Novel non-peptide ligands for the somatostatin sst3 receptor
Bioorganic & Medicinal Chemistry Letters
2001.0
Abstract
A series of imidazole derivatives has been prepared using high throughput parallel synthesis. Several compounds showed high affinity (Ki in 10(-6)-10(-8) M range) and selectivity at recombinant human somatostatin receptor subtype 3 (hsst3).