Indole-3-acetic Acid Antagonists of the Prostaglandin D₂ Receptor CRTH2

Indole-3-acetic Acid Antagonists of the Prostaglandin D₂ Receptor CRTH2 Update on the Development of Antagonists of Chemoattractant Receptor-Homologous Molecule Expressed on Th2 Cells (CRTH2). From Lead Optimization to Clinical Proof-of-Concept in Asthma and Allergic Rhinitis Discovery of selective indole-based prostaglandin D2 receptor antagonist Discovery of new chemical leads for prostaglandin D2 receptor antagonists Development and Characterization of New Inhibitors of the Human and Mouse Hematopoietic Prostaglandin D₂Synthases Acidic furo[3,2-b]indoles. A new series of potent antiallergy agents Synthesis and structure–activity relationship of 1H-indole-3-carboxylic acid pyridine-3-ylamides: A novel series of 5-HT2C receptor antagonists N-Arylsulfonyl-α-amino carboxamides are potent and selective inhibitors of the chemokine receptor CCR10 that show efficacy in the murine DNFB model of contact hypersensitivity Identification and characterisation of new inhibitors for the human hematopoietic prostaglandin D 2 synthase Pyroglutamide-Based P2X7 Receptor Antagonists Targeting Inflammatory Bowel Disease