Method for the quantitative determination of vincarine, herbadine, and herbamine in the herbage of Vinca herbacea

Chemistry of Natural Compounds
1986.0

Abstract

The alkaloids vincarine, herbadine, and herbamine isolated from the herbage of Vinca herbacea Waldstet. et Kit. are pharmacologically active. A method for their quantitative determination in plant raw material is proposed, which consists in obtaining combined alkaloids, separating them by TLC (using KSK No. 2 silica gel and ethyl acetate-methanol (95:5) system), eluting with chloroform, and determining the alkaloids in the eluates by spectrophotometry on an SF-26 instrument. The method includes steps such as extracting alkaloids from 25 g of comminuted air-dry raw material with a 2% aqueous solution of sulfuric acid, obtaining amorphous combined alkaloids, dissolving them in chloroform, depositing the solution on a TLC plate, performing ascending chromatography, staining the marker band with cerium ammonium sulfate in 85% orthophosphoric acid, extracting the corresponding sorbent sections with chloroform, evaporating the extract, dissolving the residue in methanol, and calculating the amounts using optical density and a formula. Results show the amounts of vincarine (0.064%), herbadine (0.081%), and herbamine (0.077%) in the raw material on an absolutely dry weight basis. Additionally, it is known that the oxygen radical anion (O2•−) is formed in the autooxidation of phenols in alkaline media; Renard et al. suggest it plays an active part in the oxidation of lignin by a radical chain mechanism, but there are no experimental proofs of its formation in the oxidation of lignin and its model compounds in the literature.

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