Non-steroidal glucocorticoid agonists—The discovery of aryl pyrazoles as A-ring mimetics

Non-steroidal glucocorticoid agonists—The discovery of aryl pyrazoles as A-ring mimetics Dissociated Nonsteroidal Glucocorticoid Receptor Modulators; Discovery of the Agonist Trigger in a Tetrahydronaphthalene−Benzoxazine Series Nonsteroidal Glucocorticoid Agonists: Tetrahydronaphthalenes with Alternative Steroidal A-Ring Mimetics Possessing Dissociated (Transrepression/Transactivation) Efficacy Selectivity Structure Guided Design of 5-Arylindazole Glucocorticoid Receptor Agonists and Antagonists 1H-Pyrazolo[3,4-g]hexahydro-isoquinolines as selective glucocorticoid receptor antagonists with high functional activity Octahydrophenanthrene-2,7-diol Analogues as Dissociated Glucocorticoid Receptor Agonists: Discovery and Lead Exploration 2-Benzenesulfonyl-8a-benzyl-hexahydro-2H-isoquinolin-6-ones as selective glucocorticoid receptor antagonists Trifluoromethyl group as a pharmacophore: Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand Potent nonsteroidal progesterone receptor agonists: Synthesis and SAR study of 6-aryl benzoxazines Novel pyrrole-containing progesterone receptor modulators