GABAA Receptor Agonists, Partial Agonists, and Antagonists. Design and Therapeutic Prospects

GABAA Receptor Agonists, Partial Agonists, and Antagonists. Design and Therapeutic Prospects Discovery of non-Zwitterionic GABAA receptor full agonists and a superagonist Activation of the γ-Aminobutyric Acid Type B (GABA_B) Receptor by Agonists and Positive Allosteric Modulators GABA-Activated Ligand Gated Ion Channels:  Medicinal Chemistry and Molecular Biology Partial GABAA Receptor Agonists. Synthesis and in Vitro Pharmacology of a Series of Nonannulated Analogs of 4,5,6,7-Tetrahydroisoxazolo[4,5-c]pyridin-3-ol Bioisosteric determinants for subtype selectivity of ligands for heteromeric GABAA receptors Synthesis and pharmacological evaluation of 6-aminonicotinic acid analogues as novel GABAA receptor agonists Phosphinic Acid Analogs of GABA. 1. New Potent and Selective GABAB Agonists Synthesis and Pharmacological Evaluation of Novel γ-Aminobutyric Acid Type B (GABA_B) Receptor Agonists as Gastroesophageal Reflux Inhibitors Novel γ-Aminobutyric Acid ρ₁Receptor Antagonists; Synthesis, Pharmacological Activity and Structure−Activity Relationships