Discovery of selective indole-based prostaglandin D2 receptor antagonist

Discovery of selective indole-based prostaglandin D2 receptor antagonist Discovery of new chemical leads for prostaglandin D2 receptor antagonists Indole-3-acetic Acid Antagonists of the Prostaglandin D₂ Receptor CRTH2 3-Phenyl-5-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]indole-2-carbonitrile, a potent inhibitor of prostaglandin synthetase and of platelet aggregation Discovery of benzo[g]indol-3-carboxylates as potent inhibitors of microsomal prostaglandin E2 synthase-1 Synthesis and structure–activity relationships of 4-oxo-1-phenyl-3,4,6,7-tetrahydro-[1,4]diazepino[6,7,1- hi ]indoles: novel PDE4 inhibitors Antiinflammatory activity of N-(2-benzoylphenyl)alanine derivatives From indomethacin to a selective COX-2 inhibitor: Development of indolalkanoic acids as potent and selective cyclooxygenase-2 inhibitors Antihypertensive indole derivatives of phenoxypropanolamines with .beta.-adrenergic receptor antagonist and vasodilating activity Synthesis and Structure−Activity Relationships of Novel Histamine H₁ Antagonists:  Indolylpiperidinyl Benzoic Acid Derivatives