An Evaluation of a C-Glucuronide as a liver targeting group: conjugate of a glucocorticoid antagonist

An Evaluation of a C-Glucuronide as a liver targeting group: conjugate of a glucocorticoid antagonist Bile acid conjugates of a nonsteroidal glucocorticoid receptor modulator Synthesis and activity of novel bile-acid conjugated glucocorticoid receptor antagonists Discovery of novel phosphorus-containing steroids as selective glucocorticoid receptor antagonist Parallel strategies for the preparation and selection of liver-targeted glucocorticoid receptor antagonists Liver-Selective Glucocorticoid Antagonists:  A Novel Treatment for Type 2 Diabetes Discovery of a Potent Steroidal Glucocorticoid Receptor Antagonist with Enhanced Selectivity against the Progesterone and Androgen Receptors (OP-3633) 1H-Pyrazolo[3,4-g]hexahydro-isoquinolines as selective glucocorticoid receptor antagonists with high functional activity Identification of the Clinical Candidate (R)-(1-(4-Fluorophenyl)-6-((1-methyl-1H-pyrazol-4-yl)sulfonyl)-4,4a,5,6,7,8-hexahydro-1H-pyrazolo[3,4-g]isoquinolin-4a-yl)(4-(trifluoromethyl)pyridin-2-yl)methanone (CORT125134): A Selective Glucocorticoid Receptor (GR) Antagonist Syntheses and Antigestagenic Activity of Mifepristone Derivatives