Identification of Peptide Substrate and Small Molecule Inhibitors of Testis-Specific Serine/Threonine Kinase1 (TSSK1) By the Developed Assays

Identification of Peptide Substrate and Small Molecule Inhibitors of Testis-Specific Serine/Threonine Kinase1 (TSSK1) By the Developed Assays Array-based fluorescence assay for serine/threonine kinases using specific chemical reaction In vitro and in silico studies on substrate recognition and acceptance of human PKMYT1, a Cdk1 inhibitory kinase PAIN-less identification and evaluation of small molecule inhibitors against protein tyrosine phosphatase 1B Development of a novel fluorescent probe for fluorescence correlation spectroscopic detection of kinase inhibitors Inhibitors of Tripeptidyl Peptidase II. 2. Generation of the First Novel Lead Inhibitor of Cholecystokinin-8-Inactivating Peptidase:  A Strategy for the Design of Peptidase Inhibitors Virtual Docking Approaches to Protein Kinase B Inhibition Discovery of inhibitors of the mitotic kinase TTK based on N-(3-(3-sulfamoylphenyl)-1H-indazol-5-yl)-acetamides and carboxamides Design of new inhibitors for cdc2 kinase based on a multiple pseudosubstrate structure C-terminal constrained phenylalanine as a pharmacophoric unit in peptide-based proteasome inhibitors