Synthesis and screening of ( E )-1-(β- d -galactopyranosyl)-4-(aryl)but-3-ene-2-one against Mycobacterium tuberculosis

Bioorganic & Medicinal Chemistry Letters
2011.0

Abstract

A series of galactose-derived aryl enones were synthesised and screened against Mycobacterium tuberculosis H(37)Rv. Preliminary results were promising with MIC values in the range 1.56-12.5 μg/mL.

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