Synthesis, anticholinesterase activity and structure–Activity relationships of m-Aminobenzoic acid derivatives

Bioorganic & Medicinal Chemistry Letters
2003.0

Abstract

The synthesis, acetylcholinesterase inhibitory capacity and structure-activity relationships of simple-structured m-Aminobenzoic acid derivatives are reported. Compound 1b was found to be more potent than galanthamine and tacrine in inhibiting acetylcholinesterase.

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