola (Schweinitz) Wiltshire (NRRL 1299 = ATCC 6650) have led to the isolation of brassicicolin A (6), a novel isocyanide antibiotic with potent in vitro activity against the gram-positive bacteria Bacillus subtilis and Staphylococcus aureus. Brassicicolin A is a fully acylated derivative of D-mannitol containing two D-α-hydroxyisovaleryl units, two acetyl groups, and two epimerized α-isocyanoisovaleryl units. The structure of brassicicolin A was assigned as 6 primarily through chemical degradation studies and by NMR and mass spectral analysis of its deisocyanation product. This account represents the first report of the α-isocyanoisovaleryl group as a naturally occurring structural unit.

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