Design, total synthesis, and biological evaluation of neodysiherbaine A derivative as potential probes

Design, total synthesis, and biological evaluation of neodysiherbaine A derivative as potential probes Hydroxymethyl bioisosteres of phenolic GluN2B-selective NMDA receptor antagonists: Design, synthesis and pharmacological evaluation 4-Hydroxy-1,2,5-oxadiazol-3-yl Moiety as Bioisoster of the Carboxy Function. Synthesis, Ionization Constants, and Molecular Pharmacological Characterization at Ionotropic Glutamate Receptors of Compounds Related to Glutamate and Its Homologues N-Hydroxypyrazolyl Glycine Derivatives as SelectiveN-Methyl-<scp>d</scp>-aspartic Acid Receptor Ligands 3-Hydroxy-1H-quinazoline-2,4-dione derivatives as new antagonists at ionotropic glutamate receptors: Molecular modeling and pharmacological studies Use of the 4-Hydroxytriazole Moiety as a Bioisosteric Tool in the Development of Ionotropic Glutamate Receptor Ligands Synthesis and Biological Characterization of 3-Substituted 1H-Indoles as Ligands of GluN2B-ContainingN-Methyl-<scp>d</scp>-aspartate Receptors. Part 2 Development of 2′-Substituted (2S,1′R,2′S)-2-(Carboxycyclopropyl)glycine Analogues as Potent N-Methyl-<scp>d</scp>-aspartic Acid Receptor Agonists A monocyclic neodysiherbaine analog: Synthesis and evaluation Chemo-Enzymatic Synthesis of a Series of 2,4-Syn-Functionalized (S)-Glutamate Analogues: New Insight into the Structure−Activity Relation of Ionotropic Glutamate Receptor Subtypes 5, 6, and 7