Identification of a potent analogue of Nazumamide A through iteration of combinatorial tetrapeptide libraries

Identification of a potent analogue of Nazumamide A through iteration of combinatorial tetrapeptide libraries Nazumazoles D–F, Cyclic Pentapeptides That Inhibit Chymotrypsin, from the Marine Sponge Theonella swinhoei (3S)-N-(l-Aminoacyl)-1,2,3,4-tetrahydroisoquinolines, a class of novel antithrombotic agents: Synthesis, bioassay, 3D QSAR, and ADME analysis Inhibition studies of some serine and thiol proteinases by new leupeptin analogs Total Synthesis and Full Histone Deacetylase Inhibitory Profiling of Azumamides A–E as Well as β²- epi-Azumamide E and β³-epi-Azumamide E A class of oral N-[(1S,3S)-1-methyl-1,2,3,4-tetrahydro-β-carboline-3-carbonyl]- N′-(amino-acid-acyl)hydrazine: Discovery, synthesis, in vitro anti-platelet aggregation/in vivo anti-thrombotic evaluation and 3D QSAR analysis Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor Bacithrocins A, B and C, novel thrombin inhibitors. Preparation of l-proline based aeruginosin 298-A analogs: Optimization of the P1-moiety AMP Deaminase Inhibitors. 5. Design, Synthesis, and SAR of a Highly Potent Inhibitor Series