Antibacterial p-Terphenyl with a Rare 2,2′-Bithiazole Substructure and Related Compounds Isolated from the Marine-Derived Actinomycete Nocardiopsis sp. HDN154086

Journal of Natural Products
2021.0

Abstract

Assisted by MS/MS-based molecular networking and X-ray diffraction analysis, five new <i>p</i>-terphenyl derivatives, namely, nocarterphenyls D-H (<b>1</b>-<b>5</b>), were obtained and characterized from the cultures of the marine sediment-derived actinomycete <i>Nocardiopsis</i> sp. HDN154086. The skeleton of nocarterphenyl D (<b>1</b>) was defined to possess a rare 2,2'-bithiazole scaffold, naturally occurring for the first time, and nocarterphenyls E-H (<b>2</b>-<b>5</b>) are <i>p</i>-terphenylquinones with unusual thioether linked fatty acid methyl ester substitutions. Compound <b>1</b> showed promising activity against multiple bacteria with MIC values ranging from 1.5 to 6.2 μM, and <b>2</b> exhibited notable antibacterial activity against MRSA which surpassed the positive control ciprofloxacin.

Knowledge Graph

Similar Paper

Antibacterial p-Terphenyl with a Rare 2,2′-Bithiazole Substructure and Related Compounds Isolated from the Marine-Derived Actinomycete Nocardiopsis sp. HDN154086
Journal of Natural Products 2021.0
Cytotoxic <i>p</i>-Terphenyls from a Marine-Derived <i>Nocardiopsis</i> Species
Journal of Natural Products 2019.0
Isolation and Characterization of New <i>p</i>-Terphenyls with Antifungal, Antibacterial, and Antioxidant Activities from Halophilic Actinomycete <i>Nocardiopsis gilva</i> YIM 90087
Journal of Agricultural and Food Chemistry 2013.0
Isolation and Characterization of New <i>p</i>-Terphenyls with Antifungal, Antibacterial, and Antioxidant Activities from Halophilic Actinomycete <i>Nocardiopsis gilva</i> YIM 90087
Journal of Agricultural and Food Chemistry 2013.0
α-Pyrones and Diketopiperazine Derivatives from the Marine-Derived Actinomycete Nocardiopsis dassonvillei HR10-5
Journal of Natural Products 2011.0
α-Pyrones and Diketopiperazine Derivatives from the Marine-Derived Actinomycete Nocardiopsis dassonvillei HR10-5
Journal of Natural Products 2011.0
Secondary Metabolites from an Actinomycete from Vietnam's East Sea
Natural Product Communications 2016.0
Antimicrobial metabolites from a novel halophilic actinomycete<i>Nocardiopsis terrae</i>YIM 90022
Natural Product Research 2014.0
New bioactive compounds from the marine-derived actinomycete <i>Nocardiopsis lucentensis</i> sp. ASMR2
Zeitschrift für Naturforschung B 2017.0
Nocarimidazoles A and B from a Marine-Derived Actinomycete of the Genus <i>Nocardiopsis</i>
Journal of Natural Products 2015.0