Purealidins J-R, New Bromotyrosine Alkaloids from the Okinawan Marine Sponge Psammaplysilla purea.

Chemical and Pharmaceutical Bulletin
1995.0

Abstract

Nine new bromotyrosine alkaloids, purealidins J—R (1—9), have been isolated from the Okinawan marine sponge Psammaplysilla purea and the structures were elucidated on the basis of spectroscopic data. A hydroxy group at C-1 of purealidins M—O (4—6) may be biosynthetically derived from ring-opening of a spirocyclohexadienyl-isoxazole unit of purealidin J (1), aerophobin-1 (10), and purealidin L (3), respectively. Purealidins N (5), P (7), and Q (8) were cytotoxic to tumor cell lines, while purealidins J (1), K (2), P (7), and Q (8) showed moderate inhibitory activity against epidermal growth factor (EGF) receptor kinase. © 1995, The Pharmaceutical Society of Japan. All rights reserved.

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