Synthesis, biological in vitro evaluation and stereoselectivity of ondansetron analogues: novel 5-HT2A receptor antagonists

Synthesis, biological in vitro evaluation and stereoselectivity of ondansetron analogues: novel 5-HT2A receptor antagonists 5-HT2 antagonist activity of 3-aminomethyltetralones Thiazole as a carbonyl bioisostere. A novel class of highly potent and selective 5-HT3 receptor antagonists Design and synthesis of novel ligands for the 5-HT3 and the 5-HT4 receptor Potent, Selective Tetrahydro-β-carboline Antagonists of the Serotonin 2B (5HT_2B) Contractile Receptor in the Rat Stomach Fundus New aporphinoid 5-HT2A and α1A antagonists via structural manipulations of nantenine (±)-Nantenine analogs as antagonists at human 5-HT2A receptors: C1 and flexible congeners Zatosetron, a potent, selective, and long-acting 5HT3 receptor antagonist: synthesis and structure-activity relationships Discovery of novel potent and selective ligands for 5-HT2A receptor with quinazoline scaffold Benzimidazole, Benzoxazole and Benzothiazole Derivatives as 5HT2B Receptor Ligands. Synthesis and Preliminary Pharmacological Evaluation