Nonpeptide αvβ3 antagonists. Part 2: constrained glycyl amides derived from the RGD tripeptide

Nonpeptide αvβ3 antagonists. Part 2: constrained glycyl amides derived from the RGD tripeptide Synthesis and Biological Evaluation (in Vitro and in Vivo) of Cyclic Arginine–Glycine–Aspartate (RGD) Peptidomimetic–Paclitaxel Conjugates Targeting Integrin α_Vβ₃ Rational Improvement of the Affinity and Selectivity of Integrin Binding of Grafted Lasso Peptides Synthesis of Pro-Leu-Gly-NH2 analogs modified at the prolyl residue and evaluation of their effects on the receptor binding activity of the central dopamine receptor agonist, ADTN Tri- and tetrapeptide analogs of kinins as potential renal vasodilators Dopamine receptor modulation by a highly rigid spiro bicyclic peptidomimetic of Pro-Leu-Gly-NH2 Synthesis of Novel c(AmpRGD)–Sunitinib Dual Conjugates as Molecular Tools Targeting the α_vβ₃ Integrin/VEGFR2 Couple and Impairing Tumor-Associated Angiogenesis Synthesis, biological studies and molecular dynamics of new anticancer RGD-based peptide conjugates for targeted drug delivery Multiple N-Methylation by a Designed Approach Enhances Receptor Selectivity Cyclization of RGD Peptides by Suzuki–Miyaura Cross-Coupling