Binaphthyl scaffolded peptoids via ring-closing metathesis reactions and their anti-bacterial activities

Bioorganic & Medicinal Chemistry Letters
2009.0

Abstract

An efficient synthesis of four new acyclic and four new cyclic binaphthyl-based cationic peptoids is described. These compounds had anti-bacterial activities with MIC values of 4-62 microg/mL against Staphylococcus aureus.

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