Synthesis, antimicrobial activity and binding properties of calix[4]arene based vancomycin mimics

Bioorganic & Medicinal Chemistry Letters
1996.0

Abstract

Biologically active Vancomycin antibiotic mimics have been synthesized by linking two opposite aromatic nuclei of a calix[4]arene derivative in the cone conformation with a polifunctional bridge containing D- or L- alanine units and a diethylentriamine segment.

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