Optimization of O₃-Acyl Kojic Acid Derivatives as Potent and Selective Human Neutrophil Elastase Inhibitors

Optimization of O₃-Acyl Kojic Acid Derivatives as Potent and Selective Human Neutrophil Elastase Inhibitors Exploration of nitrogen heterocycle scaffolds for the development of potent human neutrophil elastase inhibitors Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastase Simple phosphonic inhibitors of human neutrophil elastase 1,5,6,7-Tetrahydro-4H-indazol-4-ones as human neutrophil elastase (HNE) inhibitors Synthesis and pharmacological characterization of 2-aminobenzaldehyde oxime analogs as dual inhibitors of neutrophil elastase and proteinase 3 Chemical constituents from the leaves of Ilex paraguariensis inhibit human neutrophil elastase Synthesis of N-kojic-amino acid and N-kojic-amino acid-kojiate and their tyrosinase inhibitory activity Highly potent and selective inhibitors of endothelin converting enzyme Evaluation of human neutrophil elastase inhibitory effect of iridoid glycosides from Hedyotis diffusa