SGC-AAK1-1: A Chemical Probe Targeting AAK1 and BMP2K

SGC-AAK1-1: A Chemical Probe Targeting AAK1 and BMP2K SGC-GAK-1: A Chemical Probe for Cyclin G Associated Kinase (GAK) Bicyclic Heterocyclic Replacement of an Aryl Amide Leading to Potent and Kinase-Selective Adaptor Protein 2-Associated Kinase 1 Inhibitors Discovery of 2-pyrimidyl-5-amidothiophenes as potent inhibitors for AKT: Synthesis and SAR studies Design and Synthesis of Pyrazole-Based Macrocyclic Kinase Inhibitors Targeting BMPR2 Discovery of a novel protein kinase B inhibitor by structure-based virtual screening Discovery, Structure–Activity Relationships, and In Vivo Evaluation of Novel Aryl Amides as Brain Penetrant Adaptor Protein 2-Associated Kinase 1 (AAK1) Inhibitors for the Treatment of Neuropathic Pain Discovery of 2-arylquinazoline derivatives as a new class of ASK1 inhibitors Discovery of a Selective and Potent Inhibitor of Mitogen-Activated Protein Kinase-Interacting Kinases 1 and 2 (MNK1/2) Utilizing Structure-Based Drug Design A 2,6,9-hetero-trisubstituted purine inhibitor exhibits potent biological effects against multiple myeloma cells