Identification of small molecule agonists of the motilin receptor

Identification of small molecule agonists of the motilin receptor Discovery of a Potent and Novel Motilin Agonist The discovery of biaryl carboxamides as novel small molecule agonists of the motilin receptor Discovery of N-(3-Fluorophenyl)-1-[(4-([(3S)-3-methyl-1-piperazinyl]methyl)phenyl)acetyl]-4-piperidinamine (GSK962040), the First Small Molecule Motilin Receptor Agonist Clinical Candidate Investigations on the 1-(2-Biphenyl)piperazine Motif: Identification of New Potent and Selective Ligands for the Serotonin₇ (5-HT₇) Receptor with Agonist or Antagonist Action in Vitro or ex Vivo 9-Dihydroerythromycins as non-antibiotic motilin receptor agonists 9-Dihydroerythromycin ethers as motilin agonists—Developing structure–activity relationships for potency and safety Selective 5-Hydroxytryptamine 2C Receptor Agonists Derived from the Lead Compound Tranylcypromine: Identification of Drugs with Antidepressant-Like Action Heterocyclic aminopyrrolidine derivatives as melatoninergic agents Preparation and pharmacological evaluation of a novel series of 2-(phenylthio)benzo[b]thiophenes as selective MT2 receptor ligands