B-5354a, b and c, New Sphingosine Kinase Inhibitors, Produced by a Marine Bacterium. Taxonomy, Fermentation, Isolation, Physico-chemical Properties and Structure Determination.

The Journal of Antibiotics
2000.0

Abstract

In the course of our screening for inhibitors of sphingosine kinase, we found a series of active compounds in a culture broth of a novel marine bacterium, SANK71896. The structures of the compounds, named B-5354a, b and c, were elucidated by a combination of spectroscopic analyses to be new esters of 4-amino-3-hydroxybenzoic acid with long-chain unsaturated alcohols. B-5354a, b and c inhibit sphingosine kinase activity with IC50 values of 21, 58 and 38 μM, respectively. Here we report on the taxonomy of the producing organism as well as the fermentation, isolation, physico-chemical properties and structure determination of the new compounds.

Knowledge Graph

Similar Paper

B-5354a, b and c, New Sphingosine Kinase Inhibitors, Produced by a Marine Bacterium. Taxonomy, Fermentation, Isolation, Physico-chemical Properties and Structure Determination.
The Journal of Antibiotics 2000.0
Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure–activity relationship study of 4-epi-jaspine B
Bioorganic & Medicinal Chemistry 2017.0
Isolation and Structure Determination of Novel Phosphatidylinositol Kinase Inhibitors, Echiguanines A and B, from Streptomyces sp.
Journal of Natural Products 1991.0
Isolation and Structure Determination of Novel Phosphatidylinositol Kinase Inhibitors, Echiguanines A and B, from Streptomyces sp.
Journal of Natural Products 1991.0
Structure elucidation of Sch 538415, a novel acyl carrier protein synthase inhibitor from a microorganism
Bioorganic & Medicinal Chemistry Letters 2003.0
Structure-activity relationship of short-chain sphingoid bases as inhibitors of sphingosine kinase
Bioorganic & Medicinal Chemistry Letters 1999.0
Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C
Bioorganic & Medicinal Chemistry 2011.0
Synthesis and Evaluation of Sphingosine Analogues as Inhibitors of Sphingosine Kinases
Journal of Medicinal Chemistry 2009.0
Rare phenazine L-quinovose esters from a marine actinomycete
The Journal of Organic Chemistry 1992.0
A New Bicyclic Guanidine Alkaloid, Sch 575948, from a Marine Sponge, Ptilocaulis spiculifer
The Journal of Antibiotics 2003.0