The Structure−Activity Relationship of the Antimalarial Ozonide Arterolane (OZ277)

The Structure−Activity Relationship of the Antimalarial Ozonide Arterolane (OZ277) Structure–Activity Relationship of the Antimalarial Ozonide Artefenomel (OZ439) The comparative antimalarial properties of weak base and neutral synthetic ozonides Comparative Antimalarial Activities and ADME Profiles of Ozonides (1,2,4-trioxolanes) OZ277, OZ439, and Their 1,2-Dioxolane, 1,2,4-Trioxane, and 1,2,4,5-Tetraoxane Isosteres Identification and Optimization of an Aminoalcohol-Carbazole Series with Antimalarial Properties Enantioselective Synthesis and in Vivo Evaluation of Regioisomeric Analogues of the Antimalarial Arterolane Peroxide Bond-Dependent Antiplasmodial Specificity of Artemisinin and OZ277 (RBx11160) Conjugation of N -acylhydrazone and 1,2,4-oxadiazole leads to the identification of active antimalarial agents Mechanism-Based Design of Parasite-Targeted Artemisinin Derivatives:  Synthesis and Antimalarial Activity of Benzylamino and Alkylamino Ether Analogues of Artemisinin 1-Azaaurones derived from the naturally occurring aurones as potential antimalarial drugs