Rational Improvement of the Affinity and Selectivity of Integrin Binding of Grafted Lasso Peptides

Rational Improvement of the Affinity and Selectivity of Integrin Binding of Grafted Lasso Peptides Nonpeptide αvβ3 antagonists. Part 2: constrained glycyl amides derived from the RGD tripeptide Multiple N-Methylation by a Designed Approach Enhances Receptor Selectivity Synthesis, biological studies and molecular dynamics of new anticancer RGD-based peptide conjugates for targeted drug delivery Synthesis and Biological Evaluation (in Vitro and in Vivo) of Cyclic Arginine–Glycine–Aspartate (RGD) Peptidomimetic–Paclitaxel Conjugates Targeting Integrin α_Vβ₃ Small Molecule Designed to Target Metal Binding Site in the α2I Domain Inhibits Integrin Function Cyclization of RGD Peptides by Suzuki–Miyaura Cross-Coupling Determination of the Binding Specificity of an Integral Membrane Protein by Saturation Transfer Difference NMR:  RGD Peptide Ligands Binding to Integrin α_IIbβ₃ Synthesis and Biological Evaluation of Dimeric RGD Peptide−Paclitaxel Conjugate as a Model for Integrin-Targeted Drug Delivery Discovery of Cyclic Peptidomimetic Ligands Targeting the Extracellular Domain of EGFR