Design and synthesis of highly potent fumagillin analogues from homology modeling for a human MetAP-2

Design and synthesis of highly potent fumagillin analogues from homology modeling for a human MetAP-2 Fumarranol, a Rearranged Fumagillin Analogue That Inhibits Angiogenesis in Vivo Design, synthesis and evaluation of a cellular stable and detectable biotinylated fumagillin probe and investigation of cell permeability of fumagillin and its analogs to endothelial and cancer cells Synthesis and antitumor activity of 1,3,4-oxadiazole possessing 1,4-benzodioxan moiety as a novel class of potent methionine aminopeptidase type II inhibitors Metabolites of PPI-2458, a Selective, Irreversible Inhibitor of Methionine Aminopeptidase-2: Structure Determination and In Vivo Activity Antiparasitic activities of novel, orally available fumagillin analogs Total synthesis and antiangiogenic activity of cyclopentane analogues of fumagillol Discovery and Structural Modification of Inhibitors of Methionine Aminopeptidases from Escherichia coli and Saccharomyces cerevisiae Novel potent 2,5-pyrrolidinedione peptidomimetics as aminopeptidase N inhibitors. Design, synthesis and activity evaluation Synthesis and bioevaluation of 22-hydroxyacuminatine analogs