Computational discovery and biological evaluation of novel inhibitors targeting histone-lysine N-methyltransferase SET7

Computational discovery and biological evaluation of novel inhibitors targeting histone-lysine N-methyltransferase SET7 Discovery and Optimization of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Pharmacophore- and Docking-Based Virtual Screening Identifying Novel Selective Non-Nucleoside DNA Methyltransferase 1 Inhibitors through Docking-Based Virtual Screening Identification of Cyproheptadine as an Inhibitor of SET Domain Containing Lysine Methyltransferase 7/9 (Set7/9) That Regulates Estrogen-Dependent Transcription Identification of the KDM2/7 Histone Lysine Demethylase Subfamily Inhibitor and its Antiproliferative Activity 5-Aminonaphthalene derivatives as selective nonnucleoside nuclear receptor binding SET domain-protein 2 (NSD2) inhibitors for the treatment of multiple myeloma Novel and selective DNA methyltransferase inhibitors: Docking-based virtual screening and experimental evaluation Identification of DOT1L inhibitors by structure-based virtual screening adapted from a nucleoside-focused library 4-Hydroxy-3-methylbenzofuran-2-carbohydrazones as novel LSD1 inhibitors Steric structure–activity relationship of cyproheptadine derivatives as inhibitors of histone methyltransferase Set7/9