Artemisinin-dipeptidyl vinyl sulfone hybrid molecules: Design, synthesis and preliminary SAR for antiplasmodial activity and falcipain-2 inhibition

Artemisinin-dipeptidyl vinyl sulfone hybrid molecules: Design, synthesis and preliminary SAR for antiplasmodial activity and falcipain-2 inhibition Design, Synthesis, and Antiplasmodial Activity of Hybrid Compounds Based on (2R,3S)-N-Benzoyl-3-phenylisoserine N 1-{4-[(10S)-Dihydroartemisinin-10-oxyl]}phenylmethylene-N 2-(2-methylquinoline-4-yl)hydrazine derivatives as antiplasmodial falcipain-2 inhibitors A novel artemisinin–quinine hybrid with potent antimalarial activity Synthesis of Novel G Factor or Chloroquine-Artemisinin Hybrids and Conjugates with Potent Antiplasmodial Activity Artemisinin–quinoline hybrid-dimers: Synthesis and in vitro antiplasmodial activity Anti- Plasmodium falciparum activity of quinoline–sulfonamide hybrids Aza vinyl sulfones: Synthesis and evaluation as antiplasmodial agents Tetraoxane–Pyrimidine Nitrile Hybrids as Dual Stage Antimalarials Synthesis, in vitro antiplasmodial activity and cytotoxicity of a series of artemisinin–triazine hybrids and hybrid-dimers