Discovery of non-Zwitterionic GABAA receptor full agonists and a superagonist

Discovery of non-Zwitterionic GABAA receptor full agonists and a superagonist Activation of the γ-Aminobutyric Acid Type B (GABA_B) Receptor by Agonists and Positive Allosteric Modulators N-(Indol-3-ylglyoxylyl)piperidines: high affinity agonists of human GABA-A receptors containing the α1 subunit (±)-2-amino-2-thiazoline-4-ethanoic acid; a novel, specific GABAA receptor agonist GABAA Receptor Agonists, Partial Agonists, and Antagonists. Design and Therapeutic Prospects Synthesis and pharmacological evaluation of 6-aminonicotinic acid analogues as novel GABAA receptor agonists Hydroxy-1,2,5-oxadiazolyl Moiety as Bioisoster of the Carboxy Function. Synthesis, Ionization Constants, and Pharmacological Characterization of γ-Aminobutyric Acid (GABA) Related Compounds Bioisosteric determinants for subtype selectivity of ligands for heteromeric GABAA receptors GABA-Activated Ligand Gated Ion Channels:  Medicinal Chemistry and Molecular Biology Five-Membered N-Heterocyclic Scaffolds as Novel Amino Bioisosteres at γ-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters