The SAR of UK-78,282: A novel blocker of human T cell Kv1.3 potassium channels

The SAR of UK-78,282: A novel blocker of human T cell Kv1.3 potassium channels Khellinone Derivatives as Blockers of the Voltage-Gated Potassium Channel Kv1.3:  Synthesis and Immunosuppressive Activity Angular Methoxy-Substituted Furo- and Pyranoquinolinones as Blockers of the Voltage-Gated Potassium Channel Kv1.3 Development of an automated screen for Kv7.2 potassium channels and discovery of a new agonist chemotype Initial SAR studies on apamin-displacing 2-aminothiazole blockers of calcium-activated small conductance potassium channels Discovery of potent T-type calcium channel blocker Structure–activity relationship exploration of Kv1.3 blockers based on diphenoxylate Morpholin-2-one derivatives as novel selective T-type Ca2+ channel blockers Design, synthesis and biological activity of pyrazolo[1,5-a]pyrimidin-7(4H)-ones as novel Kv7/KCNQ potassium channel activators Synthesis and Pharmacological Characterization of Conformationally Restricted Retigabine Analogues as Novel Neuronal Kv7 Channel Activators