Differential binding and dopamine uptake activity of cocaine analogues modified at nitrogen

Differential binding and dopamine uptake activity of cocaine analogues modified at nitrogen Methoxylation of cocaine reduces binding affinity and produces compounds of differential binding and dopamine uptake inhibitory activity: discovery of a weak cocaine "antagonist" Structure-Activity Relationship Studies of N-Sulfonyl Analogs of Cocaine: Role of Ionic Interaction in Cocaine Binding Synthesis of 3-arylecgonine analogs as inhibitors of cocaine binding and dopamine uptake Synthesis of 3-carbamoylecgonine methyl ester analogs as inhibitors of cocaine binding and dopamine uptake N-Modified analogs of cocaine: synthesis and inhibition of binding to the cocaine receptor Synthesis of 8-oxa analogues of norcocaine endowed with interesting cocaine-like activity Novel 3.alpha.-(Diphenylmethoxy)tropane Analogs: Potent Dopamine Uptake Inhibitors without Cocaine-like Behavioral Profiles Synthesis, Dopamine Transporter Affinity, Dopamine Uptake Inhibition, and Locomotor Stimulant Activity of 2-Substituted 3β-Phenyltropane Derivatives (−)-3β-Substituted Ecgonine Methyl Esters as Inhibitors for Cocaine Binding and Dopamine Uptake