Syntheses of novel myxopyronin B analogs as potential inhibitors of bacterial RNA polymerase

Bioorganic & Medicinal Chemistry Letters
2007.0

Abstract

Based upon observations from our initial findings, additional myxopyronin B analogs have been prepared and tested for in vitro inhibitory activity against DNA-dependent RNA polymerase and antibacterial activity against Escherichia coli and Staphylococcus aureus.

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