Design, synthesis and SAR studies of tripeptide analogs with the scaffold 3-phenylpropane-1,2-diamine as aminopeptidase N/CD13 inhibitors

Design, synthesis and SAR studies of tripeptide analogs with the scaffold 3-phenylpropane-1,2-diamine as aminopeptidase N/CD13 inhibitors Novel 3-phenylpropane-1,2-diamine derivates as inhibitors of aminopeptidase N (APN) Novel aminopeptidase N (APN/CD13) inhibitors derived from 3-phenylalanyl-N′-substituted-2,6-piperidinedione Design, synthesis and primary activity assay of bi- or tri-peptide analogues with the scaffold l-arginine as amino-peptidase N/CD13 inhibitors Novel aminopeptidase N (APN/CD13) inhibitors derived from chloramphenicol amine Novel indoline-2,3-dione derivatives as inhibitors of aminopeptidase N (APN) Novel aminopeptidase N inhibitors derived from 1,3,4-thiadiazole scaffold Novel cyclic-imide peptidomimetics as aminopeptidase N inhibitors. Design, chemistry and activity evaluation. Part I Novel Human Aminopeptidase N Inhibitors: Discovery and Optimization of Subsite Binding Interactions Novel leucine ureido derivatives as aminopeptidase N inhibitors. Design, synthesis and activity evaluation