Total synthesis of a biotinylated rocaglate: Selective targeting of the translation factors eIF4AI/II

Total synthesis of a biotinylated rocaglate: Selective targeting of the translation factors eIF4AI/II Design, synthesis, and biological evaluation of biotin-labeled (−)-ternatin, a potent fat-accumulation inhibitor against 3T3-L1 adipocytes Synthesis and antitumor activity of biotinylated camptothecin derivatives as potent cytotoxic agents Design and Synthesis of Biotinylated Bivalent Carboline Derivatives as Potent Antitumor Agents Synthesis and Biological Evaluation of a Biotinylated Paclitaxel with an Extra-Long Chain Spacer Arm Design of Development Candidate eFT226, a First in Class Inhibitor of Eukaryotic Initiation Factor 4A RNA Helicase Biotin Derivatives Carrying Two Chelating DOTA Units. Synthesis, in Vitro Evaluation of Biotinidases Resistance, Avidin Binding, and Radiolabeling Tests ‘Click’ glycosylation of peptides through cysteine propargylation and CuAAC Synthetic Analogue of Rocaglaol Displays a Potent and Selective Cytotoxicity in Cancer Cells: Involvement of Apoptosis Inducing Factor and Caspase-12 Diastereoselective synthesis of (2S,4R)-4-Methylglutamic acid (sym 2081): A high affinity and selective ligand at the kainate subtype of glutamate receptors