Synthesis and evaluation of pyridyl analogs of L-735,524: Potent HIV-1 protease inhibitors

Synthesis and evaluation of pyridyl analogs of L-735,524: Potent HIV-1 protease inhibitors L-735,524: The Design of a Potent and Orally Bioavailable HIV Protease Inhibitor Identification of MK-944a:  A Second Clinical Candidate from the Hydroxylaminepentanamide Isostere Series of HIV Protease Inhibitors Synthesis and evaluation of 2-pyridinone derivatives as HIV-1-specific reverse transcriptase inhibitors. 2. Analogs of 3-aminopyridin-2(1H)-one Novel inhibitors of HIV protease HIV-1 protease inhibitory activity of L-694,746, a novel metabolite of L-689,502 Design and synthesis of potent HIV-1 protease inhibitors incorporating hydroxyprolinamides as novel P2 ligands Reduction of Peptide Character of HIV Protease Inhibitors That Exhibit Nanomolar Potency against Multidrug Resistant HIV-1 Strains Synthesis and biological evaluation of novel HIV-1 protease inhibitors using tertiary amine as P2-ligands HIV-1 Protease Inhibitors with a Transition-State Mimic Comprising a Tertiary Alcohol: Improved Antiviral Activity in Cells